Index gene_name entrez_id category interaction_types drug_claim_name drug_name PMIDs 1 1 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor SNS-032 BMS-387032 2 2 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NIFEKALANT NIFEKALANT 4 3 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PENTACHLOROPHENOL PENTACHLOROPHENOL 5 4 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE AZ6089 22869148 6 5 APOE 348 DRUGGABLE GENOME PREDNISONE PREDNISONE 3185288 8 6 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Pyridazinone derivative 1 10 7 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISOFLAVONE ISOFLAVONE 15056880 11 8 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL576982 QUIZARTINIB 12 9 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 178101832 13 10 MAPT 4137 DRUGGABLE GENOME DIHYDROXANTHOHUMOL DIHYDROXANTHOHUMOL 16 11 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME sorafenib SORAFENIB 24569458 17 12 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor PF-4691502 PF-04691502 18 13 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR JNJ-7706621 JNJ-7706621 19 14 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AG-538 CHEMBL56393 20 15 CBX1 10951 NA BENSERAZIDE BENSERAZIDE 21 16 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME BI-505 BI-505 24 17 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE BPTES 21045145 25 18 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME PMID27539678-Compound-11 26 19 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 oxazepam OXAZEPAM 27 20 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME NSC-50690 CHEMBL1388703 28 21 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE inhibitor CHEMBL2013119 RIGOSERTIB SODIUM 30 22 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE ISTAROXIME ISTAROXIME 31 23 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR GSK2816126 33 24 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GNF-PF-5510 CHEMBL578741 36 25 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SJ000113257 CHEMBL528694 37 26 PI4KB 5298 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102683 38 27 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 178103393 ALEFACEPT 39 28 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ALPRENOLOL ALPRENOLOL 41 29 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALDICARB ALDICARB 43 30 SMARCA4 6597 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING inhibitor 249565598 44 31 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR FLUTICASONE PROPIONATE 12372131 45 32 CA2 760 DRUGGABLE GENOME, ENZYME PARABEN PARABEN 46 33 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178102292 CEDIRANIB 49 34 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 13 50 35 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ROTTLERIN ROTTLERIN 52 36 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX PMID27336223-Compound-12 54 37 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL3545209 NKTR-171 55 38 FMO3 2328 ENZYME, DRUGGABLE GENOME tacrolimus TACROLIMUS 28084894 56 39 GADD45A 1647 DNA REPAIR, TUMOR SUPPRESSOR, KINASE DOXORUBICIN DOXORUBICIN 7729953 57 40 POLK 51426 DNA REPAIR, ENZYME RESVERATROL RESVERATROL 61 41 GMNN 51053 DRUGGABLE GENOME IDAZOXAN IDAZOXAN 62 42 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Mifepristone MIFEPRISTONE 64 43 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME lenalidomide LENALIDOMIDE 27458141 65 44 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR SB-202190 SB-202190 22951114 66 45 RACGAP1 29127 NA TCMDC-124522 CHEMBL526776 67 46 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CHLORAMBUCIL CHLORAMBUCIL 8621235 68 47 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME PREDNISOLONE PREDNISOLONE 12730678 69 48 ATAD5 79915 NA DOMPERIDONE DOMPERIDONE 70 49 CACNB4 785 DRUGGABLE GENOME, ION CHANNEL VERAPAMIL VERAPAMIL 71 50 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PIRINIXIC ACID PIRINIXIC ACID 74 51 RAB9A 9367 ENZYME, DRUGGABLE GENOME NSC-234945 CHEMBL260311 77 52 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CYTARABINE CYTARABINE 22931300 78 53 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-US20120277229 45(1.5) 79 54 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME ANTHRACYCLINE 15297400 80 55 KDM4A 9682 DRUGGABLE GENOME, ENZYME CLOFAZIMINE CLOFAZIMINE 81 56 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565762 83 57 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103918 MK-0249 84 58 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE DINOPROSTONE DINOPROSTONE 87 59 BCHE 590 DRUGGABLE GENOME, ENZYME RVT-103+RVT-104 88 60 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DOXACURIUM DOXACURIUM 89 61 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR VINORELBINE VINORELBINE 23038758,24647522 90 62 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 91 63 TUBB 203068 DRUGGABLE GENOME inhibitor 135652721 PACLITAXEL 95 64 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DULOXETINE DULOXETINE 96 65 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME TRAMETINIB DIMETHYL SULFOXIDE 25435907,28480077,28078132 97 66 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR Everolimus EVEROLIMUS 26951309 98 67 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SALMETEROL SALMETEROL 100 68 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FLUNISOLIDE FLUNISOLIDE 22931300 102 69 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER BRYOSTATIN BRYOSTATIN 103 70 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DOMIPHEN BROMIDE DOMIPHEN BROMIDE 104 71 TOP2B 7155 DRUGGABLE GENOME, ENZYME Salvicine 106 72 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CAULIBUGULONE D CAULIBUGULONE D 108 73 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor RUXOLITINIB RUXOLITINIB 109 74 TH 7054 ENZYME, DRUGGABLE GENOME L-Phenylalanine PHENYLALANINE 111 75 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TASOSARTAN TASOSARTAN 113 76 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME L-701324 CHEMBL31741 114 77 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor PAZOPANIB PAZOPANIB 115 78 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200434 OXTRIPHYLLINE 116 79 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor VANDETANIB VANDETANIB 117 80 GMNN 51053 DRUGGABLE GENOME DNDI1417601 CHEMBL1503729 118 81 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 119 82 HDAC11 79885 DRUGGABLE GENOME, ENZYME PMID29671355-Compound-44 120 83 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR TRIMEPRAZINE TARTRATE TRIMEPRAZINE TARTRATE 121 84 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PI3KBETA INHIBITOR AZD8186 25544636 122 85 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE ivacaftor / tezacaftor 123 86 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR ON-01910 RIGOSERTIB 25156567 128 87 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE HYDROXYCHLOROQUINE HYDROXYCHLOROQUINE 9002011 131 88 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 315661265 133 89 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545368 PANOBINOSTAT LACTATE 135 90 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GA201 IMGATUZUMAB 23209031 136 91 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE IMATINIB IMATINIB 15928335,15685537,22718859,16638875,15146165,12949711,26130666,25157968,24132921,14645423,16954519,18794084,22745105 137 92 FURIN 5045 ENZYME, PROTEASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 252166802 138 93 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE Avastin+/-Tarceva 139 94 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE NICLOSAMIDE NICLOSAMIDE 142 95 RGS4 5999 DRUGGABLE GENOME METHYLDOPA METHYLDOPA 143 96 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME SB-224289 SB-224289 144 97 LIPC 3990 ENZYME, PHOSPHOLIPASE, LIPASE, DRUGGABLE GENOME ETHANOL ALCOHOL 7163806 145 98 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 3,3'-DIMETHOXYBENZIDINE CHEMBL398363 146 99 CSNK2A2 1459 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME, TRANSCRIPTION FACTOR US8791257, 17 147 100 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 17 148 101 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR 2-ENE-VALPROATE CHEMBL117487 17566732 149 102 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR BDBM50158803 150 103 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Anti-MUC1 mab 153 104 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 310264675 CUDC-101 154 105 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE OSI-632 OSI-632 156 106 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650208 DOXEPIN 157 107 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER antiepileptics 15452306,17125969,16386926,17306068,21747585,19450124,22630058,22188362,20417680,17521963,16004559,16542858,16753003,24300029,12686700,15857428,25458099,21391884,18812236 158 108 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100518 ZIBOTENTAN 160 109 CBX1 10951 NA PURPURIN PURPURIN 163 110 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CASEARINONE B CASEARINONE B 9322361 164 111 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AMG 595 165 112 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PYRENE PYRENE 166 113 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUOCINOLONE ACETONIDE FLUOCINOLONE ACETONIDE 167 114 TUBA1A 7846 DRUGGABLE GENOME MEBENDAZOLE MEBENDAZOLE 170 115 PDE3A 5139 ENZYME, DRUGGABLE GENOME VESNARINONE VESNARINONE 171 116 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROPACHLOR PROPACHLOR 172 117 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32i 173 118 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-7387 CHEMBL119878 174 119 GGCX 2677 DRUGGABLE GENOME, ENZYME PHYTONADIONE PHYTONADIONE 175 120 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1201023 ORPHENADRINE HYDROCHLORIDE 176 121 CTH 1491 ENZYME busulfan BUSULFAN 27779248 179 122 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1742420 AMELUBANT 181 123 KMO 8564 DRUGGABLE GENOME, ENZYME Pyrimidine benzenesulfonamide derivative 2 182 124 ALOX5 240 DRUGGABLE GENOME, ENZYME SKF-105809 184 125 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SU-4312 CHEMBL328710 185 126 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 178102655 186 127 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE pravastatin PRAVASTATIN 18622257 187 128 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SANGUINARIUM SANGUINARIUM 189 129 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR SELUMETINIB SELUMETINIB 191 130 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652666 ARECOLINE 192 131 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GTF505 193 132 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor 354702260 DEBIO-1347 195 133 CBX1 10951 NA NICARDIPINE NICARDIPINE 197 134 PDE4B 5142 DRUGGABLE GENOME, ENZYME RPL-554 198 135 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TANSHINONE IIA SULFONATE TANSHINONE IIA SULFONATE 200 136 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME Sodium Tetradecyl Sulfate 201 137 HDAC11 79885 DRUGGABLE GENOME, ENZYME CUDC-101 CUDC-101 202 138 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565638 ALPELISIB 204 139 AKR1B1 231 DRUGGABLE GENOME, ENZYME Ovine corticotropin-releasing hormone 205 140 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE TEMSIROLIMUS TEMSIROLIMUS 11504908,23674493 207 141 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 208 142 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE ZSTK474 209 143 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 211 144 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 178102483 212 145 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL2107067 TESTOSTERONE UNDECANOATE 214 146 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-67 CHEMBL578512 215 147 ADAMTS5 11096 DRUGGABLE GENOME, ENZYME, PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE inhibitor 252166754 216 148 ALPL 249 ENZYME, DRUGGABLE GENOME 5,7,3',5'-TETRAHYDROXYFLAVANONE CHEMBL307893 217 149 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE DASATINIB DASATINIB 219 150 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 249565586 POZIOTINIB 220 151 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE MENADIONE MENADIONE 221 152 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME DUAL IGF-1R/INSR INHIBITOR BMS-754807 25527633 222 153 TSPO 706 DRUGGABLE GENOME Quinoline carboxamide derivative 7 223 154 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AS-013 ECRAPROST 224 155 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE KML-001 226 156 CBR1 873 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME inhibitor 178102193 WEDELOLACTONE 227 157 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME CEDIRANIB CEDIRANIB 228 158 CA1 759 DRUGGABLE GENOME, ENZYME DICHLORPHENAMIDE DICHLORPHENAMIDE 229 159 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER LIK-066 LICOGLIFLOZIN 230 160 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LOTEPREDNOL ETABONATE LOTEPREDNOL ETABONATE 231 161 PLEKHJ1 55111 NA candesartan CANDESARTAN 31327267 232 162 MAOA 4128 DRUGGABLE GENOME, ENZYME Cyclic peptide derivative 1 235 163 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Sulfamethoxazole SULFAMETHOXAZOLE 236 164 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LISINOPRIL HYDRATE LISINOPRIL HYDRATE 237 165 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Gold-complexed thiosaccharide derivative 3 240 166 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SJ000019194 CHEMBL592106 241 167 CA5A 763 ENZYME, DRUGGABLE GENOME activator 178100344 HISTIDINE 242 168 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2062265 243 169 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE TABERMINOGENE VADENOVEC 247 170 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING DIPHENHYDRAMINE HYDROCHLORIDE DIPHENHYDRAMINE HYDROCHLORIDE 248 171 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RANITIDINE RANITIDINE 22931300 249 172 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NS-398 NS-398 251 173 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CHRYSENE-1,4-DIONE CHEMBL421215 252 174 GMNN 51053 DRUGGABLE GENOME GNF-PF-3438 CHEMBL582276 254 175 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 336446935 PREXASERTIB 255 176 KLK4 9622 PROTEASE, DRUGGABLE GENOME, ENZYME Benzyl amine derivative 1 256 177 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor 178101884 GSK-690693 257 178 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-15 260 179 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE GAMMA-INTERFERON 8144393 261 180 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2105762 OMARIGLIPTIN 262 181 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-106547 CHEMBL223575 265 182 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor CUDC-101 CUDC-101 266 183 KDM4A 9682 DRUGGABLE GENOME, ENZYME MONTELUKAST SODIUM MONTELUKAST SODIUM 267 184 RACGAP1 29127 NA ISOORIENTIN ISOORIENTIN 268 185 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PROTEASE INHIBITORS 16103765 270 186 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR ILORASERTIB ILORASERTIB 271 187 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME celecoxib CELECOXIB 22336956 275 188 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DYCLONINE DYCLONINE 276 189 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-1295 CHEMBL579837 277 190 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-625137A GSK-625137A 278 191 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 336446965 279 192 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651364 ZM-241385 280 193 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000114950 CHEMBL606456 281 194 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME peginterferon alfa-2b 23360626 284 195 P4HTM 54681 TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL3544988 DAPRODUSTAT 285 196 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ISOLIQUIRITIGENIN ISOLIQUIRITIGENIN 287 197 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 838877 CHEMBL405317 290 198 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR T091317 T091317 20350005 292 199 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE fluticasone propionate 18695978 293 200 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE NINTEDANIB NINTEDANIB 294 201 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR TAE-684 TAE-684 296 202 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CID 1245272 CHEMBL408850 298 203 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649749 299 204 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Platinum IV complexe 1 300 205 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-7 301 206 MPHOSPH8 54737 NA SB-224289 SB-224289 302 207 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Oxprenolol OXPRENOLOL 305 208 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TAE-684 TAE-684 306 209 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME VILDAGLIPTIN VILDAGLIPTIN 307 210 CPB2 1361 DRUGGABLE GENOME, ENZYME, PROTEASE UK-396082 UK-396,082 308 211 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR BUDESONIDE BUDESONIDE 311 212 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Temsirolimus TEMSIROLIMUS 27016228 312 213 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PAZOPANIB PAZOPANIB 313 214 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME GATIFLOXACIN GATIFLOXACIN 315 215 SMN2 6607 DRUGGABLE GENOME APIGENIN APIGENIN 318 216 MAPT 4137 DRUGGABLE GENOME ERGOCRYPTINE ERGOCRYPTINE 319 217 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ASENAPINE ASENAPINE 320 218 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME DYRENE DYRENE 322 219 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE BAY1436032 28232670 324 220 MPHOSPH8 54737 NA BAY-11-7085 BAY-11-7085 325 221 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CHLORAMPHENICOL CHLORAMPHENICOL 326 222 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MYRICETIN MYRICETIN 329 223 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor GDC-0941 PICTILISIB 330 224 APBB1 322 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING Trimidox TRIMETHOPRIM/SULFADOXINE 331 225 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ISOPRENALINE ISOPROTERENOL 333 226 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE CYC-116 CYC-116 334 227 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME agonist 178100907 335 228 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DNR 10050715 339 229 UGCG 7357 ENZYME, DRUGGABLE GENOME Eliglustat tartrate 340 230 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Trimipramine TRIMIPRAMINE 343 231 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL956 SUPROFEN 345 232 TH 7054 ENZYME, DRUGGABLE GENOME methylphenidate METHYLPHENIDATE 26810137 347 233 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pembrolizumab PEMBROLIZUMAB 27433843 348 234 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor INK-1117 INK-1117 349 235 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME G0-203-2c 351 236 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 352 237 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GW282974X GW282974X 353 238 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME INCB53914 355 239 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BILIRUBIN BILIRUBIN 359 240 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME 1-NAPHTHYLISOTHIOCYANATE 1-NAPHTHYLISOTHIOCYANATE 360 241 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 361 242 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE paliperidone PALIPERIDONE 25714000 363 243 ALOX5AP 241 DRUGGABLE GENOME DG031 364 244 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL705 ALITRETINOIN 365 245 PRSS2 5645 DRUGGABLE GENOME, PROTEASE, ENZYME DERMOLASTIN 367 246 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BROMODIPHENHYDRAMINE BROMODIPHENHYDRAMINE 368 247 ITPA 3704 ENZYME peginterferon alfa-2b 26441325,23730840,21274861,26916827,26670100,20173735,26071337,23707372,26438033,21246582,27833958,20547162,21503919,20637204 371 248 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565578 IPATASERTIB 372 249 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200376 BETAMETHASONE BENZOATE 373 250 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BECLOMETHASONE DIPROPIONATE BECLOMETHASONE DIPROPIONATE 374 251 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545134 LY-2780301 375 252 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR CAPSAICIN CAPSAICIN 10430952 378 253 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME AZD-1152-HQPA AZD-1152-HQPA 381 254 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 383 255 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FLUOXETINE HYDROCHLORIDE FLUOXETINE HYDROCHLORIDE 387 256 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE NVP-TNKS656 26224873 389 257 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 354702297 GSK-1059615 392 258 HMGCR 3156 ENZYME, DRUGGABLE GENOME Sterol derivative 1 393 259 RAB9A 9367 ENZYME, DRUGGABLE GENOME TDR77585 CHEMBL1333386 394 260 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TICRYNAFEN TICRYNAFEN 22931300 395 261 HTT 3064 DRUGGABLE GENOME CUDC-907 FIMEPINOSTAT 398 262 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Aminocyclopentenone compound 1 399 263 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE LAK CELL 7947458,8381564,1683349 400 264 PAH 5053 DRUGGABLE GENOME, ENZYME TETRAHYDROBIOPTERIN SAPROPTERIN 401 265 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PGF2alpha 402 266 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Vedolizmab 406 267 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME CHEMBL2364609 ESKETAMINE HYDROCHLORIDE 407 268 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME 4-PAM derivative 1 408 269 PMS2 5395 CLINICALLY ACTIONABLE, DRUGGABLE GENOME NIVOLUMAB NIVOLUMAB 27001570 409 270 RRM2 6241 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL467 HYDROXYUREA 412 271 IFNG 3458 DRUGGABLE GENOME CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 10823419 413 272 CBX1 10951 NA ROTENONE ROTENONE 416 273 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE ILORASERTIB ILORASERTIB 418 274 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME RGB-286638 RGB-286638 420 275 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CHEMBL1201550 DENILEUKIN DIFTITOX 421 276 PTGES3 10728 ENZYME GENISTEIN GENISTEIN 15229138 422 277 MAGEA3 4102 ENZYME, DRUGGABLE GENOME Astuprotimut-R ASTUPROTIMUT-R 423 278 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PF-04691502 PF-04691502 21750219 424 279 COMT 1312 DRUGGABLE GENOME, ENZYME fluvoxamine FLUVOXAMINE 20619611 425 280 F11 2160 DRUGGABLE GENOME, PROTEASE, ENZYME ANTITHROMBIN 426 281 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE HYDROQUINONE HYDROQUINONE 10220568 428 282 PRPS1 5631 DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, ENZYME THIOGUANINE THIOGUANINE 25962120 431 283 RRM2 6241 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1096882 FLUDARABINE PHOSPHATE 433 284 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME QUINACRINE QUINACRINE 434 285 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CP-55940 CP-55940 435 286 ALB 213 TRANSPORTER, DRUGGABLE GENOME Sodium lauryl sulfate 436 287 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ACEBUTOLOL ACEBUTOLOL 439 288 IDO2 169355 ENZYME 2,3-diamino-benzo[b]thiophene derivative 5 440 289 NDUFB2 4708 ENZYME inhibitor CHEMBL3545135 NV-128 441 290 TNFSF13 8741 DRUGGABLE GENOME TACI-IG ATACICEPT 442 291 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Pazopanib HCl 444 292 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME WIN-552122 WIN-552122 446 293 PSMB4 5692 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL2103884 OPROZOMIB 447 294 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 178103659 449 295 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ALPHA,BETA-METHYLENE-DCTP CHEMBL1162298 18811136 450 296 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE anthracyclines and related substances 25545243,24533712,11160862,21479364,10208650,21946896,18511948 452 297 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX HELENALIN HELENALIN 453 298 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ACID BLUE 129 ACID BLUE 129 455 299 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL1200592 DESOXYCORTICOSTERONE PIVALATE 456 300 SI 6476 DRUGGABLE GENOME, ENZYME DEXAMETHASONE DEXAMETHASONE 2295387 457 301 VSIR 64115 DRUGGABLE GENOME, CLINICALLY ACTIONABLE JNJ-61610588 ONVATILIMAB 458 302 RRP7A 27341 NA methylphenidate METHYLPHENIDATE 29382897 459 303 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE DIGOXIGENIN DIGOXIGENIN 461 304 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Guadecitabine GUADECITABINE 462 305 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR WX-554 WX-554 464 306 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Metformin glycinate 22974412 465 307 BAZ2B 29994 NA ELLIPTECINE ELLIPTECINE 466 308 ATAD5 79915 NA DNDI1417132 CHEMBL1492017 467 309 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL451887 CARFILZOMIB 468 310 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER NEVIRAPINE NEVIRAPINE 17172311 469 311 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ORG 34517/34850 470 312 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Exemestane EXEMESTANE 471 313 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor CHEMBL3544942 RONICICLIB 472 314 HPSE 10855 ENZYME, DRUGGABLE GENOME TGF 16320243 473 315 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652307 474 316 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Imidazo[1,2-b]pyridazine derivative 2 478 317 HTT 3064 DRUGGABLE GENOME GNF-PF-4659 CHEMBL584442 479 318 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL levetiracetam LEVETIRACETAM 23859570,21747585,28753467,25155934 480 319 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200895 PHENELZINE SULFATE 482 320 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ZM-336372 CHEMBL186526 485 321 NR5A2 2494 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR TDR79154 CHEMBL597670 489 322 FAAH 2166 ENZYME, DRUGGABLE GENOME Azetidine urea derivative 3 490 323 SOST 50964 DRUGGABLE GENOME LY2541546 491 324 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME 3144 28235199 493 325 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 340590212 494 326 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TCDD 7530807 496 327 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SJ000147993 CHEMBL601618 497 328 PDE4B 5142 DRUGGABLE GENOME, ENZYME DYPHYLLINE DYPHYLLINE 499 329 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME BENSULIDE BENSULIDE 500 330 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME (+)-ISOBICYCLOGERMACRENAL CHEMBL2333548 503 331 ADK 132 DRUGGABLE GENOME, ENZYME, KINASE DABIGATRAN DABIGATRAN 22494098 504 332 FHIT 2272 CLINICALLY ACTIONABLE, ENZYME, TRANSPORTER TRICHOSTATIN A 17019711 505 333 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CLOBAZAM CLOBAZAM 506 334 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SANGUINARIUM SANGUINARIUM 508 335 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CYC-116 CYC-116 511 336 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SB-207266A 513 337 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE VADIMEZAN VADIMEZAN 514 338 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CHEMBL3545206 GSK1482160 516 339 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE SIBUTRAMINE HYDROCHLORIDE SIBUTRAMINE HYDROCHLORIDE 517 340 ABCA1 19 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE pravastatin PRAVASTATIN 19673941,20031551 521 341 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103498 523 342 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US8563594, 152 524 343 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4-METHOXYDALBERGIONE 4-METHOXYDALBERGIONE 525 344 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650321 526 345 SREBF1 6720 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR fluvastatin FLUVASTATIN 527 346 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME Sevoflurane SEVOFLURANE 529 347 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZD4547 26351323 531 348 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE MS417 26058079 532 349 GMNN 51053 DRUGGABLE GENOME SJ000293754 CHEMBL486706 533 350 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103646 DESOXIMETASONE 535 351 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME Oxazolyl methylthiothiazole derivative 1 536 352 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PMID26161698-Compound-18 537 353 GMNN 51053 DRUGGABLE GENOME CINACALCET CINACALCET 538 354 ATAD5 79915 NA EMETINE EMETINE 541 355 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME HALAZEPAM HALAZEPAM 542 356 APBA1 320 NA HESPERIDIN HESPERIDIN 543 357 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PARAROSANILINE PARAROSANILINE 545 358 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HISTAMINE HISTAMINE 546 359 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE UROKINASE UROKINASE 547 360 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL DWJ-208 550 361 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE LEVOMETHADYL ACETATE 551 362 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist 354702202 TROPIFEXOR 552 363 FTO 79068 ENZYME interferon alfa-2b, recombinant 25367448 553 364 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE AIKO-150 554 365 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE Verteporfin VERTEPORFIN 27308390 556 366 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME DEFEROXAMINE DEFEROXAMINE 9194688 557 367 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL190 THEOPHYLLINE 558 368 TSPO 706 DRUGGABLE GENOME Quinoline carboxamide derivative 4 563 369 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PHENIRAMINE PHENIRAMINE 564 370 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LEVOBUNOLOL LEVOBUNOLOL 565 371 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FLUACIZINE FLUACIZINE 566 372 NOS2 4843 DRUGGABLE GENOME, ENZYME GW274150 GW-274150 567 373 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CLOFENOXYDE CLOFENOXYDE 568 374 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENOXYCARB PHENOXYCARB 570 375 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME AMG 232 25567130 577 376 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME activator 53801018 SPHINGOSINE 578 377 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor LGX818 ENCORAFENIB 582 378 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DNDI1417055 CHEMBL1486366 583 379 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE ZM-447439 CHEMBL202721 584 380 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Beta-phe compound 2 586 381 SLC15A1 6564 DRUGGABLE GENOME, TRANSPORTER inhibitor 178101226 589 382 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BEZ235 DACTOLISIB 592 383 KDM4A 9682 DRUGGABLE GENOME, ENZYME CHLOROGENIC ACID CHLOROGENIC ACID 593 384 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL451887 CARFILZOMIB 597 385 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME N-(3-METHOXYPHENYL)ANTHRANILIC ACID CHEMBL1328677 599 386 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SORAFENIB SORAFENIB 602 387 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3-HYDROXY-3',4'-DIMETHOXYFLAVONE 3-HYDROXY-3',4'-DIMETHOXYFLAVONE 603 388 FFAR4 338557 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 252166628 604 389 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE O-METHYLCALOTHRIXIN A O-METHYLCALOTHRIXIN A 19203291 606 390 FKBP5 2289 DRUGGABLE GENOME escitalopram ESCITALOPRAM 607 391 RGS4 5999 DRUGGABLE GENOME PICEATANNOL PICEATANNOL 608 392 MPHOSPH8 54737 NA PROCHLORPERAZINE PROCHLORPERAZINE 610 393 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE LIF 7686393 611 394 RPTOR 57521 CLINICALLY ACTIONABLE, KINASE everolimus EVEROLIMUS 612 395 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3545324 RG-7666 613 396 CCL2 6347 DRUGGABLE GENOME NOX-E36 614 397 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Edrophonium EDROPHONIUM 615 398 ALAD 210 ENZYME Aminolevulinic acid hci 620 399 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DICHLOROPHEN DICHLOROPHEN 621 400 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE AVT-02 UE 622 401 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ANTIOXIDANT 16817236 624 402 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHIOCARB METHIOCARB 627 403 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Macrocycle derivative 13 628 404 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GOSSYPOL GOSSYPOL 629 405 PTHLH 5744 HORMONE ACTIVITY, DRUGGABLE GENOME MAGNESIUM SULFATE 11384692 630 406 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650496 631 407 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 387065584 633 408 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR vitamin d and analogues 21651652,15295697,15861036,15739035,17763859,20716226,20500803,15864137,19647104 634 409 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME SOPHORAFLAVANONE G SOPHORAFLAVANONE G 18565755 636 410 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1201827 PANITUMUMAB 637 411 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR US9006244, E2a 639 412 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE abciximab ABCIXIMAB 20938371 642 413 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER fluorouracil FLUOROURACIL 643 414 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178102626 644 415 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE MIDAZOLAM MIDAZOLAM 16406030 646 416 ATAD5 79915 NA GNF-PF-4418 CHEMBL604321 647 417 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME AMG 820 648 418 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 135650917 649 419 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE DIHYDROXANTHOHUMOL DIHYDROXANTHOHUMOL 652 420 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LISDEXAMFETAMINE LISDEXAMFETAMINE 653 421 PTGS1 5742 ENZYME, DRUGGABLE GENOME MESALAZINE MESALAMINE 654 422 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-7387 CHEMBL119878 655 423 CYTH2 9266 NA CLOTRIMAZOLE CLOTRIMAZOLE 657 424 PTGS2 5743 DRUGGABLE GENOME, ENZYME Tolmetin TOLMETIN 659 425 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TRICLOCARBAN TRICLOCARBAN 660 426 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PENTOXIFYLLINE PENTOXIFYLLINE 11836847 661 427 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ethanol ALCOHOL 24611668 664 428 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Cobimetinib COBIMETINIB 665 429 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME Tafamidis TAFAMIDIS 667 430 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650031 LEVOBUNOLOL 668 431 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE (S)-FLUOXETINE CHEMBL1169388 669 432 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALX-0061 VOBARILIZUMAB 670 433 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE inhibitor 252166838 GALETERONE 681 434 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL599 MELOXICAM 682 435 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE EMODIN EMODIN 9671406 683 436 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CUDC-101 CUDC-101 684 437 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL1742994 BRENTUXIMAB VEDOTIN 685 438 MAOA 4128 DRUGGABLE GENOME, ENZYME Tarnylcypromine derivative 3 686 439 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE Mapatumumab MAPATUMUMAB 687 440 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 223366046 AZD-7762 689 441 TSPO 706 DRUGGABLE GENOME Imidazopyridine acetamide analog 7 693 442 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 249565800 694 443 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BISPHENOL A BISPHENOL A 696 444 ATAD5 79915 NA GNF-PF-5159 CHEMBL1493528 697 445 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE SOTRASTAURIN SOTRASTAURIN 699 446 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ketorolac KETOROLAC 17986163 700 447 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ENDOTHELIN RECEPTOR ANTAGONIST 16741044 702 448 POLK 51426 DNA REPAIR, ENZYME IODOPHTHALEIN IODOPHTHALEIN 704 449 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE EVEROLIMUS EVEROLIMUS 21189378 705 450 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565687 708 451 DHFR 1719 DRUGGABLE GENOME, ENZYME 10-PROPARGYL-10-DEAZAAMINOPTERIN PRALATREXATE 710 452 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL1944698 ZOTIRACICLIB 711 453 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR LY2835219 ABEMACICLIB 712 454 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIDECYLDIMETHYLAMMONIUM CHLORIDE DIDECYLDIMETHYLAMMONIUM CHLORIDE 715 455 TUBB 203068 DRUGGABLE GENOME Simotaxel SIMOTAXEL 716 456 CP 1356 DRUGGABLE GENOME, ENZYME DEXRAZOXANE DEXRAZOXANE 8285144 719 457 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ISORHAMNETIN ISORHAMNETIN 25190466 720 458 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALITRETINOIN ALITRETINOIN 721 459 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Benzimidazole and imadazopyridine carboximidamide compound 1 722 460 BAZ2B 29994 NA 4-HYDROXYESTRADIOL CHEMBL1412489 724 461 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLEBOPRIDE CLEBOPRIDE 725 462 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1111 AMBRISENTAN 726 463 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BKM120 BUPARLISIB 26715098,22159814,26098748,24576621 727 464 CYB5R2 51700 DRUGGABLE GENOME primaquine PRIMAQUINE 729 465 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE FIRATEGRAST FIRATEGRAST 730 466 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME RIMEXOLONE RIMEXOLONE 731 467 RACGAP1 29127 NA THUNBERGINOL B THUNBERGINOL B 732 468 APOE 348 DRUGGABLE GENOME BUTHIONINE SULFOXIMINE 12615656 734 469 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101619 ERLOTINIB 735 470 TUBB2A 7280 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 736 471 FAAH 2166 ENZYME, DRUGGABLE GENOME SSR411298 737 472 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DISULFIRAM DISULFIRAM 740 473 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR ZERANOL ZERANOL 741 474 VCAM1 7412 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME TROGLITAZONE TROGLITAZONE 10626906 744 475 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 745 476 NELFCD 51497 KINASE diuretics 746 477 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650867 PYRILAMINE 747 478 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CHEMBL2108029 ERTUMAXOMAB 750 479 ALDH1A1 216 DRUGGABLE GENOME, ENZYME N- (9-FLUORENYLMETHOXYCARBONYL)-L-LEUCINE N- (9-FLUORENYLMETHOXYCARBONYL)-L-LEUCINE 751 480 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TERAZOSIN HYDROCHLORIDE TERAZOSIN HYDROCHLORIDE 752 481 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZD4785 AZD-4785 753 482 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME PYROGALLOL RED PYROGALLOL RED 754 483 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE metformin METFORMIN 28834135 755 484 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE FLUOROURACIL FLUOROURACIL 25788273 756 485 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102337 SORAFENIB 757 486 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2062264 PHENYLEPHRINE BITARTRATE 759 487 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 328083523 760 488 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE GENISTEIN GENISTEIN 9349317 761 489 GLS 2744 ENZYME CEFATRIZINE CEFATRIZINE 762 490 ABCC5 10057 DRUGGABLE GENOME, ABC TRANSPORTER, TRANSPORTER inhibitor 178101454 SILDENAFIL 763 491 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME ANTIMETABOLITE 10997587 764 492 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME INOC-005 765 493 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 187051758 INDACATEROL 766 494 GSTA1 2938 ENZYME, DRUGGABLE GENOME vincristine VINCRISTINE 29938344,19448608 767 495 CA9 768 DRUGGABLE GENOME, ENZYME inhibitor 385612194 773 496 ATAD5 79915 NA GNF-PF-5183 CHEMBL577660 775 497 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR UREA UREA 8167573 776 498 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME buprenorphine BUPRENORPHINE 29333880 777 499 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL2103975 VAPREOTIDE 778 500 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Phenindamine PHENINDAMINE 779 501 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE GPC3 targeting CAR-T cells 780 502 NRIP1 8204 NUCLEAR HORMONE RECEPTOR RETINOIC ACID 15632153,14581481 782 503 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 385612228 787 504 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135650038 788 505 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME PD-0166285 PD-0166285 791 506 MAPT 4137 DRUGGABLE GENOME FENRETINIDE FENRETINIDE 792 507 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolo[2,3-b]pyridine derivative 3 793 508 DHFR 1719 DRUGGABLE GENOME, ENZYME inhibitor 310264671 795 509 RBP4 5950 DRUGGABLE GENOME US8853215, 3 800 510 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE DASATINIB DASATINIB 20360610 801 511 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME GNF-PF-4459 CHEMBL585502 802 512 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE G007-LK 28611108 803 513 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR metoprolol METOPROLOL 15864115,20643254,15861037,16815314,20352314,12709726,12921807,15735607,18075464,12844134,22617224,17496726,14534524,21311897,14502278,20235788,16402084 805 514 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor GDC-0980 APITOLISIB 806 515 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE gefitinib GEFITINIB 18681783,17375033,22370314,14990633,16467544,16377102,17317677,14990632,18784101,17020982,19473722,21921847,16912157,19589612,20573926,16258541,19692680,22581822,17192902,16203769,16257339,17429313,18000659,17085664,18003960,19381876,17473659,15897572,22215752,26490356,23022519,21900837,20038723,16865253,11255078,17285735,15118073,20022809,16115929,19339720,18316547,19201048,22760226,16204011,16956694,17597605,12648464,21233402,18992959,22237259,22594511 809 516 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR APICIDIN APICIDIN 19705846 810 517 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE INSULIN INSULIN 15202783,8727949 811 518 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR JNJ-1661010 CHEMBL460273 812 519 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650396 813 520 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Pyrrolo[2,3-d]pyrimidine derivative 24 814 521 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE SP-600125 SP-600125 815 522 ATAD5 79915 NA DICHLORORIBOBENZIMIDAZOLE DICHLORORIBOBENZIMIDAZOLE 817 523 ATAD5 79915 NA DNDI1417195 CHEMBL1303948 819 524 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-28 820 525 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR THEOPHYLLINE THEOPHYLLINE 822 526 IL1A 3552 CELL SURFACE, DRUGGABLE GENOME RILONACEPT RILONACEPT 823 527 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL24828 VANDETANIB 824 528 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR FENRETINIDE FENRETINIDE 12234979,17273769 826 529 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NALED NALED 827 530 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SOTRASTAURIN SOTRASTAURIN 828 531 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME PD-146176 CHEMBL180917 829 532 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor BAY1000394 830 533 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE AZD-1775 ADAVOSERTIB 831 534 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME GEFITINIB GEFITINIB 832 535 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME inhibitor 135651427 ADENOSINE DIPHOSPHATE 835 536 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Flavopiridol analog 1 838 537 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ANTIOXIDANT 11274788 839 538 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL378544 VINBLASTINE SULFATE 840 539 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CARMINE CARMINE 841 540 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL16 PHENYTOIN 843 541 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MORNIFLUMATE MORNIFLUMATE 844 542 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE INC280 CAPMATINIB 28783719 847 543 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME METHOTREXATE METHOTREXATE 11237386 849 544 EIF4A1 1973 DRUGGABLE GENOME SILVESTROL SILVESTROL 22128783 859 545 TESK2 10420 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TYROSINE KINASE inhibitor 249565798 861 546 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GW7074 CHEMBL72365 862 547 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME PROTEIN SYNTHESIS INHIBITOR 10488140 863 548 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PYRROLIDINE DITHIOCARBAMATE PYRROLIDINE DITHIOCARBAMATE 866 549 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Pyrido[1,2-a]indole-1.-carboxylic acid analog 2 867 550 S100A12 6283 DRUGGABLE GENOME, KINASE Atogepant ATOGEPANT 868 551 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SITAXSENTAN SITAXENTAN 869 552 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 252166627 GLPG-0974 870 553 EIF2B1 1967 NA WORTMANNIN WORTMANNIN 10764740 872 554 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RHEIN RHEIN 873 555 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TYRPHOSTIN 23 TYRPHOSTIN 23 874 556 IGF1 3479 GROWTH FACTOR, HORMONE ACTIVITY, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE BI-836845 XENTUZUMAB 875 557 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Quinoxaline derivative 3 876 558 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL antagonist 178103764 FLUVOXAMINE 877 559 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE VANDETANIB VANDETANIB 878 560 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Premarin/Pravachol 881 561 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE QUININE SULFATE QUININE SULFATE 883 562 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 363894206 ALLITINIB 885 563 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL2138601 REFAMETINIB 886 564 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL422872 AZD-4769 887 565 TUBB 203068 DRUGGABLE GENOME Tasidotin hydrochloride 889 566 PTGS2 5743 DRUGGABLE GENOME, ENZYME IBUPROFEN IBUPROFEN 890 567 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME SU-4312 CHEMBL328710 892 568 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MEDRONIC ACID MEDRONIC ACID 894 569 HTT 3064 DRUGGABLE GENOME PMID27376512-Compound-PG-11047 896 570 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE [131I]-BC8 898 571 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 9-PHENYLIMIDAZO[1,2-H][1,7]NAPHTHYRIDINE CHEMBL455004 22503207 903 572 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-67 904 573 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PLX3397 PEXIDARTINIB 25939769 905 574 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROPYLPARABEN PROPYLPARABEN 910 575 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27551786-Compound-106 912 576 SOST 50964 DRUGGABLE GENOME inhibitor CHEMBL1742993 BLOSOZUMAB 913 577 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-202190 SB-202190 915 578 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME artemisinin ARTEMISININ 17638512,11470993 916 579 BAZ2B 29994 NA SJ000018300 CHEMBL590927 917 580 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NILUTAMIDE NILUTAMIDE 920 581 TAC1 6863 DRUGGABLE GENOME PUROMYCIN PUROMYCIN 14623771 921 582 PDE3A 5139 ENZYME, DRUGGABLE GENOME K-134 K-134 23110051 922 583 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417601 CHEMBL1503729 923 584 HKDC1 80201 DRUGGABLE GENOME, KINASE SJ000044511 CHEMBL592124 924 585 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Olaparib OLAPARIB 26909613 925 586 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 315661259 927 587 NR1D1 9572 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME SR9011 SR9011 23656296 928 588 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 363894176 931 589 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000014858 CHEMBL591628 932 590 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR PACLITAXEL PACLITAXEL 17229776 933 591 DCTD 1635 ENZYME gemcitabine GEMCITABINE 22838950 934 592 GMNN 51053 DRUGGABLE GENOME OUABAIN OUABAIN 935 593 TUBA1A 7846 DRUGGABLE GENOME CHEMBL2108628 PACLITAXEL POLIGLUMEX 936 594 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME FLUOROMETHOLONE FLUOROMETHOLONE 937 595 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CID 663143 CHEMBL1342336 938 596 MPHOSPH8 54737 NA NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 940 597 CBX1 10951 NA MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 941 598 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME A-1155463 25787766 942 599 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 249565751 945 600 FAAH 2166 ENZYME, DRUGGABLE GENOME Spirocyclic diamine urea derivative 2 947 601 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME NITROGEN MUSTARD 9459175,11839668 949 602 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 384403649 STANOZOLOL 950 603 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CAR-T cells targeting CD20 951 604 GBA 2629 DRUGGABLE GENOME, ENZYME GNF-PF-4085 CHEMBL528181 953 605 FAAH 2166 ENZYME, DRUGGABLE GENOME Propofol PROPOFOL 954 606 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER inhibitor 384403652 955 607 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL235191 TACEDINALINE 956 608 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 385612230 957 609 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL2096631 CLORAZEPATE DIPOTASSIUM 964 610 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Misoprostol MISOPROSTOL 965 611 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE Crizotinib CRIZOTINIB 27009859,25749034,24509625,18089725,25421750 967 612 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist 178103554 VISMODEGIB 969 613 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 971 614 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR UVB 14514652 972 615 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME rosuvastatin ROSUVASTATIN 973 616 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Pz-1 26126987 974 617 PLAUR 5329 DRUGGABLE GENOME, ENZYME, CELL SURFACE ADENOVIRAL VECTOR 12955075 975 618 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL3545386 BI113823 978 619 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AGROCLAVINE AGROCLAVINE 980 620 POLK 51426 DNA REPAIR, ENZYME CARMINE CARMINE 981 621 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE GNF-PF-1399 CHEMBL578504 982 622 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE BI-87E7 CHEMBL523200 984 623 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Rivastigmine RIVASTIGMINE 985 624 APH1B 83464 PROTEASE, DRUGGABLE GENOME LY-411575 CHEMBL392068 23181502,19443228 988 625 ASXL1 171023 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR N/A 24220272,26849014,20880116,21714648,23690417 989 626 KDM4A 9682 DRUGGABLE GENOME, ENZYME ERGOCRYPTINE ERGOCRYPTINE 991 627 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ARN-509 APALUTAMIDE 992 628 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME SODIUM BUTYRATE 2211839 994 629 PDE4A 5141 DRUGGABLE GENOME, ENZYME ENPROFYLLINE ENPROFYLLINE 995 630 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL932 DIPYRIDAMOLE 996 631 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CRUFOMATE CRUFOMATE 999 632 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME TAMATINIB R-406 1000 633 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 867101 CHEMBL406557 1001 634 AKR1B1 231 DRUGGABLE GENOME, ENZYME QR-333 1003 635 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE haloperidol HALOPERIDOL 27023437,18695978 1004 636 POLB 5423 DNA REPAIR, DRUGGABLE GENOME MBO7133 (CYTARABINE PRODRUG) 1005 637 ATXN2 6311 NA TCMDC-125298 CHEMBL581152 1007 638 ME3 10873 ENZYME DHT ANDROSTANOLONE 1811987 1008 639 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Thiadiazolidindione derivative 2 1010 640 PTGIS 5740 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME PHENYLBUTAZONE PHENYLBUTAZONE 1014 641 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME CLOZAPINE CLOZAPINE 12873733 1017 642 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 405067320 1018 643 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178101060 1019 644 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 223365979 PELITINIB 1020 645 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 135650006 1021 646 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000032081 CHEMBL590184 1022 647 TUBA1A 7846 DRUGGABLE GENOME CHEMBL492399 VERUBULIN 1023 648 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE SORAFENIB SORAFENIB 1025 649 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650766 1026 650 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE NSC-79888 CHEMBL1939433 22212721 1027 651 PNP 4860 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL550755 FORODESINE HYDROCHLORIDE 1028 652 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR Alpha 2 Interferon 16827904 1029 653 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE OSI-906 LINSITINIB 1031 654 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000018300 CHEMBL590927 1033 655 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE HYDROGEN PEROXIDE HYDROGEN PEROXIDE 15012988 1035 656 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PSORALEN PSORALEN 1039 657 CDK18 5129 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR inhibitor 249565897 1041 658 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Cyclic hydroxamate derivative 1 1042 659 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME RIVASTIGMINE RIVASTIGMINE 1043 660 ANO1 55107 ION CHANNEL blocker 178100996 1045 661 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR ENTRECTINIB ENTRECTINIB 28183697 1046 662 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PANITUMUMAB PANITUMUMAB 19223544 1047 663 PTGS2 5743 DRUGGABLE GENOME, ENZYME PHENYLBUTAZONE PHENYLBUTAZONE 1048 664 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DOPAMINE HYDROCHLORIDE DOPAMINE HYDROCHLORIDE 1051 665 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE RETINOL RETINOL 1576255 1052 666 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX BISINDOLYLMALEIMIDE IX BISINDOLYLMALEIMIDE IX 1053 667 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIBUTYLTIN-OXIDE TRIBUTYLTIN-OXIDE 1054 668 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME blocker 135650269 1055 669 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200602 1058 670 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-PHENYLPHENOL 2-PHENYLPHENOL 1062 671 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE BERGAMOTTIN BERGAMOTTIN 1063 672 IL13RA2 3598 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Tralokinumab TRALOKINUMAB 1064 673 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR PI-88 MUPARFOSTAT 11292191 1068 674 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PRAZOSIN HYDROCHLORIDE PRAZOSIN HYDROCHLORIDE 1070 675 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Talazoparib TALAZOPARIB 1071 676 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR 9-CIS RETINOIC ACID 9869165 1072 677 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BIPERIDEN BIPERIDEN 22793499 1073 678 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor CHEMBL403989 TG100-801 1076 679 PPP3CA 5530 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Cyclosporine CYCLOSPORINE 1077 680 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME aflatoxin b1 17638512,11470993 1078 681 TUBA4A 7277 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 1080 682 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL ZONISAMIDE ZONISAMIDE 1083 683 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1567 SUNITINIB MALATE 1084 684 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME inhibitor 178101343 1087 685 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR Gemcitabine GEMCITABINE 26853339 1089 686 KCNJ5 3762 TRANSPORTER, ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FLUPIRTINE FLUPIRTINE 1090 687 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE DIZOCILPINE DIZOCILPINE 20361801 1091 688 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME TOZASERTIB TOZASERTIB 1093 689 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TCMDC-123920 CHEMBL1606 1094 690 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 6-CHLOROMELATONIN CHEMBL34730 1096 691 GATM 2628 ENZYME, TRANSPORTER hmg coa reductase inhibitors 1097 692 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE SODIUM CROMOGLYCATE 7554404 1098 693 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SPI-1620 IRL-1620 1099 694 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE sulfasalazine SULFASALAZINE 12083967 1101 695 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SRT-1720 CHEMBL257991 1104 696 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE BAY-613606 CHEMBL541400 1106 697 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102585 DOVITINIB 1108 698 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TCMDC-125575 CHEMBL587620 1111 699 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR IDARUBICIN IDARUBICIN 1112 700 TUBA3D 113457 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 1113 701 MAPT 4137 DRUGGABLE GENOME RALOXIFENE RALOXIFENE 1114 702 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CLOROPHENE CLOROPHENE 1115 703 ATIC 471 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE FOLIC ACID 9679969 1116 704 POLB 5423 DNA REPAIR, DRUGGABLE GENOME DIOSMIN DIOSMIN 1118 705 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-1 1119 706 ATAD5 79915 NA 4,5,6,7-TETRABROMOBENZIMIDAZOLE CHEMBL373937 1120 707 KDM4A 9682 DRUGGABLE GENOME, ENZYME 4-HYDROXYESTRADIOL CHEMBL1412489 1122 708 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LAS38096 CHEMBL375293 1125 709 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CYC-116 CYC-116 1126 710 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE ERLOTINIB ERLOTINIB 22328973 1127 711 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME RAPAMYCIN SIROLIMUS 16127150 1128 712 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 1-BENZYLMALEIMIDE CHEMBL388979 1130 713 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Syntropin 1131 714 HMGCR 3156 ENZYME, DRUGGABLE GENOME CRILVASTATIN CRILVASTATIN 1132 715 HTT 3064 DRUGGABLE GENOME GNF-PF-1852 CHEMBL533293 1133 716 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor BYL719 ALPELISIB 1135 717 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SB-203580 SB-203580 1136 718 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor PKI-587 GEDATOLISIB 1137 719 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DOXORUBICIN DOXORUBICIN 22931300 1138 720 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor GSK2126458 OMIPALISIB 1139 721 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME LIF 8156996 1140 722 RGS4 5999 DRUGGABLE GENOME AM-251 CHEMBL285932 1141 723 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL522892 DOVITINIB 1143 724 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DEMETHOXYCURCUMIN DEMETHOXYCURCUMIN 19112019 1147 725 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME APICIDIN APICIDIN 19705846,17956988 1148 726 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32h 1150 727 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-55 1151 728 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CAROTENOIDS 16454745 1153 729 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Obinutuzumab OBINUTUZUMAB 1154 730 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CAPSAZEPINE CAPSAZEPINE 1156 731 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL1186894 AMRUBICIN 1157 732 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 249565691 CHEMBL1086377 1160 733 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker 135652722 TETRODOTOXIN 1161 734 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Sorafenib SORAFENIB 1165 735 ADCY9 115 KINASE, ENZYME, DRUGGABLE GENOME NSC-270718 CHEMBL401844 18630896 1167 736 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE 1168 737 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IPRATROPIUM IPRATROPIUM 22931300 1169 738 MAPT 4137 DRUGGABLE GENOME GNF-PF-5134 CHEMBL602969 1170 739 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 329968451 SOLABEGRON 1171 740 USP9Y 8287 ENZYME, PROTEASE TESTOSTERONE TESTOSTERONE 10439009 1172 741 MAOB 4129 DRUGGABLE GENOME, ENZYME PHENELZINE PHENELZINE 1173 742 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CH-5132799 PA-799 1174 743 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE LY-255283 LY-255283 1175 744 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER GARCINONE E GARCINONE E 1176 745 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TELMISARTAN TELMISARTAN 1179 746 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME BENZOQUINONE BENZOQUINONE 1180 747 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 2-AMINOFLURENE CHEMBL84472 1181 748 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor NINTEDANIB NINTEDANIB 1182 749 YEATS4 8089 TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE hydrochlorothiazide HYDROCHLOROTHIAZIDE 1183 750 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE inhibitor 381118868 BMS-823778 1184 751 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SJ000276790 CHEMBL602922 1185 752 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-156 1186 753 RIPK2 8767 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 315661219 1187 754 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR Tumor necrosis factor alpha (TNF-alpha) inhibitors 24776844,22158445 1188 755 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650167 DENOPAMINE 1189 756 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651589 1190 757 BCAT2 587 ENZYME, TRANSPORTER inhibitor 315661169 1191 758 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR NORDIHYDROGUAIARETIC ACID 2453577 1192 759 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LAROPIPRANT LAROPIPRANT 1193 760 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417031 CHEMBL1333049 1194 761 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 187051794 1195 762 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 340590273 1196 763 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TETRAHYDROAPLYSULPHURIN-1 CHEMBL1077773 19601607 1197 764 GLA 2717 ENZYME, DRUGGABLE GENOME PINDOLOL PINDOLOL 1199 765 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE afatinib AFATINIB 18681783,14990633,16467544,16377102,14990632,18784101,16257339,18003960,25611025,23022519,11255078,19339720,18316547,12648464,22594511 1202 766 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME CENISERTIB CENISERTIB 1203 767 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NGM313 1204 768 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Neu-120 1207 769 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201644 INSULIN ZINC SUSP RECOMBINANT HUMAN 1208 770 PSMD2 5708 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 1209 771 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL1237022 TOCILIZUMAB 1210 772 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE HYDROGEN PEROXIDE 16713429 1211 773 HEBP1 50865 DRUGGABLE GENOME Pyrazino[2,1-a]isoquinolin derivative 3 1212 774 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651403 1214 775 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PHENYLHYDRAZINE PHENYLHYDRAZINE 24262887 1216 776 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-20 1219 777 CAMKK2 10645 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PF-562271 PF-00562271 1220 778 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 249565627 TESEVATINIB 1221 779 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178102317 CHEMBL1908396 1224 780 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ISOTRETINOIN ISOTRETINOIN 1225 781 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE CVBT-141H 1227 782 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PHENYLPROPANOLAMINE PHENYLPROPANOLAMINE 1228 783 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 249565819 1230 784 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200844 METHYLPREDNISOLONE ACETATE 1232 785 DHFR 1719 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201746 PRALATREXATE 1233 786 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565818 1234 787 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor POZIOTINIB POZIOTINIB 1235 788 RAC1 5879 CLINICALLY ACTIONABLE, KINASE, DRUG RESISTANCE VEMURAFENIB VEMURAFENIB 25056119,24265153 1236 789 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME RG7882 1237 790 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE ACRIFLAVINE CHLORIDE ACRIFLAVINE 1239 791 TSC2 7249 CLINICALLY ACTIONABLE, KINASE, TUMOR SUPPRESSOR EVEROLIMUS EVEROLIMUS 23158522,25295501 1241 792 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SJ000111875 CHEMBL590949 1243 793 MAPT 4137 DRUGGABLE GENOME RHEIN RHEIN 1244 794 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565585 UPROSERTIB 1245 795 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE allosteric modulator 310264666 1246 796 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER agomelatine AGOMELATINE 1247 797 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Anisindione ANISINDIONE 1249 798 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR US9073931, E3 1252 799 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZACITIDINE AZACITIDINE 1253 800 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GW7647 GW7647 18162399 1254 801 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BERGAPTEN BERGAPTEN 1255 802 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE LEVONORDEFRIN LEVONORDEFRIN 1256 803 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LAS-34273 ACLIDINIUM BROMIDE 1258 804 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR inhibitor HESPERADIN HESPERADIN 19035792 1259 805 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 10-HYDROXYEVODIAMINE CHEMBL2171812 22867019 1260 806 B4GALNT1 2583 ENZYME antibody DINUTUXIMAB DINUTUXIMAB 1261 807 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CETRIMIDE CETRIMIDE 1265 808 MAPT 4137 DRUGGABLE GENOME BIIB092 GOSURANEMAB 1269 809 HKDC1 80201 DRUGGABLE GENOME, KINASE OXOPURPUREINE OXOPURPUREINE 1270 810 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TAE-684 TAE-684 1271 811 PYGL 5836 DRUGGABLE GENOME, ENZYME dexamethasone DEXAMETHASONE 23007406 1272 812 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CYT-609 20876255 1273 813 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL14762 SELICICLIB 1275 814 SMN1 6606 DRUGGABLE GENOME GNF-PF-3501 CHEMBL581910 1276 815 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 1278 816 MBNL1 4154 DRUGGABLE GENOME MITOXANTRONE MITOXANTRONE 1279 817 TPSAB1 7177 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 318164852 CHEMBL256892 1280 818 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2-(2-AMINOETHYL)ISOTHIOUREA DIHYDROBROMIDE CHEMBL1256182 1281 819 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Rituximab RITUXIMAB 1282 820 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TGFBETA1 9794232 1286 821 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-59 1288 822 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ABT-122 REMTOLUMAB 1289 823 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PTG-100 1290 824 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650378 ILOPROST 1293 825 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CAMPTOTHECIN CAMPTOTHECIN 10839298 1294 826 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME zonisamide ZONISAMIDE 24236482 1295 827 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE idarubicin IDARUBICIN 15564883 1296 828 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Capecitabine CAPECITABINE 1298 829 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHRYSENE CHRYSENE 1299 830 CBX1 10951 NA ATHRAQUINONES A ATHRAQUINONES A 1301 831 ATG5 9474 CLINICALLY ACTIONABLE, TRANSPORTER, ENZYME adalimumab ADALIMUMAB 27096233 1303 832 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody AMG-479 GANITUMAB 1304 833 RTN4 57142 DRUGGABLE GENOME HYPERBARIC OXYGEN 12951059 1306 834 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-34 1309 835 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE FAS LIGAND 10432288 1310 836 PDE3A 5139 ENZYME, DRUGGABLE GENOME 349U85.HCL 1311 837 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PLX7904 26466569,27523909 1317 838 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Indole-based analog 3 1318 839 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DIFLUFENICAN DIFLUFENICAN 1319 840 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE PROTEIN SYNTHESIS INHIBITOR 9844728 1320 841 SMN2 6607 DRUGGABLE GENOME 6-AZAURIDINE 6-AZAURIDINE 1321 842 PRMT3 10196 DRUGGABLE GENOME, METHYL TRANSFERASE, ENZYME inhibitor 310264736 1322 843 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE THYROTROPIN ALFA 1323 844 MAGEA1 4100 NA ARA-C 8749237 1324 845 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE neratinib NERATINIB 18681783,14990633,16467544,16377102,14990632,18784101,16257339,18003960,23022519,11255078,19339720,18316547,12648464,22594511 1325 846 CD74 972 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE MILATUZUMAB MILATUZUMAB 1326 847 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME SHINPTEROCARPIN SHINPTEROCARPIN 20022509 1327 848 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DNDI1417388 CHEMBL1528359 1328 849 CD3D 915 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE NI-0401 FORALUMAB 1329 850 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1521 ZALEPLON 1330 851 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PEMBROLIZUMAB PEMBROLIZUMAB 27903500,27433843 1331 852 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BCMA-CART 1332 853 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-989 CHEMBL583150 1334 854 CBX1 10951 NA METITEPINE METITEPINE 1335 855 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME COXSACKIEVIRUS TYPE A21 1336 856 TGFBR3 7049 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CYTOKINES 16634800 1338 857 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW831090X GW831090X 1339 858 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME STI571 IMATINIB MESYLATE 11439348 1341 859 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 4'-N-BENZOYLSTAUROSPORINE 1342 860 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 660258 CHEMBL259805 1343 861 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME TAE-684 TAE-684 1344 862 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SKF-82526 CHEMBL1161520 1345 863 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BUTORPHANOL BUTORPHANOL 22931300 1348 864 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE LAPATINIB LAPATINIB 1349 865 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NOSCAPINE NOSCAPINE 1351 866 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Filgrastim-SNDZ FILGRASTIM 1352 867 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL484785 CRISABOROLE 1353 868 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE DECANOIC ACID DECANOIC ACID 1355 869 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER BAS 01152706 CHEMBL2002487 1357 870 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200402 AMLODIPINE BESYLATE 1359 871 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 381118806 ACALISIB 1361 872 BAZ2B 29994 NA METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 1363 873 KDM4A 9682 DRUGGABLE GENOME, ENZYME INDAZOLE-3-CARBOXYLICACID CHEMBL502057 1364 874 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FOLFOX REGIMEN 19922504 1365 875 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR [3H]-PHORBOL 12,13-DIBUTYRATE CHEMBL27768 24794745 1367 876 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL1201733 PAZOPANIB HYDROCHLORIDE 1369 877 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Ofatumumab OFATUMUMAB 1370 878 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE VENETOCLAX VENETOCLAX 30725494 1372 879 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME BELINOSTAT BELINOSTAT 26313268 1373 880 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TRIFLUOPERAZINE TRIFLUOPERAZINE 15845548 1374 881 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DICHLOROPHEN DICHLOROPHEN 1375 882 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE SERMS 15576828 1376 883 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 363894234 1378 884 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE GNF-PF-67 CHEMBL578512 1380 885 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 384403666 1381 886 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME P-PHENYLENEDIAMINE CHEMBL403741 1384 887 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 249565869 CEP-11981 1385 888 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 328083505 1387 889 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE lonafarnib LONAFARNIB 26033044 1388 890 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MRS-1523 CHEMBL111545 1389 891 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR gemcitabine GEMCITABINE 1390 892 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103781 KETOTIFEN 1391 893 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR Belimumab BELIMUMAB 1392 894 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME CD38 and BCMA CAR-T Cells 1393 895 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Thiazole-fused cycloalkyl carboxamide derivative 1 1394 896 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3545194 LGH-447 1395 897 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL SSR-125329A 1396 898 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME SJ000001516 CHEMBL592316 1397 899 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR 1-hydroxyl-3,5-bis(4-hydroxylstyryl)benzene derivative 1 1398 900 UGT2B7 7364 DRUGGABLE GENOME methadone METHADONE 17178267,22676193 1399 901 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Pyridic ketone derivative 1 1400 902 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Gefitinib GEFITINIB 15696205,27338794,25870145 1401 903 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ANDROSTENEDIONE ANDROSTENEDIONE 1402 904 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MODAFINIL MODAFINIL 22931300 1403 905 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PERPHENAZINE PERPHENAZINE 1404 906 UGT1A6 54578 ENZYME, DRUGGABLE GENOME daunorubicin DAUNORUBICIN 1405 907 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL1201837 ECALLANTIDE 1406 908 TSPO 706 DRUGGABLE GENOME ZOPICLONE ZOPICLONE 1407 909 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545063 OSIMERTINIB MESYLATE 1409 910 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 249565748 1410 911 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor BYL719 ALPELISIB 1412 912 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME EPIPODOPHYLLOTOXIN 4-(MORPHOLINE)CARBAMATE CHEMBL1773343 21489802 1413 913 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE lithium LITHIUM 21047205,24885933 1414 914 ALB 213 TRANSPORTER, DRUGGABLE GENOME Gadofosveset GADOFOSVESET 1418 915 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor DACOMITINIB DACOMITINIB 1419 916 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1201007 HYDROXYZINE HYDROCHLORIDE 1420 917 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR VINCRISTINE VINCRISTINE 15569250 1421 918 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 178102476 1422 919 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651527 1423 920 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LEVOTHYROXINE LEVOTHYROXINE 1425 921 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ACRISORCIN ACRISORCIN 1426 922 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE AR-A014418 CHEMBL259850 1428 923 GJB3 2707 TRANSPORTER, ION CHANNEL inhibitor 178101095 OCTANOL 1429 924 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PD-332991 1430 925 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CLIOQUINOL CLIOQUINOL 1431 926 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE ETHANOL ALCOHOL 15894672 1432 927 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 5,7-DIMETHOXYISOFLAVONE 5,7-DIMETHOXYISOFLAVONE 1433 928 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CGM097 CGM-097 27659046 1436 929 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE SP-600125 SP-600125 1437 930 RBP4 5950 DRUGGABLE GENOME US8586571, 36 1439 931 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME IRX4204 1441 932 MAPT 4137 DRUGGABLE GENOME PYRANTEL PAMOATE PYRANTEL PAMOATE 1442 933 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL426084 SAMIDORPHAN 1443 934 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-13 1444 935 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 363894197 CT-7001 1445 936 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME terbinafine TERBINAFINE 1447 937 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HYDRAMETHYLNON HYDRAMETHYLNON 1449 938 SSRP1 6749 KINASE, DNA REPAIR CBL0102 1451 939 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650435 1452 940 NDUFB6 4712 ENZYME inhibitor CHEMBL3545135 NV-128 1453 941 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL3545351 AV-101 1454 942 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Exemestane EXEMESTANE 1455 943 PDE7B 27115 DRUGGABLE GENOME, ENZYME DYPHYLLINE DYPHYLLINE 1456 944 MAOB 4129 DRUGGABLE GENOME, ENZYME Phenelzine PHENELZINE 1457 945 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Pyrido[4,3-d]pyrimidin-5(6H)-one derivative 1 1458 946 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SOY PROTEIN ISOLATE 17182792 1461 947 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER OLEOYL DOPAMINE OLEOYL DOPAMINE 1462 948 RIPK2 8767 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PD-169316 PD-169316 18408713 1463 949 CSNK1E 1454 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 310264697 UMBRALISIB 1465 950 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BD-1008 CHEMBL20377 1466 951 HMGCR 3156 ENZYME, DRUGGABLE GENOME Crestor/TriLipix 1467 952 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL101 PHENYLBUTAZONE 1468 953 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 178103678 1470 954 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 381744997 REPOTRECTINIB 1472 955 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Nivolumab NIVOLUMAB 1475 956 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE LY-2584702 LY-2584702 1476 957 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NILUTAMIDE NILUTAMIDE 1478 958 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR MD1003 1479 959 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME PURPURIN PURPURIN 1480 960 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR PANITUMUMAB PANITUMUMAB 31227518 1481 961 POLK 51426 DNA REPAIR, ENZYME PYROGALLOL RED PYROGALLOL RED 1482 962 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BI-87E7 CHEMBL523200 1483 963 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-AMINO-ANTHRAQUINONE CHEMBL84685 1484 964 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME blocker 135652741 1485 965 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 178102344 TOZASERTIB 1486 966 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR inhibitor 178103592 1488 967 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROPANTHELINE BROMIDE PROPANTHELINE BROMIDE 1489 968 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 381118841 1490 969 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME PACLITAXEL PACLITAXEL 1491 970 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME MEK INHIBITOR PD0325901 26544513 1492 971 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CANDIDIN CANDIDIN 1493 972 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ALPELISIB ALPELISIB 31091374,24608574 1494 973 NQO2 4835 DRUGGABLE GENOME, ENZYME NSC-640556 CHEMBL1983317 21074425 1495 974 MAPT 4137 DRUGGABLE GENOME MMV007396 CHEMBL582286 1496 975 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor SB939 1498 976 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME SULFURETIN SULFURETIN 1499 977 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIS(2,3-DIBROMOPROPYL)PHOSPHATE TRIS(2,3-DIBROMOPROPYL)PHOSPHATE 1500 978 HSPA8 3312 TUMOR SUPPRESSOR NSC-119910 CHEMBL487046 1504 979 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME BMS-911543 BMS-911543 1505 980 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PMID27774824-Compound-Figure9Example2up 1506 981 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PROCHLORPERAZINE PROCHLORPERAZINE 1508 982 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL1200373 1509 983 KDM4A 9682 DRUGGABLE GENOME, ENZYME ALTENUSIN ALTENUSIN 1510 984 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565867 1511 985 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIFENOCONAZOLE DIFENOCONAZOLE 1512 986 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ECONAZOLE NITRATE ECONAZOLE NITRATE 1513 987 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Flufenamic Acid 1515 988 ADSS2 159 ENZYME ALANOSINE ALANOSINE 7825060 1516 989 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR GTx-758 GTX-758 1518 990 FBXW7 55294 DNA REPAIR, CLINICALLY ACTIONABLE Docetaxel DOCETAXEL 23274910 1519 991 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist,antagonist 135651233 TAMOXIFEN 1521 992 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME muraglitazar MURAGLITAZAR 18794727 1522 993 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID29757691-Compound-7 1523 994 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-840 CHEMBL601605 1524 995 BCL6 604 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE FENRETINIDE FENRETINIDE 11027625 1526 996 POLK 51426 DNA REPAIR, ENZYME AG-99 CHEMBL296407 1527 997 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CLEMASTINE CLEMASTINE 22931300 1528 998 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ZM-449829 CHEMBL154580 1529 999 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME METHOXY POLYETHYLENE GLYCOL-EPOETIN BETA 1530 1000 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME 3-METHOXYCATECHOL 3-METHOXYCATECHOL 1533 1001 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SANGUINARIUM CHLORIDE SANGUINARIUM CHLORIDE 1534 1002 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL EVT-201 1535 1003 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TAE-684 TAE-684 1536 1004 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING RESMINOSTAT RESMINOSTAT 1537 1005 MAPT 4137 DRUGGABLE GENOME CARBIDOPA CARBIDOPA 1541 1006 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SOTRASTAURIN SOTRASTAURIN 1543 1007 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME MUC-1 CART cell immunotherapy 1545 1008 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 887167 CHEMBL260342 1547 1009 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME FILGRAMSTIM 1550 1010 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME DOVITINIB DOVITINIB 28759044 1553 1011 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE LINIFANIB LINIFANIB 1554 1012 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR TPI-1020 1555 1013 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME SCOULERINE SCOULERINE 1557 1014 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME (-)-ROLIPRAM (-)-ROLIPRAM 1558 1015 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1200447 1559 1016 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Linsitinib LINSITINIB 27196766 1561 1017 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE GREEN TEA EXTRACT 17616136 1562 1018 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE CENISERTIB CENISERTIB 1563 1019 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HALOPROGIN HALOPROGIN 1565 1020 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Modafinil MODAFINIL 1566 1021 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ROCURONIUM ROCURONIUM 1568 1022 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-62 1570 1023 TUBB4B 10383 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 1571 1024 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RO-410960 CHEMBL1256291 1572 1025 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE PD-0166285 PD-0166285 1573 1026 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE DIAZEPAM DIAZEPAM 15148255 1574 1027 UGT1A6 54578 ENZYME, DRUGGABLE GENOME febuxostat FEBUXOSTAT 27798726 1575 1028 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE CAPECITABINE CAPECITABINE 1576 1029 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TCMDC-123828 CHEMBL588804 1578 1030 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TA-2005 CARMOTEROL 1580 1031 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor BAY80-6946 COPANLISIB 1581 1032 MAPT 4137 DRUGGABLE GENOME DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 1582 1033 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BUTHIONINE SULFOXIMINE BUTHIONINE SULFOXIMINE 1583 1034 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE inhibitor 249565809 1584 1035 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201754 RUFINAMIDE 1585 1036 IDS 3423 ENZYME, DRUGGABLE GENOME Recombinant human iduronate-2-sulfatase 1586 1037 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR allosteric modulator 363894205 TAK-733 1587 1038 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME Rosuvastatin ROSUVASTATIN 1588 1039 TNC 3371 DRUGGABLE GENOME, FIBRINOGEN CHEMBL2109584 F16SIP 131I 1589 1040 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR CHRYSIN CHRYSIN 19592245 1590 1041 CIP2A 57650 NA GEMCITABINE GEMCITABINE 26894380 1591 1042 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178104007 LEVOMILNACIPRAN 1592 1043 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL HALAZEPAM HALAZEPAM 1594 1044 MPHOSPH8 54737 NA TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 1595 1045 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Carbamide derivative 17 1597 1046 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 1598 1047 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME NSC-8186 CHEMBL122355 1600 1048 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-408124 CHEMBL1334465 1601 1049 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE PAZOPANIB PAZOPANIB 1602 1050 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE NVP-BEZ242 1603 1051 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Biphenyl derivative 2 1604 1052 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX MITOXANTRONE MITOXANTRONE 1607 1053 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Imidazo bicyclic iminium derivative 4 1608 1054 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102342 FEDRATINIB 1609 1055 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR ZEARALENONE ZEARALENONE 1610 1056 SERPINA5 5104 PROTEASE INHIBITOR, ENZYME, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE gemcitabine GEMCITABINE 31616045 1613 1057 ODC1 4953 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201037 EFLORNITHINE HYDROCHLORIDE 1614 1058 CBX1 10951 NA CAPSAZEPINE CAPSAZEPINE 1615 1059 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TTC-352 1616 1060 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SOTRASTAURIN SOTRASTAURIN 1617 1061 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 propofol PROPOFOL 24891132 1618 1062 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1318477 CHEMBL428064 1619 1063 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ERGOTAMINE ERGOTAMINE 1620 1064 ALOX15 246 ENZYME, DRUGGABLE GENOME inhibitor 381744944 1621 1065 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IMIPRAMINE IMIPRAMINE 1624 1066 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PLX8394 PLX8394 27834212,24422853 1625 1067 RAPGEF3 10411 ENZYME CRYPTOTANSHINONE CRYPTOTANSHINONE 1628 1068 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME CVX-060 1629 1069 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ZSTK474 26137449 1632 1070 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE BIBX-1382 FALNIDAMOL 1633 1071 IL1B 3553 KINASE, DRUGGABLE GENOME VERAPAMIL VERAPAMIL 2686646 1636 1072 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TESMILIFENE TESMILIFENE 1638 1073 CEL 1056 CELL SURFACE, DRUGGABLE GENOME, ENZYME Bucelipase alfa 1639 1074 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE OSI-7904L OSI-7904 1640 1075 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME inhibitor SORAFENIB TOSYLATE 1643 1076 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-3641 CHEMBL599098 1644 1077 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE VPI-2690B 1645 1078 NCAM1 4684 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CART-56 cells 1646 1079 PDE4A 5141 DRUGGABLE GENOME, ENZYME AVE-8112 24343458 1647 1080 BAZ2B 29994 NA GNF-PF-5381 CHEMBL578109 1648 1081 GMNN 51053 DRUGGABLE GENOME DNDI1417973 CHEMBL1572415 1650 1082 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE SORAFENIB SORAFENIB 1651 1083 TLR7 51284 DRUGGABLE GENOME agonist CHEMBL1282 IMIQUIMOD 1653 1084 TUBB2A 7280 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 1654 1085 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE JNJ-10311795 CHEMBL374027 1655 1086 PTGS2 5743 DRUGGABLE GENOME, ENZYME NEPAFENAC NEPAFENAC 1656 1087 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 348353661 1657 1088 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SORAFENIB SORAFENIB 1658 1089 NDUFB9 4715 ENZYME inhibitor CHEMBL3545135 NV-128 1659 1090 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DANTHRON DANTHRON 1662 1091 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102320 ENZASTAURIN 1663 1092 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Lucitanib LUCITANIB 27126994 1664 1093 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE NIFEDIPINE NIFEDIPINE 10051745 1665 1094 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL124660 TANDUTINIB 1666 1095 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IOXYNIL IOXYNIL 1667 1096 CRBN 51185 ENZYME, DRUG RESISTANCE inhibitor CHEMBL43452 POMALIDOMIDE 1669 1097 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR HYDROCORTAMATE HYDROCORTAMATE 1671 1098 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR R-BACLOFEN 1675 1099 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TLC-388 1678 1100 PSMC2 5701 PROTEASE, TRANSCRIPTION FACTOR inhibitor CHEMBL325041 BORTEZOMIB 1679 1101 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure3-Lycojaponicumin C 1680 1102 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 18 1681 1103 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200814 ACETAZOLAMIDE SODIUM 1682 1104 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2008005457 1684 1105 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135652435 RELAXIN 1685 1106 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TAE-684 TAE-684 1686 1107 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-209931 CHEMBL472656 1687 1108 CTNNBL1 56259 NA Beta-acetyldigoxin ACETYLDIGOXIN 1688 1109 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME RAS INHIBITOR 16985068 1691 1110 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135650308 1693 1111 GMNN 51053 DRUGGABLE GENOME NISOLDIPINE NISOLDIPINE 1694 1112 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE SORAFENIB SORAFENIB 1695 1113 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 318164808 SIPONIMOD 1696 1114 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Aminotriazolopyridine derivative 1 1697 1115 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME ANTIBIOTICS 2571317 1698 1116 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-1872 CHEMBL600103 1699 1117 KDM4A 9682 DRUGGABLE GENOME, ENZYME EUPAFOLIN EUPAFOLIN 1700 1118 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE acetaminophen / tramadol 1702 1119 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CBT-101 1705 1120 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PYRITHIONE ZINC PYRITHIONE ZINC 1706 1121 TUBB3 10381 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 1707 1122 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 178102513 PONATINIB 1708 1123 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME INSULIN INSULIN 10614629 1709 1124 PSMA2 5683 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL3545432 IXAZOMIB CITRATE 1710 1125 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649684 1711 1126 NQO2 4835 DRUGGABLE GENOME, ENZYME NSC-640584 CHEMBL476968 21074425 1712 1127 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PAZOPANIB PAZOPANIB 24625776 1713 1128 DNER 92737 NA Pyrimido-indole derivative 1 1714 1129 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR N-(3-OXODODECANOYL)HOMOSERINELACTONE CHEMBL8483 18566250 1715 1130 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Tamsulosin TAMSULOSIN 1718 1131 POLB 5423 DNA REPAIR, DRUGGABLE GENOME 3,8'-BIAPIGENIN CHEMBL515252 1720 1132 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ELLIPTECINE ELLIPTECINE 1721 1133 FAAH 2166 ENZYME, DRUGGABLE GENOME Heteroaryl-substituted urea derivative 1 1723 1134 TMEM97 27346 NA ANAVEX 1007 1724 1135 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102207 1725 1136 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TYRPHOSTIN 47 TYRPHOSTIN 47 1726 1137 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Vemurafenib VEMURAFENIB 1728 1138 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 1730 1139 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR COCAINE COCAINE 1731 1140 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652579 1732 1141 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CYCLOSPORINE CYCLOSPORINE 22931300 1733 1142 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME IRIGENOL IRIGENOL 1734 1143 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE 7-O-ACETYLAFROMOSIN CHEMBL446567 1735 1144 SOST 50964 DRUGGABLE GENOME BPS-804 SETRUSUMAB 1736 1145 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545196 PD-0166285 1739 1146 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051807 SCRIPTAID 1740 1147 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565808 1741 1148 SLC16A5 9121 DRUGGABLE GENOME, TRANSPORTER cisplatin CISPLATIN 31666714 1742 1149 TUBB3 10381 DRUGGABLE GENOME CHEMBL2304041 SAGOPILONE 1743 1150 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME allosteric modulator 223365961 COBIMETINIB 1744 1151 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Pimasertib PIMASERTIB 23629727 1746 1152 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DNDI1417085 CHEMBL1522984 1747 1153 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BELINOSTAT BELINOSTAT 25937017 1748 1154 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor ALISERTIB ALISERTIB 1751 1155 AQP1 358 ION CHANNEL, DRUGGABLE GENOME Vitamin C 1752 1156 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DNDI1340257 CHEMBL1702181 1754 1157 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1025 ISOFLUROPHATE 1755 1158 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CLOFOCTOL CLOFOCTOL 1756 1159 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 N-HISTIDYL-2-AMINONAPHTHALENE (BETANA) N-HISTIDYL-2-AMINONAPHTHALENE (BETANA) 1759 1160 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME chlorocresol CHLOROCRESOL 29344738,25086907 1761 1161 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651470 DESMOSTEROL 1763 1162 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRONE ESTRONE 1764 1163 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE MEK-1/MEKK-1 INHIBITOR E6201 32142668 1766 1164 KDM4A 9682 DRUGGABLE GENOME, ENZYME PYRIDINE-2,4-DICARBOXYLIC ACID CHEMBL316034 1767 1165 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME 135650848 PRAVASTATIN 1768 1166 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME ACOTIAMIDE ACOTIAMIDE 1769 1167 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201027 GLYCOPYRROLATE 1770 1168 DDX5 1655 CLINICALLY ACTIONABLE RX-5902 1772 1169 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TEBUFENPYRAD TEBUFENPYRAD 1773 1170 CFLAR 8837 DRUG RESISTANCE, DRUGGABLE GENOME, PROTEASE BAY-11-7085 BAY-11-7085 22326395 1775 1171 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME L-4-THIOPROLINE CHEMBL1800368 21665470 1776 1172 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME vemurafenib VEMURAFENIB 1777 1173 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME ponatinib PONATINIB 1778 1174 SV2A 9900 DRUGGABLE GENOME, TRANSPORTER Brivaracetam BRIVARACETAM 1781 1175 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 16636344,24897286,12181437,18221820 1782 1176 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135650056 CARBACYCLIN 1783 1177 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR mercaptopurine MERCAPTOPURINE 24141364 1784 1178 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-9 1785 1179 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DEXAMETHASONE DIPROPIONATE DEXAMETHASONE DIPROPIONATE 1787 1180 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Lanreotide acetate 1788 1181 MICA 100507436 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE HSP70 17911639 1789 1182 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650554 EGLUMEGAD 1790 1183 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE SULFURETIN SULFURETIN 1791 1184 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL495727 AT-9283 1794 1185 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor PF-03814735 PF-03814735 1795 1186 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR VG-101 22114467 1797 1187 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME LEPIRUDIN LEPIRUDIN 1798 1188 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME CARFILZOMIB CARFILZOMIB 24524217 1799 1189 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME AST-487 AST-487 1800 1190 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Pankomab-GEX 1801 1191 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AM580 CHEMBL69367 1802 1192 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CYTARABINE HYDROCHLORIDE CYTARABINE HYDROCHLORIDE 1803 1193 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE M4344 1804 1194 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE N,N'-DIPHENYL-P-PHENYLENEDIAMINE N,N'-DIPHENYL-P-PHENYLENEDIAMINE 1805 1195 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME TAE-684 TAE-684 1806 1196 ADGRV1 84059 G PROTEIN COUPLED RECEPTOR, TRANSPORTER, CELL SURFACE, KINASE, DRUGGABLE GENOME opioids 1808 1197 POLI 11201 DNA REPAIR RHEIN RHEIN 1810 1198 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8921389, 22 1811 1199 PIP4K2A 5305 ENZYME, KINASE SJ000201788 CHEMBL602923 1813 1200 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME TGX-221 24251790 1814 1201 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME ITRACONAZOLE ITRACONAZOLE 17518356 1815 1202 KDM4A 9682 DRUGGABLE GENOME, ENZYME 3,8'-BIAPIGENIN CHEMBL515252 1817 1203 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GlyT1 PET radiotracers 21253021 1820 1204 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE tamoxifen TAMOXIFEN 1823 1205 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE SOTRASTAURIN ACETATE 24141786 1825 1206 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ETOPOSIDE ETOPOSIDE 23999041 1826 1207 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-11437 CHEMBL1814509 1827 1208 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE (S)-VERAPAMIL (S)-VERAPAMIL 1828 1209 KAT2B 8850 ENZYME, DRUGGABLE GENOME amphetamine AMPHETAMINE 1829 1210 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 249565866 1830 1211 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135650978 SALMETEROL 1832 1212 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651366 ZOLMITRIPTAN 1835 1213 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-3350 CHEMBL600747 1837 1214 MCOLN1 57192 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER opioids 31362332 1838 1215 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CYPRODINIL CYPRODINIL 1839 1216 KLRD1 3824 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME adalimumab ADALIMUMAB 26453102 1840 1217 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme1WO2011135259 1841 1218 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor 404859154 1842 1219 RAB9A 9367 ENZYME, DRUGGABLE GENOME 7-HYDROXY ISOFLAVONE 7-HYDROXY ISOFLAVONE 1844 1220 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME BMS-387032 BMS-387032 1846 1221 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Almogran 1848 1222 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor BGJ398 INFIGRATINIB 1853 1223 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PI-103 PI-103 1856 1224 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ERYTHROPOIETIN EPOETIN BETA 16707229 1857 1225 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DNDI1417601 CHEMBL1503729 1860 1226 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE EP-51216 1864 1227 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME LEVONORDEFRIN LEVONORDEFRIN 1866 1228 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1184 ACETYLCHOLINE CHLORIDE 1867 1229 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ARZOXIFENE ARZOXIFENE 1868 1230 IDO2 169355 ENZYME 2,3-diamino-benzo[b]thiophene derivative 4 1869 1231 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE INDAPAMIDE INDAPAMIDE 1870 1232 PDE4B 5142 DRUGGABLE GENOME, ENZYME APREMILAST APREMILAST 1871 1233 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Ribavirin RIBAVIRIN 1872 1234 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RAUWOLFIA SERPENTINA RAUWOLFIA SERPENTINA 1874 1235 USP1 7398 DNA REPAIR, PROTEASE, ENZYME BENZIODARONE BENZIODARONE 1876 1236 ATAD2 29028 NUCLEAR HORMONE RECEPTOR, ENZYME inhibitor 252827390 1879 1237 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 223366125 TASELISIB 1881 1238 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 178103154 1882 1239 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME MLN-9708 IXAZOMIB CITRATE 1884 1240 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE olanzapine OLANZAPINE 24725652 1885 1241 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor ROMIDEPSIN ROMIDEPSIN 1888 1242 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TESTOSTERONE TESTOSTERONE 1890 1243 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MK2206 MK-2206 26676756,25931518,26725216,22025163,27480147 1891 1244 PSORS1C1 170679 NA carboplatin CARBOPLATIN 31616045 1892 1245 RGS4 5999 DRUGGABLE GENOME D-TRYPTOPHAN D-TRYPTOPHAN 1893 1246 TFF2 7032 DRUGGABLE GENOME HORMONES 16359755 1894 1247 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TUBERCIDIN TUBERCIDIN 1896 1248 POLI 11201 DNA REPAIR TETRAIDOFLUORESCEIN TETRAIDOFLUORESCEIN 1900 1249 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE GENTIAN VIOLET GENTIAN VIOLET 1902 1250 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor PELITINIB PELITINIB 1903 1251 UBA3 9039 TUMOR SUPPRESSOR, ENZYME inhibitor CHEMBL1231160 PEVONEDISTAT 1904 1252 TOP2B 7155 DRUGGABLE GENOME, ENZYME LYCOBETAINE LYCOBETAINE 23266176 1905 1253 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ALLITRIDIN ALLITRIDIN 1907 1254 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652751 1908 1255 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrazolo[4,3-c]pyridine derivative 2 1909 1256 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR Sirukumab SIRUKUMAB 1910 1257 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GSK9772 CHEMBL493241 18800767,22873709 1911 1258 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE Afuresertib AFURESERTIB 1912 1259 TNFRSF11A 8792 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE Pyrazolones 26398624 1913 1260 APRT 353 ENZYME, DRUGGABLE GENOME TPA ALTEPLASE 6933001 1914 1261 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 249565693 1915 1262 TXN 7295 DRUGGABLE GENOME, THIOREDOXIN GAMBOGIC ACID GAMBOGIC ACID 22663155 1916 1263 GMNN 51053 DRUGGABLE GENOME MITONAFIDE MITONAFIDE 1917 1264 POLI 11201 DNA REPAIR (-)-DICENTRINE CHEMBL478754 1920 1265 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702240 PEMIGATINIB 1921 1266 RAC1 5879 CLINICALLY ACTIONABLE, KINASE, DRUG RESISTANCE ZU-0073945 CHEMBL563777 19527032 1922 1267 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE QVA-149 1923 1268 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TREPROSTINIL TREPROSTINIL 1925 1269 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ICATIBANT ICATIBANT 1927 1270 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker 135650185 DILTIAZEM 1928 1271 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR METHOXSALEN METHOXSALEN 1929 1272 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102513 PONATINIB 1930 1273 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GSK-269962A GSK-269962A 1931 1274 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CYC-116 CYC-116 1932 1275 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME FARLETUZUMAB FARLETUZUMAB 1934 1276 CBLC 23624 CLINICALLY ACTIONABLE, KINASE, ENZYME Olaparib OLAPARIB 25883215 1935 1277 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL1645462 AC-480 1937 1278 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GRACILIN J GRACILIN J 19601607 1939 1279 ERCC4 2072 CLINICALLY ACTIONABLE, DNA REPAIR Platinum compounds 25069034 1941 1280 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CYCLOSPORINE CYCLOSPORINE 17852453 1942 1281 SMARCB1 6598 CLINICALLY ACTIONABLE radiotherapy 23190500 1943 1282 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUOXYMESTERONE FLUOXYMESTERONE 1944 1283 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ARACHIDONYL TRIFLUOROMETHYLKETONE ARACHIDONYL TRIFLUOROMETHYLKETONE 1945 1284 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CTX-1 26883273 1947 1285 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200601 NARATRIPTAN HYDROCHLORIDE 1948 1286 NOS1 4842 DRUGGABLE GENOME, ENZYME ibuprofen IBUPROFEN 25502615 1949 1287 TNFRSF4 7293 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PF-04518600 IVUXOLIMAB 1950 1288 BAZ2B 29994 NA BAS 01152706 CHEMBL2002487 1951 1289 DHODH 1723 DRUGGABLE GENOME, ENZYME LEFLUNOMIDE LEFLUNOMIDE 1952 1290 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102585 DOVITINIB 1956 1291 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL538943 VINORELBINE TARTRATE 1958 1292 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 53801005 1959 1293 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 381744939 1960 1294 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103096 APRATASTAT 1961 1295 GC 2638 DRUGGABLE GENOME inhibitor CHEMBL712 ANISINDIONE 1963 1296 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GNF-PF-2893 CHEMBL312032 1964 1297 LEPR 3953 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME antipsychotics 21510767 1967 1298 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417701 CHEMBL1326164 1969 1299 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GOSSYPETIN-8-GLUCOSIDE CHEMBL402915 18063365 1970 1300 SH2B1 25970 KINASE lithium LITHIUM 28694205 1971 1301 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 249565620 DANUSERTIB 1973 1302 F5 2153 DRUGGABLE GENOME drotrecogin alfa 15118525 1974 1303 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE Salicyclic acid 1975 1304 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Anisodine 1976 1305 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651391 1977 1306 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GNF-PF-4029 CHEMBL596633 1979 1307 NUAK1 9891 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 310264738 CERDULATINIB 1981 1308 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1370561 AMINOPHYLLINE 1983 1309 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AC480 AC-480 1985 1310 GNL3 26354 NA cyclophosphamide CYCLOPHOSPHAMIDE 1986 1311 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-123516 CHEMBL547304 1987 1312 NOS1 4842 DRUGGABLE GENOME, ENZYME BENZODIAZEPINE BENZODIAZEPINE 15136793 1988 1313 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE DNDI1417467 CHEMBL1997335 1989 1314 KDM1B 221656 DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING, ENZYME Tarnylcypromine derivative 3 1990 1315 RAB9A 9367 ENZYME, DRUGGABLE GENOME LASSBIO-123 CHEMBL573111 1993 1316 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR QUESTIOMYCIN B QUESTIOMYCIN B 1995 1317 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Oxaliplatin OXALIPLATIN 24100628 1996 1318 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER daptomycin DAPTOMYCIN 25239468 1997 1319 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME TRIAZOLAM TRIAZOLAM 22137933 1998 1320 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE sorafenib SORAFENIB 20124951,28362716 1999 1321 EGLN2 112398 ENZYME, DRUGGABLE GENOME BAY-85-3934 2000 1322 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 187051807 SCRIPTAID 2004 1323 TNFRSF14 8764 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME 178101757 2007 1324 ENPP2 5168 ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 315661229 2009 1325 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHOLECALCIFEROL CHOLECALCIFEROL 2011 1326 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 178101953 2012 1327 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565780 2016 1328 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 2017 1329 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL957 BOSENTAN 2018 1330 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME BEXAROTENE BEXAROTENE 2025 1331 CA12 771 DRUGGABLE GENOME Salicyclic acid 2026 1332 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Tricyclic compound 11 2029 1333 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE ALENDRONATE ALENDRONIC ACID 11984068 2031 1334 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHENELZINE SULFATE PHENELZINE SULFATE 2032 1335 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SULFAPHENAZOLE SULFAPHENAZOLE 2033 1336 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 310264771 NEOSTIGMINE 2034 1337 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR DACTOLISIB DACTOLISIB 2035 1338 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME SURAMIN HEXASODIUM SURAMIN HEXASODIUM 2036 1339 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor 385612188 2038 1340 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MEGESTROL ACETATE MEGESTROL ACETATE 2039 1341 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME berberine BERBERINE 21647174 2042 1342 DNER 92737 NA FT-1101 2044 1343 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR VK-2809 2045 1344 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ALLOPURINOL ALLOPURINOL 22931300 2046 1345 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE IPCONAZOLE IPCONAZOLE 2047 1346 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PD-145065 2048 1347 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE I-CBP112 26552700 2050 1348 MPHOSPH8 54737 NA EBSELEN EBSELEN 2052 1349 KDM4A 9682 DRUGGABLE GENOME, ENZYME RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 2053 1350 PDE4A 5141 DRUGGABLE GENOME, ENZYME Enprofylline ENPROFYLLINE 2054 1351 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Salicylic acid derivative 3 2055 1352 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CLONAZEPAM CLONAZEPAM 2056 1353 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651469 2057 1354 MAPT 4137 DRUGGABLE GENOME JUGLONE JUGLONE 2058 1355 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor PCI-24781 ABEXINOSTAT 2059 1356 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BAS-8770931 CHEMBL515495 2060 1357 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NSC-117079 CHEMBL471225 2061 1358 HPRT1 3251 DRUGGABLE GENOME, ENZYME NITROSOUREAS 3328039 2062 1359 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR TESTOSTERONE TESTOSTERONE 19883083 2063 1360 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Trilaciclib TRILACICLIB 26826116 2065 1361 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME RG-1530 RG-1530 2066 1362 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-18 2067 1363 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 178100865 CHEMBL597997 2068 1364 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE DACOMITINIB DACOMITINIB 26768165,28958502,21430269,18089823 2069 1365 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR simvastatin SIMVASTATIN 23930676,24598718,23252946 2071 1366 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME GSK2126458 OMIPALISIB 22389471 2073 1367 NOX1 27035 ION CHANNEL, ENZYME, TRANSPORTER, DRUGGABLE GENOME inhibitor 363894229 2074 1368 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-221466 CHEMBL95502 2075 1369 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178101423 2077 1370 HSF1 3297 TRANSCRIPTION FACTOR, DNA REPAIR QUERCETIN QUERCETIN 19296652 2079 1371 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-1211 CHEMBL600968 2080 1372 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Imidazo cyclohexylamine derivative 3 2081 1373 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ZM-336372 CHEMBL186526 2082 1374 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL1471 APREPITANT 2083 1375 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME STICTIC ACID STICTIC ACID 2084 1376 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650349 HEXOCYCLIUM 2085 1377 DPP8 54878 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103150 2086 1378 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME INU-152 28645859 2087 1379 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL1200641 CISATRACURIUM BESYLATE 2089 1380 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME METHOXSALEN METHOXSALEN 2090 1381 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME AZD-1152-HQPA AZD-1152-HQPA 2094 1382 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125653 CHEMBL580918 2095 1383 TUBB2B 347733 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 2096 1384 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEXAMETHASONE DEXAMETHASONE 10867026 2097 1385 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ZERANOL ZERANOL 2101 1386 HTT 3064 DRUGGABLE GENOME GNF-PF-67 CHEMBL578512 2102 1387 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DISULFIRAM DISULFIRAM 2103 1388 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 384403680 2104 1389 ALOX15 246 ENZYME, DRUGGABLE GENOME FEXOFENADINE HYDROCHLORIDE FEXOFENADINE HYDROCHLORIDE 2105 1390 UGT1A10 54575 DRUGGABLE GENOME, ENZYME ANTINEOPLASTIC AGENT 8689427 2106 1391 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 178102290 AT-7519 2109 1392 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HALOPERIDOL HALOPERIDOL 2110 1393 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TCMDC-125543 CHEMBL546170 2111 1394 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565579 APITOLISIB 2114 1395 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME REVERSETRIIODOTHYRONINE REVERSETRIIODOTHYRONINE 2115 1396 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-321 CHEMBL581044 2116 1397 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 11 2117 1398 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ARACHIDONIC ACID ARACHIDONIC ACID 2120 1399 E2F1 1869 TRANSCRIPTION FACTOR GP-120 12775414 2121 1400 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102592 FASCAPLYSIN 2122 1401 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL112 ACETAMINOPHEN 2123 1402 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TCMDC-125580 CHEMBL528807 2124 1403 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR OSPEMIFENE OSPEMIFENE 2129 1404 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE 2,3-DIDEOXYADENOSINE 3496090 2131 1405 PGF 5228 GROWTH FACTOR, DRUGGABLE GENOME SFLT-01 2132 1406 BCHE 590 DRUGGABLE GENOME, ENZYME rivastigmine RIVASTIGMINE 18780301,25376930,17047484,12668920 2133 1407 CALCB 797 DRUGGABLE GENOME inhibitor CHEMBL3833320 EPTINEZUMAB 2134 1408 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NALIDIXIC ACID NALIDIXIC ACID 2137 1409 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor AXITINIB AXITINIB 2138 1410 HTT 3064 DRUGGABLE GENOME GNF-PF-2947 CHEMBL581677 2139 1411 PDE10A 10846 ENZYME, DRUGGABLE GENOME PMID27321640-Compound-58 2140 1412 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR selective beta-2-adrenoreceptor agonists 15564877,16325050,11753577 2141 1413 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PROGESTERONE PROGESTERONE 2142 1414 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BIFONAZOLE BIFONAZOLE 2143 1415 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ENTRECTINIB ENTRECTINIB 2145 1416 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME quetiapine QUETIAPINE 29472872,16871470 2147 1417 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME PMID25399719-Compound-17 2153 1418 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GLUTARAL GLUTARAL 2154 1419 TAB2 23118 KINASE, DRUGGABLE GENOME gefitinib GEFITINIB 31664190 2157 1420 LAMC2 3918 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 2158 1421 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor PWT33597 2160 1422 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME U0126 18794803 2161 1423 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3544927 L-21649 2162 1424 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ZOLMITRIPTAN ZOLMITRIPTAN 2163 1425 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 315661321 UPADACITINIB 2167 1426 HSPB1 3315 DRUGGABLE GENOME DIFFERENTIATION AGENTS 8065161 2168 1427 TBX2 6909 TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX atenolol ATENOLOL 31327267 2169 1428 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-P4 2171 1429 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE 178101360 2172 1430 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHLORPYRIFOS CHLORPYRIFOS 2176 1431 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME activator 178101107 2178 1432 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Palbociclib PALBOCICLIB 2179 1433 TRPC4 7223 ION CHANNEL, KINASE, DRUGGABLE GENOME, CELL SURFACE blocker 381744969 2181 1434 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE US9156852, 105 2182 1435 POLI 11201 DNA REPAIR SCLEROTIORIN SCLEROTIORIN 2183 1436 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL585902 AMG-548 2184 1437 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR allosteric modulator 249565604 BINIMETINIB 2185 1438 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE CYC116 2186 1439 TMEM97 27346 NA N-substituted 9-azabicyclo[3.3.1]nonan-3alpha-yl-phenylcarbamate analog 3 2187 1440 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 2189 1441 CBX1 10951 NA SURAMIN SURAMIN 2190 1442 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651493 HISTAMINE 2191 1443 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1713082 TRIMEPRAZINE TARTRATE 2192 1444 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE inhibitor CHEMBL3545142 OLOCROLIMUS 2193 1445 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR antagonist 178103927 BAZEDOXIFENE 2195 1446 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3237 CHEMBL602206 2198 1447 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-2A, RECOMBINANT 2199 1448 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME ALPRAZOLAM ALPRAZOLAM 2201 1449 NDUFA2 4695 ENZYME inhibitor CHEMBL3545135 NV-128 2202 1450 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650552 2203 1451 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME MLN-0415 MLN-0415 2205 1452 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-1 2206 1453 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Sirolimus SIROLIMUS 26882569 2207 1454 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE TOLFENAMIC ACID TOLFENAMIC ACID 2208 1455 TOP2B 7155 DRUGGABLE GENOME, ENZYME DEHYDROEQUOL IDRONOXIL 2209 1456 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-acylpiperidine ether derivative 6 2210 1457 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-acylpiperidine ether derivative 3 2211 1458 RNF8 9025 KINASE, ENZYME carboplatin CARBOPLATIN 30071039 2213 1459 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 2216 1460 CCL4 6351 DRUGGABLE GENOME EPO EPOETIN ALFA 17119331 2217 1461 MAOA 4128 DRUGGABLE GENOME, ENZYME METHAMPHETAMINE METHAMPHETAMINE 2218 1462 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125544 CHEMBL533602 2221 1463 PSMB4 5692 DRUGGABLE GENOME, PROTEASE CARFILZOMIB CARFILZOMIB 24524217 2222 1464 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE DASATINIB DASATINIB 2224 1465 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ALSTERPAULLONE ALSTERPAULLONE 2225 1466 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Benzene sulfonamide derivative 11 2227 1467 PDE4D 5144 DRUGGABLE GENOME, ENZYME GPD-1116 2233 1468 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE antibody PERTUZUMAB PERTUZUMAB 2234 1469 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135649697 2235 1470 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE inhibitor 252827507 2236 1471 CP 1356 DRUGGABLE GENOME, ENZYME IMMUNOSUPPRESSIVE 8406056 2237 1472 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME RG-1530 RG-1530 2238 1473 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MECHLORETHAMINE HYDROCHLORIDE MECHLORETHAMINE HYDROCHLORIDE 2239 1474 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR CHLORPROMAZINE CHLORPROMAZINE 18408624 2241 1475 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 328083467 2242 1476 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL1944698 ZOTIRACICLIB 2243 1477 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 4-(1,1-DIETHYLPROPYL)PHENOL CHEMBL2313444 23214428 2244 1478 MAPT 4137 DRUGGABLE GENOME DAPH DAPH 2245 1479 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GW843682X GW843682X 2246 1480 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Piperidinyl pyrazole derivative 3 2251 1481 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIBUTYLCHLOROSTANNANE TRIBUTYLCHLOROSTANNANE 2252 1482 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125810 CHEMBL528119 2253 1483 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Gemcitabine GEMCITABINE 27167172,23520471,21389100,27815358,26228206 2254 1484 TNFRSF1B 7133 DRUGGABLE GENOME CARBAMAZEPINE CARBAMAZEPINE 15565432 2255 1485 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 252827529 2256 1486 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME GENISTEIN GENISTEIN 9331108 2258 1487 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHLORACYZINE CHLORACYZINE 2259 1488 CBX1 10951 NA SB-206553 CHEMBL297784 2260 1489 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME PMID27774822-Compound-Figure9Example15 2261 1490 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL52885 ENMD-981693 2262 1491 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125544 CHEMBL533602 2263 1492 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NOREPINEPHRINE NOREPINEPHRINE 2264 1493 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME CYC-116 CYC-116 2265 1494 ALPI 248 DRUGGABLE GENOME, ENZYME TIOXOLONE TIOXOLONE 2266 1495 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545085 XL-228 2269 1496 BAZ2B 29994 NA GNF-PF-4967 CHEMBL585827 2273 1497 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE Flavanone FLAVANONE 2275 1498 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL971 PENTOBARBITAL SODIUM 2276 1499 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME RHEIN RHEIN 2277 1500 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME SPERMINE SPERMINE 18366176 2278 1501 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TAMATINIB R-406 2279 1502 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 381118867 2281 1503 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR BLISIBIMOD BLISIBIMOD 2286 1504 PLD2 5338 ENZYME, DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 19136975 2287 1505 IRS1 3667 KINASE, CLINICALLY ACTIONABLE GS-101 2289 1506 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AG-528 CHEMBL56542 2290 1507 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 135651484 ESTRONE 2291 1508 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SKF-83565 HYDROBROMIDE CHEMBL541585 2292 1509 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME AG-1879 CHEMBL406845 2294 1510 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME AZD-1080 AZD-1080 2296 1511 CACNB3 784 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ION CHANNEL modulator CHEMBL593430 ATAGABALIN 2297 1512 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BAY-11-7082 CHEMBL403183 2298 1513 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PYROGALLOL PYROGALLOL 2301 1514 BAZ2B 29994 NA CEFACLOR CEFACLOR 2303 1515 TARDBP 23435 TUMOR SUPPRESSOR 1,7-O-DIACETYLMETHYLGEOPYXIN A CHEMBL1889303 2304 1516 CD27 939 PROTEASE INHIBITOR, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME 178101772 2305 1517 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE SB-222200 SB-222200 2307 1518 ATAD5 79915 NA 4'-HYDROXYPHENYL-BENZO[D]THIAZOLE CHEMBL47875 2308 1519 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 178103585 ROMIDEPSIN 2310 1520 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR SPINASAPONIN A METHYL ESTER SPINASAPONIN A METHYL ESTER 20951582 2311 1521 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME KETOTIFEN KETOTIFEN 2314 1522 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 187051792 PANOBINOSTAT 2315 1523 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE DORAMAPIMOD DORAMAPIMOD 2316 1524 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PANITUMUMAB PANITUMUMAB 2317 1525 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE trastuzumab emtansine 2318 1526 ACVR1B 91 SERINE THREONINE KINASE, CELL SURFACE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 249565824 2319 1527 HTT 3064 DRUGGABLE GENOME GNF-PF-2356 CHEMBL601547 2320 1528 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR partial agonist CHEMBL2062276 LEVALLORPHAN TARTRATE 2321 1529 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TAK-715 TAK-715 2322 1530 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PHENAZOPYRIDINE HYDROCHLORIDE PHENAZOPYRIDINE HYDROCHLORIDE 2323 1531 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-2414 CHEMBL601353 2324 1532 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CLOMIPRAMINE HYDROCHLORIDE CLOMIPRAMINE HYDROCHLORIDE 2325 1533 HPSE 10855 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1615835 MUPARFOSTAT 2328 1534 RGS4 5999 DRUGGABLE GENOME DISULFIRAM DISULFIRAM 2329 1535 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL1201178 LISDEXAMFETAMINE DIMESYLATE 2330 1536 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SJ000117451 CHEMBL592123 2331 1537 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE Imatinib IMATINIB 2332 1538 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME pitolisant PITOLISANT 2334 1539 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651408 2335 1540 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE SELENIUM 12168721,15485790 2337 1541 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-14 2338 1542 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Nilotinib NILOTINIB 2340 1543 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-64 2341 1544 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE RAZOXANE RAZOXANE 9378540 2342 1545 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3949 CHEMBL528390 2343 1546 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103522 2347 1547 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000114961 CHEMBL590168 2349 1548 TFPI2 7980 PROTEASE INHIBITOR, DRUGGABLE GENOME HEPARIN HEPARIN 2416032 2350 1549 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Indole-based analog 11 2353 1550 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL TALBUTAL TALBUTAL 2354 1551 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL2062258 2356 1552 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3,4-DIHYDROXYPHENYLACETIC ACID 3,4-DIHYDROXYPHENYLACETIC ACID 2357 1553 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PRACINOSTAT PRACINOSTAT 2359 1554 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE JNK INHIBITOR VIII CHEMBL210618 2360 1555 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BEVANTOLOL BEVANTOLOL 2361 1556 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIAMCINOLONE DIACETATE TRIAMCINOLONE DIACETATE 2363 1557 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GW7647 GW7647 2364 1558 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PURPURIN PURPURIN 2365 1559 HSPB1 3315 DRUGGABLE GENOME TRIAMTERENE TRIAMTERENE 2367 1560 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BAY 86-5044 2368 1561 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE CAR-T cells targeting GPC3 2370 1562 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-14 2371 1563 HSPA4 3308 NA UREA UREA 7548155 2373 1564 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PLK-1 INHIBITOR 2374 1565 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR OXYTOCIN OXYTOCIN 11566737 2375 1566 FAAH 2166 ENZYME, DRUGGABLE GENOME PF-04862853 CHEMBL1915783 21924613 2376 1567 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME DOXORUBICIN DOXORUBICIN 12040435 2378 1568 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Crizotinib CRIZOTINIB 28476735 2379 1569 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201024 METHSCOPOLAMINE BROMIDE 2381 1570 APC 324 CLINICALLY ACTIONABLE K-756 27196752 2382 1571 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor CARFILZOMIB CARFILZOMIB 2385 1572 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RS-67506 CHEMBL83899 2386 1573 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 178101185 2387 1574 TK1 7083 ENZYME, KINASE, DRUGGABLE GENOME zidovudine ZIDOVUDINE 22960662 2388 1575 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650471 2390 1576 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor CHEMBL1230607 PHA-793887 2391 1577 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-64 2393 1578 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR allosteric modulator 381745007 2394 1579 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR DIHYDROGAMBOGIC ACID DIHYDROGAMBOGIC ACID 2395 1580 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GNF-PF-4579 CHEMBL584626 2396 1581 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SIMOCYCLINONE D8 SIMOCYCLINONE D8 22867097 2397 1582 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME LYMPHORAD 2398 1583 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565693 2399 1584 GMNN 51053 DRUGGABLE GENOME BROQUINALDOL BROQUINALDOL 2400 1585 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE HAEMATOXYLIN HAEMATOXYLIN 2401 1586 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 252166505 TEPOTINIB 2405 1587 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME TCMDC-123916 CHEMBL493863 2406 1588 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 artemisinin ARTEMISININ 2408 1589 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DACTINOMYCIN DACTINOMYCIN 2409 1590 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CEAROIN CEAROIN 2411 1591 BAZ2B 29994 NA LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 2413 1592 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Iodine-131-tositumomab 2414 1593 CBX1 10951 NA AG-494 CHEMBL56731 2415 1594 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 374883831 PF-06751979 2417 1595 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME AZD2014 VISTUSERTIB 2418 1596 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME Pyrrolo-pyrrolone derivative 1 2420 1597 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Dihydroisoxazole derivative 1 2422 1598 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CHEMBL591 ETHCHLORVYNOL 2423 1599 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor REGORAFENIB REGORAFENIB 2425 1600 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE AZD4547 27401245 2426 1601 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRICHLORMETHINE TRICHLORMETHINE 2427 1602 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE PTX-200 2428 1603 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LIOTHYRONINE SODIUM LIOTHYRONINE SODIUM 2431 1604 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 135651551 PROGESTERONE 2432 1605 CPS1 1373 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME sodium phenylbutyrate 2434 1606 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CRIZOTINIB CRIZOTINIB 23724914,25733882,25351743,25688157,26372962 2436 1607 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ETODOLAC ETODOLAC 2437 1608 SI 6476 DRUGGABLE GENOME, ENZYME RU-38486 MIFEPRISTONE 3132399 2443 1609 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR CHLORHEXIDINE HYDROCHLORIDE CHLORHEXIDINE HYDROCHLORIDE 2444 1610 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE SCY-641 RUCLOSPORIN 2446 1611 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ZAFIRLUKAST ZAFIRLUKAST 2448 1612 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BMS-582664 BRIVANIB ALANINATE 2449 1613 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE EPTIFIBATIDE EPTIFIBATIDE 2450 1614 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL3544958 CER-002 2451 1615 ATXN2 6311 NA 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 2452 1616 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 328083490 2453 1617 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Selumetinib SELUMETINIB 26544513,27222538 2454 1618 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652339 2456 1619 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200773 TOCAINIDE HYDROCHLORIDE 2458 1620 HTT 3064 DRUGGABLE GENOME CID 94381 CHEMBL374632 2459 1621 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1201483 PSEUDOEPHEDRINE POLISTIREX 2460 1622 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ACEBUTOLOL ACEBUTOLOL 2461 1623 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 178102630 2462 1624 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GRANISETRON GRANISETRON 2463 1625 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE PIFEXOLE PIFEXOLE 2464 1626 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE ALZ-801 2465 1627 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR BAY 869766 2466 1628 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NEVIRAPINE NEVIRAPINE 22931300 2467 1629 RPTOR 57521 CLINICALLY ACTIONABLE, KINASE inhibitor AZD8055 AZD-8055 2468 1630 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL1236962 OMIPALISIB 2469 1631 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TDR77582 CHEMBL1329349 2470 1632 PDE4A 5141 DRUGGABLE GENOME, ENZYME AN-2898 2471 1633 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Peptide analog 7 2472 1634 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MEK INHIBITOR GDC-0623 23934108 2474 1635 CLCN6 1185 ION CHANNEL, DRUGGABLE GENOME blocker 178100996 2475 1636 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Olopatadine OLOPATADINE 2476 1637 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178103894 VENLAFAXINE 2477 1638 HDAC11 79885 DRUGGABLE GENOME, ENZYME PRACINOSTAT PRACINOSTAT 2478 1639 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TREQUINSIN HYDROCHLORIDE TREQUINSIN HYDROCHLORIDE 2480 1640 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2-MERCAPTOBENZIMIDAZOLE 2-MERCAPTOBENZIMIDAZOLE 2481 1641 BCHE 590 DRUGGABLE GENOME, ENZYME IMMUNOTOXIN 10198815 2485 1642 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE LUTEOLIN LUTEOLIN 2487 1643 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DICHLOROPHEN DICHLOROPHEN 2488 1644 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200982 BUTABARBITAL SODIUM 2489 1645 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Unfractionated heparin 2491 1646 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 23622981 2495 1647 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Tricyclic heterocycle derivative 1 2496 1648 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME activator 178101922 2497 1649 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME GNF-PF-5159 CHEMBL1493528 2498 1650 PDE4D 5144 DRUGGABLE GENOME, ENZYME DENBUFYLLINE DENBUFYLLINE 2501 1651 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DICLOFENAC DICLOFENAC 22931300 2503 1652 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE MARIMASTAT MARIMASTAT 2505 1653 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor BYL719 ALPELISIB 2507 1654 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME DNDI1417467 CHEMBL1997335 2509 1655 PDE4B 5142 DRUGGABLE GENOME, ENZYME RONOMILAST 2510 1656 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR 4-HYDROPEROXYCYCLOPHOSPHAMIDE PERFOSFAMIDE 1283360 2511 1657 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL49642 INDIBULIN 2512 1658 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR E-GUGGULSTERONE E-GUGGULSTERONE 2515 1659 USP1 7398 DNA REPAIR, PROTEASE, ENZYME AMYLMETACRESOL AMYLMETACRESOL 2516 1660 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TAMOXIFEN TAMOXIFEN 2517 1661 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID27336223-Compound-4 2519 1662 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING 3,8'-BIAPIGENIN CHEMBL515252 2520 1663 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-25 2521 1664 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Radiotherapy 28652249 2522 1665 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1898523 PHENDIMETRAZINE TARTRATE 2524 1666 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-67 CHEMBL578512 2526 1667 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RO5126766 26438159 2527 1668 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE fludarabine FLUDARABINE 27173875 2528 1669 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PG-490-88 2529 1670 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER nicardipine NICARDIPINE 2532 1671 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-99550 CHEMBL1288014 2533 1672 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE DASATINIB DASATINIB 15928335,15685537,22718859,16638875,15146165,12949711,26130666,25157968,14645423,16954519,18794084,22745105 2534 1673 POLK 51426 DNA REPAIR, ENZYME TETROQUINONE TETROQUINONE 2535 1674 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-29 2536 1675 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PREDNICARBATE PREDNICARBATE 2537 1676 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR rituximab RITUXIMAB 26384320 2538 1677 RAB9A 9367 ENZYME, DRUGGABLE GENOME VU0080241 CHEMBL477396 2539 1678 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME ERYTHROMYCIN ERYTHROMYCIN 18212111 2540 1679 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NALED NALED 2541 1680 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYSTEAMINE HYDROCHLORIDE CYSTEAMINE HYDROCHLORIDE 2542 1681 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EXALAMIDE EXALAMIDE 2543 1682 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE DOXORUBICIN DOXORUBICIN 12698198 2544 1683 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR WITHAFERIN A WITHAFERIN A 24079846 2546 1684 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist LY 2510924 2548 1685 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OXYMETAZOLINE OXYMETAZOLINE 2549 1686 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PYRIMETHAMINE PYRIMETHAMINE 2551 1687 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051792 PANOBINOSTAT 2552 1688 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE tramadol TRAMADOL 21837673,30549211 2553 1689 COL18A1 80781 DRUGGABLE GENOME CSF 14693162 2554 1690 METAP2 10988 ENZYME, DRUGGABLE GENOME, KINASE, PROTEASE PPI-2458 PPI-2458 2558 1691 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CYCLOVALONE CYCLOVALONE 2559 1692 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-5151 CHEMBL576208 2561 1693 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE Somatomedin-1 2563 1694 KAT2B 8850 ENZYME, DRUGGABLE GENOME TRIAZOLAM TRIAZOLAM 22137933 2564 1695 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 363894211 PEXMETINIB 2565 1696 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR Disitertide DISITERTIDE 24393789 2566 1697 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME DPX-Survivac 2570 1698 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME VALPROIC ACID VALPROIC ACID 18294844,16921367,25304896 2571 1699 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1200920 ISOETHARINE HYDROCHLORIDE 2573 1700 TH 7054 ENZYME, DRUGGABLE GENOME metyrosine METYROSINE 2574 1701 CD52 1043 DRUGGABLE GENOME antibody 178103376 ALEMTUZUMAB 2576 1702 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE leucovorin LEUCOVORIN 24980946 2577 1703 HTT 3064 DRUGGABLE GENOME FLUORESCEIN DIACETATE FLUORESCEIN DIACETATE 2580 1704 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME DIMIRACETAM DIMIRACETAM 2582 1705 ATXN2 6311 NA 4'-EPICHAETOVIRIDIN A CHEMBL1306556 2583 1706 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 252827366 GILTERITINIB 2584 1707 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 12-HYDROXY-OCTADECANOIC ACID CHEMBL292352 2585 1708 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TPCK TPCK 2587 1709 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE TCMDC-125758 CHEMBL546797 2589 1710 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178102699 BEPAFANT 2590 1711 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR BENZOTHIAZOL-2-YLAMINE CHEMBL329785 22982122 2591 1712 MAPT 4137 DRUGGABLE GENOME METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE 2592 1713 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CORTODOXONE CORTODOXONE 2593 1714 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417809 CHEMBL1442783 2594 1715 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE DNDI1417078 CHEMBL1320798 2595 1716 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 404859105 2597 1717 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME THONZONIUM THONZONIUM 2598 1718 F11 2160 DRUGGABLE GENOME, PROTEASE, ENZYME THROMBIN THROMBIN 9787166 2599 1719 CCL3 6348 KINASE, DRUGGABLE GENOME INFLIXIMAB INFLIXIMAB 16219708 2602 1720 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE 0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE 2603 1721 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FLUCONAZOLE FLUCONAZOLE 22931300 2604 1722 TUBA4A 7277 DRUGGABLE GENOME CHEMBL2304041 SAGOPILONE 2605 1723 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE GNF-PF-574 CHEMBL582737 2607 1724 TUBB 203068 DRUGGABLE GENOME ALB-109564(a) 2608 1725 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 178100555 2609 1726 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Cyclic octapeptide derivative 1 2610 1727 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565836 2611 1728 POLK 51426 DNA REPAIR, ENZYME TRYPAN BLUE TRYPAN BLUE 2612 1729 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR Analgesics 25096645 2613 1730 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW827102X GW827102X 2614 1731 BAZ2B 29994 NA DNDI1417165 CHEMBL1406948 2615 1732 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-78 CHEMBL579318 2617 1733 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR ANTIOXIDANT 12221586 2618 1734 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CONGO RED CONGO RED 2620 1735 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME SB-1578 CT-1578 2625 1736 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR T091317 T091317 22579484,24480357,24268541 2626 1737 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME DISULFIRAM DISULFIRAM 8904971 2627 1738 ELP5 23587 NA methylphenidate METHYLPHENIDATE 29382897 2629 1739 ATAD5 79915 NA TCMDC-123927 CHEMBL531268 2630 1740 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Benzene sulfonamide derivative 15 2631 1741 GHRL 51738 DRUGGABLE GENOME ROFECOXIB ROFECOXIB 16868036 2632 1742 KAT5 10524 TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, ENZYME inhibitor 187051791 2633 1743 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME LEUCETTAMINE B LEUCETTAMINE B 22998443 2634 1744 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SY-1425 2635 1745 ABCC6 368 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER HEPARAN SULFATE 12600949 2639 1746 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER N-(3,4-DICHLOROPHENYL)BENZAMIDE CHEMBL560296 2640 1747 PSMA8 143471 DRUGGABLE GENOME, PROTEASE CARFILZOMIB CARFILZOMIB 24524217 2641 1748 MAP2K5 5607 KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor AZD6244 SELUMETINIB 2643 1749 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME CYC-116 CYC-116 2644 1750 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ALVERINE CITRATE ALVERINE CITRATE 2645 1751 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178101541 FUROSEMIDE 2646 1752 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FG-2216 2648 1753 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TRIPHENYLSTANNANOL TRIPHENYLSTANNANOL 2651 1754 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20100022547C80 2653 1755 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME OPHIOBOLIN O OPHIOBOLIN O 22130129 2654 1756 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROGESTERONE PROGESTERONE 12061859 2657 1757 ALB 213 TRANSPORTER, DRUGGABLE GENOME RALTITREXED RALTITREXED 15025739 2658 1758 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor BELINOSTAT BELINOSTAT 2659 1759 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102286 QUIZARTINIB 2661 1760 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor AZD8931 SAPITINIB 2665 1761 KDM4A 9682 DRUGGABLE GENOME, ENZYME AFIMOXIFENE AFIMOXIFENE 2666 1762 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMITRIPTYLINOXIDE AMITRIPTYLINOXIDE 2667 1763 E2F1 1869 TRANSCRIPTION FACTOR NERVE GROWTH FACTOR 10454552 2669 1764 RNF8 9025 KINASE, ENZYME docetaxel DOCETAXEL 30071039 2672 1765 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 328083507 2675 1766 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GEFITINIB GEFITINIB 2678 1767 GMNN 51053 DRUGGABLE GENOME DNDI1416982 CHEMBL1479114 2680 1768 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-25 2681 1769 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE ALISERTIB ALISERTIB 2683 1770 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor SCH727965 DINACICLIB 2684 1771 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 8-OH-DPAT 8-OH-DPAT 2685 1772 PDE4B 5142 DRUGGABLE GENOME, ENZYME THEOPHYLLINE THEOPHYLLINE 2686 1773 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL ADINAZOLAM ADINAZOLAM 2687 1774 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody 252827373 ELGEMTUMAB 2688 1775 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME BUTANOIC ACID BUTANOIC ACID 19053749 2690 1776 GLCCI1 113263 NA nedocromil NEDOCROMIL 21991891 2691 1777 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE NERVE GROWTH FACTOR 11069896 2692 1778 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BLEOMYCIN BLEOMYCIN 15208274 2693 1779 IAPP 3375 DRUGGABLE GENOME, HORMONE ACTIVITY CURCUMIN CURCUMIN 2694 1780 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE OLEANOLIC_ACID OLEANOLIC_ACID 21453996 2695 1781 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIVAMPICILLIN PIVAMPICILLIN 2697 1782 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MALATHION MALATHION 2698 1783 CCL2 6347 DRUGGABLE GENOME Bindarit BINDARIT 2699 1784 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE cyclophosphamide CYCLOPHOSPHAMIDE 2700 1785 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200597 ETIDOCAINE HYDROCHLORIDE 2701 1786 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1256 ISOFLURANE 2702 1787 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650102 CIPROXIFAN 2703 1788 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PHENETHYLISOTHIOCYANATE PHENETHYLISOTHIOCYANATE 22607231 2704 1789 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PMID25656651-Compound-21a 2705 1790 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652675 CAFFEINE 2706 1791 GMNN 51053 DRUGGABLE GENOME GNF-PF-107 CHEMBL578675 2707 1792 AMH 268 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DES DIETHYLSTILBESTROL 9751506 2709 1793 LOXL2 4017 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME GS-6624 SIMTUZUMAB 2710 1794 CAMKK2 10645 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 178101957 2713 1795 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TCMDC-124354 CHEMBL546344 2714 1796 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE elexacaftor / tezacaftor / ivacaftor 2716 1797 MAP2K3 5606 KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE inhibitor TRAMETINIB TRAMETINIB 2717 1798 XPNPEP2 7512 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL2103847 TOSEDOSTAT 2721 1799 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 381118857 2722 1800 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME NRX-4204 2724 1801 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL GSK683699 2725 1802 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIPYRITHIONE DIPYRITHIONE 2726 1803 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GEMCITABINE GEMCITABINE 15581051 2727 1804 BRCA2 675 CLINICALLY ACTIONABLE Talazoparib TALAZOPARIB 2728 1805 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME gemcitabine GEMCITABINE 25162786,20665488,22705007,24475233,24361227 2729 1806 POLK 51426 DNA REPAIR, ENZYME MAREIN MAREIN 2730 1807 SETD7 80854 ENZYME, METHYL TRANSFERASE inhibitor 249565915 2731 1808 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR LY2157299 2733 1809 HCN3 57657 DRUGGABLE GENOME, ION CHANNEL blocker 135650098 CILOBRADINE 2735 1810 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102238 ROLOFYLLINE 2737 1811 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BKM120 BUPARLISIB 2740 1812 GUCY2C 2984 DRUGGABLE GENOME, KINASE agonist 178101714 LINACLOTIDE 2742 1813 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VALPROIC ACID VALPROIC ACID 22931300 2744 1814 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 223366058 2746 1815 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor PIMASERTIB PIMASERTIB 2747 1816 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DIHYDROGAMBOGIC ACID DIHYDROGAMBOGIC ACID 2748 1817 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME ACIVICIN ACIVICIN 12670536 2751 1818 PDE4A 5141 DRUGGABLE GENOME, ENZYME MM36 topical ointment 2752 1819 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE BAY1000394 2754 1820 BAZ2B 29994 NA 5,8,11,14-EICOSATETRAYNOIC ACID CHEMBL458328 2755 1821 POLK 51426 DNA REPAIR, ENZYME 3,8'-BIAPIGENIN CHEMBL515252 2757 1822 RGS4 5999 DRUGGABLE GENOME CALCIMYCIN CALCIMYCIN 2758 1823 BCHE 590 DRUGGABLE GENOME, ENZYME MEPTAZINOL MEPTAZINOL 2759 1824 ATXN2 6311 NA ERBSTATIN ERBSTATIN 2760 1825 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE N-ACETYL-L-CYSTEINE ACETYLCYSTEINE 10716998 2761 1826 CDKN2B-AS1 100048912 NA Antiinflammatory agents, non-steroids 20538124 2762 1827 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BIFONAZOLE BIFONAZOLE 2764 1828 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor 178102647 2765 1829 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 328083485 OSI-930 2767 1830 ADORA2A-AS1 646023 NA methotrexate METHOTREXATE 27399166 2770 1831 TESK2 10420 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TYROSINE KINASE inhibitor 249565799 2771 1832 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GENTIAN VIOLET GENTIAN VIOLET 2772 1833 MAOB 4129 DRUGGABLE GENOME, ENZYME METHAMPHETAMINE METHAMPHETAMINE 2773 1834 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE FENTICLOR FENTICLOR 2774 1835 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565859 PF-03715455 2775 1836 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DTS-201 2776 1837 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME TG-0054 BURIXAFOR 2778 1838 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME WHI-P154 CHEMBL473773 2779 1839 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME UNC0224 CHEMBL576781 19891491 2781 1840 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL celecoxib CELECOXIB 22336956 2782 1841 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DALBERGIONE DALBERGIONE 2783 1842 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME inhibitor 178103579 CURCUMIN 2784 1843 MAP3K7 6885 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 329968393 2785 1844 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX PYROGALLOL RED PYROGALLOL RED 16759101 2788 1845 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHENYL AMINOSALICYLATE PHENYL AMINOSALICYLATE 2789 1846 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Vidarabine VIDARABINE 2790 1847 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL1742994 BRENTUXIMAB VEDOTIN 2791 1848 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE TYRPHOSTIN A9 TYRPHOSTIN A9 2792 1849 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PROGESTOGENS 7450248 2793 1850 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GR-4661 CHEMBL344127 2796 1851 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL2107771 RALFINAMIDE 2800 1852 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR L-165041 CHEMBL153057 2802 1853 PDE4D 5144 DRUGGABLE GENOME, ENZYME BPN14770 BPN-14770 2803 1854 CBX1 10951 NA DOCEBENONE DOCEBENONE 2804 1855 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ERYTHROMYCIN ERYTHROMYCIN 22931300 2805 1856 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEGUELIN DEGUELIN 2807 1857 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE BERKELEYDIONE BERKELEYDIONE 17970594 2808 1858 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME RECOMBINANT ERYTHROPOIETIN 15957544 2809 1859 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME TOZASERTIB TOZASERTIB 2810 1860 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME PMID27828716-Compound-BIO-acetoxime 2811 1861 SLC6A15 55117 DRUGGABLE GENOME, TRANSPORTER inhibitor 178103791 LORATADINE 2812 1862 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID25991433-Compound-P6 2813 1863 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL3545327 TTP-607 2814 1864 ATAD5 79915 NA TCMDC-124356 CHEMBL22062 2816 1865 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CENISERTIB CENISERTIB 2818 1866 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR LITHOCHOLIC ACID LITHOCHOLIC ACID 17963371 2819 1867 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALSTERPAULLONE ALSTERPAULLONE 2820 1868 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Alvocidib ALVOCIDIB 12777976 2821 1869 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CPT-11 IRINOTECAN HYDROCHLORIDE 11802813 2822 1870 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME BML-210 CHEMBL324053 16921367 2823 1871 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE CELECOXIB CELECOXIB 21678971 2824 1872 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 2828 1873 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker 53801058 MIBEFRADIL 2830 1874 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER epirubicin EPIRUBICIN 22903472 2831 1875 GMNN 51053 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 2832 1876 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ERYTHROMYCIN ERYTHROMYCIN 17007374 2835 1877 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US9580418, Example 11 2837 1878 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3201 CHEMBL581872 2838 1879 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651279 TRIFLUOPERAZINE 2839 1880 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE OSI-930 OSI-930 2840 1881 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-3148 CHEMBL81782 2842 1882 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE REV-5901 REV-5901 2843 1883 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROPIOMAZINE PROPIOMAZINE 2845 1884 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Binimetinib BINIMETINIB 2847 1885 PRPS1 5631 DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, ENZYME LOMETREXOL LOMETREXOL 25962120 2848 1886 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TOPICAL CORTICOSTEROIDS 12207591 2849 1887 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BENPERIDOL BENPERIDOL 2851 1888 PIP 5304 DRUGGABLE GENOME HORMONES 7558422 2852 1889 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL antagonist CHEMBL220492 TOPIRAMATE 2854 1890 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE MEK162 BINIMETINIB 2855 1891 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BYL719 ALPELISIB 2856 1892 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE 5-FLUORODEOXYURIDINE FLOXURIDINE 15899874 2857 1893 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ALLANTODAPSONE ALLANTODAPSONE 2858 1894 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR MOTEXAFIN GADOLINIUM 2859 1895 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER atenolol ATENOLOL 2860 1896 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUOXETINE HYDROCHLORIDE FLUOXETINE HYDROCHLORIDE 2861 1897 GCLC 2729 DRUGGABLE GENOME, ENZYME BSO 9660546 2863 1898 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME GDC-0980/RG7422 2864 1899 KAT5 10524 TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, ENZYME ANACARDIC ACID 22100137 2865 1900 PDE4B 5142 DRUGGABLE GENOME, ENZYME AN-2728 CRISABOROLE 2867 1901 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE LESTAURTINIB LESTAURTINIB 2868 1902 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE TRASTUZUMAB TRASTUZUMAB 23680147 2870 1903 LMNA 4000 CLINICALLY ACTIONABLE, DRUGGABLE GENOME HISTAMINE HISTAMINE 2871 1904 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE TeloB-Vax 2872 1905 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR SULODEXIDE SULODEXIDE 2873 1906 PI3 5266 DRUGGABLE GENOME, PROTEASE INHIBITOR PROGESTERONE PROGESTERONE 14521952 2875 1907 HBB 3043 DRUGGABLE GENOME, ENZYME AZACITIDINE AZACITIDINE 2876 1908 TUBA3D 113457 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 2877 1909 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE RITONAVIR RITONAVIR 11141242 2878 1910 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 2879 1911 COL5A1 1289 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 2881 1912 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Peptide analog 47 2883 1913 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 2884 1914 TMEM97 27346 NA PMID30185082-Compound-54 2885 1915 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE PF-562271 PF-00562271 2887 1916 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-3582 CHEMBL606167 2888 1917 KDM4A 9682 DRUGGABLE GENOME, ENZYME MITOXANTRONE MITOXANTRONE 2889 1918 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MITOXANTRONE MITOXANTRONE 2890 1919 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 4-DODECYL-PHENOL CHEMBL194881 2891 1920 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME GNF-PF-2812 CHEMBL125044 2892 1921 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor PKI-587 GEDATOLISIB 2893 1922 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CARBOPLATIN CARBOPLATIN 19470925 2894 1923 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR atorvastatin ATORVASTATIN 2895 1924 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-203580 SB-203580 2896 1925 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ASTERRIC ACID ASTERRIC ACID 2897 1926 DGAT2 84649 ENZYME Vitamin B3 2901 1927 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor NILOTINIB NILOTINIB 2902 1928 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME FASUDIL FASUDIL 2906 1929 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME 681640 CHEMBL379975 2907 1930 NDUFB8 4714 ENZYME inhibitor CHEMBL3545320 ME-344 2908 1931 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CAMPTOTHECIN CAMPTOTHECIN 2910 1932 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME METHOCARBAMOL METHOCARBAMOL 22931300 2911 1933 GBA 2629 DRUGGABLE GENOME, ENZYME APTIGANEL HYDROCHLORIDE APTIGANEL HYDROCHLORIDE 2912 1934 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE TCMDC-124307 CHEMBL546865 2913 1935 HSPB1 3315 DRUGGABLE GENOME UREA UREA 9094264 2916 1936 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Neratinib NERATINIB 28274957,28679771,22908275,26874901,23953056,28363995,26333383,27078022,28539475,24323026,23220880,27697991,26243863 2917 1937 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GI-4000 2921 1938 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME Epoetin zeta 2922 1939 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME modulator CHEMBL490029 MK-0533 2923 1940 HLA-DRA 3122 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE amoxicillin AMOXICILLIN 30664875 2924 1941 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 2925 1942 KAT2B 8850 ENZYME, DRUGGABLE GENOME cannabinoids NABIXIMOLS 2926 1943 HTT 3064 DRUGGABLE GENOME TCMDC-124573 CHEMBL525826 2928 1944 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE diazepam DIAZEPAM 18695978 2929 1945 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE SB-202190 SB-202190 2930 1946 UGT2B7 7364 DRUGGABLE GENOME codeine CODEINE 25752520 2932 1947 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Aminocyclopentenone compound 6 2933 1948 POLB 5423 DNA REPAIR, DRUGGABLE GENOME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 2934 1949 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3544930 SC-80036 2935 1950 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR tacrolimus TACROLIMUS 21359536 2936 1951 PTGES 9536 DRUGGABLE GENOME, ENZYME Benzamide derivative 14 2937 1952 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Indacaterol INDACATEROL 2939 1953 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-22 2943 1954 COL11A1 1301 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 2945 1955 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Flotetuzumab FLOTETUZUMAB 2946 1956 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME paclitaxel PACLITAXEL 24361227 2947 1957 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Ruxolitinib cream 2949 1958 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ZUCAPSAICIN ZUCAPSAICIN 2950 1959 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME FLUNARIZINE DIHYDROCHLORIDE FLUNARIZINE DIHYDROCHLORIDE 2951 1960 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR heroin DIACETYLMORPHINE 24279859,28692418,26401760 2953 1961 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-124176 CHEMBL588038 2954 1962 CXCL8 3576 DRUGGABLE GENOME METHIMAZOLE METHIMAZOLE 11453524 2955 1963 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME SENNOSIDE A SENNOSIDE A 2956 1964 GPR183 1880 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651392 CHEMBL169046 2957 1965 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Indoline derivative 7 2959 1966 CBX1 10951 NA TRIMETHOPRIM TRIMETHOPRIM 2961 1967 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme15-1 2962 1968 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 2963 1969 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL blocker 381744957 2965 1970 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DOXORUBICIN DOXORUBICIN 2967 1971 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Nintedanib NINTEDANIB 22238366 2968 1972 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BUFLOMEDIL BUFLOMEDIL 2970 1973 FXYD2 486 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL1751 DIGOXIN 2972 1974 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Isoflavone derivative 2 2974 1975 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NITROGEN MUSTARD 2882834 2975 1976 CP 1356 DRUGGABLE GENOME, ENZYME AMPICILLIN AMPICILLIN 1427966 2976 1977 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SOTRASTAURIN SOTRASTAURIN 2978 1978 CA9 768 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL18 ETHOXZOLAMIDE 2980 1979 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL FLURAZEPAM FLURAZEPAM 2982 1980 SMN1 6606 DRUGGABLE GENOME NSC-234945 CHEMBL260311 2983 1981 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SOLIFENACIN SOLIFENACIN 2985 1982 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 178101311 DRAFLAZINE 2986 1983 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102729 2987 1984 FOXC2 2303 DRUG RESISTANCE, TRANSCRIPTION FACTOR OXALIPLATIN OXALIPLATIN 32110058 2988 1985 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME RAF265 RAF-265 20538618,22351689 2989 1986 POLI 11201 DNA REPAIR 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 2990 1987 RORA 6095 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE interferon beta-1a 31649263 2991 1988 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME eculizumab ECULIZUMAB 24521109 2993 1989 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME PHORBOL MYRISTATE ACETATE PHORBOL MYRISTATE ACETATE 22579485 2994 1990 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR GNF-PF-2301 CHEMBL578061 2995 1991 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE vincristine VINCRISTINE 2998 1992 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME DESIPRAMINE DESIPRAMINE 2999 1993 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALITRETINOIN ALITRETINOIN 7807131 3000 1994 RAB9A 9367 ENZYME, DRUGGABLE GENOME 7-METHOXY-BAPTIGENIN CHEMBL583578 3002 1995 SMN1 6606 DRUGGABLE GENOME CID 4101591 CHEMBL428789 3003 1996 BCAR3 8412 KINASE ANTIESTROGEN 9582273 3004 1997 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 310264675 CUDC-101 3005 1998 ALOX15 246 ENZYME, DRUGGABLE GENOME CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 3006 1999 CES1 1066 DRUGGABLE GENOME, ENZYME clopidogrel CLOPIDOGREL 23275066,27450232,25704243,24535487 3007 2000 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Apixaban APIXABAN 3009 2001 KDM4A 9682 DRUGGABLE GENOME, ENZYME N-METHYL-D-ASPARTIC ACID (NMDA) N-METHYL-D-ASPARTIC ACID (NMDA) 3011 2002 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME 681640 CHEMBL379975 3014 2003 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CCG-63802 CHEMBL1476646 3015 2004 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PWT33597 3016 2005 TUBB2A 7280 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 3019 2006 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME PACLITAXEL PACLITAXEL 9067280 3021 2007 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE IMATINIB MESYLATE IMATINIB MESYLATE 3022 2008 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody GANITUMAB GANITUMAB 3023 2009 POLI 11201 DNA REPAIR FURAMIDINE FURAMIDINE 3024 2010 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Anti-FGFR3 3028 2011 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE IFOSFAMIDE IFOSFAMIDE 3029 2012 NR1D1 9572 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME agonist 135650323 GSK-4112 3030 2013 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor BGJ398 INFIGRATINIB 3031 2014 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ANTHRACYCLINE 14978790,15068318 3032 2015 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER VINBLASTINE VINBLASTINE 21348461,20363635 3034 2016 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR METRONIDAZOLE METRONIDAZOLE 12111578 3036 2017 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR FULVESTRANT FULVESTRANT 3039 2018 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL2146883 COBIMETINIB 3040 2019 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200760 BALSALAZIDE DISODIUM 3041 2020 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL3545327 TTP-607 3042 2021 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417739 CHEMBL487356 3047 2022 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KEPONE KEPONE 3048 2023 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TOPOTECAN TOPOTECAN 3050 2024 ABCB11 8647 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CHENODIOL CHENODIOL 19102680 3051 2025 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL405821 SENICAPOC 3052 2026 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHRYSIN CHRYSIN 3053 2027 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MUTANT IDH1 INHIBITOR DS-1001 3054 2028 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TETRAHYDROCURCUMIN TETRAHYDROCURCUMIN 19112019 3055 2029 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3545096 BGT-226 3056 2030 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE modulator CHEMBL3545174 GSK2881078 3057 2031 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE I3C 11948137 3059 2032 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1578 ANISOTROPINE METHYLBROMIDE 3060 2033 MAPT 4137 DRUGGABLE GENOME MORIN MORIN 3061 2034 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL259084 MLN-8054 3062 2035 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FGF/VEGF RECEPTOR TYROSINE KINASE INHIBITOR, PD173074 27535980 3063 2036 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000032151 CHEMBL592600 3064 2037 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIMOZIDE PIMOZIDE 3065 2038 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GALANTAMINE HYDROBROMIDE GALANTAMINE HYDROBROMIDE 3066 2039 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 223366182 3067 2040 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW631581B GW631581B 3068 2041 AQP4 361 ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ZONISAMIDE ZONISAMIDE 18572411 3070 2042 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PHYSOSTIGMINE PHYSOSTIGMINE 3071 2043 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR Metelimumab METELIMUMAB 3073 2044 ATXN2 6311 NA TCMDC-125625 CHEMBL549208 3075 2045 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PYRITHIONE ZINC PYRITHIONE ZINC 3076 2046 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE PERTUZUMAB PERTUZUMAB 29802158 3077 2047 ACVR1B 91 SERINE THREONINE KINASE, CELL SURFACE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 249565787 VACTOSERTIB 3078 2048 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 381744997 REPOTRECTINIB 3080 2049 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 249565577 FAMITINIB 3081 2050 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE paclitaxel PACLITAXEL 23963862 3082 2051 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 135650760 ONAPRISTONE 3083 2052 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHYLENE BLUE CHLORIDE HYDRATE METHYLENE BLUE 3085 2053 HCP5 10866 NA gemcitabine GEMCITABINE 31616045 3086 2054 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-21588 CHEMBL1611308 3087 2055 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Isoflavone derivative 3 3088 2056 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HOECHST 33258 HOECHST 33258 3089 2057 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL1200395 ORPHENADRINE CITRATE 3090 2058 ARID1A 8289 CLINICALLY ACTIONABLE NIVOLUMAB NIVOLUMAB 29736026 3091 2059 GUCY1A2 2977 ENZYME, DRUGGABLE GENOME activator CHEMBL1200689 NITRIC OXIDE 3093 2060 ADCY1 107 DRUGGABLE GENOME, ENZYME NSC-270718 CHEMBL401844 18630896 3096 2061 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL3137336 UPROSERTIB 3097 2062 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME TAMOXIFEN TAMOXIFEN 22942317 3099 2063 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TGBA01AD 3100 2064 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652048 BQ-123 3101 2065 ATXN2 6311 NA R-N-PROPYLNORAPOMORPHINE R-N-PROPYLNORAPOMORPHINE 3102 2066 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor 249565578 IPATASERTIB 3103 2067 TARDBP 23435 TUMOR SUPPRESSOR SJ000032149 CHEMBL600778 3104 2068 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Carbamide derivative 21 3106 2069 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME EVEROLIMUS EVEROLIMUS 24625776,25295501 3107 2070 KLF4 9314 TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE APTO-253 APTO-253 3110 2071 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FLUSPIRILENE FLUSPIRILENE 3112 2072 CXCL8 3576 DRUGGABLE GENOME PROTECTIVE AGENT 9479645 3116 2073 HEBP1 50865 DRUGGABLE GENOME 3-phenyl propanoic derivative 3 3117 2074 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NIFEDIPINE NIFEDIPINE 22931300 3118 2075 IMPA1 3612 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103738 LITHIUM CITRATE 3119 2076 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Ipatasertib IPATASERTIB 27872130 3120 2077 HEXB 3074 ENZYME AMINOGLYCOSIDES 3440638 3121 2078 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLENBUTEROL HYDROCHLORIDE CLENBUTEROL HYDROCHLORIDE 3123 2079 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER TRAIL 10811986 3125 2080 CPB2 1361 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166824 3127 2081 KAT2B 8850 ENZYME, DRUGGABLE GENOME inhibitor 178103578 3128 2082 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR CYC-116 CYC-116 3129 2083 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME D-5519 3131 2084 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CLOTRIMAZOLE CLOTRIMAZOLE 3132 2085 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BENANSERIN HYDROCHLORIDE BENANSERIN HYDROCHLORIDE 3133 2086 POLI 11201 DNA REPAIR 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 3136 2087 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 348353655 OCLACITINIB 3137 2088 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BMS-687453 CHEMBL1089501 20218621 3138 2089 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OXYPHENCYCLIMINE HYDROCHLORIDE OXYPHENCYCLIMINE HYDROCHLORIDE 3139 2090 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME GEFITINIB GEFITINIB 15738541 3140 2091 KLK7 5650 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252166696 3141 2092 FOLR2 2350 CELL SURFACE, DRUGGABLE GENOME FOLIC ACID FOLIC ACID 25234128 3142 2093 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TRIFLUSAL TRIFLUSAL 3143 2094 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135652717 STAUROSPORINE 3144 2095 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME SALERMIDE SALERMIDE 3145 2096 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CV-3988 CHEMBL295212 3147 2097 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE Chloroprocaine CHLOROPROCAINE 3149 2098 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR EPINEPHRINE EPINEPHRINE 3159 2099 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE VANDETANIB VANDETANIB 3160 2100 CAT 847 ENZYME, DRUGGABLE GENOME EUK-189 3161 2101 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178103687 ALMOTRIPTAN 3162 2102 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME ANTICONVULSANT 7509966 3163 2103 KCNS3 3790 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 3164 2104 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FLUSPIRILENE FLUSPIRILENE 3166 2105 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME o-desmethyltramadol 27082504 3167 2106 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME KENPAULLONE KENPAULLONE 3170 2107 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 KENPAULLONE KENPAULLONE 3171 2108 NAPEPLD 222236 ENZYME inhibitor 405560510 HEXACHLOROPHENE 3172 2109 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 363894223 3174 2110 RBP4 5950 DRUGGABLE GENOME FENRETINIDE FENRETINIDE 16034410 3175 2111 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME LANSOPRAZOLE LANSOPRAZOLE 3176 2112 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102539 3180 2113 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SALVINORIN A SALVINORIN A 22204910 3182 2114 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Palbociclib PALBOCICLIB 3184 2115 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL918 PHENACEMIDE 3185 2116 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor IDELALISIB IDELALISIB 3186 2117 MT1G 4495 NA BSO 8966720 3187 2118 BAZ2B 29994 NA CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 3188 2119 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-4612 CHEMBL601550 3189 2120 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE LABETALOL LABETALOL 3190 2121 CA9 768 DRUGGABLE GENOME, ENZYME Sulfonamide-thiadiazole derivative 1 3191 2122 PDE10A 10846 ENZYME, DRUGGABLE GENOME 1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 6 3192 2123 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-8 3193 2124 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL538943 VINORELBINE TARTRATE 3194 2125 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33p 3195 2126 CBX1 10951 NA 2',3,4-TRIHYDROXYCHALCONE CHEMBL339587 3196 2127 PSMC5 5705 TRANSCRIPTION FACTOR BINDING, PROTEASE inhibitor IXAZOMIB IXAZOMIB 3198 2128 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Diaryl amine derivative 1 3199 2129 TUBB3 10381 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 3201 2130 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME MITOXANTRONE MITOXANTRONE 3202 2131 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 340590230 3206 2132 CA1 759 DRUGGABLE GENOME, ENZYME ZONISAMIDE ZONISAMIDE 3207 2133 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651742 3208 2134 KDM4A 9682 DRUGGABLE GENOME, ENZYME 4-METHYLDAPHNETIN 4-METHYLDAPHNETIN 3209 2135 DROSHA 29102 NA daunorubicin DAUNORUBICIN 24614921 3212 2136 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TCMDC-123992 CHEMBL530149 3213 2137 MAPT 4137 DRUGGABLE GENOME GNF-PF-5510 CHEMBL578741 3214 2138 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME PRAZEPAM PRAZEPAM 3215 2139 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 3216 2140 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ZM-449829 CHEMBL154580 3217 2141 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE P-T-OCTYLPHENOL CHEMBL259327 3218 2142 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME STROBOPININ STROBOPININ 3219 2143 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 2,4,5,10-TETRAHYDROPYRAZOLO[3,4-A]CARBAZOLE CHEMBL512649 3220 2144 RRP1B 23076 NA atenolol ATENOLOL 31327267 3221 2145 HDAC11 79885 DRUGGABLE GENOME, ENZYME APICIDIN APICIDIN 19705846 3223 2146 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2,2,3,3,4,4,5,5,6,6,7,7,8,8,8-PENTADECAFLUORO-OCTANOIC ACID CHEMBL172988 3225 2147 KMO 8564 DRUGGABLE GENOME, ENZYME Isoxazoles and isoxazoline derivative 6 3228 2148 MAPT 4137 DRUGGABLE GENOME GOSSYPOL GOSSYPOL 3229 2149 NDUFB5 4711 ENZYME inhibitor CHEMBL3545320 ME-344 3230 2150 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PHENYLPROPANOLAMINE PHENYLPROPANOLAMINE 3231 2151 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor SELUMETINIB SELUMETINIB 3232 2152 NOS1 4842 DRUGGABLE GENOME, ENZYME SOY PROTEIN 15328066 3233 2153 UBE2N 7334 ENZYME, DRUGGABLE GENOME NSC-60340 CHEMBL1534034 3234 2154 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR CI-1040 CI-1040 3235 2155 CUL4A 8451 ENZYME, DNA REPAIR, CLINICALLY ACTIONABLE inhibitor CHEMBL848 LENALIDOMIDE 3237 2156 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CISPLATIN CISPLATIN 19434073 3239 2157 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 252166843 3241 2158 CEACAM1 634 KINASE, CELL SURFACE, DRUGGABLE GENOME CHEMOKINES 15937057 3242 2159 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE TRAMETINIB TRAMETINIB 30835257 3245 2160 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ADM 9382956 3247 2161 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 8 3248 2162 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME activator 135651442 3251 2163 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 363894199 3253 2164 ALOX15B 247 DRUGGABLE GENOME, ENZYME E324 E324 3254 2165 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PANITUMUMAB PANITUMUMAB 3255 2166 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 223365885 DOTHIEPIN 3256 2167 ATXN2 6311 NA SJ000154295 CHEMBL578502 3257 2168 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US20138552206 5 3259 2169 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FANDOSENTAN POTASSIUM FANDOSENTAN POTASSIUM 3260 2170 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME BREVAREX MAB 3261 2171 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CSA CYCLOSPORINE 17477024 3262 2172 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 387065614 3263 2173 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME RG2833 3265 2174 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 187051805 QUISINOSTAT 3266 2175 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GNF-PF-3716 CHEMBL609606 3267 2176 CELSR2 1952 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME hmg coa reductase inhibitors 25350695 3269 2177 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE PAZOPANIB PAZOPANIB 3272 2178 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR conjugated estrogens 9860300 3273 2179 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AGM-1470 O-CHLOROACETYLCARBAMOYLFUMAGILLOL 8012959 3275 2180 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650527 3276 2181 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist 404859091 CILOFEXOR 3277 2182 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THIOGUANOSINE THIOGUANOSINE 3279 2183 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR PF-562271 PF-00562271 3280 2184 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker 135651305 VERAPAMIL 3283 2185 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE AP1903 RIMIDUCID 3284 2186 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Seribantumab SERIBANTUMAB 3285 2187 TRH 7200 DRUGGABLE GENOME ERYTHRO 4219111 3286 2188 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME FENOFIBRATE FENOFIBRATE 11356390 3287 2189 POLB 5423 DNA REPAIR, DRUGGABLE GENOME STREPTONIGRIN STREPTONIGRIN 3288 2190 CBX1 10951 NA DNDI1417614 CHEMBL1567571 3289 2191 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME ENALAPRIL ENALAPRIL 16678199 3290 2192 BAZ2B 29994 NA GNF-PF-4992 CHEMBL275177 3291 2193 PPCDC 60490 ENZYME trastuzumab TRASTUZUMAB 3292 2194 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CB7969312 CHEMBL599255 3293 2195 UBE2N 7334 ENZYME, DRUGGABLE GENOME THONZONIUM BROMIDE THONZONIUM BROMIDE 3294 2196 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565648 3295 2197 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor 178102596 3298 2198 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-209931 CHEMBL472656 3300 2199 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-3561 CHEMBL599712 3301 2200 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ICI-164384 CHEMBL1222035 20659801 3303 2201 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-34a 3305 2202 F5 2153 DRUGGABLE GENOME rivaroxaban RIVAROXABAN 3307 2203 ATXN2 6311 NA PYRITHIONE PYRITHIONE 3308 2204 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE 178101724 3310 2205 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME BELINOSTAT BELINOSTAT 25937017 3311 2206 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545296 ARQ-736 3314 2207 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 384403668 3318 2208 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL2105728 CRENOLANIB 3319 2209 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PMID27376512-Compound-MTC-423 3320 2210 TAC1 6863 DRUGGABLE GENOME HUMAN CHORIONIC GONADOTROPIN 14706561 3321 2211 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Trametinib TRAMETINIB 27659046 3322 2212 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME DASATINIB DASATINIB 3323 2213 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor 178103434 METHAZOLAMIDE 3325 2214 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DIHYDRO-OBLIQUIN DIHYDRO-OBLIQUIN 3327 2215 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AMILORIDE HYDROCHLORIDE AMILORIDE HYDROCHLORIDE 3328 2216 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Piperazine derivative 6 3329 2217 HDAC11 79885 DRUGGABLE GENOME, ENZYME DAUNORUBICIN DAUNORUBICIN 22260166 3331 2218 PPAT 5471 DRUGGABLE GENOME, ENZYME Azathioprine AZATHIOPRINE 3332 2219 MPHOSPH8 54737 NA INDIRUBIN SULFATE SU-9516 3333 2220 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME paclitaxel PACLITAXEL 22441531 3334 2221 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME ATryn antithrombin 24391399 3338 2222 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AG-370 CHEMBL59150 3339 2223 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 3340 2224 CMKLR1 1240 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100364 3341 2225 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME DICHLOROPHEN DICHLOROPHEN 3342 2226 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 252166657 3347 2227 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ETHANOL ALCOHOL 8576634 3348 2228 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL49642 INDIBULIN 3349 2229 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1201570 ANAKINRA 3350 2230 MARK1 4139 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565590 CHEMBL1236539 3352 2231 HPSE 10855 ENZYME, DRUGGABLE GENOME ANTIESTROGEN 14695198 3353 2232 GJA3 2700 ION CHANNEL, TRANSPORTER inhibitor 135652731 3354 2233 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME THALIDOMIDE THALIDOMIDE 15939924 3355 2234 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702262 ROGARATINIB 3356 2235 DPP9 91039 PROTEASE, ENZYME, DRUGGABLE GENOME Talabostat TALABOSTAT 3357 2236 TK1 7083 ENZYME, KINASE, DRUGGABLE GENOME Thymidine kinase-expressing adenovirus and ganciclovir suicide gene therapy 3360 2237 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RAPAMYCIN SIROLIMUS 17652445 3361 2238 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2016054807Example71 3363 2239 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20100022547C86 3367 2240 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME PMID27998201-Compound-6 3369 2241 PSMB9 5698 DRUGGABLE GENOME, PROTEASE, ENZYME CARFILZOMIB CARFILZOMIB 24524217 3370 2242 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME QUERCETIN QUERCETIN 3372 2243 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME ELLIPTECINE ELLIPTECINE 3373 2244 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BRIMONIDINE BRIMONIDINE 3374 2245 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650038 3375 2246 AKR1C3 8644 ENZYME, DRUGGABLE GENOME ASP-9521 3378 2247 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GDC-0941 PICTILISIB 23674493,27174596,24601221,22084396,27020857,23136191,24339963,27197306,26058079,27604488,27196766,28119489 3379 2248 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-724440 CHEMBL515617 3380 2249 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE CYC-116 CYC-116 3381 2250 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY PMA 8879350 3382 2251 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME VANOXERINE VANOXERINE 3383 2252 ALOX15 246 ENZYME, DRUGGABLE GENOME ATHRAQUINONES A ATHRAQUINONES A 3385 2253 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIPYRIDAMOLE DIPYRIDAMOLE 3388 2254 ANGPTL3 27329 DRUGGABLE GENOME, FIBRINOGEN, CELL SURFACE, GROWTH FACTOR AKCEA-ANGPTL3-LRX VUPANORSEN 3389 2255 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PLX7486 3390 2256 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CB7969312 CHEMBL599255 3393 2257 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TROVAFLOXACIN MESYLATE TROVAFLOXACIN MESYLATE 3394 2258 IFNG 3458 DRUGGABLE GENOME CIGB-128 3395 2259 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME BENZOTHIAZOL-2-YLAMINE CHEMBL329785 22982122 3396 2260 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PF-3463275 PF-03463275 3397 2261 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor 328083505 3399 2262 SMN2 6607 DRUGGABLE GENOME DESMETHOXYYANGONIN DESMETHOXYYANGONIN 3400 2263 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 187051807 SCRIPTAID 3402 2264 PTGES 9536 DRUGGABLE GENOME, ENZYME Benzimidazole derivative 13 3404 2265 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR TESTOSTERONE TESTOSTERONE 3405 2266 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME activator 135650283 3406 2267 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 187051792 PANOBINOSTAT 3407 2268 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME RO-5212054 RG-7256 3409 2269 BIRC7 79444 PROTEASE INHIBITOR, TUMOR SUPPRESSOR, DRUG RESISTANCE antagonist 223366066 GDC-0152 3410 2270 SMN2 6607 DRUGGABLE GENOME 3',4'-DIHYDROXYFLAVONE CHEMBL222556 3411 2271 MLKL 197259 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE inhibitor 336446900 3412 2272 CSF3 1440 GROWTH FACTOR, DRUGGABLE GENOME TALABOSTAT TALABOSTAT 3414 2273 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1951071 ARFORMOTEROL TARTRATE 3420 2274 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2011137219 37(4-6) 3421 2275 GBA 2629 DRUGGABLE GENOME, ENZYME AFEGOSTAT AFEGOSTAT 21250698 3423 2276 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE trastuzumab emtansine 28040715,24879797,21458915,26920887 3425 2277 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME TURBINATINE TURBINATINE 15568781 3428 2278 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR CYC-116 CYC-116 3432 2279 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135650094 CICAPROST 3434 2280 HSPB1 3315 DRUGGABLE GENOME QUERCETIN QUERCETIN 19296652 3435 2281 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR FURAFYLLINE FURAFYLLINE 3437 2282 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CXR-1002 3438 2283 XDH 7498 DRUGGABLE GENOME, ENZYME Azaindole derivative 4 3439 2284 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652642 3441 2285 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY RETINOIDS 12182039 3444 2286 KDM4A 9682 DRUGGABLE GENOME, ENZYME PYRITHIONE PYRITHIONE 3445 2287 GMNN 51053 DRUGGABLE GENOME FALNIDAMOL FALNIDAMOL 3447 2288 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL1950289 TANZISERTIB 3448 2289 ATAD5 79915 NA DNDI1417013 CHEMBL1452227 3449 2290 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CANTHARIDIN CANTHARIDIN 3450 2291 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME noroxymorphone 3451 2292 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-48 3453 2293 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE irinotecan IRINOTECAN 21273624,16456808 3454 2294 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL6318 IDOXIFENE 3455 2295 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AGROCLAVINE AGROCLAVINE 3456 2296 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 OMEPRAZOLE OMEPRAZOLE 22931300 3457 2297 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649910 3459 2298 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Paroxetine PAROXETINE 3460 2299 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051797 APICIDIN 3464 2300 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DOCONEXENT DOCONEXENT 20695472 3466 2301 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE BC21 22224445 3467 2302 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GLIQUIDONE GLIQUIDONE 3468 2303 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 252827493 3471 2304 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE CYC-116 CYC-116 3472 2305 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME ARQ 736 3476 2306 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Anakinra ANAKINRA 3477 2307 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LAPATINIB LAPATINIB 25590338,19718025 3478 2308 TUBB 203068 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 3479 2309 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LOPERAMIDE LOPERAMIDE 3481 2310 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 405067321 3482 2311 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PANOBINOSTAT PANOBINOSTAT 3484 2312 KCNT2 343450 ION CHANNEL, DRUGGABLE GENOME blocker 135651249 3486 2313 GMNN 51053 DRUGGABLE GENOME MECLIZINE DIHCL MECLIZINE DIHCL 3488 2314 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE GAMBOGIC AMIDE GAMBOGIC AMIDE 17911251 3494 2315 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651094 SULPROSTONE 3495 2316 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor SORAFENIB SORAFENIB 3496 2317 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 252827496 3498 2318 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545420 AG-24322 3500 2319 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE TAK-114 3503 2320 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Losartan LOSARTAN 3504 2321 HSPB1 3315 DRUGGABLE GENOME TYROSINE KINASE INHIBITOR 8875961 3505 2322 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 flutamide FLUTAMIDE 9187528 3508 2323 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE 12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE 3509 2324 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE glucocorticoids 25157341 3510 2325 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 223366031 3511 2326 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BAS-8770957 CHEMBL500812 19179076 3512 2327 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker 178101077 3514 2328 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER TETRAETHYLAMMONIUM CHLORIDE TETRAETHYLAMMONIUM CHLORIDE 3515 2329 RORA 6095 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE agonist 381118853 3516 2330 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HARMAN HARMAN 3518 2331 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL1946170 REGORAFENIB 3520 2332 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE SUNITINIB SUNITINIB 23583911 3521 2333 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR PROTEIN SYNTHESIS INHIBITOR 1735464 3524 2334 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME GW441756X GW441756X 3525 2335 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Quinoline derivative 11 3526 2336 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GUAIFENESIN GUAIFENESIN 22931300 3527 2337 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME YUANHUADINE YUANHUADINE 21916433 3528 2338 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME BUSULFAN BUSULFAN 9389690 3529 2339 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR BUTYRYLHYDROXAMIC ACID BUTYRYLHYDROXAMIC ACID 21874153 3532 2340 ATXN2 6311 NA SANGUINARIUM SANGUINARIUM 3536 2341 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE DEXPROPRANOLOL DEXPROPRANOLOL 3537 2342 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GRAMINE GRAMINE 3538 2343 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AZD1480 AZD-1480 21926964 3539 2344 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Aryl carboxamide derivative 4 3540 2345 UBE2N 7334 ENZYME, DRUGGABLE GENOME AMINODIMETHOXYQUINAZOLINYLPIPERAZINE AMINODIMETHOXYQUINAZOLINYLPIPERAZINE 3541 2346 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL3545188 PASIREOTIDE PAMOATE 3542 2347 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 223366064 SARACATINIB 3543 2348 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor MIDOSTAURIN MIDOSTAURIN 3545 2349 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Carboxamide derivative 10 3546 2350 ATXN2 6311 NA (+/-)-OCTOCLOTHEPIN MALEATE CHEMBL1256660 3550 2351 MUC16 94025 DRUGGABLE GENOME CHEMBL1742981 ABAGOVOMAB 3552 2352 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME FLUDIOXONIL FLUDIOXONIL 3553 2353 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565922 3554 2354 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Pyrrolo-pyridone derivative 3 3555 2355 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME MYRICETIN MYRICETIN 3556 2356 KDM4A 9682 DRUGGABLE GENOME, ENZYME DIMETHYLPHENYLPIPERAZINIUM IODIDE DIMETHYLPHENYLPIPERAZINIUM IODIDE 3557 2357 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER TCMDC-125620 CHEMBL530291 3558 2358 RTN4 57142 DRUGGABLE GENOME inhibitor CHEMBL2108679 OZANEZUMAB 3559 2359 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Etirinotecan pegol 3560 2360 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CGRP CALCITONIN GENE-RELATED PEPTIDE 3563 2361 ABHD6 57406 PHOSPHOLIPASE, ENZYME Piperazine carbamic compound 2 3564 2362 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME flupirtine FLUPIRTINE 26959717 3565 2363 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR 5-BROMODEOXYURIDINE 2537681 3568 2364 ATIC 471 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE METHOTREXATE METHOTREXATE 3860829 3569 2365 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-33 3570 2366 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE ACETYLDIGITOXIN ACETYLDIGITOXIN 3571 2367 DES 1674 NA TPA ALTEPLASE 7507197 3572 2368 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME METHACYCLINE HYDROCHLORIDE METHACYCLINE HYDROCHLORIDE 3573 2369 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR antagonist 135650518 3574 2370 ARID1A 8289 CLINICALLY ACTIONABLE GSK126 25686104 3577 2371 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 252166602 NANATINOSTAT 3578 2372 GJA3 2700 ION CHANNEL, TRANSPORTER inhibitor 135650269 3580 2373 DHFR 1719 DRUGGABLE GENOME, ENZYME METHOTREXATE METHOTREXATE 3581 2374 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-720622 CHEMBL1287980 3586 2375 ATAD5 79915 NA DOXAZOSIN DOXAZOSIN 3589 2376 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME activator 336446902 SRT-2104 3590 2377 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-699479 CHEMBL1701915 3591 2378 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LY-2090314 LY-2090314 3592 2379 HTT 3064 DRUGGABLE GENOME PMID28092474-Compound-33 3593 2380 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR tideglusib TIDEGLUSIB 3594 2381 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME CID 3237815 CHEMBL410484 3595 2382 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER DEXTROMETHORPHAN DEXTROMETHORPHAN 15582917 3597 2383 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SJ000293754 CHEMBL486706 3600 2384 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-27 3602 2385 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Isoflavone derivative 5 3604 2386 GLS 2744 ENZYME THUNBERGINOL B THUNBERGINOL B 3606 2387 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CI-218872 CI-218872 3607 2388 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE GNF-PF-2272 CHEMBL601757 3608 2389 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROPERICIAZINE PERICIAZINE 3609 2390 HTT 3064 DRUGGABLE GENOME GNF-PF-2324 CHEMBL577419 3610 2391 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1417097 CHEMBL1531222 3611 2392 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NITAZOXANIDE NITAZOXANIDE 3612 2393 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-54 3613 2394 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-(2-HYDROXYBENZYL)PHENOL CHEMBL148831 3614 2395 PTGDS 5730 ENZYME, TRANSPORTER, DRUGGABLE GENOME HORMONES 10387044 3615 2396 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-12 3617 2397 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PAZOPANIB PAZOPANIB 28221861 3618 2398 BAZ2B 29994 NA GNF-PF-5029 CHEMBL600360 3619 2399 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE PRT-062607 PRT-2607 24419749 3620 2400 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200472 QUAZEPAM 3622 2401 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL3545295 AVE0847 3623 2402 CYB5R3 1727 DRUGGABLE GENOME, ENZYME methylene blue 3628 2403 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 3629 2404 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 315661144 PF-04995274 3630 2405 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE acetaminophen / codeine 3631 2406 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SALMETEROL SALMETEROL 3632 2407 GLA 2717 ENZYME, DRUGGABLE GENOME Deoxynojirimycin DUVOGLUSTAT 3633 2408 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GOSSYPETIN GOSSYPETIN 3634 2409 MAPT 4137 DRUGGABLE GENOME NSC-632536 CHEMBL1367933 3636 2410 VKORC1 79001 DRUGGABLE GENOME, ENZYME Tecarfarin TECARFARIN 3639 2411 MAPT 4137 DRUGGABLE GENOME 3,3',4'-TRIHYDROXYFLAVONE CHEMBL122701 3640 2412 STAT2 6773 TRANSCRIPTION FACTOR, KINASE 13-CIS-RETINOIC ACID 11032398 3641 2413 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SELEGILINE SELEGILINE 22931300 3642 2414 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE inhibitor 249565754 3644 2415 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENPYROXYMATE FENPYROXYMATE 3645 2416 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM BROMIDE 3646 2417 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1201012 FLURANDRENOLIDE 3647 2418 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Porfimer Sodium 3648 2419 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102905 3649 2420 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DESIPRAMINE DESIPRAMINE 3650 2421 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER cyclophosphamide CYCLOPHOSPHAMIDE 3655 2422 ARRB2 409 ION CHANNEL, G PROTEIN COUPLED RECEPTOR tramadol TRAMADOL 30549211 3656 2423 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR 12-EPISCALARIN CHEMBL269105 17988093 3657 2424 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR L-PHENYLALANINE PHENYLALANINE 3658 2425 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME DCC-3014 3660 2426 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL1079593 VS-5584 3661 2427 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 310264724 LY-3009120 3662 2428 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PODOFILOX PODOFILOX 3663 2429 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Navitoclax NAVITOCLAX 27197306 3665 2430 GJB2 2706 ION CHANNEL, TRANSPORTER inhibitor 135652731 3668 2431 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ALSTERPAULLONE ALSTERPAULLONE 3669 2432 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135652725 VINCAMINE 3670 2433 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PX-478 PX-478 3671 2434 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 3672 2435 TAT 6898 ENZYME TETRACYCLINE TETRACYCLINE 2154 3674 2436 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200602 3675 2437 DTNBP1 84062 KINASE methamphetamine METHAMPHETAMINE 17555717 3676 2438 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200703 CHLORDIAZEPOXIDE HYDROCHLORIDE 3677 2439 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417055 CHEMBL1486366 3678 2440 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-124266 CHEMBL124006 3680 2441 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ETHANOL ALCOHOL 12641735 3685 2442 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL236593 TELCAGEPANT 3686 2443 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR GM-CSF REGRAMOSTIM 8662788 3687 2444 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 252827520 DUBERMATINIB 3688 2445 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PMID29130358-Compound-SB-3CT 3690 2446 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL378544 VINBLASTINE SULFATE 3691 2447 TDO2 6999 ENZYME, DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 6136271 3692 2448 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SR-59230A CHEMBL1326499 3693 2449 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR AFIMOXIFENE AFIMOXIFENE 20334368,24805199 3694 2450 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-125034 CHEMBL239439 3696 2451 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MEDROXYPROGESTERONE ACETATE MEDROXYPROGESTERONE ACETATE 3697 2452 KDM4A 9682 DRUGGABLE GENOME, ENZYME 2-HYDROXYPHENAZINE 5,10-DIOXIDE CHEMBL179611 3698 2453 ALDH1A1 216 DRUGGABLE GENOME, ENZYME Z-PRO-PROLINAL Z-PRO-PROLINAL 3701 2454 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR VEMURAFENIB VEMURAFENIB 22197931,7651428,18632602,19915144,23569304,25157968 3703 2455 MIF 4282 DRUGGABLE GENOME, CELL SURFACE ANTI-MIF MONOCLONAL ANTIBODY 3704 2456 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ETHYL EICOSAPENTAENOIC ACID 3705 2457 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545396 BMS-690514 3706 2458 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL592445 GEDATOLISIB 3707 2459 ALOX15B 247 DRUGGABLE GENOME, ENZYME DIENESTROL DIENESTROL 3709 2460 PRMT3 10196 DRUGGABLE GENOME, METHYL TRANSFERASE, ENZYME inhibitor 178103611 3712 2461 NOX4 50507 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 363894228 3713 2462 SLC28A2 9153 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME ADENOSINE ADENOSINE 23388705 3717 2463 GMNN 51053 DRUGGABLE GENOME NIFURALDEZONE NIFURALDEZONE 3718 2464 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CHEMBL591 ETHCHLORVYNOL 3720 2465 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR CENISERTIB CENISERTIB 3721 2466 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DIFLUNISAL DIFLUNISAL 3722 2467 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TERAZOSIN TERAZOSIN 3723 2468 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BUTYLATED HYDROXYTOLUENE BUTYLATED HYDROXYTOLUENE 22931300 3724 2469 FGB 2244 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, FIBRINOGEN, DRUGGABLE GENOME inhibitor CHEMBL1201505 FIBRINOLYSIN, HUMAN 3725 2470 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-23 3727 2471 PTGS1 5742 ENZYME, DRUGGABLE GENOME MEFENAMIC ACID 3728 2472 MYO9B 4650 NA SALT VOLANESORSEN SODIUM 8987990 3729 2473 CXCL2 2920 DRUGGABLE GENOME BCG BCG VACCINE 18217952 3730 2474 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 252827368 PEXIDARTINIB 3731 2475 NT5C2 22978 ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE didanosine DIDANOSINE 23315321 3732 2476 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Quinoline and quinazoline derivative 4 3735 2477 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR RADANAMYCIN RADANAMYCIN 16464590 3736 2478 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PD-0166285 PD-0166285 3738 2479 SCNN1A 6337 DRUGGABLE GENOME, ION CHANNEL triamterene TRIAMTERENE 23788015 3740 2480 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ZARDAVERINE ZARDAVERINE 3742 2481 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL2177390 IPATASERTIB 3743 2482 MAPT 4137 DRUGGABLE GENOME GNF-PF-4085 CHEMBL528181 3746 2483 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Dacomitinib DACOMITINIB 3747 2484 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2109621 ABITUZUMAB 3748 2485 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME methimazole METHIMAZOLE 3749 2486 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE IL-1 8844493,9923819,2162889 3750 2487 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW837331X GW837331X 3751 2488 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2326966 SF-1126 3752 2489 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE HYPERICIN HYPERICIN 3754 2490 SERPINA6 866 DRUGGABLE GENOME, PROTEASE INHIBITOR RIMEXOLONE RIMEXOLONE 3756 2491 RRM2 6241 DRUGGABLE GENOME, ENZYME Hydroxyurea HYDROXYUREA 3757 2492 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Indolinone derivative 1 3758 2493 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 3759 2494 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9216972, 67 3760 2495 MAPT 4137 DRUGGABLE GENOME HOE-33342 CHEMBL343002 3761 2496 XDH 7498 DRUGGABLE GENOME, ENZYME FEBUXOSTAT FEBUXOSTAT 3762 2497 CD52 1043 DRUGGABLE GENOME Alemtuzumab ALEMTUZUMAB 3764 2498 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650081 3765 2499 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 223366182 3766 2500 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DEXAMETHASONE DEXAMETHASONE 16482568 3767 2501 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-93817 CHEMBL1509789 3768 2502 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME inhibitor GDC-0973 COBIMETINIB 3770 2503 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE E7449 2X-121 3771 2504 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE antibody 178101775 TRASTUZUMAB 3774 2505 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1307 CHEMBL585030 3775 2506 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE CP-868596 CRENOLANIB 3776 2507 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor DASATINIB DASATINIB 3777 2508 IFNG 3458 DRUGGABLE GENOME Emapalumab EMAPALUMAB 3781 2509 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 249565599 3782 2510 TUBA4A 7277 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 3784 2511 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR NORELGESTROMIN NORELGESTROMIN 3785 2512 CDKAL1 54901 ENZYME Dipeptidyl peptidase 4 (DPP-4) inhibitors 3787 2513 KDM4A 9682 DRUGGABLE GENOME, ENZYME APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 3788 2514 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME SELENIUM 16648561 3789 2515 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ranolazine RANOLAZINE 24433361 3790 2516 TPBG 7162 CELL SURFACE, DRUGGABLE GENOME CHEMBL1743045 NAPTUMOMAB ESTAFENATOX 3793 2517 RACGAP1 29127 NA GNF-PF-321 CHEMBL581044 3794 2518 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 681640 CHEMBL379975 3795 2519 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ZAPA ZAPA 3796 2520 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NSC-228155 CHEMBL505670 3799 2521 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-3149 CHEMBL582507 3800 2522 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 252166704 3801 2523 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 2-ANILINOPYRIDINE CHEMBL555260 3802 2524 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE NILOTINIB NILOTINIB 3803 2525 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 3804 2526 HSPB1 3315 DRUGGABLE GENOME inhibitor OGX-427 APATORSEN 3805 2527 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MIFEPRISTONE MIFEPRISTONE 3806 2528 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 404859135 3808 2529 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MESO-HEXESTROL MESO-HEXESTROL 3809 2530 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NIACIN RECEPTOR AGONIST 3812 2531 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 gliquidone GLIQUIDONE 24442125 3814 2532 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME ALTISSIMACOUMARIN C ALTISSIMACOUMARIN C 22799262 3815 2533 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE LOVASTATIN LOVASTATIN 2351867,7662319,1588827 3816 2534 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CARTEOLOL CARTEOLOL 3817 2535 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR HYDROMORPHONE HYDROMORPHONE 3818 2536 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 2',3'-DIHYDROXYFLAVONE CHEMBL242171 3820 2537 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AMIODARONE AMIODARONE 3821 2538 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE CB7969312 CHEMBL599255 3822 2539 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE KUL-7211 3824 2540 GMNN 51053 DRUGGABLE GENOME XANTHOANGELOL B XANTHOANGELOL B 3825 2541 RNASEH2A 10535 ENZYME PROGESTERONE PROGESTERONE 12080023 3826 2542 POLK 51426 DNA REPAIR, ENZYME RACEPINEPHRINE RACEPINEPHRINE 3830 2543 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme6Pyrrolo[2,3-d]pyrimidines 3831 2544 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545263 LGX-806 3832 2545 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE DACTOLISIB DACTOLISIB 3833 2546 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 135650271 FLUOXYMESTERONE 3834 2547 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL RO-229735 CHEMBL2170369 21751815 3835 2548 KDM4A 9682 DRUGGABLE GENOME, ENZYME LOMOFUNGIN LOMOFUNGIN 3836 2549 MYLK 4638 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor TOZASERTIB TOZASERTIB 19035792 3838 2550 TSPO 706 DRUGGABLE GENOME Imidazo[1,2-b]pyridazine acetamide derivative 5 3839 2551 TMEM97 27346 NA Fused aryl carbocycle derivative 3 3840 2552 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME IL-12 12895357 3842 2553 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ICARITIN ICARITIN 3844 2554 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor CHEMBL565612 SOTRASTAURIN 3845 2555 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER spironolactone SPIRONOLACTONE 3848 2556 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME mitotane MITOTANE 23524664 3849 2557 NAAA 27163 ENZYME, DRUGGABLE GENOME inhibitor 381118830 3851 2558 KRT19 3880 DRUGGABLE GENOME PD-98059 CHEMBL35482 15793288 3852 2559 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FELODIPINE FELODIPINE 3853 2560 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135651263 TIMOLOL 3856 2561 SMN2 6607 DRUGGABLE GENOME HYDRALAZINE HYDRALAZINE 3859 2562 CGA 1081 DRUGGABLE GENOME, HORMONE ACTIVITY VINBLASTINE VINBLASTINE 6181870 3862 2563 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ENOXAMAST ENOXAMAST 3863 2564 MAFB 9935 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Tumor necrosis factor alpha (TNF-alpha) inhibitors 3864 2565 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE lapatinib LAPATINIB 3865 2566 NDUFC2 4718 ENZYME inhibitor CHEMBL3545135 NV-128 3867 2567 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PIMETHIXENE PIMETHIXENE 3868 2568 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-2954 CHEMBL582722 3869 2569 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME PMID27774822-Compound-Figure10Example1 3870 2570 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE DETD-35 27048951 3871 2571 IL23A 51561 DRUGGABLE GENOME BRIAKINUMAB BRIAKINUMAB 3873 2572 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MONATEPIL MONATEPIL 3874 2573 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR allosteric modulator 223365961 COBIMETINIB 3876 2574 PSMD13 5719 NA inhibitor CARFILZOMIB CARFILZOMIB 3877 2575 GLA 2717 ENZYME, DRUGGABLE GENOME EBSELEN EBSELEN 3879 2576 PDE7A 5150 ENZYME, DRUGGABLE GENOME DYPHYLLINE DYPHYLLINE 3880 2577 GC 2638 DRUGGABLE GENOME cetuximab CETUXIMAB 29208668 3881 2578 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DESVENLAFAXINE DESVENLAFAXINE 3882 2579 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE MERCURIC CHLORIDE MERCURIC CHLORIDE 3884 2580 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2105683 NAPROXEN ETEMESIL 3885 2581 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME RESVERATROL RESVERATROL 23316803,23859249,18046409 3886 2582 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE VEMURAFENIB VEMURAFENIB 23288408 3889 2583 PTGS2 5743 DRUGGABLE GENOME, ENZYME atenolol ATENOLOL 3891 2584 GPR68 8111 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 404859017 3892 2585 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME thiotepa THIOTEPA 3893 2586 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CCT196969 25500121,15294323,17210691 3894 2587 TUBB 203068 DRUGGABLE GENOME Sphingosome Encapsulated Vinorelbine 3895 2588 MAPT 4137 DRUGGABLE GENOME DIHYDROERGOCRISTINE DIHYDROERGOCRISTINE 3896 2589 COMT 1312 DRUGGABLE GENOME, ENZYME methylphenidate METHYLPHENIDATE 29230023,23131881,24763183,18214865,18703939,22149470,24035255,21550019 3897 2590 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SJ000071854 CHEMBL602127 3898 2591 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 178102337 SORAFENIB 3899 2592 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AZITHROMYCIN AZITHROMYCIN 22931300 3900 2593 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ETHANOL ALCOHOL 8803617 3903 2594 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX ACACETIN ACACETIN 25190466 3904 2595 ALOX15 246 ENZYME, DRUGGABLE GENOME QUINOXALINE-2-CARBOXYLIC ACID CHEMBL151797 3906 2596 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000119988 CHEMBL589694 3908 2597 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102618 3909 2598 NT5C2 22978 ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE THIOGUANINE THIOGUANINE 23377183,23377281 3910 2599 CIC 23152 CLINICALLY ACTIONABLE, DRUG RESISTANCE TRAMETINIB TRAMETINIB 28178529 3911 2600 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545111 HEMAY-022 3912 2601 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135650378 ILOPROST 3914 2602 ATAD5 79915 NA N,N-HEXAMETHYLENEAMILORIDE N,N-HEXAMETHYLENEAMILORIDE 3915 2603 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 QUINIDINE QUINIDINE 22931300,19117415 3916 2604 HTT 3064 DRUGGABLE GENOME DNDI1417599 CHEMBL2094833 3917 2605 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER propranolol PROPRANOLOL 3918 2606 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TERBUTALINE TERBUTALINE 3920 2607 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR ROFECOXIB ROFECOXIB 15613743 3921 2608 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CEDIRANIB CEDIRANIB 3923 2609 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SJ000018300 CHEMBL590927 3924 2610 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme23MPPDerivatives 3925 2611 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CADMIUM DICHLORIDE CADMIUM DICHLORIDE 3927 2612 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TS-022 3929 2613 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE DS-7423 DS-7423 3930 2614 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 3931 2615 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME CLOCORTOLONE CLOCORTOLONE 3932 2616 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME TAMATINIB R-406 3933 2617 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor 178103723 CILOSTAZOL 3935 2618 HTT 3064 DRUGGABLE GENOME DNDI1416955 CHEMBL1327172 3936 2619 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 terfenadine TERFENADINE 15861034 3937 2620 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE AZD-1775 ADAVOSERTIB 3940 2621 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE AMINOGLUTETHIMIDE AMINOGLUTETHIMIDE 18256205 3941 2622 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DROSPIRENONE DROSPIRENONE 3942 2623 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650468 3943 2624 MPHOSPH8 54737 NA BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 3944 2625 ATAD5 79915 NA ANGUIDIN ANGUIDIN 3945 2626 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 16 3946 2627 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL876 MECLOFENAMATE SODIUM 3949 2628 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2-NITRO-ETHANOL CHEMBL324774 3950 2629 FOXO3 2309 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE RESVERATROL RESVERATROL 17513867 3951 2630 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200341 INDECAINIDE HYDROCHLORIDE 3952 2631 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor XL147 PILARALISIB 3953 2632 TH 7054 ENZYME, DRUGGABLE GENOME EPO EPOETIN ALFA 16368081 3958 2633 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 249565576 ENMD-2076 3960 2634 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME VERAPAMIL HYDROCHLORIDE VERAPAMIL HYDROCHLORIDE 3961 2635 RACGAP1 29127 NA KAEMPFEROL KAEMPFEROL 3963 2636 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR GANODERIOL F GANODERIOL F 22014750 3964 2637 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Navicixizumab NAVICIXIZUMAB 3966 2638 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DOMIPHEN BROMIDE DOMIPHEN BROMIDE 3967 2639 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CITRIC ACID CITRIC ACID 3968 2640 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE PENTOSTATIN PENTOSTATIN 3970 2641 ITGB5 3693 CELL SURFACE, DRUGGABLE GENOME CNTO-95 INTETUMUMAB 3972 2642 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TYRPHOSTIN 23 TYRPHOSTIN 23 3976 2643 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Ficlatuzumab FICLATUZUMAB 24901237 3977 2644 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CANAVANINE CANAVANINE 3978 2645 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-44 3980 2646 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-30 3982 2647 BRD7 29117 ENZYME inhibitor 252166773 3983 2648 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NSC-753576 CHEMBL2088731 22982122 3984 2649 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor DASATINIB DASATINIB 3985 2650 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MICHLER'S KETONE MICHLER'S KETONE 3986 2651 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PROPYLPYRAZOLETRIOL PROPYLPYRAZOLETRIOL 3987 2652 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE cisplatin CISPLATIN 3990 2653 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE QUINALIZARIN QUINALIZARIN 3993 2654 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BDBM50080559 3994 2655 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3301595 DASOTRALINE 3996 2656 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200903 SECOBARBITAL SODIUM 3998 2657 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Tamoxifen TAMOXIFEN 3999 2658 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PF-03715455 PF-03715455 21888439 4000 2659 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CHLORAMBUCIL CHLORAMBUCIL 4001 2660 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649887 4002 2661 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME P-BCMA-101 CAR-T cells 4003 2662 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Copanlisib COPANLISIB 27672108 4004 2663 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEFEROXAMINE MESYLATE DEFEROXAMINE MESYLATE 4006 2664 ADH1A 124 DRUGGABLE GENOME FOMEPIZOLE FOMEPIZOLE 4009 2665 ATAD5 79915 NA FLUSPIRILENE FLUSPIRILENE 4010 2666 ATXN2 6311 NA CYCLOVALONE CYCLOVALONE 4011 2667 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CHRYSENE-1,4-DIONE CHEMBL421215 4013 2668 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NU-1025 CHEMBL123904 4014 2669 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody FIGITUMUMAB FIGITUMUMAB 4015 2670 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ERGOCRYPTINE ERGOCRYPTINE 4018 2671 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE DOXYCYCLINE HYCLATE DOXYCYCLINE HYCLATE 4020 2672 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MPA PROGESTERONE 14659903 4022 2673 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR TRAMETINIB TRAMETINIB 4024 2674 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR VTP-43742 4026 2675 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE HYDROCORTISONE HYDROCORTISONE 2707640 4027 2676 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR VERTEPORFIN VERTEPORFIN 15505074 4028 2677 POLK 51426 DNA REPAIR, ENZYME SURAMIN HEXASODIUM SURAMIN HEXASODIUM 4029 2678 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-12 4030 2679 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR DEFIBROTIDE DEFIBROTIDE 12745658 4031 2680 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor AP26113 CHEMBL3397300 4033 2681 COL1A2 1278 DRUGGABLE GENOME Solubilized type 1 native bovine collagen 4035 2682 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 4036 2683 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-663284 CHEMBL337173 25703307 4037 2684 MAPT 4137 DRUGGABLE GENOME NSC-228155 CHEMBL505670 4038 2685 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 249565616 SAPANISERTIB 4039 2686 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Lapatinib LAPATINIB 4040 2687 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE CAR-GPC3 T cell 4041 2688 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE methamphetamine METHAMPHETAMINE 23880023 4042 2689 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2103795 AZILSARTAN KAMEDOXOMIL 4043 2690 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AKOS004227608 4044 2691 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME inhibitor ODANACATIB ODANACATIB 4045 2692 RRM2 6241 DRUGGABLE GENOME, ENZYME cytarabine CYTARABINE 24024897 4046 2693 CYP26B1 56603 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME TALAROZOLE TALAROZOLE 4048 2694 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SYM004 4049 2695 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR ALPHA-DIFLUOROMETHYLORNITHINE 15075199 4052 2696 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE METHOTREXATE METHOTREXATE 23652803 4053 2697 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME TERFENADINE TERFENADINE 4054 2698 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-132 4055 2699 CA12 771 DRUGGABLE GENOME celecoxib CELECOXIB 22336956 4057 2700 CCNK 8812 KINASE fluorouracil FLUOROURACIL 4058 2701 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL RANOLAZINE RANOLAZINE 4059 2702 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME CISPLATIN CISPLATIN 25924824,25082261 4060 2703 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME GALANTAMINE GALANTAMINE 4061 2704 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Ramucirumab RAMUCIRUMAB 4062 2705 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor MK0752 4063 2706 HTRA1 5654 ENZYME, DRUGGABLE GENOME, PROTEASE bevacizumab BEVACIZUMAB 22594510,23559864,23842101,23337555 4064 2707 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME KD-025 CHEMBL2005186 4065 2708 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME AMORFRUTIN A AMORFRUTIN A 25938459 4066 2709 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME MMV009085 CHEMBL581225 4067 2710 VIM 7431 DRUGGABLE GENOME ENU 3440878 4069 2711 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER vaccine AD.P53-DC 4070 2712 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ANDROGENS 12796696 4071 2713 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-29 4073 2714 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650947 4075 2715 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Sodium Ascorbate 4080 2716 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-US20130053382 37(4-6) 4081 2717 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 249565672 4082 2718 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SEMAPIMOD SEMAPIMOD 4085 2719 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1200485 SORAFENIB TOSYLATE 4086 2720 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 252827368 PEXIDARTINIB 4088 2721 TDO2 6999 ENZYME, DRUGGABLE GENOME inhibitor 315661101 4090 2722 FAAH 2166 ENZYME, DRUGGABLE GENOME ACETAMINOPHEN ACETAMINOPHEN 15987694 4091 2723 HSPA8 3312 TUMOR SUPPRESSOR CISPLATIN CISPLATIN 15378690 4093 2724 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PYRROLIDINE DITHIOCARBAMATE PYRROLIDINE DITHIOCARBAMATE 4094 2725 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME GW843682X GW843682X 4095 2726 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MINOXIDIL MINOXIDIL 22931300 4096 2727 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201638 INSULIN SUSP PROTAMINE ZINC PURIFIED PORK 4097 2728 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE INDIMITECAN INDIMITECAN 20630766 4098 2729 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PRACINOSTAT PRACINOSTAT 4100 2730 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLUFENAMIC ACID FLUFENAMIC ACID 4101 2731 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE THONZONIUM BROMIDE THONZONIUM BROMIDE 4102 2732 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER venetoclax VENETOCLAX 4105 2733 ARSA 410 DRUGGABLE GENOME, ENZYME RO-410960 CHEMBL1256291 4107 2734 SFTPB 6439 DRUGGABLE GENOME STZ STREPTOZOCIN 1386745 4108 2735 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-107022 CHEMBL1601846 4111 2736 ATAD5 79915 NA TCMDC-124353 CHEMBL529918 4112 2737 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MELPHALAN MELPHALAN 4114 2738 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME WIN-55212-2 WIN-552122 4115 2739 COMT 1312 DRUGGABLE GENOME, ENZYME Opicapone OPICAPONE 4117 2740 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE BMS-275291 REBIMASTAT 15041713 4118 2741 ALOX5 240 DRUGGABLE GENOME, ENZYME MESALAZINE MESALAMINE 4120 2742 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CRIZOTINIB CRIZOTINIB 26870817 4122 2743 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NLG8189 4123 2744 SLC33A1 9197 TRANSPORTER 178101262 4124 2745 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME CID 100335 CHEMBL1520346 4125 2746 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME TANNIC ACID TANNIC ACID 4128 2747 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PROPRANOLOL PROPRANOLOL 2903243,16680159 4129 2748 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME AICAR CHEMBL483849 17181154 4130 2749 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER HETEROCODEINE HETEROCODEINE 18311899 4131 2750 MAP2K5 5607 KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor SELUMETINIB SELUMETINIB 4132 2751 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 384403638 4133 2752 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME VORINOSTAT VORINOSTAT 19344175,19966789,26211462,23622981,22260166,20491440,21548582,19084294 4134 2753 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051799 DACINOSTAT 4135 2754 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TIMOLOL TIMOLOL 4136 2755 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AMDINOCILLIN AMDINOCILLIN 4137 2756 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-25 4139 2757 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER QUINONE 11713586 4140 2758 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651213 4144 2759 MR1 3140 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ANTITHYMOCYTE GLOBULIN 4145 2760 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY PC4 12665168 4146 2761 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MEPIVACAINE MEPIVACAINE 22931300 4147 2762 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE flucloxacillin FLOXACILLIN 30664875 4148 2763 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178102588 4149 2764 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TRIFLUOPERAZINE TRIFLUOPERAZINE 4150 2765 E2F1 1869 TRANSCRIPTION FACTOR DES DIETHYLSTILBESTROL 15545218 4151 2766 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 249565806 SILMITASERTIB 4153 2767 SPINT1 6692 PROTEASE INHIBITOR, DRUGGABLE GENOME SURAMIN SURAMIN 15590895 4155 2768 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor TRAMETINIB TRAMETINIB 4156 2769 TOP2B 7155 DRUGGABLE GENOME, ENZYME CAP-7.1 4157 2770 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Cyclic sulfonamide derivative 3 4159 2771 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178103560 AMLODIPINE 4161 2772 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ASARININ ASARININ 4162 2773 FMO3 2328 ENZYME, DRUGGABLE GENOME nicotine NICOTINE 28290528 4164 2774 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GENISTEIN GENISTEIN 16380645 4165 2775 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SOTRASTAURIN SOTRASTAURIN 4167 2776 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ABIETIC ACID ABIETIC ACID 24799257 4171 2777 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Nalidixic Acid 4172 2778 POLK 51426 DNA REPAIR, ENZYME PIRENOXINE PIRENOXINE 4173 2779 PLAUR 5329 DRUGGABLE GENOME, ENZYME, CELL SURFACE UROKINASE UROKINASE 4174 2780 RHBDF2 79651 ENZYME opioids 21622719 4175 2781 KDM4A 9682 DRUGGABLE GENOME, ENZYME MERCAPTOPURINE HYDRATE MERCAPTOPURINE 4176 2782 PTGS2 5743 DRUGGABLE GENOME, ENZYME OXAPROZIN OXAPROZIN 4177 2783 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TEGASEROD MALEATE TEGASEROD MALEATE 4179 2784 CAMKK2 10645 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE US9623028, Compound 101 4181 2785 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR Pirfenidone PIRFENIDONE 4182 2786 POLB 5423 DNA REPAIR, DRUGGABLE GENOME DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 4185 2787 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DNDI1417400 CHEMBL1362503 4186 2788 SLC28A2 9153 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME tenofovir disoproxil fumarate 31619748 4187 2789 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PAZOPANIB PAZOPANIB 4188 2790 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist CHEMBL38 TRETINOIN 4189 2791 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Quinazolinedione derivative 2 4190 2792 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL371405 MARIZOMIB 4195 2793 CNPY4 245812 NA Tumor necrosis factor alpha (TNF-alpha) inhibitors 24776844 4197 2794 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Dutogliptin DUTOGLIPTIN 4198 2795 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE SP-600125 SP-600125 4199 2796 DHFR 1719 DRUGGABLE GENOME, ENZYME inhibitor 178103443 PEMETREXED 4200 2797 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor CHEMBL428690 ALVOCIDIB 4202 2798 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE HEXACHLOROPHENE HEXACHLOROPHENE 4203 2799 ATAD5 79915 NA P-HYDROXYPHENETHYL ANISATE CHEMBL1078244 4204 2800 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Six-membered heterocyclic benzamide derivative 7 4205 2801 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody 310264711 ISTIRATUMAB 4206 2802 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR GO-6976 GO-6976 4207 2803 ALOX5 240 DRUGGABLE GENOME, ENZYME 6-DECYLSALICYLIC ACID CHEMBL416038 24231650 4209 2804 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE VX-809 LUMACAFTOR 4210 2805 RAB9A 9367 ENZYME, DRUGGABLE GENOME SB-206553 CHEMBL297784 4211 2806 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER inhibitor 252827460 4212 2807 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE LINIFANIB LINIFANIB 4213 2808 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME BRYOSTATIN-1 16483930 4214 2809 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-5007 CHEMBL1989853 4215 2810 GJB1 2705 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER inhibitor 135652731 4216 2811 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME aspirin ASPIRIN 15784113,19392989 4218 2812 HEXB 3074 ENZYME CIS-PLATINUM 6987030 4220 2813 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROGESTERONE PROGESTERONE 4222 2814 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124416 CHEMBL530664 4223 2815 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-133896 CHEMBL512908 4224 2816 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CROMOLYN CROMOLYN 22931300 4225 2817 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER 2'-HYDROXYCHALCONE 2'-HYDROXYCHALCONE 22112540 4228 2818 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME CID 4970947 CHEMBL1451921 4229 2819 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-130 CHEMBL578890 4232 2820 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PRODINE HYDROCHLORIDE ALPHAPRODINE HYDROCHLORIDE 4233 2821 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1120 BISMUTH SUBSALICYLATE 4234 2822 SF3B3 23450 DRUGGABLE GENOME PLADIENOLIDE B PLADIENOLIDE B 17643112 4236 2823 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CYSTEAMINE HYDROCHLORIDE CYSTEAMINE HYDROCHLORIDE 4238 2824 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL1201748 CABAZITAXEL 4240 2825 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TCMDC-125758 CHEMBL546797 4243 2826 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LY-367265 CHEMBL1079460 4245 2827 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER (S)-VERAPAMIL (S)-VERAPAMIL 17646169 4246 2828 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-37 4247 2829 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE TT-100 4249 2830 CSNK1E 1454 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor HTS-466284 CHEMBL261454 19035792 4250 2831 CD83 9308 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SULFASALAZINE SULFASALAZINE 11471196 4251 2832 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NORETHYNODREL NORETHYNODREL 4252 2833 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME GNF-PF-3023 CHEMBL535331 4253 2834 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DINACICLIB DINACICLIB 4255 2835 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LIPOTECAN 4256 2836 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE lumacaftor LUMACAFTOR 22698459,24561283,26137539,24038832,22293084,24973281,21825083,24392786,26823392,28325531,24796242,27334259,21976485,23891399 4257 2837 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Isosteric imidazolyl pyrimidine derivative 1 4261 2838 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME rucaparib RUCAPARIB 4262 2839 TXNRD1 7296 DRUGGABLE GENOME 4-aryl quinol derivative 7 4266 2840 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody NIMOTUZUMAB NIMOTUZUMAB 4268 2841 ATAD5 79915 NA 2-HYDROXY-NAPHTHALDEHYDE THIOSEMICARBAZONE CHEMBL505209 4269 2842 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DACTINOMYCIN DACTINOMYCIN 4270 2843 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR antagonist LCL161 LCL-161 4271 2844 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER ALTENUSIN ALTENUSIN 4272 2845 TOP2B 7155 DRUGGABLE GENOME, ENZYME VORELOXIN VOSAROXIN 4273 2846 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR Lenzilumab LENZILUMAB 4274 2847 ALAD 210 ENZYME Porphobilinogen 4275 2848 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR GLUCOCORTICOID 17079862 4278 2849 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103105 CANDOXATRILAT 4280 2850 CCL21 6366 DRUGGABLE GENOME ADENOVIRAL VECTOR 14613584 4285 2851 RGS4 5999 DRUGGABLE GENOME inhibitor 252827382 CHEMBL1476646 4288 2852 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 363894199 4289 2853 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME BIOCHANIN BIOCHANIN 4290 2854 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL30219 METHOHEXITAL SODIUM 4291 2855 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL315985 ESLICARBAZEPINE 4294 2856 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME FORMONONETIN FORMONONETIN 4295 2857 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME PACLITAXEL PACLITAXEL 16211241,15347474 4296 2858 RAB9A 9367 ENZYME, DRUGGABLE GENOME GRINIMIBINE GRINIMIBINE 4297 2859 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL526 PROPOFOL 4299 2860 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME ALPRAZOLAM ALPRAZOLAM 4302 2861 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AEE788 AEE-788 22046346 4304 2862 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 7,8,2'-TRIHYDROXYFLAVONE CHEMBL244707 4305 2863 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103884 OPROZOMIB 4306 2864 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE agonist CHEMBL1201716 MECASERMIN 4307 2865 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME NBQX NBQX 4308 2866 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX ANTISENSE OLIGONUCLEOTIDES 8035811 4309 2867 EPHA7 2045 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 4310 2868 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME FLUORANTHEN-3-YLAMINE CHEMBL103583 4312 2869 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Pitolisant PITOLISANT 4317 2870 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652031 4318 2871 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 310264675 CUDC-101 4319 2872 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL1743014 ETARACIZUMAB 4320 2873 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SERTRALINE HYDROCHLORIDE SERTRALINE HYDROCHLORIDE 4323 2874 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METHOCTRAMINE METHOCTRAMINE 4325 2875 PPCDC 60490 ENZYME FEC100 4326 2876 ALDH1A1 216 DRUGGABLE GENOME, ENZYME RETINOL RETINOL 4327 2877 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FUSARIC ACID FUSARIC ACID 4328 2878 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650477 4329 2879 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 4330 2880 PSMC6 5706 NA inhibitor CARFILZOMIB CARFILZOMIB 4332 2881 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME QUERCETIN QUERCETIN 4333 2882 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALL-TRANS RETINOIC ACID 9792441 4335 2883 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135651147 4336 2884 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR TRAMETINIB TRAMETINIB 4337 2885 TLR7 51284 DRUGGABLE GENOME MEDI9197 TELRATOLIMOD 4338 2886 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE DES DIETHYLSTILBESTROL 15545218 4339 2887 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Salicylic acid derivative 1 4342 2888 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor BKM120 BUPARLISIB 4343 2889 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 385612234 4345 2890 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LAROPIPRANT LAROPIPRANT 4346 2891 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GERONTOXANTHONE A GERONTOXANTHONE A 25838141 4347 2892 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME (-)-EPICATECHIN (-)-EPICATECHIN 4348 2893 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL2219421 RECILISIB 4349 2894 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME agonist CHEMBL1201566 DARBEPOETIN ALFA 4350 2895 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1416934 CHEMBL1989750 4351 2896 LSS 4047 ENZYME, DRUGGABLE GENOME inhibitor 178103329 4352 2897 SMN2 6607 DRUGGABLE GENOME RUTAECARPINE RUTAECARPINE 4355 2898 CACNA2D3 55799 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200382 BEPRIDIL HYDROCHLORIDE 4357 2899 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RP-67580 CHEMBL131171 4358 2900 ALOX15 246 ENZYME, DRUGGABLE GENOME MERCURIC CHLORIDE MERCURIC CHLORIDE 4359 2901 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME WITHAFERIN A WITHAFERIN A 22705001 4361 2902 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ALX-5407 CHEMBL180966 4363 2903 BAZ2B 29994 NA NSC-234945 CHEMBL260311 4364 2904 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VB4-845 OPORTUZUMAB MONATOX 4365 2905 PLD1 5337 ENZYME, DRUGGABLE GENOME inhibitor 252827439 4367 2906 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AZD4547 4370 2907 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ENALAPRIL ENALAPRIL 4371 2908 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker 135652715 SAXITOXIN 4373 2909 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME ethanol ALCOHOL 31595439 4374 2910 GLS 2744 ENZYME 2,3,4-TRIHYDROXYBENZOPHENONE CHEMBL1527 4375 2911 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME CHIR-99021 CHIR-99021 4376 2912 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor SB939 4380 2913 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER U-50488 U-50488 METHANE SULFONATE 4381 2914 SERPINB2 5055 PROTEASE INHIBITOR, DRUGGABLE GENOME UROKINASE UROKINASE 4382 2915 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME CA4P 12171907 4385 2916 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PREDNISOLONE PREDNISOLONE 4386 2917 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR VITAMIN K3H2 VITAMIN K3H2 4389 2918 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME hormonal contraceptives for systemic use 15208046,28750087,12069454,16769590 4390 2919 CES1 1066 DRUGGABLE GENOME, ENZYME inhibitor 178103312 4391 2920 MAPT 4137 DRUGGABLE GENOME NOREPINEPHRINE NOREPINEPHRINE 4392 2921 RGS4 5999 DRUGGABLE GENOME DIMETHYLPINOCEMBRIN DIMETHYLPINOCEMBRIN 4394 2922 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALSTERPAULLONE ALSTERPAULLONE 4395 2923 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BECATECARIN BECATECARIN 4397 2924 ATAD5 79915 NA 2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE CHEMBL502774 4398 2925 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 A-315456 CHEMBL362863 4402 2926 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE DEOXYCOFORMYCIN PENTOSTATIN 11969266 4403 2927 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME IMATINIB IMATINIB 4404 2928 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE IPP-204106 4405 2929 KLC1 3831 NA fluorouracil FLUOROURACIL 17549067 4406 2930 CXCL8 3576 DRUGGABLE GENOME E319 E319 4407 2931 COL1A2 1278 DRUGGABLE GENOME TNF-ALPHA 12393755 4408 2932 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103141 4410 2933 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor PCI-24781 ABEXINOSTAT 4412 2934 NQO2 4835 DRUGGABLE GENOME, ENZYME NSC-640566 CHEMBL1287867 21074425 4413 2935 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME PREDNISOLONE PREDNISOLONE 4418 2936 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 135651401 4419 2937 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor CHEMBL3545052 FIMEPINOSTAT 4420 2938 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE LOPERAMIDE LOPERAMIDE 4424 2939 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PENDIMETHALIN PENDIMETHALIN 4426 2940 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR (+)-THALIPORPHINE CHEMBL1397308 4427 2941 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LUCATUMUMAB LUCATUMUMAB 4428 2942 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR L-796568 CHEMBL111201 4430 2943 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 381744937 4431 2944 SOD2 6648 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE cyclophosphamide CYCLOPHOSPHAMIDE 4434 2945 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE UNOPROSTONE ISOPROPYL UNOPROSTONE ISOPROPYL 4435 2946 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR LAUROGUADINE LAUROGUADINE 4438 2947 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ESTRIOL E3 4439 2948 FGA 2243 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, FIBRINOGEN RETEPLASE RETEPLASE 4440 2949 LNPEP 4012 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, TRANSPORTER, PROTEASE US10059720, Example 82 4441 2950 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 329968432 4442 2951 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-3964 CHEMBL599088 4443 2952 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR PREDNISOLONE PREDNISOLONE 18447956 4444 2953 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor PANOBINOSTAT PANOBINOSTAT 4445 2954 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER Benzbromarone BENZBROMARONE 4446 2955 MDH2 4191 NA ALBUMIN ALBUMIN HUMAN 2932302 4448 2956 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 223366052 OSIMERTINIB 4450 2957 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CHIDAMIDE CHIDAMIDE 4451 2958 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL OPC-14523 4452 2959 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME agonist 348353636 CIBINETIDE 4453 2960 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL activator CHEMBL119549 ANDOLAST 4454 2961 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE TAK-700 ORTERONEL 4455 2962 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME SB-202190 SB-202190 4456 2963 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 felbamate FELBAMATE 9187528 4458 2964 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VORELOXIN VOSAROXIN 4460 2965 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 135649993 BICALUTAMIDE 4464 2966 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ARACHIDONYL TRIFLUOROMETHYLKETONE ARACHIDONYL TRIFLUOROMETHYLKETONE 4466 2967 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Dipivefrin DIPIVEFRIN 4467 2968 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BUSULFAN BUSULFAN 22931300 4468 2969 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Fasitibant chloride 4469 2970 RAB9A 9367 ENZYME, DRUGGABLE GENOME GENISTEIN GENISTEIN 4470 2971 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650469 4472 2972 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME ETAZOLATE ETAZOLATE 4473 2973 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 178104017 MIRABEGRON 4474 2974 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME THYROXINE THYROXINE 11059392 4476 2975 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR 2,3,4-TRIHYDROXYBENZOPHENONE CHEMBL1527 4477 2976 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 4-TERT-BUTYLCATECHOL CHEMBL220845 4479 2977 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MAO INHIBITORS 16669850 4481 2978 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DOXORUBICIN DOXORUBICIN 4483 2979 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE AZD-1480 AZD-1480 21138246,24978112 4484 2980 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NIACIN NIACIN 25737085 4485 2981 COMT 1312 DRUGGABLE GENOME, ENZYME TOLCAPONE TOLCAPONE 4486 2982 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME PROPOFOL PROPOFOL 4487 2983 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CAROTENOIDS 11237167 4489 2984 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ospemifene OSPEMIFENE 4490 2985 BAZ2B 29994 NA LANSOPRAZOLE LANSOPRAZOLE 4491 2986 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102101 4492 2987 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor VORINOSTAT VORINOSTAT 4493 2988 PBRM1 55193 CLINICALLY ACTIONABLE inhibitor 249565598 4495 2989 BRDT 676 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE TRIAZOLAM TRIAZOLAM 22137933 4496 2990 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME L-MIMOSINE L-MIMOSINE 4497 2991 TUBA1B 10376 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 4499 2992 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR EC145 VINTAFOLIDE 4501 2993 IL11 3589 DRUGGABLE GENOME, KINASE, GROWTH FACTOR ALENDRONATE ALENDRONIC ACID 12522661 4502 2994 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-48 4503 2995 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE ALISERTIB ALISERTIB 4505 2996 ALDH1A1 216 DRUGGABLE GENOME, ENZYME HOMOVANILLIC ACID HOMOVANILLIC ACID 4509 2997 HEBP1 50865 DRUGGABLE GENOME Trepenoid derivative 1 4510 2998 TAT 6898 ENZYME PROGESTERONE PROGESTERONE 9744518 4512 2999 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 249565718 CHEMBL573107 4515 3000 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR STAUROSPORINE STAUROSPORINE 9359403 4516 3001 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 249565928 LY-2584702 4517 3002 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL2103851 AMUVATINIB 4518 3003 GABBR2 9568 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL ARBACLOFEN ARBACLOFEN 4522 3004 TXNRD1 7296 DRUGGABLE GENOME ARSENIC TRIOXIDE 4524 3005 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME CERC-301 RISLENEMDAZ 4526 3006 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME AG-1879 CHEMBL406845 4527 3007 POLI 11201 DNA REPAIR CEPHALOCHROMIN CEPHALOCHROMIN 4529 3008 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL3545160 SU-014813 4530 3009 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-53 4531 3010 DGKB 1607 KINASE antipsychotics 31447353 4532 3011 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 3238892 CHEMBL261118 4534 3012 DGAT1 8694 ENZYME, DRUGGABLE GENOME Pyrazolo[1,5-a]pyrimidine derivative 29 4535 3013 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SNS-314 SNS-314 4536 3014 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL52885 ENMD-981693 4537 3015 NOS1 4842 DRUGGABLE GENOME, ENZYME PRAZOSIN PRAZOSIN 9322222 4538 3016 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist,antagonist 135650883 RALOXIFENE 4540 3017 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Fam-Trastuzumab Deruxtecan-nxki 4541 3018 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE rosuvastatin ROSUVASTATIN 20207952 4542 3019 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 3-(DIMETHYLAMINO)PHENOL CHEMBL225257 4544 3020 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME YUANHUADINE YUANHUADINE 21916433 4545 3021 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR antagonist 223366065 CHEMBL504559 4548 3022 IL18 3606 DRUGGABLE GENOME PPD 11882036 4550 3023 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135652701 LOVASTATIN 4552 3024 TSPO 706 DRUGGABLE GENOME Imidazo[1,2-b]pyridazine acetamide derivative 6 4553 3025 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME BAY 10-00394 4554 3026 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIOGLITAZONE PIOGLITAZONE 16447051 4555 3027 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3833357 BEGELOMAB 4556 3028 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME LY3202626 4557 3029 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE THYROXINE THYROXINE 12433937 4558 3030 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 tropisetron TROPISETRON 9187528 4560 3031 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE benazepril BENAZEPRIL 20079160 4561 3032 BAZ2B 29994 NA TCMDC-125134 CHEMBL546975 4563 3033 GCLM 2730 ENZYME PMSG 11780957 4564 3034 CRP 1401 DRUGGABLE GENOME rosuvastatin ROSUVASTATIN 21094359 4565 3035 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE GDC-0068 IPATASERTIB 4566 3036 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Five-and-six-membered heterocyclic compound 1 4567 3037 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1201754 RUFINAMIDE 4568 3038 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LEVOTHYROXINE LEVOTHYROXINE 4572 3039 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 223366208 BMS-690514 4574 3040 PGD 5226 ENZYME, DRUGGABLE GENOME PENICILLAMINE PENICILLAMINE 289317 4576 3041 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME N-PHENETHYLCINNAMAMIDE CHEMBL1305393 4578 3042 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Neratinib NERATINIB 26627007,26333383,26243863 4580 3043 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1742982 AFLIBERCEPT 4581 3044 PTGS1 5742 ENZYME, DRUGGABLE GENOME IBUPROFEN IBUPROFEN 4587 3045 ERAP2 64167 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE inhibitor 348353642 4588 3046 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME STREPTONIGRIN STREPTONIGRIN 4589 3047 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PHENAZINE PHENAZINE 4592 3048 CEACAM1 634 KINASE, CELL SURFACE, DRUGGABLE GENOME ARCITUMOMAB ARCITUMOMAB 4593 3049 PDE4A 5141 DRUGGABLE GENOME, ENZYME RONOMILAST 4595 3050 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BRADANICLINE BRADANICLINE 23126648 4596 3051 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PHA-767491 CHEMBL225519 4598 3052 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor PIMASERTIB PIMASERTIB 4599 3053 CDH23 64072 NA methylphenidate METHYLPHENIDATE 29382897 4600 3054 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE SIMVASTATIN SIMVASTATIN 16436088 4601 3055 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE PENICILLAMINE PENICILLAMINE 17666490 4602 3056 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SELEGILINE SELEGILINE 22931300 4603 3057 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GEFITINIB GEFITINIB 4604 3058 MUC5AC 4586 DRUGGABLE GENOME CHEMBL1743013 ENSITUXIMAB 4605 3059 BAZ2B 29994 NA GNF-PF-1947 CHEMBL585591 4606 3060 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE MK-2637 4607 3061 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-29 4608 3062 FAAH 2166 ENZYME, DRUGGABLE GENOME Imidazolyl urea derivative 1 4609 3063 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE Everolimus EVEROLIMUS 27507190 4611 3064 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME ABC294640 4612 3065 CA2 760 DRUGGABLE GENOME, ENZYME ACETAZOLAMIDE ACETAZOLAMIDE 4615 3066 ATXN2 6311 NA GNF-PF-211 CHEMBL582699 4616 3067 SLC6A15 55117 DRUGGABLE GENOME, TRANSPORTER LORATADINE LORATADINE 25318072 4618 3068 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CARBAMAZEPINE CARBAMAZEPINE 22931300 4619 3069 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist CHEMBL2105738 GALETERONE 4620 3070 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-50 4621 3071 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 363894186 TALABOSTAT 4622 3072 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE OLAPARIB OLAPARIB 20739657,26510020,32343890,28363999,20124459,24841718 4624 3073 GMNN 51053 DRUGGABLE GENOME ASTEMIZOLE ASTEMIZOLE 4626 3074 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME OSI-632 OSI-632 4628 3075 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TAK-285 TAK-285 23983820 4630 3076 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME JNJ-7706621 JNJ-7706621 4631 3077 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ROSE BENGAL ROSE BENGAL 4632 3078 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ENNIATIN B ENNIATIN B 4633 3079 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GO-6976 GO-6976 4637 3080 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SALICYLURIC ACID SALICYLURIC ACID 4638 3081 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 artesunate ARTESUNATE 18064444,18979093,19926036,19851082,18350255,12920490,12844133 4639 3082 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR VERAPAMIL VERAPAMIL 4640 3083 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE doxorubicin DOXORUBICIN 16330681 4641 3084 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-1134 CHEMBL600694 4642 3085 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME IMD-1041 IMD-1041 4643 3086 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PIMOZIDE PIMOZIDE 4645 3087 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME SJ000019194 CHEMBL592106 4646 3088 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MEQUITAZINE MEQUITAZINE 4647 3089 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME EBSELEN EBSELEN 4648 3090 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME RG-1530 RG-1530 4649 3091 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PLATINUM COMPOUND 25636205 4650 3092 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20169447134C85 4651 3093 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PIPOBROMAN PIPOBROMAN 4653 3094 SLC14A2 8170 TRANSPORTER nifedipine NIFEDIPINE 17344938 4655 3095 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Carboxamide derivative 6 4656 3096 GMNN 51053 DRUGGABLE GENOME GNF-PF-4659 CHEMBL584442 4658 3097 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE Tolperisone TOLPERISONE 4659 3098 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651481 DOXERCALCIFEROL 4660 3099 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178101947 RUBOXISTAURIN 4661 3100 CBX1 10951 NA DOPAMINE HYDROCHLORIDE DOPAMINE HYDROCHLORIDE 4664 3101 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 348353648 4666 3102 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650983 4667 3103 IL1B 3553 KINASE, DRUGGABLE GENOME ERYTHROMYCIN ERYTHROMYCIN 2534682 4668 3104 BAP1 8314 PROTEASE, TUMOR SUPPRESSOR, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE APITOLISIB APITOLISIB 28389374 4669 3105 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-20 4670 3106 FECH 2235 ENZYME Methyl aminolevulinate 4671 3107 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLORANIL CHLORANIL 4673 3108 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE VANDETANIB VANDETANIB 4674 3109 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME Nilotinib NILOTINIB 4675 3110 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE CYC-116 CYC-116 4677 3111 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor PALBOCICLIB PALBOCICLIB 4678 3112 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 223366077 RGB-286638 4680 3113 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 178102482 GRAPIPRANT 4685 3114 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AG-1288 CHEMBL166486 4686 3115 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 405067337 4688 3116 GPR68 8111 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 178102508 LORAZEPAM 4689 3117 ALPI 248 DRUGGABLE GENOME, ENZYME ISOQUERCETIN ISOQUERCETIN 4690 3118 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR goserelin GOSERELIN 4692 3119 SV2A 9900 DRUGGABLE GENOME, TRANSPORTER BRIVARACETAM BRIVARACETAM 4693 3120 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME rigosertib RIGOSERTIB 27104980 4695 3121 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-52 4696 3122 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING COLCHICINE COLCHICINE 4697 3123 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ZM-39923 HCL CHEMBL538798 4698 3124 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BVT.2733 4700 3125 CES1 1066 DRUGGABLE GENOME, ENZYME K-604 4701 3126 MAP3K9 4293 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL290352 CEP-1347 4703 3127 HMGCR 3156 ENZYME, DRUGGABLE GENOME SIMVASTATIN SIMVASTATIN 4704 3128 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TRICLABENDAZOLE TRICLABENDAZOLE 4705 3129 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE AR-12286 VEROSUDIL 4708 3130 CA9 768 DRUGGABLE GENOME, ENZYME 90Y-cG250 4709 3131 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PARTHENOLIDE PARTHENOLIDE 25190466 4710 3132 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TESTOSTERONE TESTOSTERONE 12796696 4711 3133 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME PENTOSAN POLYSULFATE 17071199 4712 3134 VIM 7431 DRUGGABLE GENOME GANGLIOSIDE GM2 7923401 4713 3135 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SALMETEROL XINAFOATE SALMETEROL XINAFOATE 4714 3136 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 citalopram CITALOPRAM 21546862 4715 3137 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor ARQ 197 4718 3138 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (R)-FLECAINIDE (R)-FLECAINIDE 4719 3139 TYMSOS 494514 NA azathioprine AZATHIOPRINE 26332308 4720 3140 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 25-HYDROXYCHOLESTEROL CHEMBL169046 23830695 4723 3141 MGLL 11343 DRUGGABLE GENOME, ENZYME inhibitor 252166807 4724 3142 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GENTIAN VIOLET GENTIAN VIOLET 4725 3143 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 363894177 4727 3144 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METRONIDAZOLE METRONIDAZOLE 4728 3145 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Affitope AD-01 22506132 4729 3146 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE CLOTRIMAZOLE CLOTRIMAZOLE 4730 3147 BAZ2B 29994 NA ZINC 02849675 CHEMBL605959 4731 3148 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3544999 SAMOTOLISIB 4732 3149 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Carbamide derivative 20 4734 3150 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SK&F-86002 CHEMBL313417 4735 3151 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-34 4736 3152 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE REGORAFENIB REGORAFENIB 4739 3153 GC 2638 DRUGGABLE GENOME Isosorbide Dinitrate 4740 3154 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME THALIDOMIDE THALIDOMIDE 4744 3155 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE prilocaine PRILOCAINE 4747 3156 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE SIROLIMUS SIROLIMUS 19122144 4750 3157 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PIMASERTIB PIMASERTIB 4752 3158 AOX1 316 DRUGGABLE GENOME Menadione MENADIONE 4754 3159 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE modulator CHEMBL1812161 VATIQUINONE 4755 3160 AKR1B1 231 DRUGGABLE GENOME, ENZYME inhibitor 178103983 LIDORESTAT 4756 3161 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL2104954 BALAMAPIMOD 4757 3162 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIAZOXIDE DIAZOXIDE 4758 3163 SMN1 6606 DRUGGABLE GENOME DESMETHOXYYANGONIN DESMETHOXYYANGONIN 4759 3164 CA2 760 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL17 DICHLORPHENAMIDE 4760 3165 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ENTRECTINIB ENTRECTINIB 4763 3166 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME (S)-NOMIFENSINE CHEMBL51697 4764 3167 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR neratinib NERATINIB 4765 3168 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ZM-39923 HCL CHEMBL538798 4766 3169 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3137317 SONIDEGIB PHOSPHATE 4767 3170 TUBA1C 84790 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 4768 3171 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SORAFENIB SORAFENIB 4769 3172 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR KAEMPFEROL KAEMPFEROL 4771 3173 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME fluvastatin FLUVASTATIN 27839692 4772 3174 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME VIRAL VECTOR 10911621 4773 3175 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33i 4775 3176 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR GDC-0068 IPATASERTIB 4777 3177 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE SOTRASTAURIN SOTRASTAURIN 4778 3178 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100381 4779 3179 TOP2B 7155 DRUGGABLE GENOME, ENZYME Nemorubicin NEMORUBICIN 4780 3180 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Bipyrazole derivative 1 4781 3181 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Doxorubicin DOXORUBICIN 26552700 4784 3182 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650582 4785 3183 TMEM97 27346 NA Fused aryl carbocycle derivative 4 4787 3184 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565907 4789 3185 ALOX15B 247 DRUGGABLE GENOME, ENZYME 3,3',4'-TRIHYDROXYFLAVONE CHEMBL122701 4790 3186 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-2844 CHEMBL576353 4792 3187 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor CHEMBL3545110 RIBOCICLIB 4793 3188 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c][1,2,4]benzotriazine derivative 2 4794 3189 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SURAMIN SURAMIN 4795 3190 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Imatinib IMATINIB 28514312 4796 3191 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Cetuximab CETUXIMAB 25838391,27002107,28179366,25605843 4797 3192 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE MK2206 MK-2206 4798 3193 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME PHA-767491 CHEMBL225519 4799 3194 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3544942 RONICICLIB 4800 3195 ALCAM 214 DRUG RESISTANCE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE FLUOROURACIL FLUOROURACIL 24708484 4802 3196 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Venetoclax VENETOCLAX 4803 3197 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Asciminib ASCIMINIB 4804 3198 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE THIOMERSAL THIMEROSAL 4805 3199 ORAI1 84876 TRANSCRIPTION FACTOR, ION CHANNEL, TRANSPORTER CM2489 4807 3200 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Fulvestrant FULVESTRANT 4808 3201 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GW843682X GW843682X 4809 3202 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE TAZAROTENE TAZAROTENE 16109552 4810 3203 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE SEMAGACESTAT SEMAGACESTAT 19443228 4812 3204 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GALETERONE GALETERONE 4813 3205 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 249565646 PILARALISIB 4815 3206 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HOMATROPINE METHYLBROMIDE HOMATROPINE METHYLBROMIDE 22931300 4816 3207 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE XL647 TESEVATINIB 4817 3208 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2218887 4818 3209 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE BETAMETHASONE BETAMETHASONE 17515865 4819 3210 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME antibody 315661194 4820 3211 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MANUMYCIN A MANUMYCIN A 4821 3212 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE PLX3397 PEXIDARTINIB 24583793 4824 3213 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker 135651503 4825 3214 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR TAXOL PACLITAXEL 8554977 4826 3215 ATXN2 6311 NA RALOXIFENE RALOXIFENE 4828 3216 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CEDIRANIB CEDIRANIB 4829 3217 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME INOSITOL INOSITOL 2847980 4830 3218 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE DS-7423 DS-7423 24504419 4831 3219 GMNN 51053 DRUGGABLE GENOME EFAROXAN EFAROXAN 4832 3220 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody TREMELIMUMAB TREMELIMUMAB 4833 3221 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1201141 IBUPROFEN LYSINE 4834 3222 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CID 867101 CHEMBL406557 4835 3223 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLOTRIMAZOLE CLOTRIMAZOLE 4836 3224 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MEPANIPYRIM MEPANIPYRIM 4837 3225 GATA2 2624 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX 5-AZACYTIDINE AZACITIDINE 12706120 4838 3226 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CHIR-99021 CHIR-99021 4841 3227 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MESTANOLONE MESTANOLONE 4842 3228 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL2103743 TOFACITINIB CITRATE 4843 3229 PTGS2 5743 DRUGGABLE GENOME, ENZYME KETOPROFEN KETOPROFEN 4844 3230 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200982 BUTABARBITAL SODIUM 4846 3231 NCOA1 8648 ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX TCMDC-123764 CHEMBL533226 4847 3232 NCOA3 8202 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, ENZYME TAMOXIFEN TAMOXIFEN 12618500 4848 3233 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ETHYNODIOL DIACETATE 4850 3234 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 249565693 4851 3235 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270010-Compound-Figure5-2 4853 3236 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE Sapanisertib SAPANISERTIB 25261369 4854 3237 USP1 7398 DNA REPAIR, PROTEASE, ENZYME BEXAROTENE BEXAROTENE 4855 3238 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME RHEIN RHEIN 4856 3239 CBX1 10951 NA U-73122 CHEMBL1256678 4857 3240 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PHENAZINE-1-CARBOXYLIC ACID PHENAZINE-1-CARBOXYLIC ACID 4859 3241 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Pyrimidinedione derivative 1 4860 3242 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TEPOTINIB TEPOTINIB 32469185,24061647 4861 3243 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE PMID25726713-Compound-48 4862 3244 FAAH 2166 ENZYME, DRUGGABLE GENOME Ketoheterocycle derivative 1 4863 3245 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME mycophenolate mofetil 24681964 4864 3246 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL741 LAMOTRIGINE 4866 3247 GMNN 51053 DRUGGABLE GENOME SORAFENIB SORAFENIB 4867 3248 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL1201748 CABAZITAXEL 4868 3249 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE AZD0530 SARACATINIB 4873 3250 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE VINBLASTINE SULFATE VINBLASTINE SULFATE 4875 3251 POLI 11201 DNA REPAIR HOMIDIUM BROMIDE HOMIDIUM BROMIDE 4876 3252 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER MYCOPHENOLIC ACID MYCOPHENOLIC ACID 4877 3253 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SJ000032152 CHEMBL590665 4878 3254 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME HAEMATOXYLIN HAEMATOXYLIN 4879 3255 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR sorafenib SORAFENIB 20124951 4880 3256 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650340 GW7845 4881 3257 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator CHEMBL1201476 ENOXAPARIN SODIUM 4883 3258 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TOZASERTIB TOZASERTIB 4884 3259 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE SAR245409 VOXTALISIB 24634413 4885 3260 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-20 4886 3261 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor GIVINOSTAT GIVINOSTAT 4887 3262 MPHOSPH8 54737 NA TAMOXIFEN CITRATE TAMOXIFEN CITRATE 4889 3263 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE MMV009085 CHEMBL581225 4890 3264 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME ROMIDEPSIN ROMIDEPSIN 4891 3265 GMNN 51053 DRUGGABLE GENOME TCMDC-124356 CHEMBL22062 4893 3266 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING ENTINOSTAT ENTINOSTAT 19966789,20491440 4896 3267 GUCY1B1 2983 DRUGGABLE GENOME positive modulator CHEMBL2107834 RIOCIGUAT 4897 3268 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE 2,2-dimethylbenzopyran derivative 1 4898 3269 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VALPROIC ACID 16328060 4899 3270 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE LYMPHOKINE-ACTIVATED KILLER CELLS 15893691 4901 3271 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650689 NALTRINDOLE 4902 3272 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HALOBETASOL PROPIONATE HALOBETASOL PROPIONATE 4903 3273 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL FLUDIAZEPAM FLUDIAZEPAM 4905 3274 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-13 4906 3275 SCARB1 949 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME peginterferon alfa-2a 4908 3276 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME quetiapine QUETIAPINE 23859574 4909 3277 NCAM1 4684 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CHEMBL2109634 ONCOLYSIN S 4911 3278 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ETAZOLATE ETAZOLATE 4915 3279 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME (-)-U-50488 (-)-U-50488 4918 3280 TUBB6 84617 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 4919 3281 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NITROXOLINE NITROXOLINE 4921 3282 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1228 OXYPHENBUTAZONE 4922 3283 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE propofol PROPOFOL 26771271 4924 3284 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR THROMBIN THROMBIN 10952976 4925 3285 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PMID29671355-Compound-62 4926 3286 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR VER-49009 CHEMBL365617 4927 3287 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE SJ000036432 CHEMBL591135 4929 3288 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1421 DASATINIB 4930 3289 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1779046 TARAFENACIN 4931 3290 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PILOCARPINE PILOCARPINE 15183516 4932 3291 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL allosteric modulator 135652747 4933 3292 PSMD11 5717 KINASE inhibitor CHEMBL325041 BORTEZOMIB 4936 3293 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Dapagliflozin Propanediol; Saxagliptin Hydrochloride 4937 3294 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME BRYOSTATIN BRYOSTATIN 22579485 4938 3295 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME MK2206 MK-2206 24265152 4939 3296 AQP9 366 ION CHANNEL HORMONES 15647391 4940 3297 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME Everolimus EVEROLIMUS 4941 3298 KCNH6 81033 DRUGGABLE GENOME, ION CHANNEL inhibitor 135652149 4942 3299 GMNN 51053 DRUGGABLE GENOME LIOTHYRONINE SODIUM LIOTHYRONINE SODIUM 4943 3300 POLI 11201 DNA REPAIR LAVENDUSTIN B LAVENDUSTIN B 4944 3301 CXCL8 3576 DRUGGABLE GENOME YANGONIN YANGONIN 4945 3302 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE agonist CHEMBL2108621 MAPATUMUMAB 4947 3303 PTGS2 5743 DRUGGABLE GENOME, ENZYME THALIDOMIDE THALIDOMIDE 4949 3304 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Durvalumab DURVALUMAB 27225694 4950 3305 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AV-412 MP-412 17888033 4954 3306 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CGP-53353 CGP-53353 4955 3307 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR IL-12 16026835 4957 3308 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR ETHANOL ALCOHOL 1744136 4958 3309 RGS4 5999 DRUGGABLE GENOME inhibitor 252827384 4962 3310 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL1614707 MUBRITINIB 4963 3311 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 nifedipine NIFEDIPINE 15634941 4965 3312 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3352 CHEMBL600306 4969 3313 BAZ2B 29994 NA 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 4971 3314 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE OSI-632 OSI-632 4973 3315 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME TCMDC-123749 CHEMBL524376 4974 3316 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE ANASTROZOLE ANASTROZOLE 18256205 4976 3317 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME rocuronium ROCURONIUM 25279974 4977 3318 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME Sorafenib SORAFENIB 4978 3319 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1079593 VS-5584 4979 3320 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE TYROSINE KINASE INHIBITOR 15383630 4980 3321 PDE4D 5144 DRUGGABLE GENOME, ENZYME ROLIPRAM ROLIPRAM 4981 3322 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMG-232 AMG-232 24456472 4982 3323 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE ANTI-HER3 MONOCLONAL ANTIBODY GSK2849330 29610121 4985 3324 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor SB939 4986 3325 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Phenylpyridine derivative 3 4990 3326 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-159 CHEMBL599924 4992 3327 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103487 4993 3328 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PYRILAMINE PYRILAMINE 22007643,16408006 4996 3329 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE IL-7 17023582 4997 3330 TXNRD1 7296 DRUGGABLE GENOME Binuclear gold(I) compound 1 4998 3331 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PEMBROLIZUMAB PEMBROLIZUMAB 31086949 4999 3332 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-15 5000 3333 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OXPRENOLOL OXPRENOLOL 5001 3334 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AMPEROZIDE HYDROCHLORIDE AMPEROZIDE HYDROCHLORIDE 5002 3335 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME GNF-PF-1702 CHEMBL600313 5003 3336 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER BAFETINIB BAFETINIB 18191450 5005 3337 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME BRYOSTATIN-1 5006 3338 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL2387080 TASELISIB 5007 3339 PMM2 5373 ENZYME EBSELEN EBSELEN 5008 3340 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-PG-11048 5010 3341 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE Belnacasan BELNACASAN 5012 3342 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME N-METHYL-D-ASPARTIC ACID (NMDA) N-METHYL-D-ASPARTIC ACID (NMDA) 5013 3343 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000047240 CHEMBL590706 5014 3344 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME ticagrelor TICAGRELOR 25935875 5015 3345 ARSA 410 DRUGGABLE GENOME, ENZYME GOSSYPOL GOSSYPOL 5016 3346 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 itraconazole ITRACONAZOLE 9187528 5018 3347 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417523 CHEMBL598663 5019 3348 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME Benzoimidazole derivative 2 5020 3349 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651269 TOLTERODINE 5022 3350 IL6ST 3572 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE BAZEDOXIFENE BAZEDOXIFENE 24456369 5023 3351 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME ERLOTINIB ERLOTINIB 5024 3352 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR Radiotherapy 26853339 5028 3353 ATAD5 79915 NA 5,8-DIPRENYLOXYPSORALEN CHEMBL1710181 5029 3354 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CLODRONATE DISODIUM CLODRONATE DISODIUM 5030 3355 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER antineoplastic agents 29546524 5032 3356 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist 135650348 HEXESTROL 5033 3357 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-3265 CHEMBL581868 5034 3358 TLR7 51284 DRUGGABLE GENOME ANA773 5035 3359 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-14 5037 3360 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR ELLIPTECINE ELLIPTECINE 5039 3361 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-4798 CHEMBL584635 5040 3362 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AMILORIDE AMILORIDE 5041 3363 HYAL2 8692 DRUGGABLE GENOME, CELL SURFACE EPINEPHRINE EPINEPHRINE 212383 5042 3364 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor BMS-599626 AC-480 5044 3365 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist CHEMBL2108061 VOLOCIXIMAB 5045 3366 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME TAMATINIB R-406 5046 3367 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GNF-PF-4283 CHEMBL606166 5047 3368 LEPR 3953 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME valproic acid 5049 3369 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Estetrol ESTETROL 5050 3370 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE OBTUSAQUINONE OBTUSAQUINONE 5052 3371 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL3545217 NS-018 5053 3372 ATAD5 79915 NA DNDI1417157 CHEMBL1576659 5054 3373 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Cisplatin CISPLATIN 25376608,25567130,25964101,23428903,26086967,27179933,23839309,28652249,18618574,26294215 5055 3374 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1237055 HYDROMORPHONE HYDROCHLORIDE 5056 3375 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 249565842 5057 3376 HSPB1 3315 DRUGGABLE GENOME PHENANTHROLINE PHENANTHROLINE 5059 3377 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 328083524 LENIOLISIB 5060 3378 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME vaccine PRINOMASTAT PRINOMASTAT 5061 3379 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 381118852 5064 3380 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200602 5066 3381 SMN2 6607 DRUGGABLE GENOME METHYL ROBUSTONE METHYL ROBUSTONE 5067 3382 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyridopyrimidinone derivative 2 5068 3383 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIAZOXIDE DIAZOXIDE 8301566 5069 3384 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor TOZASERTIB TOZASERTIB 19035792 5070 3385 ADH1B 125 DRUGGABLE GENOME, ENZYME acetaldehyde ACETALDEHYDE 31002879 5071 3386 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR AZ20 25593184 5072 3387 EIF3A 8661 NA Platinum compounds 5073 3388 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE ALMITRINE ALMITRINE 5074 3389 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PD-174265 CHEMBL188762 19969465 5076 3390 PTPRF 5792 DRUGGABLE GENOME, ENZYME, PROTEIN PHOSPHATASE ERLOTINIB HYDROCHLORIDE 26291013 5081 3391 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-23 5082 3392 TUBB4B 10383 DRUGGABLE GENOME CHEMBL492399 VERUBULIN 5083 3393 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-2776 CHEMBL578294 5084 3394 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL3039511 BEVENOPRAN 5085 3395 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TCMDC-123653 CHEMBL548540 5086 3396 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ROSE BENGAL ROSE BENGAL 5088 3397 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME BORTEZOMIB BORTEZOMIB 24524217 5089 3398 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME TAE-684 TAE-684 5090 3399 GLS 2744 ENZYME CEFMETAZOLE SODIUM CEFMETAZOLE SODIUM 5091 3400 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME EPINEPHRINE EPINEPHRINE 5092 3401 GPR37 2861 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist 178102688 5093 3402 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME OSI-632 OSI-632 5094 3403 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TEMEFOS TEMEFOS 5095 3404 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL856 PRIMIDONE 5097 3405 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR SURAMIN SURAMIN 15833899,11473364 5101 3406 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DOVITINIB DOVITINIB 5103 3407 PDE10A 10846 ENZYME, DRUGGABLE GENOME PMID27321640-Compound-59 5104 3408 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE SERM 11901050 5105 3409 TRPC4 7223 ION CHANNEL, KINASE, DRUGGABLE GENOME, CELL SURFACE blocker 381744967 5107 3410 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME PMA 12118374 5108 3411 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ZAFIRLUKAST ZAFIRLUKAST 5111 3412 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist CHEMBL547 ISOTRETINOIN 5112 3413 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER ERYTHROMYCIN ERYTHROMYCIN 10817732 5113 3414 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX AZACITIDINE AZACITIDINE 5116 3415 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 384403668 5117 3416 PTCH1 5727 CLINICALLY ACTIONABLE, TRANSPORTER SONIDEGIB SONIDEGIB 24651015 5118 3417 TLR7 51284 DRUGGABLE GENOME Isatoribine ISATORIBINE 5119 3418 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL166863 POLMACOXIB 5120 3419 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1201184 LANREOTIDE ACETATE 5122 3420 KDM4A 9682 DRUGGABLE GENOME, ENZYME 1-AMINOCYCLOPROPANECARBOXYLIC ACID HCL CHEMBL1255660 5124 3421 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GW3965 CHEMBL59030 18800767 5125 3422 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 gefitinib GEFITINIB 24433361 5126 3423 APH1B 83464 PROTEASE, DRUGGABLE GENOME GSI-136 GSI-136 5128 3424 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE ACCCRETROPIN 5130 3425 ALDH1A1 216 DRUGGABLE GENOME, ENZYME RIBAVIRIN RIBAVIRIN 5131 3426 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ELLIPTECINE ELLIPTECINE 18816045,19783445 5133 3427 NOS1 4842 DRUGGABLE GENOME, ENZYME DHT ANDROSTANOLONE 10725371 5134 3428 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME BIBT986 TANOGITRAN 5135 3429 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000047241 CHEMBL601933 5136 3430 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565693 5139 3431 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LUTEOLIN LUTEOLIN 5140 3432 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-102742 CHEMBL1519374 5141 3433 GMNN 51053 DRUGGABLE GENOME GNF-PF-3286 CHEMBL581880 5142 3434 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AMG 853 5144 3435 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SHP099 27362227 5145 3436 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE rifampin RIFAMPIN 22151084 5147 3437 IL18 3606 DRUGGABLE GENOME MEDI-2338 MEDI-2338 24812504 5148 3438 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME GW632580X GW632580X 5150 3439 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER YONDELIS YONDELIS 16888811 5152 3440 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE OXPRENOLOL OXPRENOLOL 5153 3441 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Binimetinib BINIMETINIB 5155 3442 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 384403651 5156 3443 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IDAZOXAN IDAZOXAN 5157 3444 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor CHEMBL565612 SOTRASTAURIN 5158 3445 IGFBP6 3489 DRUGGABLE GENOME ANTISERUM 8940357 5159 3446 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Arsenic trioxide 5160 3447 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PRODIGIOSIN PRODIGIOSIN 18922034 5161 3448 ABHD6 57406 PHOSPHOLIPASE, ENZYME Pyrazole derivative 80 5162 3449 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FLUSPIRILENE FLUSPIRILENE 5163 3450 AKR1B1 231 DRUGGABLE GENOME, ENZYME Sulindac SULINDAC 5164 3451 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DEPSIPEPTIDE ROMIDEPSIN 11929951 5165 3452 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE MEDROXYPROGESTERONE ACETATE MEDROXYPROGESTERONE ACETATE 5166 3453 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-123916 CHEMBL493863 5168 3454 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DITHIAZANINE DITHIAZANINE 5169 3455 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME CALCITONIN CALCITONIN 16222118 5170 3456 ABO 28 NA Ace Inhibitors, Plain 21832968 5171 3457 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tacrine-indole hybrid derivative 2 5172 3458 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME SNS-314 SNS-314 5173 3459 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CARBOPLATIN CARBOPLATIN 5176 3460 TXK 7294 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 178102336 BOSUTINIB 5177 3461 UCHL5 51377 DNA REPAIR, TUMOR SUPPRESSOR, ENZYME, PROTEASE PMID26077642-Compound-Figure3A 5178 3462 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Sulodexide SULODEXIDE 5179 3463 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 L-694247 L-694247 5180 3464 GMNN 51053 DRUGGABLE GENOME CID 663143 CHEMBL1342336 5182 3465 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TOSYL-L-LYSINE CHLOROMETHYL KETONE CHEMBL466465 5183 3466 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ANDALUSOL ANDALUSOL 23046382 5185 3467 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ELLIPTECINE ELLIPTECINE 5186 3468 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER risperidone RISPERIDONE 29723928,24589909,26129906,29443543,19997080,23609392 5190 3469 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 178102312 5191 3470 TUBA3D 113457 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 5192 3471 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE DOVITINIB DOVITINIB 5193 3472 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 5194 3473 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 223366203 RONICICLIB 5195 3474 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME KANZONOL W KANZONOL W 20022509 5197 3475 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE CIXUTUMUMAB CIXUTUMUMAB 5198 3476 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE ALSTERPAULLONE ALSTERPAULLONE 5199 3477 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 405067336 5201 3478 HTT 3064 DRUGGABLE GENOME NIHYDRAZONE NIHYDRAZONE 5202 3479 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor XL-765 VOXTALISIB 5203 3480 USP1 7398 DNA REPAIR, PROTEASE, ENZYME inhibitor 223366218 5204 3481 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ASN003 5206 3482 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ARRY-334543 VARLITINIB 5208 3483 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE HIF-1alpha 5210 3484 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Pyrrolo-pyridinone derivative 5 5211 3485 XDH 7498 DRUGGABLE GENOME, ENZYME allopurinol ALLOPURINOL 27798726,24915143 5212 3486 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR SURAMIN SURAMIN 9586958 5213 3487 MAPT 4137 DRUGGABLE GENOME ITRAZOLE ITRACONAZOLE 5215 3488 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200873 PHENTOLAMINE MESYLATE 5216 3489 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-376719 CHEMBL156263 5218 3490 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Epinastine EPINASTINE 5219 3491 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CABOZANTINIB CABOZANTINIB 25242168 5220 3492 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ITF2357 GIVINOSTAT 5221 3493 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME modulator CHEMBL1236924 INT131 5223 3494 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-2844 CHEMBL576353 5224 3495 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Zalutumumab ZALUTUMUMAB 5225 3496 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME AZD-1775 ADAVOSERTIB 5226 3497 HCN3 57657 DRUGGABLE GENOME, ION CHANNEL blocker 135651356 ZATEBRADINE 5227 3498 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME AST-487 AST-487 5229 3499 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CHEMBL2108660 TUCOTUZUMAB CELMOLEUKIN 5230 3500 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-95397 CHEMBL429095 5232 3501 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR DICLOFENAC DICLOFENAC 15131590 5233 3502 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PENTOSALEN PENTOSALEN 5234 3503 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME EVEROLIMUS EVEROLIMUS 26176165,24836070 5235 3504 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor ERLOTINIB HYDROCHLORIDE 5236 3505 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102783 5237 3506 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL1642 IMATINIB MESYLATE 5238 3507 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 1,3-DIPHENYLTHIOUREA CHEMBL275260 5239 3508 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL628 PENTOXIFYLLINE 5243 3509 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GTF505 5246 3510 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Trimidox TRIMETHOPRIM/SULFADOXINE 5249 3511 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1200992 5250 3512 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-56 5251 3513 HTT 3064 DRUGGABLE GENOME PERHEXILINE MALEATE PERHEXILINE MALEATE 5252 3514 ATXN2 6311 NA GEOPYXIN A GEOPYXIN A 5254 3515 FBXW7 55294 DNA REPAIR, CLINICALLY ACTIONABLE Sirolimus SIROLIMUS 24586741,18787170,23558291 5255 3516 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178100430 5256 3517 MGAT2 4247 ENZYME Phenylmethanesulfonamide derivative 1 5258 3518 MAOA 4128 DRUGGABLE GENOME, ENZYME Heteroaryl-cyclopropylamine derivative 1 5259 3519 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME haloperidol HALOPERIDOL 27023437 5260 3520 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Trametinib TRAMETINIB 26343583,28783719,28344857,25370473,27797976,25309914,22798288,28268064,24265153,28512244,25665005,25706985,27760111,27770002,24265152,26732095,26469692,22805292,27297867,22663011,27488531,27338794,27500726,26811525,27048246,27222538,25265492,27697975,22389471,26392102,28784858,28891408,27312529,26916115,23248257,26369631,24265154 5261 3521 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE SARACATINIB SARACATINIB 26191369 5262 3522 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME HL010183 CHEMBL2348411 23490148 5263 3523 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME ILORASERTIB ILORASERTIB 5264 3524 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Peptide analog 49 5265 3525 PDE4B 5142 DRUGGABLE GENOME, ENZYME DENBUFYLLINE DENBUFYLLINE 5267 3526 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR FONDAPARINUX FONDAPARINUX 5268 3527 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-1477 CHEMBL582675 5269 3528 SPP1 6696 DRUGGABLE GENOME SODIUM BUTYRATE 9224725 5270 3529 TH 7054 ENZYME, DRUGGABLE GENOME TETRAHYDROBIOPTERIN SAPROPTERIN 5271 3530 XIRP2 129446 NA atenolol ATENOLOL 5272 3531 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR MEDICATION 16456494 5273 3532 GSTZ1 2954 ENZYME, DRUGGABLE GENOME dichloroacetic acid 27143230 5274 3533 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-220455 CHEMBL95207 5275 3534 ADM 133 DRUGGABLE GENOME, HORMONE ACTIVITY PD-98059 CHEMBL35482 10830296 5280 3535 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Six-membered heterocyclic benzamide derivative 3 5282 3536 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ACETOCHLOR ACETOCHLOR 5283 3537 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000113107 CHEMBL589245 5284 3538 BCHE 590 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 2 5286 3539 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME WORTMANNIN WORTMANNIN 12401608,9502808,14574224 5287 3540 AREG 374 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE panitumumab PANITUMUMAB 23959273 5289 3541 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor PCI-24781 ABEXINOSTAT 5291 3542 KLK6 5653 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 404859022 5292 3543 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL2326966 SF-1126 5293 3544 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 223365967 CHEMBL523685 5294 3545 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LY-367265 CHEMBL1079460 5295 3546 ATAD5 79915 NA GNF-PF-1083 CHEMBL530361 5296 3547 AKR1B1 231 DRUGGABLE GENOME, ENZYME inhibitor 178103990 ZENARESTAT 5297 3548 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL2106798 NERAMEXANE MESYLATE 5298 3549 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME ISIS-TTRRx 5299 3550 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PHENYLBUTANOIC ACID PHENYLBUTANOIC ACID 24044874 5300 3551 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR RUCAPARIB RUCAPARIB 5301 3552 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DMSO DIMETHYL SULFOXIDE 9067579 5303 3553 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545427 CM-082 5304 3554 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER EPIPODOPHYLLOTOXINS 9719484 5305 3555 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200578 THEOPHYLLINE SODIUM GLYCINATE 5306 3556 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME OSI-774 ERLOTINIB 18723475 5307 3557 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE IBANDRONATE IBANDRONIC ACID 5308 3558 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME OCTADEC-17-YNOIC ACID CHEMBL182310 5310 3559 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-119915 CHEMBL1481974 5314 3560 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE TELATINIB TELATINIB 5315 3561 MPHOSPH8 54737 NA PICEATANNOL PICEATANNOL 5316 3562 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME infliximab INFLIXIMAB 5317 3563 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 336446944 5319 3564 IL18 3606 DRUGGABLE GENOME tacrolimus TACROLIMUS 25712187,25487141 5321 3565 STK4 6789 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 252827426 5322 3566 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Vorinostat VORINOSTAT 5323 3567 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME XL019 XL-019 5324 3568 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME DOVITINIB DOVITINIB 5325 3569 MSH6 2956 CLINICALLY ACTIONABLE, DNA REPAIR Temozolomide TEMOZOLOMIDE 19584161 5327 3570 ATAD5 79915 NA GNF-PF-2272 CHEMBL601757 5328 3571 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100466 5329 3572 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EXIFONE EXIFONE 5331 3573 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyridone 6 22916261 5332 3574 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 318164839 PONESIMOD 5334 3575 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THIOSALICYLIC ACID THIOSALICYLIC ACID 5336 3576 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME tegafur TEGAFUR 12209976,28950804,24923815,30858516,23603345,16115930,27122156,31382864,22490566,9470816,18600527,15944764,26603945,18443386,17700593,17165084,17000685,19530960,26794347,19795123,12360106,19473056,9439663,26099996,26216193,27864592,17121937,18299612,28295243,15132136,20819423,27995989,16151913,15017333,24817302,30114658,29846282,9323575,29134491,23988873,17203168,11895907,32378051,25677447,17064846,20385995,25796495,26265035,17417073,30723313,17848752,23930673,20665215,26804652,28929491,11350878,11555601,23942539,18452418,27454530,25410891,16361556,21077799,10803677,29889674,14635116,11156223,26846104,21498394,19858398,10071185,23585145 5338 3577 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRADIOL BENZOATE 521021 5340 3578 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AST-487 AST-487 5341 3579 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-126757 CHEMBL228132 5343 3580 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TAG-72 2316628 5345 3581 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CARBOPLATIN CARBOPLATIN 22139083 5346 3582 PTGS2 5743 DRUGGABLE GENOME, ENZYME ThermoProfen 5347 3583 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE TRIDOLGOSIR TRIDOLGOSIR 17897956 5348 3584 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CEPHALOCHROMIN CEPHALOCHROMIN 5349 3585 TNFRSF4 7293 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE 315661177 5350 3586 EED 8726 ENZYME, CLINICALLY ACTIONABLE MAK683 5353 3587 GSTM1 2944 DRUGGABLE GENOME, ENZYME doxorubicin DOXORUBICIN 23323945 5354 3588 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 223366069 RUCAPARIB 5355 3589 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1169880 BITOPERTIN 5356 3590 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AG-808 CHEMBL68534 5360 3591 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FENRETINIDE FENRETINIDE 5361 3592 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE aspirin ASPIRIN 17559347,22940005,15757620 5362 3593 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PURPURIN PURPURIN 5363 3594 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ZYH-1 5364 3595 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RIFAMPICIN RIFAMPIN 22931300 5365 3596 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GNF-PF-321 CHEMBL581044 5369 3597 HBB 3043 DRUGGABLE GENOME, ENZYME voxelotor VOXELOTOR 5370 3598 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL182066 RADIPRODIL 5371 3599 ATXN2 6311 NA GNF-PF-1678 CHEMBL580340 5372 3600 MAOB 4129 DRUGGABLE GENOME, ENZYME 4-hydroxybenzaldehyde 4-HYDROXYBENZALDEHYDE 5373 3601 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CHOLECALCIFEROL CHOLECALCIFEROL 9811059 5375 3602 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRICIRIBINE TRICIRIBINE 5376 3603 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 310264738 CERDULATINIB 5378 3604 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 135651428 5379 3605 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME BECLOMETHASONE BECLOMETHASONE 5381 3606 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565694 CHIR-99021 5382 3607 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme13INDY 5383 3608 EYA2 2139 DNA REPAIR NSC-127133 CHEMBL1172911 5384 3609 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME inhibitor 178103614 5385 3610 STAT5A 6776 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TOFACITINIB TOFACITINIB 14593182,19053756 5386 3611 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME GDC-0941 PICTILISIB 24265153,26577700,19276360 5387 3612 TOP1MT 116447 DRUGGABLE GENOME, ENZYME TOPOTECAN TOPOTECAN 5389 3613 FOXO1 2308 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR fluorouracil FLUOROURACIL 5390 3614 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DEOXIEPINEPHRINE DEOXIEPINEPHRINE 5391 3615 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME AZACITIDINE AZACITIDINE 5393 3616 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL DSP-3905 5394 3617 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TRIFLUOPERAZINE TRIFLUOPERAZINE 5395 3618 HTT 3064 DRUGGABLE GENOME DNDI1416969 CHEMBL1453126 5396 3619 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME APS-2-79 27556948 5397 3620 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Ertumaxomab ERTUMAXOMAB 5398 3621 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FELBAMATE FELBAMATE 22931300 5399 3622 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL VERAPAMIL VERAPAMIL 5400 3623 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME UREA UREA 17312972 5401 3624 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GYROPHORIC ACID GYROPHORIC ACID 5404 3625 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL572881 MOTESANIB 5405 3626 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR HYDROCORTAMATE HYDROCORTAMATE 5406 3627 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL PF-05186462 5407 3628 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-747267 CHEMBL610767 5410 3629 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX BISDEMETHOXYCURCUMIN BISDEMETHOXYCURCUMIN 23145932 5411 3630 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME ASPIRIN ASPIRIN 11981761 5412 3631 ATAD5 79915 NA GNF-PF-5217 CHEMBL601970 5413 3632 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-353263 CHEMBL1383812 5416 3633 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME PHA-767491 CHEMBL225519 5417 3634 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE GNF-PF-3060 CHEMBL581449 5418 3635 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PALIFERMIN PALIFERMIN 5419 3636 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RANITIDINE RANITIDINE 22931300 5420 3637 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SNS-314 SNS-314 5422 3638 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650720 5423 3639 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR AUTOLOGOUS DENDRITIC CELLS 16997859 5424 3640 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 2 5425 3641 PRKAB1 5564 ENZYME, KINASE, DRUGGABLE GENOME ANTIOXIDANT 14502105 5426 3642 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE THYROTROPIN ALFA 5427 3643 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PHENAMIPHOS PHENAMIPHOS 5429 3644 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE MEDI-546 ANIFROLUMAB 5430 3645 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE RETINOID 12697904 5431 3646 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE BECLOMETHASONE BECLOMETHASONE 5433 3647 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565590 CHEMBL1236539 5434 3648 SF3B1 23451 CLINICALLY ACTIONABLE N/A 24220272,21998214,22096241 5435 3649 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor 178101947 RUBOXISTAURIN 5436 3650 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PAZOPANIB PAZOPANIB 5437 3651 KDM4A 9682 DRUGGABLE GENOME, ENZYME CYCLOHETERPHYLLIN CYCLOHETERPHYLLIN 5439 3652 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 340590283 5441 3653 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR goserelin GOSERELIN 5442 3654 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TAE-684 TAE-684 5443 3655 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PHENINDIONE PHENINDIONE 5444 3656 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CCG-63802 CHEMBL1476646 5445 3657 CLK1 1195 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor 249565795 5446 3658 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1711 ISOPROTERENOL HYDROCHLORIDE 5448 3659 TSPO 706 DRUGGABLE GENOME PMID27599163-Compound-76 5451 3660 POLI 11201 DNA REPAIR QUERCITRIN QUERCITRIN 5452 3661 SGK1 6446 SERINE THREONINE KINASE, KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME, DRUG RESISTANCE ALPELISIB ALPELISIB 27451907 5453 3662 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR ABBV-744 ABBV-744 5455 3663 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE CENISERTIB CENISERTIB 5457 3664 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Meloxicam MELOXICAM 5458 3665 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME PHENYLEPHRINE PHENYLEPHRINE 10220693 5459 3666 ALOX15 246 ENZYME, DRUGGABLE GENOME CISPLATIN CISPLATIN 5463 3667 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PD-98059 CHEMBL35482 5464 3668 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE AMENTOFLAVONE AMENTOFLAVONE 5465 3669 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR modulator CHEMBL3137316 FOSDAGROCORAT 5466 3670 PTGES 9536 DRUGGABLE GENOME, ENZYME VEGF 16155957 5467 3671 ITGA11 22801 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE IFN 16697656 5468 3672 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ANGUIDIN ANGUIDIN 5469 3673 SLC12A2 6558 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE BUMETANIDE BUMETANIDE 5470 3674 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE GELDANAMYCIN GELDANAMYCIN 12811834 5471 3675 NPEPPS 9520 PROTEASE, ENZYME, DRUGGABLE GENOME CHR-2797 TOSEDOSTAT 5472 3676 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME DAUNORUBICIN DAUNORUBICIN 22260166 5473 3677 BAZ2B 29994 NA TCMDC-123769 CHEMBL534353 5476 3678 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME AG-808 CHEMBL68534 5478 3679 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME KITE-585 5480 3680 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody RO5083945 IMGATUZUMAB 5481 3681 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME ICA-105665 5482 3682 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650787 5483 3683 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200586 PRILOCAINE HYDROCHLORIDE 5484 3684 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 5485 3685 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE (5Z,9Z)-5,9-HEXADECADIENOIC ACID CHEMBL464637 12444712 5486 3686 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE DOVITINIB DOVITINIB 5487 3687 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE dabrafenib DABRAFENIB 5488 3688 TSPO 706 DRUGGABLE GENOME Diazepam DIAZEPAM 5489 3689 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE DOLASTATIN 10 9615758 5490 3690 STK4 6789 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 178102336 BOSUTINIB 5491 3691 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME SAR302503 24398328,21926964 5492 3692 XPO1 7514 CLINICALLY ACTIONABLE, KINASE inhibitor CHEMBL3545185 SELINEXOR 5495 3693 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MALATHION MALATHION 5496 3694 PSMB3 5691 PROTEASE, DRUGGABLE GENOME inhibitor BORTEZOMIB BORTEZOMIB 5497 3695 GMNN 51053 DRUGGABLE GENOME GNF-PF-1134 CHEMBL600694 5498 3696 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING CIPROFIBRATE CIPROFIBRATE 16680159 5499 3697 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME efavirenz EFAVIRENZ 18301070 5500 3698 TUBB2B 347733 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 5501 3699 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OLOMOUCINE OLOMOUCINE 5502 3700 ALOX15 246 ENZYME, DRUGGABLE GENOME EHNA EHNA 5503 3701 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C5 5505 3702 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING VINBLASTINE SULFATE VINBLASTINE SULFATE 5507 3703 TPCN2 219931 ION CHANNEL, DRUGGABLE GENOME blocker 135651305 VERAPAMIL 5508 3704 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 385612219 BREPOCITINIB 5509 3705 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE FLUOROURACIL FLUOROURACIL 24450514 5510 3706 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1231 OXYBUTYNIN 5513 3707 DHODH 1723 DRUGGABLE GENOME, ENZYME inhibitor 375973210 5516 3708 POLB 5423 DNA REPAIR, DRUGGABLE GENOME DITHIAZANINE IODIDE DITHIAZANINE IODIDE 5517 3709 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor 252827519 5518 3710 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE AM-111 BRIMAPITIDE, C-TERMINAL ACID 5520 3711 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIETHYLCARBAMAZINE CITRATE DIETHYLCARBAMAZINE CITRATE 5523 3712 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125319 CHEMBL527586 5524 3713 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-348401 CHEMBL515505 5526 3714 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME SAPONIN 12451485 5527 3715 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIGOXIN DIGOXIN 5528 3716 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-stenine 5529 3717 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FLUDROCORTISONE FLUDROCORTISONE 5530 3718 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE poziotinib POZIOTINIB 5531 3719 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME MOCETINOSTAT MOCETINOSTAT 23829483,26287310 5532 3720 PDE3B 5140 ENZYME, DRUGGABLE GENOME US8741907-compound-3 5534 3721 ATXN2 6311 NA A-77636 CHEMBL291143 5535 3722 CES1 1066 DRUGGABLE GENOME, ENZYME mycophenolate mofetil 24220207 5536 3723 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DIFLORASONE DIFLORASONE 5538 3724 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME VENLAFAXINE VENLAFAXINE 5539 3725 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 318164850 ETRASIMOD 5540 3726 RAB9A 9367 ENZYME, DRUGGABLE GENOME NSC-44661 CHEMBL571228 5541 3727 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE MK2206 MK-2206 26106072 5543 3728 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL3545252 DOCETAXEL 5544 3729 CYP27B1 1594 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 20S-HYDROXYVITAMIN D3 CHEMBL2036072 22404326 5545 3730 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Fulvestrant FULVESTRANT 26733612 5549 3731 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME OXYGEN THERAPY 9736447 5551 3732 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BENZO[B]THIOPHEN-2-YLMETHANAMINE CHEMBL1770735 25458499 5552 3733 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE MORPHINE MORPHINE 12373743 5554 3734 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 310264749 SERABELISIB 5555 3735 TUBA3C 7278 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 5556 3736 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE PROGESTERONE PROGESTERONE 12529413 5558 3737 MPHOSPH8 54737 NA DOPAMINE DOPAMINE 5559 3738 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SAR-405838 SAR-405838 5560 3739 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 249565765 5561 3740 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor MK-2206 MK-2206 5562 3741 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME MASITINIB MASITINIB 5568 3742 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME tolperisone TOLPERISONE 25953735 5570 3743 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1023 BEXAROTENE 5573 3744 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MITOGEN-ACTIVATED PROTEIN KINASE INHIBITOR 16123320 5574 3745 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417086 CHEMBL1224755 5575 3746 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME MOMETASONE MOMETASONE 5577 3747 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US8975409, Example 9(3) 5578 3748 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE AZD6482 AZD-6482 5579 3749 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-62 5581 3750 BAZ2B 29994 NA TCMDC-125298 CHEMBL581152 5582 3751 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GNF-PF-2262 CHEMBL577862 5583 3752 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651378 5584 3753 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TAMATINIB R-406 5585 3754 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZYL ISOTHIOCYANATE BENZYL ISOTHIOCYANATE 5586 3755 CBX1 10951 NA NSC-7387 CHEMBL119878 5587 3756 LAMC2 3918 DRUGGABLE GENOME BST-1005 5588 3757 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME TYRPHOSTIN A9 11112699 5589 3758 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PRULIFLOXACIN PRULIFLOXACIN 5590 3759 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 381118865 5593 3760 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME KX2-361 KX2-361 5594 3761 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME FBT-A05 FBT-A05 5596 3762 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME BACILLUS CALMETTE-GUERIN 11025701 5597 3763 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HYDRAMETHYLNON HYDRAMETHYLNON 5598 3764 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE SB-242235 SB-242235 5599 3765 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SB-224289 SB-224289 5600 3766 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR PHOTOSENSITIZER 15611953 5601 3767 TUBA1A 7846 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 5602 3768 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR RO-14 5604 3769 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR KB002/003 5607 3770 ATF2 1386 TRANSCRIPTION FACTOR 2-METHOXYESTRADIOL 2-METHOXYESTRADIOL 15691880 5609 3771 USP1 7398 DNA REPAIR, PROTEASE, ENZYME FLUPIRTINE MALEATE FLUPIRTINE MALEATE 5610 3772 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW680191X GW680191X 5611 3773 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL258805 SU-9516 5614 3774 GMNN 51053 DRUGGABLE GENOME TCMDC-123947 CHEMBL525098 5615 3775 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DIBENZ[A,H]ANTHRACENE DIBENZ[A,H]ANTHRACENE 5616 3776 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GOSSYPOL GOSSYPOL 5617 3777 PHEX 5251 ENZYME, PROTEASE, DRUGGABLE GENOME RHGH 9323282 5618 3778 PTGS2 5743 DRUGGABLE GENOME, ENZYME Indomethacin INDOMETHACIN 5619 3779 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME N-(pyridin-2-yl)pyrimidin-4-amine derivative 2 5620 3780 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME BAY-613606 CHEMBL541400 5623 3781 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CYPROHEPTADINE CYPROHEPTADINE 5627 3782 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE DLX-105 5629 3783 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Edasalonexent EDASALONEXENT 5630 3784 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1201022 PHENAZOPYRIDINE HYDROCHLORIDE 5631 3785 DGAT1 8694 ENZYME, DRUGGABLE GENOME inhibitor 223366160 PF-04620110 5635 3786 ITPA 3704 ENZYME ribavirin RIBAVIRIN 26441325,25713999,23730840,21274861,26916827,26670100,20173735,26071337,23707372,26438033,21246582,27833958,20547162,21503919,20637204 5636 3787 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE CAMPTOTHECIN CAMPTOTHECIN 5637 3788 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-123852 CHEMBL547656 5638 3789 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME EUPATORIN EUPATORIN 5639 3790 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker 135650484 5641 3791 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051798 BELINOSTAT 5642 3792 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TETRABROMOBENZOTRIAZOLE TETRABROMOBENZOTRIAZOLE 5643 3793 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME inhibitor 249565696 5645 3794 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774822-Compound-Figure2Example1-1left 5646 3795 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TCMDC-125353 CHEMBL547924 5648 3796 NDUFS8 4728 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 5649 3797 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE SORAFENIB SORAFENIB 5651 3798 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ZOXAZOLAMINE ZOXAZOLAMINE 22931300 5652 3799 USP1 7398 DNA REPAIR, PROTEASE, ENZYME 2-METHOXY-1,4-NAPHTHOQUINONE 2-METHOXY-1,4-NAPHTHOQUINONE 5653 3800 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Entinostat ENTINOSTAT 18483379,23498719 5655 3801 FNTA 2339 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL298734 LONAFARNIB 5656 3802 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MM-111 MM-111 5660 3803 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NSC-607097 CHEMBL1374370 5661 3804 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL527 PIROXICAM 5662 3805 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE PEG-INTERFERON ALFACON-1 5663 3806 PSENEN 55851 DRUGGABLE GENOME inhibitor RO 4929097 5665 3807 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME BIRABRESIB BIRABRESIB 26976114 5666 3808 TSPO 706 DRUGGABLE GENOME Midazolam MIDAZOLAM 5667 3809 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME MLN-9708 IXAZOMIB CITRATE 5668 3810 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565807 5672 3811 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 385612218 5674 3812 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DOXORUBICIN DOXORUBICIN 5675 3813 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL THIOPENTAL THIOPENTAL 5676 3814 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Cyclophosphamide CYCLOPHOSPHAMIDE 25589624 5677 3815 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200463 OXAPROZIN POTASSIUM 5678 3816 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-5510 CHEMBL578741 5679 3817 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME PAC-1 PAC-1 5680 3818 DPEP1 1800 PROTEASE, DRUGGABLE GENOME, ENZYME CILASTATIN CILASTATIN 5681 3819 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 5683 3820 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME ENTINOSTAT ENTINOSTAT 21696956,19966789,20491440 5684 3821 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME R-N-PROPYLNORAPOMORPHINE R-N-PROPYLNORAPOMORPHINE 5685 3822 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649752 5688 3823 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201560 PEGINTERFERON ALFA-2A 5689 3824 VPS37A 137492 DRUG RESISTANCE CETUXIMAB CETUXIMAB 22016507 5691 3825 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270010-Compound-Figure24-b 5692 3826 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 318164802 5694 3827 KDM4A 9682 DRUGGABLE GENOME, ENZYME BAS 01152706 CHEMBL2002487 5696 3828 SLC29A4 222962 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 135652709 QUININE 5697 3829 MAPT 4137 DRUGGABLE GENOME GNF-PF-1919 CHEMBL576409 5698 3830 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker 53801058 MIBEFRADIL 5699 3831 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178101480 5701 3832 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TEPROTUMUMAB TEPROTUMUMAB 21985784 5702 3833 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-278539 CHEMBL275168 5704 3834 TXNRD1 7296 DRUGGABLE GENOME Disulfide compound 1 5706 3835 ALDH1A2 8854 DRUGGABLE GENOME, ENZYME RETINOL RETINOL 9666306 5709 3836 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Indazole derivative 2 5710 3837 BRD1 23774 ENZYME inhibitor 252166774 5712 3838 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE modulator CHEMBL3545046 GSK2849466 5714 3839 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-134 5715 3840 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CUDC-101 CUDC-101 5716 3841 UGT1A7 54577 DRUGGABLE GENOME, ENZYME NICOTINE NICOTINE 12167564 5717 3842 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32o 5718 3843 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE DOVITINIB DOVITINIB 5719 3844 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Estrogen receptor beta-selective phytoestrogenic formulation 5720 3845 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR GAMBOGIC ACID GAMBOGIC ACID 21486005 5721 3846 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHLORPROMAZINE HYDROCHLORIDE CHLORPROMAZINE HYDROCHLORIDE 5722 3847 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 3-METHYLCHOLANTHRENE 3-METHYLCHOLANTHRENE 5724 3848 KDM4A 9682 DRUGGABLE GENOME, ENZYME TOSUFLOXACIN TOSYLATE TOSUFLOXACIN TOSYLATE 5725 3849 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Doxorubicin DOXORUBICIN 25658463,21399868,16243804,23165797,26826118 5726 3850 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SORAFENIB SORAFENIB 5727 3851 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor 385612193 5728 3852 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR BENZO(K)FLUORANTHENE BENZO(K)FLUORANTHENE 5729 3853 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BROMODEOXYURIDINE 8008235 5730 3854 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR QUINONE 8794898 5731 3855 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DOXEPIN DOXEPIN 5733 3856 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL QUAZEPAM QUAZEPAM 5735 3857 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OXYBUTYNIN OXYBUTYNIN 22931300 5736 3858 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE activator 135650906 5737 3859 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 178102645 5741 3860 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME PHA-767491 CHEMBL225519 5742 3861 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME inhibitor 135650306 GLYBURIDE 5743 3862 TUBA1A 7846 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 5744 3863 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GDC0879 19276360 5746 3864 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CAMBINOL CAMBINOL 5747 3865 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650868 QUADAZOCINE 5749 3866 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE NSC-663284 CHEMBL337173 5750 3867 FST 10468 DRUGGABLE GENOME ANTI-ANDROGEN 14761877 5753 3868 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME GSK 2118436 5754 3869 SPATA5 166378 NA paclitaxel PACLITAXEL 24444404 5757 3870 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 135650105 5758 3871 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME Mibefradil MIBEFRADIL 5759 3872 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FENBUCONAZOLE FENBUCONAZOLE 5760 3873 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME TESTOSTERONE TESTOSTERONE 8779895 5761 3874 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Bosutinib BOSUTINIB 5762 3875 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME BAY-613606 CHEMBL541400 5764 3876 TARDBP 23435 TUMOR SUPPRESSOR SJ000260153 CHEMBL589717 5766 3877 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DIHYDROXIDINE DIHYDROXIDINE 5769 3878 POLK 51426 DNA REPAIR, ENZYME JUGLONE JUGLONE 21903399 5770 3879 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Piperidinyl triazole derivative 3 5771 3880 F5 2153 DRUGGABLE GENOME Rivaroxaban RIVAROXABAN 5772 3881 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antibody OLARATUMAB OLARATUMAB 5773 3882 NR0B2 8431 TRANSCRIPTION FACTOR BINDING, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 252827495 5774 3883 GMNN 51053 DRUGGABLE GENOME 2-METHOXY-1,4-NAPHTHOQUINONE 2-METHOXY-1,4-NAPHTHOQUINONE 5775 3884 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103513 AZD-3839 5777 3885 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 375973222 5779 3886 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER opioids 23803057,25794200,24950410,27061230,28379874,21398039,24034787,19514130 5780 3887 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CX-6258 27486174 5783 3888 UGT2B7 7364 DRUGGABLE GENOME lamotrigine LAMOTRIGINE 26213157,26790665,27096250,23263737 5785 3889 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Genz-644282 5786 3890 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX FLUAZINAM FLUAZINAM 5787 3891 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103483 AZILSARTAN 5788 3892 MAPT 4137 DRUGGABLE GENOME GNF-PF-5007 CHEMBL1989853 5789 3893 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL antagonist CHEMBL14935 TEZAMPANEL 5790 3894 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PENTAZOCINE PENTAZOCINE 5791 3895 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL2068724 ACAMPROSATE CALCIUM 5795 3896 ALDH1A1 216 DRUGGABLE GENOME, ENZYME KOPARIN KOPARIN 5796 3897 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME peginterferon alfa-2a 23360626 5798 3898 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME AMOXAPINE AMOXAPINE 5799 3899 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178103575 5801 3900 CBL 867 KINASE, ENZYME, CLINICALLY ACTIONABLE Fasudil FASUDIL 26177294 5802 3901 PTGS1 5742 ENZYME, DRUGGABLE GENOME ASPIRIN ASPIRIN 23651359 5803 3902 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-628113 CHEMBL176599 5804 3903 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX RESACTIN A RESACTIN A 5805 3904 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PROTOPORPHYRIN PROTOPORPHYRIN 5807 3905 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME FLUNARIZINE FLUNARIZINE 5808 3906 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DNDI1417346 CHEMBL1490332 5809 3907 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR GW685698X FLUTICASONE FUROATE 5810 3908 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME ISOTHYMONIN ISOTHYMONIN 5811 3909 PTGS2 5743 DRUGGABLE GENOME, ENZYME SULINDAC SULINDAC 5813 3910 PSMD2 5708 NA MLN-9708 IXAZOMIB CITRATE 5814 3911 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 354702204 DEZAPELISIB 5815 3912 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PHYSODIC ACID PHYSODIC ACID 5816 3913 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME METHYLDOPA METHYLDOPA 5818 3914 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ethanol ALCOHOL 29588096,26049587,15902904,25514903 5819 3915 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE BAY-613606 CHEMBL541400 5821 3916 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME QUERCETIN DIHYDRATE QUERCETIN DIHYDRATE 5822 3917 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIMETHYL-TETRADECYL-AMMONIUM CHLORIDE TRIMETHYL-TETRADECYL-AMMONIUM CHLORIDE 5823 3918 TOP2B 7155 DRUGGABLE GENOME, ENZYME NK-314 5824 3919 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL29919 ELPETRIGINE 5825 3920 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR LAS-41002 22956938 5826 3921 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR INTERLEUKIN-4 9352015 5827 3922 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL (+)-[3H]-PENTAZOCINE CHEMBL2311194 22853801 5828 3923 ATAD5 79915 NA GNF-PF-2335 CHEMBL601146 5829 3924 NAMPT 10135 DRUGGABLE GENOME GMX1777 TEGLARINAD CHLORIDE 5830 3925 PGGT1B 5229 ENZYME, DRUGGABLE GENOME GGTI-2418 5831 3926 CECR2 27443 NA inhibitor 252827481 5832 3927 CXCL8 3576 DRUGGABLE GENOME CHLORDANE CHLORDANE 5834 3928 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHEMBL1341 METHOXYFLURANE 5836 3929 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2011801300410 5837 3930 ATAD5 79915 NA KAMEBANIN KAMEBANIN 5838 3931 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME BEZ235 DACTOLISIB 5839 3932 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALVAC 12855617 5840 3933 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Falecalcitrol 5844 3934 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PIPLARTINE PIPLARTINE 5847 3935 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ERYTHROSINE ERYTHROSINE 5848 3936 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Odiparcil ODIPARCIL 5851 3937 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR NICARDIPINE NICARDIPINE 10748141 5853 3938 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL924 ZOLEDRONIC ACID 5854 3939 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3545243 AS-703988 5856 3940 MAPT 4137 DRUGGABLE GENOME HEXACHLOROPHENE HEXACHLOROPHENE 5857 3941 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651391 5859 3942 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 223365984 LUCITANIB 5860 3943 ALDH1A1 216 DRUGGABLE GENOME, ENZYME RABEPRAZOLE RABEPRAZOLE 5861 3944 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME 3-acylidene-2-oxoindole derivative 1 5863 3945 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE ATEZOLIZUMAB ATEZOLIZUMAB 29773717 5864 3946 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PANITUMUMAB PANITUMUMAB 26644315,23404247,20921465,18316791,28275037,19223544 5866 3947 DPYSL3 1809 NA METHIMAZOLE METHIMAZOLE 11694350 5867 3948 RACGAP1 29127 NA TCMDC-138263 CHEMBL535307 5868 3949 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ERLOTINIB ERLOTINIB 5869 3950 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL2146883 COBIMETINIB 5872 3951 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIAMCINOLONE TRIAMCINOLONE 5873 3952 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 249565738 5875 3953 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DNDI1417776 CHEMBL1585652 5876 3954 ALOX15 246 ENZYME, DRUGGABLE GENOME 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 5877 3955 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE CEDIRANIB CEDIRANIB 5878 3956 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MK-212 MK-212 5879 3957 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 252166524 SOTAGLIFLOZIN 5881 3958 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE DCC-2036 REBASTINIB 5882 3959 SOD2 6648 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE asparaginase ASPARAGINASE 27019981 5883 3960 USP1 7398 DNA REPAIR, PROTEASE, ENZYME KHELLIN KHELLIN 5884 3961 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE TRAFERMIN TRAFERMIN 5887 3962 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE PHILANTHOTOXIN 343 PHILANTHOTOXIN 343 20873775 5888 3963 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE PF-562271 PF-00562271 5889 3964 HNMT 3176 ENZYME, DRUGGABLE GENOME Amodiaquine AMODIAQUINE 5891 3965 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL393220 ATORVASTATIN CALCIUM 5893 3966 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME REOLYSIN PELAREOREP 5895 3967 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE LY-367265 CHEMBL1079460 5903 3968 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651592 5905 3969 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME NICOXAMAT NICOXAMAT 25937017 5906 3970 MAGEA1 4100 NA 5-AZA-2-DEOXYCYTIDINE 9247253 5909 3971 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME FLUTAMIDE FLUTAMIDE 15735703 5910 3972 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR Buparlisib BUPARLISIB 5911 3973 F2RL3 9002 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 381744952 5912 3974 TOP2B 7155 DRUGGABLE GENOME, ENZYME Epirubicin EPIRUBICIN 5913 3975 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR CI-1040 CI-1040 12370306,19915144 5914 3976 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MMV009085 CHEMBL581225 5915 3977 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PMID27774824-Compound-Figure11Example1up 5917 3978 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE FISETIN FISETIN 8759170 5918 3979 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMPHOTERICIN B 15969931 5920 3980 RAD50 10111 CLINICALLY ACTIONABLE, KINASE, DNA REPAIR CHECKPOINT KINASE INHIBITOR AZD7762 24934408 5924 3981 SLC38A2 54407 TRANSPORTER 178101264 5925 3982 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX N,N'-DIPHENYL-GUANIDINE CHEMBL77675 5926 3983 PNPLA3 80339 ENZYME vincristine VINCRISTINE 28744905 5928 3984 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-61836 CHEMBL521171 5930 3985 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER NOVOBIOCIN NOVOBIOCIN 10901300 5931 3986 PRKAB1 5564 ENZYME, KINASE, DRUGGABLE GENOME METFORMIN METFORMIN 26471090 5932 3987 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200500 BECLOMETHASONE DIPROPIONATE 5933 3988 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650427 5935 3989 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 178101156 URB-597 5936 3990 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GOSSYPOL GOSSYPOL 5937 3991 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL PRIMIDONE PRIMIDONE 5938 3992 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ANTIBIOTICS 14736076 5940 3993 PTGS2 5743 DRUGGABLE GENOME, ENZYME ACETAMINOPHEN ACETAMINOPHEN 5941 3994 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR CHLORAMBUCIL CHLORAMBUCIL 5943 3995 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SB-408124 CHEMBL1334465 5944 3996 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME AS-1402 HUHMFG1 5945 3997 FTO 79068 ENZYME mercaptopurine MERCAPTOPURINE 27558924 5946 3998 ALOX5 240 DRUGGABLE GENOME, ENZYME Rilopirox RILOPIROX 5948 3999 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Oxymetazoline OXYMETAZOLINE 5950 4000 POLI 11201 DNA REPAIR DEPHOSTATIN DEPHOSTATIN 5952 4001 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PD-98059 CHEMBL35482 5953 4002 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SEROTONIN SEROTONIN 5955 4003 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR UCN-01 UCN-01 12244092 5956 4004 TSPO 706 DRUGGABLE GENOME Clorazepate CLORAZEPIC ACID 5957 4005 MAPT 4137 DRUGGABLE GENOME PD-98059 CHEMBL35482 5958 4006 ALDH1A1 216 DRUGGABLE GENOME, ENZYME INAMRINONE INAMRINONE 5959 4007 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MEPIVACAINE MEPIVACAINE 22931300 5960 4008 NFATC2 4773 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME asparaginase ASPARAGINASE 25987655 5961 4009 P2RX4 5025 ION CHANNEL, DRUGGABLE GENOME P2X4 inhibitora 5963 4010 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Emicizumab EMICIZUMAB 5964 4011 GMNN 51053 DRUGGABLE GENOME DNDI1417560 CHEMBL1373255 5965 4012 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor DACTOLISIB DACTOLISIB 5966 4013 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650178 DICYCLOMINE 5967 4014 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TAMIBAROTENE TAMIBAROTENE 5968 4015 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ANAZOLENE ANAZOLENE 5969 4016 ADAM17 6868 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, NEUTRAL ZINC METALLOPEPTIDASE, TRANSPORTER, ENZYME inhibitor 178103981 ILOMASTAT 5971 4017 IL1B 3553 KINASE, DRUGGABLE GENOME BECLOMETHASONE DIPROPIONATE 9176529 5975 4018 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME R-phenserine 5976 4019 DPP7 29952 PROTEASE, ENZYME, DRUGGABLE GENOME CRWCYVOHVXAEMF-LBPRGKRZSA-N 5978 4020 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TCMDC-124327 CHEMBL581929 5979 4021 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME SLV-338 5980 4022 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651172 5981 4023 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Venetoclax VENETOCLAX 5982 4024 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor SODIUM PHENYLBUTYRATE 5983 4025 QRFPR 84109 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102518 5984 4026 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME ALISERTIB ALISERTIB 5987 4027 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor PIVANEX AN-9 5990 4028 TUBB4B 10383 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 5992 4029 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL464 ETRETINATE 5993 4030 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Paclitaxel PACLITAXEL 5994 4031 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR ALPRAZOLAM ALPRAZOLAM 22137933 5996 4032 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE HORMONES 9133444 5997 4033 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PALBOCICLIB PALBOCICLIB 6000 4034 KDM4A 9682 DRUGGABLE GENOME, ENZYME MICONAZOLE MICONAZOLE 6002 4035 ALOX5 240 DRUGGABLE GENOME, ENZYME SELENIUM 14975747 6003 4036 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545002 MP-412 6005 4037 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545195 LY-3009120 6006 4038 KDM1A 23028 DRUGGABLE GENOME, ENZYME, CELL SURFACE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING inhibitor 178103603 6008 4039 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ANTISENSE C-FOS 12215476 6009 4040 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PODOFILOX PODOFILOX 6010 4041 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SILODOSIN SILODOSIN 6011 4042 STK16 8576 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME inhibitor 249565890 6013 4043 MAP4K3 8491 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 384403668 6014 4044 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AC480 AC-480 6015 4045 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL OXAZEPAM OXAZEPAM 6019 4046 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYCLANDELATE CYCLANDELATE 6020 4047 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor BGJ398 INFIGRATINIB 6021 4048 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CID 4970947 CHEMBL1451921 6022 4049 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RO-0506220 CHEMBL1956069 16476733 6023 4050 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR calcitriol CALCITRIOL 15883634,18470879,17274004,21651652,10707958,333287,9933478,21418277,15295697,15861036,16210379,15739035,17763859,20716226,14685227,20500803,15864137,20727239,11450701,19647104,18827005,10320522 6027 4051 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING NSC-60339 CHEMBL1448793 6028 4052 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE ILORASERTIB ILORASERTIB 6029 4053 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME AZATADINE AZATADINE 6030 4054 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000294102 CHEMBL607309 6031 4055 MAPT 4137 DRUGGABLE GENOME NSC-367089 CHEMBL1543865 6032 4056 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LITHIUM LITHIUM 18619545 6033 4057 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE 2-Methoxyestradiol 2-METHOXYESTRADIOL 24162827 6036 4058 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CILOSTAMIDE CILOSTAMIDE 6037 4059 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUFENOXURON FLUFENOXURON 6039 4060 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178101956 6041 4061 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SULFASALAZINE SULFASALAZINE 22931300 6042 4062 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE STIROFOS STIROFOS 6043 4063 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Antibodie derivative 1 6045 4064 CD37 951 DRUGGABLE GENOME IMGN529 NARATUXIMAB EMTANSINE 6046 4065 UGT1A6 54578 ENZYME, DRUGGABLE GENOME risperidone RISPERIDONE 6047 4066 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE 6049 4067 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PAEONOL PAEONOL 6050 4068 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Aromatic bicyclic compound 2 6051 4069 CPB2 1361 DRUGGABLE GENOME, ENZYME, PROTEASE DS-1040 6052 4070 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR POLYSIALIC ACID 16903870 6053 4071 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHLORDANE CHLORDANE 6055 4072 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE PROTEASOME INHIBITOR 17910634 6056 4073 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LIGNOCAINE LIDOCAINE 9832299 6057 4074 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE ENTRECTINIB ENTRECTINIB 6060 4075 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200802 TALBUTAL 6061 4076 POLI 11201 DNA REPAIR 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 6062 4077 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 405560505 6063 4078 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-58 6064 4079 RABEP1 9135 CLINICALLY ACTIONABLE, GROWTH FACTOR lithium LITHIUM 28694205 6065 4080 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE LANATOSIDE C LANATOSIDE C 6066 4081 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649998 6067 4082 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PARICALCITOL PARICALCITOL 6069 4083 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE AST-487 AST-487 6070 4084 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME PMA 15707698,9502808,14574224 6071 4085 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32s 6072 4086 GJB6 10804 ION CHANNEL inhibitor 178101095 OCTANOL 6073 4087 PMEL 6490 DRUGGABLE GENOME Multi-epitope tyrosinase/gp100 vaccine 6074 4088 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME DNDI1417467 CHEMBL1997335 6076 4089 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID25726713-Compound-51 6078 4090 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE WIN-55212-2 WIN-552122 6080 4091 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CEFMETAZOLE SODIUM CEFMETAZOLE SODIUM 6084 4092 CPS1 1373 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Polidocanol - BioForm Medical/Chemische Fabrik Kreussler & Co 6085 4093 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE TEGAFUR TEGAFUR 6087 4094 STK38L 23012 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565890 6088 4095 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME adalimumab ADALIMUMAB 6089 4096 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 336446930 6090 4097 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135649878 CHEMBL351231 6091 4098 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor MASITINIB MASITINIB 6093 4099 PRSS3 5646 ENZYME, PROTEASE, DRUGGABLE GENOME CYANOPEPTOLIN SS CYANOPEPTOLIN SS 6094 4100 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor TEMSIROLIMUS TEMSIROLIMUS 6095 4101 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 178103650 ETHINYL ESTRADIOL 6096 4102 CA2 760 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL220491 BRINZOLAMIDE 6098 4103 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME METHYLPREDNISOLONE METHYLPREDNISOLONE 6100 4104 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR QUINAPRIL QUINAPRIL 12693379,11849656 6101 4105 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Difelikefalin DIFELIKEFALIN 6103 4106 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE PLX-4720 PLX-4720 6104 4107 IPO8 10526 NA MKC-1 ENMD-981693 6105 4108 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PREDNISONE PREDNISONE 11186134 6106 4109 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Atezolizumab ATEZOLIZUMAB 6107 4110 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME LAS38096 CHEMBL375293 6108 4111 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME TAE-684 TAE-684 6110 4112 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor AUY922 6111 4113 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Tricyclic compound 1 6112 4114 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME Ponatinib PONATINIB 6113 4115 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE celecoxib CELECOXIB 22336956 6119 4116 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE PHLORETIN PHLORETIN 6120 4117 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALCITRIOL CALCITRIOL 11158396 6121 4118 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE AAB-003/PF-05236812 6122 4119 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME ISOPROTERENOL ISOPROTERENOL 6124 4120 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR AMMONIA SOLUTION, STRONG AMMONIA SOLUTION, STRONG 22324546 6125 4121 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE rigosertib RIGOSERTIB 6127 4122 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TIOCONAZOLE TIOCONAZOLE 6128 4123 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Pimasertib PIMASERTIB 23629727 6129 4124 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL BUTALBITAL BUTALBITAL 6131 4125 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING BUTANOIC ACID BUTANOIC ACID 19053749 6133 4126 SMN1 6606 DRUGGABLE GENOME GNF-PF-1872 CHEMBL600103 6136 4127 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME HISPIDIN HISPIDIN 6137 4128 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME CLOFIBRATE CLOFIBRATE 16316932 6138 4129 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER GABAPENTIN GABAPENTIN 17328248 6139 4130 KCNA7 3743 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107762 NERISPIRDINE 6140 4131 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR BAY1000394 6141 4132 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE PEMETREXED PEMETREXED 6143 4133 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR CLADRIBINE CLADRIBINE 12948851 6144 4134 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650568 6145 4135 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PMID25726713-Compound-49 6146 4136 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FLUVOXAMINE FLUVOXAMINE 22931300 6147 4137 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ILORASERTIB ILORASERTIB 6148 4138 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650110 CLOFIBRATE 6149 4139 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE TOZASERTIB TOZASERTIB 6150 4140 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CIS-2,4,3',5'-TETRAMETHOXYSTILBENE CHEMBL221300 6151 4141 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLOPERASTINE HYDROCLORIDE CLOPERASTINE HYDROCLORIDE 6152 4142 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE S-110 6153 4143 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME inhibitor 249565918 6155 4144 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 249565863 6156 4145 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ADM 17121723 6158 4146 ALB 213 TRANSPORTER, DRUGGABLE GENOME Activated recombinant FVII-albumin fusion protein 6159 4147 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR APX005M APX-005M 6160 4148 PTCH1 5727 CLINICALLY ACTIONABLE, TRANSPORTER inhibitor VISMODEGIB VISMODEGIB 6161 4149 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-124573 CHEMBL525826 6162 4150 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER DENDROAMIDE A DENDROAMIDE A 8786364 6163 4151 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR PROTOPORPHYRIN PROTOPORPHYRIN 6166 4152 GRK2 156 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, G PROTEIN COUPLED RECEPTOR, ENZYME US9493490, L 6167 4153 REEP5 7905 NA sertraline SERTRALINE 22795047 6168 4154 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID25991433-Compound-P4 6170 4155 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NITROMIDE NITROMIDE 6171 4156 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE MITOMYCIN C 15782115 6174 4157 MMP16 4325 CELL SURFACE, DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166829 6176 4158 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ABBV-399 TELISOTUZUMAB VEDOTIN 6177 4159 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENOTHIAZINE PHENOTHIAZINE 6178 4160 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER CEFMETAZOLE CEFMETAZOLE 22166395 6179 4161 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE ISOPROTERENOL ISOPROTERENOL 14732742 6180 4162 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ANGIOGENESIS INHIBITOR 15457133 6181 4163 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BUTYRYLHYDROXAMIC ACID BUTYRYLHYDROXAMIC ACID 21874153 6182 4164 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME AZATADINE AZATADINE 6183 4165 XDH 7498 DRUGGABLE GENOME, ENZYME CLARITHROMYCIN CLARITHROMYCIN 14730107 6184 4166 MAPT 4137 DRUGGABLE GENOME GNF-PF-2755 CHEMBL600738 6186 4167 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1234354 PF-04691502 6187 4168 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR LAUROGUADINE LAUROGUADINE 6188 4169 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-743899 CHEMBL101804 6190 4170 FMO3 2328 ENZYME, DRUGGABLE GENOME sulindac SULINDAC 6191 4171 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (R,S)-INDATRALINE (R,S)-INDATRALINE 6196 4172 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NORBINALTORPHIMINE NORBINALTORPHIMINE 6197 4173 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TENIPOSIDE TENIPOSIDE 9543255 6198 4174 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER TENOFOVIR TENOFOVIR 17172311 6199 4175 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AT-7519 AT-7519 18656911 6200 4176 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 178102559 NINTEDANIB 6203 4177 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1280 VERAPAMIL HYDROCHLORIDE 6205 4178 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor RUXOLITINIB RUXOLITINIB 6206 4179 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103435 METHOCARBAMOL 6207 4180 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-57 6208 4181 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CPI-0610 6209 4182 ARID1A 8289 CLINICALLY ACTIONABLE DASATINIB DASATINIB 27364904 6210 4183 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (-)-THALIPORPHINE CHEMBL1394328 6211 4184 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME LY2181308 GATAPARSEN 6212 4185 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MAPROTILINE HYDROCHLORIDE MAPROTILINE HYDROCHLORIDE 6213 4186 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE DHT ANDROSTANOLONE 17657240 6216 4187 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651330 XAMOTEROL 6217 4188 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SERTINDOLE SERTINDOLE 6218 4189 MVK 4598 KINASE, ENZYME inhibitor 135651475 6219 4190 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME SANGUINARIUM SANGUINARIUM 6221 4191 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Xanthine derivative 1 6222 4192 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME GINSENOSIDE RH1 GINSENOSIDE RH1 26420067 6223 4193 TUBB2A 7280 DRUGGABLE GENOME ANHYDROVINBLASTIN 6224 4194 NDUFS2 4720 ENZYME inhibitor CHEMBL3545135 NV-128 6225 4195 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER LIPOSOMAL DOXORUBICIN 12138343 6227 4196 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE AMG 0001 6229 4197 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR WEDELOLACTONE WEDELOLACTONE 6232 4198 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LOVASTATIN LOVASTATIN 22931300 6235 4199 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME RVX-208 APABETALONE 6238 4200 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL190 THEOPHYLLINE 6240 4201 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE DEPHOSTATIN DEPHOSTATIN 6241 4202 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Biaromatic compound 1 6243 4203 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL751 BROMFENAC SODIUM 6244 4204 CP 1356 DRUGGABLE GENOME, ENZYME SODIUM MOLYBDATE 7504610 6245 4205 TUBB 203068 DRUGGABLE GENOME inhibitor 178103457 VINBLASTINE 6246 4206 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE ABT-767 6247 4207 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650332 CHEMBL435278 6249 4208 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE ANTIINFLAMMATORY AGENTS 8423594 6250 4209 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BAS 01152706 CHEMBL2002487 6252 4210 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-47a 6254 4211 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 363894214 SITRAVATINIB 6255 4212 RHOA 387 KINASE, CLINICALLY ACTIONABLE pravastatin PRAVASTATIN 23166513 6256 4213 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565648 6257 4214 GAPDH 2597 DRUGGABLE GENOME, ENZYME PURPUROGALLIN PURPUROGALLIN 6258 4215 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR GEFITINIB GEFITINIB 6261 4216 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SULFINPYRAZONE SULFINPYRAZONE 6262 4217 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE LITHOGLYCOCHOLATE LITHOGLYCOCHOLATE 23489211 6263 4218 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102586 6264 4219 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PACLITAXEL PACLITAXEL 29584549 6266 4220 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME RHAMNETIN RHAMNETIN 24397781 6269 4221 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TERTATOLOL TERTATOLOL 2903243 6272 4222 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME SPERMINE BIS-1-NAPG CHEMBL2347630 23434419 6273 4223 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME KO-947 6274 4224 TFAP2A 7020 TRANSCRIPTION FACTOR HORMONES 12704799 6277 4225 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SJ000113972 CHEMBL591137 6278 4226 POLI 11201 DNA REPAIR 2,3,4-TRIHYDROXYBENZOPHENONE CHEMBL1527 6279 4227 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE fluorouracil FLUOROURACIL 23567490 6280 4228 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE phenazopyridine PHENAZOPYRIDINE 24372186,20701405,6125724,6410650 6282 4229 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME AMOXAPINE AMOXAPINE 6283 4230 ALDH3A1 218 DRUGGABLE GENOME, ENZYME DISULFIRAM DISULFIRAM 2185582 6286 4231 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR RESMINOSTAT RESMINOSTAT 6287 4232 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor BGJ398 INFIGRATINIB 6288 4233 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Eliglustat ELIGLUSTAT 6289 4234 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 7-NITROINDAZOLE 7-NITROINDAZOLE 6290 4235 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652666 ARECOLINE 6292 4236 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 381118846 6295 4237 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NALTREXONE HYDROCHLORIDE NALTREXONE HYDROCHLORIDE 6296 4238 PSMA8 143471 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL3545432 IXAZOMIB CITRATE 6297 4239 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 404859021 6298 4240 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME N-(BENZYLCARBAMOTHIOYL)BENZAMIDE CHEMBL1478462 6300 4241 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR olaparib OLAPARIB 6301 4242 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 310264720 6302 4243 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME ASTERRIC ACID ASTERRIC ACID 6304 4244 TARDBP 23435 TUMOR SUPPRESSOR DNDI1416982 CHEMBL1479114 6306 4245 SV2A 9900 DRUGGABLE GENOME, TRANSPORTER modulator CHEMBL1286 LEVETIRACETAM 6310 4246 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE E-7050 GOLVATINIB 6313 4247 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TRASTUZUMAB TRASTUZUMAB 27900589,20504363,16091755,31453370,22257673,30452336,26598547,11248153,27108243,18555254,26296355,22149875,29523624,26874901,25601188,20728210,30857956,19289619,23204226,15911866,29320312,25693012,29146401,25370464,29584549,22493419,27697991,26243863,16236737,20124187 6314 4248 SRSF10 10772 NA Cynarin CYNARIN 6315 4249 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32u 6316 4250 SMN1 6606 DRUGGABLE GENOME XANTHYLETIN XANTHYLETIN 6318 4251 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE IRINOTECAN IRINOTECAN 6319 4252 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor NINTEDANIB NINTEDANIB 6320 4253 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR deferasirox DEFERASIROX 30651574 6321 4254 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE Lestaurtinib LESTAURTINIB 16258068 6322 4255 HBB 3043 DRUGGABLE GENOME, ENZYME OXY-111A 6323 4256 TARDBP 23435 TUMOR SUPPRESSOR DEXIBUPROFEN DEXIBUPROFEN 6324 4257 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE peginterferon alfa-2b 6325 4258 KDM4A 9682 DRUGGABLE GENOME, ENZYME AG-528 CHEMBL56542 6327 4259 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 9-CIS RETINOIC ACID 12644300 6330 4260 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100293 6332 4261 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CLORAZEPATE CLORAZEPIC ACID 6334 4262 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565924 6335 4263 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FOMEPIZOLE FOMEPIZOLE 6337 4264 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ZINC CHLORIDE 16585387 6339 4265 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1194 PRILOCAINE 6340 4266 MIF 4282 DRUGGABLE GENOME, CELL SURFACE COR100140 6341 4267 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME PF-562271 PF-00562271 6343 4268 UMPS 7372 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE capecitabine CAPECITABINE 20647221,28347776,16818689 6346 4269 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ETHINYL ESTRADIOL ETHINYL ESTRADIOL 22931300 6347 4270 PSMA7 5688 PROTEASE, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 24524217 6348 4271 RACGAP1 29127 NA 4-(N,NDIMETHYLAMINO)BENZALDOXIME CHEMBL498513 6350 4272 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 inhibitor 252827405 6351 4273 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR GW441756X GW441756X 6353 4274 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AGI-5198 23558169 6355 4275 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER remifentanil REMIFENTANIL 29755652 6356 4276 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Pyrido[1,2-a]indole-1.-carboxylic acid analog 4 6357 4277 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE BAY1125976 6358 4278 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 340590280 DAGROCORAT 6359 4279 GBA 2629 DRUGGABLE GENOME, ENZYME 404859139 AMBROXOL 6361 4280 CD37 951 DRUGGABLE GENOME antibody 374883837 6362 4281 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 374883878 ABROCITINIB 6363 4282 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 310264724 LY-3009120 6365 4283 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE IMATINIB IMATINIB 6366 4284 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GO-6976 GO-6976 6367 4285 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103641 6369 4286 PTGS1 5742 ENZYME, DRUGGABLE GENOME DIFLUNISAL DIFLUNISAL 6370 4287 ALOX15 246 ENZYME, DRUGGABLE GENOME DITHIOLETHIONE DITHIOLETHIONE 6371 4288 SUMO2 6613 ENZYME BITHIONOLOXIDE BITHIONOLOXIDE 6372 4289 TSPO 706 DRUGGABLE GENOME Benzothiazepine analog 2 6374 4290 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE MK-0354 CHEMBL456145 6375 4291 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME EPINEPHRINE BITARTRATE EPINEPHRINE BITARTRATE 6376 4292 NOS2 4843 DRUGGABLE GENOME, ENZYME TILARGININE TILARGININE 6377 4293 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE TCDD 7530807 6378 4294 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHLOROETHYLCLONIDINE CHLOROETHYLCLONIDINE 6379 4295 PRRC2A 7916 NA carbamazepine CARBAMAZEPINE 16538176 6380 4296 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL1201023 ORPHENADRINE HYDROCHLORIDE 6381 4297 ACAT1 38 ENZYME SULFASALAZINE SULFASALAZINE 6382 4298 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PHENELZINE PHENELZINE 6383 4299 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-34a 6385 4300 IGFBP1 3484 DRUGGABLE GENOME ORAL CONTRACEPTIVE 8530593 6386 4301 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME antibody ZALTRAP ZALTRAP 6387 4302 GMNN 51053 DRUGGABLE GENOME PROTOAPIGENONE PROTOAPIGENONE 6388 4303 MAPT 4137 DRUGGABLE GENOME GNF-PF-840 CHEMBL601605 6389 4304 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME NITAZOXANIDE NITAZOXANIDE 6390 4305 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Aminopyrimidine derivative 5 6391 4306 TUBA4A 7277 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 6393 4307 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3545091 XEN403 6394 4308 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 lovastatin LOVASTATIN 6395 4309 CFB 629 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166853 6397 4310 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650917 6398 4311 RGS4 5999 DRUGGABLE GENOME OXITRIPTAN OXITRIPTAN 6399 4312 ORAI2 80228 ION CHANNEL blocker 381118798 6400 4313 GATA4 2626 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE NSC-85661 CHEMBL1684098 21310620 6401 4314 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL1201585 TRASTUZUMAB 6402 4315 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL inhibitor 135650722 NISOLDIPINE 6403 4316 PTGES 9536 DRUGGABLE GENOME, ENZYME Imidazopyridine derivative 5 6404 4317 CDH11 1009 CLINICALLY ACTIONABLE RG6125 6407 4318 ATP5F1E 514 TRANSPORTER glucocorticoids 26307125 6409 4319 BRCA2 675 CLINICALLY ACTIONABLE Niraparib NIRAPARIB 6410 4320 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME QUERCETIN QUERCETIN 6411 4321 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR MOMETASONE MOMETASONE 6412 4322 POLI 11201 DNA REPAIR DNDI1417523 CHEMBL598663 6414 4323 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE PMID26882240-Compound-32 6415 4324 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PD-0325901 PD-0325901 26272063 6416 4325 KDM4A 9682 DRUGGABLE GENOME, ENZYME STICTIC ACID STICTIC ACID 6417 4326 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BKM120 BUPARLISIB 6419 4327 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME TAE-684 TAE-684 6420 4328 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR ORTHO-PHTHALALDEHYDE ORTHO-PHTHALALDEHYDE 6421 4329 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL586701 ZSTK-474 6422 4330 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545246 LIFIRAFENIB 6423 4331 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE II-B08 20170098 6424 4332 KDM4A 9682 DRUGGABLE GENOME, ENZYME (S)-MAP4 HCL CHEMBL1256510 6426 4333 TNKS2 80351 DRUGGABLE GENOME, ENZYME inhibitor 404859121 6427 4334 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-175743 CHEMBL1609016 6428 4335 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER Lobeline LOBELINE 6429 4336 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Merestinib, LY2801653 6430 4337 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Eniluracil ENILURACIL 6431 4338 RAPGEF3 10411 ENZYME 8-BROMO-CAMP SODIUM CHEMBL1256796 6432 4339 AKT1S1 84335 KINASE, DRUGGABLE GENOME GEDATOLISIB GEDATOLISIB 20166697 6433 4340 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ABEMACICLIB ABEMACICLIB 27217383 6434 4341 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-49 6436 4342 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-33 6439 4343 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIMPINELLIN PIMPINELLIN 6440 4344 AKR1C3 8644 ENZYME, DRUGGABLE GENOME docetaxel DOCETAXEL 23116553 6441 4345 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ABIETIC ACID ABIETIC ACID 24799257 6444 4346 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR TCDD 12606293 6445 4347 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DNDI1417072 CHEMBL1310701 6446 4348 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Regorafenib REGORAFENIB 21170960,27371698,25239608 6447 4349 HMGCR 3156 ENZYME, DRUGGABLE GENOME FLUVASTATIN FLUVASTATIN 6449 4350 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PHA-767491 CHEMBL225519 6451 4351 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Ulocuplumab ULOCUPLUMAB 6454 4352 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor SF1126 6455 4353 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW280670X GW280670X 6456 4354 MICB 4277 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE peginterferon alfa-2a 6457 4355 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200618 FEXOFENADINE HYDROCHLORIDE 6458 4356 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PHTHALAZINONE PHTHALAZINONE 6459 4357 CCND3 896 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PALBOCICLIB PALBOCICLIB 23079656 6461 4358 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1237135 MAPROTILINE HYDROCHLORIDE 6462 4359 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE Cisplatin CISPLATIN 28652249 6463 4360 SCTR 6344 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651884 SECRETIN 6464 4361 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR partial agonist CHEMBL1516474 TEGASEROD MALEATE 6465 4362 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE CEDIRANIB CEDIRANIB 6466 4363 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME TRIMIPRAMINE TRIMIPRAMINE 6467 4364 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651328 6471 4365 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE cilostazol CILOSTAZOL 6473 4366 KAT2B 8850 ENZYME, DRUGGABLE GENOME opioids 6475 4367 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL154 NAPROXEN 6477 4368 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME AST-487 AST-487 6478 4369 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME LEUCETTAMINE B LEUCETTAMINE B 22998443 6479 4370 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 6-CHLOROMELATONIN CHEMBL34730 6481 4371 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LINURON LINURON 6482 4372 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME PRT4445 6483 4373 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME celecoxib CELECOXIB 22336956 6484 4374 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE Dendritic cell vaccine 6485 4375 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE MRX-801 6486 4376 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ALEXIDINE DIHYDROCHLORIDE ALEXIDINE DIHYDROCHLORIDE 6487 4377 BAZ2B 29994 NA NSC-71033 CHEMBL116548 6488 4378 UBE2N 7334 ENZYME, DRUGGABLE GENOME SPHINGOSINE SPHINGOSINE 6489 4379 MAP3K9 4293 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 310264738 CERDULATINIB 6490 4380 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE LORATADINE LORATADINE 6492 4381 PLCG1 5335 ENZYME, KINASE, PHOSPHOLIPASE, DRUGGABLE GENOME propionic acid derivatives 26398624 6493 4382 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 249565688 CHEMBL1765740 6494 4383 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 252166845 6496 4384 PSORS1C1 170679 NA etanercept ETANERCEPT 6498 4385 GATA4 2626 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE Drugs used in alcohol dependence 20585342 6499 4386 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-1008 CHEMBL602424 6500 4387 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHENOBARBITAL PHENOBARBITAL 22931300 6502 4388 RACGAP1 29127 NA COUMESTROL COUMESTROL 6503 4389 HTT 3064 DRUGGABLE GENOME EDO-S101 TINOSTAMUSTINE 6504 4390 MEG3 55384 NA Platinum compounds 6505 4391 TXNRD1 7296 DRUGGABLE GENOME Metal complex derivative 3 6507 4392 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3039504 NINTEDANIB ESYLATE 6508 4393 CPB2 1361 DRUGGABLE GENOME, ENZYME, PROTEASE SAR-126119 6509 4394 SH2B1 25970 KINASE valproic acid 28694205 6510 4395 IL13RA1 3597 EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE, DRUGGABLE GENOME CINTREDEKIN BESUDOTOX 6511 4396 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR muraglitazar MURAGLITAZAR 18794727 6512 4397 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE VEMURAFENIB VEMURAFENIB 27325282,26359985 6513 4398 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME DNDI1417195 CHEMBL1303948 6514 4399 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LAPATINIB LAPATINIB 19718025 6516 4400 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME 178101632 FILGRASTIM 6517 4401 PDE5A 8654 ENZYME, DRUGGABLE GENOME ICARIIN ICARIIN 6518 4402 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME AZD-1775 ADAVOSERTIB 6519 4403 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2103827 DROXIDOPA 6520 4404 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE CS1229 6522 4405 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL2103878 ODELEPRAN 6526 4406 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL XEN402 6527 4407 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE docetaxel DOCETAXEL 21783417,22285168 6528 4408 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE WZ4002 22046346 6529 4409 TUBA1A 7846 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 6530 4410 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR RAPAMYCIN SIROLIMUS 12907620 6532 4411 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme4Upper 6533 4412 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Vemurafenib VEMURAFENIB 27312529 6534 4413 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GREEN TEA POLYPHENOLS 11830514 6535 4414 TUBA1B 10376 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 6537 4415 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PD-0166285 PD-0166285 6538 4416 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL2103847 TOSEDOSTAT 6539 4417 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PKI-402 CHEMBL589258 20371716 6540 4418 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 E-GUGGULSTERONE E-GUGGULSTERONE 6541 4419 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEXTRAN SULFATE SODIUM 17178849 6542 4420 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME L-751250 6544 4421 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE SB-220025 SB-220025 6546 4422 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649983 BERAPROST 6548 4423 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 THIOPERAMIDE THIOPERAMIDE 6549 4424 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 405560501 6550 4425 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135652434 RELAXIN 6551 4426 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME methadone METHADONE 17329992,27286724,17178267,17502774,28320034,21902500,17638512,23249875,16338275,11470993,27289271,30907440,21790905,25556837 6552 4427 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CEFOTAXIME CEFOTAXIME 6553 4428 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GW0742 CHEMBL38508 6554 4429 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME CARFILZOMIB CARFILZOMIB 6555 4430 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR ENOXOLONE ENOXOLONE 24461294 6556 4431 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE buprenorphine BUPRENORPHINE 18695978 6557 4432 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 1,6-diazanaphthalenes and pyrido[2,3-d] pyrimidine derivative 1 6558 4433 ATAD5 79915 NA PICEATANNOL PICEATANNOL 6559 4434 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR SP-600125 SP-600125 6560 4435 HTT 3064 DRUGGABLE GENOME OXYBENZONE OXYBENZONE 6562 4436 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE HYDROCORTISONE HYDROCORTISONE 6565 4437 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 6567 4438 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 252166595 BIMIRALISIB 6568 4439 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Chloroquine CHLOROQUINE 6569 4440 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR H2O2 18006461 6570 4441 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE ZSTK474 6572 4442 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LABETALOL LABETALOL 6575 4443 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ACID BLUE 129 ACID BLUE 129 6578 4444 BRCA2 675 CLINICALLY ACTIONABLE RUCAPARIB RUCAPARIB 6579 4445 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102743 6580 4446 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 5,7,3',5'-TETRAHYDROXYFLAVANONE CHEMBL307893 6582 4447 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Donepezil DONEPEZIL 6583 4448 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL1567 SUNITINIB MALATE 6584 4449 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Ospemifene OSPEMIFENE 6585 4450 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ENTINOSTAT ENTINOSTAT 6586 4451 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME AMCINONIDE AMCINONIDE 6588 4452 BMP7 655 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR pegaspargase PEGASPARGASE 26590194 6589 4453 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103585 ROMIDEPSIN 6590 4454 KDM6A 7403 ENZYME, CLINICALLY ACTIONABLE Tazemetostat TAZEMETOSTAT 6591 4455 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHANESULFONIC ACID METHYL ESTER METHANESULFONIC ACID METHYL ESTER 6592 4456 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ARSENIC TRIOXIDE 16613325 6594 4457 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CHEMBL2109300 GSK933776 6595 4458 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BETAXOLOL BETAXOLOL 2903243 6596 4459 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CO-1686 ROCILETINIB 6597 4460 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28117607-Compound-21 6599 4461 PDE9A 5152 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL628 PENTOXIFYLLINE 6600 4462 ADH4 127 DRUGGABLE GENOME, ENZYME ETHANOL ALCOHOL 3610585 6601 4463 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL2103836 IMAGABALIN 6604 4464 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE raltegravir RALTEGRAVIR 6605 4465 SMPD1 6609 ENZYME, DRUGGABLE GENOME inhibitor 404859087 6606 4466 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ETHYNODIOL DIACETATE ETHYNODIOL DIACETATE 6607 4467 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Olaparib OLAPARIB 6608 4468 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TENIPOSIDE TENIPOSIDE 6609 4469 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER quinine QUININE 6611 4470 GHRL 51738 DRUGGABLE GENOME RALOXIFENE RALOXIFENE 18164562 6614 4471 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE GSK2141795 UPROSERTIB 6616 4472 MAOA 4128 DRUGGABLE GENOME, ENZYME Psoralen PSORALEN 6617 4473 CRTC1 23373 CLINICALLY ACTIONABLE XL765 6618 4474 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR ARSENIC TRIOXIDE 16638192 6619 4475 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME LEVONORDEFRIN LEVONORDEFRIN 6620 4476 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ZEARALENONE ZEARALENONE 6621 4477 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor GDC-0941 PICTILISIB 6622 4478 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR VORINOSTAT VORINOSTAT 6623 4479 KDM4A 9682 DRUGGABLE GENOME, ENZYME GUAIAZULENE GUAIAZULEN 6624 4480 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TOSYL-L-LYSINE CHLOROMETHYL KETONE CHEMBL466465 6625 4481 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR UVB 11874477 6626 4482 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE AZD-1152-HQPA AZD-1152-HQPA 6628 4483 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR AZD3463 26372962 6630 4484 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER QUINACRINE DIHYDROCHLORIDE QUINACRINE DIHYDROCHLORIDE 6631 4485 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM BROMIDE 6632 4486 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201639 INSULIN ZINC SUSP BEEF 6633 4487 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Fused benzoheterocycle amide derivative 1 6635 4488 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SB-431542 SB-431542 6637 4489 AMH 268 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GONADOTROPINS 347363,8810722 6638 4490 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME DNDI1417467 CHEMBL1997335 6639 4491 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL2062261 LEVORPHANOL TARTRATE 6640 4492 NOS2 4843 DRUGGABLE GENOME, ENZYME HP-228 6643 4493 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME ANTIPLATELET AGENT 15253106 6644 4494 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE 12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE 6647 4495 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor BAY1000394 6649 4496 LTF 4057 CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, PROTEASE BACITRACIN BACITRACIN 12042436 6651 4497 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178102191 6652 4498 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417827 CHEMBL1363249 6654 4499 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 363894185 6655 4500 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ANISALDEHYDE ANISALDEHYDE 6657 4501 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE FORMESTANE FORMESTANE 18256205 6658 4502 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORALIN CHLORALIN 6659 4503 KLK4 9622 PROTEASE, DRUGGABLE GENOME, ENZYME Ecallantide ECALLANTIDE 6661 4504 BAZ2B 29994 NA BENZTHIAZIDE BENZTHIAZIDE 6662 4505 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME PMID27998201-Compound-7 6663 4506 ATXN2 6311 NA AMSACRINE AMSACRINE 6665 4507 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-100 6666 4508 MAOB 4129 DRUGGABLE GENOME, ENZYME Coumaricacid 6670 4509 POLI 11201 DNA REPAIR NSC-69187 CHEMBL19954 6675 4510 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FF-284 25169980,28034880,25589496 6676 4511 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL2068839 RISLENEMDAZ 6677 4512 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CGM097 CGM-097 27659046 6678 4513 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ERB-257 6679 4514 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor ERLOTINIB ERLOTINIB 6680 4515 TNNT2 7139 DRUGGABLE GENOME PYROGALLOL RED PYROGALLOL RED 6681 4516 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE SB-0304 CHEMBL409225 21978284 6682 4517 PAEP 5047 DRUGGABLE GENOME GENISTEIN GENISTEIN 12820358 6683 4518 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652022 LANREOTIDE 6684 4519 GLS 2744 ENZYME LINOLENIC ACID LINOLENIC ACID 6685 4520 PLIN3 10226 NA IDURSULFASE IDURSULFASE 6686 4521 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BROMOCHLOROACETIC ACID BROMOCHLOROACETIC ACID 6688 4522 DHFR 1719 DRUGGABLE GENOME, ENZYME CH-4051 6689 4523 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL445813 AT-7519 6690 4524 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 405067325 OTAMIXABAN 6691 4525 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ARACHIDONIC ACID ARACHIDONIC ACID 6692 4526 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GNF-PF-2893 CHEMBL312032 6694 4527 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL2103840 DINACICLIB 6695 4528 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME HOMOHARRINGTONINE OMACETAXINE MEPESUCCINATE 15854289 6697 4529 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR N'-(2,4-DIHYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE CHEMBL199592 6698 4530 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TYRPHOSTIN AG-112 CHEMBL76589 6699 4531 PDE9A 5152 DRUGGABLE GENOME, ENZYME inhibitor 135651355 ZAPRINAST 6702 4532 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ANTI-CD20 (HA20) MONOCLONAL ANTIBODY 6704 4533 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-2359 CHEMBL610622 6705 4534 ATP2A3 489 DRUGGABLE GENOME, TRANSPORTER, ENZYME celecoxib CELECOXIB 22336956 6706 4535 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200903 SECOBARBITAL SODIUM 6707 4536 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL445813 AT-7519 6708 4537 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NS-1619 CHEMBL384903 6709 4538 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME MK 1775 6710 4539 BPI 671 DRUGGABLE GENOME XOMA-629 6711 4540 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME Neu-2000 6712 4541 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME KETOTIFEN KETOTIFEN 6714 4542 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SIMAZINE SIMAZINE 6715 4543 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 405560506 6717 4544 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SODIUM LAURYL SULFATE SODIUM LAURYL SULFATE 6719 4545 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1722 METHYLPHENIDATE HYDROCHLORIDE 6721 4546 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PENFLURIDOL PENFLURIDOL 6722 4547 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME rhodamine 123 11559526 6723 4548 ALDH1A2 8854 DRUGGABLE GENOME, ENZYME hydrochlorothiazide HYDROCHLOROTHIAZIDE 29097388 6724 4549 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PMID30107136-Compound-Example2 6725 4550 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2-(ALPHA-NAPHTHOYL)ETHYLTRIMETHYLAMMONIUM IODIDE CHEMBL1255936 6726 4551 RRM2 6241 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200983 GALLIUM NITRATE 6727 4552 IL1B 3553 KINASE, DRUGGABLE GENOME RESVERATROL RESVERATROL 16389574 6728 4553 ATAD5 79915 NA TRIPHENYLSTANNYL ACETATE TRIPHENYLSTANNYL ACETATE 6730 4554 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Azilsartan AZILSARTAN 6733 4555 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ARA-C 14713572 6734 4556 ALOX15B 247 DRUGGABLE GENOME, ENZYME CAPSAZEPINE CAPSAZEPINE 6736 4557 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Dihydroergotamine nasal 6738 4558 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Imidazo bicyclic iminium derivative 9 6741 4559 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Dasatinib DASATINIB 6743 4560 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHENOXYBENZAMINE PHENOXYBENZAMINE 22931300 6744 4561 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8987457, 198 6745 4562 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME atrasentan ATRASENTAN 16513443 6746 4563 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CID 887167 CHEMBL260342 6748 4564 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 178103880 TICLOPIDINE 6749 4565 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CAPSAZEPINE CAPSAZEPINE 6750 4566 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Indole-based analog 2 6751 4567 POLI 11201 DNA REPAIR TOLONIUM CHLORIDE TOLONIUM CHLORIDE 6752 4568 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME SR-123781A 6753 4569 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 374883876 6754 4570 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CELECOXIB CELECOXIB 6755 4571 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor BAY80-6946 COPANLISIB 6756 4572 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE M9831 6759 4573 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Fludarabine FLUDARABINE 20739657 6760 4574 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor SORAFENIB SORAFENIB 6761 4575 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PRAZOSIN HYDROCHLORIDE 11406472 6762 4576 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 315661256 REBASTINIB 6763 4577 HR 55806 NUCLEAR HORMONE RECEPTOR Levomequitazine 6764 4578 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 6-METHYLCOUMARIN CHEMBL443436 6765 4579 KDM6A 7403 ENZYME, CLINICALLY ACTIONABLE inhibitor 178103606 6766 4580 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651282 NALFURAFINE 6768 4581 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DEMETHYLENCECALIN DEMETHYLENCECALIN 6769 4582 GGCT 79017 ENZYME inhibitor 381744946 6770 4583 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 12 6771 4584 POLI 11201 DNA REPAIR CEFOTAXIME SODIUM CEFOTAXIME SODIUM 6773 4585 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 fesoterodine FESOTERODINE 6774 4586 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME CS-038 6775 4587 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor DASATINIB DASATINIB 6776 4588 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME GEFITINIB GEFITINIB 6777 4589 POLK 51426 DNA REPAIR, ENZYME DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 6778 4590 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE inhibitor 223366154 6779 4591 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BETANAPHTHOL BETANAPHTHOL 6780 4592 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME propafenone PROPAFENONE 2713973,14653957,17001296,12421483,17460029 6781 4593 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565579 APITOLISIB 6783 4594 GMNN 51053 DRUGGABLE GENOME GNF-PF-5151 CHEMBL576208 6784 4595 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DEXMEDETOMIDINE DEXMEDETOMIDINE 6785 4596 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXYQUINOLINE SULFATE OXYQUINOLINE SULFATE 6786 4597 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR antagonist 135650105 6790 4598 MAOB 4129 DRUGGABLE GENOME, ENZYME Ethylvanillin 6791 4599 BAZ2B 29994 NA NSC-353720 CHEMBL1408276 6795 4600 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE NSC-695801 CHEMBL461193 6796 4601 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 6797 4602 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CARBOPLATIN CARBOPLATIN 12360105 6798 4603 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID27724045-Compound-15 6799 4604 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor GSK2126458 OMIPALISIB 6801 4605 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor AMUVATINIB AMUVATINIB 6802 4606 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor SOPHORETIN QUERCETIN 6804 4607 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201063 PROPAFENONE HYDROCHLORIDE 6805 4608 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 223366076 6806 4609 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 erlotinib ERLOTINIB 6807 4610 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME HMBA 9067579 6809 4611 NAPEPLD 222236 ENZYME ETHANOL ALCOHOL 17302558 6812 4612 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Decitabine DECITABINE 24874286 6813 4613 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE DOXORUBICIN DOXORUBICIN 23585524 6814 4614 MARCKSL1 65108 KINASE IFN 11483670 6815 4615 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GSK-961081 6816 4616 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 (S)-NIMODIPINE (S)-NIMODIPINE 6817 4617 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-38 6819 4618 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PURPUROGALLIN PURPUROGALLIN 6820 4619 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DZNeP 25605023 6822 4620 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CETUXIMAB CETUXIMAB 21163703,19223544 6823 4621 FGA 2243 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, FIBRINOGEN RECOMBINANT FACTOR IX FC FUSION PROTEIN 6824 4622 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR LACTULOSE LACTULOSE 11355146 6825 4623 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME 5,8,11,14-EICOSATETRAYNOIC ACID CHEMBL458328 6826 4624 TUBB3 10381 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 6827 4625 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR GP100 15665624 6829 4626 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME OPHIOBOLIN O OPHIOBOLIN O 22130129 6833 4627 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 315661321 UPADACITINIB 6837 4628 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL1952329 SGI-1776 6838 4629 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME HMPL-004 ANDROGRAPHOLIDE 6839 4630 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1201463 CODEINE POLISTIREX 6842 4631 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME METHOTRIMEPRAZINE LEVOMEPROMAZINE 6843 4632 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ESMOLOL ESMOLOL 6844 4633 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Sym015 6846 4634 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR lisinopril LISINOPRIL 12522467 6848 4635 RACGAP1 29127 NA SULFURETIN SULFURETIN 6849 4636 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE BDBM50061612 6850 4637 MKNK1 8569 SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, ENZYME CGP-57380 CHEMBL1240885 25800647 6851 4638 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 348353623 6852 4639 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Clemastine CLEMASTINE 6853 4640 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 lidocaine LIDOCAINE 9187528 6855 4641 NOS1 4842 DRUGGABLE GENOME, ENZYME DHEA PRASTERONE 16836960 6856 4642 POR 5447 ENZYME, DRUGGABLE GENOME sirolimus SIROLIMUS 23974086 6857 4643 ATAD5 79915 NA GNF-PF-3546 CHEMBL598680 6858 4644 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamate derivative 16 6861 4645 TGFB2 7042 GROWTH FACTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME FANG vaccine 6862 4646 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR TCMDC-123591 CHEMBL588234 6863 4647 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL1879463 DACTOLISIB 6864 4648 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652338 6865 4649 GMNN 51053 DRUGGABLE GENOME SEW-03621 CHEMBL1271059 6866 4650 MAP3K14 9020 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE inhibitor 374883851 6867 4651 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Gefitinib GEFITINIB 6869 4652 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Codeine CODEINE 6871 4653 TUBB4B 10383 DRUGGABLE GENOME CHEMBL2108628 PACLITAXEL POLIGLUMEX 6873 4654 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-42 6874 4655 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrimidopyridazinone derivative 2 6875 4656 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FENTICLOR FENTICLOR 6877 4657 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE methotrexate METHOTREXATE 12972956,16870553 6878 4658 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME KETOCONAZOLE KETOCONAZOLE 6881 4659 GLS 2744 ENZYME ANTIANGIOGENIC 15743040 6882 4660 ADAMTS5 11096 DRUGGABLE GENOME, ENZYME, PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE AGG-523 AGG-523 6883 4661 ATAD5 79915 NA 8-FLUOROTRYPTANTHRIN CHEMBL1098875 6884 4662 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME LINOLENIC ACID LINOLENIC ACID 6885 4663 ALOX15 246 ENZYME, DRUGGABLE GENOME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 6887 4664 PTGS2 5743 DRUGGABLE GENOME, ENZYME BALSALAZIDE BALSALAZIDE 6888 4665 MYD88 4615 CLINICALLY ACTIONABLE Ibrutinib IBRUTINIB 6889 4666 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID27744724-Compound-18 6890 4667 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE FPL-55712 FPL-55712 6891 4668 DGAT1 8694 ENZYME, DRUGGABLE GENOME PMID25470667-Compound-Figure4-1A 6892 4669 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SAPPANONE A DIMETHYL ETHER SAPPANONE A DIMETHYL ETHER 6893 4670 HTT 3064 DRUGGABLE GENOME DNDI1417346 CHEMBL1490332 6894 4671 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE MARIMASTAT MARIMASTAT 6896 4672 KDM4A 9682 DRUGGABLE GENOME, ENZYME MMV006513 CHEMBL585622 6897 4673 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Everolimus EVEROLIMUS 26544513 6899 4674 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME Platinum compounds 22441531 6900 4675 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor SELICICLIB SELICICLIB 6901 4676 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OXYPHENBUTAZONE OXYPHENBUTAZONE 6902 4677 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Biomed 101 6903 4678 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651301 6904 4679 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-11 6905 4680 ATXN2 6311 NA DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 6906 4681 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2'-HYDROXYCHALCONE 2'-HYDROXYCHALCONE 6908 4682 HSPB1 3315 DRUGGABLE GENOME DIFFERENTIATION INDUCER 7500647 6910 4683 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650158 DAMGO 6911 4684 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1417132 CHEMBL1492017 6912 4685 COIL 8161 NA EGCG EPIGALOCATECHIN GALLATE 16046615 6913 4686 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR SHIKONIN SHIKONIN 6915 4687 ATAD5 79915 NA 3,5-DIPHENYLISOXAZOLE 3,5-DIPHENYLISOXAZOLE 6919 4688 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME NSC-44661 CHEMBL571228 6920 4689 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME PURPURIN PURPURIN 6921 4690 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor XL147 PILARALISIB 6924 4691 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME Xentuzumab XENTUZUMAB 6926 4692 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3641 CHEMBL599098 6927 4693 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RITONAVIR RITONAVIR 21393461,21953914 6929 4694 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 328083469 6930 4695 TARDBP 23435 TUMOR SUPPRESSOR NSC-407228 CHEMBL74852 6932 4696 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-5510 CHEMBL578741 6936 4697 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME AZD0530 SARACATINIB 6938 4698 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME irinotecan IRINOTECAN 25127363 6939 4699 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE ORNITHINE DECARBOXYLASE INHIBITOR 11876528 6940 4700 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR FULVESTRANT FULVESTRANT 19133777,26407012,25879485,17337183,17275315,19845386,20621492 6942 4701 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-204741 CHEMBL323356 6943 4702 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR KEYHOLE LIMPET HEMOCYANIN 15857404 6947 4703 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 404859078 6948 4704 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME Rilimogene galvacirepvec 6949 4705 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417941 CHEMBL2095095 6950 4706 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL979 MEPROBAMATE 6951 4707 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650941 CHEMBL88272 6954 4708 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ALEFACEPT ALEFACEPT 6956 4709 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRIBROMSALAN TRIBROMSALAN 6959 4710 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR P-PHENYLENEDIAMINE CHEMBL403741 6961 4711 CD83 9308 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CD40L 11093145 6962 4712 RAPGEF3 10411 ENZYME HEXACHLOROPHENE HEXACHLOROPHENE 6963 4713 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor ENMD-2076 ENMD-2076 6964 4714 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135649939 AMITRIPTYLINE 6966 4715 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR PMID26924192-Compound-102 6967 4716 ITGB6 3694 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor 385612210 6968 4717 GMNN 51053 DRUGGABLE GENOME THUNBERGINOL A THUNBERGINOL A 6973 4718 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL BROMAZEPAM BROMAZEPAM 6974 4719 DGAT1 8694 ENZYME, DRUGGABLE GENOME Pyridine-amide derivative 1 6975 4720 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2,4-HEXADIENAL 2,4-HEXADIENAL 6976 4721 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ISOKAEMPFERIDE ISOKAEMPFERIDE 6981 4722 PMEL 6490 DRUGGABLE GENOME Melanoma vaccine 6982 4723 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TOLMETIN SODIUM TOLMETIN SODIUM 6984 4724 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CEFOTAXIME CEFOTAXIME 8354907,10989981 6986 4725 UBE2N 7334 ENZYME, DRUGGABLE GENOME CHLORHEXIDINE CHLORHEXIDINE 6987 4726 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor CHEMBL1200826 LITHIUM CARBONATE 6988 4727 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE nivolumab NIVOLUMAB 6990 4728 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650687 NALTREXONE 6991 4729 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME GSK2798745 GSK2798745 6992 4730 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE inhibitor 384403654 6993 4731 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR DDTC 17052849 6995 4732 CBX1 10951 NA METHYLDOPA (RACEMIC) METHYLDOPA (RACEMIC) 6997 4733 USP1 7398 DNA REPAIR, PROTEASE, ENZYME METHYLBENZETHONIUM METHYLBENZETHONIUM 7004 4734 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102722 7006 4735 DHFR 1719 DRUGGABLE GENOME, ENZYME ANTITUMOR ANTIBIOTIC 8117738 7008 4736 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE Sapanisertib SAPANISERTIB 26574479 7010 4737 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR TPX-0005 7011 4738 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1555 GALANTAMINE HYDROBROMIDE 7015 4739 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL PENTOBARBITAL PENTOBARBITAL 7020 4740 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 135651724 7021 4741 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545283 RIVICICLIB 7025 4742 TARDBP 23435 TUMOR SUPPRESSOR TCMDC-123862 CHEMBL533074 7027 4743 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Triazolo-pyrimidinedione derivative 2 7028 4744 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER Sotrastaurin acetate 7029 4745 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE MABT5102A CRENEZUMAB 7032 4746 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE allosteric modulator 315661107 7033 4747 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PONATINIB PONATINIB 20513156 7034 4748 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR inhibitor CRIZOTINIB CRIZOTINIB 7035 4749 CD37 951 DRUGGABLE GENOME TRU-016 OTLERTUZUMAB 7036 4750 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE SCH-53020 CHEMBL66279 7037 4751 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CARMINE CARMINE 7038 4752 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR DIFFRACTAIC ACID DIFFRACTAIC ACID 7039 4753 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ARACHIDONOYL DOPAMINE ARACHIDONOYL DOPAMINE 7040 4754 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ETHYL VANILLIN ETHYL VANILLIN 7042 4755 MDM4 4194 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, DRUGGABLE GENOME NIVOLUMAB NIVOLUMAB 28351930 7043 4756 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME PF-562271 PF-00562271 7044 4757 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME HOMATROPINE METHYLBROMIDE 7046 4758 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CD20Bi aATC 23529012 7049 4759 CYP4B1 1580 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME thalidomide THALIDOMIDE 20038957 7051 4760 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHLORPROMAZINE CHLORPROMAZINE 22931300 7052 4761 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor AMG900 AMG-900 7053 4762 CYP4B1 1580 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME DEXTRAN SULFATE 15039297 7056 4763 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE tramadol TRAMADOL 18695978 7058 4764 PSMC5 5705 TRANSCRIPTION FACTOR BINDING, PROTEASE inhibitor CARFILZOMIB CARFILZOMIB 7059 4765 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE Indapamide INDAPAMIDE 7060 4766 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEFEROXAMINE DEFEROXAMINE 16950787 7062 4767 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2107779 SEMAPIMOD 7063 4768 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 328083491 SB590885 7064 4769 AOX1 316 DRUGGABLE GENOME azathioprine AZATHIOPRINE 19500084 7065 4770 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL411907 SONOLISIB 7066 4771 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DAIDZEIN DAIDZEIN 7067 4772 KCNC2 3747 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 7069 4773 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Safotibant SAFOTIBANT 7070 4774 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BITHIONOLATE SODIUM BITHIONOLATE SODIUM 7071 4775 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE DICHLOROISOPROTERENOL DICHLOROISOPROTERENOL 2903243 7072 4776 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 178102670 7073 4777 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL49642 INDIBULIN 7074 4778 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME NSC-102045 CHEMBL483633 7075 4779 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Fluocinolone Acetonide 7076 4780 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Ipatasertib IPATASERTIB 26725216 7077 4781 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL3545108 AZD9056 7078 4782 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME LABETALOL HYDROCHLORIDE LABETALOL HYDROCHLORIDE 7081 4783 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ADAPALENE ADAPALENE 7082 4784 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRADIOL ACETATE 7083 4785 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE U0126 17942397 7084 4786 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME MK-2461 MK-2461 7087 4787 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SAR-100842 25593637 7088 4788 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL2107313 BECATECARIN 7089 4789 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME AR-A014418 CHEMBL259850 7090 4790 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774822-Compound-Figure3CompoundI-165 7091 4791 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Hepatitis vaccines 21111021 7093 4792 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 187051820 7094 4793 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME epirubicin EPIRUBICIN 25008867,21362365,20568049 7095 4794 POLK 51426 DNA REPAIR, ENZYME PHENYLSTIBONIC ACID PHENYLSTIBONIC ACID 7096 4795 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CENISERTIB CENISERTIB 7097 4796 TASP1 55617 PROTEASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 252827510 7098 4797 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR N-quinolin-benzene sulphonamide derivative 1 7099 4798 RBX1 9978 DNA REPAIR, ENZYME inhibitor CHEMBL468 THALIDOMIDE 7100 4799 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CPL-7075 LENABASUM 7101 4800 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-48 7102 4801 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-53 7103 4802 SCNN1A 6337 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL585 TRIAMTERENE 7104 4803 ATP5F1E 514 TRANSPORTER etanercept ETANERCEPT 26307125 7106 4804 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE BAY-613606 CHEMBL541400 7107 4805 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE N/A 7108 4806 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR RETINOID 8498603 7109 4807 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL473417 VISMODEGIB 7110 4808 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL429876 CILENGITIDE 7111 4809 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-4481 CHEMBL597251 7113 4810 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE CYC-116 CYC-116 7115 4811 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-25 7118 4812 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 187051793 GIVINOSTAT 7119 4813 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME DABRAFENIB DABRAFENIB 23020132,22608338,24265155,29072975,25399551,23463675,25673644,25452114,25265494,31811016,27283860,27048246,24583796,23031422,25265492,25435907,28947956,28480077,28891408,29431699,28078132 7120 4814 ALOX5 240 DRUGGABLE GENOME, ENZYME MECLOFENAMIC ACID 7123 4815 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME AZD-0837 ATECEGATRAN METOXIL 7124 4816 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BYL719 ALPELISIB 24569456 7125 4817 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME VEMURAFENIB VEMURAFENIB 23020132,22608338,26619011,21483012,22351686,19001320,21156289,20368568,19255327,22048237,19561230,19010912,23549875,25024077,23489023,18541894,24586605,24508103,22773810,23833300,23812671,24576830,19238210,20818844,23612012,23251002,22356324,20857202,22536370,22997239,21163703,15035987,23470635,21663470,24594804,22586120,20413299,22805292,19537845,14679157,22663011,21975775,22038996,22448344,12068308,24163374,19773371,24354346,23325582,24583796,23031422,22735384,21683865,25370471,21639808,22281684,22649091,22241789,24570209,23918947,25989278,22389471,23934108,22180495,23524406,26678033,19018267,24388723,23845441,23614898,25157968,20619739,12460919,24107445,12460918,21594703,20350999,20630094,21426297,19404918,22743296,24396464,22972589,21129611,23406027,25656898 7126 4818 HCN3 57657 DRUGGABLE GENOME, ION CHANNEL blocker 135651358 7127 4819 PSENEN 55851 DRUGGABLE GENOME inhibitor CHEMBL1090771 AVAGACESTAT 7128 4820 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME bromazepam BROMAZEPAM 7130 4821 HTT 3064 DRUGGABLE GENOME GNF-PF-78 CHEMBL579318 7132 4822 PSMD4 5710 NA PROTEASOME INHIBITOR 15899868 7133 4823 NDUFS8 4728 ENZYME inhibitor CHEMBL3545135 NV-128 7134 4824 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME Cyclopenta[d]pyrimidine derivative 1 7135 4825 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-23 7137 4826 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 5-AZACYTIDINE AZACITIDINE 11696442 7138 4827 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME LINIFANIB LINIFANIB 7139 4828 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME CHS-131 7141 4829 MAP3K5 4217 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, ENZYME GS-4997 SELONSERTIB 7143 4830 ARG1 383 ENZYME sodium benzoate / sodium phenylacetate 7144 4831 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME LY-2090314 LY-2090314 7145 4832 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PENTABROMOPHENOL PENTABROMOPHENOL 7148 4833 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-8 7149 4834 PDE4A 5141 DRUGGABLE GENOME, ENZYME OX914 7151 4835 SMN2 6607 DRUGGABLE GENOME GNF-PF-3501 CHEMBL581910 7153 4836 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 249565632 AT-9283 7154 4837 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RETASPIMYCIN RETASPIMYCIN 7155 4838 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME clomipramine CLOMIPRAMINE 10867985 7156 4839 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 halothane HALOTHANE 12386121,19702528,19442086,11038165,14704462,8886611 7157 4840 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME CHEMBL1371 CHLORZOXAZONE 7158 4841 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor PANOBINOSTAT PANOBINOSTAT 7159 4842 RACGAP1 29127 NA NSC-60339 CHEMBL1448793 7161 4843 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE BCNU CARMUSTINE 9219734 7164 4844 CD248 57124 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE OntecizumabAmatuximab 7165 4845 ACP3 55 ENZYME, DRUGGABLE GENOME MVA-BN 7167 4846 CTSC 1075 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 252166823 7168 4847 HAS3 3038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME HYDROCORTISONE HYDROCORTISONE 13130151 7169 4848 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Indole-based analog 2 7170 4849 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Onartuzumab ONARTUZUMAB 24101053,27918764,23882082 7171 4850 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor PX-866 SONOLISIB 7172 4851 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-327705 CHEMBL1317986 7173 4852 HSPA4 3308 NA PHOSPHODIESTERASE INHIBITOR 9383212 7175 4853 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MBX-102 ARHALOFENATE 7176 4854 USP1 7398 DNA REPAIR, PROTEASE, ENZYME L-745870 L-745870 7178 4855 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-21 7179 4856 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE DNDI1417099 CHEMBL1565444 7181 4857 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL1421 DASATINIB 7182 4858 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3545065 VEROSUDIL 7184 4859 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SCOULERINE SCOULERINE 7185 4860 PDGFC 56034 DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR inhibitor SUNITINIB SUNITINIB 7186 4861 NDUFAF3 25915 NA inhibitor CHEMBL3545320 ME-344 7188 4862 PTMA 5757 NA THYMALFASIN THYMALFASIN 7189 4863 PTGES 9536 DRUGGABLE GENOME, ENZYME Imidazole benzamide derivative 1 7190 4864 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 inhibitor 252827435 7191 4865 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 387065612 7192 4866 PPAT 5471 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1542 AZATHIOPRINE 7193 4867 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ETHANOL ALCOHOL 16930224 7194 4868 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist 249565879 SONIDEGIB 7195 4869 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135649957 ARPROMIDINE 7196 4870 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor PKI-587 GEDATOLISIB 7197 4871 TUBB2B 347733 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 7198 4872 GPR12 2835 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NEOCYCLOCITRINOL B NEOCYCLOCITRINOL B 18656987 7199 4873 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CAULIBUGULONE B CAULIBUGULONE B 7200 4874 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME DESMOSTEROL DESMOSTEROL 23910990 7202 4875 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ALPHA INTERFERON CETUXIMAB 8777337 7204 4876 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROGESTERONE PROGESTERONE 7205 4877 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PK11007 7206 4878 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR DS6051b 7207 4879 TUBA1A 7846 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 7210 4880 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Belotecan hydrocholoride 7211 4881 STING1 340061 CLINICALLY ACTIONABLE, KINASE agonist 381118902 ADU-S100 7212 4882 ACADSB 36 ENZYME VALPROIC ACID 7214 4883 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RESVERATROL RESVERATROL 7215 4884 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GFT14 7216 4885 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3039504 NINTEDANIB ESYLATE 7218 4886 HPN 3249 DRUGGABLE GENOME, PROTEASE, CELL SURFACE BENTIROMIDE BENTIROMIDE 7219 4887 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ESTRIOL ESTRIOL 7222 4888 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 2056784 CHEMBL261123 7223 4889 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-1644 CHEMBL600734 7224 4890 GRB2 2885 NA LIPOSOMAL GRB-2 7225 4891 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ACITRETIN ACITRETIN 7227 4892 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE PD-0166285 PD-0166285 7228 4893 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR Premarin/Pravachol 7231 4894 GALNS 2588 DRUGGABLE GENOME, ENZYME BMN-110 ELOSULFASE ALFA 7234 4895 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME CYC-116 CYC-116 7235 4896 TARDBP 23435 TUMOR SUPPRESSOR 3-PHENYLUMBELLIFERONE CHEMBL153505 7236 4897 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TOCILIZUMAB TOCILIZUMAB 7237 4898 PDE4A 5141 DRUGGABLE GENOME, ENZYME THEOPHYLLINE THEOPHYLLINE 7238 4899 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-720622 CHEMBL1287980 7239 4900 CYP27A1 1593 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 HORMONES 12597773 7242 4901 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649754 7243 4902 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 315661313 7244 4903 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Pyrazole derivative 66 7248 4904 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor 178103455 TOPIRAMATE 7249 4905 FCER1G 2207 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE R112 7250 4906 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PROPIDIUM PROPIDIUM 7252 4907 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SCLEROTIORIN SCLEROTIORIN 7254 4908 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PF-562271 PF-00562271 7255 4909 BRCA2 675 CLINICALLY ACTIONABLE Niraparib NIRAPARIB 27717299 7256 4910 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME ILORASERTIB ILORASERTIB 7257 4911 PRF1 5551 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME IL-2 ALDESLEUKIN 15893691 7259 4912 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME HGS1029 7261 4913 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102478 7262 4914 TUBB2B 347733 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 7264 4915 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651514 7265 4916 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103480 TASOSARTAN 7266 4917 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102315 RUXOLITINIB 7268 4918 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 223366184 7269 4919 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 20(S)-GINSENOSIDE RG3 CHEMBL398412 21956953 7273 4920 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417024 CHEMBL1462710 7275 4921 CASP4 837 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL197672 EMRICASAN 7276 4922 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AMO-02 7277 4923 CTSC 1075 ENZYME, DRUGGABLE GENOME, PROTEASE PROGESTERONE PROGESTERONE 17916955 7278 4924 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135650848 PRAVASTATIN 7280 4925 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL3545257 MIROGABALIN BESYLATE 7281 4926 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE ANGUSTIBALIN ANGUSTIBALIN 7282 4927 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR hydrochlorothiazide HYDROCHLOROTHIAZIDE 15864129,14553962,16109321 7283 4928 TK1 7083 ENZYME, KINASE, DRUGGABLE GENOME Ad-OC-hsvTK/valacyclovir 7284 4929 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SNA-120 PEGCANTRATINIB 7289 4930 BMPR1A 657 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 249565824 7291 4931 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Imatinib IMATINIB 7293 4932 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE GLUFOSFAMIDE GLUFOSFAMIDE 7294 4933 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-37642 CHEMBL1707907 7295 4934 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME rifampin RIFAMPIN 22562052,21709081,24420746,19374892 7297 4935 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME enflurane ENFLURANE 25989378,12411786,26951757,8828983,19919814,17710899,7829078,9334205,21965348,11063719,10823104,20681998,25611019,19648156,25256590,12220451,11668625,23736090,14500992,9066328,14641996,18945287,25960145,7889656,11575529,18212565,16284304,8602662,18306019,28326467,11928716,18502356,10352931,12151923,11525881,17122579,16917943,8220422,10700782,16163667,17226826,9389851,16732128,16835904,11448278,29101530,9450902,7547049,23628358,9543323,24361844,26994242,12208234,15448513,16621918,21455645,11553045,12124989,19020143,19191329,27918309,8220423,12059893,10612851,16732084,10793526,27382027,15108991,12709367,12123492,26381711,25268394,28063098,11493496,12434264,12411788,19685112,25735680,8902717,29608462,27663056,7751854,8012359,9520251,15731587,15210166,1510267,10888602,22030266,25466363,17483490,28403410,12237752,1774074,17081152,18564801,10484775,21282829,16244001,7586638,19191333,25086907,7633940,17667581,12883402,19346234,1354642,22415532 7298 4936 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TCMDC-125321 CHEMBL587449 7299 4937 PTGS2 5743 DRUGGABLE GENOME, ENZYME IBUPROFEN IBUPROFEN 7301 4938 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME TRIAZOLAM TRIAZOLAM 22137933 7302 4939 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BAY1125976 27699769 7305 4940 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2103873 MACITENTAN 7306 4941 GSTT1 2952 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 12851839 7308 4942 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE EVEROLIMUS EVEROLIMUS 7310 4943 HCN3 57657 DRUGGABLE GENOME, ION CHANNEL blocker 135650438 IVABRADINE 7312 4944 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME NV-52 7313 4945 APOE 348 DRUGGABLE GENOME LORAZEPAM LORAZEPAM 15699298 7314 4946 TUBB 203068 DRUGGABLE GENOME ZD-6126 ZD-6126 7315 4947 PSMD3 5709 NA inhibitor BORTEZOMIB BORTEZOMIB 7316 4948 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX PMID27336223-Compound-11 7317 4949 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR partial agonist CHEMBL2027925 CAPESEROD 7318 4950 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-117199 CHEMBL502257 7319 4951 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL371405 MARIZOMIB 7320 4952 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CISPLATIN CISPLATIN 31316618,29941343 7322 4953 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME INDOCATE INDOCATE 7323 4954 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME modulator CHEMBL2103824 ARHALOFENATE 7326 4955 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR ENOXAPARIN ENOXAPARIN 7327 4956 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102724 7329 4957 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-14 7330 4958 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME VORICONAZOLE VORICONAZOLE 19029318 7331 4959 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL1908371 IDRAPARINUX SODIUM 7332 4960 TUBA1A 7846 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 7333 4961 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KBP-5074 7338 4962 MAPT 4137 DRUGGABLE GENOME NORDEFRIN NORDEFRIN 7339 4963 RBBP9 10741 ENZYME, DRUGGABLE GENOME inhibitor 252166808 7341 4964 HTT 3064 DRUGGABLE GENOME SJ000120081 CHEMBL606532 7342 4965 GAA 2548 DRUGGABLE GENOME, ENZYME CID 667285 CHEMBL267160 7343 4966 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME CIMIRACEMATE A CIMIRACEMATE A 19835377 7344 4967 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BUTAMBEN BUTAMBEN 7345 4968 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Temozolomide TEMOZOLOMIDE 21730979 7346 4969 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PREGNENOLONE CARBONITRILE PREGNENOLONE CARBONITRILE 7347 4970 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PSB-1115 CHEMBL8565 7348 4971 ATAD5 79915 NA NILE RED NILE RED 7349 4972 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AMCINONIDE AMCINONIDE 7350 4973 POLI 11201 DNA REPAIR TAXIFOLIN TAXIFOLIN 7351 4974 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 178100554 7352 4975 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 7354 4976 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-156744 CHEMBL1481453 22524450 7356 4977 CYP24A1 1591 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME tenofovir disoproxil fumarate 31619748 7357 4978 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 363894214 SITRAVATINIB 7361 4979 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SB-220025 SB-220025 7362 4980 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201091 TERAZOSIN HYDROCHLORIDE HYDRATE 7363 4981 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (S)-FLUOXETINE CHEMBL1169388 7364 4982 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PROPYLTHIOURACIL PROPYLTHIOURACIL 22931300 7366 4983 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR DNDI1417548 CHEMBL2094789 7367 4984 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIHYDROSPINGOSINE DIHYDROSPINGOSINE 7368 4985 ALOX15 246 ENZYME, DRUGGABLE GENOME PHENOTHIAZINE PHENOTHIAZINE 7369 4986 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR VORINOSTAT VORINOSTAT 24694055,19344175,19966789,26211462,23622981,22260166,17447750,20491440,21548582,24074025,23672185,19084294 7374 4987 LTF 4057 CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, PROTEASE HLF 1-11 7375 4988 DHFR 1719 DRUGGABLE GENOME, ENZYME pemetrexed PEMETREXED 24732178,23709418 7376 4989 ARRB2 409 ION CHANNEL, G PROTEIN COUPLED RECEPTOR fentanyl FENTANYL 30549211 7379 4990 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PHENYLBUTYRYLHYDROXAMIC ACID PHENYLBUTYRYLHYDROXAMIC ACID 21874153 7381 4991 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BROMEBRIC ACID BROMEBRIC ACID 7383 4992 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200440 MEPIVACAINE HYDROCHLORIDE 7384 4993 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME INCB054828 PEMIGATINIB 7385 4994 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Olaratumab OLARATUMAB 7386 4995 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR INDOCYANINE GREEN SODIUM INDOCYANINE GREEN 7387 4996 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL538943 VINORELBINE TARTRATE 7388 4997 KDM4A 9682 DRUGGABLE GENOME, ENZYME PRALIDOXIME IODIDE PRALIDOXIME IODIDE 7389 4998 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME ALISERTIB SODIUM 7392 4999 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Ocrelizumab OCRELIZUMAB 7393 5000 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW785804X GW785804X 7395 5001 PSMC1 5700 PROTEASE inhibitor CHEMBL3545432 IXAZOMIB CITRATE 7396 5002 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE ALLYL ISOTHIOCYANATE ALLYL ISOTHIOCYANATE 26338358 7398 5003 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417759 CHEMBL1446254 7399 5004 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor CHEMBL1084546 PF-00562271 7400 5005 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102239 TONAPOFYLLINE 7401 5006 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ROTENONE ROTENONE 7402 5007 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME SJ000150791 CHEMBL600572 7403 5008 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-83217 CHEMBL120806 7404 5009 POLD1 5424 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME inhibitor CHEMBL1637 GEMCITABINE HYDROCHLORIDE 7405 5010 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BI 655064 7406 5011 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-228155 CHEMBL505670 7407 5012 TARDBP 23435 TUMOR SUPPRESSOR CEPHALOCHROMIN CEPHALOCHROMIN 7408 5013 PSMD2 5708 NA BORTEZOMIB BORTEZOMIB 7411 5014 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE PROTEASOME INHIBITOR 16186809 7412 5015 PTBP1 5725 DRUGGABLE GENOME MMV085203 CHEMBL586031 7413 5016 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor 223366040 7414 5017 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor GSK2636771 GSK-2636771 7415 5018 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL1094636 NIRAPARIB 7416 5019 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PANOBINOSTAT PANOBINOSTAT 7423 5020 TMSB10 9168 NA RETINOIDS 2059565,2169566,1846397,1315216 7424 5021 BRCA2 675 CLINICALLY ACTIONABLE Etoposide ETOPOSIDE 26116172 7426 5022 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR XL844 7427 5023 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE NADOLOL NADOLOL 1681747 7428 5024 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102733 7429 5025 TAC1 6863 DRUGGABLE GENOME GINGER GINGER 1282221 7430 5026 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BENZQUINAMIDE BENZQUINAMIDE 7431 5027 ATAT1 79969 ENZYME gemcitabine GEMCITABINE 31616045 7433 5028 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE N/A 19047294,26586702,16109776,26676635,26239249,25281355,24573385,25713434 7434 5029 SHMT1 6470 ENZYME fluorouracil FLUOROURACIL 22044939 7435 5030 GMNN 51053 DRUGGABLE GENOME DNDI1416924 CHEMBL156959 7436 5031 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NITROXOLINE NITROXOLINE 7437 5032 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME KENPAULLONE KENPAULLONE 7438 5033 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Antiinflammatory agents, non-steroids 28750137 7440 5034 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME METHYLENE BLUE METHYLENE BLUE 7444 5035 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL Mirogabalin MIROGABALIN 7445 5036 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME CAR-T cells targeting Mesothelin 7449 5037 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CLORAZEPATE CLORAZEPIC ACID 7450 5038 SGPL1 8879 ENZYME, DRUGGABLE GENOME inhibitor 252166675 7451 5039 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Cyclopropyl-spiro piperidine derivative 3 7452 5040 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME Curcumin CURCUMIN 7454 5041 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME PEPSTATIN PEPSTATIN 7455 5042 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHENOXYBENZAMINE PHENOXYBENZAMINE 22931300 7456 5043 MAP3K1 4214 CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME cisplatin CISPLATIN 21636554 7459 5044 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650120 7460 5045 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE GS-9820 ACALISIB 7461 5046 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BENZQUINAMIDE BENZQUINAMIDE 7462 5047 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME blocker 135651426 ADENOSINE 7464 5048 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DEBRISOQUIN DEBRISOQUIN 7465 5049 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MMV007764 CHEMBL609628 7466 5050 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TC-A2317 22293494 7467 5051 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE OUABAIN OUABAIN 7468 5052 ERAP1 51752 PROTEASE, ENZYME, DRUGGABLE GENOME TCMDC-124377 CHEMBL531269 7469 5053 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Pyrimidinyl compound 6 7471 5054 FAM178B 51252 NA lithium LITHIUM 29121268 7472 5055 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE S-222611 S-222611 7473 5056 HTT 3064 DRUGGABLE GENOME KENPAULLONE KENPAULLONE 7475 5057 GMNN 51053 DRUGGABLE GENOME TRICLABENDAZOLE TRICLABENDAZOLE 7476 5058 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME E-6700 7477 5059 MPHOSPH8 54737 NA MORIN MORIN 7478 5060 SRI 6717 NA ADM 2568983 7479 5061 MAZ 4150 TRANSCRIPTION FACTOR IL-1 11809795 7481 5062 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE TGR-1202 UMBRALISIB TOSYLATE 7482 5063 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR GDC-0973 COBIMETINIB 7484 5064 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Tosagestin TOSAGESTIN 7485 5065 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DOCEBENONE DOCEBENONE 7487 5066 BAZ2B 29994 NA GALLIC ACID METHYL ESTER GALLIC ACID METHYL ESTER 7489 5067 DGAT1 8694 ENZYME, DRUGGABLE GENOME Pyrazolo[1,5-a]pyrimidine derivative 28 7493 5068 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME (RS)-ROSCOVITINE (RS)-ROSCOVITINE 7494 5069 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PMID29671355-Compound-25 7495 5070 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZOLPIDEM ZOLPIDEM 7496 5071 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR SOBETIROME SOBETIROME 7497 5072 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING PATULIN PATULIN 16680159 7498 5073 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE ASPIRIN ASPIRIN 10921413 7499 5074 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR HE3286 HE3286 7500 5075 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR Erteberel ERTEBEREL 7501 5076 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-172033 CHEMBL238624 7502 5077 BAZ2B 29994 NA ROSMARINIC ACID ROSMARINIC ACID 7507 5078 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-20 7508 5079 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE OSI-632 OSI-632 7509 5080 POLI 11201 DNA REPAIR SCOULERINE SCOULERINE 7511 5081 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 178102906 SITAGLIPTIN 7512 5082 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE ALBUMIN ALBUMIN HUMAN 11531629 7513 5083 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201496 INSULIN ASPART 7514 5084 SLCO2A1 6578 TRANSPORTER, DRUGGABLE GENOME Thiazides, plain 28783044 7515 5085 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE TAK-659 TAK-659 7516 5086 CCN1 3491 DRUGGABLE GENOME ANTISENSE OLIGONUCLEOTIDES 18381294 7517 5087 TFF2 7032 DRUGGABLE GENOME VT-111a 21683260 7518 5088 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100426 7519 5089 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIGITOXIN DIGITOXIN 7522 5090 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE ENTRECTINIB ENTRECTINIB 7523 5091 EIF4H 7458 DRUGGABLE GENOME GNF-PF-4618 CHEMBL585964 7524 5092 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 (S)-NITRENDIPINE (S)-NITRENDIPINE 7525 5093 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME 1,2-dihydroindazolo[4,3-bc][1,5]benzoxazepine derivative 1 7526 5094 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PROPOXYCAINE PROPOXYCAINE 7527 5095 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE NSC-728558 CHEMBL457246 19167892 7528 5096 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL415049 BARASERTIB 7530 5097 PIGM 93183 NA methylphenidate METHYLPHENIDATE 29382897 7532 5098 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR LETROZOLE LETROZOLE 26715889 7535 5099 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME RG-1530 RG-1530 7537 5100 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME nilotinib NILOTINIB 7538 5101 IL1A 3552 CELL SURFACE, DRUGGABLE GENOME Xilonix BERMEKIMAB 7540 5102 ABCG8 64241 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER atorvastatin ATORVASTATIN 16103896,15262185,20592455 7542 5103 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME VITAMIN E 2035236 7543 5104 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Alpelisib ALPELISIB 7546 5105 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 7547 5106 KAT2B 8850 ENZYME, DRUGGABLE GENOME DIETHYL-2-DODECYLIDENEMALONATE CHEMBL1797708 21292492 7548 5107 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRIOL ESTRIOL 7549 5108 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE AZD5363 CAPIVASERTIB 26116361,19755509,24088382,22294718 7552 5109 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Bendamustine BENDAMUSTINE 20739657 7555 5110 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE BUTORPHANOL BUTORPHANOL 7556 5111 CYP4B1 1580 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME docetaxel DOCETAXEL 20038957 7557 5112 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PALMITOYL-DL-CARNITINE CHLORIDE CHEMBL1256761 7558 5113 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PYRITHIONE ZINC PYRITHIONE ZINC 7559 5114 HTT 3064 DRUGGABLE GENOME MITOXANTRONE MITOXANTRONE 7562 5115 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BETAMETHASONE BETAMETHASONE 7563 5116 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE DIMETHYLCURCUMIN DIMETHYLCURCUMIN 25753330 7564 5117 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Cycloalkyl nitrile pyrazolo pyridone derivative 1 7565 5118 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme12-3 7566 5119 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE apixaban APIXABAN 28678049,29457840 7567 5120 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME RVX-208 APABETALONE 7568 5121 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 vemurafenib VEMURAFENIB 23116250 7572 5122 PSMD6 9861 NA inhibitor CHEMBL451887 CARFILZOMIB 7573 5123 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SORAFENIB SORAFENIB 7574 5124 GMNN 51053 DRUGGABLE GENOME BROMHEXINE HYDROCHLORIDE BROMHEXINE HYDROCHLORIDE 7577 5125 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE NINTEDANIB NINTEDANIB 7578 5126 AKR1C3 8644 ENZYME, DRUGGABLE GENOME INDOMETHACIN INDOMETHACIN 23432095 7579 5127 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL TRIAZOLAM TRIAZOLAM 7582 5128 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Famitinib FAMITINIB 7583 5129 SMN2 6607 DRUGGABLE GENOME DNDI1417031 CHEMBL1333049 7584 5130 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 135651472 DIETHYLSTILBESTROL 7586 5131 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL2109047 INTERFERON ALFA-N3 7587 5132 GSTM1 2944 DRUGGABLE GENOME, ENZYME CAROTENOID 15095308 7588 5133 EYA2 2139 DNA REPAIR SJ000018309 CHEMBL591363 7589 5134 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER OLEAMIDE OLEAMIDE 7590 5135 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR ENALAPRIL ENALAPRIL 18812665 7592 5136 FAAH 2166 ENZYME, DRUGGABLE GENOME Piperazine urea derivative 1 7593 5137 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PMID27336223-Compound-7 7595 5138 USP1 7398 DNA REPAIR, PROTEASE, ENZYME BUNAMIDINE BUNAMIDINE 7596 5139 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR LY2127399 7599 5140 BAZ2B 29994 NA 3,3'-DIMETHOXYBENZIDINE CHEMBL398363 7600 5141 POLI 11201 DNA REPAIR S(+)-ISOPROTERENOL-BITARTRATE CHEMBL1257092 7601 5142 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR US9714230, 46 7602 5143 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE imatinib IMATINIB 30237583 7603 5144 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CINOLAZEPAM CINOLAZEPAM 7605 5145 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Pyrazolopyrimidine and thienopyrimidine amide derivative 1 7607 5146 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 315661099 7608 5147 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 252166579 TACEDINALINE 7609 5148 PTGS1 5742 ENZYME, DRUGGABLE GENOME diclofenac sodium patch 7612 5149 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE agonist CHEMBL2107846 DULANERMIN 7614 5150 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 310264764 7615 5151 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL1201748 CABAZITAXEL 7616 5152 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER nortriptyline NORTRIPTYLINE 12082591 7617 5153 COMT 1312 DRUGGABLE GENOME, ENZYME ENTACAPONE ENTACAPONE 7618 5154 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135651045 SIMVASTATIN 7620 5155 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TEMSIROLIMUS TEMSIROLIMUS 7621 5156 PCSK7 9159 ENZYME, PROTEASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 252166868 7624 5157 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME TRICHOSTATIN TRICHOSTATIN 21055848,16921367,19966789,19385600 7625 5158 RRM2 6241 DRUGGABLE GENOME, ENZYME GEMCITABINE GEMCITABINE 7627 5159 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Laquinimod LAQUINIMOD 7628 5160 POLK 51426 DNA REPAIR, ENZYME OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 7629 5161 DPP9 91039 PROTEASE, ENZYME, DRUGGABLE GENOME Thiomorpholine derivative 2 7630 5162 GUCY1A1 2982 ENZYME, DRUGGABLE GENOME activator CHEMBL730 NITROGLYCERIN 7631 5163 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GDC-0980 APITOLISIB 26951309,26787751,21998291 7632 5164 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME GISENOSIDE RK1 GISENOSIDE RK1 26420067 7633 5165 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CLOTIAZEPAM CLOTIAZEPAM 7634 5166 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE PMID26394986-Compound-10 7636 5167 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME LY-2624803 LY2624803 7637 5168 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GNF-PF-2301 CHEMBL578061 7639 5169 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME BUTYRYLHYDROXAMIC ACID BUTYRYLHYDROXAMIC ACID 21874153 7640 5170 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 310264705 PITOLISANT 7642 5171 NECTIN4 81607 DRUGGABLE GENOME antibody 405067331 7643 5172 AIFM1 9131 DRUGGABLE GENOME HSP70 12022952 7644 5173 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 7645 5174 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Metformin METFORMIN 26921394,24077915 7647 5175 CA5A 763 ENZYME, DRUGGABLE GENOME activator 178101506 AMPHETAMINE 7651 5176 CA9 768 DRUGGABLE GENOME, ENZYME CHEMBL3707297 CG250 177LU 7653 5177 TLE3 7090 TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR DOCETAXEL DOCETAXEL 7656 5178 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL517712 ATROPINE 7657 5179 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BKM120 BUPARLISIB 28108151 7658 5180 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GDC-0032 TASELISIB 26589432 7659 5181 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR GIVINOSTAT GIVINOSTAT 7660 5182 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 348353623 7664 5183 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME LINAGLIPTON 7665 5184 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GIPARMEN GIPARMEN 7666 5185 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME SNS-314 SNS-314 7667 5186 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRICLABENDAZOLE TRICLABENDAZOLE 7668 5187 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME LASSBIO-123 CHEMBL573111 7670 5188 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME GOSSYPOL GOSSYPOL 7672 5189 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE imatinib IMATINIB 11526490 7673 5190 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 12548406 7674 5191 CD37 951 DRUGGABLE GENOME Otlertuzumab OTLERTUZUMAB 7675 5192 DNER 92737 NA Dihydropyrido pyrazinone compound 1 7676 5193 MAPT 4137 DRUGGABLE GENOME ZK-93423 CHEMBL1518572 7677 5194 GABPA 2551 TRANSCRIPTION FACTOR QUERCETIN QUERCETIN 17462537 7678 5195 UBA2 10054 DRUGGABLE GENOME, ENZYME LOBARIC ACID LOBARIC ACID 7679 5196 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CYC-116 CYC-116 7680 5197 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PERPHENAZINE PERPHENAZINE 7681 5198 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE DACOMITINIB DACOMITINIB 23930994 7683 5199 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565642 RALIMETINIB 7684 5200 NQO2 4835 DRUGGABLE GENOME, ENZYME NSC-640559 CHEMBL1287866 21074425 7685 5201 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRICLOFENOL TRICLOFENOL 7686 5202 NOS2 4843 DRUGGABLE GENOME, ENZYME BENZODIAZEPINE BENZODIAZEPINE 12106778 7688 5203 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SAR153191 7689 5204 SMN1 6606 DRUGGABLE GENOME CID 5310655 CHEMBL408563 7690 5205 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TAE-684 TAE-684 7691 5206 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUNISOLIDE FLUNISOLIDE 7692 5207 HEBP1 50865 DRUGGABLE GENOME Pyrazino[2,1-a]isoquinolin derivative 2 7693 5208 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2-MERCAPTOBENZIMIDAZOLE 2-MERCAPTOBENZIMIDAZOLE 7696 5209 RPS6KA4 8986 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 7698 5210 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR allosteric modulator 405560349 7700 5211 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GSK0660 CHEMBL592652 22369181 7702 5212 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE 6,4'-DIHYDROXYFLAVONE CHEMBL484663 7703 5213 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125653 CHEMBL580918 7704 5214 MYO9B 4650 NA STREPTOZOTOCIN STREPTOZOCIN 2523196 7705 5215 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER granisetron GRANISETRON 29177570,27241063 7707 5216 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL289351 FOSBRETABULIN DISODIUM 7709 5217 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME INDIGO INDIGO 7711 5218 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME PPD 11468004 7712 5219 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME FOLIC ACID 15047700 7715 5220 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor HESPERADIN HESPERADIN 19035792 7716 5221 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CRYPTOTANSHINONE CRYPTOTANSHINONE 7717 5222 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651375 7718 5223 ATXN2 6311 NA GEDUNIN GEDUNIN 7719 5224 DHRS9 10170 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE (+)-ISOZONARONE CHEMBL459574 19188072 7721 5225 CBX1 10951 NA TCMDC-125544 CHEMBL533602 7722 5226 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL Dantrolene DANTROLENE 7723 5227 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-70 7725 5228 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE inhibitor 249565620 DANUSERTIB 7726 5229 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME NSC-92207 CHEMBL139935 7727 5230 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker 135650617 DIZOCILPINE 7728 5231 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL378544 VINBLASTINE SULFATE 7729 5232 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR HYPERICIN HYPERICIN 7734 5233 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE AZAKENPAULLONE AZAKENPAULLONE 7735 5234 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOREMIFENE CITRATE TOREMIFENE CITRATE 7736 5235 MAP3K1 4214 CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME gefitinib GEFITINIB 21636554 7738 5236 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME MEK162 BINIMETINIB 26577700 7739 5237 TXNDC11 51061 DRUGGABLE GENOME, THIOREDOXIN hydrochlorothiazide HYDROCHLOROTHIAZIDE 7740 5238 KDM4A 9682 DRUGGABLE GENOME, ENZYME CARMINIC ACID CARMINIC ACID 7741 5239 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist CHEMBL2103864 NAVARIXIN 7742 5240 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME TAE-684 TAE-684 7743 5241 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME M-carboxycinnamic acid bishydroxamide 7746 5242 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL3545272 LAS190792 7748 5243 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3545092 CR 1447 7749 5244 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Radiotherapy 26589432 7750 5245 GAA 2548 DRUGGABLE GENOME, ENZYME TCMDC-124544 CHEMBL531322 7751 5246 SMARCA2 6595 NA GNF-PF-3736 CHEMBL583824 7752 5247 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102599 7753 5248 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME EVEROLIMUS EVEROLIMUS 24625776,24622468 7754 5249 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX KENPAULLONE KENPAULLONE 7756 5250 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR COUMESTROL COUMESTROL 7757 5251 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NU6027 21730979 7758 5252 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor 404859010 7759 5253 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHINIOFON CHINIOFON 7760 5254 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Fluvoxamine FLUVOXAMINE 7761 5255 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE meperidine MEPERIDINE 18695978 7762 5256 GMNN 51053 DRUGGABLE GENOME NSC-145669 CHEMBL191611 7763 5257 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650558 LY-510929 7765 5258 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 7766 5259 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 7767 5260 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL2062276 LEVALLORPHAN TARTRATE 7770 5261 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BETULINIC ACID BETULINIC ACID 19716700 7771 5262 RACGAP1 29127 NA NSC-645827 CHEMBL95704 7773 5263 TFF2 7032 DRUGGABLE GENOME Nafamostat NAFAMOSTAT 7774 5264 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR RHEIN RHEIN 7775 5265 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 310264782 7776 5266 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE pegloticase PEGLOTICASE 26906307,25224415 7778 5267 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE agonist 178100830 SUXAMETHONIUM 7779 5268 CBX1 10951 NA NSC-9037 CHEMBL1451216 7782 5269 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 178102666 7783 5270 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME FEXOFENADINE FEXOFENADINE 7784 5271 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MEPANIPYRIM MEPANIPYRIM 7785 5272 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ALSTERPAULLONE ALSTERPAULLONE 7786 5273 ADCY6 112 ENZYME, KINASE, DRUGGABLE GENOME inhibitor 178101917 7787 5274 PSMA8 143471 DRUGGABLE GENOME, PROTEASE inhibitor BORTEZOMIB BORTEZOMIB 7794 5275 APBB1 322 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING G-207 virus construct 7795 5276 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE activator 375973253 7797 5277 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRICIFEROL TRICIFEROL 20452225 7800 5278 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME GNF-PF-3023 CHEMBL535331 7801 5279 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Isoindoline derivative 1 7803 5280 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE UO126 28215740 7804 5281 AREG 374 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE capecitabine CAPECITABINE 25026457 7805 5282 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHIR-99021 CHIR-99021 7806 5283 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-46 7807 5284 GMNN 51053 DRUGGABLE GENOME FLUNARIZINE FLUNARIZINE 7808 5285 POLK 51426 DNA REPAIR, ENZYME RHAMNETIN RHAMNETIN 7809 5286 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CYC-116 CYC-116 7811 5287 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100615 7812 5288 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ECONAZOLE NITRATE ECONAZOLE NITRATE 7813 5289 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE ALTEPLASE ALTEPLASE 7815 5290 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor MOTESANIB MOTESANIB 7816 5291 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME L-655240 CHEMBL362223 7817 5292 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME IMATINIB IMATINIB 18971950 7818 5293 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 381118861 7819 5294 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE POLYPHENOL 15324350 7820 5295 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-25 7821 5296 HP 3240 DRUGGABLE GENOME, PROTEASE, ENZYME HEPATITIS B VACCINE 8256500 7822 5297 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-4029 CHEMBL596633 7824 5298 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DAB 8185829 7827 5299 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE SURAMIN SURAMIN 7829 5300 ALOX15 246 ENZYME, DRUGGABLE GENOME FISETIN FISETIN 17869117 7830 5301 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SCARLET RED SCARLET RED 7831 5302 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1256958 EPINEPHRINE BITARTRATE 7833 5303 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE TELATINIB TELATINIB 7834 5304 CYB5R2 51700 DRUGGABLE GENOME metoclopramide METOCLOPRAMIDE 7835 5305 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER 4-((2-PHENETHYLPHENOXY)METHYL)PYRIDINE CHEMBL270688 18257545 7837 5306 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Parthenolide PARTHENOLIDE 7838 5307 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-640566 CHEMBL1287867 21074425 7839 5308 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor BGJ398 INFIGRATINIB 7840 5309 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-39 7842 5310 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME DHEA PRASTERONE 9177459 7843 5311 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor DOVITINIB DOVITINIB 7844 5312 TJP1 7082 KINASE, TRANSCRIPTION FACTOR risperidone RISPERIDONE 7845 5313 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE JNJ 38877605 23729478 7846 5314 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME simvastatin SIMVASTATIN 7847 5315 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL1742994 BRENTUXIMAB VEDOTIN 7848 5316 DIABLO 56616 NA CEPHALOSTATIN 14695204 7850 5317 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000113107 CHEMBL589245 7851 5318 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GLUCOCORTICOID 9275052 7852 5319 EML4 27436 CLINICALLY ACTIONABLE, KINASE TAE226 26090892 7853 5320 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR SELENIUM 16036356 7858 5321 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Carmoterol CARMOTEROL 7859 5322 HTT 3064 DRUGGABLE GENOME Ampicidin analog 1 7860 5323 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OXYBUTYNIN OXYBUTYNIN 7861 5324 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2013009582Example76 7862 5325 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor CHEMBL574737 UCN-01 7863 5326 MAOB 4129 DRUGGABLE GENOME, ENZYME P2B-001 7865 5327 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CHEMBL2068724 ACAMPROSATE CALCIUM 7867 5328 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BERAPROST BERAPROST 7868 5329 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME GEMFIBROZIL GEMFIBROZIL 16316932 7870 5330 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CODEINE CODEINE 7871 5331 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 7874 5332 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE cisplatin CISPLATIN 22901187 7876 5333 MAPT 4137 DRUGGABLE GENOME DOCEBENONE DOCEBENONE 7877 5334 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR isoproterenol ISOPROTERENOL 7878 5335 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-2357 CHEMBL578257 7879 5336 SMN2 6607 DRUGGABLE GENOME NICLOSAMIDE NICLOSAMIDE 7880 5337 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME ARRY-382 ARRY-382 7885 5338 NDUFB4 4710 ENZYME inhibitor CHEMBL3545320 ME-344 7886 5339 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE PREDNISONE PREDNISONE 17063711 7887 5340 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Indoline derivative 3 7888 5341 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor SORAFENIB SORAFENIB 7889 5342 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TAK-715 TAK-715 7890 5343 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL Amlodipine AMLODIPINE 7891 5344 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER IGF-1R antibody 27196767 7893 5345 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor RO5212054 7894 5346 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHENANTHROLINE PHENANTHROLINE 7898 5347 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VESNARINONE VESNARINONE 9226479 7901 5348 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME desflurane DESFLURANE 25989378,12411786,26951757,8828983,19919814,17710899,7829078,9334205,21965348,11063719,10823104,20681998,25611019,19648156,25256590,12220451,11668625,23736090,14500992,9066328,14641996,18945287,25960145,7889656,11575529,18212565,16284304,8602662,18306019,28326467,11928716,18502356,10352931,12151923,11525881,17122579,16917943,8220422,10700782,16163667,17226826,9389851,16732128,16835904,11448278,29101530,9450902,7547049,23628358,9543323,24361844,26994242,12208234,15448513,16621918,21455645,11553045,12124989,19020143,19191329,27918309,8220423,12059893,10612851,16732084,10793526,27382027,15108991,12709367,12123492,26381711,25268394,28063098,11493496,12434264,12411788,19685112,25735680,8902717,29608462,27663056,7751854,8012359,9520251,15731587,15210166,1510267,10888602,22030266,25466363,17483490,28403410,12237752,1774074,17081152,18564801,10484775,21282829,16244001,7586638,19191333,25086907,7633940,17667581,12883402,19346234,1354642,22415532 7902 5349 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Trametinib TRAMETINIB 27338794 7904 5350 COMT 1312 DRUGGABLE GENOME, ENZYME Entacapone ENTACAPONE 7905 5351 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY ANTIDEPRESSANT 10889291 7907 5352 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR METHOTREXATE METHOTREXATE 7908 5353 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 178103523 OBINUTUZUMAB 7909 5354 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Alitretinoin ALITRETINOIN 7910 5355 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GSK369796 GSK-369796 19222165 7911 5356 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1766582 R-1487 7912 5357 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PF-03715455 PF-03715455 21888439 7913 5358 BAZ2B 29994 NA DITHIAZANINE IODIDE DITHIAZANINE IODIDE 7916 5359 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ALPROSTADIL ALPROSTADIL 22931300 7917 5360 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME PL37 7919 5361 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR GSK2126458 OMIPALISIB 22389471 7920 5362 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TRANSTORINE TRANSTORINE 7921 5363 ALPL 249 ENZYME, DRUGGABLE GENOME NSC-353720 CHEMBL1408276 7922 5364 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE BLU-285 AVAPRITINIB 7924 5365 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 7925 5366 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor MOTESANIB MOTESANIB 7926 5367 MGLL 11343 DRUGGABLE GENOME, ENZYME Pyrazole derivative 81 7927 5368 POLA1 5422 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, DNA REPAIR BROMOVINYL DEOXYURIDINE 7928 5369 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME MUSTARD 15102853 7929 5370 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ZIPRASIDONE ZIPRASIDONE 7930 5371 SERPING1 710 DRUGGABLE GENOME, PROTEASE INHIBITOR Rhucin RHUCIN 7931 5372 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 348353620 7932 5373 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME METHYLENE BLUE CHLORIDE HYDRATE METHYLENE BLUE 7933 5374 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR QUERCETAGETIN QUERCETAGETIN 25190466 7934 5375 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR FLUTAMIDE FLUTAMIDE 7935 5376 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 178102082 ADAPALENE 7936 5377 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME ANACARDIC ACID 18215015 7938 5378 MGLL 11343 DRUGGABLE GENOME, ENZYME Azetidinyl-piperidine derivative 1 7941 5379 GBP6 163351 NA Tumor necrosis factor alpha (TNF-alpha) inhibitors 7942 5380 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE D-DOPA CHEMBL211670 7943 5381 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor BMS-754807 BMS-754807 7944 5382 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 5,7-DIHYDROXY-4-METHYLCOUMARIN 5,7-DIHYDROXY-4-METHYLCOUMARIN 7945 5383 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL1421 DASATINIB 7946 5384 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Hirudin 7948 5385 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE ALISERTIB ALISERTIB 7949 5386 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IMIPRAMINE IMIPRAMINE 22931300 7950 5387 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Poziotinib POZIOTINIB 7951 5388 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL260933 GS 6201 7952 5389 CREB1 1385 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR citalopram CITALOPRAM 20643483,17548750 7953 5390 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE GW459057A GW459057A 16890436 7954 5391 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27551786-Compound-II 7956 5392 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PATULIN PATULIN 7957 5393 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-102742 CHEMBL1519374 7958 5394 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE COLFORSIN COLFORSIN 7959 5395 PARP3 10039 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR inhibitor CHEMBL506871 VELIPARIB 7960 5396 UGT2B7 7364 DRUGGABLE GENOME oxycodone OXYCODONE 29502154 7961 5397 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME PMID27774822-Compound-Figure3CompoundI-165 7962 5398 APOA2 336 DRUGGABLE GENOME RETINOIDS 7918317 7965 5399 TMEM97 27346 NA Benzamide derivative 9 7968 5400 PDE7B 27115 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL628 PENTOXIFYLLINE 7969 5401 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DNDI1417331 CHEMBL1092508 7972 5402 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 404859078 7973 5403 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565691 CHEMBL1086377 7974 5404 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR OLEIC ACID OLEIC ACID 7975 5405 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651150 7976 5406 WDR5 11091 DRUGGABLE GENOME, TUMOR SUPPRESSOR antagonist 249565911 7977 5407 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL495727 AT-9283 7978 5408 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-CROs 7980 5409 TARDBP 23435 TUMOR SUPPRESSOR TCMDC-124425 CHEMBL548681 7981 5410 ALOX5 240 DRUGGABLE GENOME, ENZYME ZILEUTON ZILEUTON 7982 5411 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-130 7983 5412 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR LAUROGUADINE LAUROGUADINE 7984 5413 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OLANZAPINE OLANZAPINE 7985 5414 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DESOXIMETASONE DESOXIMETASONE 7986 5415 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102259 7987 5416 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE NIVOLUMAB NIVOLUMAB 31086949 7988 5417 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Thiadiazolyl carboxamide derivative 1 7989 5418 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE TRIAMTERENE TRIAMTERENE 7991 5419 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PALMITIC ACID PALMITIC ACID 7994 5420 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR CIPROFIBRATE CIPROFIBRATE 7995 5421 TUBB3 10381 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 7996 5422 TNFSF10 8743 DRUGGABLE GENOME Ad5-TRAIL 7998 5423 POLK 51426 DNA REPAIR, ENZYME DEMECLOCYCLINE HYDROCHLORIDE DEMECLOCYCLINE HYDROCHLORIDE 8000 5424 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102257 8002 5425 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor 178101942 8007 5426 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME LAK 3489774 8008 5427 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 8009 5428 POLI 11201 DNA REPAIR NSC-22225 CHEMBL462314 8010 5429 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DOMPERIDONE DOMPERIDONE 8011 5430 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178102559 NINTEDANIB 8012 5431 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125140 CHEMBL525106 8013 5432 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme18 8014 5433 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE XL281 8015 5434 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE allosteric modulator 328083529 MIRANSERTIB 8016 5435 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor SOPHORETIN QUERCETIN 8017 5436 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE ALTEPLASE ALTEPLASE 8018 5437 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Galnobax 8019 5438 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102307 ALVOCIDIB 8020 5439 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 223365981 FALNIDAMOL 8022 5440 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE AZD3463 27009859 8023 5441 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW780056X GW780056X 8025 5442 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME BELINOSTAT BELINOSTAT 8026 5443 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Trametinib TRAMETINIB 26343583,27659046,25665005,26324075,26882569,26582713,27338794,27222538,27556948,22805291,27312529,27876675,26369631,28179366 8029 5444 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL2109406 PATRITUMAB 8032 5445 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE GALETERONE GALETERONE 8033 5446 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Rubitecan RUBITECAN 8035 5447 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME ODANACATIB ODANACATIB 8036 5448 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL1569 AMANTADINE HYDROCHLORIDE 8038 5449 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ROLIPRAM ROLIPRAM 19464886 8039 5450 AKR1C1 1645 DRUGGABLE GENOME, ENZYME 2-(4-CHLOROBENZYLIDENE)CYCLOPENTANONE CHEMBL562352 19237229 8040 5451 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3360203 PILARALISIB 8041 5452 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE HEPARAN SULFATE 12972284 8042 5453 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CATECHIN CATECHIN 8045 5454 BRCA2 675 CLINICALLY ACTIONABLE KU-0063794 26546619 8046 5455 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR MF-101 MF101 8047 5456 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE VINBLASTINE SULFATE VINBLASTINE SULFATE 8048 5457 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor CHEMBL1695 TIAGABINE HYDROCHLORIDE 8049 5458 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-158389 CHEMBL192626 8050 5459 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1722209 TOLTERODINE TARTRATE 8051 5460 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE MER-5101 8052 5461 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PIRIBEDIL PIRIBEDIL 8054 5462 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PRAVASTATIN PRAVASTATIN 15842807 8055 5463 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME verubecestat VERUBECESTAT 8056 5464 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL482968 ENMD-2076 8057 5465 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW795493X GW795493X 8058 5466 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102998 DABIGATRAN 8061 5467 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PROSTAGLANDIN E1 7492761 8062 5468 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME CENISERTIB CENISERTIB 8063 5469 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME LY-2090314 LY-2090314 8066 5470 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 dolasetron DOLASETRON 9187528 8067 5471 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR ALL-TRANS-RETINOIC ACID 11927016 8069 5472 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650183 DIHYDROMORPHINE 8070 5473 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CHLORANIL CHLORANIL 8072 5474 FCGR2A 2212 CLINICALLY ACTIONABLE, DRUGGABLE GENOME infliximab INFLIXIMAB 25823785,24667440,24048425,27044681 8074 5475 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Quinoline derivative 10 8075 5476 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRIAMTERENE TRIAMTERENE 8076 5477 TXNRD1 7296 DRUGGABLE GENOME inhibitor CHEMBL1200978 ARSENIC TRIOXIDE 8078 5478 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE SULFASALAZINE SULFASALAZINE 8079 5479 APC 324 CLINICALLY ACTIONABLE Ibuprofen IBUPROFEN 17909047 8080 5480 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR GNF-PF-4371 CHEMBL585651 8081 5481 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Thiomorpholine derivative 2 8082 5482 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE mycophenolic acid 25163792,28624888 8083 5483 P4HB 5034 THIOREDOXIN, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 8084 5484 CACNB3 784 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ION CHANNEL VERAPAMIL VERAPAMIL 8085 5485 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-O1 8086 5486 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PD-98059 CHEMBL35482 15930183 8087 5487 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME EMODIN EMODIN 8088 5488 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR IMIDOCARB DIPROPIONATE IMIDOCARB DIPROPIONATE 8090 5489 KDM4A 9682 DRUGGABLE GENOME, ENZYME MESO-2,3-DIMERCAPTOSUCCINIC ACID CHEMBL28721 8092 5490 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 8093 5491 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR TRICIRIBINE TRICIRIBINE 8096 5492 CD8A 925 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE Protein vaccines 8097 5493 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PLX8394 PLX8394 8098 5494 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME SJ000202381 CHEMBL591598 8099 5495 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NAPHTHYLAMINE NAPHTHYLAMINE 8100 5496 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL1852688 INFIGRATINIB 8101 5497 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Desoxypeganine 8104 5498 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651386 8105 5499 HTT 3064 DRUGGABLE GENOME KAMEBANIN KAMEBANIN 8106 5500 CDH1 999 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Volasertib VOLASERTIB 26597303 8107 5501 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 9 8109 5502 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545335 AG-13958 8110 5503 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme9EHT1610 8113 5504 LIPF 8513 ENZYME, DRUGGABLE GENOME GT 389-255 8114 5505 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE KMN-21 CHEMBL570176 19892550 8115 5506 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NANAOMYCIN NANAOMYCIN 8116 5507 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME SELICICLIB SELICICLIB 8117 5508 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NALOXONE BENZOYLHYDRAZONE NALOXONE BENZOYLHYDRAZONE 8118 5509 PDE4A 5141 DRUGGABLE GENOME, ENZYME DYPHYLLINE DYPHYLLINE 8119 5510 FHL2 2274 TRANSCRIPTION FACTOR BINDING gemcitabine GEMCITABINE 24444404 8120 5511 SMN1 6606 DRUGGABLE GENOME (E)-2-STYRYLCHROMONE CHEMBL388823 8121 5512 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE BARDOXOLONE METHYL BARDOXOLONE METHYL 25675144 8122 5513 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME NORGESTREL NORGESTREL 8123 5514 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652220 8124 5515 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER methylprednisolone METHYLPREDNISOLONE 14583680 8125 5516 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER FENTICLOR FENTICLOR 8126 5517 MAPT 4137 DRUGGABLE GENOME NBQX NBQX 8127 5518 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEFOTAXIME SODIUM CEFOTAXIME SODIUM 8129 5519 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL296468 BMS-387032 8131 5520 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor CHEMBL3545085 XL-228 8133 5521 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100365 POBILUKAST 8134 5522 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW806742X GW806742X 8135 5523 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 363894135 MERESTINIB 8136 5524 EPHX2 2053 DRUGGABLE GENOME, ENZYME inhibitor 178101928 8137 5525 PTGS2 5743 DRUGGABLE GENOME, ENZYME CIMICOXIB CIMICOXIB 8139 5526 FGG 2266 DRUGGABLE GENOME, FIBRINOGEN, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE ALFIMEPRASE ALFIMEPRASE 8140 5527 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME VM-202 8143 5528 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL PROPOFOL PROPOFOL 8144 5529 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE BLEOMYCIN A5 14675139 8145 5530 PSMD3 5709 NA inhibitor CHEMBL2103884 OPROZOMIB 8146 5531 XRCC1 7515 CLINICALLY ACTIONABLE CARBOPLATIN CARBOPLATIN 16875718 8149 5532 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CI-1040 CI-1040 8151 5533 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL1201619 APROTININ 8152 5534 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE TCMDC-125758 CHEMBL546797 8153 5535 MAOB 4129 DRUGGABLE GENOME, ENZYME 4-Hydroxybenzylalcohol 8154 5536 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME GEMFIBROZIL GEMFIBROZIL 9409246 8156 5537 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME warfarin WARFARIN 26223945,29737521 8157 5538 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545179 AZD-7451 8158 5539 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PT2399 27595393 8159 5540 REG1A 5967 DRUGGABLE GENOME, GROWTH FACTOR LINOMIDE ROQUINIMEX 9564847 8160 5541 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYLERGONOVINE METHYLERGONOVINE 8162 5542 B2M 567 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE AMIKACIN AMIKACIN 7672871 8164 5543 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TIMOLOL TIMOLOL 8166 5544 PSMC3IP 29893 NUCLEAR HORMONE RECEPTOR inhibitor BORTEZOMIB BORTEZOMIB 8167 5545 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME PMID27828716-Compound-17 8169 5546 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE SP-600125 SP-600125 8170 5547 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CLOBETASOL PROPIONATE CLOBETASOL PROPIONATE 8171 5548 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR GSK2636771 GSK-2636771 8172 5549 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SELENIUM 14744887 8173 5550 ALOX5 240 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL421 SULFASALAZINE 8175 5551 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME evolocumab EVOLOCUMAB 8176 5552 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME CID 4101591 CHEMBL428789 8179 5553 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYTARABINE CYTARABINE 8180 5554 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR ROQUINIMEX ROQUINIMEX 9811314 8181 5555 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL FLURAZEPAM FLURAZEPAM 8183 5556 PDE4B 5142 DRUGGABLE GENOME, ENZYME MEM 1414 8185 5557 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME ADENOVIRAL VECTOR 10911621 8186 5558 PSMB10 5699 PROTEASE, DRUGGABLE GENOME inhibitor BORTEZOMIB BORTEZOMIB 8189 5559 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME Imidazo[4,5-c]pyridine derivative 1 8190 5560 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TRETINOIN TRETINOIN 8192 5561 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME STZ STREPTOZOCIN 8171758 8194 5562 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR N-(3-METHOXYPHENYL)ANTHRANILIC ACID CHEMBL1328677 8195 5563 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102608 IC261 8197 5564 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME DEBIO-9902 SR 8198 5565 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3445 CHEMBL582697 8202 5566 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR CYC-116 CYC-116 8203 5567 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor TIVOZANIB TIVOZANIB 8206 5568 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650021 8207 5569 ECE1 1889 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE inhibitor 178103120 DAGLUTRIL 8210 5570 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME granisetron GRANISETRON 16551910 8212 5571 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE BMN673 8215 5572 CTSA 5476 DRUGGABLE GENOME, ENZYME, PROTEASE SAR164653 8217 5573 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HELENALIN HELENALIN 8219 5574 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-630812 CHEMBL237570 8221 5575 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SALBUTAMOL ALBUTEROL 8223 5576 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CHRYSOPHANOL CHRYSOPHANOL 8224 5577 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Palbociclib PALBOCICLIB 27020857,26369631 8225 5578 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE MGD006 FLOTETUZUMAB 8228 5579 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Vandetanib VANDETANIB 25910950 8229 5580 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME DASATINIB DASATINIB 8231 5581 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102416 8233 5582 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OXETHAZAINE OXETHAZAINE 8234 5583 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652727 YOHIMBINE 8235 5584 SLC7A5 8140 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 328083449 8236 5585 SMAD2 4087 KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GERANIIN GERANIIN 26169124 8237 5586 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE ERLOTINIB ERLOTINIB 8238 5587 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME AC-55541 CHEMBL493076 18720984 8239 5588 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR lithium LITHIUM 24885933 8243 5589 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TETRAPHENYL-UREA CHEMBL169335 8244 5590 PTGS1 5742 ENZYME, DRUGGABLE GENOME SALSALATE SALSALATE 8245 5591 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER CISPLATIN CISPLATIN 19274060 8247 5592 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-60 8248 5593 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 lornoxicam LORNOXICAM 15764711,16342679,16182270 8249 5594 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 etoposide ETOPOSIDE 8251 5595 SMN1 6606 DRUGGABLE GENOME CID 3237815 CHEMBL410484 8252 5596 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR CYCLIRAMINE MALEATE CYCLIRAMINE MALEATE 8254 5597 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Valsartan VALSARTAN 8255 5598 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 8256 5599 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME TCMDC-125758 CHEMBL546797 8257 5600 RAB9A 9367 ENZYME, DRUGGABLE GENOME 6,4'-DIMETHOXYFLAVONE 6,4'-DIMETHOXYFLAVONE 8258 5601 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 315661180 ZOTIRACICLIB 8259 5602 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 vindesine VINDESINE 9187528 8261 5603 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME CEFOTETAN CEFOTETAN 8262 5604 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Everolimus EVEROLIMUS 23629727 8263 5605 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR (R)-SARGACHROMENOL (R)-SARGACHROMENOL 21142112 8264 5606 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Nomegestrol acetate 8265 5607 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL2105743 OLODATEROL HYDROCHLORIDE 8267 5608 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SALUBRINAL SALUBRINAL 8268 5609 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME LEVAMISOLE LEVAMISOLE 17669706 8270 5610 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4459 CHEMBL585502 8273 5611 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR CDNA vaccine 8274 5612 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE allosteric modulator 315661241 8275 5613 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 XANTHONE XANTHONE 8276 5614 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DESLORATADINE DESLORATADINE 8280 5615 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR CLOFARABINE CLOFARABINE 8282 5616 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GTF505 8286 5617 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417941 CHEMBL2095095 8287 5618 ALDH1A1 216 DRUGGABLE GENOME, ENZYME OSAJIN OSAJIN 8288 5619 PGC 5225 DRUGGABLE GENOME, ENZYME, PROTEASE ECABET ECABET 8289 5620 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME Ficlatuzumab FICLATUZUMAB 8290 5621 PTGES 9536 DRUGGABLE GENOME, ENZYME inhibitor 252827532 8292 5622 COMT 1312 DRUGGABLE GENOME, ENZYME ENTACAPONE ENTACAPONE 8293 5623 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 8296 5624 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE NP-506 CHEMBL480356 19110422 8297 5625 RAB9A 9367 ENZYME, DRUGGABLE GENOME 7-METHOXYISOFLAVONE CHEMBL563919 8298 5626 M6PR 4074 ENZYME, DRUGGABLE GENOME Alglucosidase alfa 8299 5627 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PAC-1 PAC-1 27297867 8301 5628 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX OXYPHENBUTAZONE OXYPHENBUTAZONE 8302 5629 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE DS-7423 DS-7423 8303 5630 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HTS-05058 CHEMBL261692 8305 5631 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRADIOL ENANTHATE ESTRADIOL ENANTHATE 8306 5632 HMGCR 3156 ENZYME, DRUGGABLE GENOME Pravastatin PRAVASTATIN 8307 5633 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DINOPROSTONE DINOPROSTONE 8310 5634 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME activator 135650900 RILUZOLE 8314 5635 SCAP 22937 TRANSCRIPTION FACTOR simvastatin SIMVASTATIN 16158080 8316 5636 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE AZACITIDINE AZACITIDINE 8317 5637 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE APD-209 23976842 8318 5638 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-4992 CHEMBL275177 8320 5639 TGFB2 7042 GROWTH FACTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME LERDELIMUMAB LERDELIMUMAB 8321 5640 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE BARASERTIB BARASERTIB 8322 5641 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR Genistein GENISTEIN 8323 5642 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GOSSYPETIN GOSSYPETIN 8324 5643 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PF-06700841 BREPOCITINIB 8325 5644 POLI 11201 DNA REPAIR PROTOAPIGENONE PROTOAPIGENONE 8326 5645 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE N/A 21881046,25281355,22490330,21670448 8327 5646 MAPT 4137 DRUGGABLE GENOME DANTROLENE DANTROLENE 8328 5647 PDE4A 5141 DRUGGABLE GENOME, ENZYME TOFIMILAST TOFIMILAST 8333 5648 CXCL8 3576 DRUGGABLE GENOME ALPRAZOLAM ALPRAZOLAM 12218154 8334 5649 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 178103585 ROMIDEPSIN 8335 5650 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AFATINIB AFATINIB 26619011,19455431,22452896,23102728,20068085,16707764,17653080,15710947,20479403,25668228,16912157,24893891,15728811,20573926,16258541,19692680,15118125,18227510,24658966,18199554,19922469,20033049,26515464,25923549,21783417,19692684,22753918,16187797,22452895,23945392,15329413,24636847,23816963,24729716,23816960,22285168,19096302,16204070,24894453,16043828,22215752,21194487,24065731,15118073,20022809,23948351,16115929,18458038,17332364,24623981,19147750,25157968,16011858,21430269,2302402,15737014,26720284,21670455,21233402,23242437,25923550,22588155,21531810,18303429,19671738 8336 5651 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER CYCLOSPORINE CYCLOSPORINE 23017888 8337 5652 SLC9A3 6550 DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE, EXCHANGER GLUCOCORTICOID 9727362 8339 5653 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NIMETAZEPAM NIMETAZEPAM 8341 5654 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME GW441756X GW441756X 8342 5655 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME RESVERATROL RESVERATROL 16116226 8343 5656 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME ENTRECTINIB ENTRECTINIB 8344 5657 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME OSI-632 OSI-632 8345 5658 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ANTISENSE OLIGONUCLEOTIDES 15141022 8346 5659 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102917 8347 5660 KCNS3 3790 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL284348 DALFAMPRIDINE 8348 5661 POLB 5423 DNA REPAIR, DRUGGABLE GENOME LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 8349 5662 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME ENMD-2076 ENMD-2076 8350 5663 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME (R,S)-INDATRALINE (R,S)-INDATRALINE 8351 5664 HTT 3064 DRUGGABLE GENOME SJ000113972 CHEMBL591137 8352 5665 GSTM1 2944 DRUGGABLE GENOME, ENZYME anthracyclines and related substances 27785604 8357 5666 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1706 NAPHAZOLINE HYDROCHLORIDE 8358 5667 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650950 8359 5668 EIF4A1 1973 DRUGGABLE GENOME HIPPURISTANOL HIPPURISTANOL 16532013 8360 5669 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor PF-4691502 PF-04691502 8361 5670 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Antiinflammatory agents, non-steroids 17681167 8362 5671 ALOX15 246 ENZYME, DRUGGABLE GENOME SANGUINARIUM SANGUINARIUM 8363 5672 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BUFOGENIN BUFOGENIN 8364 5673 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER (R,S)-INDATRALINE (R,S)-INDATRALINE 8368 5674 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE oxycodone OXYCODONE 25239082,31773688,21209234 8369 5675 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING MOCETINOSTAT MOCETINOSTAT 23829483,26287310 8372 5676 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING ALPHA-DIFLUOROMETHYLORNITHINE 9950818 8373 5677 APC 324 CLINICALLY ACTIONABLE Sulindac SULINDAC 19755659 8374 5678 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PRX-3140 8376 5679 LSS 4047 ENZYME, DRUGGABLE GENOME inhibitor 178103323 8377 5680 ATAD5 79915 NA TPCK TPCK 8379 5681 ATXN2 6311 NA NSC-348401 CHEMBL515505 8380 5682 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US10149841, Compound 19 8381 5683 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32z 8382 5684 PDF 64146 DRUGGABLE GENOME Ustekinumab USTEKINUMAB 8383 5685 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE DIFFERENTIATION INDUCER 8595156 8385 5686 SMN1 6606 DRUGGABLE GENOME 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 8386 5687 HSD11B2 3291 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME RG-7234 8387 5688 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE LY2780301 28750271,25902900 8388 5689 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TIOTROPIUM TIOTROPIUM 8390 5690 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor BEZ235 DACTOLISIB 8391 5691 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR NIMESULIDE NIMESULIDE 8392 5692 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 354702300 GELDANAMYCIN 8393 5693 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME SB-202190 SB-202190 8395 5694 MPHOSPH8 54737 NA PD-404182 CHEMBL595227 8396 5695 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER FEXOFENADINE HYDROCHLORIDE 15536457 8397 5696 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102662 8399 5697 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENTANYL FENTANYL 8400 5698 TNFRSF14 8764 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME 178101763 8403 5699 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-35 8405 5700 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE LAK 8895065 8407 5701 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL agonist 178101134 8408 5702 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 11437491 8409 5703 TAF1 6872 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE inhibitor 336446910 8410 5704 PSMA6 5687 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL451887 CARFILZOMIB 8412 5705 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-3286 CHEMBL581880 8413 5706 HTT 3064 DRUGGABLE GENOME GNF-PF-3996 CHEMBL584458 8414 5707 CMKLR1 1240 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100428 8415 5708 PDE4B 5142 DRUGGABLE GENOME, ENZYME ethanol ALCOHOL 32451486 8416 5709 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201141 IBUPROFEN LYSINE 8419 5710 ACTB 60 TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE ETHINYLESTRADIOL ETHINYL ESTRADIOL 17288598 8420 5711 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651094 SULPROSTONE 8421 5712 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Beta-Lapachone LAPACHONE 8422 5713 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 223366126 DUVELISIB 8423 5714 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME LY-2090314 LY-2090314 8425 5715 MTTP 4547 DRUGGABLE GENOME BMS-201038 LOMITAPIDE MESYLATE 8426 5716 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 4,4'-DITHIODIPYRIDINE CHEMBL1232076 8429 5717 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650717 8430 5718 ATAD5 79915 NA EUPAFOLIN EUPAFOLIN 8431 5719 EPHX2 2053 DRUGGABLE GENOME, ENZYME inhibitor 178103826 OXAPROZIN 8432 5720 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME PAPAVERINE HYDROCHLORIDE PAPAVERINE HYDROCHLORIDE 8433 5721 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CRLX101 8434 5722 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US10100051, Compound 1 8435 5723 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR TAXIFOLIN TAXIFOLIN 8436 5724 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Pentoxifylline PENTOXIFYLLINE 8437 5725 CPT2 1376 DRUGGABLE GENOME PERHEXILINE PERHEXILINE 8438 5726 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SB-202190 SB-202190 8441 5727 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE Methimazole METHIMAZOLE 8442 5728 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW819077X GW819077X 8443 5729 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME fluorouracil FLUOROURACIL 27995989,21449681,18540691 8444 5730 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR CB-839 TELAGLENASTAT 28346230 8446 5731 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TANNIN PYROGALLOL TANNIN PYROGALLOL 8447 5732 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE N-ACETYLCOLCHINOL CHEMBL486504 8449 5733 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER THYMIDINE THYMIDINE 9379682 8450 5734 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2107911 ONERCEPT 8451 5735 E2F1 1869 TRANSCRIPTION FACTOR BCNU CARMUSTINE 11445852 8452 5736 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor SUNITINIB SUNITINIB 8453 5737 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME RESVERATROL RESVERATROL 8455 5738 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME PHENOBARBITAL PHENOBARBITAL 9230198 8456 5739 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TAMOXIFEN CITRATE TAMOXIFEN CITRATE 8457 5740 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Liproca Depot 8458 5741 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1200893 PROTOKYLOL HYDROCHLORIDE 8460 5742 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545006 PWT-33587 8461 5743 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NALBUPHINE NALBUPHINE 22204910 8463 5744 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1201765 FESOTERODINE FUMARATE 8464 5745 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEFOXITIN SODIUM CEFOXITIN SODIUM 8468 5746 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME NIMESULIDE NIMESULIDE 8469 5747 CA2 760 DRUGGABLE GENOME, ENZYME BRINZOLAMIDE BRINZOLAMIDE 8471 5748 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR SJ000113257 CHEMBL528694 8473 5749 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE Ac-YVAD-cmk 8474 5750 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHENFORMIN HYDROCHLORIDE PHENFORMIN HYDROCHLORIDE 8475 5751 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME VORTIOXETINE VORTIOXETINE 8476 5752 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Dextrothyroxine Sodium 8478 5753 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135649872 CHEMBL361355 8479 5754 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Everolimus EVEROLIMUS 24742739 8480 5755 CXCL8 3576 DRUGGABLE GENOME FENTANYL FENTANYL 9527747 8481 5756 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME RUPATADINE RUPATADINE 8482 5757 RACGAP1 29127 NA PHENOTHIAZINE PHENOTHIAZINE 8484 5758 HTT 3064 DRUGGABLE GENOME N-(3,4-DIMETHOXYPHENETHYL)BENZENESULFONAMIDE CHEMBL258316 8487 5759 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BENZAMIL BENZAMIL 8488 5760 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 178102315 RUXOLITINIB 8489 5761 VEGFB 7423 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL2108313 CONBERCEPT 8491 5762 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Ribociclib Succinate 8492 5763 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3545412 K-877 8495 5764 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MINOXIDIL MINOXIDIL 22931300 8499 5765 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE DEXAMETHASONE DEXAMETHASONE 7599067 8500 5766 GJB1 2705 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER inhibitor 178100972 CARBENOXOLONE 8501 5767 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1509 DROSPIRENONE 8502 5768 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545265 MLN-0415 8503 5769 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR TAXOTERE TAXOTERE 10470115 8505 5770 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Maleimides derivative 3 8508 5771 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE HESPERETIN HESPERETIN 8509 5772 BAZ2B 29994 NA PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE CHEMBL114544 8511 5773 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 178103833 8512 5774 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 8517 5775 NDUFS1 4719 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 8518 5776 KAT2B 8850 ENZYME, DRUGGABLE GENOME cocaine COCAINE 8519 5777 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 363894187 8520 5778 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BRONOPOL BRONOPOL 8521 5779 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MESALAZINE MESALAMINE 8522 5780 F5 2153 DRUGGABLE GENOME estrogens ESTRONE SODIUM SULFATE 11532625,16113779,12067913,12869355,16301339,9459317,10073976,15467059,11859850,10943572,12069454,12138364,14551147,7968118,11703344 8523 5781 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER erlotinib ERLOTINIB 8524 5782 ATAD5 79915 NA PIFEXOLE PIFEXOLE 8525 5783 ATAD5 79915 NA NSC-319994 CHEMBL1329443 8526 5784 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE RAS INHIBITOR 12137763 8529 5785 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 2-BFI CHEMBL404505 8530 5786 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER zidovudine ZIDOVUDINE 22960662,16791115 8531 5787 KMT5C 84787 ENZYME, METHYL TRANSFERASE, DNA REPAIR inhibitor 310264730 8532 5788 ALOX15 246 ENZYME, DRUGGABLE GENOME Isothiazolone derivative 1 8533 5789 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE modulator ENOBOSARM ENOBOSARM 8537 5790 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL49642 INDIBULIN 8538 5791 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (R,S)-INDATRALINE (R,S)-INDATRALINE 8540 5792 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MAKALUVAMINE C TFA SALT MAKALUVAMINE C TFA SALT 8691207 8541 5793 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE NSC-348401 CHEMBL515505 8542 5794 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-1000163A GSK-1000163A 8543 5795 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Indazole derivative 6 8546 5796 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Seocalcitol SEOCALCITOL 8547 5797 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL1683544 ERIBULIN MESYLATE 8548 5798 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Trifluridine TRIFLURIDINE 8549 5799 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650473 8551 5800 TUBA1A 7846 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 8552 5801 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME BICALUTAMIDE BICALUTAMIDE 11845989 8555 5802 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CENISERTIB CENISERTIB 8556 5803 FKBP5 2289 DRUGGABLE GENOME gemcitabine GEMCITABINE 23936393 8557 5804 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Selumetinib SELUMETINIB 24971884 8560 5805 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE AMUVATINIB AMUVATINIB 8561 5806 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME KENPAULLONE KENPAULLONE 8562 5807 MAPT 4137 DRUGGABLE GENOME 4-HYDROXYDERRICIN CHEMBL458094 8563 5808 BAZ2B 29994 NA CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 8564 5809 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR inhibitor BORTEZOMIB BORTEZOMIB 8566 5810 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME DNDI1417467 CHEMBL1997335 8569 5811 GCLM 2730 ENZYME ANTIOXIDANT 12637989 8570 5812 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME zidovudine ZIDOVUDINE 23089673 8571 5813 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME PIRARUBICIN PIRARUBICIN 8572 5814 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BAS-8770951 CHEMBL478323 19179076 8573 5815 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CANERTINIB CANERTINIB 8575 5816 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW829055X GW829055X 8576 5817 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHYLTESTOSTERONE METHYLTESTOSTERONE 8577 5818 PKN1 5585 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565832 8578 5819 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE FORMOTEROL FORMOTEROL 8579 5820 SMN2 6607 DRUGGABLE GENOME GNF-PF-992 CHEMBL602561 8580 5821 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SPIPERONE SPIPERONE 8581 5822 XDH 7498 DRUGGABLE GENOME, ENZYME IMMUNOMODULATORS 8046245 8583 5823 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Arformoterol ARFORMOTEROL 8584 5824 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THIOINOSINE THIOINOSINE 8585 5825 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME APICIDIN APICIDIN 19705846 8586 5826 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE AST-487 AST-487 8587 5827 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051793 GIVINOSTAT 8588 5828 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 8590 5829 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE GM6001 8591 5830 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE LEVODOPA LEVODOPA 14514477 8594 5831 HEBP1 50865 DRUGGABLE GENOME 4-(2-cyclohexylethoxy) aniline derivative 2 8595 5832 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178103821 NEFAZODONE 8598 5833 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE SULINDAC SULINDAC 16030090 8599 5834 HBB 3043 DRUGGABLE GENOME, ENZYME negative modulator CHEMBL18901 EFAPROXIRAL 8600 5835 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor 249565784 LY-2874455 8601 5836 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR toremifene TOREMIFENE 8602 5837 SMN1 6606 DRUGGABLE GENOME 2-METHOXYPHENAZINE CHEMBL1420181 8603 5838 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME activator 178102951 8604 5839 MAPT 4137 DRUGGABLE GENOME ISOEUGENITOL ISOEUGENITOL 8606 5840 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR inhibitor 252827512 CHEMBL481422 8607 5841 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL450 METHARBITAL 8608 5842 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MIDOSTAURIN MIDOSTAURIN 15448205 8609 5843 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1626570 HEXOCYCLIUM METHYLSULFATE 8612 5844 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR 2,3,5-TRIS(4-HYDROXYPHENYL)THIOPHENE CHEMBL2332580 23586645 8613 5845 GABBR2 9568 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL R-BACLOFEN 8616 5846 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TETRAMETHRIN TETRAMETHRIN 8618 5847 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-17 8620 5848 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TRIFLUOPERAZINE TRIFLUOPERAZINE 8621 5849 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR RHEIN RHEIN 8622 5850 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GI-4000 25044103,25585100,24372276 8623 5851 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-US20130053382 38(5-7) 8625 5852 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MESOTRIONE MESOTRIONE 8626 5853 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IDEBENONE IDEBENONE 8627 5854 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME CAR-T cells targeting mesothelin 8628 5855 ACP1 52 ENZYME, DRUGGABLE GENOME, PROTEIN PHOSPHATASE GNF-PF-4353 CHEMBL527307 8629 5856 MPHOSPH8 54737 NA N,N-HEXAMETHYLENEAMILORIDE N,N-HEXAMETHYLENEAMILORIDE 8630 5857 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102573 8631 5858 BCHE 590 DRUGGABLE GENOME, ENZYME Succinylcholine SUXAMETHONIUM 8632 5859 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 315661321 UPADACITINIB 8633 5860 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Benzodihydroisofuran derivative 2 8635 5861 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545283 RIVICICLIB 8637 5862 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE HGF 16616440 8638 5863 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ALLOPURINOL ALLOPURINOL 22931300 8639 5864 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200764 METHACHOLINE CHLORIDE 8641 5865 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor MK 1775 8643 5866 ATAD5 79915 NA FLAVONE FLAVONE 8646 5867 HPSE 10855 ENZYME, DRUGGABLE GENOME 2-O, 3-O DESULFATED HEPARIN 8647 5868 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 363894208 ILORASERTIB 8648 5869 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135649698 8650 5870 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Vorinostat VORINOSTAT 18483379,23498719 8651 5871 PDE10A 10846 ENZYME, DRUGGABLE GENOME Triazolo-pyridine derivative 6 8652 5872 CBX1 10951 NA EXISULIND EXISULIND 8654 5873 MIF 4282 DRUGGABLE GENOME, CELL SURFACE PPD 393437 8655 5874 TSPO 706 DRUGGABLE GENOME Benzothiazepine analog 9 8657 5875 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor CHEMBL19 METHAZOLAMIDE 8661 5876 BAZ2B 29994 NA GNF-PF-3909 CHEMBL599304 8663 5877 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LEVOTHYROXINE LEVOTHYROXINE 8664 5878 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME inhibitor 178103594 8665 5879 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BKM120 BUPARLISIB 8666 5880 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL235191 TACEDINALINE 8667 5881 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 310264784 CHEMBL442577 8668 5882 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Apremilast APREMILAST 8670 5883 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-747267 CHEMBL610767 8671 5884 POLK 51426 DNA REPAIR, ENZYME IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 8672 5885 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-1702 CHEMBL600313 8674 5886 CD3D 915 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE MUROMONAB MUROMONAB-CD3 8679 5887 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1416988 CHEMBL1389794 8680 5888 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME NSC-753574 CHEMBL2088730 22982122 8681 5889 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TETRADECYLTHIOACETIC ACID TETRADECYLTHIOACETIC ACID 20036122 8684 5890 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL435224 LAPAQUISTAT ACETATE 8686 5891 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME ELIPRODIL ELIPRODIL 8687 5892 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE LAS-100977 ABEDITEROL 8688 5893 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE LIGNAN 15671223 8689 5894 STK33 65975 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565870 8691 5895 HBB 3043 DRUGGABLE GENOME, ENZYME Luspatercept–aamt 8692 5896 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 178103584 8693 5897 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL738 THIOPENTAL SODIUM 8695 5898 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME DNDI1417467 CHEMBL1997335 8696 5899 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Dihydropyrido pyrazinone compound 3 8697 5900 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR BAY 1082439 8698 5901 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME NU-6027 CHEMBL303958 8699 5902 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 5310655 CHEMBL408563 8700 5903 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Bococizumab BOCOCIZUMAB 8701 5904 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME inhibitor 249565704 LONAFARNIB 8702 5905 BRCA2 675 CLINICALLY ACTIONABLE niraparib NIRAPARIB 8703 5906 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE HISTONE DEACETYLASE INHIBITOR 15474507 8705 5907 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Irinotecan IRINOTECAN 26842236 8708 5908 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE ACARBOSE ACARBOSE 8886823 8710 5909 APC 324 CLINICALLY ACTIONABLE NC043 21321609 8711 5910 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RS-39604 CHEMBL66114 8715 5911 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 249565626 SCH-900776 8716 5912 POLG 5428 ENZYME Valproic Acid 8717 5913 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PMID29671355-Compound-31 8718 5914 CA12 771 DRUGGABLE GENOME inhibitor CHEMBL1200814 ACETAZOLAMIDE SODIUM 8720 5915 POLI 11201 DNA REPAIR NSC-95397 CHEMBL429095 8721 5916 KDM4A 9682 DRUGGABLE GENOME, ENZYME OXYTETRACYCLINE OXYTETRACYCLINE 8723 5917 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TRIFLUOPERAZINE TRIFLUOPERAZINE 8724 5918 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ACRYLAMIDE ACRYLAMIDE 8726 5919 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1200665 DIPHENOXYLATE HYDROCHLORIDE 8727 5920 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ANS-6637 8729 5921 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-742865 CHEMBL102936 8730 5922 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW301888X GW301888X 8731 5923 MAP4K3 8491 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565855 8733 5924 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISOLIQUIRITIGENIN ISOLIQUIRITIGENIN 8734 5925 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565851 8735 5926 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME BI-853520 BI-853520 8736 5927 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2011806744710 8738 5928 POLK 51426 DNA REPAIR, ENZYME CARBOFENOTION CARBOFENOTION 8739 5929 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2103803 DAROTROPIUM BROMIDE 8740 5930 CD44 960 DRUGGABLE GENOME, CELL SURFACE GENTAMICIN GENTAMICIN 14967965 8741 5931 PDE4A 5141 DRUGGABLE GENOME, ENZYME Ronomilast 8742 5932 BAZ2B 29994 NA ZAFIRLUKAST ZAFIRLUKAST 8743 5933 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 sildenafil SILDENAFIL 28440343 8744 5934 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3545081 RG-7304 8745 5935 TNC 3371 DRUGGABLE GENOME, FIBRINOGEN F-16-131I 8746 5936 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Cetuximab CETUXIMAB 27207775 8747 5937 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor VISMODEGIB VISMODEGIB 8748 5938 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENANTHROLINE PHENANTHROLINE 8749 5939 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE EMTRICITABINE EMTRICITABINE 17172311 8753 5940 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL628 PENTOXIFYLLINE 8757 5941 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 252166770 8759 5942 ACVR2A 92 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CELL SURFACE BYM338 BIMAGRUMAB 8760 5943 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Anti-EGFR CAR T 8761 5944 UGT1A10 54575 DRUGGABLE GENOME, ENZYME mycophenolic acid 24220207 8762 5945 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 223366120 LANABECESTAT 8763 5946 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135650308 8764 5947 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135649895 8765 5948 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME POTASSIUM DICHROMATE POTASSIUM DICHROMATE 8766 5949 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PANITUMUMAB PANITUMUMAB 8767 5950 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Bisphosphonates 18687167,24311107,21151198 8769 5951 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CETYLPYRIDINIUM CHLORIDE CETYLPYRIDINIUM CHLORIDE 8770 5952 ATXN2 6311 NA PD-173074 PD-173074 8771 5953 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE BARDOXOLONE METHYL BARDOXOLONE METHYL 25675144 8773 5954 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-60340 CHEMBL1534034 8774 5955 FGB 2244 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, FIBRINOGEN, DRUGGABLE GENOME RECOMBINANT FACTOR IX FC FUSION PROTEIN 8776 5956 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME L-Tryptophan TRYPTOPHAN 8777 5957 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SOTRASTAURIN SOTRASTAURIN 8778 5958 CA2 760 DRUGGABLE GENOME, ENZYME Ethoxzolamide ETHOXZOLAMIDE 8779 5959 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HERBIMYCIN HERBIMYCIN 23947794 8780 5960 TOP2B 7155 DRUGGABLE GENOME, ENZYME DIGITOXIN DIGITOXIN 16309315 8781 5961 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME AZD-1775 ADAVOSERTIB 8783 5962 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE allosteric modulator 381745019 8787 5963 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker 252166811 8788 5964 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE RISPERIDONE RISPERIDONE 15567770,11545247 8789 5965 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LY2835219 ABEMACICLIB 8790 5966 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME MYRICETIN MYRICETIN 8792 5967 PTK6 5753 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, ENZYME inhibitor 249565866 8793 5968 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE KETAMINE KETAMINE 20361801 8794 5969 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR BRYOSTATIN BRYOSTATIN 8795 5970 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 328083468 8796 5971 HOMER1 9456 KINASE levodopa LEVODOPA 24126708 8797 5972 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178101025 8798 5973 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BENZALDEHYDE BENZALDEHYDE 8799 5974 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor VALPROIC ACID DEPAKOTE 8800 5975 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135649926 ALPRENOLOL 8802 5976 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DYCLONINE HYDROCHLORIDE DYCLONINE HYDROCHLORIDE 8803 5977 SMN2 6607 DRUGGABLE GENOME CID 3237815 CHEMBL410484 8805 5978 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 340590249 DELGOCITINIB 8808 5979 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Carvedilol CARVEDILOL 8810 5980 TMEM97 27346 NA PMID30185082-Compound-57 8812 5981 POLK 51426 DNA REPAIR, ENZYME ISOKAEMPFERIDE ISOKAEMPFERIDE 8813 5982 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZD5363 CAPIVASERTIB 19755509,24088382 8815 5983 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME OXYTETRACYCLINE HYDROCHLORIDE OXYTETRACYCLINE HYDROCHLORIDE 8816 5984 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 252166570 GSK-1070916 8817 5985 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200584 AMINOSALICYLATE POTASSIUM 8819 5986 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PHENOXODIOL 8820 5987 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME DINACICLIB DINACICLIB 8821 5988 HEXA 3073 DRUGGABLE GENOME, ENZYME N-ACETYLGLUCOSAMINE THIAZOLINE CHEMBL257158 20822912 8822 5989 GMNN 51053 DRUGGABLE GENOME DNDI1417099 CHEMBL1565444 8823 5990 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE allosteric modulator 178102419 8824 5991 PDE7A 5150 ENZYME, DRUGGABLE GENOME ISOBUTYLMETHYLXANTHINE ISOBUTYLMETHYLXANTHINE 24239625 8825 5992 MAOB 4129 DRUGGABLE GENOME, ENZYME Coumarin/resveratrol hybrid derivative 1 8826 5993 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE MLN-576 8827 5994 FN1 2335 DRUGGABLE GENOME CHEMBL2109608 L19IL2 8828 5995 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CYPROTERONE ACETATE CYPROTERONE ACETATE 8829 5996 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR isoproterenol ISOPROTERENOL 27643874 8830 5997 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-O3 8831 5998 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HER2/neu peptide vaccine 8835 5999 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME FK-614 ATX08-001 8836 6000 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE blocker CHEMBL473 DOFETILIDE 8838 6001 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE RETINOIC ACID 12485937,11426618 8839 6002 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 2',3'-DIHYDROXYFLAVONE CHEMBL242171 8840 6003 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE AZAKENPAULLONE AZAKENPAULLONE 8841 6004 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL984 MIVACURIUM CHLORIDE 8842 6005 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1201729 DRONEDARONE HYDROCHLORIDE 8843 6006 TUBB 203068 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 8844 6007 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Trilaciclib TRILACICLIB 8845 6008 EPHX2 2053 DRUGGABLE GENOME, ENZYME lithium LITHIUM 29121268 8846 6009 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE 178101617 8847 6010 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE 2-CHLOROADENOSINE CHEMBL285819 8848 6011 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CID 887167 CHEMBL260342 8849 6012 USP7 7874 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME, PROTEASE PMID26077642-Compound-Vif1 8851 6013 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME agonist CHEMBL312443 GABOXADOL 8854 6014 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Tivantinib TIVANTINIB 8855 6015 FAAH2 158584 DRUGGABLE GENOME, ENZYME inhibitor 310264767 8856 6016 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ZK-93423 CHEMBL1518572 8857 6017 MAOB 4129 DRUGGABLE GENOME, ENZYME Heteroaryl-cyclopropylamine derivative 1 8858 6018 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR PHA-767491 CHEMBL225519 8859 6019 TMEM97 27346 NA Piperazinyl methyl quinazolinone derivative 3 8860 6020 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME PROTEOLYTIC ENZYMES 9502079 8862 6021 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178101837 BATIMASTAT 8863 6022 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE INSULIN INSULIN 17182020 8864 6023 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME MIDAZOLAM MIDAZOLAM 17093965 8865 6024 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME FACTOR IX 8866 6025 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 310264749 SERABELISIB 8867 6026 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178101497 KETOPROFEN 8868 6027 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME PSEUDOEPHEDRINE PSEUDOEPHEDRINE 8869 6028 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 8873 6029 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CROMOLYN CROMOLYN 22931300 8874 6030 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE TESTOSTERONE PROPIONATE TESTOSTERONE PROPIONATE 8875 6031 ALOX15 246 ENZYME, DRUGGABLE GENOME CHLORANIL CHLORANIL 8876 6032 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 8877 6033 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME PF-562271 PF-00562271 8880 6034 FANCC 2176 CLINICALLY ACTIONABLE, DNA REPAIR MITOMYCIN MITOMYCIN 16243825 8881 6035 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DACTINOMYCIN DACTINOMYCIN 22931300 8882 6036 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE antisense oligonucleotide ISIS 5132 8883 6037 TAOK3 51347 DNA REPAIR, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565794 8884 6038 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PRX-321 PRX-321 8886 6039 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-125252 CHEMBL1408031 22524450 8887 6040 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL GABOXADOL GABOXADOL 8890 6041 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE BCL201 8891 6042 ATAD5 79915 NA DAPH DAPH 8892 6043 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 739615 CHEMBL260560 8893 6044 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AGEN1884 ZALIFRELIMAB 8897 6045 RAB9A 9367 ENZYME, DRUGGABLE GENOME SIB-1893 CHEMBL88612 8898 6046 SMN1 6606 DRUGGABLE GENOME LASSBIO-294 CHEMBL233194 8900 6047 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL2140408 AMG-900 8901 6048 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BISMUTH SUBSALICYLATE BISMUTH SUBSALICYLATE 8902 6049 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME LY3009120 LY-3009120 26343583 8903 6050 GLS 2744 ENZYME ASTERRIC ACID ASTERRIC ACID 8904 6051 MLST8 64223 KINASE inhibitor AZD8055 AZD-8055 8905 6052 SLCO4C1 353189 TRANSPORTER, DRUGGABLE GENOME 178101436 8906 6053 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME PD-98059 CHEMBL35482 11313272 8907 6054 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PMID26924192-Compound-102 8908 6055 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR GM-CSF REGRAMOSTIM 15126418 8909 6056 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR METHOTREXATE METHOTREXATE 8911 6057 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor VANDETANIB VANDETANIB 8912 6058 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Loratadine LORATADINE 8915 6059 S100A2 6273 NA ANTISENSE OLIGONUCLEOTIDES 11304580 8916 6060 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 310264699 SAMOTOLISIB 8917 6061 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CISPLATIN CISPLATIN 8918 6062 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME LBR-101 FREMANEZUMAB 8919 6063 CSNK2A2 1459 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME, TRANSCRIPTION FACTOR US8940736, 23 8921 6064 CBX1 10951 NA MIFEPRISTONE MIFEPRISTONE 8922 6065 HYAL2 8692 DRUGGABLE GENOME, CELL SURFACE HORMONES 7215332 8923 6066 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545285 XL-999 8924 6067 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME FLUDIAZEPAM FLUDIAZEPAM 8925 6068 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Pyrazolopyridine derivative 3 8927 6069 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR inhibitor CHEMBL1200983 GALLIUM NITRATE 8928 6070 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CEDIRANIB CEDIRANIB 8929 6071 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PHENYLBUTANOIC ACID PHENYLBUTANOIC ACID 24044874 8930 6072 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME PD-153035 CHEMBL29197 17681471 8931 6073 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE Triciribine TRICIRIBINE 26224873 8932 6074 TLR7 51284 DRUGGABLE GENOME antagonist 178103773 HYDROXYCHLOROQUINE 8933 6075 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR norepinephrine NOREPINEPHRINE 8934 6076 PLD2 5338 ENZYME, DRUGGABLE GENOME VU0364739 8936 6077 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Bosutinib BOSUTINIB 8937 6078 KRT18 3875 DRUGGABLE GENOME ANTIVIRAL 17713161 8938 6079 IL1B 3553 KINASE, DRUGGABLE GENOME AC-201 DIACEREIN 8942 6080 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Cediranib CEDIRANIB 26461489 8945 6081 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME LEVOCABASTINE LEVOCABASTINE 8946 6082 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL blocker 178101035 8949 6083 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE ENTINOSTAT ENTINOSTAT 8951 6084 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Sorafenib SORAFENIB 8953 6085 ERAP1 51752 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 252166866 8954 6086 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME AMG-131 INT131 8957 6087 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL2103836 IMAGABALIN 8958 6088 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX L-DOPA LEVODOPA 16930409,15896973 8959 6089 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR PHENELZINE SULFATE PHENELZINE SULFATE 8965 6090 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor ODM-201 DAROLUTAMIDE 8967 6091 PDE4A 5141 DRUGGABLE GENOME, ENZYME Revamilast REVAMILAST 8968 6092 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyridopyrimidinone derivative 1 8969 6093 POLI 11201 DNA REPAIR ASTERRIC ACID ASTERRIC ACID 8970 6094 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650251 FARGLITAZAR 8972 6095 SLC31A1 1317 TRANSPORTER cisplatin CISPLATIN 22725681,22516052 8975 6096 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR 2'-EPI-TUBERATOLIDE B 2'-EPI-TUBERATOLIDE B 21142112 8976 6097 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Olaratumab OLARATUMAB 8978 6098 CPM 1368 PROTEASE, DRUGGABLE GENOME, CELL SURFACE, ENZYME inhibitor 252166875 8980 6099 CBX1 10951 NA GW7647 GW7647 8981 6100 MAPT 4137 DRUGGABLE GENOME SJ000294102 CHEMBL607309 8982 6101 GMNN 51053 DRUGGABLE GENOME TCMDC-125254 CHEMBL547313 8983 6102 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL190333 RWJ-67657 8984 6103 TUBB2A 7280 DRUGGABLE GENOME VINORELBINE VINORELBINE 8986 6104 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651128 8987 6105 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor 374883860 8989 6106 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR TESTOSTERONE TESTOSTERONE 8994 6107 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrrole derivative 7 8996 6108 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEXEFAROXAN DEXEFAROXAN 8997 6109 SLC16A1 6566 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME BUTYRATE 11882670 8998 6110 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor LENVATINIB LENVATINIB 8999 6111 SPSB2 84727 DRUGGABLE GENOME, B30_2 SPRY DOMAIN PHENYLTHIAZOL-2-AMINE CHEMBL175296 25559643 9000 6112 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME antibody RILOTUMUMAB RILOTUMUMAB 9004 6113 PTGES 9536 DRUGGABLE GENOME, ENZYME Alpha-substituted pirinixic acid and pirinixic acid ester derivative 1 9005 6114 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX 2-PHENYLACETYLAMINOBENZOTHIAZOLE CHEMBL1405979 9006 6115 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Ifosfamide IFOSFAMIDE 23165797 9007 6116 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Tamoxifen TAMOXIFEN 26116361 9008 6117 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE Peptidomimetic analog 5 9009 6118 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Rhopressa NETARSUDIL DIMESYLATE 9010 6119 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GUTHION GUTHION 9011 6120 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LOFEPRAMINE HYDROCHLORIDE LOFEPRAMINE HYDROCHLORIDE 9013 6121 PLCG1 5335 ENZYME, KINASE, PHOSPHOLIPASE, DRUGGABLE GENOME Pyrazolones 26398624 9014 6122 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE XL999 9015 6123 MAOB 4129 DRUGGABLE GENOME, ENZYME 3-Hydroxy-2-butanone 9016 6124 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor AZD6244 SELUMETINIB 9017 6125 TUBB2A 7280 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 9019 6126 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor LDE 225 9024 6127 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR TAK-828 9025 6128 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR BELINOSTAT BELINOSTAT 9026 6129 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME simeprevir SIMEPREVIR 9030 6130 MAPT 4137 DRUGGABLE GENOME ALTENUSIN ALTENUSIN 9031 6131 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME G-573 23934108 9034 6132 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Trametinib TRAMETINIB 27659046,27797976,26882569,26469692,26627007,26369631 9035 6133 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Erdafitinib ERDAFITINIB 9036 6134 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON BETA-1B 9040 6135 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 3,4-DICHLOROISOCOUMARIN CHEMBL24983 9041 6136 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ETHINYL ESTRADIOL 9042 6137 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135650928 ROSUVASTATIN 9043 6138 RGS12 6002 DRUGGABLE GENOME LAVENDUSTIN C LAVENDUSTIN C 9046 6139 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE 0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE 9047 6140 PTGS2 5743 DRUGGABLE GENOME, ENZYME Tiaprofenic acid 9049 6141 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR RECOMBINANT HUMAN IL-4 11228246 9050 6142 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor SELUMETINIB SELUMETINIB 9051 6143 TOP2B 7155 DRUGGABLE GENOME, ENZYME Berubicin BERUBICIN 9052 6144 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME GDC-0973 COBIMETINIB 9053 6145 SAP130 79595 NA SPLICEOSTATIN-A CHEMBL1221944 17643111 9055 6146 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE RAPAMYCIN SIROLIMUS 15878982 9056 6147 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-52 9057 6148 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9522888, 412 9060 6149 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME CENISERTIB CENISERTIB 9061 6150 BAZ2B 29994 NA CICLOPIROX OLAMINE CICLOPIROX OLAMINE 9062 6151 IL1B 3553 KINASE, DRUGGABLE GENOME XOMA 052 9063 6152 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2031465 AZD-6703 9064 6153 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME EMBELIN EMBELIN 9065 6154 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHEMBL407 FLUMAZENIL 9066 6155 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200996 MEPHENTERMINE SULFATE 9067 6156 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565631 TIVANTINIB 9070 6157 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GNF-PF-5294 CHEMBL579725 9071 6158 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL1742994 BRENTUXIMAB VEDOTIN 9072 6159 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE LICOAGRODIN LICOAGRODIN 24047800 9073 6160 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME avatrombopag AVATROMBOPAG 9074 6161 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MRS-1220 CHEMBL88147 9075 6162 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL HEXOBARBITAL HEXOBARBITAL 9076 6163 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE CIGLITAZONE CIGLITAZONE 20170185 9077 6164 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-62 9078 6165 MAPT 4137 DRUGGABLE GENOME CRYPTOTANSHINONE CRYPTOTANSHINONE 9080 6166 CDK18 5129 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR inhibitor CHEMBL488436 AZD-5438 9081 6167 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RELCOVAPTAN RELCOVAPTAN 9082 6168 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TRAMETINIB TRAMETINIB 25504439,23515407,25452114,23431193 9083 6169 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-13 9085 6170 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE RO-26-2853 9086 6171 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE BMS-345541 BMS-345541 9087 6172 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE SULFISOXAZOLE SULFISOXAZOLE 9088 6173 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE THERAPEUTIC TUMOR INFILTRATING LYMPHOCYTES 27959684 9089 6174 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE RG7686 9090 6175 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ACEPROMETAZINE ACEPROMETAZINE 9091 6176 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME propylthiouracil PROPYLTHIOURACIL 9092 6177 BAZ2B 29994 NA SR-2640 SR-2640 9094 6178 VEGFC 7424 GROWTH FACTOR, TRANSPORTER, DRUGGABLE GENOME bevacizumab BEVACIZUMAB 20124951 9096 6179 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME modulator CHEMBL940 GABAPENTIN 9097 6180 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650496 9098 6181 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE FF-284 26438159 9099 6182 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 178101884 GSK-690693 9100 6183 GBA 2629 DRUGGABLE GENOME, ENZYME SJ000170251 CHEMBL603154 9101 6184 TUBA3D 113457 DRUGGABLE GENOME CHEMBL2105643 FOSBRETABULIN TROMETHAMINE 9102 6185 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 381118865 9104 6186 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME TCMDC-124266 CHEMBL124006 9106 6187 RGS4 5999 DRUGGABLE GENOME perphenazine PERPHENAZINE 9107 6188 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL931 HALOTHANE 9108 6189 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE RHGH 7762644 9109 6190 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200363 PENBUTOLOL SULFATE 9111 6191 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1201731 NEBIVOLOL HYDROCHLORIDE 9112 6192 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME inhibitor 404859088 9115 6193 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ARASERTACONAZOLE ARASERTACONAZOLE 9116 6194 EEF1A1 1915 TRANSCRIPTION FACTOR SPARSOMYCIN SPARSOMYCIN 20118940 9117 6195 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-124176 CHEMBL588038 9118 6196 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist 135650918 9119 6197 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PATULIN PATULIN 9120 6198 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heteroaryl-carboxamide derivative 10 9121 6199 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE GSK1325756 DANIRIXIN 9122 6200 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME BI 860585 9124 6201 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL2105741 TRAMETINIB DIMETHYL SULFOXIDE 9125 6202 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZK-159222 CHEMBL2112314 20883026 9127 6203 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE Ibrolipim IBROLIPIM 9131 6204 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME L-701324 CHEMBL31741 9132 6205 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CI-1040 CI-1040 20538618,19915144,19018267 9133 6206 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHOTREXATE METHOTREXATE 22931300 9134 6207 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE gemcitabine GEMCITABINE 31616045 9136 6208 MGLL 11343 DRUGGABLE GENOME, ENZYME Azetidine-benzoxazin-3(4H)-one derivative 2 9137 6209 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRELANSERIN TRELANSERIN 9138 6210 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME HARMINE HARMINE 22998443 9139 6211 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-61836 CHEMBL521171 9140 6212 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MALTOTRIOSE MALTOTRIOSE 9141 6213 IGFBP1 3484 DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 7683312,1714534 9142 6214 ACACA 31 ENZYME, DRUGGABLE GENOME inhibitor 252827541 9143 6215 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-133896 CHEMBL512908 9145 6216 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2- (2,6-DIMETHOXYPHENOXYETHYL)AMINOMETHYL-1,4-BENZODIOXANE HYDROCHLORIDE (WB 4101) 2- (2,6-DIMETHOXYPHENOXYETHYL)AMINOMETHYL-1,4-BENZODIOXANE HYDROCHLORIDE (WB 4101) 9147 6217 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BN-OD-026 9148 6218 ATAD5 79915 NA OUABAIN OUABAIN 9150 6219 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME BALSALAZIDE BALSALAZIDE 9151 6220 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 249565724 9152 6221 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Olenolic acid acetate derivative 1 9154 6222 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DIOTYROSINE DIOTYROSINE 9155 6223 HLA-DRB5 3127 DRUGGABLE GENOME, CLINICALLY ACTIONABLE amoxicillin AMOXICILLIN 10535882 9156 6224 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 223366077 RGB-286638 9158 6225 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE ARQ 751 9159 6226 ALOX15B 247 DRUGGABLE GENOME, ENZYME HEXACHLOROPHENE HEXACHLOROPHENE 9161 6227 VKORC1 79001 DRUGGABLE GENOME, ENZYME inhibitor 178103444 PHENINDIONE 9162 6228 PRDX5 25824 ENZYME 2-(2-HYDROXYBENZYL)PHENOL CHEMBL148831 26492576 9163 6229 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR 7-O-METHYLCRYPTOCHINONE A 7-O-METHYLCRYPTOCHINONE A 25127166 9164 6230 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124240 CHEMBL582764 9165 6231 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME P-BCMA-101 9166 6232 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL TRIAZOLAM TRIAZOLAM 9170 6233 SMN2 6607 DRUGGABLE GENOME 2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE CHEMBL412603 9171 6234 F5 2153 DRUGGABLE GENOME Drotrecogin alfa 9172 6235 ALOX15B 247 DRUGGABLE GENOME, ENZYME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 9174 6236 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL FLURAZEPAM FLURAZEPAM 9175 6237 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200492 NEFAZODONE HYDROCHLORIDE 9176 6238 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AV-412 MP-412 17888033,19459856 9178 6239 TARDBP 23435 TUMOR SUPPRESSOR DNDI1417411 CHEMBL1445650 9179 6240 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650307 9180 6241 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE BSO 15127200 9181 6242 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME IPRIFLAVONE IPRIFLAVONE 9183 6243 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Anti-CD19/BCMA CAR-T cells 9184 6244 IFNG 3458 DRUGGABLE GENOME METHYLPREDNISOLONE METHYLPREDNISOLONE 9396353 9185 6245 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING CUDC-101 CUDC-101 9188 6246 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HYDRASTININE HYDRASTININE 9190 6247 FGA 2243 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, FIBRINOGEN ALFIMEPRASE ALFIMEPRASE 9192 6248 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PLUMBAGIN PLUMBAGIN 9194 6249 CDKN2B 1030 CLINICALLY ACTIONABLE, KINASE PALBOCICLIB PALBOCICLIB 23898052 9195 6250 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 249565824 9196 6251 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 178102309 PICTILISIB 9198 6252 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GW843682X GW843682X 9199 6253 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201731 NEBIVOLOL HYDROCHLORIDE 9200 6254 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CEFPODOXIME PROXETIL CEFPODOXIME PROXETIL 9201 6255 PDE7A 5150 ENZYME, DRUGGABLE GENOME DYPHYLLINE DYPHYLLINE 9206 6256 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE BMS-708163 AVAGACESTAT 9207 6257 TNFRSF11A 8792 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE 178101759 9208 6258 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE N/A 26711002,10086740,26102509,26606880,9462753,26522332,21714648,26769228,25807284,8609706,21877899,11432885,24517889,15704129 9209 6259 BCL2L2 599 CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor NAVITOCLAX NAVITOCLAX 9210 6260 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER EGFR antibody 27196767 9211 6261 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AZD-1152-HQPA AZD-1152-HQPA 9212 6262 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE VATALANIB VATALANIB 9213 6263 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 3,4-DICHLOROISOCOUMARIN CHEMBL24983 9214 6264 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHIR-99021 CHIR-99021 9215 6265 IMPDH2 3615 DRUGGABLE GENOME, ENZYME MYCOPHENOLATE MOFETIL 9216 6266 DHODH 1723 DRUGGABLE GENOME, ENZYME LEFLUNOMIDE LEFLUNOMIDE 9217 6267 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX PF-06463922 LORLATINIB 28285684 9218 6268 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME AR-12 AR-12 9219 6269 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 2-ENE-VALPROATE CHEMBL117487 17566732 9220 6270 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR VEMURAFENIB VEMURAFENIB 24265155 9223 6271 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME s 1 (combination) 24923815,30858516,16115930,22490566,19530960,26794347,19473056,29845393,26099996,26216193,18299612,20819423,30114658,28614820,11895907,25677447,26265035,30723313,26804652,29239269,25410891,10803677,14635116,11156223,26846104,21498394 9225 6272 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NITROXOLINE NITROXOLINE 9226 6273 NDUFA9 4704 ENZYME inhibitor CHEMBL3545135 NV-128 9227 6274 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE IPRIFLAVONE IPRIFLAVONE 9229 6275 POLK 51426 DNA REPAIR, ENZYME PROFLAVINE PROFLAVINE 9230 6276 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ANTIVIRAL 8211145 9233 6277 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NISOLDIPINE NISOLDIPINE 9234 6278 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME MADOLIN A MADOLIN A 9236 6279 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Salicylic acid derivative 5 9237 6280 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ETHACRYNIC ACID ETHACRYNIC ACID 9238 6281 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PROTRIPTYLINE HYDROCHLORIDE PROTRIPTYLINE HYDROCHLORIDE 9240 6282 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL190 THEOPHYLLINE 9241 6283 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOLUIC ACID TOLUIC ACID 9243 6284 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIBUTYLDICHLOROSTANNANE DIBUTYLDICHLOROSTANNANE 9244 6285 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Atezolizumab ATEZOLIZUMAB 27225694 9246 6286 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR GS 6201 GS 6201 9248 6287 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE TGX-221 26137449 9249 6288 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL OXAZEPAM OXAZEPAM 9250 6289 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL2107877 BLISIBIMOD 9251 6290 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR AM-111 BRIMAPITIDE, C-TERMINAL ACID 9252 6291 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CO1686 27252416,27283993 9253 6292 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE INDOMETHACIN INDOMETHACIN 2707640 9255 6293 HMGCR 3156 ENZYME, DRUGGABLE GENOME fluvastatin FLUVASTATIN 17563401,18815589,18332269,16103896,18261733,15199031 9256 6294 PRKAB1 5564 ENZYME, KINASE, DRUGGABLE GENOME activator 252827478 9258 6295 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PKI-587 GEDATOLISIB 9263 6296 GMNN 51053 DRUGGABLE GENOME A-443654 A-443654 9265 6297 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE H2O2 18299966 9266 6298 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NSC-675972 CHEMBL1379243 9267 6299 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TCMDC-124416 CHEMBL530664 9268 6300 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE AAB-002 9269 6301 TARDBP 23435 TUMOR SUPPRESSOR SJ000260158 CHEMBL601918 9270 6302 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME TRAMADOL TRAMADOL 9271 6303 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PAPAVERINE PAPAVERINE 9272 6304 GABBR2 9568 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL448343 LESOGABERAN 9274 6305 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL861 MEPHENYTOIN 9275 6306 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL919 FOSPHENYTOIN SODIUM 9276 6307 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DOFETILIDE DOFETILIDE 22931300 9279 6308 TUBA1A 7846 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 9280 6309 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NITROXOLINE NITROXOLINE 9281 6310 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR IPI-504 RETASPIMYCIN HYDROCHLORIDE 9283 6311 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-56 9284 6312 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1131 ACITRETIN 9286 6313 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TCMDC-125813 CHEMBL580076 9287 6314 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR TOREMIFENE TOREMIFENE 12476040 9289 6315 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE Gilteritinib GILTERITINIB 9290 6316 HTT 3064 DRUGGABLE GENOME MMV009085 CHEMBL581225 9291 6317 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SJ000044511 CHEMBL592124 9292 6318 TH 7054 ENZYME, DRUGGABLE GENOME SERTRALINE HYDROCHLORIDE 8629887 9293 6319 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ADIPHENINE ADIPHENINE 9295 6320 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650286 9297 6321 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SLAZINIC ACID SLAZINIC ACID 9299 6322 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE LY3300054 LODAPOLIMAB 9300 6323 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER RITONAVIR RITONAVIR 17664327 9302 6324 MTRF1L 54516 NA antidepressants 9303 6325 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUTICASONE FUROATE 9305 6326 UGT1A7 54577 DRUGGABLE GENOME, ENZYME allopurinol ALLOPURINOL 27798726 9306 6327 PSMB3 5691 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 9307 6328 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2-CHLORO-ADENOSINETRIPHOSPHATE CHEMBL1368696 9309 6329 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-1852 CHEMBL533293 9312 6330 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 328083499 SNS-314 9316 6331 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1200430 ESTRADIOL ACETATE 9318 6332 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE (20S,21S)-7-CYCLOHEXYLFLUOROCAMPTOTHECIN (20S,21S)-7-CYCLOHEXYLFLUOROCAMPTOTHECIN 24069881 9321 6333 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL107367 FARGLITAZAR 9322 6334 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DACTINOMYCIN DACTINOMYCIN 9324 6335 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUMETHASONE PIVALATE 9325 6336 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TANNIC ACID TANNIC ACID 9326 6337 PRKAB1 5564 ENZYME, KINASE, DRUGGABLE GENOME PROGESTERONE PROGESTERONE 16020477 9327 6338 FTH1 2495 NA Ferritarg P 9330 6339 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102413 9331 6340 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651503 9332 6341 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LY-255283 LY-255283 9333 6342 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BYL719 ALPELISIB 9334 6343 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 375973268 9335 6344 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME AZAKENPAULLONE AZAKENPAULLONE 9337 6345 F12 2161 DRUGGABLE GENOME, ENZYME, PROTEASE ANTITHROMBIN 9338 6346 BAZ2B 29994 NA GNF-PF-3237 CHEMBL602206 9339 6347 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR STF-62247 18769110,18598947 9340 6348 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE CUDC-101 CUDC-101 9341 6349 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AZETIDINE-2,4-DICARBOXYLIC ACID 9345 6350 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-1656 CHEMBL579028 9347 6351 PREP 5550 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 405560408 9348 6352 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER prednisolone PREDNISOLONE 14583680,25582575 9349 6353 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor BYL719 ALPELISIB 9350 6354 AKR1B1 231 DRUGGABLE GENOME, ENZYME Epalrestat EPALRESTAT 9352 6355 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL3187723 BINIMETINIB 9354 6356 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545133 JNJ-26483327 9355 6357 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 404859065 9356 6358 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE WISTIN WISTIN 9357 6359 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER IL-12 16751417 9359 6360 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 223366033 9361 6361 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 178102837 9363 6362 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ISOVELLERAL ISOVELLERAL 9364 6363 PYGL 5836 DRUGGABLE GENOME, ENZYME methotrexate METHOTREXATE 23007406 9365 6364 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL79 LIDOCAINE 9367 6365 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103666 METHYLPREDNISOLONE 9368 6366 SMARCA4 6597 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING PALBOCICLIB PALBOCICLIB 30718512,30718506 9370 6367 GFRA1 2674 KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE 178101552 9371 6368 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor GDC-0032 TASELISIB 9373 6369 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE MPA PROGESTERONE 7872957 9375 6370 ATXN2 6311 NA PIPLARTINE PIPLARTINE 9378 6371 HSF1 3297 TRANSCRIPTION FACTOR, DNA REPAIR CYCLOHEXIMIDE CYCLOHEXIMIDE 9379 6372 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MK2206 MK-2206 21289267 9380 6373 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUFURALOL BUFURALOL 2903243 9384 6374 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ANTIOXIDANT 16139439 9385 6375 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor BEZ235 DACTOLISIB 9389 6376 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DISULFOTON DISULFOTON 9390 6377 COL1A1 1277 CLINICALLY ACTIONABLE, DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 9391 6378 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CUCURBITACIN B CUCURBITACIN B 9392 6379 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DNDI1417309 CHEMBL1341830 9393 6380 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER valinomycin VALINOMYCIN 9394 6381 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME sorafenib SORAFENIB 28362716 9395 6382 ALDH3A1 218 DRUGGABLE GENOME, ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 9396 6383 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DUP-697 DUP-697 9398 6384 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE Deslanoside DESLANOSIDE 9399 6385 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE FIIN-01 20338520 9400 6386 XPNPEP2 7512 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252827461 9402 6387 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565827 9403 6388 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE E-10030 PEGPLERANIB SODIUM 9404 6389 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 178102626 9405 6390 ATXN2 6311 NA 1-O-ACETYLGEOPYXIN A CHEMBL1902074 9406 6391 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 249565930 9407 6392 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-17 9408 6393 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME citalopram CITALOPRAM 9409 6394 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-21 9410 6395 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR KMN-21 CHEMBL570176 19892550 9411 6396 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PI-103 PI-103 9412 6397 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor AZD8931 SAPITINIB 9414 6398 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AZOCYCLOTIN AZOCYCLOTIN 9415 6399 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor 348353622 9416 6400 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL289351 FOSBRETABULIN DISODIUM 9417 6401 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270010-Compound-Figure16-b-2 9418 6402 TH 7054 ENZYME, DRUGGABLE GENOME DEHYDROEPIANDROSTERONE PRASTERONE 8704732 9419 6403 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME MEN-10376 CHEMBL412982 9420 6404 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 8 9422 6405 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651895 9425 6406 MAPT 4137 DRUGGABLE GENOME 3-METHOXYCATECHOL 3-METHOXYCATECHOL 9426 6407 GUCY1B1 2983 DRUGGABLE GENOME activator CHEMBL136478 SODIUM NITROPRUSSIDE 9427 6408 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (-)-U-50488 (-)-U-50488 9428 6409 ATAD5 79915 NA 5-FLUOROURIDINE CHEMBL54918 9429 6410 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MEVASTATIN MEVASTATIN 9430 6411 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL679 EPINEPHRINE 9431 6412 KMO 8564 DRUGGABLE GENOME, ENZYME Cyclopropane 1-carboxylic acid derivative 1 9432 6413 NCL 4691 NA AS1411 9433 6414 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TYROSOL SINAPATE TYROSOL SINAPATE 23403296 9434 6415 SLC1A2 6506 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE inhibitor 178101134 9435 6416 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BYL719 ALPELISIB 9436 6417 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR 178100609 9437 6418 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR LIDOCAINE LIDOCAINE 16210356 9438 6419 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR IPRIFLAVONE IPRIFLAVONE 9439 6420 TRPV2 51393 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker 135652740 9441 6421 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 theophylline THEOPHYLLINE 9187528 9444 6422 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER midazolam MIDAZOLAM 9446 6423 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor REGORAFENIB REGORAFENIB 9448 6424 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DEFERASIROX DEFERASIROX 9449 6425 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME PACLITAXEL PACLITAXEL 12559175 9450 6426 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Rucaparib RUCAPARIB 28588062,26779812,27002934,27454289 9451 6427 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OXICONAZOLE NITRATE OXICONAZOLE NITRATE 9454 6428 RAB9A 9367 ENZYME, DRUGGABLE GENOME N-(3,4-DICHLOROPHENYL)BENZAMIDE CHEMBL560296 9455 6429 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FLUOXETINE FLUOXETINE 21393461 9458 6430 CAMK4 814 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ESTRADIOL BENZOATE 11588616 9459 6431 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RALOXIFENE RALOXIFENE 22931300 9460 6432 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135649983 BERAPROST 9462 6433 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178104017 MIRABEGRON 9463 6434 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR IFOSFAMIDE IFOSFAMIDE 9260581 9464 6435 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ERDAFITINIB ERDAFITINIB 26324363,31340094 9465 6436 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR KAI-9803 DELCASERTIB 9469 6437 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 rosiglitazone ROSIGLITAZONE 9470 6438 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL3545252 DOCETAXEL 9471 6439 CPB1 1360 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166875 9472 6440 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME IMMUNOCONJUGATE 7523704,10368631 9473 6441 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GEFITINIB GEFITINIB 21258250,23470965,27664271,22370314,31605797,18386816,25179728,15728811,19692680,15118125,18227510,20826716,16707605,22901364,17085664,24353160,26124334,24736073,15329413,15897572,16282176,12748244,19020901,20038723,15118073,20022809,25948633,19147750,18509184,24457318,27304188,21531810,16818686,24755888,16730237 9474 6442 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TRAMADOL TRAMADOL 9475 6443 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CODEINE CODEINE 9476 6444 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROPIOMAZINE PROPIOMAZINE 9478 6445 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ABT-414 DEPATUXIZUMAB MAFODOTIN 26846818 9479 6446 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 S-ETOMIDATE S-ETOMIDATE 9481 6447 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ISIS-104838 9482 6448 TXNRD1 7296 DRUGGABLE GENOME Terpyridineplatinum(II) complexe 2 9483 6449 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME RAFAMETINIB 9484 6450 PDE4A 5141 DRUGGABLE GENOME, ENZYME ENPROFYLLINE ENPROFYLLINE 9485 6451 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME WIN-62577 CHEMBL1256845 9487 6452 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE 178101337 9488 6453 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR LY-2090314 LY-2090314 9489 6454 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE antagonist 252166530 VENETOCLAX 9491 6455 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Pyrimidinyl compound 7 9492 6456 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME TARIQUIDAR TARIQUIDAR 20621487 9493 6457 AKR1C3 8644 ENZYME, DRUGGABLE GENOME ANDROGENS 10998348 9494 6458 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Baricitinib BARICITINIB 9495 6459 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor PANOBINOSTAT PANOBINOSTAT 9497 6460 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE (R)-MELPHALAN (R)-MELPHALAN 9498 6461 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 340590256 TRILACICLIB 9499 6462 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Tamibarotene TAMIBAROTENE 9500 6463 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100307 9501 6464 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GAMOLENIC ACID GAMOLENIC ACID 9502 6465 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 310264718 PF-03758309 9503 6466 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 354702286 9505 6467 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL113 CAFFEINE 9507 6468 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME KENPAULLONE KENPAULLONE 9508 6469 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-83217 CHEMBL120806 9509 6470 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL714 ALBUTEROL 9510 6471 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME ALN-TTR 9513 6472 BAZ2B 29994 NA 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 9514 6473 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MITOMYCIN-C 8162589 9516 6474 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL68055 ACOLBIFENE 9519 6475 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200864 9521 6476 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX N-ACETYLCOLCHINOL CHEMBL486504 9522 6477 NOS2 4843 DRUGGABLE GENOME, ENZYME inhibitor 363894143 GW-274150 9523 6478 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME blocker 135650723 NITRENDIPINE 9526 6479 MVD 4597 DRUGGABLE GENOME, ENZYME inhibitor 135649848 9527 6480 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor AZD8931 SAPITINIB 9528 6481 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Toremifene TOREMIFENE 9529 6482 POLR2A 5430 NA 3'-DCTP CHEMBL480328 20516278 9531 6483 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME IL-2 ALDESLEUKIN 10201984 9533 6484 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CAFFEIC ACID CAFFEIC ACID 9534 6485 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SSR-504734 9535 6486 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PROPRANOLOL PROPRANOLOL 9536 6487 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Folic Acid 9537 6488 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PIMOZIDE PIMOZIDE 9538 6489 ALOX15 246 ENZYME, DRUGGABLE GENOME PURPUROGALLIN PURPUROGALLIN 9540 6490 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AZD1208 26472029 9541 6491 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHLORETIN PHLORETIN 9542 6492 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor AZD8330 9543 6493 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE MILVETEROL MILVETEROL 9544 6494 COIL 8161 NA ACTINOMYCIN D 2088441 9546 6495 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL3545330 MSX-122 9549 6496 CA5A 763 ENZYME, DRUGGABLE GENOME activator 135651493 HISTAMINE 9551 6497 NME1 4830 KINASE tenofovir TENOFOVIR 9553 6498 HSPA4 3308 NA AEG-33773 9554 6499 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FPL-64176 CHEMBL93655 9556 6500 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR ECHINACEA ECHINACEA, UNSPECIFIED 9568541 9558 6501 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 9560 6502 CA9 768 DRUGGABLE GENOME, ENZYME SULFAMIDE SULFAMIDE 9561 6503 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor 178101473 9563 6504 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL431651 ENRASENTAN 9564 6505 CES2 8824 DRUGGABLE GENOME, ENZYME SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 9567 6506 ODC1 4953 DRUGGABLE GENOME, ENZYME Eflornithine EFLORNITHINE 9568 6507 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE SULFONE 9125494 9570 6508 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME HYPERICIN HYPERICIN 9574 6509 ABCB11 8647 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE lapatinib LAPATINIB 23556451 9576 6510 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME AR-42 AR-42 9577 6511 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE 4-HYDRAZINYLBENZENESULFONIC ACID CHEMBL510966 19007293 9578 6512 NDUFAF4 29078 NA inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 9579 6513 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565765 9580 6514 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PARAROSANILINE PARAROSANILINE 9581 6515 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1237102 LEVOCABASTINE HYDROCHLORIDE 9584 6516 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651236 TAPROSTENE 9585 6517 CD58 965 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE ALBUMIN ALBUMIN HUMAN 8697653 9586 6518 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER METHIMAZOLE METHIMAZOLE 7790147 9589 6519 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 9590 6520 FLCN 201163 CLINICALLY ACTIONABLE SIROLIMUS SIROLIMUS 26418749 9593 6521 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ROBINETIN ROBINETIN 9594 6522 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CYTOREDUCTIVE SURGERY 20942962 9599 6523 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417147 CHEMBL2094484 9600 6524 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIBROMOACETIC ACID TRIBROMOACETIC ACID 9601 6525 PTGS2 5743 DRUGGABLE GENOME, ENZYME capecitabine CAPECITABINE 19219602 9602 6526 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-68b 9603 6527 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NIFEDIPINE NIFEDIPINE 9604 6528 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3360203 PILARALISIB 9606 6529 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545006 PWT-33587 9607 6530 TUBB2B 347733 DRUGGABLE GENOME CHEMBL2304041 SAGOPILONE 9608 6531 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GSK610677 GSK-610677 9611 6532 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Pegamotecan PEGAMOTECAN 9613 6533 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE QUIZARTINIB QUIZARTINIB 21689725,24045550,19164557,15972446,16384925,18024392,18986703,22504184,16912224,23714533,25157968,17259998,23582185,16731599 9614 6534 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Sorafenib SORAFENIB 25363205 9615 6535 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE 178101724 9616 6536 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 252166735 9617 6537 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BACLOFEN BACLOFEN 9618 6538 HDAC11 79885 DRUGGABLE GENOME, ENZYME VORINOSTAT VORINOSTAT 9619 6539 UGCG 7357 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103853 9620 6540 PTGS2 5743 DRUGGABLE GENOME, ENZYME TOLMETIN TOLMETIN 9622 6541 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE OLODATEROL OLODATEROL 9623 6542 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE Imetelstat IMETELSTAT 9625 6543 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE 131I-radretumab 9628 6544 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 9630 6545 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TCMDC-123868 CHEMBL548615 9631 6546 TUBA4A 7277 DRUGGABLE GENOME CHEMBL2103826 DAVUNETIDE 9632 6547 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 363894197 CT-7001 9633 6548 PBRM1 55193 CLINICALLY ACTIONABLE ALPRAZOLAM ALPRAZOLAM 22137933 9635 6549 MMP15 4324 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166829 9637 6550 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GNF-PF-3148 CHEMBL81782 9639 6551 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL1116 RALOXIFENE HYDROCHLORIDE 9640 6552 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HEXACHLOROPHENE HEXACHLOROPHENE 9641 6553 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1201032 RIZATRIPTAN BENZOATE 9643 6554 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL3545274 MK-6913 9644 6555 IMPDH2 3615 DRUGGABLE GENOME, ENZYME 6-CL-PRT-BIOTIN CHEMBL1683024 21295473 9646 6556 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor IPI-926 PATIDEGIB 9647 6557 KDM4A 9682 DRUGGABLE GENOME, ENZYME TYRPHOSTIN 51 TYRPHOSTIN 51 9648 6558 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER voriconazole VORICONAZOLE 19033450 9649 6559 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AG-494 CHEMBL56731 9650 6560 APCS 325 TRANSPORTER, DRUGGABLE GENOME GSK2398852 DEZAMIZUMAB 9651 6561 MAPT 4137 DRUGGABLE GENOME OXYPHENBUTAZONE OXYPHENBUTAZONE 9652 6562 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Gedatolisib GEDATOLISIB 21325073 9653 6563 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PMID29671355-Compound-62 9654 6564 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME HYDROXYUREA HYDROXYUREA 12041671 9655 6565 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME DIFLUOROMETHYLORNITHINE 10716720 9657 6566 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE risperidone RISPERIDONE 18855532 9658 6567 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-23 9659 6568 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME MYRICETIN MYRICETIN 9660 6569 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102561 BOHEMINE 9661 6570 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-60 9662 6571 MAP3K9 4293 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, ENZYME, SERINE THREONINE KINASE CEP1347 9663 6572 TPBG 7162 CELL SURFACE, DRUGGABLE GENOME antibody 374883834 9665 6573 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 135650719 NILUTAMIDE 9666 6574 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702242 SURUFATINIB 9667 6575 LDHA 3939 DRUGGABLE GENOME ANTHRACYCLINES 3458424 9669 6576 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-117079 CHEMBL471225 9670 6577 GMNN 51053 DRUGGABLE GENOME TCMDC-125298 CHEMBL581152 9671 6578 ALOX5 240 DRUGGABLE GENOME, ENZYME ZILEUTON ZILEUTON 9672 6579 HSPA4 3308 NA TRAIL 12460647 9673 6580 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NSC-3323 CHEMBL1270169 9675 6581 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HALOPERIDOL HALOPERIDOL 9676 6582 MAPT 4137 DRUGGABLE GENOME GW282974X GW282974X 9677 6583 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 nelfinavir NELFINAVIR 9678 6584 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR YSIL6 9680 6585 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME CID 752709 CHEMBL429335 9681 6586 SMN1 6606 DRUGGABLE GENOME DNDI1416969 CHEMBL1453126 9688 6587 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CAPENSIN CAPENSIN 9689 6588 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3-METHOXYCATECHOL 3-METHOXYCATECHOL 9690 6589 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE remifentanil REMIFENTANIL 26771271 9691 6590 SMN1 6606 DRUGGABLE GENOME AG-1296 CHEMBL71191 9695 6591 BAZ2B 29994 NA NIFLUMIC ACID NIFLUMIC ACID 9701 6592 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ZM-449829 CHEMBL154580 9702 6593 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SILMITASERTIB SILMITASERTIB 9703 6594 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME SAR-566658 SAR-566658 9705 6595 ITPR1 3708 ION CHANNEL, KINASE, DRUGGABLE GENOME, TRANSPORTER antagonist 135651544 9706 6596 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2219421 RECILISIB 9707 6597 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565803 9710 6598 USP1 7398 DNA REPAIR, PROTEASE, ENZYME INAMRINONE INAMRINONE 9711 6599 COL18A1 80781 DRUGGABLE GENOME GLUTAMINE GLUTAMINE 16572858 9714 6600 CTNNA2 1496 NA Tumor necrosis factor alpha (TNF-alpha) inhibitors 27670765 9716 6601 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PREDNISOLONE PREDNISOLONE 9717 6602 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-32 9721 6603 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor AZD4547 9723 6604 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME agonist 310264755 9724 6605 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-159 CHEMBL599924 9727 6606 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 9728 6607 HNF1A 6927 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR N/A 26961851,25434466,25076298 9729 6608 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DIMETHYL GAMBOGATE DIMETHYL GAMBOGATE 9732 6609 RAB9A 9367 ENZYME, DRUGGABLE GENOME 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 9733 6610 KMO 8564 DRUGGABLE GENOME, ENZYME Isoxazoles and isoxazoline derivative 2 9734 6611 KDM4A 9682 DRUGGABLE GENOME, ENZYME ENCLOMIPHENE CITRATE ENCLOMIPHENE CITRATE 9735 6612 TPSAB1 7177 PROTEASE, DRUGGABLE GENOME, ENZYME Lactoferrin 9739 6613 PTPRM 5797 DRUGGABLE GENOME, PROTEIN PHOSPHATASE methotrexate METHOTREXATE 24583629 9740 6614 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Brompheniramine BROMPHENIRAMINE 9742 6615 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PMID27774824-Compound-Figure9Example2down 9745 6616 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Bosentan BOSENTAN 9746 6617 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE Deguelin DEGUELIN 25348016,25242579 9747 6618 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR EPOPROSTENOL EPOPROSTENOL 9748 6619 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIBEKACIN DIBEKACIN 9750 6620 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TYRPHOSTIN A9 TYRPHOSTIN A9 9752 6621 HPSE 10855 ENZYME, DRUGGABLE GENOME ASTEMIZOLE ASTEMIZOLE 23415087 9753 6622 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ADRIAMYCIN ADRIAMYCIN 9494516 9755 6623 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 348353622 9756 6624 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE REC-02 9757 6625 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME BMS-387032 BMS-387032 9758 6626 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 nabumetone NABUMETONE 19923256 9759 6627 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TCMDC-125758 CHEMBL546797 9760 6628 PTGS2 5743 DRUGGABLE GENOME, ENZYME FLURBIPROFEN FLURBIPROFEN 9763 6629 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GNF-PF-5510 CHEMBL578741 9765 6630 GAL 51083 DRUGGABLE GENOME Selective serotonin reuptake inhibitors 9767 6631 MAP2K6 5608 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE, TUMOR SUPPRESSOR inhibitor TRAMETINIB TRAMETINIB 9768 6632 MPHOSPH8 54737 NA A-77636 HCL CHEMBL1256876 9769 6633 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SAPPANONE A TRIMETHYL ETHER SAPPANONE A TRIMETHYL ETHER 9771 6634 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME RETINOIC ACID 2119291 9772 6635 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Alvespimycin hydrochloride 9774 6636 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE clarithromycin CLARITHROMYCIN 18695978 9776 6637 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE DESMOTEPLASE DESMOTEPLASE 9777 6638 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PD-0325901 PD-0325901 26272063 9779 6639 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME PMID29130358-Compound-Figure18(14a) 9780 6640 CBL 867 KINASE, ENZYME, CLINICALLY ACTIONABLE ANTISENSE OLIGONUCLEOTIDES 8849724 9781 6641 RAB9A 9367 ENZYME, DRUGGABLE GENOME TCMDC-124307 CHEMBL546865 9782 6642 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME 7-azaindole derivative 1 9784 6643 TOP2B 7155 DRUGGABLE GENOME, ENZYME SNS-595 VOSAROXIN 9786 6644 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY SODIUM BUTYRATE 3550424 9787 6645 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL1289926 AXITINIB 9788 6646 KDM4A 9682 DRUGGABLE GENOME, ENZYME SOLYPERTINE TARTRATE SOLYPERTINE TARTRATE 9790 6647 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX MMV009085 CHEMBL581225 9791 6648 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565728 9793 6649 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL1200993 GALLAMINE TRIETHIODIDE 9796 6650 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 223366042 CAPIVASERTIB 9798 6651 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TILNOPROFEN ARBAMEL TILNOPROFEN ARBAMEL 9801 6652 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 187051777 DIFLUPREDNATE 9802 6653 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 135651389 9803 6654 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE DNDI1416917 CHEMBL1335833 9804 6655 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE LGX818 ENCORAFENIB 26577700 9805 6656 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PALBOCICLIB PALBOCICLIB 9806 6657 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME MIDAZOLAM MIDAZOLAM 9807 6658 TUBA1C 84790 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 9808 6659 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE DOVITINIB DOVITINIB 9810 6660 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 2',3'-DIHYDROXYFLAVONE CHEMBL242171 9812 6661 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME NAVITOCLAX, ABT-263 9815 6662 MGLL 11343 DRUGGABLE GENOME, ENZYME Azetidine-benzoxazin-3(4H)-one derivative 1 9816 6663 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME CNS-5161 CNS-5161 9817 6664 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE ofloxacin OFLOXACIN 9820 6665 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE MLN-8054 MLN-8054 9821 6666 HSPA4 3308 NA GOSSYPOL GOSSYPOL 2193225 9823 6667 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CETUXIMAB CETUXIMAB 26812186,19075190,19255327,22734028,23182985,21228335,17384584,26623049,2278970,19114683,21398618,20921465,18316791,19679400,18794081,21975775,16361624,16618717,19773371,26371285,24558511,3122217,16434492,19018267,20921462,25157968,12460918,20978259,22407852,22392911,23406027 9824 6668 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL2105395 OSPEMIFENE 9825 6669 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR 3',4'-DIHYDROXYFLAVONE CHEMBL222556 9826 6670 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649995 BIMATOPROST 9827 6671 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RS-23597-190 CHEMBL83954 9828 6672 PAH 5053 DRUGGABLE GENOME, ENZYME activator CHEMBL1201775 SAPROPTERIN DIHYDROCHLORIDE 9830 6673 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DOX 15659049 9831 6674 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DEPHOSTATIN DEPHOSTATIN 9832 6675 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417080 CHEMBL1498652 9834 6676 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR avatrombopag AVATROMBOPAG 9839 6677 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME LINIFANIB LINIFANIB 9840 6678 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DITHIANON DITHIANON 9842 6679 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201765 FESOTERODINE FUMARATE 9843 6680 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME Benzoheterocyclic compound 1 9844 6681 MBP 4155 CELL SURFACE BIOFLAVONOID 9482255 9847 6682 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME METHYLENE BLUE METHYLENE BLUE 9848 6683 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE TCDD 12883080 9849 6684 PDE5A 8654 ENZYME, DRUGGABLE GENOME PENTOXIFYLLINE PENTOXIFYLLINE 9852 6685 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ATRACURIUM BESYLATE ATRACURIUM BESYLATE 9853 6686 ADH1B 125 DRUGGABLE GENOME, ENZYME FOMEPIZOLE FOMEPIZOLE 9855 6687 PTGS2 5743 DRUGGABLE GENOME, ENZYME FLURBIPROFEN FLURBIPROFEN 9856 6688 KAT8 84148 ENZYME inhibitor 187051791 9857 6689 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE INCB40093 9858 6690 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 249565632 AT-9283 9859 6691 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2109390 MAB-425 9861 6692 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING METHIMAZOLE METHIMAZOLE 9862 6693 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32g 9864 6694 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 223366185 9865 6695 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR GNF-PF-3037 CHEMBL600336 9868 6696 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIMETHOMORPH DIMETHOMORPH 9869 6697 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 252166689 9870 6698 PDE10A 10846 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL932 DIPYRIDAMOLE 9871 6699 CBX1 10951 NA GR-127935 GR-127935 9872 6700 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ABAMECTIN ABAMECTIN 9873 6701 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-640558 CHEMBL1288281 21074425 9874 6702 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IRIGENOL IRIGENOL 9875 6703 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE ILORASERTIB ILORASERTIB 9877 6704 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE fenofibrate FENOFIBRATE 19207029 9878 6705 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BERGAPTEN BERGAPTEN 9879 6706 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102689 9882 6707 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 178102620 9883 6708 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER FENRETINIDE FENRETINIDE 9886 6709 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ENDRIN ENDRIN 9887 6710 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 9888 6711 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SULFADIAZINE, SILVER SULFADIAZINE, SILVER 9890 6712 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME Sodium phenylbutyrate 9891 6713 LGALS9 3965 DRUGGABLE GENOME, TRANSPORTER LACTOSE, ANHYDROUS LACTOSE, ANHYDROUS 21524586 9895 6714 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME AST-487 AST-487 9896 6715 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE THROMBIN THROMBIN 16720831 9897 6716 GMNN 51053 DRUGGABLE GENOME TCMDC-123634 CHEMBL530499 9898 6717 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL288441 BOSUTINIB 9899 6718 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TCMDC-124063 CHEMBL534535 9900 6719 SMN2 6607 DRUGGABLE GENOME BIOCHANIN BIOCHANIN 9903 6720 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME 3,4-methylenedioxymethamphetamine 28117133,17638512,11470993 9907 6721 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1549 HYDROCORTISONE CYPIONATE 9908 6722 MPHOSPH8 54737 NA GALLAMINE GALLAMINE 9910 6723 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BENZAMIL BENZAMIL 9911 6724 ATAD5 79915 NA CYCLOHEXIMIDE CYCLOHEXIMIDE 9912 6725 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL27759 ENTINOSTAT 9913 6726 PHB2 11331 CELL SURFACE STEROID HORMONE 10850416 9914 6727 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650789 PAXILLINE 9915 6728 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXAZEPAM OXAZEPAM 9917 6729 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651281 TRIPROLIDINE 9918 6730 CD14 929 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME IC14 IC14 9920 6731 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME OXAZEPAM OXAZEPAM 9922 6732 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL52885 ENMD-981693 9923 6733 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME ANTITHROMBIN 9924 6734 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME tamoxifen TAMOXIFEN 9926 6735 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 354702284 9927 6736 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME ESTRADIOL BENZOATE 10211766 9930 6737 POLB 5423 DNA REPAIR, DRUGGABLE GENOME AG-538 CHEMBL56393 9931 6738 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Reteplase RETEPLASE 9934 6739 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE MICELLAR PACLITAXEL 10620631 9936 6740 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 404859006 VOXELOTOR 9937 6741 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL403989 TG100-801 9938 6742 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor XL-765 VOXTALISIB 9941 6743 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MEPHENTERMINE MEPHENTERMINE 9942 6744 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Cytarabine CYTARABINE 9945 6745 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Phenylpyrrolidinone derivative 1 9946 6746 CXCL8 3576 DRUGGABLE GENOME Ibuprofen IBUPROFEN 9947 6747 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 4-Carboxamido-isoindolinone derivative 2 9948 6748 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 178102646 9949 6749 POLB 5423 DNA REPAIR, DRUGGABLE GENOME PENTAMIDINE ISETHIONATE PENTAMIDINE ISETHIONATE 9952 6750 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BENZETHONIUM BENZETHONIUM 9955 6751 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR antagonist 135650608 MIFEPRISTONE 9956 6752 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR MPC-3100 9957 6753 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MODAFINIL MODAFINIL 10820139 9960 6754 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AEZS-112, ZEN-012 9961 6755 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178101860 9964 6756 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Avatrombopag AVATROMBOPAG 9965 6757 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651873 9967 6758 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CEP-11981 CEP-11981 22148921 9968 6759 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CHIR-99021 CHIR-99021 9969 6760 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE chlorpropamide CHLORPROPAMIDE 9970 6761 RPS6KA5 9252 DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 9971 6762 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL1721885 SU-014813 9972 6763 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-24047 CHEMBL1288013 9973 6764 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GUAIAZULENE GUAIAZULEN 9974 6765 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565621 MILCICLIB 9976 6766 IMPDH2 3615 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1456 MYCOPHENOLATE MOFETIL 9977 6767 PTGS1 5742 ENZYME, DRUGGABLE GENOME BALSALAZIDE BALSALAZIDE 9978 6768 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FENTICLOR FENTICLOR 9979 6769 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME NSC-66209 CHEMBL175266 9980 6770 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Dexbrompheniramine DEXBROMPHENIRAMINE 9983 6771 PRMT1 3276 ENZYME, METHYL TRANSFERASE FURAMIDINE FURAMIDINE 24564570 9984 6772 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE Quinazoline derivative 9 9985 6773 NDUFS4 4724 ENZYME inhibitor CHEMBL3545320 ME-344 9987 6774 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME PYRIDINE-2,4-DICARBOXYLIC ACID CHEMBL316034 9988 6775 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CEFSULODIN SODIUM CEFSULODIN SODIUM 9990 6776 SLC1A3 6507 TRANSPORTER, DRUGGABLE GENOME, CELL SURFACE 178101410 9991 6777 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME IMATINIB IMATINIB 22148584,24681986 9993 6778 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE BYL719 ALPELISIB 28119489 9994 6779 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NANAOMYCIN NANAOMYCIN 9995 6780 PTGES 9536 DRUGGABLE GENOME, ENZYME Imidazopyridine derivative 6 9997 6781 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ixabepilone IXABEPILONE 9999 6782 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TALMAPIMOD TALMAPIMOD 19195885 10000 6783 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PYROGALLOL PYROGALLOL 10001 6784 TXNRD1 7296 DRUGGABLE GENOME Fotemustine FOTEMUSTINE 10002 6785 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 178102681 WORTMANNIN 10003 6786 POLI 11201 DNA REPAIR HYCANTHONE HYCANTHONE 10004 6787 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME BETA-LAPACHONE LAPACHONE 10005 6788 NOS1 4842 DRUGGABLE GENOME, ENZYME RETINOIC ACID 9635256 10006 6789 PSMC2 5701 PROTEASE, TRANSCRIPTION FACTOR BORTEZOMIB BORTEZOMIB 24524217 10007 6790 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650684 NALOXONE 10009 6791 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GDC-0068 IPATASERTIB 10010 6792 CXCL8 3576 DRUGGABLE GENOME CI-1033 CANERTINIB 15956251 10011 6793 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR BBI-6000 10012 6794 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9409892, 148 10016 6795 ABAT 18 DRUGGABLE GENOME, ENZYME valproic acid 23407051 10017 6796 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ONONIN ONONIN 10019 6797 ALOX15 246 ENZYME, DRUGGABLE GENOME BITHIONOL BITHIONOL 10020 6798 ATXN2 6311 NA SJ000001516 CHEMBL592316 10022 6799 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TROPISETRON TROPISETRON 9826103 10023 6800 PTGS2 5743 DRUGGABLE GENOME, ENZYME CARPROFEN CARPROFEN 10025 6801 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE amlodipine AMLODIPINE 17178265 10028 6802 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SAPPANONE A DIMETHYL ETHER SAPPANONE A DIMETHYL ETHER 10031 6803 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1683 HYDROCORTISONE BUTYRATE 10033 6804 MAPT 4137 DRUGGABLE GENOME SANGUINARIUM CHLORIDE SANGUINARIUM CHLORIDE 10035 6805 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DAUNORUBICIN DAUNORUBICIN 10038 6806 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR BETA-LAPACHONE LAPACHONE 10039 6807 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 10040 6808 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651794 10041 6809 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Mequitazine MEQUITAZINE 10043 6810 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR MEDICATION 15488477 10045 6811 APH1B 83464 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL463981 BEGACESTAT 10046 6812 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL52885 ENMD-981693 10048 6813 NAMPT 10135 DRUGGABLE GENOME GMX1777 TEGLARINAD CHLORIDE 10049 6814 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME AG-528 CHEMBL56542 10050 6815 CXCL8 3576 DRUGGABLE GENOME ALPHA INTERFERON CETUXIMAB 10614716 10051 6816 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME N/A 10053 6817 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Tarizine derivative 1 10054 6818 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME BMS-387032 BMS-387032 10055 6819 RPS6KA6 27330 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME inhibitor 249565632 AT-9283 10056 6820 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BUTANOIC ACID BUTANOIC ACID 19053749 10057 6821 SPG7 6687 PROTEASE, ENZYME docetaxel DOCETAXEL 20038957 10058 6822 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-2905 CHEMBL582694 10059 6823 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TERAZOSIN TERAZOSIN 22931300 10060 6824 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE CEFUROXIME SODIUM CEFUROXIME SODIUM 10061 6825 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR TAMOXIFEN TAMOXIFEN 8019941 10063 6826 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE modulator CHEMBL1738889 ENOBOSARM 10064 6827 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102762 10065 6828 OASL 8638 NA peginterferon alfa-2b 21993426 10070 6829 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PREDNICARBATE PREDNICARBATE 10073 6830 ATXN2 6311 NA 4-HYDROXYDERRICIN CHEMBL458094 10076 6831 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 178102666 10077 6832 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Influenza vaccines 11756990 10078 6833 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME PURPURIN PURPURIN 10079 6834 DIO1 1733 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1518 PROPYLTHIOURACIL 10081 6835 USP1 7398 DNA REPAIR, PROTEASE, ENZYME THONZONIUM THONZONIUM 10084 6836 CARM1 10498 ENZYME, METHYL TRANSFERASE, DRUGGABLE GENOME inhibitor 336446915 10086 6837 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200472 QUAZEPAM 10088 6838 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE NAFTIFINE HYDROCHLORIDE NAFTIFINE HYDROCHLORIDE 10089 6839 BAP1 8314 PROTEASE, TUMOR SUPPRESSOR, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE VALPROIC ACID 22038994 10092 6840 KLC3 147700 NA gemcitabine GEMCITABINE 10093 6841 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DNDI1417234 CHEMBL2094549 10094 6842 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE IFN 11352647 10095 6843 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL580 LORAZEPAM 10096 6844 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE LAS38096 CHEMBL375293 10097 6845 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE E7046 10098 6846 CYP27A1 1593 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 inhibitor 252827509 10099 6847 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR GEFITINIB GEFITINIB 26124204 10100 6848 BAZ2B 29994 NA TRYPTOPHAN TRYPTOPHAN 10101 6849 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE paclitaxel PACLITAXEL 21151855,24599932 10102 6850 HLA-E 3133 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE glucocorticoids 10103 6851 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651136 10104 6852 ATAD5 79915 NA GALANGIN GALANGIN 10105 6853 NDUFAB1 4706 NA inhibitor CHEMBL3545320 ME-344 10106 6854 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OXYMETAZOLINE OXYMETAZOLINE 10108 6855 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME RHEIN RHEIN 10109 6856 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 tacrolimus TACROLIMUS 29318894 10110 6857 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR STAUROSPORINE STAUROSPORINE 7588324 10112 6858 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 178100874 10115 6859 PTGS2 5743 DRUGGABLE GENOME, ENZYME meloxicam MELOXICAM 19602986 10116 6860 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE GLUCOCORTICOID 2973444 10117 6861 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME GENTAMICIN GENTAMICIN 15736857 10118 6862 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME inhibitor 252827512 CHEMBL481422 10119 6863 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DNDI1318477 CHEMBL428064 10120 6864 HEBP1 50865 DRUGGABLE GENOME Chalcone derivative 1 10122 6865 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor PCI-24781 ABEXINOSTAT 10123 6866 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor CHEMBL608533 MIDOSTAURIN 10124 6867 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CITROPTEN CITROPTEN 10125 6868 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A2 10126 6869 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 252827493 10127 6870 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE CISPLATIN CISPLATIN 23390248 10130 6871 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE TCMDC-125528 CHEMBL375673 10131 6872 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Cetuximab CETUXIMAB 26715098,26666244,25714871,26341921,27458141,28280091,25838391,24304820,18202412,28632865,27312529,20570890,27002107,28179366,25605843,19064407 10132 6873 ALOX15B 247 DRUGGABLE GENOME, ENZYME TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 10134 6874 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 223366125 TASELISIB 10135 6875 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 4-IMIDAZOLEACRYLIC ACID CHEMBL1236602 10136 6876 CCNG1 900 KINASE MX-DNG1 10137 6877 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE DIGOXIN DIGOXIN 10139 6878 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ERLOTINIB ERLOTINIB 10141 6879 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER inhibitor 252827420 10142 6880 KCNF1 3754 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107762 NERISPIRDINE 10143 6881 PTGS2 5743 DRUGGABLE GENOME, ENZYME Meloxicam MELOXICAM 10144 6882 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 7,12-DIMETHYL-BENZO[A]ANTHRACENE CHEMBL329673 10146 6883 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME LINIFANIB LINIFANIB 10147 6884 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Benzene sulfonamide derivative 12 10148 6885 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CHEMBL1102 GLUTETHIMIDE 10149 6886 GAA 2548 DRUGGABLE GENOME, ENZYME ISOTHYMONIN ISOTHYMONIN 10150 6887 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER BISINDOLYLMALEIMIDE IX BISINDOLYLMALEIMIDE IX 25058929 10152 6888 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL231779 APIXABAN 10153 6889 MGA 23269 TRANSCRIPTION FACTOR inhibitor CHEMBL1561 MIGLITOL 10154 6890 SOD2 6648 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE heroin DIACETYLMORPHINE 29459008 10155 6891 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545308 ROCILETINIB 10157 6892 NQO2 4835 DRUGGABLE GENOME, ENZYME NSC-640558 CHEMBL1288281 21074425 10158 6893 BAZ2B 29994 NA GNF-PF-1731 CHEMBL581251 10159 6894 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME BML-210 CHEMBL324053 16921367 10163 6895 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME CANDOXATRIL CANDOXATRIL 10164 6896 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Blinatumomab BLINATUMOMAB 10165 6897 BAZ2B 29994 NA 2-HYDROXYPHENAZINE 5,10-DIOXIDE CHEMBL179611 10167 6898 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME inhibitor BORTEZOMIB BORTEZOMIB 10169 6899 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE Selumetinib SELUMETINIB 27821489 10174 6900 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ALPRAZOLAM ALPRAZOLAM 22137933 10176 6901 VKORC1L1 154807 DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 10177 6902 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 404859105 10179 6903 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR RETINYL PALMITATE 17377406 10181 6904 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME FENOFIBRATE FENOFIBRATE 16316932 10182 6905 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200806 NAPROXEN SODIUM 10185 6906 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE TIVOZANIB TIVOZANIB 10186 6907 ACE2 59272 ENZYME, TRANSPORTER, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, CELL SURFACE, PROTEASE inhibitor 223366196 ORE-1001 10187 6908 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545250 GSK-2269557 10188 6909 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Candesartan CANDESARTAN 10189 6910 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-124557 CHEMBL530682 10190 6911 NDUFB1 4707 ENZYME inhibitor CHEMBL3545320 ME-344 10191 6912 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme2WO2012/098065upper 10194 6913 CBX1 10951 NA GNF-PF-5510 CHEMBL578741 10195 6914 LIPG 9388 DRUGGABLE GENOME, ENZYME, LIPASE, CELL SURFACE, PHOSPHOLIPASE GSK-264220A 10196 6915 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR METHYLTESTOSTERONE METHYLTESTOSTERONE 10198 6916 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor SOPHORETIN QUERCETIN 10199 6917 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1200323 LABETALOL HYDROCHLORIDE 10200 6918 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME DNDI1417457 CHEMBL1530911 10201 6919 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 381118834 10202 6920 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME TAMATINIB R-406 10203 6921 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1752 DYPHYLLINE 10204 6922 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TEMSIROLIMUS TEMSIROLIMUS 10205 6923 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 thioridazine THIORIDAZINE 19923256 10207 6924 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor MOTESANIB MOTESANIB 10209 6925 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650857 PROPANTHELINE 10210 6926 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SULFORAPHANE SULFORAPHANE 20304643 10211 6927 HMOX1 3162 ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE ZNCL2 9175711 10214 6928 ALOX5 240 DRUGGABLE GENOME, ENZYME inhibitor 375973266 10216 6929 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE SPC5001 10217 6930 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[4,3-h]quinazoline-3-carboxamide derivative 1 10218 6931 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL932 DIPYRIDAMOLE 10219 6932 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME Avastin+/-Tarceva 10220 6933 RAB9A 9367 ENZYME, DRUGGABLE GENOME IPRIFLAVONE IPRIFLAVONE 10221 6934 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BOSENTAN BOSENTAN 10222 6935 NEDD8 4738 ENZYME MLN4924 10226 6936 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FENOLDOPAM BROMIDE FENOLDOPAM BROMIDE 10227 6937 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Gantenerumab GANTENERUMAB 10228 6938 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102599 10229 6939 ALOX15 246 ENZYME, DRUGGABLE GENOME NSC-172033 CHEMBL238624 10230 6940 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RO-046790 CHEMBL433461 10231 6941 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME U-50488 U-50488 METHANE SULFONATE 10233 6942 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ribociclib RIBOCICLIB 10234 6943 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 10235 6944 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TD-8954 TAK-954 10238 6945 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE PF-562271 PF-00562271 10239 6946 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Vinorelbine VINORELBINE 26801247 10240 6947 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist 381745014 TALADEGIB 10242 6948 NDUFA5 4698 ENZYME inhibitor CHEMBL3545320 ME-344 10243 6949 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CAPSAICIN CAPSAICIN 10246 6950 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING DFMO 9950818 10248 6951 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650383 IMIGLITAZAR 10250 6952 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME WITHAFERIN A WITHAFERIN A 24079846 10251 6953 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SNS-314 SNS-314 10252 6954 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME CIGB-M3 10253 6955 MAP2K3 5606 KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE inhibitor AZD6244 SELUMETINIB 10255 6956 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL activator 135651219 SURAMIN 10256 6957 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-11437 CHEMBL1814509 10257 6958 ABHD6 57406 PHOSPHOLIPASE, ENZYME inhibitor 178101972 10261 6959 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HYDROCOTARNINE HYDROCOTARNINE 10262 6960 ALOX15 246 ENZYME, DRUGGABLE GENOME CATECHIN CATECHIN 10264 6961 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYTARABINE CYTARABINE 21343560 10265 6962 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CXB909 10266 6963 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME THONZONIUM BROMIDE THONZONIUM BROMIDE 10268 6964 BAZ2B 29994 NA SJ000032153 CHEMBL600862 10269 6965 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE VU001171 CHEMBL515763 10270 6966 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX antagonist 135649903 10271 6967 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 3-HYDROXYEVODIAMINE CHEMBL2171793 22867019 10274 6968 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE blocker 178101015 10275 6969 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 178102620 10276 6970 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE JNJ-7706621 JNJ-7706621 10277 6971 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DESLORATADINE DESLORATADINE 10278 6972 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 10280 6973 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ISIS 3521 11723237,11906253 10281 6974 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE CLOCINNAMOX CLOCINNAMOX 17004724 10282 6975 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200330 PILOCARPINE HYDROCHLORIDE 10283 6976 KDM4A 9682 DRUGGABLE GENOME, ENZYME TENOXICAM TENOXICAM 10284 6977 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME VEDOLIZUMAB VEDOLIZUMAB 10285 6978 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DIETHYL-2-UNDECYLIDENEMALONATE CHEMBL1797707 21292492 10287 6979 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 381118808 PARSACLISIB 10290 6980 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774824-Compound-Figure8Example99 10291 6981 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor RAF265 RAF-265 10292 6982 ATAD5 79915 NA TCMDC-123770 CHEMBL533529 10293 6983 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR METHYLENE BLUE METHYLENE BLUE 10294 6984 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 1245272 CHEMBL408850 10295 6985 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1946170 REGORAFENIB 10297 6986 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Cetuximab CETUXIMAB 10299 6987 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME palonosetron PALONOSETRON 10304 6988 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AM-281 CHEMBL476833 10305 6989 TUSC2 11334 NA CNVN-202 10307 6990 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 328083526 CITARINOSTAT 10310 6991 TUBB4B 10383 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 10311 6992 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE LY3039478 CRENIGACESTAT 10312 6993 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3301609 TOREFORANT 10313 6994 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR BORTEZOMIB BORTEZOMIB 15657181 10315 6995 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2009153313 10317 6996 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 etoposide ETOPOSIDE 10318 6997 ATAD5 79915 NA MMV085203 CHEMBL586031 10320 6998 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PRACINOSTAT PRACINOSTAT 10321 6999 SMN1 6606 DRUGGABLE GENOME CID 1225609 CHEMBL444376 10323 7000 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR MACROLIDE ANTIBIOTIC 16476120 10325 7001 CBR1 873 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME doxorubicin DOXORUBICIN 21048526,19016765,19022938,19204081 10326 7002 LOXL2 4017 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 385612245 10327 7003 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME CYC-116 CYC-116 10329 7004 GMNN 51053 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 10330 7005 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor 249565629 SOTRASTAURIN 10331 7006 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME LORAZEPAM LORAZEPAM 10332 7007 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 223366122 MOMELOTINIB 10333 7008 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CINOLAZEPAM CINOLAZEPAM 10334 7009 RPS6KA6 27330 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME inhibitor 249565718 CHEMBL573107 10336 7010 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ISOETHARINE ISOETHARINE 10337 7011 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE GEFITINIB GEFITINIB 17575239 10338 7012 GSTT1 2952 DRUGGABLE GENOME imatinib IMATINIB 25188725 10339 7013 SLC1A3 6507 TRANSPORTER, DRUGGABLE GENOME, CELL SURFACE inhibitor 178101349 10342 7014 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ARN-6039 10343 7015 TSPO 706 DRUGGABLE GENOME Iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivative 3 10344 7016 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Sirolimus SIROLIMUS 18708578 10345 7017 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 381118815 10347 7018 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 16-DEHYDROPREGNENOLONE ACETATE CHEMBL1761683 10348 7019 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR LEVOTHYROXINE LEVOTHYROXINE 16075920 10350 7020 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Tafenoquine TAFENOQUINE 10355 7021 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor CHEMBL521686 OLAPARIB 10356 7022 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME AT001/r84 10359 7023 GAA 2548 DRUGGABLE GENOME, ENZYME LUTEOLIN LUTEOLIN 10360 7024 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme9EHT9851 10361 7025 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000128325 CHEMBL602718 10362 7026 GART 2618 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200373 10366 7027 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 178103824 METAPROTERENOL 10367 7028 POLI 11201 DNA REPAIR CARMINE CARMINE 10368 7029 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650557 10369 7030 ATXN2 6311 NA MEFLOQUINE HYDROCHLORIDE MEFLOQUINE HYDROCHLORIDE 10370 7031 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BLZ945 27199435 10371 7032 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME morphine MORPHINE 32432768 10373 7033 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PHENOXYBENZAMINE HYDROCHLORIDE PHENOXYBENZAMINE HYDROCHLORIDE 10374 7034 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER LEUCOVORIN LEUCOVORIN 12036927 10375 7035 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME RUTIN RUTIN 25496805 10377 7036 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor ROMIDEPSIN ROMIDEPSIN 10379 7037 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Heparin Calcium 10380 7038 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-348401 CHEMBL515505 10382 7039 PDE6A 5145 DRUGGABLE GENOME, ENZYME inhibitor 252827469 10383 7040 TAC1 6863 DRUGGABLE GENOME GP-120 10597775 10384 7041 SMN1 6606 DRUGGABLE GENOME TDR77585 CHEMBL1333386 10387 7042 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX PYRROLIDINE DITHIOCARBAMATE PYRROLIDINE DITHIOCARBAMATE 10388 7043 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200578 THEOPHYLLINE SODIUM GLYCINATE 10390 7044 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 252827520 DUBERMATINIB 10392 7045 PTGS1 5742 ENZYME, DRUGGABLE GENOME Naproxen NAPROXEN 10393 7046 ECE1 1889 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE SLV 306 10395 7047 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 10396 7048 MT1A 4489 NA arsenic trioxide 24924344 10397 7049 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIHYDROTESTOSTERONE ANDROSTANOLONE 12500968 10398 7050 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 1-AMINOBENZOTRIAZOLE CHEMBL101168 10399 7051 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME DHT ANDROSTANOLONE 15517879 10400 7052 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 223366137 10401 7053 PTGS1 5742 ENZYME, DRUGGABLE GENOME INDOMETHACIN INDOMETHACIN 10406 7054 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-N1 10407 7055 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Go 6976 16956345 10408 7056 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2,4-DINITROTOLUENE CHEMBL259865 10409 7057 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ZOLMITRIPTAN ZOLMITRIPTAN 10410 7058 ATXN2 6311 NA NSC-699479 CHEMBL1701915 10411 7059 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-56 10412 7060 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME RESVERATROL RESVERATROL 15672869 10414 7061 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME OTAMIXABAN OTAMIXABAN 10415 7062 CBX1 10951 NA TREQUINSIN TREQUINSIN 10416 7063 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Anti-CD20 CAR-T cells 10418 7064 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor 384403635 10420 7065 TGFB2 7042 GROWTH FACTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TRABEDERSEN TRABEDERSEN 10421 7066 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE ARQ092 26469692 10422 7067 PTGS1 5742 ENZYME, DRUGGABLE GENOME E163 E163 10075763 10424 7068 BHMT 635 DRUGGABLE GENOME, ENZYME CHEMBL1201130 BETAINE HYDROCHLORIDE 10427 7069 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TCDD 16598927 10428 7070 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GLABRANIN GLABRANIN 10429 7071 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ANDROGENS 8577638 10430 7072 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 385612197 10431 7073 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TELMISARTAN TELMISARTAN 10432 7074 IPO7 10527 NA MKC-1 ENMD-981693 10434 7075 SOAT1 6646 DRUGGABLE GENOME NIFEDIPINE NIFEDIPINE 3341992,2829803 10437 7076 APC 324 CLINICALLY ACTIONABLE JW67 21199802 10438 7077 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME NITRAZEPAM NITRAZEPAM 10442 7078 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Oral paclitaxel 10443 7079 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CIPROFLOXACIN CIPROFLOXACIN 15194011 10444 7080 EEF2 1938 DRUGGABLE GENOME, KINASE SS1(DSFV)-PE38 10445 7081 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME OLEIC ACID OLEIC ACID 10446 7082 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ERBB3 INHIBITOR 25952648 10447 7083 TK1 7083 ENZYME, KINASE, DRUGGABLE GENOME HQK-1004 ARGININE BUTYRATE 10448 7084 STK39 27347 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME losartan LOSARTAN 21993215 10450 7085 CXCR6 10663 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 178100558 10451 7086 ATP5F1D 513 TRANSPORTER ENFLURANE ENFLURANE 10452 7087 PRMT1 3276 ENZYME, METHYL TRANSFERASE NSC-45174 CHEMBL221047 20666457 10453 7088 PDE4D 5144 DRUGGABLE GENOME, ENZYME Oglemilast OGLEMILAST 18660832 10454 7089 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE VOLOCIXIMAB VOLOCIXIMAB 10455 7090 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE AZD-1152-HQPA AZD-1152-HQPA 10456 7091 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417420 CHEMBL1546223 10458 7092 MAPT 4137 DRUGGABLE GENOME BI-87E7 CHEMBL523200 10460 7093 EIF4E 1977 DRUGGABLE GENOME ETOPOSIDE ETOPOSIDE 11956083 10461 7094 CXCL2 2920 DRUGGABLE GENOME NEUROTROPHIC FACTOR 15194436 10462 7095 CYP27B1 1594 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 peginterferon alfa-2b 21145801 10463 7096 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME MIANSERIN MIANSERIN 10465 7097 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME thioridazine THIORIDAZINE 19604081,2007317 10467 7098 ALB 213 TRANSPORTER, DRUGGABLE GENOME Oxyphenbutazone OXYPHENBUTAZONE 10469 7099 NME1 4830 KINASE lamivudine LAMIVUDINE 10470 7100 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Inotuzumab Ozogamicin 10471 7101 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME SKF-38393 SKF-38393 10472 7102 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RO-0505124 CHEMBL1956070 16476733 10473 7103 PSMA5 5686 PROTEASE, DRUGGABLE GENOME inhibitor CARFILZOMIB CARFILZOMIB 10475 7104 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CUDC-101 CUDC-101 20388807 10476 7105 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME GATIFLOXACIN GATIFLOXACIN 10477 7106 NR5A2 2494 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 385612243 10479 7107 AKR1B1 231 DRUGGABLE GENOME, ENZYME T2c-003 10483 7108 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Cyclopenta[d]pyrimidine derivative 1 10487 7109 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CARNOSIC ACID CARNOSIC ACID 10490 7110 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR chlorthalidone CHLORTHALIDONE 10491 7111 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER morphine MORPHINE 24703092,25311385,16580900,29474345,25155932,19514130,17898703 10492 7112 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FGF-1 FIBROBLAST GROWTH FACTOR-1 15870071 10493 7113 TUBA1C 84790 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 10494 7114 POLG 5428 ENZYME KASANOSIN A KASANOSIN A 18308572 10495 7115 ABHD6 57406 PHOSPHOLIPASE, ENZYME PMID29053063-Compound-11d 10496 7116 TGFBR3 7049 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 8143777 10497 7117 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFACON-1 10498 7118 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1201159 FENTANYL HYDROCHLORIDE 10499 7119 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Insulin-lispro 10500 7120 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME CHEMBL1714 KETAMINE HYDROCHLORIDE 10503 7121 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 6 10504 7122 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE tiotropium TIOTROPIUM 19183167 10505 7123 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PD-168393 CHEMBL285063 17334377,23988354,10346932 10508 7124 PCSK6 5046 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE inhibitor 252166858 10509 7125 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CELECOXIB CELECOXIB 10510 7126 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE PD-325901 10514 7127 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 249565843 10515 7128 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 178101880 10518 7129 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BISPHENOL A BISPHENOL A 10520 7130 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-40 10521 7131 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY FDG FLUDEOXYGLUCOSE-F18 10452315 10522 7132 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 252166594 VS-5584 10523 7133 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PNU-99194A PNU-99194A 10524 7134 ADAM8 101 ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, CELL SURFACE, DRUGGABLE GENOME, PROTEASE inhibitor 252166879 10525 7135 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PENTABROMOPHENOL PENTABROMOPHENOL 10527 7136 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178104021 ACLIDINIUM 10529 7137 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 252166594 VS-5584 10530 7138 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME CITALOPRAM CITALOPRAM 10531 7139 LPAR2 9170 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135650457 10532 7140 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LESTAURTINIB LESTAURTINIB 10534 7141 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL agonist 178100898 10535 7142 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651980 10536 7143 SLC12A7 10723 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178101310 10537 7144 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 381744997 REPOTRECTINIB 10538 7145 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545050 BMS-817378 10539 7146 POLI 11201 DNA REPAIR TYRPHOSTIN 51 TYRPHOSTIN 51 10541 7147 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-3201 CHEMBL581872 10546 7148 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR THIETHYLPERAZINE THIETHYLPERAZINE 10547 7149 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051820 10548 7150 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LITHIUM LITHIUM 15475000 10549 7151 PSMC1 5700 PROTEASE inhibitor CHEMBL451887 CARFILZOMIB 10550 7152 GMNN 51053 DRUGGABLE GENOME TRYPTANTHRIN TRYPTANTHRIN 10554 7153 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ILORASERTIB ILORASERTIB 10555 7154 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor ZELBORAF ZELBORAF 10556 7155 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650563 10557 7156 NTF4 4909 GROWTH FACTOR BDNF 7552337 10558 7157 ATXN2 6311 NA AROMOLINE AROMOLINE 10559 7158 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 3 10560 7159 TDP2 51567 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 10563 7160 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME agonist CHEMBL1201568 PEGFILGRASTIM 10564 7161 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE R1678 10566 7162 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL1683544 ERIBULIN MESYLATE 10568 7163 FGFR1OP2 26127 NA brivanib BRIVANIB 20124951 10570 7164 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR tamoxifen TAMOXIFEN 17713466 10571 7165 TUBB 203068 DRUGGABLE GENOME KOS-1803 10572 7166 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 348353655 OCLACITINIB 10573 7167 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GEFITINIB GEFITINIB 10574 7168 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME OXYTETRACYCLINE OXYTETRACYCLINE 10576 7169 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 252166516 10577 7170 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE OMACETAXINE MEPESUCCINATE 19322212,22896000 10578 7171 PTGS1 5742 ENZYME, DRUGGABLE GENOME FENOPROFEN FENOPROFEN 10580 7172 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE BLU-285 AVAPRITINIB 10583 7173 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PIOGLITAZONE PIOGLITAZONE 17251278 10585 7174 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE FOLIC ACID 3479800 10586 7175 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUSPIRILENE FLUSPIRILENE 10587 7176 AQP9 366 ION CHANNEL ANDROGENS 12021052 10591 7177 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1480 FELODIPINE 10592 7178 TARDBP 23435 TUMOR SUPPRESSOR GRINIMIBINE GRINIMIBINE 10593 7179 CCL18 6362 DRUGGABLE GENOME IMMUNOMODULATORS 12161279 10594 7180 NCOA1 8648 ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX ETOPOSIDE ETOPOSIDE 10595 7181 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178102313 NERATINIB 10598 7182 RACGAP1 29127 NA RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 10599 7183 TSPO 706 DRUGGABLE GENOME Pyrazolopyrimidine acetamide analog 2 10600 7184 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SOTRASTAURIN SOTRASTAURIN 10601 7185 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 178103840 PHENELZINE 10602 7186 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE GO-6976 GO-6976 10604 7187 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME US9024044, 62 10605 7188 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL LORAZEPAM LORAZEPAM 10607 7189 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR TANNIC ACID TANNIC ACID 10608 7190 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYPERICIN HYPERICIN 17219054 10609 7191 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME LFG-316 TESIDOLUMAB 24860651 10610 7192 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME OXYTETRACYCLINE OXYTETRACYCLINE 10612 7193 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CYC-116 CYC-116 10613 7194 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102295 AFATINIB 10614 7195 GMNN 51053 DRUGGABLE GENOME CYCLOVALONE CYCLOVALONE 10615 7196 PTGES 9536 DRUGGABLE GENOME, ENZYME PMID28627961-Compound-30 10617 7197 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON BETA-1B 10618 7198 CSNK1E 1454 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 328083473 CHEMBL1951415 10619 7199 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME PMID28594589-Compound-TABLE3C12 10620 7200 AKR1C1 1645 DRUGGABLE GENOME, ENZYME HUMAN CHORIONIC GONADOTROPIN 436730 10622 7201 FZD7 8324 G PROTEIN COUPLED RECEPTOR, KINASE antagonist 381745004 10623 7202 ACAT1 38 ENZYME PMID25470667-Compound-K-604 10624 7203 TLR7 51284 DRUGGABLE GENOME agonist 178101715 LOXORIBINE 10625 7204 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178103000 MELAGATRAN 10627 7205 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DEL-22379 DEL-22379 26267534 10628 7206 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME 4-(thiazol-5-yl)-pyrimidine derivative 2 10629 7207 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NICERGOLINE NICERGOLINE 10632 7208 ATXN2 6311 NA KAMEBANIN KAMEBANIN 10635 7209 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR olaparib OLAPARIB 10636 7210 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME LITHIUM LITHIUM 12614997 10638 7211 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL403989 TG100-801 10639 7212 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3545337 C-1311 10641 7213 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX THIOMERSAL THIMEROSAL 10642 7214 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME JNK INHIBITOR VIII CHEMBL210618 10643 7215 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 340590232 BETRIXABAN 10644 7216 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-50 10645 7217 GLS 2744 ENZYME OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 10646 7218 GNA11 2767 CLINICALLY ACTIONABLE MEK INHIBITOR PD0325901 24141786 10647 7219 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1,2-DINITRO-BENZENE CHEMBL168075 10648 7220 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME ANTIESTROGENS 12782587 10649 7221 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CISPLATIN CISPLATIN 10650 7222 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME ESTAZOLAM ESTAZOLAM 22137933 10651 7223 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME S-(P-AZIDOPHENACYL)GLUTATHIONE CHEMBL1256813 10653 7224 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER H2O2 14622133,12514119 10654 7225 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME tipiracil / trifluridine 10655 7226 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHOSALONE PHOSALONE 10657 7227 TOP2B 7155 DRUGGABLE GENOME, ENZYME Cinoxacin CINOXACIN 10658 7228 CPB1 1360 DRUGGABLE GENOME, PROTEASE, ENZYME US8710232, 7 10659 7229 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BAY80-6946 COPANLISIB 10660 7230 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR S-06911 10661 7231 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME Avatrombopag AVATROMBOPAG 10663 7232 TET2 54790 CLINICALLY ACTIONABLE, ENZYME Azacitidine AZACITIDINE 25224413,21494260 10666 7233 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 6-AMINONICOTINAMIDE 6-AMINONICOTINAMIDE 10667 7234 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR IMIPRAMINE HYDROCHLORIDE IMIPRAMINE HYDROCHLORIDE 10668 7235 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE CHEMOPREVENTIVE AGENT 16041863 10670 7236 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR AR-42 AR-42 10671 7237 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME ANTI-INFLAMMATORY DRUGS 2571317 10672 7238 ALOX15B 247 DRUGGABLE GENOME, ENZYME N,N'-DIPHENYL-P-PHENYLENEDIAMINE N,N'-DIPHENYL-P-PHENYLENEDIAMINE 10674 7239 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 15 10675 7240 MPHOSPH8 54737 NA METHOCTRAMINE HYDROCHLORIDE METHOCTRAMINE HYDROCHLORIDE 10677 7241 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GW9662 CHEMBL375270 10678 7242 RAB9A 9367 ENZYME, DRUGGABLE GENOME HYDRALAZINE HYDRALAZINE 10680 7243 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE BAY-613606 CHEMBL541400 10682 7244 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AG-024322 AG-24322 10683 7245 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE STREPTOZOTOCIN STREPTOZOCIN 16954344 10687 7246 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-P4 10688 7247 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NSC-102742 CHEMBL1519374 10689 7248 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ENDO-ATROPINE ENDO-ATROPINE 22931300 10691 7249 SLC1A7 6512 TRANSPORTER, DRUGGABLE GENOME 178101255 10693 7250 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL PHENOBARBITAL PHENOBARBITAL 10694 7251 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRADIOL VALERATE ESTRADIOL VALERATE 10697 7252 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME TOZASERTIB TOZASERTIB 10698 7253 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID25656651-Compound-42 10699 7254 CXCL8 3576 DRUGGABLE GENOME HISTONE DEACETYLASE INHIBITOR 12010777 10700 7255 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NORETHINDRONE NORETHINDRONE 10703 7256 USP1 7398 DNA REPAIR, PROTEASE, ENZYME LAWSONE LAWSONE 10704 7257 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-27 10709 7258 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENZOXIQUINE BENZOXIQUINE 10710 7259 ATXN2 6311 NA L-162313 CHEMBL288174 10712 7260 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE antibody 329968449 ANDECALIXIMAB 10713 7261 NDUFA7 4701 ENZYME inhibitor CHEMBL3545320 ME-344 10714 7262 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR 1190312-92-5 10715 7263 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME GW441756X GW441756X 10717 7264 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME MEK162 BINIMETINIB 10718 7265 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178102311 GSK-461364 10722 7266 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CAMPTOTHECIN CAMPTOTHECIN 10724 7267 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME PRAZEPAM PRAZEPAM 10725 7268 ATXN2 6311 NA NICARDIPINE NICARDIPINE 10727 7269 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW643971X GW643971X 10730 7270 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME EFALIZUMAB EFALIZUMAB 10732 7271 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR ADJUVANT 15161015 10733 7272 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME activator 135651544 10735 7273 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME PF-562271 PF-00562271 10737 7274 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ARI-3037MO 10738 7275 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TRAFERMIN TRAFERMIN 10739 7276 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME Dimethoxybenzylidene-2-thio-imidazole-4-one derivative 1 10740 7277 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE Drugs For Treatment Of Tuberculosis 31648372 10741 7278 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 10742 7279 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-43 10745 7280 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME RG7625 PETESICATIB 10746 7281 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Trastuzumab TRASTUZUMAB 26432108 10748 7282 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor LY2784544 GANDOTINIB 10749 7283 CCR7 1236 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR agonist 135651670 10750 7284 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ELLAGIC ACID ELLAGIC ACID 10752 7285 BAZ2B 29994 NA CEPHALOTHIN SODIUM CEPHALOTHIN SODIUM 10753 7286 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200440 MEPIVACAINE HYDROCHLORIDE 10754 7287 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR OCTREOTIDE OCTREOTIDE 16452215 10755 7288 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME MYRICETIN MYRICETIN 10756 7289 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 135651303 10757 7290 POLI 11201 DNA REPAIR CEFIXIME CEFIXIME 10758 7291 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 867101 CHEMBL406557 10759 7292 MAPT 4137 DRUGGABLE GENOME NIFEDIPINE NIFEDIPINE 10760 7293 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 178101973 10761 7294 PLD1 5337 ENZYME, DRUGGABLE GENOME US9127005, P0L 10762 7295 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLORFENAPYR CHLORFENAPYR 10764 7296 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OLANZAPINE OLANZAPINE 10765 7297 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 354702238 MAVELERTINIB 10767 7298 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ACETOPHENAZINE ACETOPHENAZINE 17606915 10768 7299 CAT 847 ENZYME, DRUGGABLE GENOME ethanol ALCOHOL 25514903 10769 7300 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Systebryl 10770 7301 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor ENMD-2076 ENMD-2076 10771 7302 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE BFGF 15924676 10772 7303 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE carboplatin CARBOPLATIN 23963862 10775 7304 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME pioglitazone PIOGLITAZONE 12610044 10777 7305 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 252827496 10778 7306 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE (S)-THIORPHAN (S)-THIORPHAN 10779 7307 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL1200485 SORAFENIB TOSYLATE 10781 7308 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor MASITINIB MASITINIB 10782 7309 SEM1 7979 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 10783 7310 ALPL 249 ENZYME, DRUGGABLE GENOME RETINOIC ACID 10691970 10786 7311 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE DOVITINIB DOVITINIB 10788 7312 LIMK2 3985 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565831 10789 7313 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Desirudin Recombinant 10790 7314 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ISOTHYMONIN ISOTHYMONIN 10792 7315 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652136 10793 7316 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE PIPERINE PIPERINE 10794 7317 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MGAH22 MARGETUXIMAB 22129105 10795 7318 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000113972 CHEMBL591137 10796 7319 GMNN 51053 DRUGGABLE GENOME GNF-PF-4998 CHEMBL585795 10797 7320 GAA 2548 DRUGGABLE GENOME, ENZYME GNF-PF-3537 CHEMBL601110 10798 7321 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ARRY-334543 VARLITINIB 10799 7322 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR SAPPANONE A TRIMETHYL ETHER SAPPANONE A TRIMETHYL ETHER 10803 7323 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE ERLOTINIB ERLOTINIB 10805 7324 RPA1 6117 DNA REPAIR, KINASE NSC-15520 CHEMBL1765371 21459001 10806 7325 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE GLN GLUTAMINE 16898871 10807 7326 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Quinoxaline derivative 6 10808 7327 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SIDURON SIDURON 10809 7328 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DICLOFENAC SODIUM DICLOFENAC SODIUM 10811 7329 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ARS-853 26739882 10814 7330 ASNS 440 CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE ASPARAGINASE ASPARAGINASE 28069604 10817 7331 NFKBIA 4792 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME 6-METHOXYCOMAPARVIN CHEMBL401565 18088098 10819 7332 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME MELATONIN MELATONIN 15205854 10820 7333 PIEZO1 9780 ION CHANNEL, TRANSPORTER inhibitor 381118822 10821 7334 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 178103443 PEMETREXED 10822 7335 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE AT9283 AT-9283 10824 7336 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 diazepam DIAZEPAM 22641027 10826 7337 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHENYLBUTAZONE PHENYLBUTAZONE 22931300 10827 7338 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DACTOLISIB DACTOLISIB 19029981,22392911 10828 7339 SLC9A1 6548 TRANSPORTER, DRUGGABLE GENOME, EXCHANGER, CELL SURFACE CARIPORIDE CARIPORIDE 17493937 10830 7340 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-348401 CHEMBL515505 10831 7341 BMP2 650 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BUTAMBEN BUTAMBEN 22041064 10833 7342 AKR1C4 1109 DRUGGABLE GENOME, ENZYME daunorubicin DAUNORUBICIN 20837989 10834 7343 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Coagulation Factor IX 10837 7344 CCL3 6348 KINASE, DRUGGABLE GENOME Nagrestipen NAGRESTIPEN 10838 7345 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Dasatinib DASATINIB 27222538 10839 7346 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NSC-180246 CHEMBL484640 10840 7347 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Demecarium bromide 10841 7348 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-3716 CHEMBL609606 10842 7349 CBX1 10951 NA NSC-348401 CHEMBL515505 10843 7350 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR TESTOSTERONE TESTOSTERONE 9260906 10844 7351 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 178103081 PRALNACASAN 10845 7352 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 223366125 TASELISIB 10847 7353 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 223366148 TALMAPIMOD 10848 7354 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME GW441756X GW441756X 10850 7355 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MEDROXYPROGESTERONE MEDROXYPROGESTERONE ACETATE 12846422 10852 7356 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-51 10853 7357 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL3545287 LY2624803 10854 7358 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME CAR-T cells targeting BCMA 10855 7359 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor CHEMBL3545133 JNJ-26483327 10857 7360 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565843 10858 7361 TUBA3D 113457 DRUGGABLE GENOME CHEMBL2304041 SAGOPILONE 10860 7362 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE Rapamycin SIROLIMUS 10861 7363 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417614 CHEMBL1567571 10863 7364 EPRS1 2058 DRUGGABLE GENOME, ENZYME HALOFUGINONE HALOFUGINONE 10864 7365 CYP27A1 1593 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 URSODEOXYCHOLIC ACID 12011083 10867 7366 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103751 EPINASTINE 10869 7367 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME GNF-PF-3314 CHEMBL582287 10870 7368 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DIETHANOLAMINE DIETHANOLAMINE 10871 7369 RGS4 5999 DRUGGABLE GENOME CAMBINOL CAMBINOL 10872 7370 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PD-169316 PD-169316 10873 7371 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL3545295 AVE0847 10874 7372 DNER 92737 NA Isoxazole-based bicyclic compound 2 10878 7373 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-2950 CHEMBL602807 10879 7374 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ACITRETIN ACITRETIN 10882 7375 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 178100943 10883 7376 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME SP-600125 SP-600125 10884 7377 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Rucaparib RUCAPARIB 26779812 10885 7378 PSMD8 5714 NA inhibitor BORTEZOMIB BORTEZOMIB 10886 7379 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator 178103417 ENOXAPARIN 10887 7380 NECTIN4 81607 DRUGGABLE GENOME ASG-22ME ENFORTUMAB VEDOTIN 10888 7381 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME VALPROIC ACID VALPROIC ACID 18294844,16921367,25304896 10889 7382 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CUDC-907 FIMEPINOSTAT 22693356,20570890 10891 7383 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE AN-9 AN-9 8348968 10894 7384 APOA2 336 DRUGGABLE GENOME GLUCOCORTICOID 8706754 10895 7385 TUBB 203068 DRUGGABLE GENOME inhibitor 178103415 DOCETAXEL 10896 7386 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 187051839 10897 7387 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 OLEOYL DOPAMINE OLEOYL DOPAMINE 10899 7388 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 223365885 DOTHIEPIN 10902 7389 KDM5B 10765 ENZYME inhibitor 375973270 10905 7390 MAPT 4137 DRUGGABLE GENOME 2',3,4-TRIHYDROXYCHALCONE CHEMBL339587 10906 7391 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GALANGIN GALANGIN 10907 7392 MAOB 4129 DRUGGABLE GENOME, ENZYME 4-Hydroxybenzoicacid 10908 7393 NDUFA13 51079 ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545135 NV-128 10909 7394 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY IMMUNOMODULATORS 7769089 10910 7395 HSPB2 3316 KINASE PS-341 BORTEZOMIB 15004512 10911 7396 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME BMS-345541 BMS-345541 10912 7397 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IODOFORM IODOFORM 10914 7398 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CARNOSIC ACID CARNOSIC ACID 10922 7399 NAPEPLD 222236 ENZYME inhibitor 405560495 10923 7400 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 252827484 10924 7401 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1389 LEVONORGESTREL 10925 7402 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL QUAZEPAM QUAZEPAM 10926 7403 CBX1 10951 NA OMEPRAZOLE OMEPRAZOLE 10927 7404 CBX1 10951 NA ISOXANTHOPTERIN ISOXANTHOPTERIN 10928 7405 TUBB4B 10383 DRUGGABLE GENOME DOLASTATIN-10 DOLASTATIN-10 10929 7406 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Parthenolide PARTHENOLIDE 10930 7407 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE Gemfibrozil GEMFIBROZIL 10931 7408 SEM1 7979 NA inhibitor CHEMBL2103884 OPROZOMIB 10934 7409 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER anthracyclines and related substances 23441093,21900104 10936 7410 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE Venetoclax VENETOCLAX 10940 7411 TUBB2B 347733 DRUGGABLE GENOME CHEMBL492399 VERUBULIN 10942 7412 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR HORMONES 17131419 10945 7413 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME hydrochlorothiazide HYDROCHLOROTHIAZIDE 10946 7414 TOP2B 7155 DRUGGABLE GENOME, ENZYME Idarubicin IDARUBICIN 10947 7415 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1648 ISRADIPINE 10948 7416 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME lovastatin LOVASTATIN 16103896 10949 7417 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 315661202 MIVEBRESIB 10950 7418 MBNL1 4154 DRUGGABLE GENOME GNF-PF-5149 CHEMBL600309 10954 7419 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Gefitinib GEFITINIB 10958 7420 PSMA5 5686 PROTEASE, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 24524217 10959 7421 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE PROTOPORPHYRIN PROTOPORPHYRIN 9868803 10960 7422 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Actinomycines 10961 7423 PSMC2 5701 PROTEASE, TRANSCRIPTION FACTOR inhibitor CHEMBL3545432 IXAZOMIB CITRATE 10963 7424 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-30 10965 7425 IFNG 3458 DRUGGABLE GENOME PEFLOXACIN PEFLOXACIN 8673851 10966 7426 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ABBV-323 RAVAGALIMAB 10967 7427 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AC430 AC-430 10968 7428 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE 5-(N-ETHYL-N-ISOPROPYL)AMILORIDE 5-(N-ETHYL-N-ISOPROPYL)AMILORIDE 10971 7429 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TERPYRIDINE TERPYRIDINE 10972 7430 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist 178100827 PANCURONIUM 10973 7431 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SILDENAFIL SILDENAFIL 10974 7432 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE BARASERTIB BARASERTIB 10975 7433 KRT18 3875 DRUGGABLE GENOME MITOMYCIN-C 11968007 10976 7434 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL allosteric modulator 178100982 10979 7435 OASL 8638 NA ribavirin RIBAVIRIN 21993426 10980 7436 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE NSC-649410 CHEMBL177126 22921742 10982 7437 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME ENTINOSTAT ENTINOSTAT 19966789,20491440 10983 7438 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME ROTENONE ROTENONE 21875114 10984 7439 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME TRIAMTERENE TRIAMTERENE 10985 7440 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PROPRANOLOL PROPRANOLOL 10395986 10987 7441 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 381118866 10989 7442 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE INSM-18 INSM-18 10991 7443 IL1A 3552 CELL SURFACE, DRUGGABLE GENOME ABT-981 10993 7444 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 8-(P-SULFOPHENYL)THIOPHYLLINE CHEMBL8488 10994 7445 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CYCLOBENZAPRINE CYCLOBENZAPRINE 10995 7446 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR THIRAM THIRAM 10996 7447 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME 3',4'-DIMETHOXYFLAVONE 3',4'-DIMETHOXYFLAVONE 10998 7448 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL inhibitor 135651976 10999 7449 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME RUXOLITINIB RUXOLITINIB 26701727,31372595 11000 7450 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE LOMOFUNGIN LOMOFUNGIN 11001 7451 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME BACLOFEN BACLOFEN 11301212 11002 7452 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MK-1029 MK-1029 11003 7453 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor NINTEDANIB NINTEDANIB 11004 7454 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE LEOIDIN LEOIDIN 11005 7455 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME SU-6656 CHEMBL605003 11006 7456 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565788 11008 7457 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE DNDI1418024 CHEMBL1333798 11009 7458 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME cevimeline CEVIMELINE 11010 7459 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE PENTAZOCINE PENTAZOCINE 11011 7460 PGP 283871 NA ETOPOSIDE ETOPOSIDE 11012 7461 PTP4A3 11156 DRUGGABLE GENOME, PROTEIN PHOSPHATASE CETUXIMAB CETUXIMAB 23867504 11013 7462 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Venetoclax VENETOCLAX 27974663 11014 7463 CMPK1 51727 KINASE, ENZYME lamivudine LAMIVUDINE 11015 7464 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE BI-505 BI-505 11016 7465 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL GABOXADOL GABOXADOL 11017 7466 CBL 867 KINASE, ENZYME, CLINICALLY ACTIONABLE Gemcitabine GEMCITABINE 25348515 11018 7467 MAPT 4137 DRUGGABLE GENOME DEXKETOPROFEN DEXKETOPROFEN 11019 7468 PTPN6 5777 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE BDBM50054344 11020 7469 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE VS-5584 VS-5584 23270925 11021 7470 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PLUMBAGIN PLUMBAGIN 11022 7471 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE CEQ508 11024 7472 MAPT 4137 DRUGGABLE GENOME O-DEMETHYLATED ADAPALENE O-DEMETHYLATED ADAPALENE 11025 7473 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR UREA UREA 9458825 11026 7474 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor 374883861 MK-8353 11027 7475 MUC16 94025 DRUGGABLE GENOME Oregovomab OREGOVOMAB 24886523 11028 7476 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 178101743 11030 7477 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE DERMOLASTIN 11031 7478 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651193 11032 7479 PBK 55872 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, ENZYME LINIFANIB LINIFANIB 11034 7480 KCNJ3 3760 EXTERNAL SIDE OF PLASMA MEMBRANE, ION CHANNEL, DRUGGABLE GENOME activator 135652743 11035 7481 XDH 7498 DRUGGABLE GENOME, ENZYME Fused heterocyclic compound 3 11037 7482 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR OSPEMIFENE OSPEMIFENE 11038 7483 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME 6-METHOXYCOMAPARVIN 5-METHYL ETHER CHEMBL256967 18088098 11039 7484 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652108 11041 7485 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Foretinib FORETINIB 26779812 11043 7486 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE motesanib MOTESANIB 20124951 11044 7487 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NORGESTREL NORGESTREL 11045 7488 MAPT 4137 DRUGGABLE GENOME DITHIAZANINE IODIDE DITHIAZANINE IODIDE 11047 7489 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PNEUMOCOCCAL POLYSACCHARIDE VACCINE 10225849 11048 7490 KDM4A 9682 DRUGGABLE GENOME, ENZYME METHYLMALONIC ACID METHYLMALONIC ACID 11049 7491 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Erenumab ERENUMAB 11050 7492 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652215 11051 7493 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Esmolol ESMOLOL 11052 7494 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME nateglinide NATEGLINIDE 18187595 11053 7495 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENZOPHENONE BENZOPHENONE 11056 7496 PTCH1 5727 CLINICALLY ACTIONABLE, TRANSPORTER RETINOIC ACID 12455633 11057 7497 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL964 DISULFIRAM 11058 7498 PLA2G7 7941 DRUGGABLE GENOME, ENZYME inhibitor 178103948 RILAPLADIB 11059 7499 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR MEK162 BINIMETINIB 11060 7500 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME mitoxantrone MITOXANTRONE 26663398 11061 7501 IL11 3589 DRUGGABLE GENOME, KINASE, GROWTH FACTOR AZACYTIDINE AZACITIDINE 12543079 11062 7502 CDKAL1 54901 ENZYME Tumor necrosis factor alpha (TNF-alpha) inhibitors 27670765 11063 7503 CYP27B1 1594 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 tenofovir disoproxil fumarate 31619748 11064 7504 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TDR78026 CHEMBL1483413 11066 7505 POLI 11201 DNA REPAIR NSC-7387 CHEMBL119878 11067 7506 BAZ2B 29994 NA DEOXYVASICINONE DEOXYVASICINONE 11068 7507 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE GANTOFIBAN GANTOFIBAN 11070 7508 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TANNIC ACID TANNIC ACID 11071 7509 GAPDH 2597 DRUGGABLE GENOME, ENZYME NSC-228155 CHEMBL505670 11072 7510 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL2105732 LEVOMILNACIPRAN HYDROCHLORIDE 11073 7511 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE SALICYLHYDROXAMIC ACID SALICYLHYDROXAMIC ACID 11074 7512 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL2219416 NALOXEGOL OXALATE 11075 7513 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651542 11076 7514 SMN1 6606 DRUGGABLE GENOME 5,7-DIMETHOXYISOFLAVONE 5,7-DIMETHOXYISOFLAVONE 11077 7515 CSF3 1440 GROWTH FACTOR, DRUGGABLE GENOME Interleukin-3 MUPLESTIM 11078 7516 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE MONOMETHYL AURISTATIN E 18593940 11080 7517 HSPB1 3315 DRUGGABLE GENOME DICARBONODITHIOIMIDIC DIAMIDE DICARBONODITHIOIMIDIC DIAMIDE 11081 7518 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR G1T38 LEROCICLIB 11082 7519 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000124275 CHEMBL602150 11083 7520 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL16 PHENYTOIN 11085 7521 MYB 4602 CLINICALLY ACTIONABLE RETINOID 8670250 11086 7522 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-3725 CHEMBL598695 11087 7523 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME ARRY-162 BINIMETINIB 11088 7524 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-109483 CHEMBL507159 22524450 11090 7525 ATAD5 79915 NA GNF-PF-1969 CHEMBL601364 11091 7526 VASP 7408 KINASE hydrochlorothiazide HYDROCHLOROTHIAZIDE 11092 7527 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER TCMDC-124353 CHEMBL529918 11093 7528 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 1,2-DINITRO-BENZENE CHEMBL168075 11094 7529 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Zoledronate ZOLEDRONIC ACID 11097 7530 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BRIMONIDINE BRIMONIDINE 11098 7531 MGLL 11343 DRUGGABLE GENOME, ENZYME Azetidinyl-piperidine derivative 3 11099 7532 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SJ000120515 CHEMBL592314 11100 7533 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE WORTMANNIN WORTMANNIN 10559227 11102 7534 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER reserpine RESERPINE 11104 7535 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME WAY-629 CHEMBL258465 11105 7536 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417597 CHEMBL1330352 11106 7537 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME N-naphtyl-N-benzylurea derivative 1 11107 7538 CDK18 5129 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR inhibitor CHEMBL1230607 PHA-793887 11108 7539 PTGS2 5743 DRUGGABLE GENOME, ENZYME PHENYLBUTAZONE PHENYLBUTAZONE 11110 7540 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PHENYLBUTAZONE PHENYLBUTAZONE 22931300 11111 7541 NEDD4L 23327 ENZYME diuretics 18591455,21052022 11112 7542 PDE7B 27115 DRUGGABLE GENOME, ENZYME DYPHYLLINE DYPHYLLINE 11113 7543 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME BORTEZOMIB BORTEZOMIB 11114 7544 BAZ2B 29994 NA TCMDC-124518 CHEMBL527584 11115 7545 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker 135652722 TETRODOTOXIN 11117 7546 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE NYSTATIN NYSTATIN 7721938 11119 7547 PRMT6 55170 ENZYME, METHYL TRANSFERASE inhibitor 310264736 11120 7548 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200386 PREDNICARBATE 11121 7549 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ABT-414 DEPATUXIZUMAB MAFODOTIN 24424355 11122 7550 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PYRAZOLE PYRAZOLE 16374848 11124 7551 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 1,3-DI(4-AMINOPHENYLCARBOXAMIDO)BENZENE CHEMBL421431 11125 7552 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME NS1 27820802 11126 7553 KDM1A 23028 DRUGGABLE GENOME, ENZYME, CELL SURFACE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING inhibitor 310264760 11128 7554 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AMSACRINE HYDROCHLORIDE AMSACRINE HYDROCHLORIDE 11129 7555 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE H2O2 2138680 11130 7556 USP1 7398 DNA REPAIR, PROTEASE, ENZYME 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 11133 7557 TCF7L2 6934 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR sulfonamides, urea derivatives 21114608,17519421 11134 7558 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Encorafenib ENCORAFENIB 27312529 11135 7559 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME PF-04554878 DEFACTINIB 11136 7560 CBX1 10951 NA XCT790 CHEMBL189753 11137 7561 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135652750 11140 7562 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE GPC-3298306 11141 7563 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR PKC412 MIDOSTAURIN 11719451 11142 7564 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AMOXAPINE AMOXAPINE 11143 7565 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Cyclic cyanoethypypazole derivative 1 11146 7566 HTT 3064 DRUGGABLE GENOME PMID28092474-Compound-34 11147 7567 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Methscopolamine Bromide 11148 7568 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METYROSINE METYROSINE 22931300 11150 7569 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SOFALCONE SOFALCONE 11153 7570 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME AEW-541 AEW-541 11155 7571 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME ROXITHROMYCIN ROXITHROMYCIN 18212111 11156 7572 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SB-202190 SB-202190 11157 7573 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 381118891 11160 7574 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101402 GLYCYRRHIZIN 11161 7575 PNP 4860 ENZYME, DRUGGABLE GENOME Guanosine GUANOSINE 11162 7576 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR modulator CHEMBL146506 MOFAROTENE 11164 7577 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CONGO RED CONGO RED 11165 7578 PSMC1 5700 PROTEASE BORTEZOMIB BORTEZOMIB 24524217 11166 7579 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GW7074 CHEMBL72365 11168 7580 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BUDESONIDE BUDESONIDE 22931300 11169 7581 PSMA8 143471 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL371405 MARIZOMIB 11173 7582 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Telmisartan TELMISARTAN 11174 7583 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL421 SULFASALAZINE 11175 7584 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUCYTOSINE FLUCYTOSINE 11178 7585 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR antagonist 223366062 AT-406 11179 7586 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102568 11180 7587 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BECLOMETHASONE BECLOMETHASONE 22931300 11181 7588 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-44 11183 7589 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4'-HYDROXYCHALCONE 4'-HYDROXYCHALCONE 11184 7590 GMNN 51053 DRUGGABLE GENOME OXIBENDAZOLE OXIBENDAZOLE 11185 7591 GPR68 8111 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 404859018 11186 7592 GMNN 51053 DRUGGABLE GENOME DIHYDROERGOCRISTINE MESYLATE DIHYDROERGOCRISTINE MESYLATE 11188 7593 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR BECLOMETHASONE BECLOMETHASONE 11189 7594 PTPN6 5777 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE IL-4 15613279 11190 7595 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-695801 CHEMBL461193 11192 7596 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE METIPRANOLOL METIPRANOLOL 11193 7597 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 385612206 AVITRIPTAN 11195 7598 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 363894179 11197 7599 CA2 760 DRUGGABLE GENOME, ENZYME Benzthiazide BENZTHIAZIDE 11200 7600 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Isoflavone derivative 1 11204 7601 PTGS1 5742 ENZYME, DRUGGABLE GENOME NABUMETONE NABUMETONE 11205 7602 ADH1C 126 ENZYME, DRUGGABLE GENOME FOMEPIZOLE FOMEPIZOLE 11206 7603 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME CHRYSENE CHRYSENE 11207 7604 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AMIODARONE AMIODARONE 11209 7605 MAPT 4137 DRUGGABLE GENOME PIPLARTINE PIPLARTINE 11210 7606 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000120081 CHEMBL606532 11213 7607 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR CICLESONIDE CICLESONIDE 11214 7608 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME AG-490 CHEMBL56543 11215 7609 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-44 11216 7610 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Cycloalkyl nitrile pyrazolo pyridone derivative 2 11217 7611 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 348353661 11218 7612 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR CELASTROL CELASTROL 25756299,21129982 11219 7613 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR L-DOPA LEVODOPA 15081599 11220 7614 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE OXYBENZONE OXYBENZONE 11221 7615 SH2B1 25970 KINASE olanzapine OLANZAPINE 28694205 11222 7616 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING 2-MERCAPTOPYRIMIDINE 2-MERCAPTOPYRIMIDINE 11223 7617 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Celiprolol CELIPROLOL 11224 7618 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor REGORAFENIB REGORAFENIB 11225 7619 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEMETON-S-METHYL DEMETON-S-METHYL 11227 7620 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME JNJ-7706621 JNJ-7706621 11228 7621 NT5C2 22978 ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE gemcitabine GEMCITABINE 22838949,24300978 11229 7622 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102276 11231 7623 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 nateglinide NATEGLINIDE 22842957 11232 7624 EIF4E 1977 DRUGGABLE GENOME H2O2 12151318 11233 7625 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor OBATOCLAX OBATOCLAX 11234 7626 ALDH1A1 216 DRUGGABLE GENOME, ENZYME LEAD DIACETATE TRIHYDRATE LEAD DIACETATE TRIHYDRATE 11235 7627 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417809 CHEMBL1442783 11236 7628 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME Alpha 1-PI 11238 7629 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antibody ATEZOLIZUMAB ATEZOLIZUMAB 11239 7630 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DNDI1417132 CHEMBL1492017 11240 7631 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ARTESUNATE ARTESUNATE 25074847 11244 7632 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650833 PIRIBEDIL 11246 7633 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE APOMORPHINE APOMORPHINE 11247 7634 ADM 133 DRUGGABLE GENOME, HORMONE ACTIVITY NSC-87877 CHEMBL472004 22884224 11248 7635 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID29757691-Compound-8b 11249 7636 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 4-NONYLPHENOL 4-NONYLPHENOL 11251 7637 TUBB6 84617 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 11252 7638 EPHX1 2052 ENZYME, DRUGGABLE GENOME docetaxel DOCETAXEL 20157331 11254 7639 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CY-208243 CHEMBL313737 11255 7640 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor FOSTAMATINIB FOSTAMATINIB 11256 7641 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3996 CHEMBL584458 11258 7642 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR P276-00 RIVICICLIB 11259 7643 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE INGLIFORIB INGLIFORIB 11260 7644 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 11261 7645 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER CALCDPWW CALCDPWW 19597508 11262 7646 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL538943 VINORELBINE TARTRATE 11263 7647 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650246 ETORPHINE 11264 7648 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ARGENTEOSIDE A ARGENTEOSIDE A 23362862 11265 7649 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX ISOLIQUIRITIGENIN ISOLIQUIRITIGENIN 21866899 11266 7650 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 10 11267 7651 BAZ2B 29994 NA PROCHLORPERAZINE EDISYLATE PROCHLORPERAZINE EDISYLATE 11268 7652 TRAF3IP2 10758 TRANSCRIPTION FACTOR, KINASE nevirapine NEVIRAPINE 11269 7653 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102422 D-PHENYLALANINE 11274 7654 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 135650927 ROSIGLITAZONE 11275 7655 TFAP2A 7020 TRANSCRIPTION FACTOR NELFINAVIR NELFINAVIR 10996400 11276 7656 RHBDF2 79651 ENZYME fentanyl FENTANYL 21622719 11277 7657 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Epacadostat EPACADOSTAT 11278 7658 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 187051834 LIFITEGRAST 11279 7659 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 methadone METHADONE 9187528,21902501 11280 7660 GMNN 51053 DRUGGABLE GENOME MERADIMATE MERADIMATE 11281 7661 PKD2 5311 DRUGGABLE GENOME, TUMOR SUPPRESSOR, ION CHANNEL, TRANSPORTER allopurinol ALLOPURINOL 30924126 11282 7662 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CARBARIL CARBARIL 11283 7663 HEXB 3074 ENZYME TAMOXIFEN TAMOXIFEN 8577454 11284 7664 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE GW441756X GW441756X 11285 7665 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR DASATINIB DASATINIB 11286 7666 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SANGUINARINE SULFATE SANGUINARINE SULFATE 11288 7667 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME 1,4-DICHLOROBENZENE 1,4-DICHLOROBENZENE 16699520 11291 7668 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME BAY-613606 CHEMBL541400 11292 7669 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR citalopram CITALOPRAM 18794724 11293 7670 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL193240 ROFLUMILAST 11295 7671 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3545088 PUQUITINIB 11296 7672 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 310264675 CUDC-101 11297 7673 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 11298 7674 USP1 7398 DNA REPAIR, PROTEASE, ENZYME FLAVIN ADENINE DINUCLEOTIDE FLAVIN ADENIN DINUCLEOTIDE 11299 7675 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIGOXIGENIN DIGOXIGENIN 11300 7676 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ivabradine IVABRADINE 11301 7677 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DEQUALINIUM CHLORIDE DEQUALINIUM CHLORIDE 11303 7678 SMN2 6607 DRUGGABLE GENOME RESVERATROL RESVERATROL 11304 7679 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Cediranib CEDIRANIB 22238366 11305 7680 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR BAZEDOXIFENE BAZEDOXIFENE 11307 7681 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TOLONIUM CHLORIDE TOLONIUM CHLORIDE 11308 7682 IGF1 3479 GROWTH FACTOR, HORMONE ACTIVITY, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE Xentuzumab XENTUZUMAB 11310 7683 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Sirukumab SIRUKUMAB 11311 7684 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651509 11312 7685 ADO 84890 NA hydrochlorothiazide HYDROCHLOROTHIAZIDE 31327267 11316 7686 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SP-600125 SP-600125 23634759 11317 7687 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 249565660 11319 7688 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ZIPRASIDONE ZIPRASIDONE 11320 7689 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 249565850 11321 7690 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Hydroxyflutamide HYDROXYFLUTAMIDE 11323 7691 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ADALIMUMAB ADALIMUMAB 11324 7692 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE deferasirox DEFERASIROX 25348619,26403473 11325 7693 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Bis-aminopyrimidine derivative 5 11326 7694 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ABT-414 DEPATUXIZUMAB MAFODOTIN 26846818 11329 7695 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RTA-901 11330 7696 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 315661271 11331 7697 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR EPLERENONE EPLERENONE 11332 7698 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antagonist CHEMBL2109393 RG-7160 11334 7699 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-EP20041486488 11335 7700 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-95397 CHEMBL429095 11336 7701 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE R-IFN-1a 11337 7702 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SB-220025 SB-220025 11339 7703 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178103752 ESCITALOPRAM 11341 7704 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ENDO-ATROPINE ENDO-ATROPINE 22931300 11343 7705 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor SODIUM PHENYLBUTYRATE 11344 7706 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3184679 AZD-4547 11346 7707 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MYL-1401O 11347 7708 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BUSPIRONE BUSPIRONE 11348 7709 SERPINA6 866 DRUGGABLE GENOME, PROTEASE INHIBITOR Ciclesonide CICLESONIDE 11349 7710 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME PD-98059 CHEMBL35482 11350 7711 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-1134 CHEMBL600694 11352 7712 TUBA1A 7846 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 11354 7713 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE tamoxifen TAMOXIFEN 11130383,15197194,16331614,16636335 11355 7714 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME Platinum compounds 19525887 11356 7715 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME VOLVALERENAL D VOLVALERENAL D 11358 7716 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor AS703569 CENISERTIB 11359 7717 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE perindopril PERINDOPRIL 11361 7718 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DAMNACANTHAL DAMNACANTHAL 11362 7719 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650275 FLUPHENAZINE 11363 7720 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER Alkavervir ALKAVERVIR 11364 7721 TCF7L2 6934 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR tacrolimus TACROLIMUS 23041303,21857094 11365 7722 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME PROTOPORPHYRIN DISODIUM PROTOPORPHYRIN DISODIUM 11366 7723 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE BAY-613606 CHEMBL541400 11368 7724 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody AVE1642 11370 7725 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PARTHENOLIDE PARTHENOLIDE 25190466 11371 7726 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME E-4716 11372 7727 SERPINA6 866 DRUGGABLE GENOME, PROTEASE INHIBITOR PARAMETHASONE PARAMETHASONE 11373 7728 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FENAMIDONE FENAMIDONE 11374 7729 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE Crizotinib CRIZOTINIB 23811600 11375 7730 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR BRDU 10495776 11376 7731 TAOK3 51347 DNA REPAIR, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME morphine MORPHINE 11377 7732 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL428647 PACLITAXEL 11378 7733 HNMT 3176 ENZYME, DRUGGABLE GENOME DABIGATRAN DABIGATRAN 22494098 11379 7734 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER aliskiren ALISKIREN 11381 7735 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor METFORMIN METFORMIN 11382 7736 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200479 DICYCLOMINE HYDROCHLORIDE 11385 7737 NPC1L1 29881 DRUGGABLE GENOME, TRANSPORTER EZETIMIBE EZETIMIBE 11386 7738 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Tubastatin A 25957812 11387 7739 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL antagonist 135650660 11389 7740 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR ABEXINOSTAT ABEXINOSTAT 28221861 11390 7741 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME TAK-701 11391 7742 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE hydroxyzine HYDROXYZINE 18695978 11393 7743 MAPT 4137 DRUGGABLE GENOME EPALRESTAT EPALRESTAT 11394 7744 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE DASATINIB DASATINIB 32092139,21953054,17372901,19671763,17699867,16434489 11395 7745 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2,4,6-TRIHYDROXYACETOPHENONE 2,4,6-TRIHYDROXYACETOPHENONE 11396 7746 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR WZ4002 22961667 11397 7747 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL552212 LEXIBULIN 11398 7748 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL RO-4882224 CHEMBL1077391 19762240 11399 7749 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE F200 11400 7750 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR CLIOQUINOL CLIOQUINOL 11401 7751 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR AM-111 BRIMAPITIDE, C-TERMINAL ACID 11402 7752 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR CHLORPROMAZINE HYDROCHLORIDE CHLORPROMAZINE HYDROCHLORIDE 11403 7753 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE TRAIL 12642685 11404 7754 PTGS1 5742 ENZYME, DRUGGABLE GENOME Carbamate derivative 2 11407 7755 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME LORAZEPAM LORAZEPAM 11408 7756 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 amlodipine AMLODIPINE 11410 7757 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME BAY-613606 CHEMBL541400 11411 7758 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 387065613 11413 7759 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-acylpiperidine ether derivative 2 11415 7760 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PHYSOSTIGMINE PHYSOSTIGMINE 11417 7761 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PRIMAQUINE PHOSPHATE PRIMAQUINE PHOSPHATE 11419 7762 MPHOSPH8 54737 NA SIB-1757 CHEMBL88553 11420 7763 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE SALINE SODIUM CHLORIDE 12688543 11422 7764 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135649888 11424 7765 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR 2,3,4,6-TETRACHLORO-PHENOL CHEMBL320361 11425 7766 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DORAMAPIMOD DORAMAPIMOD 11426 7767 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ERGOCRYPTINE ERGOCRYPTINE 11430 7768 TMPRSS2 7113 CLINICALLY ACTIONABLE, PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178103048 CAMOSTAT 11433 7769 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BMS-816336 11434 7770 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE inhibitor 252827403 11435 7771 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor NINTEDANIB NINTEDANIB 11436 7772 GAA 2548 DRUGGABLE GENOME, ENZYME 4-HYDROXYESTRADIOL CHEMBL1412489 11438 7773 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Lapatinib LAPATINIB 26270481,26627007,23940356,26245675,26920887 11440 7774 POLK 51426 DNA REPAIR, ENZYME GNF-PF-1852 CHEMBL533293 11441 7775 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR dobutamine DOBUTAMINE 15564877,16325050,11753577 11442 7776 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 310264692 VEROSUDIL 11444 7777 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Capecitabine CAPECITABINE 26432108 11445 7778 CBX1 10951 NA ML-10302 CHEMBL286136 11446 7779 CD47 961 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE ABT-510 ABT-510 11447 7780 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME MK-8808 11449 7781 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE V3381 INDANTADOL 11451 7782 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TACROLIMUS TACROLIMUS 17202802 11453 7783 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor PANOBINOSTAT PANOBINOSTAT 11456 7784 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FEBUXOSTAT FEBUXOSTAT 11457 7785 CUX2 23316 TRANSCRIPTION FACTOR rifampin RIFAMPIN 11458 7786 TUBA1A 7846 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 11459 7787 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Nalbuphine hydrochloride ER 11461 7788 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MELEVODOPA MELEVODOPA 11465 7789 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR AMOXICILLIN AMOXICILLIN 16815316 11467 7790 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PARATHION PARATHION 11469 7791 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID30259754-Compound-LY2562175 11470 7792 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR US10022354, Example 152 11471 7793 KDM6A 7403 ENZYME, CLINICALLY ACTIONABLE inhibitor 381118851 11473 7794 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME QUINACRINE DIHYDROCHLORIDE QUINACRINE DIHYDROCHLORIDE 11474 7795 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME PMID29130358-Compound-Figure18(14a) 11477 7796 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor CHEMBL1976040 ADAVOSERTIB 11478 7797 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Trimeprazine METHYLPROMAZINE 11479 7798 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE ANTIESTROGEN 10908655 11480 7799 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME XL844 11481 7800 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME VTB-38543 11482 7801 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME TPX-0005 11483 7802 TARDBP 23435 TUMOR SUPPRESSOR FLURBIPROFEN FLURBIPROFEN 11484 7803 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Paclitaxel PACLITAXEL 28514312,26432108 11486 7804 MAPT 4137 DRUGGABLE GENOME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 11487 7805 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 363894139 CR-6086 11488 7806 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE MANGOSTIN MANGOSTIN 11489 7807 LGR6 59352 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102181 11492 7808 P4HB 5034 THIOREDOXIN, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE ASTRAGALIN ASTRAGALIN 11493 7809 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZANOTERONE ZANOTERONE 11494 7810 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1-HEXYLPYRIDINIUM IODIDE CHEMBL555242 11499 7811 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE pioglitazone PIOGLITAZONE 11503 7812 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-27 11504 7813 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 252166527 PEFICITINIB 11505 7814 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE lapuleucel-T LAPULEUCEL-T 11507 7815 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE RG-1530 RG-1530 11510 7816 BAZ2B 29994 NA DNDI1417447 CHEMBL1307453 11511 7817 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE EPIRUBICIN EPIRUBICIN 11759828 11512 7818 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GEFITINIB GEFITINIB 21258250,15696205,19794967,23313110 11515 7819 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Quizartinib QUIZARTINIB 23497317 11516 7820 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE HYDROQUINONE HYDROQUINONE 11518 7821 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649831 11519 7822 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Citalopram derivative 1 11520 7823 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651488 11522 7824 EPHX2 2053 DRUGGABLE GENOME, ENZYME inhibitor 363894191 11523 7825 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR CX-4945 SILMITASERTIB 11524 7826 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4-PHENYLAZO-PHENYLAMINE CHEMBL83761 11525 7827 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102296 DORAMAPIMOD 11526 7828 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ERGOCORNINE ERGOCORNINE 11527 7829 TARDBP 23435 TUMOR SUPPRESSOR TCMDC-124336 CHEMBL527271 11529 7830 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROPIOMAZINE PROPIOMAZINE 11530 7831 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ISOFENPHOS ISOFENPHOS 11532 7832 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650113 CLOPROSTENOL 11536 7833 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME ETHINYL ESTRADIOL 12312052 11538 7834 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-47 11540 7835 ASL 435 ENZYME sodium benzoate / sodium phenylacetate 11541 7836 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME CITALOPRAM CITALOPRAM 11542 7837 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE inhibitor 187051756 CROFELEMER 11544 7838 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Avastin+/-Tarceva 11546 7839 HTT 3064 DRUGGABLE GENOME Remetinostat REMETINOSTAT 11547 7840 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2109621 ABITUZUMAB 11549 7841 TOP2B 7155 DRUGGABLE GENOME, ENZYME dexrazoxane DEXRAZOXANE 21048526 11550 7842 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Ortataxel ORTATAXEL 11551 7843 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROPICONAZOLE PROPICONAZOLE 11554 7844 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Lenvatinib LENVATINIB 25295214 11555 7845 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR N-PHENETHYLCINNAMAMIDE CHEMBL1305393 11557 7846 KDM4A 9682 DRUGGABLE GENOME, ENZYME 4-HYDROXYBENZALDEHYDE PHENYLHYDRAZONE CHEMBL224032 11560 7847 ADAM17 6868 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, NEUTRAL ZINC METALLOPEPTIDASE, TRANSPORTER, ENZYME MARIMASTAT MARIMASTAT 26192023 11561 7848 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE ADJUVANT 7787697 11562 7849 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME methylcholanthrene 17481570 11564 7850 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27551786-Compound-III 11565 7851 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROROXAN PROROXAN 11567 7852 APOE 348 DRUGGABLE GENOME hmg coa reductase inhibitors 11568 7853 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME GDC0879 19276360 11569 7854 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NALOXONE NALOXONE 17616524 11570 7855 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 2890444 11572 7856 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME bleomycin BLEOMYCIN 11573 7857 EYA2 2139 DNA REPAIR FLUAZINAM FLUAZINAM 11574 7858 GLCCI1 113263 NA budesonide BUDESONIDE 21991891 11576 7859 HDAC11 79885 DRUGGABLE GENOME, ENZYME PMID29671355-Compound-21 11577 7860 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PENICILLIN PENICILLIN G POTASSIUM 12530481 11579 7861 GMNN 51053 DRUGGABLE GENOME DEMETHOXYCURCUMIN DEMETHOXYCURCUMIN 11580 7862 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 348353652 11581 7863 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-39 11582 7864 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TAK-715 TAK-715 11583 7865 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALFUZOSIN HYDROCHLORIDE ALFUZOSIN HYDROCHLORIDE 11584 7866 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OLVANIL OLVANIL 11585 7867 POLK 51426 DNA REPAIR, ENZYME PYRONIN Y PYRONIN Y 11588 7868 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR CETRORELIX CETRORELIX 16391860 11589 7869 NCOA1 8648 ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX inhibitor 252827441 11592 7870 PTGS2 5743 DRUGGABLE GENOME, ENZYME MESALAZINE MESALAMINE 11594 7871 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE neratinib NERATINIB 23220880 11595 7872 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649794 11596 7873 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 178100968 11597 7874 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Neratinib NERATINIB 11598 7875 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE DOVITINIB DOVITINIB 11601 7876 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID25656651-Compound-34a 11602 7877 BAZ2B 29994 NA 6-METHOXY-HARMALAN CHEMBL338115 11603 7878 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HYDROCORTISONE HYDROCORTISONE 7909787 11604 7879 CTSF 8722 DRUGGABLE GENOME, PROTEASE, ENZYME PMID27998201-Compound-12 11605 7880 HEBP1 50865 DRUGGABLE GENOME Omaveloxolone OMAVELOXOLONE 11606 7881 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist,antagonist 135651233 TAMOXIFEN 11607 7882 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BI-69A11 19175524 11608 7883 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME NSC-37136 CHEMBL1370674 11609 7884 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE inhibitor 404859129 11610 7885 MAPT 4137 DRUGGABLE GENOME OSAJIN OSAJIN 11611 7886 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 7,8,3'-TRIHYDROXYFLAVONE CHEMBL225513 11616 7887 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL2107771 RALFINAMIDE 11618 7888 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CLOTRIMAZOLE CLOTRIMAZOLE 11620 7889 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-3314 CHEMBL582287 11622 7890 MAPT 4137 DRUGGABLE GENOME GNF-PF-5052 CHEMBL601367 11623 7891 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Roscovitine derivative 1 11624 7892 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1034 DICLOFENAC SODIUM 11626 7893 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ESTRADIOL ESTRADIOL 23448346 11629 7894 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417181 CHEMBL1537417 11630 7895 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565699 CHEMBL322970 11631 7896 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE DESLANOSIDE DESLANOSIDE 11632 7897 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE IDH305 11633 7898 CMTM8 152189 NA methylphenidate METHYLPHENIDATE 29382897 11635 7899 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Pegsunercept PEGSUNERCEPT 11637 7900 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER FLUOROURACIL FLUOROURACIL 19274060 11640 7901 MKNK1 8569 SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, ENZYME EFT508 TOMIVOSERTIB 11642 7902 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME UNC1062 23585477 11643 7903 CBX1 10951 NA TRIMIPRAMINE TRIMIPRAMINE 11644 7904 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SP-600125 SP-600125 11647 7905 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DIPHENHYDRAMINE DIPHENHYDRAMINE 11648 7906 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PORFIROMYCIN PORFIROMYCIN 11650 7907 TGFBR3 7049 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME RANTES 14637022 11651 7908 SMN1 6606 DRUGGABLE GENOME CID 1540951 CHEMBL259421 11652 7909 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166854 11653 7910 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR aspirin ASPIRIN 17496729 11654 7911 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL717 MEDROXYPROGESTERONE ACETATE 11655 7912 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME DASATINIB DASATINIB 11656 7913 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 381118859 11657 7914 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR TNF-ALPHA 9751175 11658 7915 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-19 11659 7916 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE RALOXIFENE RALOXIFENE 15590986 11662 7917 USP1 7398 DNA REPAIR, PROTEASE, ENZYME 1,4-DIMETHOXYANTHRAQUINONE 1,4-DIMETHOXYANTHRAQUINONE 11664 7918 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CANDESARTAN CILEXETIL CANDESARTAN CILEXETIL 11665 7919 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR RESMINOSTAT RESMINOSTAT 11666 7920 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CAMBINOL CAMBINOL 11668 7921 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DG3173 VELDOREOTIDE 11669 7922 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE MDX-214 11672 7923 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME DAUNORUBICIN DAUNORUBICIN 22260166 11673 7924 GUCY1A1 2982 ENZYME, DRUGGABLE GENOME activator CHEMBL136478 SODIUM NITROPRUSSIDE 11674 7925 TBP 6908 TRANSCRIPTION FACTOR HORMONES 7848271 11675 7926 HEXB 3074 ENZYME ESTRAMUSTINE ESTRAMUSTINE 6795611 11677 7927 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME Progesterone PROGESTERONE 11679 7928 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 178103981 ILOMASTAT 11680 7929 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178101522 FENOPROFEN 11681 7930 MAPT 4137 DRUGGABLE GENOME DNDI1417025 CHEMBL1320453 11682 7931 NCAM1 4684 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CD56 CAR T cells 11685 7932 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor 178103494 IBRUTINIB 11687 7933 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER O-DEMETHYLATED ADAPALENE O-DEMETHYLATED ADAPALENE 11688 7934 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565793 11689 7935 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Gefitinib GEFITINIB 23242808,22448344,27312529 11690 7936 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE SB-202190 SB-202190 22951114 11691 7937 TNFRSF11A 8792 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE propionic acid derivatives 26398624 11693 7938 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MRS-1220 CHEMBL88147 11695 7939 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TALMAPIMOD TALMAPIMOD 11696 7940 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME NIVOLUMAB NIVOLUMAB 28525386 11697 7941 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125298 CHEMBL581152 11699 7942 TUBA1B 10376 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 11700 7943 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-407228 CHEMBL74852 11701 7944 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 252827368 PEXIDARTINIB 11702 7945 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NEUROPROTECTIVE AGENT 17530460 11703 7946 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2013161919Example85-117 11707 7947 ATXN2 6311 NA (R,S)-INDATRALINE (R,S)-INDATRALINE 11708 7948 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CEPHALORIDINE CEPHALORIDINE 11710 7949 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ANGUSTIBALIN ANGUSTIBALIN 11712 7950 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE 385612241 11715 7951 EYA2 2139 DNA REPAIR (R)-EDELFOSINE (R)-EDELFOSINE 11716 7952 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PANITUMUMAB PANITUMUMAB 26812186,19075190,19255327,22734028,23182985,21228335,17384584,26623049,2278970,19114683,21398618,20921465,18316791,19679400,18794081,21975775,16361624,16618717,19773371,26371285,24558511,3122217,16434492,19018267,20921462,25157968,12460918,20978259,22407852,22392911,23406027 11718 7953 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 381118891 11719 7954 NGFR 4804 CELL SURFACE, DRUGGABLE GENOME Fulranumab FULRANUMAB 11720 7955 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL3545134 LY-2780301 11721 7956 KDM4A 9682 DRUGGABLE GENOME, ENZYME EMODIN EMODIN 11723 7957 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE ANISTREPLASE ANISTREPLASE 11725 7958 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SALSOLINOL HYDROBROMIDE SALSOLINOL HYDROBROMIDE 11726 7959 TUBA3C 7278 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 11728 7960 PDE3A 5139 ENZYME, DRUGGABLE GENOME RPL-554 11730 7961 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Vemurafenib VEMURAFENIB 27312529 11731 7962 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR MONOETHANOLAMINE MONOETHANOLAMINE 11732 7963 TMEM167A 153339 NA fluorouracil FLUOROURACIL 28796378 11733 7964 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-123579 CHEMBL533954 11734 7965 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CORYNANTHEINE CORYNANTHEINE 11735 7966 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME SAXAGLIPTIN SAXAGLIPTIN 11736 7967 MAOB 4129 DRUGGABLE GENOME, ENZYME VITAMIN-B12 8043706 11737 7968 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME inhibitor 135652711 RIFAMPIN 11740 7969 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR BVD-523 ULIXERTINIB 11745 7970 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Imidazopyridazine derivative 1 11746 7971 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Peptidomimetic analog 3 11747 7972 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1567 SUNITINIB MALATE 11749 7973 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 178102515 TEMSIROLIMUS 11750 7974 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-102049 CHEMBL74675 11751 7975 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BDBM50177019 11752 7976 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Docetaxel DOCETAXEL 21399868 11755 7977 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR BENZYL SALICYLATE BENZYL SALICYLATE 11757 7978 BAZ2B 29994 NA inhibitor 249565913 11759 7979 NOS1 4842 DRUGGABLE GENOME, ENZYME DEXTRAN SULFATE SODIUM 15613746,17160477 11760 7980 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1201089 DIPHENHYDRAMINE CITRATE 11761 7981 XRCC5 7520 KINASE CAMPTOTHECIN CAMPTOTHECIN 16230379 11762 7982 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DROSPIRENONE DROSPIRENONE 11763 7983 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR inhibitor CHEMBL1096882 FLUDARABINE PHOSPHATE 11766 7984 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 2-BROMO-HEXADECANOIC ACID CHEMBL118417 11767 7985 PNP 4860 ENZYME, DRUGGABLE GENOME ULODESINE ULODESINE 11770 7986 GUCY2C 2984 DRUGGABLE GENOME, KINASE agonist 178101551 11774 7987 SF3B2 10992 NA SPLICEOSTATIN-A CHEMBL1221944 17643111 11775 7988 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME GEFITINIB GEFITINIB 11776 7989 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE fluorouracil FLUOROURACIL 24958282 11777 7990 POLB 5423 DNA REPAIR, DRUGGABLE GENOME DNDI1416969 CHEMBL1453126 11778 7991 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 178103082 TANOMASTAT 11781 7992 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AG-494 CHEMBL56731 11782 7993 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PHENELZINE SULFATE PHENELZINE SULFATE 11785 7994 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DEPHOSTATIN DEPHOSTATIN 11786 7995 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME DICHLON DICHLON 11787 7996 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL3545252 DOCETAXEL 11789 7997 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ritonavir RITONAVIR 9187528 11792 7998 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHENYLSTIBONIC ACID PHENYLSTIBONIC ACID 11795 7999 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME CHLORQUINALDOL CHLORQUINALDOL 11796 8000 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PROPYLTHIOURACIL PROPYLTHIOURACIL 7790147 11797 8001 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Thiazole derivative 4 11798 8002 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIACEREIN DIACEREIN 11799 8003 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER MTX METHOTREXATE 12036927 11800 8004 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME 5-FU FLUOROURACIL 8888499 11802 8005 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651740 11803 8006 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME GENISTEIN GENISTEIN 16203797 11804 8007 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Autologous Anti-BCMA-CAR-expressing CD4+/CD8+ T-lymphocytes FCARH143 11805 8008 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ERYTHROPOIETIN EPOETIN BETA 16468051 11806 8009 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE KD025 11807 8010 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME HARMINE HARMINE 11808 8011 CYB5R3 1727 DRUGGABLE GENOME, ENZYME primaquine PRIMAQUINE 25058800 11811 8012 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CC-8490 11812 8013 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Gestrinone GESTRINONE 11813 8014 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103588 11814 8015 PDE10A 10846 ENZYME, DRUGGABLE GENOME Triazolo-pyridine derivative 3 11815 8016 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 4'-O-ACETYLPATENTIFLORIN B 4'-O-ACETYLPATENTIFLORIN B 22119124 11816 8017 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ERLOTINIB ERLOTINIB 26181029 11819 8018 UBA1 7317 ENZYME HYRTIOERECTINE B HYRTIOERECTINE B 22695182 11820 8019 PTGS2 5743 DRUGGABLE GENOME, ENZYME NIFLUMIC ACID 11821 8020 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 STAVUDINE STAVUDINE 22931300 11822 8021 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 3-METHOXYCATECHOL 3-METHOXYCATECHOL 11823 8022 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-17 11824 8023 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AZAKENPAULLONE AZAKENPAULLONE 11825 8024 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SPERMINE SPERMINE 11826 8025 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE AE-941 11827 8026 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Selumetinib SELUMETINIB 26272063,26351322,26438159,26666244,27231576,23200175,22271687,27655129,24935174,26676756,24939055,25870145,27222538,19029981,27556948,26232337,27422710,26725216,27312529,22952903,27480147,26125448,28492898,25322874 11829 8027 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MK-212 MK-212 11830 8028 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME IOFETAMINE HYDROCHLORIDE IOFETAMINE HYDROCHLORIDE 11833 8029 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METHYLMALONIC ACID METHYLMALONIC ACID 11835 8030 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DESERPIDINE DESERPIDINE 11837 8031 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE modulator CHEMBL3545356 VK5211 11838 8032 PSMD13 5719 NA inhibitor CHEMBL325041 BORTEZOMIB 11839 8033 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME NSC-36398 CHEMBL483206 11840 8034 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PROTEASE INHIBITORS 14520092 11841 8035 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME INGENOL MEBUTATE 11842 8036 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL488436 AZD-5438 11844 8037 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME LY-2090314 LY-2090314 11845 8038 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE antagonist 405560412 11847 8039 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME (+)-JQ1 11849 8040 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SALMETEROL XINAFOATE SALMETEROL XINAFOATE 11850 8041 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE BRM 1832500 11852 8042 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME EVEROLIMUS EVEROLIMUS 26821351 11853 8043 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-663 CHEMBL596847 11855 8044 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL1201010 FLUDROCORTISONE ACETATE 11856 8045 ATAD5 79915 NA [3H]-PHORBOL 12,13-DIBUTYRATE CHEMBL27768 11858 8046 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000018309 CHEMBL591363 11861 8047 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AMLEXANOX AMLEXANOX 11862 8048 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Pazopanib PAZOPANIB 11863 8049 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRAMUSTINE PHOSPHATE SODIUM ESTRAMUSTINE PHOSPHATE SODIUM 11864 8050 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 328083494 11865 8051 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME ANTI-INFLAMMATORY DRUGS 11164833 11866 8052 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX STROPHANTHIDIN ACETATE STROPHANTHIDIN ACETATE 11867 8053 GNA11 2767 CLINICALLY ACTIONABLE AEB071 SOTRASTAURIN 24141786,27507190 11868 8054 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ziprasidone ZIPRASIDONE 18695978 11870 8055 HSPB1 3315 DRUGGABLE GENOME BENZENETHIOL BENZENETHIOL 11872 8056 APC 324 CLINICALLY ACTIONABLE Leucovorin LEUCOVORIN 27626067 11873 8057 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GSK642444 11877 8058 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 249565817 11878 8059 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 11879 8060 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL586701 ZSTK-474 11880 8061 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 18 11881 8062 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2-PHENYLPHENOL 2-PHENYLPHENOL 11882 8063 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE unspecified PD-1 antibody 26645196 11883 8064 MAOB 4129 DRUGGABLE GENOME, ENZYME RWJ-416457 CHEMBL221877 11884 8065 CP 1356 DRUGGABLE GENOME, ENZYME TUMOR NECROSIS FACTOR 2439635 11885 8066 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME LINIFANIB LINIFANIB 11886 8067 FAAH 2166 ENZYME, DRUGGABLE GENOME opioids 11887 8068 BCHE 590 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 1 11889 8069 POLB 5423 DNA REPAIR, DRUGGABLE GENOME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 11890 8070 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 249565578 IPATASERTIB 11891 8071 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651493 HISTAMINE 11893 8072 ASNS 440 CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE asparaginase ASPARAGINASE 24268318 11895 8073 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 348353655 OCLACITINIB 11897 8074 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 385612170 KZR-616 11898 8075 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652249 11899 8076 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE AG-1879 CHEMBL406845 11900 8077 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR ANTIOXIDANT 12023887 11902 8078 MPI 4351 ENZYME, DRUGGABLE GENOME GNF-PF-5134 CHEMBL602969 11903 8079 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME FLAVOPIRIDOL ALVOCIDIB 11205902 11904 8080 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrido[3,2-d]pyrimidine derivative 2 11905 8081 IL1R2 7850 DRUGGABLE GENOME ANAKINRA ANAKINRA 11906 8082 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHLORPROMAZINE HYDROCHLORIDE CHLORPROMAZINE HYDROCHLORIDE 11907 8083 BHLHE40 8553 NA TRICHOSTATIN A 10737769 11909 8084 HDAC11 79885 DRUGGABLE GENOME, ENZYME HINOKITIOL HINOKITIOL 11910 8085 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor BUPARLISIB HYDROCHLORIDE 11911 8086 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR trastuzumab TRASTUZUMAB 11914 8087 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SP-600125 SP-600125 11915 8088 IL1B 3553 KINASE, DRUGGABLE GENOME CHINESE HERBS 8871284 11916 8089 MAOA 4128 DRUGGABLE GENOME, ENZYME 8-{[(4-BROMOPHENYL)METHYL]SULFANYL}CAFFEINE CHEMBL1927670 22055712 11919 8090 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL1683544 ERIBULIN MESYLATE 11920 8091 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME KAINIC ACID KAINIC ACID 11921 8092 NOS1AP 9722 NA verapamil VERAPAMIL 19247217 11922 8093 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME CIS-RESVERATROL CIS-RESVERATROL 11923 8094 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE GEDATOLISIB GEDATOLISIB 20166697 11924 8095 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME NITROSOUREAS 9393761 11925 8096 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME CARFILZOMIB CARFILZOMIB 24524217 11926 8097 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Ibrutinib IBRUTINIB 26563132 11927 8098 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RTA 744 11928 8099 VCAM1 7412 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMA 7678355 11929 8100 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ISOKAEMPFERIDE ISOKAEMPFERIDE 11930 8101 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE modafinil MODAFINIL 18695978 11931 8102 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100403 11934 8103 MGLL 11343 DRUGGABLE GENOME, ENZYME ABX-1431 11936 8104 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CABOZANTINIB CABOZANTINIB 27694386,29061793,21926191 11937 8105 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650293 FURTRETHONIUM 11939 8106 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME VORINOSTAT VORINOSTAT 24694055,19344175,19966789,26211462,23622981,22260166,17447750,20491440,21548582,23672185,19084294 11940 8107 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Capecitabine CAPECITABINE 17679724,26432108,26487584,26920887 11941 8108 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR SANT1 26781311 11942 8109 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 384403681 11943 8110 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor PI-103 PI-103 11944 8111 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME ARRY-382 ARRY-382 11945 8112 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2017974 BUPARLISIB 11946 8113 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CHLORANIL CHLORANIL 11947 8114 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE S-222611 S-222611 11950 8115 SOAT1 6646 DRUGGABLE GENOME 6-HYDROXYDOPAMINE 1559138 11952 8116 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 11953 8117 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Heparin low molecular weight 11955 8118 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE E2012 11956 8119 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102332 VATALANIB 11960 8120 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178102613 ISOGRANULATIMIDE 11961 8121 PDE6A 5145 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL628 PENTOXIFYLLINE 11962 8122 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1631 CHEMBL577222 11964 8123 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME ENMD-2076 ENMD-2076 11965 8124 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR US9006244, E2b 11966 8125 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR AMPICILLIN TRIHYDRATE AMPICILLIN TRIHYDRATE 11967 8126 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor 178103971 IBUDILAST 11969 8127 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RG-1530 RG-1530 11970 8128 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZD4785 AZD-4785 28615361 11971 8129 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135649956 ARIPIPRAZOLE 11975 8130 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER INC280 CAPMATINIB 25971938 11976 8131 IL17RC 84818 DRUGGABLE GENOME IL-17 16785495 11977 8132 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE GNF-PF-4085 CHEMBL528181 11978 8133 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 252166609 11980 8134 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GSK-269962A GSK-269962A 11981 8135 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor BMS777607 11982 8136 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Tricyclic compound 1 11983 8137 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DOXEPIN DOXEPIN 22007643 11985 8138 GLS 2744 ENZYME ISOTHYMONIN ISOTHYMONIN 11987 8139 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650653 11989 8140 IL23A 51561 DRUGGABLE GENOME Ustekinumab USTEKINUMAB 11990 8141 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Afimoxifene AFIMOXIFENE 11992 8142 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE SOTRASTAURIN SOTRASTAURIN 11994 8143 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Atenolol ATENOLOL 11995 8144 GMNN 51053 DRUGGABLE GENOME TCMDC-123650 CHEMBL580727 11996 8145 PDE10A 10846 ENZYME, DRUGGABLE GENOME Pyrido[1,2,4]triazolo[4,3-a]pyrazine derivative 2 11997 8146 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Selumetinib SELUMETINIB 26272063,22271687,24939055,21358673,26232337,26137449 11999 8147 BCHE 590 DRUGGABLE GENOME, ENZYME RIVASTIGMINE RIVASTIGMINE 12001 8148 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 328083488 CHEMBL401930 12002 8149 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 12004 8150 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor INCB028060 CAPMATINIB 12005 8151 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ATENOLOL ATENOLOL 2903243 12006 8152 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417776 CHEMBL1585652 12008 8153 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GSK2126458 OMIPALISIB 26603258 12010 8154 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME GNF-PF-5114 CHEMBL601952 12011 8155 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME IFN 15875206 12012 8156 NPR3 4883 DRUGGABLE GENOME agonist 178101592 12013 8157 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 354702292 12014 8158 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME IDAZOXAN IDAZOXAN 12015 8159 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051793 GIVINOSTAT 12016 8160 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 7,8,2'-TRIHYDROXYFLAVONE CHEMBL244707 12017 8161 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME cerivastatin CERIVASTATIN 15970799 12018 8162 AQP9 366 ION CHANNEL TESTOSTERONE TESTOSTERONE 12021052,12002438 12019 8163 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-16 12020 8164 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL ATRA TRETINOIN 18404486 12021 8165 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CARINATIN G CARINATIN G 12022 8166 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PYROGALLOL PYROGALLOL 12024 8167 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SOTALOL SOTALOL 22931300 12029 8168 GMNN 51053 DRUGGABLE GENOME GR-4661 CHEMBL344127 12031 8169 MARK4 57787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME JNJ-7706621 JNJ-7706621 12032 8170 NOTCH2 4853 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE inhibitor MK0752 12033 8171 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PROMETHAZINE HYDROCHLORIDE PROMETHAZINE HYDROCHLORIDE 12034 8172 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE MULTIKINASE INHIBITOR AEE788 18227510,19147750 12035 8173 GMNN 51053 DRUGGABLE GENOME FLUNARIZINE HYDROCHLORIDE FLUNARIZINE HYDROCHLORIDE 12036 8174 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NORDEXFENFLURAMINE NORDEXFENFLURAMINE 12037 8175 RAB9A 9367 ENZYME, DRUGGABLE GENOME TCMDC-125321 CHEMBL587449 12038 8176 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE TCMDC-124327 CHEMBL581929 12039 8177 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OLEOYL DOPAMINE OLEOYL DOPAMINE 12041 8178 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME IFX-1 12042 8179 IL24 11009 DRUGGABLE GENOME, KINASE INGN-241 12043 8180 HSPB2 3316 KINASE PROTEASOME INHIBITOR 15004512 12045 8181 MAPT 4137 DRUGGABLE GENOME PICEATANNOL PICEATANNOL 12046 8182 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NIACIN NIACIN 22931300 12047 8183 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650584 METITEPINE 12048 8184 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 404859149 12049 8185 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE DNDI1417467 CHEMBL1997335 12051 8186 GBA 2629 DRUGGABLE GENOME, ENZYME GENISTEIN GENISTEIN 12052 8187 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME GNF-PF-1919 CHEMBL576409 12053 8188 MUC16 94025 DRUGGABLE GENOME DMUC-5754A SOFITUZUMAB VEDOTIN 12054 8189 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Z-PRO-PROLINAL Z-PRO-PROLINAL 12056 8190 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CICLOPIROX OLAMINE CICLOPIROX OLAMINE 12057 8191 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Drugs For Treatment Of Tuberculosis 19686464,22162992,29036176 12058 8192 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIOGLITAZONE HYDROCHLORIDE PIOGLITAZONE HYDROCHLORIDE 12059 8193 SMN1 6606 DRUGGABLE GENOME GNF-PF-1000 CHEMBL600554 12060 8194 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME FLURANDRENOLIDE FLURANDRENOLIDE 12061 8195 GLS 2744 ENZYME DAPHNORIN DAPHNORIN 12062 8196 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2165191 AZD-6482 12063 8197 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Ponatinib PONATINIB 12064 8198 MMP7 4316 NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166768 12065 8199 CXCL8 3576 DRUGGABLE GENOME HEPTACHLOR HEPTACHLOR 12066 8200 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 249565706 BMS-214662 12067 8201 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CDDP CISPLATIN 16043385 12068 8202 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ALPROSTADIL ALPROSTADIL 12069 8203 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ICI-199,441 ICI-199,441 12071 8204 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME RUPATADINE RUPATADINE 12073 8205 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME GW843682X GW843682X 12074 8206 SMN2 6607 DRUGGABLE GENOME NABUMETONE NABUMETONE 12077 8207 CHN2 1124 NA fluorouracil FLUOROURACIL 24444404 12078 8208 TDO2 6999 ENZYME, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 4 12079 8209 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor 178103254 RASAGILINE 12081 8210 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME antagonist 381744949 12082 8211 SFTPA1 653509 DRUGGABLE GENOME IL-1RA ANAKINRA 8996657 12083 8212 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE SELECTIVE ESTROGEN RECEPTOR MODULATOR 11901050 12084 8213 MAP2K3 5606 KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE inhibitor DABRAFENIB MESYLATE 12086 8214 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER DELAVIRDINE DELAVIRDINE 21189339 12087 8215 EEF2K 29904 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Lapatinib LAPATINIB 12092 8216 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor CHEMBL3544942 RONICICLIB 12093 8217 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR antagonist 249565759 12094 8218 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CALANOLIDE A CALANOLIDE A 12095 8219 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GNF-PF-3537 CHEMBL601110 12096 8220 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 7,4'-DIHYDROXYFLAVONE CHEMBL294878 12097 8221 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GSK2334470 CHEMBL1765740 28178345 12099 8222 MAOA 4128 DRUGGABLE GENOME, ENZYME IncarviatoneA 12100 8223 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor ROMIDEPSIN ROMIDEPSIN 12101 8224 MAPT 4137 DRUGGABLE GENOME ZK-164015 CHEMBL184074 12102 8225 PDE5A 8654 ENZYME, DRUGGABLE GENOME AVANAFIL AVANAFIL 12103 8226 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME SULFORAPHANE SULFORAPHANE 15753404 12107 8227 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR VALSARTAN VALSARTAN 12108 8228 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME EMODIN EMODIN 12109 8229 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PF-04449913 GLASDEGIB 12110 8230 CBX1 10951 NA CLOFAZIMINE CLOFAZIMINE 12112 8231 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor DACOMITINIB DACOMITINIB 12114 8232 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE METMAB ONARTUZUMAB 12116 8233 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE SIROLIMUS SIROLIMUS 12119 8234 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Aromatic bicyclic compound 4 12120 8235 HPSE 10855 ENZYME, DRUGGABLE GENOME LABETALOL LABETALOL 23415087 12121 8236 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AG-527 CHEMBL258767 12125 8237 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3545097 SAPANISERTIB 12126 8238 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME PROTOPORPHYRIN PROTOPORPHYRIN 12127 8239 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 249565824 12129 8240 CCND3 896 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME LY2835219 ABEMACICLIB 12131 8241 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LONIDAMINE LONIDAMINE 12133 8242 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY ANDROSTENEDIONE ANDROSTENEDIONE 8404664 12134 8243 GMNN 51053 DRUGGABLE GENOME DIENESTROL DIENESTROL 12136 8244 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PYROGALLOL PYROGALLOL 12137 8245 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 252166498 TRAMADOL 12138 8246 PLA2G7 7941 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2104981 RILAPLADIB 12139 8247 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Aminopyridine derivative 2 12141 8248 RACGAP1 29127 NA HARMOL HARMOL 12142 8249 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR CISPLATIN CISPLATIN 10071988,8554977 12143 8250 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-636948 CHEMBL1998001 12144 8251 TICAM1 148022 TRANSCRIPTION FACTOR VACCINE 18217948 12145 8252 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR TAMATINIB R-406 12152 8253 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE VER-49009 CHEMBL365617 12154 8254 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE HOMIDIUM BROMIDE HOMIDIUM BROMIDE 12155 8255 TUBB2A 7280 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 12156 8256 ITPKA 3706 KINASE, ENZYME inhibitor 336446934 12157 8257 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist 252166707 12158 8258 GHRL 51738 DRUGGABLE GENOME HUMAN CHORIONIC GONADOTROPIN 17535999 12159 8259 RPTOR 57521 CLINICALLY ACTIONABLE, KINASE inhibitor MLN0128 SAPANISERTIB 12160 8260 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NVP-LAQ824 DACINOSTAT 12161 8261 COMT 1312 DRUGGABLE GENOME, ENZYME methadone METHADONE 28006928,32407152,23686330,21398039,23302985,26902643,29474345,23773341,25155931,25185591,19514130,28745577,27027462 12162 8262 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PHENYLBUTYRYLHYDROXAMIC ACID PHENYLBUTYRYLHYDROXAMIC ACID 21874153 12163 8263 DROSHA 29102 NA vincristine VINCRISTINE 24614921 12164 8264 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PATULIN PATULIN 16680159 12168 8265 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE INDOMETHACIN INDOMETHACIN 17329922 12169 8266 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME LUTEOLIN LUTEOLIN 12170 8267 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR TACEDINALINE TACEDINALINE 18692397 12172 8268 PCYT1A 5130 ENZYME lamivudine LAMIVUDINE 12173 8269 ATXN2 6311 NA TCMDC-123808 CHEMBL546493 12174 8270 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME HORMONES 11589623 12175 8271 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565576 ENMD-2076 12176 8272 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME 1,4-BIS(4-METHOXYPHENYLSULFONYL)PIPERAZINE CHEMBL1091502 12177 8273 SMN1 6606 DRUGGABLE GENOME GNF-PF-992 CHEMBL602561 12178 8274 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE DRF-1042 12179 8275 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE WP-1066 12180 8276 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME RIBAVIRIN RIBAVIRIN 16699498 12181 8277 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME DNDI1417156 CHEMBL1504679 12183 8278 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL activator 178101089 CHEMBL1290115 12184 8279 LPAR2 9170 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE CAFFEINE CAFFEINE 10199823 12186 8280 SI 6476 DRUGGABLE GENOME, ENZYME INSULIN INSULIN 9585003 12187 8281 CCNK 8812 KINASE epirubicin EPIRUBICIN 12188 8282 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ZYH-1 12189 8283 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE NSC-21588 CHEMBL1611308 12190 8284 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker 53801037 12193 8285 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DNDI1417478 CHEMBL1972216 12194 8286 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR PIRFENIDONE PIRFENIDONE 12907346 12196 8287 SRD5A3 79644 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200969 DUTASTERIDE 12197 8288 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor AT9283 AT-9283 12199 8289 ATXN2 6311 NA TCMDC-125544 CHEMBL533602 12200 8290 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 752709 CHEMBL429335 12201 8291 ZNF804A 91752 NA antipsychotics 21892778 12203 8292 HMGCR 3156 ENZYME, DRUGGABLE GENOME SIMVASTATIN SIMVASTATIN 16680159 12204 8293 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL593430 ATAGABALIN 12205 8294 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AZD3759 AZD-3759 27928026 12206 8295 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME (S)-methadone 17178267 12207 8296 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545119 BMS-794833 12209 8297 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 zidovudine ZIDOVUDINE 22960662 12210 8298 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE ACU-XSP-001 12211 8299 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE CDX-3379 12213 8300 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE spironolactone SPIRONOLACTONE 22543981 12215 8301 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-14 12216 8302 MAP3K7 6885 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 223366077 RGB-286638 12221 8303 ARSA 410 DRUGGABLE GENOME, ENZYME DESIPRAMINE DESIPRAMINE 12222 8304 PTGES 9536 DRUGGABLE GENOME, ENZYME Methyl-piperidine compound 1 12223 8305 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME repaglinide REPAGLINIDE 17923851,15961978,14534525,18388877,21270106 12224 8306 TOP2B 7155 DRUGGABLE GENOME, ENZYME Podofilox PODOFILOX 12225 8307 CP 1356 DRUGGABLE GENOME, ENZYME ORAL CONTRACEPTIVE 12616983 12226 8308 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AZD-1775 ADAVOSERTIB 12227 8309 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ticlopidine TICLOPIDINE 17339877 12228 8310 POLK 51426 DNA REPAIR, ENZYME PINOPHILIN A PINOPHILIN A 22264170 12229 8311 MAPT 4137 DRUGGABLE GENOME TRICLABENDAZOLE TRICLABENDAZOLE 12231 8312 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CC-90003 12232 8313 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ISOTRETINOIN ISOTRETINOIN 12233 8314 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200733 DESFLURANE 12235 8315 KCNH6 81033 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL284348 DALFAMPRIDINE 12236 8316 TPM3 7170 KINASE, CLINICALLY ACTIONABLE METHOTREXATE METHOTREXATE 8509220 12238 8317 STING1 340061 CLINICALLY ACTIONABLE, KINASE agonist 315661283 12239 8318 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER ADRIAMYCIN ADRIAMYCIN 15130309 12241 8319 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX APIGENIN APIGENIN 25190466 12242 8320 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor MIDOSTAURIN MIDOSTAURIN 12243 8321 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DHT ANDROSTANOLONE 16990489,16482568 12244 8322 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PMID25416646-Compound-Figure5-H 12245 8323 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ERLOTINIB ERLOTINIB 12246 8324 HR 55806 NUCLEAR HORMONE RECEPTOR Histamine Phosphate 12248 8325 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GENISTEIN GENISTEIN 8621505 12249 8326 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME BAY 869766 12250 8327 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME PALBOCICLIB PALBOCICLIB 12251 8328 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME IDRABIOTAPARINUX 12252 8329 TSPO 706 DRUGGABLE GENOME Benzothiazepine analog 3 12254 8330 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200982 BUTABARBITAL SODIUM 12255 8331 MYO9B 4650 NA PTHRP 10985428 12256 8332 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID29166791-Compound-AMPCP 12257 8333 PSME2 5721 NA inhibitor CARFILZOMIB CARFILZOMIB 12259 8334 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OFLOXACIN OFLOXACIN 22931300 12260 8335 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METITEPINE METITEPINE 12261 8336 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NITROFURANTOIN NITROFURANTOIN 22931300 12262 8337 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650943 12263 8338 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HOMIDIUM HOMIDIUM 12264 8339 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PROTOPORPHYRIN PROTOPORPHYRIN 12265 8340 PDE5A 8654 ENZYME, DRUGGABLE GENOME ENALAPRIL ENALAPRIL 15452190 12266 8341 ATXN2 6311 NA ALOXISTATIN ALOXISTATIN 12267 8342 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METITEPINE METITEPINE 12268 8343 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME GO-203-2c GO-203-2C 12269 8344 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-25 12271 8345 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201540 INSULIN SUSP ISOPHANE RECOMBINANT HUMAN 12272 8346 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OXYPHENONIUM BROMIDE OXYPHENONIUM BROMIDE 12274 8347 CIC 23152 CLINICALLY ACTIONABLE, DRUG RESISTANCE SELUMETINIB SELUMETINIB 28178529 12275 8348 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME INCB57643 12277 8349 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR BML-210 CHEMBL324053 16921367 12278 8350 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR DEHYDROEQUOL IDRONOXIL 12280 8351 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME ethinyl estradiol 17638512 12281 8352 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PTAEROXYLIN PTAEROXYLIN 12282 8353 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 12284 8354 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE venetoclax VENETOCLAX 12285 8355 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor 223366063 BOCOCIZUMAB 12286 8356 LST1 7940 NA abacavir ABACAVIR 12287 8357 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HALAZONE HALAZONE 12288 8358 MAPT 4137 DRUGGABLE GENOME QUINOLIN-6-YLAMINE CHEMBL99408 12289 8359 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200461 MIDODRINE HYDROCHLORIDE 12290 8360 ALOX15 246 ENZYME, DRUGGABLE GENOME PH-011685 CHEMBL126804 12291 8361 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 12294 8362 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MGCD-0103 MOCETINOSTAT 12296 8363 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE SELUMETINIB SELUMETINIB 12298 8364 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RALOXIFENE RALOXIFENE 22931300,21393461,21447734 12301 8365 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-24 12303 8366 GHRL 51738 DRUGGABLE GENOME PIOGLITAZONE PIOGLITAZONE 16682836 12304 8367 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER amiodarone AMIODARONE 12308 8368 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200334 MORICIZINE HYDROCHLORIDE 12309 8369 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200788 CISAPRIDE 12312 8370 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Doxepin DOXEPIN 12313 8371 VPS35 55737 ENZYME MELAGATRAN MELAGATRAN 22494098 12314 8372 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME omeprazole OMEPRAZOLE 15860653 12315 8373 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Saracatinib SARACATINIB 27231123 12316 8374 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME ALISERTIB ALISERTIB 12317 8375 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650744 CHEMBL270960 12318 8376 TARDBP 23435 TUMOR SUPPRESSOR NSC-92207 CHEMBL139935 12320 8377 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A11 12321 8378 PSMA2 5683 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL451887 CARFILZOMIB 12324 8379 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR NSC-88915 CHEMBL387152 19883083 12326 8380 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125149 CHEMBL547175 12327 8381 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME TRANILAST TRANILAST 12329 8382 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-12 12330 8383 GMNN 51053 DRUGGABLE GENOME TCMDC-124316 CHEMBL534214 12331 8384 COMT 1312 DRUGGABLE GENOME, ENZYME oxycodone OXYCODONE 28006928,23686330,21398039,23302985,26902643,29474345,23773341,25155931,25185591,19514130,28745577,27027462 12332 8385 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL2387080 TASELISIB 12334 8386 CPT1A 1374 DRUGGABLE GENOME, ENZYME PERHEXILINE PERHEXILINE 12335 8387 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CISATRACURIUM BESYLATE CISATRACURIUM BESYLATE 12336 8388 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE U0126 21358673 12337 8389 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL2103884 OPROZOMIB 12338 8390 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200705 HYDROXYAMPHETAMINE HYDROBROMIDE 12339 8391 ATXN2 6311 NA ENPIROLINE ENPIROLINE 12340 8392 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME REMOXIPRIDE REMOXIPRIDE 22931300 12341 8393 PRKG1 5592 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME GSK-269962A GSK-269962A 12342 8394 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124585 CHEMBL587856 12343 8395 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYSTAMINE CYSTAMINE 12345 8396 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE FASUDIL FASUDIL 22257127 12346 8397 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL576982 QUIZARTINIB 12347 8398 DNER 92737 NA Pyrimido-indole derivative 2 12350 8399 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR 12-EPI-SALVINORIN A 12-EPI-SALVINORIN A 22204910 12351 8400 PSMB9 5698 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 385612170 KZR-616 12352 8401 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 249565835 12353 8402 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 405067317 12354 8403 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GSK1059615 GSK-1059615 12356 8404 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FENRETINIDE FENRETINIDE 12357 8405 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102336 BOSUTINIB 12359 8406 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PKI-402 CHEMBL589258 20371716 12360 8407 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CERITINIB CERITINIB 23837797 12362 8408 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME tamsulosin TAMSULOSIN 12363 8409 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME INDIGOTINDISULFONATE INDIGOTINDISULFONATE 12364 8410 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor CHEMBL109480 TANESPIMYCIN 12365 8411 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID29324067-Compound-40 12367 8412 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PD-0166285 PD-0166285 12368 8413 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Ketotifen KETOTIFEN 12369 8414 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYDROCORTISONE HYDROCORTISONE 12371 8415 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL1200549 RAPACURONIUM BROMIDE 12375 8416 TUBA1A 7846 DRUGGABLE GENOME CHEMBL2105643 FOSBRETABULIN TROMETHAMINE 12376 8417 FAAH 2166 ENZYME, DRUGGABLE GENOME IPI-940 12378 8418 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Dipeptide analog 4 12379 8419 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651570 12381 8420 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545340 R-343 12383 8421 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR PROTEASOME INHIBITOR 16550004 12384 8422 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME CYC-116 CYC-116 12385 8423 KDM4A 9682 DRUGGABLE GENOME, ENZYME CLOTRIMAZOLE CLOTRIMAZOLE 12386 8424 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BIFEMELANE BIFEMELANE 12387 8425 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE MECASERMIN MECASERMIN 12390 8426 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 310264738 CERDULATINIB 12391 8427 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME IMATINIB IMATINIB 12392 8428 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AB928 AB-928 12395 8429 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR AKOS020330481 12396 8430 ALOX5 240 DRUGGABLE GENOME, ENZYME Tepoxalin TEPOXALIN 12399 8431 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor 178103171 12400 8432 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135649840 12403 8433 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4803 CHEMBL585240 12404 8434 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME RETINOIC ACID 17001699 12405 8435 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE 2-METHOXYPHENAZINE CHEMBL1420181 12406 8436 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist 135649905 12407 8437 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DIPYRIDAMOLE DIPYRIDAMOLE 12408 8438 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GEFITINIB GEFITINIB 12411 8439 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1059 PREGABALIN 12415 8440 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102549 12416 8441 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CAFFEINE CAFFEINE 10537077 12417 8442 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649649 12420 8443 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ACETYLSEROTONIN ACETYLSEROTONIN 12421 8444 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE AXITINIB AXITINIB 12423 8445 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ANTITHYMOCYTE GLOBULIN 12424 8446 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor 381744902 12425 8447 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE VANDETANIB VANDETANIB 12427 8448 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Bosutinib BOSUTINIB 12428 8449 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE YUANHUADINE YUANHUADINE 21916433 12430 8450 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-431542 SB-431542 12431 8451 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE HGF 18362143 12432 8452 HSPA9 3313 NA MKT-077 CHEMBL33859 12433 8453 DTNBP1 84062 KINASE citalopram CITALOPRAM 19065121 12434 8454 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE GDC-0068 IPATASERTIB 12439 8455 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-343227 CHEMBL1329326 12441 8456 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FINASTERIDE FINASTERIDE 10386468 12442 8457 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ANTHRALIN ANTHRALIN 12443 8458 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR LINIFANIB LINIFANIB 12444 8459 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702260 DEBIO-1347 12445 8460 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME XIMELAGATRAN XIMELAGATRAN 12446 8461 KMO 8564 DRUGGABLE GENOME, ENZYME PMID27172114-Compound-49 12447 8462 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200875 FLAVOXATE HYDROCHLORIDE 12448 8463 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE MSB2311 12449 8464 HTT 3064 DRUGGABLE GENOME INDOPROFEN INDOPROFEN 12450 8465 BAZ2B 29994 NA NALIDIXATE SODIUM NALIDIXATE SODIUM 12451 8466 GMNN 51053 DRUGGABLE GENOME DNDI1417447 CHEMBL1307453 12452 8467 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 5-AZA-2'-DEOXYCYTIDINE 14559817 12453 8468 H2AX 3014 NA TEMOZOLOMIDE TEMOZOLOMIDE 16024643 12454 8469 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR BIOFLAVONOID 16619521 12455 8470 KDM4A 9682 DRUGGABLE GENOME, ENZYME RAFOXANIDE RAFOXANIDE 12456 8471 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR STAUROSPORINE STAUROSPORINE 17167033 12458 8472 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR inhibitor 178103590 TAZEMETOSTAT 12459 8473 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME BESTATIN METHYL ESTER BESTATIN METHYL ESTER 21515062 12462 8474 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Lomustine LOMUSTINE 26762204 12463 8475 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE lapatinib LAPATINIB 12464 8476 POR 5447 ENZYME, DRUGGABLE GENOME midazolam MIDAZOLAM 23324807,19801957 12466 8477 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2011796857710 12467 8478 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-30 12468 8479 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Everolimus EVEROLIMUS 23629727,27797976,20664174,20664172,27217440 12469 8480 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ALFENTANIL HYDROCHLORIDE ALFENTANIL HYDROCHLORIDE 12473 8481 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-27 12475 8482 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 318164845 ABEDITEROL 12483 8483 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 381118872 12484 8484 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 135650608 MIFEPRISTONE 12485 8485 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL1201748 CABAZITAXEL 12486 8486 CRP 1401 DRUGGABLE GENOME fenofibrate FENOFIBRATE 12487 8487 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 381118812 MIZOLASTINE 12488 8488 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME KEPONE KEPONE 12489 8489 PCSK1 5122 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103178 12493 8490 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AZD8055 AZD-8055 26359452 12495 8491 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrazolopyridine derivative 4 12498 8492 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME agonist 178101085 N-METHYL-D-ASPARTIC ACID (NMDA) 12499 8493 ALOX15 246 ENZYME, DRUGGABLE GENOME NSC-119915 CHEMBL1481974 12500 8494 CBX1 10951 NA HYDROXYAMINE HYDROXYAMINE 12502 8495 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649987 BETAXOLOL 12503 8496 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PROPYLPYRAZOLETRIOL PROPYLPYRAZOLETRIOL 12504 8497 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 irbesartan IRBESARTAN 16094537,12359989,21842338 12505 8498 GAK 2580 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME SB-202190 SB-202190 22951114 12506 8499 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102697 12507 8500 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE MEK INHIBITOR PD0325901 23171796 12508 8501 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 12509 8502 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PSEUDOEPHEDRINE PSEUDOEPHEDRINE 12510 8503 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE R(-)-PROPYLNORAPOMORPHINE HCL CHEMBL538542 12511 8504 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Pembrolizumab PEMBROLIZUMAB 12512 8505 CBLC 23624 CLINICALLY ACTIONABLE, KINASE, ENZYME N/A 17671213 12513 8506 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE NEU-2000 12514 8507 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYDROQUINONE HYDROQUINONE 12515 8508 TLR7 51284 DRUGGABLE GENOME DSP-0509 12516 8509 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3,5-DIMETHOXYISONAPHTHOIC ACID CHEMBL1608067 12518 8510 NOTCH3 4854 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TAREXTUMAB TAREXTUMAB 25934888,24525742 12519 8511 HTT 3064 DRUGGABLE GENOME TRYPAN BLUE TRYPAN BLUE 12520 8512 PDE4A 5141 DRUGGABLE GENOME, ENZYME MILRINONE MILRINONE 12521 8513 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME HOMATROPINE METHYLBROMIDE 12523 8514 PSMD7 5713 PROTEASE PROTEASOME INHIBITOR 15221960 12524 8515 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 L-165041 CHEMBL153057 12525 8516 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL2110725 VINFLUNINE 12526 8517 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Cetuximab CETUXIMAB 26644315,27312529,28179366 12527 8518 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102817 12528 8519 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 12529 8520 CLCN6 1185 ION CHANNEL, DRUGGABLE GENOME antipsychotics 17976958 12530 8521 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE fam-trastuzumab deruxtecan-nxki 12535 8522 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200602 12536 8523 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000294102 CHEMBL607309 12537 8524 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor TRAMETINIB TRAMETINIB 12538 8525 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MONENSIN SODIUM MONENSIN SODIUM 12539 8526 RNASEH2A 10535 ENZYME TGFBETA1 15084595 12541 8527 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE CC-486 12542 8528 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102613 ISOGRANULATIMIDE 12543 8529 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME REGN-910 NESVACUMAB 12544 8530 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-159 CHEMBL599924 12545 8531 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 249565863 12546 8532 THBD 7056 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME SIMVASTATIN SIMVASTATIN 18663903 12547 8533 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE BROMODEOXYURIDINE 177889 12548 8534 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor XL-765 VOXTALISIB 12552 8535 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Pyrimidinyl compound 1 12553 8536 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1752 DYPHYLLINE 12556 8537 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE CYC-116 CYC-116 12557 8538 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor BELINOSTAT BELINOSTAT 12558 8539 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME CYANIDIN CYANIDIN 12559 8540 HMGCR 3156 ENZYME, DRUGGABLE GENOME Fluvastatin FLUVASTATIN 12560 8541 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102285 LINIFANIB 12561 8542 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR BUTANOIC ACID BUTANOIC ACID 19053749 12564 8543 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist 178100790 12565 8544 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME HPP-607 12566 8545 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PMID29130358-Compound-Figure10(2a) 12568 8546 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE MRX-4 CONTEZOLID ACEFOSAMIL 12570 8547 MAPT 4137 DRUGGABLE GENOME CARBOPLATIN CARBOPLATIN 12572 8548 TUBB 203068 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 12574 8549 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE IL-1RA ANAKINRA 9555664 12577 8550 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE IL-5 10961875 12578 8551 TSPO 706 DRUGGABLE GENOME Pyrazolopyrimidine acetamide analog 1 12581 8552 DYRK2 8445 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID28766366-Compound-Scheme21Left 12582 8553 ENO2 2026 CELL SURFACE NERVE GROWTH FACTOR 6793214 12583 8554 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME activator 53801022 12584 8555 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1201020 DISOPYRAMIDE PHOSPHATE 12585 8556 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BCMA CART and huCART19 12586 8557 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME EVT-201 12587 8558 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-228155 CHEMBL505670 12588 8559 PREP 5550 PROTEASE, ENZYME, DRUGGABLE GENOME ONO-1603 CHEMBL1087333 12591 8560 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME LY-2090314 LY-2090314 12592 8561 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ERLOTINIB ERLOTINIB 17877814,21258250,23470965,27664271,26773740,15310767,26768165,32193290,21841502,25668228,25179728,20826716,21783417,22901364,17085664,24353160,26124334,24736073,15329413,24636847,22285168,29290255,16282176,28874593,20942962,16014883,25521405,19147750,24868098,24457318,17177598,27304188,21531810,21969500,16818686 12594 8562 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME HYDROGEN PEROXIDE 15304367 12595 8563 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE US9567304, Compound N-9 12596 8564 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ANTISENSE OLIGONUCLEOTIDES 9092554 12597 8565 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 315661343 12600 8566 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME DDP 15970709 12601 8567 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 2-MERCAPTOBENZOTHIAZOLE 2-MERCAPTOBENZOTHIAZOLE 24262887 12602 8568 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME dapoxetine DAPOXETINE 26937172 12603 8569 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CHEMBL1743058 PONEZUMAB 12606 8570 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CONJUGATED ESTROGENS 12607 8571 KCNA7 3743 ION CHANNEL, DRUGGABLE GENOME blocker 135649937 AMIODARONE 12608 8572 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR ESTAZOLAM ESTAZOLAM 22137933 12609 8573 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 6'-IODONONIVAMIDE CHEMBL177809 12614 8574 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ZIRAM ZIRAM 12615 8575 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE MOMELOTINIB MOMELOTINIB 12616 8576 C1S 716 ENZYME, PROTEASE, DRUGGABLE GENOME TNT009 12617 8577 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME BIVALIRUDIN BIVALIRUDIN 12619 8578 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL3301587 DURVALUMAB 12620 8579 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE OPIOIDS 10232386 12621 8580 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TRAZODONE TRAZODONE 12624 8581 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE NINTEDANIB NINTEDANIB 12625 8582 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PWT-33597 23066039 12626 8583 CSNK2A2 1459 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME, TRANSCRIPTION FACTOR inhibitor HESPERADIN HESPERADIN 19035792 12628 8584 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CYPROTERONE CYPROTERONE 22931300 12629 8585 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ZAPA ZAPA 12631 8586 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270010-Compound-Figure17-2 12632 8587 KRT10 3858 CELL SURFACE EGFR TYROSINE KINASE INHIBITOR 10601294 12634 8588 POLK 51426 DNA REPAIR, ENZYME PIRARUBICIN PIRARUBICIN 12635 8589 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR PD 0332991 12636 8590 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR MECHLORETHAMINE HYDROCHLORIDE MECHLORETHAMINE HYDROCHLORIDE 12638 8591 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor 178101328 12640 8592 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME 681640 CHEMBL379975 12641 8593 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545339 FRUQUINTINIB 12643 8594 SLC16A1 6566 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME SODIUM BUTYRATE 11882670 12645 8595 SRPK2 6733 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565786 12646 8596 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GUTHION GUTHION 12648 8597 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY NALTREXONE NALTREXONE 9623517 12650 8598 GUCY1A2 2977 ENZYME, DRUGGABLE GENOME activator CHEMBL1311 ISOSORBIDE MONONITRATE 12651 8599 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-24 12653 8600 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2165191 AZD-6482 12655 8601 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE ISOPRENALINE ISOPROTERENOL 12656 8602 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651541 EPOPROSTENOL 12657 8603 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1200335 TESTOSTERONE ENANTHATE 12658 8604 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DNDI1417072 CHEMBL1310701 12659 8605 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4832 CHEMBL601137 12660 8606 BRCA2 675 CLINICALLY ACTIONABLE PR-104 PR-104 25193512 12662 8607 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 6 12664 8608 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 alprazolam ALPRAZOLAM 32112986 12665 8609 F2RL3 9002 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 329968398 12666 8610 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SCH-58261 SCH-58261 12667 8611 TAC1 6863 DRUGGABLE GENOME FUROSEMIDE FUROSEMIDE 2048822 12668 8612 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL190 THEOPHYLLINE 12669 8613 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME CLOBETASOL CLOBETASOL 12674 8614 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL1683544 ERIBULIN MESYLATE 12675 8615 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME METIZOLINE METIZOLINE 12676 8616 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME RHEIN RHEIN 12677 8617 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL2105081 FRAKEFAMIDE 12678 8618 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR CYCLOSPORIN A 10642325 12679 8619 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-20 12682 8620 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME activator 135650820 12686 8621 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 VISNAGIN VISNAGIN 12690 8622 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 178102513 PONATINIB 12691 8623 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME N/A 12692 8624 INHBA 3624 CLINICALLY ACTIONABLE, GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME inhibitor CHEMBL1743073 SOTATERCEPT 12693 8625 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CINNARIZINE CINNARIZINE 16680159 12695 8626 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 THIAMYLAL SODIUM THIAMYLAL SODIUM 12697 8627 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 fluvastatin FLUVASTATIN 16103896 12698 8628 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TRIAMCINOLONE TRIAMCINOLONE 10199793 12699 8629 KCNA7 3743 ION CHANNEL, DRUGGABLE GENOME blocker 135651305 VERAPAMIL 12701 8630 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-34b 12702 8631 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Six-membered heterocyclic benzamide derivative 6 12703 8632 SMN1 6606 DRUGGABLE GENOME 7-HYDROXY ISOFLAVONE 7-HYDROXY ISOFLAVONE 12704 8633 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CYC-116 CYC-116 12706 8634 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE ABBV-2451 12708 8635 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TELENZEPINE TELENZEPINE 12710 8636 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR MADOLIN U MADOLIN U 12712 8637 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME CTS-21166 12713 8638 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ISIS-CRP 12714 8639 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CEFACLOR CEFACLOR 22166395 12715 8640 GMNN 51053 DRUGGABLE GENOME GNF-PF-2272 CHEMBL601757 12716 8641 ST14 6768 ENZYME, DRUGGABLE GENOME, PROTEASE US8569313, Inhibitor 14 12717 8642 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE benzene BENZENE 15935810 12719 8643 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL580 LORAZEPAM 12721 8644 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE CORTISOL HYDROCORTISONE 2115769 12722 8645 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PROTOPORPHYRIN PROTOPORPHYRIN 12723 8646 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE LAPATINIB LAPATINIB 23404373,22511346 12725 8647 SMN1 6606 DRUGGABLE GENOME CID 1245272 CHEMBL408850 12726 8648 SORCS2 57537 NA atazanavir ATAZANAVIR 31562781 12727 8649 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME FLUORODIFEN FLUORODIFEN 12728 8650 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PERTUZUMAB PERTUZUMAB 29320312 12733 8651 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME ILORASERTIB ILORASERTIB 12734 8652 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE CHEMBL1742992 BLINATUMOMAB 12736 8653 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PD98059 14534538 12737 8654 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MELATONIN MELATONIN 12740 8655 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor TOZASERTIB TOZASERTIB 12742 8656 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL289351 FOSBRETABULIN DISODIUM 12743 8657 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178103273 KETOROLAC 12744 8658 BAZ2B 29994 NA CHLORTETRACYCLINE HYDROCHLORIDE CHLORTETRACYCLINE HYDROCHLORIDE 12745 8659 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GW775608X GW775608X 18602262 12746 8660 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor CHEMBL3544967 GSK-2256098 12747 8661 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL3545167 FE 202767 12748 8662 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME STEARIC ACID STEARIC ACID 12749 8663 IDS 3423 ENZYME, DRUGGABLE GENOME Idursulfase IDURSULFASE 12750 8664 GMNN 51053 DRUGGABLE GENOME CGP-74514A CHEMBL1256911 12752 8665 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ATORVASTATIN ATORVASTATIN 16139565 12755 8666 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL1980297 ILORASERTIB 12757 8667 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE CAR-GPC3 T Cells 12759 8668 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME SB19065 12760 8669 GADD45A 1647 DNA REPAIR, TUMOR SUPPRESSOR, KINASE WORTMANNIN WORTMANNIN 12066222 12761 8670 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NORTRIPTYLINE HYDROCHLORIDE NORTRIPTYLINE HYDROCHLORIDE 12762 8671 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 135650365 IBUPROFEN 12763 8672 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GSK1482160 GSK1482160 12764 8673 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME PROGESTIN PROGESTERONE 9052414 12765 8674 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MK-571 MK-571 12767 8675 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME LOMOFUNGIN LOMOFUNGIN 12768 8676 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BUFLOMEDIL BUFLOMEDIL 12769 8677 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ENMD-2076 ENMD-2076 12770 8678 KMO 8564 DRUGGABLE GENOME, ENZYME Cyclopropane 1-carboxylic acid derivative 8 12771 8679 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BACLOFEN BACLOFEN 7674378,9486305 12772 8680 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-67436 CHEMBL1331995 12774 8681 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE FENRETINIDE FENRETINIDE 12775 8682 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CARMINE CARMINE 12776 8683 GMNN 51053 DRUGGABLE GENOME VINCRISTINE SULFATE VINCRISTINE SULFATE 12777 8684 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR GO-6976 GO-6976 12778 8685 ALPL 249 ENZYME, DRUGGABLE GENOME CEPHALOCHROMIN CEPHALOCHROMIN 12779 8686 TUBA3C 7278 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 12780 8687 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME DONEPEZIL DONEPEZIL 12781 8688 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY DES DIETHYLSTILBESTROL 10650935 12782 8689 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9522888, 575 12783 8690 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR SJ000029700 CHEMBL591864 12784 8691 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE FLUSPIRILENE FLUSPIRILENE 12785 8692 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME PIROXICAM PIROXICAM 10716720 12787 8693 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ITRACONAZOLE ITRACONAZOLE 15969931 12788 8694 SERPINA5 5104 PROTEASE INHIBITOR, ENZYME, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE THROMBIN THROMBIN 8136018 12789 8695 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE BENZANTHRONE BENZANTHRONE 12790 8696 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME HUMAN CHORIONIC GONADOTROPIN 17823853 12792 8697 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME SEIMATOPOLIDE A SEIMATOPOLIDE A 22424300 12796 8698 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE partial agonist CHEMBL3545230 APIMOSTINEL 12799 8699 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 649849 CHEMBL405914 12800 8700 H2AW 92815 NA TRICHOSTATIN A 15292402 12801 8701 SMN1 6606 DRUGGABLE GENOME INDOPROFEN INDOPROFEN 12802 8702 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE OSI-632 OSI-632 12803 8703 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME dextromethorphan / quinidine 12804 8704 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE G-CSF FILGRASTIM 11391619 12807 8705 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-1241 CHEMBL528724 12808 8706 LSS 4047 ENZYME, DRUGGABLE GENOME inhibitor 178103320 12809 8707 GNMT 27232 ENZYME l-methionine METHIONINE 24651765 12812 8708 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY CORTISOL HYDROCORTISONE 7716064 12814 8709 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE GW441756X GW441756X 12815 8710 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL2103868 CABOZANTINIB S-MALATE 12817 8711 CD38 952 CELL SURFACE, DRUGGABLE GENOME CART-38 cells 12819 8712 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565850 12820 8713 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor SORAFENIB SORAFENIB 12821 8714 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051802 12822 8715 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 310264749 SERABELISIB 12827 8716 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TREQUINSIN TREQUINSIN 12830 8717 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL428690 ALVOCIDIB 12831 8718 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DESOXIMETASONE DESOXIMETASONE 12832 8719 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200472 QUAZEPAM 12833 8720 NDUFA13 51079 ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 12834 8721 BAZ2B 29994 NA NSC-377852 CHEMBL1466186 12835 8722 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUTICASONE PROPIONATE 12836 8723 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME AS1402 HUHMFG1 12837 8724 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR CISPLATIN CISPLATIN 21273582 12838 8725 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 178101973 12839 8726 PDE10A 10846 ENZYME, DRUGGABLE GENOME 1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 4 12843 8727 NDUFS5 4725 ENZYME inhibitor CHEMBL3545135 NV-128 12846 8728 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME SERTRALINE SERTRALINE 12847 8729 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Sodium butyrate 12849 8730 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER bupropion BUPROPION 22947179 12850 8731 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DOXACURIUM DOXACURIUM 12851 8732 CYP27B1 1594 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ribavirin RIBAVIRIN 21145801 12854 8733 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Gold-complexed thiosaccharide derivative 1 12855 8734 ATAD5 79915 NA DIGITOXIN DIGITOXIN 12860 8735 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200914 TAMSULOSIN HYDROCHLORIDE 12862 8736 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL1795071 RUXOLITINIB PHOSPHATE 12864 8737 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1719 OLOPATADINE HYDROCHLORIDE 12865 8738 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 12866 8739 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR CISPLATIN CISPLATIN 12917817 12868 8740 DNPEP 23549 ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE inhibitor 252166877 12869 8741 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178103087 MORPHANTHRIDINE 12870 8742 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MAPROTILINE MAPROTILINE 12871 8743 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MK-886 CHEMBL29097 12872 8744 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650568 12873 8745 PPIB 5479 ENZYME, DRUGGABLE GENOME L-Proline PROLINE 12874 8746 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CAFFEINE CAFFEINE 1339096 12875 8747 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR TRIAMCINOLONE TRIAMCINOLONE 12174062 12877 8748 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL3545079 PLX-5622 12878 8749 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor LINSITINIB LINSITINIB 12879 8750 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AZD-1152-HQPA AZD-1152-HQPA 12880 8751 ABCC5 10057 DRUGGABLE GENOME, ABC TRANSPORTER, TRANSPORTER irinotecan IRINOTECAN 26352872 12881 8752 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Troglitazone TROGLITAZONE 12882 8753 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL haloperidol HALOPERIDOL 27023437 12883 8754 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR REL-BENDIGOLE F CHEMBL1915271 21684166 12884 8755 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE SNS-314 SNS-314 12885 8756 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545052 FIMEPINOSTAT 12886 8757 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 310264675 CUDC-101 12887 8758 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AG-490 CHEMBL56543 12888 8759 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME PF-562271 PF-00562271 12889 8760 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE quetiapine QUETIAPINE 24240480,18695978 12890 8761 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Bevacizumab BEVACIZUMAB 21216929 12894 8762 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NORETHINDRONE ACETATE NORETHINDRONE ACETATE 12895 8763 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650339 GW7647 12896 8764 ALDH1A1 216 DRUGGABLE GENOME, ENZYME AZACITIDINE AZACITIDINE 12898 8765 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MEFENAMIC ACID MEFENAMIC ACID 22931300 12899 8766 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL52885 ENMD-981693 12900 8767 RBP4 5950 DRUGGABLE GENOME US9434727, 120 12901 8768 ATXN2 6311 NA GNF-PF-1644 CHEMBL600734 12902 8769 XDH 7498 DRUGGABLE GENOME, ENZYME FENTANYL FENTANYL 9637647 12903 8770 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME GNF-PF-1969 CHEMBL601364 12904 8771 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 isoniazid ISONIAZID 20941486 12905 8772 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AZD-5438 AZD-5438 12906 8773 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER oxycodone OXYCODONE 21209234,19514130 12908 8774 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IODOACETAMIDE IODOACETAMIDE 12909 8775 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE leucovorin LEUCOVORIN 18245544,17700593,29845393,27864592,20819423,29134491,25331073,20385995,27557140,24980946,23407049 12913 8776 HPGDS 27306 ENZYME, DRUGGABLE GENOME Praziquantel PRAZIQUANTEL 12914 8777 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER STZ STREPTOZOCIN 1722397 12916 8778 IL23A 51561 DRUGGABLE GENOME ustekinumab USTEKINUMAB 12917 8779 CCL21 6366 DRUGGABLE GENOME LT-BETA 15632007 12918 8780 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PF-04691502 PF-04691502 12921 8781 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CID 1540951 CHEMBL259421 12922 8782 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1684984 PA-799 12923 8783 SH2B1 25970 KINASE risperidone RISPERIDONE 28694205 12925 8784 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 4,4'-DITHIODIPYRIDINE CHEMBL1232076 12926 8785 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE GNF-PF-3955 CHEMBL605747 12928 8786 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 310264688 EDAGLITAZONE 12929 8787 PTHLH 5744 HORMONE ACTIVITY, DRUGGABLE GENOME DIFFERENTIATION AGENTS 10839458 12930 8788 APC 324 CLINICALLY ACTIONABLE DIFLUOROMETHYLORNITHINE 10766173 12931 8789 NOS2 4843 DRUGGABLE GENOME, ENZYME KD7040 KD7040 12933 8790 WNK1 65125 SERINE THREONINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 252827493 12935 8791 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 223366141 12936 8792 ARG1 383 ENZYME L-2-AMINOHISTIDINE CHEMBL1099167 20441173 12937 8793 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME HEPARIN CALCIUM 17322644 12938 8794 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9670220, 33 12939 8795 KDM4A 9682 DRUGGABLE GENOME, ENZYME KAINIC ACID KAINIC ACID 12940 8796 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE dexamethasone DEXAMETHASONE 26521987 12942 8797 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 1-NAPHTHYLISOTHIOCYANATE 1-NAPHTHYLISOTHIOCYANATE 12944 8798 TXNRD1 7296 DRUGGABLE GENOME 4-aryl quinol derivative 4 12945 8799 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR PLATINUM PLATINUM 8110490 12947 8800 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME GABOXADOL GABOXADOL 12949 8801 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR THIOMERSAL THIMEROSAL 12950 8802 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135649941 AMOXAPINE 12952 8803 CACNB4 785 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1059 PREGABALIN 12954 8804 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME Pyrazolo-triazine derivative 2 12955 8805 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NITROMIDE NITROMIDE 12957 8806 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYCLOVALONE CYCLOVALONE 12958 8807 ELAVL1 1994 DRUGGABLE GENOME DEHYDROMUTACTIN DEHYDROMUTACTIN 17632515 12960 8808 PACSIN2 11252 KINASE, TRANSPORTER methotrexate METHOTREXATE 22846425 12962 8809 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME NICLOSAMIDE NICLOSAMIDE 12964 8810 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RG-1530 RG-1530 12965 8811 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALUM 11768621 12966 8812 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ASTEMIZOLE ASTEMIZOLE 12967 8813 PARG 8505 ENZYME BENZAMIDE BENZAMIDE 21692479 12968 8814 HTT 3064 DRUGGABLE GENOME BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 12970 8815 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BPDE 8866791 12971 8816 IMPDH1 3614 ENZYME, DRUGGABLE GENOME VX-944 12973 8817 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME MGCD-0103 MOCETINOSTAT 12974 8818 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE VINBLASTINE VINBLASTINE 10590059 12977 8819 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrrolo-pyridine derivative 3 12979 8820 POLK 51426 DNA REPAIR, ENZYME AMINACRINE AMINACRINE 12982 8821 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME LY294002 23039341 12984 8822 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE POH 16439861 12985 8823 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR QUERCETIN QUERCETIN 25190466 12987 8824 ATXN2 6311 NA PERPHENAZINE PERPHENAZINE 12989 8825 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ZOLANTIDINE ZOLANTIDINE 12991 8826 BAZ2B 29994 NA 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 12992 8827 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor 178103691 ANAGRELIDE 12994 8828 SPP1 6696 DRUGGABLE GENOME TYROSINE KINASE INHIBITOR 12176960 12995 8829 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-34c 12996 8830 CBX1 10951 NA FLUPHENAZINE FLUPHENAZINE 12997 8831 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FAMPROFAZONE FAMPROFAZONE 12999 8832 AREG 374 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE CETUXIMAB CETUXIMAB 23374602 13000 8833 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2015042088Example11 13002 8834 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL1944698 ZOTIRACICLIB 13003 8835 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Obatoclax OBATOCLAX 13004 8836 GBA 2629 DRUGGABLE GENOME, ENZYME SULFANITRAN SULFANITRAN 13005 8837 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mercaptopurine MERCAPTOPURINE 13006 8838 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Duloxetine DULOXETINE 13007 8839 GMNN 51053 DRUGGABLE GENOME TCMDC-125733 CHEMBL530788 13008 8840 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE NAC ACETYLCYSTEINE 12485928 13009 8841 UGT2B7 7364 DRUGGABLE GENOME buprenorphine BUPRENORPHINE 24256307 13010 8842 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565876 13012 8843 CALM1 801 ION CHANNEL, KINASE, ENZYME, DRUGGABLE GENOME FLUNARIZINE FLUNARIZINE 13013 8844 DDC 1644 ENZYME, DRUGGABLE GENOME Benserazide BENSERAZIDE 13014 8845 MAPT 4137 DRUGGABLE GENOME INDIGOTINDISULFONATE INDIGOTINDISULFONATE 13015 8846 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 385612249 13016 8847 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CITROPTEN CITROPTEN 13017 8848 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME NITRAZEPAM NITRAZEPAM 13018 8849 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650029 13019 8850 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-3407 CHEMBL602990 13020 8851 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 12-METHYL TETRADECANOIC ACID CHEMBL495852 13021 8852 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103856 PROMETHAZINE 13025 8853 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 404859096 13027 8854 NDUFB3 4709 ENZYME inhibitor CHEMBL3545320 ME-344 13028 8855 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MITOXANTRONE MITOXANTRONE 9494516,9426516 13029 8856 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE PINOCEMBRIN PINOCEMBRIN 13031 8857 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME ETRAVIRINE ETRAVIRINE 21189339 13032 8858 NEK4 6787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TAMATINIB R-406 13033 8859 TYMP 1890 GROWTH FACTOR, DRUGGABLE GENOME FLUOROURACIL FLUOROURACIL 11205264 13034 8860 PDE4A 5141 DRUGGABLE GENOME, ENZYME ROLIPRAM ROLIPRAM 13036 8861 SULT1A1 6817 DRUGGABLE GENOME, ENZYME acetaminophen ACETAMINOPHEN 30908574,23462933,26049587,6957279 13038 8862 MAPT 4137 DRUGGABLE GENOME DEPHOSTATIN DEPHOSTATIN 13039 8863 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MUNDULONE MUNDULONE 13042 8864 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ORYZALIN ORYZALIN 13043 8865 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLOBAZAM CLOBAZAM 13045 8866 PTGS1 5742 ENZYME, DRUGGABLE GENOME ETODOLAC ETODOLAC 13046 8867 COMT 1312 DRUGGABLE GENOME, ENZYME Analgesics 25096645 13047 8868 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR ZINC915379 13048 8869 GMNN 51053 DRUGGABLE GENOME LORATADINE LORATADINE 13049 8870 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME sorafenib SORAFENIB 22736425,24510746 13052 8871 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME interferons 23360626 13053 8872 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME L-alanyl-l-glutamine ALANYL GLUTAMINE 13054 8873 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME DABRAFENIB DABRAFENIB 24265153,25452114 13055 8874 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE NILOTINIB NILOTINIB 18191450 13056 8875 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LIOTHYRONINE LIOTHYRONINE 13058 8876 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR 2-CDA CLADRIBINE 15813915 13059 8877 DNER 92737 NA RG6146 13061 8878 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL661 ALPRAZOLAM 13064 8879 DHFR 1719 DRUGGABLE GENOME, ENZYME MITOMYCIN-C 1332730 13065 8880 PLA2G7 7941 DRUGGABLE GENOME, ENZYME Rilapladib RILAPLADIB 13068 8881 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PMID28048944-Compound-7 13070 8882 IL1B 3553 KINASE, DRUGGABLE GENOME aspirin ASPIRIN 19448967 13071 8883 ALDH1A1 216 DRUGGABLE GENOME, ENZYME VALERENIC ACID VALERENIC ACID 13074 8884 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME ribavirin RIBAVIRIN 13077 8885 MAPT 4137 DRUGGABLE GENOME DIHYDROERGOTAMINE DIHYDROERGOTAMINE 13078 8886 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CARBIDOPA CARBIDOPA 13079 8887 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME CENISERTIB CENISERTIB 13080 8888 OGDH 4967 NA CPI-613 13081 8889 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GNF-PF-5134 CHEMBL602969 13082 8890 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Bicyclic heteroaryl benzamide derivative 9 13083 8891 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-32984 CHEMBL1339015 13085 8892 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565850 13087 8893 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-11437 CHEMBL1814509 13088 8894 MAPT 4137 DRUGGABLE GENOME DAUNORUBICIN DAUNORUBICIN 13089 8895 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-5061 CHEMBL601385 13090 8896 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 2-(STYRYL)-BENZIMIDAZOLE CHEMBL473721 13091 8897 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CETIRIZINE CETIRIZINE 13092 8898 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ANESTHETICS 15041592 13093 8899 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SUFENTANIL CITRATE SUFENTANIL CITRATE 13095 8900 ECE1 1889 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE SLV-338 13097 8901 GMNN 51053 DRUGGABLE GENOME CILNIDIPINE CILNIDIPINE 13098 8902 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE XL880 FORETINIB 13099 8903 CXCL8 3576 DRUGGABLE GENOME IL-1 2250017 13101 8904 STX11 8676 NA emapalumab EMAPALUMAB 13103 8905 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL Diquafosol DIQUAFOSOL 13104 8906 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME PI-103 PI-103 13106 8907 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR ADENOVIRUS VECTOR 16014023 13109 8908 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ANTISERUM 10962349 13111 8909 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HOMIDIUM BROMIDE HOMIDIUM BROMIDE 13115 8910 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (+/-)-PENTAACETYLCATECHIN (+/-)-PENTAACETYLCATECHIN 13118 8911 POLI 11201 DNA REPAIR NSC-348401 CHEMBL515505 13120 8912 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME isoniazid ISONIAZID 25798582,29036176,27281183 13122 8913 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2387080 TASELISIB 13123 8914 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME DOXORUBICIN DOXORUBICIN 18174247 13124 8915 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PIPERTRAMINE AMIDE PIPERTRAMINE AMIDE 13126 8916 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE l-methylfolate 27035272,27520898,31058543 13128 8917 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Isoindoline derivative 2 13129 8918 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE citalopram CITALOPRAM 18695978 13130 8919 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR DOXORUBICIN DOXORUBICIN 10728907 13132 8920 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR ACACETIN ACACETIN 25190466 13133 8921 VKORC1 79001 DRUGGABLE GENOME, ENZYME DICUMAROL DICUMAROL 13134 8922 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Tri-substituted purine derivative 1 13135 8923 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178100911 13137 8924 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Indoline derivative 20 13138 8925 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL6318 IDOXIFENE 13139 8926 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2105732 LEVOMILNACIPRAN HYDROCHLORIDE 13141 8927 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR AFURESERTIB HYDROCHLORIDE 13142 8928 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 223366204 COPANLISIB 13143 8929 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SILODOSIN SILODOSIN 13144 8930 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME REPOTRECTINIB REPOTRECTINIB 30093503 13147 8931 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL940 GABAPENTIN 13149 8932 MAPT 4137 DRUGGABLE GENOME EMODIC ACID EMODIC ACID 13151 8933 MBTPS1 8720 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, PROTEASE inhibitor 252827485 13152 8934 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL AZIETOMIDATE AZIETOMIDATE 16884293 13155 8935 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103857 EDIVOXETINE 13156 8936 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME CD10-CART 13157 8937 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR UROKINASE UROKINASE 13159 8938 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LOMOFUNGIN LOMOFUNGIN 13160 8939 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE XL-820 XL-820 13161 8940 RGS4 5999 DRUGGABLE GENOME DIGOXIN DIGOXIN 13162 8941 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ORTHO-PHTHALALDEHYDE ORTHO-PHTHALALDEHYDE 13163 8942 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor PD 0325901 13164 8943 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME ARQ092 26469692 13165 8944 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME AG-881 13166 8945 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX CID 739615 CHEMBL260560 13167 8946 PTGS2 5743 DRUGGABLE GENOME, ENZYME SC-75416 13170 8947 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL403989 TG100-801 13172 8948 AKR1B1 231 DRUGGABLE GENOME, ENZYME GROWTH AGENTS 9371720 13173 8949 PNPLA3 80339 ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 28744905 13174 8950 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CALCIPOTRIENE CALCIPOTRIENE 13175 8951 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CISPLATIN CISPLATIN 25010864 13176 8952 TUBB6 84617 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 13177 8953 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER pentazocine PENTAZOCINE 13179 8954 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME EVT-101 EVT-101 13181 8955 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Brexpiprazole BREXPIPRAZOLE 13182 8956 MAPT 4137 DRUGGABLE GENOME GNF-PF-5114 CHEMBL601952 13183 8957 PDE3A 5139 ENZYME, DRUGGABLE GENOME hydrochlorothiazide HYDROCHLOROTHIAZIDE 31327267 13184 8958 EPHA4 2043 DRUGGABLE GENOME, KINASE, CELL SURFACE, TYROSINE KINASE inhibitor CHEMBL24828 VANDETANIB 13185 8959 PTGS1 5742 ENZYME, DRUGGABLE GENOME PIROXICAM PIROXICAM 13186 8960 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE OSI-632 OSI-632 13187 8961 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CID 867101 CHEMBL406557 13188 8962 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME INDINAVIR INDINAVIR 22931300 13189 8963 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GW7647 GW7647 13190 8964 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 13191 8965 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL ALPRAZOLAM ALPRAZOLAM 13193 8966 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME EC0489 13194 8967 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody CIXUTUMUMAB CIXUTUMUMAB 13197 8968 LRP2 4036 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, KINASE cisplatin CISPLATIN 23274376,31666714,17457342 13198 8969 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CYPATE CYPATE 22871580 13199 8970 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME MEDROXYPROGESTERONE MEDROXYPROGESTERONE ACETATE 15885761 13202 8971 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME ETOPOSIDE ETOPOSIDE 15454884 13203 8972 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ENZYME INHIBITOR 15619341 13204 8973 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR PHA-767491 CHEMBL225519 13205 8974 KDM4A 9682 DRUGGABLE GENOME, ENZYME S-NITROSOGLUTATHIONE S-NITROSOGLUTATHIONE 13206 8975 NEK4 6787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DOVITINIB DOVITINIB 13208 8976 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR PQR309 BIMIRALISIB 13209 8977 SMN1 6606 DRUGGABLE GENOME DIBENZOYLMETHANE DIBENZOYLMETHANE 13212 8978 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NVP-AUY922 LUMINESPIB 13213 8979 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 249565749 13215 8980 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 387065624 13216 8981 POLK 51426 DNA REPAIR, ENZYME EMODIC ACID EMODIC ACID 13217 8982 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BELINOSTAT BELINOSTAT 13220 8983 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-228155 CHEMBL505670 13222 8984 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR L-165041 CHEMBL153057 13223 8985 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME METHYLDOPA METHYLDOPA 13224 8986 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE ZAPRINAST ZAPRINAST 13225 8987 SMN1 6606 DRUGGABLE GENOME PIPERINE PIPERINE 13227 8988 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor TAK901 13230 8989 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE MEK162 BINIMETINIB 26577700 13232 8990 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545154 POZIOTINIB 13233 8991 GMNN 51053 DRUGGABLE GENOME E319 E319 13234 8992 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor BI847325 13235 8993 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE DNDI1417467 CHEMBL1997335 13236 8994 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE allosteric modulator 315661243 13237 8995 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 893238 CHEMBL473735 13239 8996 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Dextromethorphan DEXTROMETHORPHAN 13240 8997 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE IL-2 ALDESLEUKIN 8938794 13241 8998 HSPA4 3308 NA NIMESULIDE NIMESULIDE 9645681 13242 8999 COMT 1312 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1324 TOLCAPONE 13246 9000 PSENEN 55851 DRUGGABLE GENOME BMS-299897 CHEMBL247471 13248 9001 FABP3 2170 NA inhibitor 252827455 13250 9002 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Gemcitabine GEMCITABINE 28750271 13251 9003 VKORC1 79001 DRUGGABLE GENOME, ENZYME inhibitor 135651418 ALITRETINOIN 13252 9004 MAOA 4128 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 3 13253 9005 TOP2B 7155 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL452231 TENIPOSIDE 13254 9006 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE BKM120 BUPARLISIB 28119489 13257 9007 RAB9A 9367 ENZYME, DRUGGABLE GENOME PTEROSTILBENE PTEROSTILBENE 13258 9008 CTSE 1510 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103180 13259 9009 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PSEUDOEPHEDRINE PSEUDOEPHEDRINE 13260 9010 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 310264784 CHEMBL442577 13263 9011 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE G-CSF FILGRASTIM 16331631 13266 9012 ST6GAL1 6480 DRUGGABLE GENOME flucloxacillin FLOXACILLIN 19483685 13267 9013 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CETUXIMAB CETUXIMAB 29196463,24653627,24934779,26888827,28287083,18003960,22152101,22270724,24894453,18794099 13268 9014 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME METHAMPHETAMINE METHAMPHETAMINE 13269 9015 TMEM97 27346 NA PMID30185082-Compound-28 13271 9016 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 53801090 CAPSAICIN 13272 9017 CACNB4 785 DRUGGABLE GENOME, ION CHANNEL SAFINAMIDE SAFINAMIDE 13273 9018 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME Rosiglitazone + metformin 13275 9019 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SAR245409 VOXTALISIB 24634413 13276 9020 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE DNDI1417353 CHEMBL1481721 13277 9021 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME bevacizumab BEVACIZUMAB 27503580 13279 9022 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 660258 CHEMBL259805 13280 9023 KLB 152831 ENZYME NGM313 13283 9024 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME LORAZEPAM LORAZEPAM 13284 9025 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650309 13285 9026 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Quinoline carboxamide derivative 3 13287 9027 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TAMOXIFEN TAMOXIFEN 13288 9028 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 13289 9029 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER agonist CHEMBL983 SUCCINYLCHOLINE CHLORIDE 13291 9030 UBE2I 7329 TRANSCRIPTION FACTOR BINDING, ENZYME cisplatin CISPLATIN 19859084 13293 9031 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178102633 MUBRITINIB 13295 9032 EYA2 2139 DNA REPAIR GNF-PF-3418 CHEMBL582099 13296 9033 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL ARVERAPAMIL 13297 9034 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Rosiglitazone + metformin 13298 9035 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652006 13299 9036 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ARQ092 26469692 13301 9037 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE MANSONONE F MANSONONE F 21600681 13302 9038 MAPT 4137 DRUGGABLE GENOME DIHYDROERGOCRISTINE MESYLATE DIHYDROERGOCRISTINE MESYLATE 13304 9039 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL phenytoin PHENYTOIN 17001291 13305 9040 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR CI-1040 CI-1040 13306 9041 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE GARCINOL GARCINOL 13308 9042 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1370561 AMINOPHYLLINE 13309 9043 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME VANDETANIB VANDETANIB 13310 9044 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CORALYNE CORALYNE 13311 9045 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135649880 13312 9046 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 252166787 13314 9047 KDM4A 9682 DRUGGABLE GENOME, ENZYME 5-NITRO-[1,10]PHENANTHROLINE CHEMBL101815 13315 9048 FXYD2 486 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL3545057 ACETYLDIGITOXIN 13316 9049 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME PREGABALIN PREGABALIN 13319 9050 RPS6KB2 6199 DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME, KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545003 MSC-2363318A 13322 9051 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PD-81723 CHEMBL59532 13323 9052 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME CENISERTIB CENISERTIB 13324 9053 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FIPRONIL FIPRONIL 13325 9054 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME R(-)-PROPYLNORAPOMORPHINE HCL CHEMBL538542 13327 9055 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR JNJ-7777120 JNJ-7777120 21920751 13329 9056 XPO1 7514 CLINICALLY ACTIONABLE, KINASE Selinexor oral 13330 9057 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR U-74389G MALEATE CHEMBL1256186 13331 9058 MAPT 4137 DRUGGABLE GENOME GNF-PF-5061 CHEMBL601385 13332 9059 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE MODIFIED IFN-ALPHA 13333 9060 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW810372X GW810372X 13336 9061 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Triazole derivative 6 13337 9062 CBX1 10951 NA CLOTRIMAZOLE CLOTRIMAZOLE 13338 9063 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649837 13339 9064 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME NN1952 13342 9065 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME (R,S)-INDATRALINE (R,S)-INDATRALINE 13344 9066 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR TRIMETREXATE TRIMETREXATE 13346 9067 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIDANOSINE DIDANOSINE 22931300 13347 9068 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FUSARIC ACID FUSARIC ACID 13348 9069 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MEFLOQUINE HYDROCHLORIDE MEFLOQUINE HYDROCHLORIDE 13349 9070 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME MG-132 MG-132 24321833,18801655 13350 9071 SFTPA1 653509 DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 9486201,2015097,10781428,8969273,3194412,8906664,3382698,12538780,2610267,2014154,8572233 13351 9072 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME KENPAULLONE KENPAULLONE 13353 9073 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CI-966 CHEMBL77287 13354 9074 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650782 OXOTREMORINE 13356 9075 CTSC 1075 ENZYME, DRUGGABLE GENOME, PROTEASE PENTOSAN POLYSULFATE 17826736 13358 9076 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER dexmedetomidine DEXMEDETOMIDINE 13359 9077 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TRIFLUPROMAZINE TRIFLUPROMAZINE 13362 9078 TUBA3D 113457 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 13363 9079 TUBA1B 10376 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 13364 9080 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR TCMDC-124518 CHEMBL527584 13367 9081 POLB 5423 DNA REPAIR, DRUGGABLE GENOME PHYSODIC ACID PHYSODIC ACID 13368 9082 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417185 CHEMBL1549738 13370 9083 TAC1 6863 DRUGGABLE GENOME ANDROGENS 7982063 13372 9084 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 249565861 13374 9085 DPP8 54878 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166751 13376 9086 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Antithyroid Preparations 27157822 13377 9087 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHENOBARBITAL PHENOBARBITAL 22931300 13378 9088 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-4 13379 9089 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE peginterferon alfa-2b 13380 9090 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652036 13382 9091 MBD4 8930 DNA REPAIR PD1 INHIBITOR 29760383 13383 9092 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE CAPIVASERTIB CAPIVASERTIB 26351323,28489509 13385 9093 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SP-600125 SP-600125 13386 9094 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GARLIC GARLIC 15974642 13387 9095 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME Aminotriazolopyridine derivative 1 13389 9096 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650464 CHEMBL153057 13390 9097 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200464 PROPARACAINE HYDROCHLORIDE 13391 9098 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RO-194603 RO-194603 13393 9099 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE THIOTEPA THIOTEPA 13394 9100 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102670 13395 9101 VAMP2 6844 DRUGGABLE GENOME BOTULINUM TOXIN TYPE B 13396 9102 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE IB-MECA IB-MECA 13397 9103 BAZ2B 29994 NA 1,2-NAPHTHOQUINONE 1,2-NAPHTHOQUINONE 13398 9104 CYB5R1 51706 DRUGGABLE GENOME primaquine PRIMAQUINE 13399 9105 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DRONEDARONE DRONEDARONE 13400 9106 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AMIODARONE AMIODARONE 13401 9107 ALOX5 240 DRUGGABLE GENOME, ENZYME WY-50295-tromethamine 13402 9108 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody MM151 13403 9109 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR KW-3357 ANTITHROMBIN ALFA 13405 9110 NAAA 27163 ENZYME, DRUGGABLE GENOME inhibitor 178101852 13406 9111 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PHENETHYLISOTHIOCYANATE PHENETHYLISOTHIOCYANATE 21241062 13408 9112 RNPEP 6051 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor CHEMBL2103847 TOSEDOSTAT 13409 9113 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR MF101 MF101 13411 9114 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIPHENYLBISMUTHINE TRIPHENYLBISMUTHINE 13412 9115 PROS1 5627 DRUGGABLE GENOME Warfarin WARFARIN 13413 9116 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1255654 TETRACAINE HYDROCHLORIDE 13415 9117 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME TGFBETA1 11262404 13416 9118 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor DACOMITINIB DACOMITINIB 13417 9119 DPP9 91039 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 252166752 13418 9120 CA9 768 DRUGGABLE GENOME, ENZYME inhibitor 385612193 13419 9121 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME FX125L 13420 9122 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 187051754 TAFLUPROST 13421 9123 POLI 11201 DNA REPAIR NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 13423 9124 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 94381 CHEMBL374632 13426 9125 JUND 3727 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR CLOZAPINE CLOZAPINE 12093589 13429 9126 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Panitumumab PANITUMUMAB 23729478 13430 9127 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3545058 DEXTROTHYROXINE SODIUM 13432 9128 HTT 3064 DRUGGABLE GENOME CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM BROMIDE 13433 9129 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR ENTINOSTAT ENTINOSTAT 19966789,20491440 13434 9130 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor XL228 XL-228 13436 9131 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ENTRECTINIB ENTRECTINIB 13439 9132 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE sulfadiazine SULFADIAZINE 24372186 13440 9133 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR P-T-OCTYLPHENOL CHEMBL259327 13441 9134 TAC1 6863 DRUGGABLE GENOME FAMOTIDINE FAMOTIDINE 12495560 13442 9135 TARDBP 23435 TUMOR SUPPRESSOR SJ000262868 CHEMBL589444 13443 9136 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX (S,R)-MEFLOQUINE (S,R)-MEFLOQUINE 13444 9137 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME PMID27998201-Compound-10 13445 9138 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BGJ398 INFIGRATINIB 28119489 13446 9139 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Bevacizumab BEVACIZUMAB 13447 9140 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME minocycline MINOCYCLINE 13448 9141 HLA-DQB1 3119 CLINICALLY ACTIONABLE ticlopidine TICLOPIDINE 17339877 13450 9142 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651323 13451 9143 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME TOZASERTIB TOZASERTIB 13453 9144 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME RALTITREXED RALTITREXED 21879757 13454 9145 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 3',4'-DIHYDROXYFLAVONE CHEMBL222556 13455 9146 ABAT 18 DRUGGABLE GENOME, ENZYME Divalproex sodium 13456 9147 POLK 51426 DNA REPAIR, ENZYME DAPHNETIN DAPHNETIN 13459 9148 HLA-DRA 3122 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE NIVOLUMAB NIVOLUMAB 26822383 13460 9149 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METARAMINOL METARAMINOL 13461 9150 MTAP 4507 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE L-ALANOSINE ALANOSINE 16505107 13462 9151 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME MLN-8054 MLN-8054 20684549,17360485 13463 9152 KDM4A 9682 DRUGGABLE GENOME, ENZYME PROTOPORPHYRIN DISODIUM PROTOPORPHYRIN DISODIUM 13464 9153 SMOX 54498 ENZYME, DRUGGABLE GENOME DFMO 10409651 13466 9154 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE LOBARIC ACID LOBARIC ACID 13467 9155 HTT 3064 DRUGGABLE GENOME CAPTAN CAPTAN 13470 9156 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100421 13471 9157 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2062262 METARAMINOL BITARTRATE 13472 9158 GMNN 51053 DRUGGABLE GENOME TCMDC-125587 CHEMBL532160 13473 9159 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DYDROGESTERONE DYDROGESTERONE 13474 9160 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor 363894204 13476 9161 AMH 268 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HUMAN CHORIONIC GONADOTROPIN 10443662 13477 9162 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3545209 NKTR-171 13479 9163 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RECOMBINANT HUMAN IL-2 10383947 13480 9164 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ENNIATIN B ENNIATIN B 13481 9165 PON1 5444 ENZYME, TRANSPORTER, DRUGGABLE GENOME epirubicin EPIRUBICIN 13484 9166 CRISPLD2 83716 DRUGGABLE GENOME dexamethasone DEXAMETHASONE 24926665 13485 9167 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME LTB4 13486 9168 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL1683544 ERIBULIN MESYLATE 13487 9169 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PLX4720 PLX-4720 24265153 13488 9170 ITPR1 3708 ION CHANNEL, KINASE, DRUGGABLE GENOME, TRANSPORTER activator 178101039 13489 9171 FAAH 2166 ENZYME, DRUGGABLE GENOME PMID29053063-Compound-14 13491 9172 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Probenecid PROBENECID 13492 9173 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor 178103355 ALIROCUMAB 13493 9174 CD38 952 CELL SURFACE, DRUGGABLE GENOME CD38-specific gene-engineered T cells 13494 9175 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME OBTUSAQUINONE OBTUSAQUINONE 13497 9176 HDC 3067 DRUGGABLE GENOME, ENZYME BF-DERM1 13502 9177 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR SPIRUCHOSTATIN C SPIRUCHOSTATIN C 21967146 13503 9178 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE ZSTK474 13505 9179 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BGJ398 INFIGRATINIB 13507 9180 BAZ2B 29994 NA DNDI1417529 CHEMBL1990783 13508 9181 TMX2 51075 THIOREDOXIN, DRUGGABLE GENOME ethanol ALCOHOL 32451486 13510 9182 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CHLOROTRIANISENE CHLOROTRIANISENE 13511 9183 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 EUPARIN EUPARIN 13512 9184 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR 3-EPI-ISOCUCURBITACIN D CHEMBL2022241 25756299 13514 9185 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33k 13515 9186 POLB 5423 DNA REPAIR, DRUGGABLE GENOME DIGALLIC ACID DIGALLIC ACID 1705574 13517 9187 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor MK0752 13518 9188 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER fluvastatin FLUVASTATIN 16002074 13520 9189 E2F1 1869 TRANSCRIPTION FACTOR QUERCETIN QUERCETIN 16274926 13521 9190 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 4-METHOXYDALBERGIONE 4-METHOXYDALBERGIONE 13522 9191 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Galantamine analog 1 13523 9192 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR OPK-0018 13524 9193 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME GANCICLOVIR GANCICLOVIR 10766345 13525 9194 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SAR351034 25537454 13526 9195 CBX1 10951 NA IDARUBICIN IDARUBICIN 13527 9196 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PD-0166285 PD-0166285 13528 9197 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor CHEMBL3545368 PANOBINOSTAT LACTATE 13530 9198 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 328083498 13531 9199 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125488 METHOTREXATE 13532 9200 MMP14 4323 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166779 13533 9201 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-44 13535 9202 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SULFINPYRAZONE SULFINPYRAZONE 13536 9203 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE ENTRECTINIB ENTRECTINIB 13537 9204 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME Beta Blocking Agents 18425130,21127457 13538 9205 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8481586, 15 13540 9206 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MESTRANOL MESTRANOL 22931300 13541 9207 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR L-165041 CHEMBL153057 13542 9208 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PROGESTERONE PROGESTERONE 13545 9209 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US10149841, Compound 5 13546 9210 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NITAZOXANIDE NITAZOXANIDE 13548 9211 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR HYDROQUINONE HYDROQUINONE 13549 9212 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER Bisphosphonates 13551 9213 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR NOREPINEPHRINE NOREPINEPHRINE 13552 9214 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE CUCURBITACIN B CUCURBITACIN B 20347305 13554 9215 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME TCMDC-123912 CHEMBL106525 13555 9216 EPHA1 2041 DRUGGABLE GENOME, KINASE, TYROSINE KINASE inhibitor 249565804 13557 9217 BRCA2 675 CLINICALLY ACTIONABLE talazoparib TALAZOPARIB 13558 9218 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR Tazemetostat TAZEMETOSTAT 13560 9219 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 249565645 MK-2461 13561 9220 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Imatinib IMATINIB 13562 9221 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME SJ000040549 CHEMBL589421 13563 9222 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR TRACAZOLATE TRACAZOLATE 13564 9223 MGLL 11343 DRUGGABLE GENOME, ENZYME 1,4-BIS(MALIMIDO)XYLENE CHEMBL565711 19583260 13565 9224 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650328 13566 9225 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE BAY 80-6946 13568 9226 SDC1 6382 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CAR138 T Cells 13569 9227 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103926 UMECLIDINIUM 13570 9228 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE IL-8 1827816 13571 9229 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774824-Compound-Figure6Example6 13572 9230 ATXN2 6311 NA GNF-PF-67 CHEMBL578512 13573 9231 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR MOCETINOSTAT MOCETINOSTAT 23829483,26287310 13574 9232 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor MEK162 BINIMETINIB 13575 9233 CA1 759 DRUGGABLE GENOME, ENZYME Ethoxzolamide ETHOXZOLAMIDE 13576 9234 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ZILEUTON ZILEUTON 22931300 13580 9235 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HERCEPTIN HERCEPTIN 17216002,15581051 13582 9236 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 178103782 LABETALOL 13583 9237 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR 2,4-HEXADIENAL 2,4-HEXADIENAL 13584 9238 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME SRIF-28 CHEMBL442494 18410083 13585 9239 HPN 3249 DRUGGABLE GENOME, PROTEASE, CELL SURFACE AC1LFXA6 13588 9240 KAT2B 8850 ENZYME, DRUGGABLE GENOME DIETHYL-2-TETRADECYLIDENEMALONATE CHEMBL257748 21292492 13589 9241 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL402548 DANUSERTIB 13591 9242 TUBB2B 347733 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 13592 9243 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE docetaxel DOCETAXEL 21151855 13593 9244 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CNF1010 TANESPIMYCIN 13594 9245 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AMSACRINE AMSACRINE 22931300 13595 9246 KDM4A 9682 DRUGGABLE GENOME, ENZYME PYROGALLOL RED PYROGALLOL RED 13597 9247 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL fentanyl FENTANYL 13598 9248 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME METHYLCELLULOSE METHYLCELLULOSE 9016860 13600 9249 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE IVACAFTOR IVACAFTOR 13601 9250 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE ANTHRACYCLINE 12611456 13603 9251 DPEP1 1800 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201057 CILASTATIN SODIUM 13604 9252 MAPT 4137 DRUGGABLE GENOME COUMESTROL COUMESTROL 13605 9253 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2,2,3,3,4,4,5,5,6,6,7,7,8,8,9,9,9-HEPTADECAFLUORO-NONANOIC ACID CHEMBL426404 13606 9254 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Prodigiosin PRODIGIOSIN 26759239 13607 9255 CYB5R3 1727 DRUGGABLE GENOME, ENZYME mepivacaine MEPIVACAINE 13608 9256 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 13610 9257 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME letermovir LETERMOVIR 31022310 13611 9258 ATAD5 79915 NA PYROGALLOL RED PYROGALLOL RED 13612 9259 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Salirasib SALIRASIB 13613 9260 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE SCYLLO-INOSITOL SCYLLITOL 13614 9261 COL1A1 1277 CLINICALLY ACTIONABLE, DRUGGABLE GENOME somatropin recombinant 22026923 13615 9262 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor PF04449913 13616 9263 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE SDF-1 13620 9264 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor GIVINOSTAT GIVINOSTAT 13622 9265 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NRX-5183 13623 9266 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR VORINOSTAT VORINOSTAT 13625 9267 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 328083505 13626 9268 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor 249565728 13627 9269 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker 187051775 ERLOSAMIDE 13628 9270 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR ZK304709 18829975 13630 9271 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL482967 CYC-116 13631 9272 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 249565820 13632 9273 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME SULFADIAZINE, SILVER SULFADIAZINE, SILVER 13633 9274 XPO1 7514 CLINICALLY ACTIONABLE, KINASE SL-801 CBS-9106 13634 9275 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL527 PIROXICAM 13635 9276 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE D-ASPARTATE D-ASPARTATE 13637 9277 SCARB1 949 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME ribavirin RIBAVIRIN 13638 9278 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor PCI-24781 ABEXINOSTAT 13639 9279 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME ABARELIX ABARELIX 11342922 13640 9280 SLC9A1 6548 TRANSPORTER, DRUGGABLE GENOME, EXCHANGER, CELL SURFACE Zoniporide hydrochloride 13642 9281 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIGOXIN DIGOXIN 13643 9282 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 135652070 13644 9283 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RG-1530 RG-1530 13646 9284 CBX1 10951 NA TYRPHOSTIN A9 TYRPHOSTIN A9 13648 9285 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR PROCARBAZINE PROCARBAZINE 23904111 13650 9286 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER bleomycin BLEOMYCIN 25637052 13651 9287 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-67 13652 9288 HTT 3064 DRUGGABLE GENOME CALYCULIN A CALYCULIN A 13653 9289 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THIOGUANINE THIOGUANINE 13655 9290 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TRAMETINIB TRAMETINIB 26644315,24685132,22169769,24915778,27876675 13657 9291 MAPT 4137 DRUGGABLE GENOME ERGOCRISTINE ERGOCRISTINE 13658 9292 TMPRSS2 7113 CLINICALLY ACTIONABLE, PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166870 13659 9293 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE VITAMIN E 15582575 13660 9294 POLK 51426 DNA REPAIR, ENZYME 2,3,4-TRIHYDROXYBENZOPHENONE CHEMBL1527 13662 9295 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME RG-1530 RG-1530 13663 9296 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Ponezumab PONEZUMAB 13664 9297 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE ARSENIC TRIOXIDE 17332940 13665 9298 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE antibody REGN421 13666 9299 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-1919 CHEMBL576409 13667 9300 GLS 2744 ENZYME PMID30273516-Compound-22b 13671 9301 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 178102614 13672 9302 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GNF-PF-5183 CHEMBL577660 13673 9303 TARDBP 23435 TUMOR SUPPRESSOR BIFONAZOLE BIFONAZOLE 13674 9304 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLARITHROMYCIN CLARITHROMYCIN 17635500 13677 9305 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CINNARIZINE CINNARIZINE 13678 9306 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME CART-meso-19 T cells 13683 9307 CD52 1043 DRUGGABLE GENOME inhibitor CHEMBL1201587 ALEMTUZUMAB 13684 9308 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME RETINOL RETINOL 2920014 13686 9309 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME SCLEROTIORIN SCLEROTIORIN 13687 9310 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL68117 VOSAROXIN 13688 9311 NOS1 4842 DRUGGABLE GENOME, ENZYME SALT VOLANESORSEN SODIUM 11243307 13689 9312 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL971 PENTOBARBITAL SODIUM 13690 9313 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL405 AMPHETAMINE 13691 9314 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE UCN-01 UCN-01 15534092 13692 9315 SLC3A2 6520 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER IGN523 13696 9316 FANCC 2176 CLINICALLY ACTIONABLE, DNA REPAIR CHLORAMBUCIL CHLORAMBUCIL 16243825 13700 9317 GAA 2548 DRUGGABLE GENOME, ENZYME ACRIDIN-1-YLAMINE CHEMBL146525 13701 9318 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME inhibitor 187051830 13704 9319 ICAM3 3385 DRUGGABLE GENOME CSA CYCLOSPORINE 15732868 13705 9320 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR FENTICLOR FENTICLOR 13706 9321 HTT 3064 DRUGGABLE GENOME NSC-105827 CHEMBL171699 13708 9322 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CURCUMIN CURCUMIN 23276449 13709 9323 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE GS-9973 ENTOSPLETINIB 13710 9324 PNP 4860 ENZYME, DRUGGABLE GENOME FORODESINE FORODESINE 13711 9325 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201168 ISOCARBOXAZID 13712 9326 CBX1 10951 NA L-METHIONINE-SULFOXIMINE CHEMBL1627202 13713 9327 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102761 13715 9328 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Romidepsin ROMIDEPSIN 13719 9329 MAPT 4137 DRUGGABLE GENOME DANTROLENE SODIUM DANTROLENE SODIUM 13720 9330 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PMID27376512-Compound-Figure2aExample1 13722 9331 MPHOSPH8 54737 NA TRIFLUOPERAZINE HYDROCHLORIDE TRIFLUOPERAZINE HYDROCHLORIDE 13723 9332 CTSD 1509 PROTEASE, DRUGGABLE GENOME, ENZYME STREPTOZOTOCIN STREPTOZOCIN 3282952 13724 9333 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE GENISTEIN GENISTEIN 17539658 13727 9334 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor MASITINIB MASITINIB 13729 9335 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE panitumumab PANITUMUMAB 13730 9336 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 5-HYDROXYINDOLACETIC ACID CHEMBL395915 13732 9337 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME HTS-05057 CHEMBL372629 13733 9338 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT 13735 9339 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME LOPERAMIDE LOPERAMIDE 13737 9340 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32k 13740 9341 ATXN2 6311 NA T091317 T091317 13741 9342 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 348353628 13743 9343 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545398 PG-760564 13744 9344 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR N6-PHENYLADENOSINE N6-PHENYLADENOSINE 13745 9345 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CLONIDINE CLONIDINE 13747 9346 HTT 3064 DRUGGABLE GENOME CHEMBL1200595 CHLORPHENTERMINE HYDROCHLORIDE 13748 9347 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR QUINESTROL QUINESTROL 13749 9348 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY BISPECIFIC ANTIBODY 10433080 13750 9349 GLS 2744 ENZYME MMV000704 CHEMBL582478 13751 9350 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE E-10030 PEGPLERANIB SODIUM 13752 9351 ROR1 4919 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CELL SURFACE Cirmtuzumab CIRMTUZUMAB 13753 9352 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MORICIZINE MORICIZINE 13754 9353 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-309895 CHEMBL552439 13757 9354 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000001516 CHEMBL592316 13758 9355 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2103827 DROXIDOPA 13759 9356 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-2947 CHEMBL581677 13760 9357 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BGJ398 INFIGRATINIB 28119489 13761 9358 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE Gemcitabine GEMCITABINE 22753594 13762 9359 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 374883850 ATABECESTAT 13763 9360 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR FG-3019 PAMREVLUMAB 13764 9361 GAA 2548 DRUGGABLE GENOME, ENZYME 4-METHYLUMBELLIFERYL ACETATE CHEMBL12019 13766 9362 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR cytarabine CYTARABINE 24024897 13767 9363 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GR-127935 GR-127935 13768 9364 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SELICICLIB SELICICLIB 13769 9365 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE ANTI-PD-L1 MONOCLONAL ANTIBODY 25970248 13772 9366 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-23 13773 9367 CACNB3 784 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ION CHANNEL ARVERAPAMIL 13774 9368 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252827503 CGS-27023A 13775 9369 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3039558 ETIRINOTECAN PEGOL 13776 9370 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist,allosteric modulator 387065586 GSK1482160 13778 9371 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SPIRAMIDE SPIRAMIDE 13779 9372 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 315661288 13780 9373 ATXN2 6311 NA (S)-ROSCOVITINE (S)-ROSCOVITINE 13781 9374 SLC47A2 146802 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 178101296 13782 9375 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME ENTRECTINIB ENTRECTINIB 13783 9376 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor MSC1936369B PIMASERTIB HYDROCHLORIDE 13785 9377 SHMT1 6470 ENZYME leucovorin LEUCOVORIN 22044939 13786 9378 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TCMDC-125758 CHEMBL546797 13787 9379 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 381118895 13788 9380 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE OMP-52M51 BRONTICTUZUMAB 13789 9381 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE IRINOTECAN HYDROCHLORIDE HYDRATE IRINOTECAN HYDROCHLORIDE HYDRATE 13790 9382 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME LARGAZOLE LARGAZOLE 21420302,21936551,25203782,20491440 13792 9383 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-33 13793 9384 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BERGAMOTTIN BERGAMOTTIN 21393461 13795 9385 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C12 13796 9386 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PANTOPRAZOLE SODIUM PANTOPRAZOLE SODIUM 13798 9387 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MELENGESTROL ACETATE MELENGESTROL ACETATE 13799 9388 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR GSK-269962A GSK-269962A 13800 9389 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHOCARBAMOL METHOCARBAMOL 22931300 13801 9390 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor SARACATINIB SARACATINIB 13802 9391 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME INDOMETHACIN INDOMETHACIN 22931300 13803 9392 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 249565927 13804 9393 HTT 3064 DRUGGABLE GENOME methylphenidate METHYLPHENIDATE 29382897 13805 9394 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PURPUROGALLIN PURPUROGALLIN 13806 9395 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL456237 LXR-623 13810 9396 MAOA 4128 DRUGGABLE GENOME, ENZYME Clorgyline CLORGILINE 13811 9397 GMNN 51053 DRUGGABLE GENOME FANGCHINOLINE FANGCHINOLINE 13812 9398 EPHB2 2048 KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME MK-8353 MK-8353 13814 9399 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 223366184 13816 9400 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SEMUSTINE SEMUSTINE 13818 9401 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME USL311 USL-311 13819 9402 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE BAY-613606 CHEMBL541400 13820 9403 AKR1B1 231 DRUGGABLE GENOME, ENZYME inhibitor 178103991 ZOPOLRESTAT 13821 9404 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200878 TRIAMCINOLONE HEXACETONIDE 13822 9405 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR Antiinflammatory agents, non-steroids 20538124 13823 9406 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 249565654 XL-019 13824 9407 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL TETRODOTOXIN TETRODOTOXIN 13825 9408 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-25 13826 9409 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL1200475 DAUNORUBICIN CITRATE 13831 9410 NOS1 4842 DRUGGABLE GENOME, ENZYME ANTI-INFLAMMATORY DRUGS 7827327 13833 9411 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER NICLOSAMIDE NICLOSAMIDE 13834 9412 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE IMATINIB IMATINIB 22148584,24681986 13835 9413 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 3,4-METHYLENEDIOXYB-NITROSTYRENE CHEMBL596380 13836 9414 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE AZD5991 AZD-5991 13837 9415 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200948 TRIMIPRAMINE MALEATE 13840 9416 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CLONAZEPAM CLONAZEPAM 13842 9417 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR SCH772984 27312529 13843 9418 F2RL3 9002 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100603 13844 9419 TUBB3 10381 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 13845 9420 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CRENOLANIB CRENOLANIB 13846 9421 GSTA1 2938 ENZYME, DRUGGABLE GENOME rituximab RITUXIMAB 29938344,19448608 13847 9422 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME AZD4547 22869148 13849 9423 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PYRIDALYL PYRIDALYL 13850 9424 ADD1 118 KINASE bumetanide BUMETANIDE 20877298 13851 9425 GAA 2548 DRUGGABLE GENOME, ENZYME 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 13852 9426 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ZOLEDRONIC ACID 20504363 13855 9427 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649971 ATENOLOL 13857 9428 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR TGFBETA1 15153523 13859 9429 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE chlorambucil CHLORAMBUCIL 27173875 13861 9430 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME UM-164 27154914 13862 9431 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GBR-12935 CHEMBL26320 13863 9432 DSG3 1830 NA DESMOGLEIN-3 13864 9433 CYP24A1 1591 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME deferasirox DEFERASIROX 29160302,29099735 13865 9434 S100A10 6281 KINASE GONADOTROPINS 11356677 13867 9435 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TRICETIN TRICETIN 13869 9436 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME TOFACITINIB TOFACITINIB 26231159 13870 9437 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702240 PEMIGATINIB 13871 9438 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 23622981 13872 9439 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME NSC-60340 CHEMBL1534034 13873 9440 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE ERYTHROPOIETIN EPOETIN BETA 1713254 13874 9441 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-677438 CHEMBL118678 13875 9442 KLRD1 3824 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME methotrexate METHOTREXATE 26453102 13876 9443 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 13878 9444 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME zidovudine ZIDOVUDINE 22960662 13880 9445 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE Decamethonium DECAMETHONIUM 13881 9446 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Lapatinib LAPATINIB 13882 9447 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME FOLFOX 28280091,26766738,27002107 13883 9448 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32t 13888 9449 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL408513 BELINOSTAT 13889 9450 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE ANTIOXIDANT 9573532 13891 9451 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1160544 TERBUTALINE SULFATE 13893 9452 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE THALIDOMIDE THALIDOMIDE 13894 9453 ICAM3 3385 DRUGGABLE GENOME INTERFERONS 14989786 13895 9454 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR inhibitor 328083500 CHEMBL592893 13896 9455 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME KINASE INHIBITOR 17041089 13897 9456 GMNN 51053 DRUGGABLE GENOME NSC-1010 CHEMBL1688556 13898 9457 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME EVEROLIMUS EVEROLIMUS 29156677 13899 9458 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TAZAROTENE TAZAROTENE 13900 9459 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 8 13901 9460 MAOA 4128 DRUGGABLE GENOME, ENZYME CX157 13902 9461 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RESERPINE RESERPINE 11743742 13903 9462 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE L6 15764607 13904 9463 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 6,4'-DIMETHOXYFLAVONE 6,4'-DIMETHOXYFLAVONE 13905 9464 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR ELR510444 22295124 13906 9465 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 135650723 NITRENDIPINE 13908 9466 PDE5A 8654 ENZYME, DRUGGABLE GENOME Udenafil UDENAFIL 13909 9467 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-2657 CHEMBL578944 13910 9468 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME 178103302 13913 9469 ITPA 3704 ENZYME peginterferon alfa-2a 25713999 13915 9470 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE inhibitor CHEMBL3833321 BAN2401 13917 9471 PDE4A 5141 DRUGGABLE GENOME, ENZYME APREMILAST APREMILAST 13918 9472 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE MEMANTINE MEMANTINE 20361801 13919 9473 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor 178103971 IBUDILAST 13920 9474 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHOLECALCIFEROL CHOLECALCIFEROL 13922 9475 GLS 2744 ENZYME ABIETIC ACID ABIETIC ACID 13923 9476 GJC1 10052 ION CHANNEL inhibitor 135650269 13924 9477 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3107 CHEMBL602383 13925 9478 CTSC 1075 ENZYME, DRUGGABLE GENOME, PROTEASE GSK2793660 13926 9479 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME MSX-122 MSX-122 13927 9480 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME lapatinib LAPATINIB 24687830,28786423 13928 9481 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BRIMONIDINE BRIMONIDINE 13929 9482 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178103612 MOLIBRESIB 13930 9483 ALDH1A1 216 DRUGGABLE GENOME, ENZYME LY-2183240 CHEMBL509860 13931 9484 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Methylscopolamine METHSCOPOLAMINE 13932 9485 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 13934 9486 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DICHLOROPHEN DICHLOROPHEN 13935 9487 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE JQ1 COMPOUND 24373973 13936 9488 TARDBP 23435 TUMOR SUPPRESSOR TPCK TPCK 13937 9489 MAP2 4133 NA MELATONIN MELATONIN 8829136 13939 9490 PTGES 9536 DRUGGABLE GENOME, ENZYME Pyrimidine derivative 2 13940 9491 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DAUNORUBICIN DAUNORUBICIN 13941 9492 USP1 7398 DNA REPAIR, PROTEASE, ENZYME BENZETHONIUM BENZETHONIUM 13942 9493 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME TAE-684 TAE-684 13943 9494 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME HAEMATOXYLIN HAEMATOXYLIN 13944 9495 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROGESTERONE PROGESTERONE 13945 9496 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AG-490 CHEMBL56543 21185195 13946 9497 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME MLN-8054 MLN-8054 13947 9498 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SUBEROHYDROXAMIC ACID SUBEROHYDROXAMIC ACID 16921367 13948 9499 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker 135649885 13950 9500 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL3544935 XL-418 13951 9501 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL898 DIFLUNISAL 13952 9502 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DIHYDROSPINGOSINE DIHYDROSPINGOSINE 13953 9503 KCNJ3 3760 EXTERNAL SIDE OF PLASMA MEMBRANE, ION CHANNEL, DRUGGABLE GENOME activator 223366101 13954 9504 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE NIMOTUZUMAB NIMOTUZUMAB 13955 9505 POLI 11201 DNA REPAIR NSC-121858 CHEMBL483838 13956 9506 GMNN 51053 DRUGGABLE GENOME ACITRETIN ACITRETIN 13958 9507 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 5-FLUOROINDOLE-2-CARBOXYLIC ACID 5-FLUOROINDOLE-2-CARBOXYLIC ACID 13959 9508 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565589 BAFETINIB 13961 9509 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE DS-8895 13962 9510 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651405 TIRATRICOL 13963 9511 TUBA1A 7846 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 13964 9512 ALOX15 246 ENZYME, DRUGGABLE GENOME BAICALEIN BAICALEIN 17869117 13966 9513 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BACLOFEN BACLOFEN 13967 9514 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME midazolam MIDAZOLAM 17638512,11470993 13968 9515 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135652126 13969 9516 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL activator 135652668 13970 9517 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE CHLOROETHYLCLONIDINE CHLOROETHYLCLONIDINE 13971 9518 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ASTERRIC ACID ASTERRIC ACID 13972 9519 BAZ2B 29994 NA SJ000114741 CHEMBL591370 13973 9520 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER CEFUROXIME CEFUROXIME 22166395 13974 9521 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102019 13975 9522 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GITOXIGENIN GITOXIGENIN 13976 9523 RACGAP1 29127 NA NSC-69187 CHEMBL19954 13977 9524 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME CHEMBL2103837 TAFAMIDIS 13979 9525 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650288 13980 9526 LPAR2 9170 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 178103194 13984 9527 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DOVITINIB DOVITINIB 13985 9528 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME ISIS-CRP 13986 9529 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE SNN-0031 13987 9530 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE blocker CHEMBL1700 SOTALOL HYDROCHLORIDE 13988 9531 ETV5 2119 DRUG RESISTANCE, CLINICALLY ACTIONABLE TRAMETINIB TRAMETINIB 28178529 13990 9532 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SB-242235 SB-242235 13991 9533 HSPB1 3315 DRUGGABLE GENOME TEROXIRONE TEROXIRONE 13992 9534 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TANSHINONE IIA TANSHINONE IIA 13993 9535 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR LY-2382770 LY-2382770 13995 9536 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE metoclopramide METOCLOPRAMIDE 13998 9537 POLK 51426 DNA REPAIR, ENZYME SHIKONIN SHIKONIN 13999 9538 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PRASTERONE PRASTERONE 14000 9539 TMEM97 27346 NA PMID30185082-Compound-56 14002 9540 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE partial agonist CHEMBL1685 DEZOCINE 14005 9541 TUBA4A 7277 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 14006 9542 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Carteolol CARTEOLOL 14007 9543 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER modafinil MODAFINIL 26757307 14011 9544 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE VINCRISTINE VINCRISTINE 17999741 14012 9545 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME TANDUTINIB TANDUTINIB 14013 9546 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GEFITINIB GEFITINIB 14014 9547 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE Tricyclic compound 4 14015 9548 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 348353621 PYROTINIB 14016 9549 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 felodipine FELODIPINE 9187528 14018 9550 ADK 132 DRUGGABLE GENOME, ENZYME, KINASE GP-3269 14019 9551 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 381118807 14020 9552 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEXTROMETHORPHAN HYDROBROMIDE MONOHYDRATE DEXTROMETHORPHAN HYDROBROMIDE 14021 9553 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor ENTINOSTAT ENTINOSTAT 14022 9554 PSMD1 5707 NA OPROZOMIB OPROZOMIB 14023 9555 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE GNF-PF-2301 CHEMBL578061 14024 9556 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL962 EPOPROSTENOL SODIUM 14025 9557 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME 1,2,4-triazolo[1,5a]pyridine derivative 1 14026 9558 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Bambuterol BAMBUTEROL 14028 9559 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody CIXUTUMUMAB CIXUTUMUMAB 14032 9560 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE 252166786 EMI-137 14034 9561 ATXN2 6311 NA 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 14035 9562 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 223366142 14037 9563 ALOX5 240 DRUGGABLE GENOME, ENZYME NDGA 15694390 14038 9564 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE RETEPLASE RETEPLASE 14039 9565 GADD45G 10912 KINASE, TUMOR SUPPRESSOR ANDROGENS 15062559 14042 9566 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Fluoxymesterone FLUOXYMESTERONE 14043 9567 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CIMETIDINE CIMETIDINE 22931300 14044 9568 C1QA 712 DRUGGABLE GENOME, CELL SURFACE IMMUNE GLOBULIN 14045 9569 SMN2 6607 DRUGGABLE GENOME CID 1540951 CHEMBL259421 14046 9570 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME PD-0166285 PD-0166285 14047 9571 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-3165 CHEMBL581257 14049 9572 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER NPT-200-11 14050 9573 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR BAICALEIN BAICALEIN 19592245 14052 9574 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PROTEIN KINASE C INHIBITOR 9223624 14053 9575 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166828 14054 9576 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Estradiol Acetate 14056 9577 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor GEFITINIB GEFITINIB 14057 9578 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor 178103251 PIRLINDOLE 14058 9579 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1768 BETHANECHOL CHLORIDE 14064 9580 HTT 3064 DRUGGABLE GENOME TCMDC-123764 CHEMBL533226 14065 9581 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME ALOGLIPTIN ALOGLIPTIN 14067 9582 ATXN2 6311 NA MITOXANTRONE MITOXANTRONE 14068 9583 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135651495 14069 9584 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME RAFAMETINIB 14070 9585 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR antagonist 310264686 14071 9586 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME NU-172 21838685 14073 9587 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE CILENGITIDE CILENGITIDE 12154028 14074 9588 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME GNF-PF-2272 CHEMBL601757 14075 9589 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CHEMBL1743072 SOLANEZUMAB 14077 9590 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CIANIDANOL CIANIDANOL 14078 9591 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32y 14079 9592 HEBP1 50865 DRUGGABLE GENOME Chalcone derivative 4 14081 9593 F7 2155 ENZYME, DRUGGABLE GENOME, PROTEASE Vatreptacog alfa (activated) 14083 9594 HTRA1 5654 ENZYME, DRUGGABLE GENOME, PROTEASE ranibizumab RANIBIZUMAB 22594510,23559864,23842101,23337555 14084 9595 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE OSI-632 OSI-632 14085 9596 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 25 14087 9597 BUB1 699 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565789 14090 9598 CLU 1191 CELL SURFACE, DRUGGABLE GENOME OGX-011 CUSTIRSEN SODIUM 14091 9599 BAZ2B 29994 NA METHYLDOPA METHYLDOPA 14092 9600 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CINTAZONE CINTAZONE 14094 9601 AKR1B1 231 DRUGGABLE GENOME, ENZYME Oxilofrine OXILOFRINE 14095 9602 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor 178101910 MILRINONE 14098 9603 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PD-0166285 PD-0166285 14099 9604 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 178101101 14100 9605 GAPDH 2597 DRUGGABLE GENOME, ENZYME NSC-92207 CHEMBL139935 14102 9606 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE GNF-PF-2301 CHEMBL578061 14104 9607 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE HYDROCODONE HYDROCODONE 14105 9608 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 315661317 14106 9609 PSMA3 5684 PROTEASE, DRUGGABLE GENOME inhibitor CARFILZOMIB CARFILZOMIB 14107 9610 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL2105395 OSPEMIFENE 14108 9611 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2387080 TASELISIB 14110 9612 GMNN 51053 DRUGGABLE GENOME GNF-PF-1295 CHEMBL579837 14112 9613 PLAUR 5329 DRUGGABLE GENOME, ENZYME, CELL SURFACE RECOMBINANT INTERFERON GAMMA 8049441 14113 9614 PXN 5829 NA H2O2 9590268 14114 9615 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BYL719 ALPELISIB 27126994 14115 9616 NEU3 10825 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE OSELTAMIVIR OSELTAMIVIR 18694948 14117 9617 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME LY-517717 CHEMBL1271162 14118 9618 PTPRB 5787 DRUGGABLE GENOME, PROTEIN PHOSPHATASE AKB-9778 RAZUPROTAFIB 14119 9619 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RALOXIFENE RALOXIFENE 14122 9620 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Aniline derivative 1 14123 9621 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR UCCF-029 CHEMBL177991 14124 9622 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL272980 MOCETINOSTAT 14125 9623 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565869 CEP-11981 14126 9624 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR OUABAIN HYDRATE OUABAIN 14127 9625 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE BORTEZOMIB BORTEZOMIB 20875739 14128 9626 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DIALLYLDISULFIDE DIALLYLDISULFIDE 14129 9627 MAP3K7 6885 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 348353658 14130 9628 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME UREA UREA 9726418 14131 9629 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BENFLUOREX HYDROCHLORIDE BENFLUOREX HYDROCHLORIDE 14132 9630 PLTP 5360 DRUGGABLE GENOME VITAMIN E 15734742,15576481,12105225 14133 9631 HLA-DQA1 3117 CLINICALLY ACTIONABLE LYMPHOKINES 2166625 14134 9632 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-3266 CHEMBL581869 14136 9633 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Gossypol GOSSYPOL 14137 9634 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TYRPHOSTIN A9 TYRPHOSTIN A9 14138 9635 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CBP-501 CBP-501 14139 9636 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME EV-077 14140 9637 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 354702287 14142 9638 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ZNFTXQFGUIKQQE-UHFFFAOYSA-N 14143 9639 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR CORTISOL HYDROCORTISONE 15576665 14146 9640 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR IL-2 ALDESLEUKIN 10229082 14148 9641 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AUY922 26832792 14150 9642 RGS4 5999 DRUGGABLE GENOME 3,4-DICHLOROISOCOUMARIN CHEMBL24983 14154 9643 TYMSOS 494514 NA capecitabine CAPECITABINE 25677447 14155 9644 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHA-767491 CHEMBL225519 14156 9645 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME GSK2636771 GSK-2636771 26577700,26645196 14157 9646 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SIMVASTATIN SIMVASTATIN 10543307 14159 9647 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 252827412 14161 9648 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LINIFANIB LINIFANIB 14162 9649 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE 5-(4-PHENYLBUTOXY)PSORALEN CHEMBL1256851 14163 9650 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE DASATINIB DASATINIB 14164 9651 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor PF-4691502 PF-04691502 14165 9652 MAPT 4137 DRUGGABLE GENOME DOCONEXENT DOCONEXENT 14167 9653 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Selumetinib SELUMETINIB 26343583,25870145,23406027 14168 9654 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE GSK2126458 OMIPALISIB 14170 9655 CBX1 10951 NA RESERPINE RESERPINE 14171 9656 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE N,N'-DIPHENYL-GUANIDINE CHEMBL77675 14172 9657 BRD9 65980 ENZYME inhibitor 252166773 14173 9658 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor NINTEDANIB NINTEDANIB 14174 9659 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DOPAMINE HYDROCHLORIDE DOPAMINE HYDROCHLORIDE 14175 9660 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME inhibitor 336446964 14179 9661 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE WORTMANNIN WORTMANNIN 11598141,12490950,12743033,18366935 14180 9662 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL521851 PICTILISIB 14182 9663 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2,4-DIHYDROXYBENZOPHENONE 2,4-DIHYDROXYBENZOPHENONE 14183 9664 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Pyrazole and thiophene derivative 1 14184 9665 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 14185 9666 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE 178101305 14187 9667 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2109332 MLNM-2201 14189 9668 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME gefitinib GEFITINIB 25554506,21332310,20035425,17148776 14191 9669 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1237105 CARBOPROST TROMETHAMINE 14192 9670 PTGS2 5743 DRUGGABLE GENOME, ENZYME ETORICOXIB ETORICOXIB 14193 9671 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LAPATINIB LAPATINIB 14194 9672 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CUDC-101 CUDC-101 14196 9673 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-45 14198 9674 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME DOX 1387586 14199 9675 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor XL147 PILARALISIB 14201 9676 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545201 TA-5493 14202 9677 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AM-251 CHEMBL285932 14203 9678 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PD173074 27998968,23558953,21119661 14206 9679 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 QUERCETIN QUERCETIN 14207 9680 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamide derivative 1 14210 9681 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ALSTERPAULLONE ALSTERPAULLONE 14211 9682 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BGT226 BGT-226 23705826 14213 9683 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RABEPRAZOLE RABEPRAZOLE 14214 9684 POLK 51426 DNA REPAIR, ENZYME CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 14216 9685 TXNRD1 7296 DRUGGABLE GENOME vitamin c 23913015 14218 9686 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Ponatinib PONATINIB 22238366,25294908,28034880 14219 9687 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHLORETIN PHLORETIN 14221 9688 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME GEFITINIB GEFITINIB 22281684 14222 9689 ALOX15 246 ENZYME, DRUGGABLE GENOME Indole and benzimidazole derivative 1 14223 9690 RRM2B 50484 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL1200983 GALLIUM NITRATE 14225 9691 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME ARRY-300 ARRY-300 14226 9692 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1657 TAZAROTENE 14228 9693 MPI 4351 ENZYME, DRUGGABLE GENOME DNDI1417614 CHEMBL1567571 14229 9694 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL607707 PELITINIB 14230 9695 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE 5-FLUORODEOXYURIDINE FLOXURIDINE 8324744 14231 9696 HDC 3067 DRUGGABLE GENOME, ENZYME inhibitor 178101877 14232 9697 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 7 14233 9698 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-47b 14234 9699 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME DIETHYL-2-TETRADECYLMALONATE CHEMBL1797712 21292492 14235 9700 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107647 LANICEMINE 14236 9701 KDM4A 9682 DRUGGABLE GENOME, ENZYME CETIRIZINE HYDROCHLORIDE CETIRIZINE HYDROCHLORIDE 14238 9702 MAGEA3 4102 ENZYME, DRUGGABLE GENOME KITE-718 14239 9703 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME AZD-1775 ADAVOSERTIB 14241 9704 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 14243 9705 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antibody PF-04605412 PF-04605412 14244 9706 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR CLIOQUINOL CLIOQUINOL 14245 9707 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME LATREPIRDINE LATREPIRDINE 14246 9708 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 14247 9709 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamate derivative 10 14248 9710 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LAGASCATRIOL LAGASCATRIOL 23046382 14252 9711 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 385612234 14253 9712 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME ILORASERTIB ILORASERTIB 14254 9713 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE CEDIRANIB CEDIRANIB 14256 9714 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CGS-12066B CHEMBL27403 14257 9715 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COUMARIN COUMARIN 14258 9716 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL SSR-125047 14259 9717 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE 2-CHLORO-ADENOSINETRIPHOSPHATE CHEMBL1368696 14260 9718 HMGCR 3156 ENZYME, DRUGGABLE GENOME simvastatin SIMVASTATIN 17563401,18815589,18332269,16103896,18261733,15199031 14261 9719 USP1 7398 DNA REPAIR, PROTEASE, ENZYME 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 14262 9720 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GR-55562 GR-55562 14266 9721 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME THIOMERSAL THIMEROSAL 14267 9722 ESRRG 2104 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DES DIETHYLSTILBESTROL 12579585 14268 9723 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR MK2206 MK-2206 26676756 14269 9724 KCNG1 3755 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL113461 TEDISAMIL 14270 9725 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME volatile anesthetics 25989378,12411786,21965348,20837722,20301325,9037193,12467748,19648156,23223104,25960145,26031886,28326467,25424378,12761368,11725865,16917943,24291096,16163667,23628358,19807743,18313359,21455645,10625004,12124989,3177917,15537710,12059893,23069638,27382027,19018722,10360872,17182726,25735680,27663056,15731587,26068069,28403410,9873004,20888934,15299003,19346234,22415532 14272 9726 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NIHYDRAZONE NIHYDRAZONE 14273 9727 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051805 QUISINOSTAT 14274 9728 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL1200512 IRINOTECAN HYDROCHLORIDE HYDRATE 14276 9729 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565904 TRYPTANTHRIN 14278 9730 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE CVBT-141B 14279 9731 PTBP1 5725 DRUGGABLE GENOME DNDI1417941 CHEMBL2095095 14281 9732 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650557 14283 9733 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE DIPHENYLETHER DIPHENYLETHER 18952425 14284 9734 TUBA3C 7278 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 14285 9735 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 178102937 ALOGLIPTIN 14286 9736 EIF2AK1 27102 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 381118865 14287 9737 PTGS2 5743 DRUGGABLE GENOME, ENZYME LICOFELONE LICOFELONE 14288 9738 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 187051843 LASOFOXIFENE 14289 9739 GGH 8836 PROTEASE, ENZYME, DRUGGABLE GENOME methotrexate METHOTREXATE 15284538,22763757,17286537,19827168,16999998,15564880 14290 9740 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ISOTRETINOIN ISOTRETINOIN 14291 9741 WNT7A 7476 DRUGGABLE GENOME, CELL SURFACE DES DIETHYLSTILBESTROL 9806537 14292 9742 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DNDI1417941 CHEMBL2095095 14293 9743 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 381118891 14295 9744 MGLL 11343 DRUGGABLE GENOME, ENZYME Azetidinyl-piperazine derivative 3 14299 9745 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BGJ398 INFIGRATINIB 27338794 14300 9746 TCF7L2 6934 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Dipeptidyl peptidase 4 (DPP-4) inhibitors 27166975 14301 9747 NDUFB10 4716 ENZYME inhibitor CHEMBL3545320 ME-344 14305 9748 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178104021 ACLIDINIUM 14306 9749 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 252827463 14308 9750 METAP2 10988 ENZYME, DRUGGABLE GENOME, KINASE, PROTEASE PPI-2458 PPI-2458 14309 9751 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL276711 SEMAXANIB 14310 9752 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GENTIAN VIOLET GENTIAN VIOLET 14311 9753 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR VASOPRESSIN VASOPRESSIN 16457953 14312 9754 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650891 UPIDOSIN 14313 9755 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Beta Blocking Agents 22543981,16189366 14314 9756 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ALFENTANIL ALFENTANIL 14316 9757 GCLC 2729 DRUGGABLE GENOME, ENZYME BUTHIONINE SULPHOXIMINE 11705692 14317 9758 ATP5F1E 514 TRANSPORTER adalimumab ADALIMUMAB 26307125 14318 9759 PRORP 9692 NA zileuton ZILEUTON 25963335 14320 9760 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR GOSSYPETIN GOSSYPETIN 25190466 14322 9761 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE NILOTINIB NILOTINIB 23676790,12623848,20367437,17114651,18828913,21895409,21489624,11964322,25157968,21605905,21562040 14323 9762 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CAPTAN CAPTAN 14324 9763 NDUFS7 374291 ENZYME inhibitor CHEMBL3545320 ME-344 14325 9764 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545200 S-222611 14326 9765 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 249565627 TESEVATINIB 14327 9766 FCGRT 2217 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antibody 374883846 14328 9767 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE AGN-211745 14330 9768 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ISA-P53-01 14333 9769 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CRIZOTINIB CRIZOTINIB 29596029,23724914,25264305,24875859,25922291,22215748,25688157,26372962,25667280,30980071,29333528 14334 9770 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE PURPURIN PURPURIN 14336 9771 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker 223366057 14337 9772 MAP2K6 5608 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE, TUMOR SUPPRESSOR inhibitor BAY869766 14339 9773 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE RG-1530 RG-1530 14340 9774 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR HUMAN CHORIONIC GONADOTROPIN 15941869 14341 9775 ALOX15 246 ENZYME, DRUGGABLE GENOME FLAVANONE FLAVANONE 14342 9776 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ARS-853 26739882,26841430 14344 9777 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TCMDC-125293 CHEMBL548629 14345 9778 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Bevacizumab + Erlotinib 14346 9779 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME MSDC-0602 14347 9780 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650388 IMPROMIDINE 14348 9781 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 14350 9782 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TOZASERTIB TOZASERTIB 14351 9783 ALOX15 246 ENZYME, DRUGGABLE GENOME ZIRAM ZIRAM 14352 9784 KDM1A 23028 DRUGGABLE GENOME, ENZYME, CELL SURFACE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING TRANYLCYPROMINE HYDROCHLORIDE TRANYLCYPROMINE HYDROCHLORIDE 14353 9785 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650082 14355 9786 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Bis-aminopyrimidine derivative 5 14356 9787 PTGS1 5742 ENZYME, DRUGGABLE GENOME Curcumin CURCUMIN 14358 9788 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR HEXACHLOROPHENE HEXACHLOROPHENE 14359 9789 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SAQUINAVIR MESYLATE SAQUINAVIR MESYLATE 14362 9790 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Betamethasone BETAMETHASONE 14363 9791 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE ANTIESTROGEN 12556556 14364 9792 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE CEP-11981 CEP-11981 14365 9793 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 249565693 14366 9794 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650752 14367 9795 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE AM-630 CHEMBL181633 14368 9796 POLI 11201 DNA REPAIR NCG-C00094421-01 CHEMBL553503 14369 9797 GRK2 156 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 405560387 14370 9798 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE erdafitinib ERDAFITINIB 14371 9799 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME ENTRECTINIB ENTRECTINIB 26884591,29237803,28183697 14372 9800 HLA-DQB1 3119 CLINICALLY ACTIONABLE carbamazepine CARBAMAZEPINE 24399721 14374 9801 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR RG-1530 RG-1530 14375 9802 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GNF-PF-2950 CHEMBL602807 14376 9803 SLC38A5 92745 TRANSPORTER 178101385 14377 9804 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ARA-C 1849032 14378 9805 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SB-207710 CHEMBL114112 20812727 14379 9806 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ANTIBIOTICS 9470171 14380 9807 TUBB4B 10383 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 14382 9808 POLB 5423 DNA REPAIR, DRUGGABLE GENOME EPHEDRINE SULFATE EPHEDRINE SULFATE 14383 9809 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME COBALT 14741615 14385 9810 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Panitumumab PANITUMUMAB 28404754,26540314,23625191,24919569,18316791,26341920,19064407 14386 9811 CA2 760 DRUGGABLE GENOME, ENZYME COBALT 107027 14387 9812 SULT1A3 6818 DRUGGABLE GENOME, ENZYME acetaminophen ACETAMINOPHEN 23462933,26049587 14388 9813 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME TCMDC-125758 CHEMBL546797 14389 9814 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Imidazo[1,2-b]pyridazine derivative 1 14390 9815 SLC28A1 9154 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE gemcitabine GEMCITABINE 18538445,25162786,30889042 14393 9816 GAA 2548 DRUGGABLE GENOME, ENZYME DNDI1417523 CHEMBL598663 14396 9817 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Dromostanolone DROMOSTANOLONE 14397 9818 POLI 11201 DNA REPAIR QUINACRINE DIHYDROCHLORIDE QUINACRINE DIHYDROCHLORIDE 14398 9819 RIPK3 11035 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 384403680 14400 9820 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 252166793 14402 9821 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SJ000173328 CHEMBL591613 14404 9822 PRKACB 5567 ENZYME, KINASE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 178101884 GSK-690693 14405 9823 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NEOCUPROINE NEOCUPROINE 14406 9824 EPHB4 2050 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL3544983 TESEVATINIB 14408 9825 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Quinolone Antibacterials 24372186 14410 9826 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AZD5363 CAPIVASERTIB 26351323 14411 9827 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Dinoprost Tromethamine 14413 9828 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE Pyridone 6 22916261 14414 9829 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178100902 14416 9830 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 328083479 14418 9831 KDM4A 9682 DRUGGABLE GENOME, ENZYME CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 14419 9832 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000001516 CHEMBL592316 14420 9833 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 2',3'-DIHYDROXYFLAVONE CHEMBL242171 14421 9834 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE vincristine VINCRISTINE 27173875 14423 9835 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID27336223-Compound-5 14426 9836 TPCN1 53373 ION CHANNEL, DRUGGABLE GENOME blocker 135652732 14427 9837 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 4-(thiazol-5-yl)-pyrimidine derivative 1 14428 9838 RAB9A 9367 ENZYME, DRUGGABLE GENOME TCMDC-124522 CHEMBL526776 14429 9839 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-124557 CHEMBL530682 14431 9840 CXCL8 3576 DRUGGABLE GENOME ACETAMINOPHEN ACETAMINOPHEN 15878691 14434 9841 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-133896 CHEMBL512908 14435 9842 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9409892, 19 14438 9843 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE REL-HUEAFURANOID A CHEMBL2207339 23141910 14439 9844 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL PRAZEPAM PRAZEPAM 14441 9845 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE propranolol PROPRANOLOL 14443 9846 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 310264733 FIMEPINOSTAT 14445 9847 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ACRISORCIN ACRISORCIN 14446 9848 MAPT 4137 DRUGGABLE GENOME PROTOPORPHYRIN PROTOPORPHYRIN 14447 9849 CASP14 23581 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166874 14448 9850 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW279320X GW279320X 14449 9851 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-80 14450 9852 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL107 COLCHICINE 14451 9853 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Ro 31-7453 14452 9854 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE LAPATINIB LAPATINIB 25953157,25398453 14453 9855 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE AST-487 AST-487 14455 9856 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OESTRADIOL ESTRADIOL 3033233 14456 9857 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417185 CHEMBL1549738 14457 9858 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR SLAZINIC ACID SLAZINIC ACID 14458 9859 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 354702260 DEBIO-1347 14459 9860 ERAP2 64167 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE inhibitor 252166866 14461 9861 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX FLUORESCEIN FLUORESCEIN 14462 9862 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE PERTUZUMAB PERTUZUMAB 23680147 14464 9863 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE OBP-301 14466 9864 TUBB3 10381 DRUGGABLE GENOME IXABEPILONE IXABEPILONE 14467 9865 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650066 14468 9866 ENOSF1 55556 ENZYME fluorouracil FLUOROURACIL 17549067,27995989,20714149,27001118,23263912 14472 9867 TSPO 706 DRUGGABLE GENOME ONO-2952 ONO-2952 14473 9868 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 14474 9869 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE chloroprocaine CHLOROPROCAINE 14475 9870 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE LIPOIC ACID THIOCTIC ACID 23984871 14477 9871 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1201466 ESTROGENS, CONJUGATED SYNTHETIC A 14478 9872 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME ROEMERINE ROEMERINE 14480 9873 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PALOMID 529 14481 9874 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PMID26924192-Compound-103 14484 9875 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE POLYPHENOL 14633667 14485 9876 NEK4 6787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME BAY-613606 CHEMBL541400 14486 9877 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE DASATINIB DASATINIB 21689725,24045550,19164557,15972446,16384925,18024392,15685537,23149070,18986703,22504184,16912224,18559612,23714533,25157968,17699867,22932406,17259998,21642685,23582185,16731599 14487 9878 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME MITOXANTRONE MITOXANTRONE 14488 9879 NDUFA8 4702 ENZYME inhibitor CHEMBL3545135 NV-128 14489 9880 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE JNJ-7706621 JNJ-7706621 14490 9881 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME TOZASERTIB TOZASERTIB 14492 9882 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME (R,S)-AMPA (R,S)-AMPA 14493 9883 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CARBINOXAMINE CARBINOXAMINE 14494 9884 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE 6,6'-DISELANEDIYLBIS(N-PHENYLHEXANAMIDE) CHEMBL1086397 20855208 14495 9885 XYLT2 64132 ENZYME gemcitabine GEMCITABINE 31616045 14497 9886 VEGFC 7424 GROWTH FACTOR, TRANSPORTER, DRUGGABLE GENOME aflibercept AFLIBERCEPT 20124951 14498 9887 GATA2 2624 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX fasudil FASUDIL 22541434 14500 9888 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565797 14501 9889 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 178101691 14503 9890 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME OCINAPLON OCINAPLON 14504 9891 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE SORAFENIB SORAFENIB 14506 9892 CBX1 10951 NA PROMETHAZINE PROMETHAZINE 14507 9893 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE PMID29130358-Compound-Figure17(11) 14511 9894 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1079593 VS-5584 14512 9895 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE MEDI-547 14513 9896 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649841 14515 9897 SMN2 6607 DRUGGABLE GENOME AG1295 AG1295 14517 9898 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME BRYOSTATIN-1 14518 9899 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME PMID27828716-Compound-19 14519 9900 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-108783 CHEMBL1489812 14521 9901 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 artemether ARTEMETHER 14524 9902 IL18 3606 DRUGGABLE GENOME MYCOPHENOLIC ACID 12907250 14527 9903 POLK 51426 DNA REPAIR, ENZYME PROTOPORPHYRIN PROTOPORPHYRIN 14528 9904 RGS19 10287 NA opioids 14530 9905 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL blocker,inhibitor 178101028 14531 9906 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor 385612194 14533 9907 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BML-210 CHEMBL324053 16921367 14534 9908 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1614702 SCIO-323 14535 9909 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor CUDC-101 CUDC-101 14536 9910 GMNN 51053 DRUGGABLE GENOME TERFENADINE TERFENADINE 14538 9911 HEBP1 50865 DRUGGABLE GENOME Pyrazino[2,1-a]isoquinolin derivative 4 14539 9912 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME VX-11e 27974663 14540 9913 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33h 14542 9914 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR allosteric modulator 249565628 MK-2206 14543 9915 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 2-STYRYL-QUINOLINE CHEMBL127579 14544 9916 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US9434725, 113 14545 9917 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER DIGOXIN DIGOXIN 15969931,16674925 14547 9918 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE carboplatin CARBOPLATIN 30071039 14548 9919 SFTPA1 653509 DRUGGABLE GENOME PMA 8810290 14550 9920 HTT 3064 DRUGGABLE GENOME SJ000128325 CHEMBL602718 14552 9921 AKR1C3 8644 ENZYME, DRUGGABLE GENOME TESTOSTERONE TESTOSTERONE 10998348 14553 9922 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR HORMONES 12082616 14554 9923 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Ureido-phenyl-substituted triazine derivative 2 14555 9924 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-acylpiperidine ether derivative 5 14558 9925 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME C5A 16634840 14562 9926 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE 681640 CHEMBL379975 14564 9927 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR A-007 SIVIFENE 14565 9928 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20128202889C90 14566 9929 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ADAPALENE ADAPALENE 14567 9930 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR P-T-OCTYLPHENOL CHEMBL259327 14569 9931 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIPHENHYDRAMINE DIPHENHYDRAMINE 22931300 14570 9932 CBX1 10951 NA DISULFIRAM DISULFIRAM 14574 9933 ALB 213 TRANSPORTER, DRUGGABLE GENOME EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 20598557 14576 9934 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME QUERCETIN QUERCETIN 25190466 14578 9935 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE AG-1879 CHEMBL406845 14582 9936 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER NIFEDIPINE NIFEDIPINE 10213372 14584 9937 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE Seribantumab SERIBANTUMAB 14585 9938 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor VORINOSTAT VORINOSTAT 14586 9939 POLK 51426 DNA REPAIR, ENZYME 9-AMINOCAMPTOTHECIN 9-AMINOCAMPTOTHECIN 14587 9940 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker 135650296 GALLAMINE 14588 9941 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR LOVASTATIN LOVASTATIN 9072409 14589 9942 POLI 11201 DNA REPAIR PYROGALLOL RED PYROGALLOL RED 14590 9943 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Margetuximab MARGETUXIMAB 14591 9944 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE ANTIDEPRESSANTS 16890384 14592 9945 NDUFB3 4709 ENZYME inhibitor CHEMBL3545135 NV-128 14597 9946 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME SCH 66336 15090542 14598 9947 PDE10A 10846 ENZYME, DRUGGABLE GENOME Pyrido[1,2,4]triazolo[4,3-a]pyrazine derivative 1 14599 9948 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 315661273 ATICAPRANT 14600 9949 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1370561 AMINOPHYLLINE 14601 9950 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 135649892 ACROLEIN 14602 9951 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Ribociclib RIBOCICLIB 14604 9952 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Asparaginase ASPARAGINASE 28151717 14605 9953 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME Hu-CART meso cells 14608 9954 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE MEPINDOLOL MEPINDOLOL 2903243 14609 9955 SMARCA2 6595 NA NSC-69187 CHEMBL19954 14611 9956 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CGM097 CGM-097 27659046 14612 9957 MAPT 4137 DRUGGABLE GENOME DAMNACANTHAL DAMNACANTHAL 14614 9958 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1479 DANAZOL 14615 9959 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Acyl piperidine derivative 2 14616 9960 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 135652717 STAUROSPORINE 14618 9961 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TRIDIHEXETHYL TRIDIHEXETHYL 14619 9962 GLS 2744 ENZYME AMPICILLIN SODIUM AMPICILLIN SODIUM 14621 9963 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 252166792 14622 9964 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE LYMPHOKINES 7586221 14623 9965 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MEPREDNISONE MEPREDNISONE 14624 9966 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565686 BX-795 14626 9967 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE inhibitor CHEMBL413 SIROLIMUS 14627 9968 SQLE 6713 DRUGGABLE GENOME, ENZYME inhibitor 252827452 14628 9969 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Prasterone PRASTERONE 14630 9970 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NIALAMIDE NIALAMIDE 14631 9971 AKR1B1 231 DRUGGABLE GENOME, ENZYME AR08 24707983 14633 9972 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TRIPELENNAMINE TRIPELENNAMINE 14636 9973 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL3545215 BMS-911543 14637 9974 IDE 3416 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, ENZYME, PROTEASE CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 14638 9975 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CP-339818 CP-339818 14639 9976 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE CISPLATIN CISPLATIN 14640 9977 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Isoetharine ISOETHARINE 14643 9978 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME S-(P-AZIDOPHENACYL)GLUTATHIONE CHEMBL1256813 14644 9979 ADH1C 126 ENZYME, DRUGGABLE GENOME cyclophosphamide CYCLOPHOSPHAMIDE 24533712 14646 9980 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545325 SAR-125844 14647 9981 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Obatoclax OBATOCLAX 22460902 14648 9982 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Oxatomide OXATOMIDE 14649 9983 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650532 LOSARTAN 14650 9984 MAOB 4129 DRUGGABLE GENOME, ENZYME Schiff base compound 2 14651 9985 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1544 LIOTHYRONINE 14653 9986 SLC28A2 9153 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME URIDINE URIDINE 11641443 14654 9987 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME FENOFIBRIC ACID FENOFIBRIC ACID 22579484,23566516 14655 9988 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652101 14656 9989 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 223366195 14657 9990 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR CHLORPYRIFOS CHLORPYRIFOS 14658 9991 GUCY1A2 2977 ENZYME, DRUGGABLE GENOME RIOCIGUAT RIOCIGUAT 14659 9992 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178103589 RICOLINOSTAT 14660 9993 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565621 MILCICLIB 14661 9994 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR RXI-109 24587648 14662 9995 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TRAMETINIB TRAMETINIB 14664 9996 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL1980297 ILORASERTIB 14665 9997 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1232583 INDEGLITAZAR 14666 9998 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ROSMARINIC ACID ROSMARINIC ACID 14668 9999 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL INS37217 14669 10000 UGT1A7 54577 DRUGGABLE GENOME, ENZYME methotrexate METHOTREXATE 29791011 14670 10001 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE AMG-191 AMG-191 14671 10002 CAPG 822 NA vincristine VINCRISTINE 14673 10003 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 178100383 14674 10004 TUBB6 84617 DRUGGABLE GENOME CHEMBL492399 VERUBULIN 14676 10005 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102678 14677 10006 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE LY3039478 CRENIGACESTAT 14678 10007 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE GLPG0187 GLPG-0187 14679 10008 VIM 7431 DRUGGABLE GENOME CHEMBL2108045 PRITUMUMAB 14680 10009 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE TAMOXIFEN TAMOXIFEN 9615734 14682 10010 IL1B 3553 KINASE, DRUGGABLE GENOME ACITRETIN ACITRETIN 1431212 14683 10011 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor 249565822 BALANOL 14684 10012 PTGS2 5743 DRUGGABLE GENOME, ENZYME Antiinflammatory agents, non-steroids 25876828,19602986 14685 10013 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BITHIONOL BITHIONOL 14686 10014 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME 1H-PYRROLO[2,3-B]PYRIDINE CHEMBL389685 26492576 14688 10015 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME Birinapant BIRINAPANT 14690 10016 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 223366123 BARICITINIB 14691 10017 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HEPTANE HEPTANE 14692 10018 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 310264692 VEROSUDIL 14694 10019 PLCG2 5336 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE, PHOSPHOLIPASE inhibitor 252827477 14695 10020 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417309 CHEMBL1341830 14696 10021 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL124660 TANDUTINIB 14697 10022 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103657 FLUOCINONIDE 14701 10023 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME idarubicin IDARUBICIN 22584460 14702 10024 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AM580 CHEMBL69367 14703 10025 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652301 14704 10026 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor DOVITINIB DOVITINIB 14705 10027 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME XANTHOHUMOL XANTHOHUMOL 22111577 14706 10028 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME PURPUROGALLIN PURPUROGALLIN 14707 10029 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545213 BENTAMAPIMOD 14708 10030 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR ARTESUNATE ARTESUNATE 25074847 14710 10031 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME daunorubicin DAUNORUBICIN 25119182 14711 10032 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR GNF-PF-2301 CHEMBL578061 14712 10033 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200759 ANAGRELIDE HYDROCHLORIDE 14713 10034 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125738 CHEMBL527585 14714 10035 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE CART-117 cells 14715 10036 POLB 5423 DNA REPAIR, DRUGGABLE GENOME 2-AMINOPHENOXAZINONE CHEMBL146710 14716 10037 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 223366126 DUVELISIB 14719 10038 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor 178103777 INAMRINONE 14722 10039 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE KX2-391 KX2-391 20038108 14726 10040 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GZ402674 14727 10041 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE MAPROTILINE MAPROTILINE 14728 10042 LGALS3 3958 CELL SURFACE, DRUGGABLE GENOME LACTOSE, ANHYDROUS LACTOSE, ANHYDROUS 21524586 14729 10043 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103398 ACETAZOLAMIDE 14730 10044 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CASEARINOL B CASEARINOL B 9322361 14731 10045 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Edotecarin EDOTECARIN 14733 10046 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME LITHIUM LITHIUM 12558976 14734 10047 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GNF-PF-1307 CHEMBL585030 14735 10048 BCHE 590 DRUGGABLE GENOME, ENZYME ISOFLUROPHATE ISOFLUROPHATE 14736 10049 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CNS-7056 REMIMAZOLAM 14737 10050 BAZ2B 29994 NA OMEPRAZOLE OMEPRAZOLE 14738 10051 CBX1 10951 NA PROCHLORPERAZINE PROCHLORPERAZINE 14739 10052 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE ETICLOPRIDE ETICLOPRIDE 14740 10053 HDAC11 79885 DRUGGABLE GENOME, ENZYME MOCETINOSTAT MOCETINOSTAT 23829483,26287310 14741 10054 FFAR4 338557 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100239 14742 10055 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE BVT-A 14743 10056 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE BGJ398 INFIGRATINIB 27401245,23443805,24122810,26036639,28034880,27870574,28119489,24563622,26048680 14744 10057 MFGE8 4240 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TRIAB 14747 10058 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178101324 14748 10059 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1417472 CHEMBL1563896 14749 10060 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME NAFTOPIDIL NAFTOPIDIL 14750 10061 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 249565764 14752 10062 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE TAE-684 TAE-684 14754 10063 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME Imatinib IMATINIB 18971950 14755 10064 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE L-733060 CHEMBL27006 14756 10065 TFF2 7032 DRUGGABLE GENOME Sivelestat sodium hydrate 14757 10066 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE AZD1390 14758 10067 MAPT 4137 DRUGGABLE GENOME GNF-PF-186 CHEMBL601140 14759 10068 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR SODIUM SALICYLATE 10574634 14761 10069 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR dopamine DOPAMINE 14763 10070 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LAVENDUSTIN A LAVENDUSTIN A 14765 10071 KCNH8 131096 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 14767 10072 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2062265 14768 10073 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 178103215 RIVASTIGMINE 14769 10074 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545154 POZIOTINIB 14770 10075 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ROBUSTONE ROBUSTONE 14772 10076 EGLN2 112398 ENZYME, DRUGGABLE GENOME GSK1278863 DAPRODUSTAT 14774 10077 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SB-220025 SB-220025 14775 10078 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME HYDROXYZINE HYDROXYZINE 14778 10079 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TOREMIFENE TOREMIFENE 14779 10080 PLA2G7 7941 DRUGGABLE GENOME, ENZYME DARAPLADIB DARAPLADIB 14780 10081 MAPT 4137 DRUGGABLE GENOME GNF-PF-3996 CHEMBL584458 14781 10082 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PROPAFENONE HYDROCHLORIDE PROPAFENONE HYDROCHLORIDE 14785 10083 GABBR2 9568 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL GAMMA HYDROXYBUTYRIC ACID 14787 10084 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2109587 AZ9773 14789 10085 SMN1 6606 DRUGGABLE GENOME MYCOPHENOLIC ACID MYCOPHENOLIC ACID 14792 10086 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR RALOXIFENE RALOXIFENE 14793 10087 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYDROCORTISONE ACETATE HYDROCORTISONE ACETATE 14795 10088 POLK 51426 DNA REPAIR, ENZYME AG-808 CHEMBL68534 14796 10089 CTH 1491 ENZYME Hydrazinoacetic acid 14797 10090 APOE 348 DRUGGABLE GENOME fenofibrate FENOFIBRATE 12042669 14798 10091 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE ORPHENADRINE ORPHENADRINE 14800 10092 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME URSODEOXYCHOLIC ACID 7712308 14801 10093 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor BUPARLISIB HYDROCHLORIDE 14802 10094 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TETRADECYLTHIOACETIC ACID TETRADECYLTHIOACETIC ACID 14803 10095 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor CHEMBL18 ETHOXZOLAMIDE 14804 10096 TYMP 1890 GROWTH FACTOR, DRUGGABLE GENOME S-1 16685374 14805 10097 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-37 14807 10098 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE Bafetinib BAFETINIB 14808 10099 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125734 CHEMBL586195 14809 10100 DOT1L 84444 CLINICALLY ACTIONABLE, DNA REPAIR, METHYL TRANSFERASE, DRUGGABLE GENOME, ENZYME inhibitor 178103597 14810 10101 TNNC1 7134 DRUGGABLE GENOME TIRAMSETIV 14811 10102 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME QUINOLINIC ACID QUINOLINIC ACID 14812 10103 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE PHENFORMIN PHENFORMIN 14813 10104 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102418 14818 10105 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BITHIONOLOXIDE BITHIONOLOXIDE 14820 10106 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR agonist 384403637 PURMORPHAMINE 14821 10107 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CITICOLINE SODIUM CITICOLINE SODIUM 14822 10108 CA1 759 DRUGGABLE GENOME, ENZYME activator 178100344 HISTIDINE 14824 10109 KCNA7 3743 ION CHANNEL, DRUGGABLE GENOME blocker 135650266 FLECAINIDE 14825 10110 XPC 7508 DNA REPAIR, CLINICALLY ACTIONABLE Platinum compounds 28791697 14826 10111 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME SP-600125 SP-600125 14827 10112 THBD 7056 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CILOSTAZOL CILOSTAZOL 10918946 14828 10113 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 223366195 14829 10114 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 14830 10115 PDE3A 5139 ENZYME, DRUGGABLE GENOME MILRINONE MILRINONE 14831 10116 HMGCR 3156 ENZYME, DRUGGABLE GENOME Hexahydro naphthalene derivative 2 14832 10117 UGT2B15 7366 DRUGGABLE GENOME phenobarbital PHENOBARBITAL 26049587 14836 10118 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME ANTIOXIDANT 17016661 14839 10119 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL2103856 ATOPAXAR 14841 10120 CBX1 10951 NA NSC-95397 CHEMBL429095 14843 10121 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Lenalidomide LENALIDOMIDE 14844 10122 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9181182, 34 14845 10123 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENCHLORAZOL-ETHYL FENCHLORAZOL-ETHYL 14846 10124 XDH 7498 DRUGGABLE GENOME, ENZYME Azaindole derivative 6 14847 10125 ATXN2 6311 NA TCMDC-125587 CHEMBL532160 14848 10126 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-36398 CHEMBL483206 14851 10127 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE FASUDIL FASUDIL 14852 10128 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME Zotarolimus ZOTAROLIMUS 14853 10129 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METIPRANOLOL METIPRANOLOL 14854 10130 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR VITAMIN A 9627692,10609868 14858 10131 NCL 4691 NA IPP-204106 14859 10132 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME inotersen INOTERSEN 14860 10133 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-17 14861 10134 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652116 14862 10135 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1201047 ANILERIDINE HYDROCHLORIDE 14863 10136 GZMA 3001 PROTEASE, DRUGGABLE GENOME, ENZYME CYCLOSPORINE CYCLOSPORINE 8420038 14864 10137 ANO1 55107 ION CHANNEL blocker 178100993 14865 10138 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FREUND'S ADJUVANT 15637741 14866 10139 MAOB 4129 DRUGGABLE GENOME, ENZYME ISOCARBOXAZID ISOCARBOXAZID 14867 10140 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME inhibitor CHEMBL1743016 FARLETUZUMAB 14868 10141 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METHYL 3-(2,5-DIHYDROXYPHENYL)ACRYLATE CHEMBL17329 14869 10142 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PURGIN II PURGIN II 23273047 14870 10143 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Tranexamic Acid 14872 10144 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2096626 14875 10145 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METACRESOL METACRESOL 14876 10146 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PF3644022 26140595 14878 10147 CP 1356 DRUGGABLE GENOME, ENZYME CLOMIPHENE CITRATE 1692793 14880 10148 TSPO 706 DRUGGABLE GENOME ESZOPICLONE ESZOPICLONE 14881 10149 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME NITROFURANTOIN NITROFURANTOIN 17093006 14884 10150 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME 20(S)-PROTOPANAXADIOL CHEMBL375563 26420067 14885 10151 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GELDANAMYCIN GELDANAMYCIN 25756299,25277067,21129982,18408713,18020309,21273068,21861487,23947794,23859777 14886 10152 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2103827 DROXIDOPA 14888 10153 PRSS2 5645 DRUGGABLE GENOME, PROTEASE, ENZYME CYANOPEPTOLIN S CYANOPEPTOLIN S 14889 10154 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL2104753 RIVOGLITAZONE 14891 10155 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Pyrrolidine derivative 11 14893 10156 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PERTUZUMAB PERTUZUMAB 14894 10157 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-59 14896 10158 NCOA3 8202 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, ENZYME TCMDC-123764 CHEMBL533226 14897 10159 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-108 CHEMBL578929 14899 10160 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 178101749 14900 10161 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZENE-1,2-DIAMINE CHEMBL70582 14901 10162 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL2408045 SAPITINIB 14902 10163 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ADRIAMYCIN ADRIAMYCIN 16893460 14903 10164 BAZ2B 29994 NA RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 14904 10165 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-38 14906 10166 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody DALOTUZUMAB DALOTUZUMAB 14907 10167 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Lofexidine LOFEXIDINE 14908 10168 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651497 14909 10169 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE RECOMBINANT INTERFERON ALFA-2B 14910 10170 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL TEZAMPANEL TEZAMPANEL 14912 10171 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 14913 10172 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Curcumin CURCUMIN 14914 10173 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR (S)-SARGACHROMENOL (S)-SARGACHROMENOL 21142112 14915 10174 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1744447 ROSUVASTATIN CALCIUM 14918 10175 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY DEXAMETHASONE DEXAMETHASONE 10468226 14919 10176 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME CENISERTIB CENISERTIB 14920 10177 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GYKI-52466 GYKI-52466 14921 10178 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103175 CHEMBL482436 14922 10179 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME DOCETAXEL DOCETAXEL 16983095 14923 10180 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PROTOAPIGENONE PROTOAPIGENONE 16038533 14926 10181 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AG-537 CHEMBL67535 14928 10182 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 1,6-diazanaphthalenes and pyrido[2,3-d] pyrimidine derivative 2 14929 10183 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NALMEFENE NALMEFENE 14930 10184 MPHOSPH8 54737 NA FIDUXOSIN HYDROCHLORIDE FIDUXOSIN HYDROCHLORIDE 14931 10185 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SUVN-D4010 SUVN-D4010 14932 10186 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE ritonavir RITONAVIR 26287941 14933 10187 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NOLATREXED NOLATREXED 14934 10188 TMPRSS2 7113 CLINICALLY ACTIONABLE, PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 405067326 14937 10189 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE OXYMORPHONE OXYMORPHONE 14938 10190 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR 6-HYDROXYMETHYLACYLFULVENE IROFULVEN 12014623 14939 10191 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-58 14940 10192 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PMID25726713-Compound-48 14941 10193 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SRA737 27167172 14942 10194 CEBPA 1050 TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE OICR-9429 26167872 14943 10195 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE KINETIN KINETIN 14944 10196 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 187051799 DACINOSTAT 14946 10197 MAPT 4137 DRUGGABLE GENOME 2,5-BIS(4-METHOXYSTYRYL)PYRAZINE CHEMBL2181039 22913544 14949 10198 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor DOVITINIB DOVITINIB 14950 10199 SMN1 6606 DRUGGABLE GENOME 2-AMINO-ANTHRAQUINONE CHEMBL84685 14951 10200 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME CHIR-99021 CHIR-99021 14953 10201 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME LORAZEPAM LORAZEPAM 14954 10202 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 5-O-methyl-M30 14955 10203 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GRISEOFULVIN GRISEOFULVIN 14956 10204 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR BDBM50363782 14957 10205 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE TANDUTINIB TANDUTINIB 14961 10206 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 328083483 PF-00562271 14962 10207 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-1872 CHEMBL600103 14964 10208 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PHENYLEPHRINE PHENYLEPHRINE 7567780 14965 10209 PSMD9 5715 NA inhibitor BORTEZOMIB BORTEZOMIB 14966 10210 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE DANAZOL DANAZOL 8529771,3146615,7607583 14968 10211 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652551 14969 10212 REG3A 5068 DRUGGABLE GENOME ALF-5755 25493266 14970 10213 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1723343 ZOLPIDEM TARTRATE 14971 10214 PRF1 5551 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME emapalumab EMAPALUMAB 14972 10215 ZSCAN25 221785 NA lumefantrine LUMEFANTRINE 14973 10216 KDM4A 9682 DRUGGABLE GENOME, ENZYME 2-PICOLINIC ACID 2-PICOLINIC ACID 14974 10217 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MITOXANTRONE MITOXANTRONE 14975 10218 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 695758 CHEMBL260028 14976 10219 NAT1 9 ENZYME, DRUGGABLE GENOME mesalazine MESALAMINE 14977 10220 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE TRASTUZUMAB TRASTUZUMAB 21594665,19010894,20453058,22294718,26920887 14980 10221 BRCA2 675 CLINICALLY ACTIONABLE YU238259 26116172 14983 10222 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE DWP-09031 14985 10223 USP1 7398 DNA REPAIR, PROTEASE, ENZYME RU-24969 RU-24969 14986 10224 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR AT-406 AT-406 25520882 14987 10225 GPA33 10223 DRUGGABLE GENOME MGD007 MGD-007 14988 10226 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE CODEINE CODEINE 14989 10227 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL antagonist 385612191 14991 10228 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102596 14992 10229 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NIFEDIPINE NIFEDIPINE 14993 10230 KLF5 688 TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, DRUGGABLE GENOME OUABAIN OUABAIN 14994 10231 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Quinoline derivative 15 14997 10232 ALOX15 246 ENZYME, DRUGGABLE GENOME CATECHOL CATECHOL 14998 10233 DYRK2 8445 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 249565847 15001 10234 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME MTX METHOTREXATE 15670151 15002 10235 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MECLIZINE MECLIZINE 15003 10236 POLI 11201 DNA REPAIR AG-808 CHEMBL68534 15004 10237 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417221 CHEMBL1459280 15005 10238 CACNB4 785 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1628502 GABAPENTIN ENACARBIL 15006 10239 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 249565855 15007 10240 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ESREBOXETINE ESREBOXETINE 15008 10241 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ESTRAMUSTINE ESTRAMUSTINE 15009 10242 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102585 DOVITINIB 15010 10243 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME dapsone DAPSONE 28885988,23604100,24152261,29512326,29458119 15011 10244 TMEM97 27346 NA N-substituted 9-azabicyclo[3.3.1]nonan-3alpha-yl-phenylcarbamate analog 1 15012 10245 TUBA4A 7277 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 15014 10246 ATAD5 79915 NA RO-5-3335 CHEMBL91609 15015 10247 HDAC11 79885 DRUGGABLE GENOME, ENZYME PANOBINOSTAT PANOBINOSTAT 15018 10248 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE ISIS-CRP 15019 10249 OGG1 4968 ENZYME CAFFEINE CAFFEINE 18557781 15020 10250 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE GW843682X GW843682X 15023 10251 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIFLUBENZURON DIFLUBENZURON 15026 10252 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL2364574 DOXYCYCLINE CALCIUM 15027 10253 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE LAPATINIB LAPATINIB 19010894,22294718,26920887 15028 10254 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER lopinavir LOPINAVIR 23996099 15029 10255 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME DA-1229 EVOGLIPTIN 15030 10256 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE DIPYRIDAMOLE DIPYRIDAMOLE 15031 10257 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 328083494 15032 10258 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER lamivudine LAMIVUDINE 15033 10259 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103532 15034 10260 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE LEVORPHANOL LEVORPHANOL 15041 10261 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ELATOSIDE D ELATOSIDE D 21889336 15043 10262 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Muc1-specific gene-engineered T cells 15044 10263 CDH2 1000 CELL SURFACE, DRUGGABLE GENOME ADH-1 ADH-1 15047 10264 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PRACTOLOL PRACTOLOL 2903243 15050 10265 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID27724045-Compound-29 15051 10266 ATXN2 6311 NA THIRAM THIRAM 15052 10267 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102421 15053 10268 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649735 15054 10269 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 310264726 15055 10270 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Beperminogene perplasmid 15056 10271 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RESOKAEMPFEROL RESOKAEMPFEROL 15058 10272 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME hmg coa reductase inhibitors 15059 10273 MGLL 11343 DRUGGABLE GENOME, ENZYME Piperazine carbamic compound 1 15060 10274 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FST-201 15063 10275 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE ENPIROLINE ENPIROLINE 15064 10276 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME AG1295 AG1295 15065 10277 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GUANIDINONALTRINDOLE GUANIDINONALTRINDOLE 15068 10278 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR JTE-451 15069 10279 HTRA1 5654 ENZYME, DRUGGABLE GENOME, PROTEASE HYDROGEN PEROXIDE 10517331 15071 10280 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SJ000044511 CHEMBL592124 15072 10281 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IPRONIAZID IPRONIAZID 22931300 15073 10282 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PADIMATE O PADIMATE O 15075 10283 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor BI-2536 BI-2536 15076 10284 GMNN 51053 DRUGGABLE GENOME DNDI1417185 CHEMBL1549738 15078 10285 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME S-49076 23175443,23804704 15080 10286 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ISOPROTERENOL ISOPROTERENOL 15081 10287 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TAE-684 TAE-684 15083 10288 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE RIGOSERTIB RIGOSERTIB 15085 10289 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N/A 25326232 15086 10290 GMNN 51053 DRUGGABLE GENOME TRIFLUOPERAZINE HYDROCHLORIDE TRIFLUOPERAZINE HYDROCHLORIDE 15087 10291 RAB9A 9367 ENZYME, DRUGGABLE GENOME SB-204741 CHEMBL323356 15089 10292 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Cycloalkyl nitrile pyrazolo pyridone derivative 2 15091 10293 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NICLOSAMIDE NICLOSAMIDE 15092 10294 PTGES 9536 DRUGGABLE GENOME, ENZYME Benzimidazole derivative 16 15093 10295 DHX36 170506 NA MANOALIDE MANOALIDE 22394195 15094 10296 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR MECHLORETHAMINE MECHLORETHAMINE 10640980 15096 10297 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ORAL CONTRACEPTIVE 15298951 15097 10298 PDE4B 5142 DRUGGABLE GENOME, ENZYME TCMDC-125454 CHEMBL535714 15098 10299 TUBB3 10381 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 15099 10300 CD8A 925 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE Fluoropeptide vaccine 15103 10301 ATAD5 79915 NA IPRIFLAVONE IPRIFLAVONE 15106 10302 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR inhibitor CHEMBL467 HYDROXYUREA 15107 10303 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417264 CHEMBL1467200 15108 10304 ZSCAN25 221785 NA lopinavir LOPINAVIR 15109 10305 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545052 FIMEPINOSTAT 15110 10306 PYY 5697 DRUGGABLE GENOME, HORMONE ACTIVITY Peptide YY 3-36 15113 10307 DGAT1 8694 ENZYME, DRUGGABLE GENOME Lactam derivative 2 15117 10308 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2010077680 495 15118 10309 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR SALINE SODIUM CHLORIDE 17334244 15120 10310 MAPT 4137 DRUGGABLE GENOME PH-011685 CHEMBL126804 15121 10311 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME ORPHENADRINE ORPHENADRINE 15122 10312 CD3D 915 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE CHEMBL1742992 BLINATUMOMAB 15123 10313 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PHA-767491 CHEMBL225519 15124 10314 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR candesartan CANDESARTAN 18594050 15126 10315 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SJ000032152 CHEMBL590665 15128 10316 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-102 15129 10317 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DROLOXIFENE DROLOXIFENE 11721384 15130 10318 MGLL 11343 DRUGGABLE GENOME, ENZYME Pyrazole derivative 84 15131 10319 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100315 15132 10320 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565590 CHEMBL1236539 15133 10321 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXYPHENBUTAZONE OXYPHENBUTAZONE 15134 10322 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY PHENYTOIN PHENYTOIN 3935423 15135 10323 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE lapatinib LAPATINIB 26570998,23220880 15137 10324 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR risperidone RISPERIDONE 23422377 15140 10325 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL451 CHLORDIAZEPOXIDE 15144 10326 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Autologous T Cells Expressing MET scFv CAR 15147 10327 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 15148 10328 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE LEVALLORPHAN LEVALLORPHAN 15149 10329 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME daunorubicin DAUNORUBICIN 26663398 15150 10330 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR spironolactone SPIRONOLACTONE 22543981 15152 10331 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-139459 CHEMBL86464 15153 10332 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID28048944-Compound-11 15155 10333 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE CHOLIC ACID CHOLIC ACID 19102680 15156 10334 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BI 882370 26916115 15157 10335 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME DM-71 15158 10336 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-137192 CHEMBL268584 15159 10337 TARDBP 23435 TUMOR SUPPRESSOR PTEROSTILBENE PTEROSTILBENE 15161 10338 ALDH5A1 7915 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL433 VALPROATE SODIUM 15162 10339 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEXRAZOXANE DEXRAZOXANE 12911317 15164 10340 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR BUTANOIC ACID BUTANOIC ACID 19053749 15165 10341 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE simvastatin SIMVASTATIN 24598718,23252946,17192506,18695978,17289397,26164721,16321621,15284534 15166 10342 ENOSF1 55556 ENZYME methotrexate METHOTREXATE 18322994,16130010 15167 10343 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 178103995 LINSITINIB 15168 10344 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor 178101944 ROLIPRAM 15170 10345 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE NPS-1034 24165158,23542356 15171 10346 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NALOXONE NALOXONE 15172 10347 BCOR 54880 CLINICALLY ACTIONABLE N/A 26150234,26098867,26573325,26516930 15174 10348 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GW7074 CHEMBL72365 15175 10349 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Niraparib NIRAPARIB 15176 10350 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL ANAVEX 2-73 15178 10351 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL2331680 RG-7603 15180 10352 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GSK3787 CHEMBL598608 25768705 15181 10353 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ORTHO-METHOXYCINNAMALDEHYDE CHEMBL83159 15182 10354 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GEMCITABINE HYDROCHLORIDE GEMCITABINE HYDROCHLORIDE 15184 10355 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 IPRATROPIUM IPRATROPIUM 22931300 15185 10356 SMN1 6606 DRUGGABLE GENOME PT-103 CHEMBL398765 15186 10357 POLI 11201 DNA REPAIR ERGOCRYPTINE ERGOCRYPTINE 15187 10358 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE RG-7010 15188 10359 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE ACETAMINOPHEN ACETAMINOPHEN 11896290 15190 10360 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Dasatinib DASATINIB 15191 10361 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME PAPAVERINE PAPAVERINE 15193 10362 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor CHEMBL445813 AT-7519 15194 10363 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE R-flurbiprofen 15195 10364 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor PWT33597 15196 10365 LAMB2 3913 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 15197 10366 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GRAVEOLINE GRAVEOLINE 15200 10367 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-1030062A GSK-1030062A 15201 10368 PRKAG2 51422 ENZYME, KINASE SAPONARIN SAPONARIN 26471090 15202 10369 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME R3Mab 25326231,19381019 15203 10370 GMNN 51053 DRUGGABLE GENOME TYRPHOSTIN A9 TYRPHOSTIN A9 15204 10371 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CDX-3379 26880266,18441328 15205 10372 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CUDC-101 CUDC-101 15206 10373 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GW3965 CHEMBL59030 15207 10374 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125784 CHEMBL581574 15210 10375 KDM4A 9682 DRUGGABLE GENOME, ENZYME GLYASPERIN D GLYASPERIN D 15212 10376 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SUBEROHYDROXAMIC ACID SUBEROHYDROXAMIC ACID 16921367 15213 10377 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 385612233 15214 10378 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist 252166532 ABT 737 15215 10379 DNER 92737 NA PLX51107 15216 10380 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ILOPROST ILOPROST 15217 10381 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 223366077 RGB-286638 15218 10382 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHR-3996 NANATINOSTAT 15219 10383 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TYRPHOSTIN 1 TYRPHOSTIN 1 15220 10384 POLK 51426 DNA REPAIR, ENZYME SENNOSIDE B SENNOSIDE B 15221 10385 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CARBENOXOLONE DISODIUM CARBENOXOLONE SODIUM 15222 10386 PBK 55872 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, ENZYME BAY-613606 CHEMBL541400 15225 10387 SGK1 6446 SERINE THREONINE KINASE, KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME, DRUG RESISTANCE CI-1040 CI-1040 15227 10388 REG3A 5068 DRUGGABLE GENOME SALT VOLANESORSEN SODIUM 9024308 15228 10389 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE 404859000 ELEXACAFTOR 15230 10390 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE AFATINIB AFATINIB 27044931,24685132 15231 10391 GLS 2744 ENZYME GARENOXACIN GARENOXACIN 15233 10392 RUNX2 860 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR ANTISENSE OLIGONUCLEOTIDES 10722711 15234 10393 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8829193, 1 15235 10394 DDC 1644 ENZYME, DRUGGABLE GENOME carbidopa CARBIDOPA 15236 10395 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE TASELISIB TASELISIB 26589432 15238 10396 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE Famitinib FAMITINIB 15239 10397 SMN1 6606 DRUGGABLE GENOME AZARIBINE AZARIBINE 15240 10398 EIF2AK2 5610 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR RICIN 18599499 15242 10399 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor CHEMBL3545377 LY-2606368 15244 10400 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE VANDETANIB VANDETANIB 15245 10401 HMGCR 3156 ENZYME, DRUGGABLE GENOME 2-cyclopropyl-4-substituted-phenoxy-quinoline derivative 1 15246 10402 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LENVATINIB LENVATINIB 15247 10403 XPO1 7514 CLINICALLY ACTIONABLE, KINASE KOS-1815 24631834 15248 10404 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME CHZ868 26175413 15249 10405 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TDR77585 CHEMBL1333386 15250 10406 CBX1 10951 NA NSC-107022 CHEMBL1601846 15251 10407 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ARRY-797 ARRY-797 15255 10408 GAA 2548 DRUGGABLE GENOME, ENZYME inhibitor 381118910 MIGALASTAT 15256 10409 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 223366206 INFIGRATINIB 15258 10410 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ELLAGIC ACID ELLAGIC ACID 15261 10411 NR1D1 9572 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME antagonist 135651083 15263 10412 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE TCMDC-125221 CHEMBL546649 15264 10413 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650925 15266 10414 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME NITRAZEPAM NITRAZEPAM 15267 10415 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE BOVINE CARTILAGE 9085145 15268 10416 MEGF11 84465 NA fluorouracil FLUOROURACIL 24444404 15269 10417 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE Elisidepsin 15271 10418 DPP6 1804 DRUGGABLE GENOME, ENZYME, TRANSPORTER, PROTEASE ethanol ALCOHOL 32451486 15274 10419 GLS 2744 ENZYME OXYTETRACYCLINE OXYTETRACYCLINE 15276 10420 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200873 PHENTOLAMINE MESYLATE 15277 10421 TRIB3 57761 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE methylphenidate METHYLPHENIDATE 29382897 15278 10422 ATXN2 6311 NA SCLEROTIORIN SCLEROTIORIN 15279 10423 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR CLOBETASOL CLOBETASOL 15280 10424 RABEP1 9135 CLINICALLY ACTIONABLE, GROWTH FACTOR amisulpride AMISULPRIDE 28694205 15281 10425 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME donepezil DONEPEZIL 24433464,26952092 15283 10426 AQP9 366 ION CHANNEL ANTISERUM 16035648 15284 10427 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER RITUXIMAB RITUXIMAB 16971809 15285 10428 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TCMDC-124240 CHEMBL582764 15286 10429 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ISOLIQUIRITIGENIN ISOLIQUIRITIGENIN 15288 10430 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLOFAZIMINE CLOFAZIMINE 15289 10431 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME inhibitor 178102814 VERLUKAST 15290 10432 TUBB2B 347733 DRUGGABLE GENOME ABT-751 ABT-751 25468039 15291 10433 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 15292 10434 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PI3-KINASE INHIBITORS 12736339 15294 10435 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL27759 ENTINOSTAT 15295 10436 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TRANSPLATIN TRANSPLATIN 15296 10437 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2004087707 15297 10438 PTGS1 5742 ENZYME, DRUGGABLE GENOME NABUMETONE NABUMETONE 15298 10439 SCG5 6447 CLINICALLY ACTIONABLE, DRUGGABLE GENOME CAPSAICIN CAPSAICIN 3858706 15300 10440 JUNB 3726 TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR UVB 9607142 15301 10441 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME IMATINIB IMATINIB 15805252 15302 10442 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PD-169316 PD-169316 15304 10443 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SALVINORIN A 15305 10444 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ondansetron ONDANSETRON 25012726,20707787 15307 10445 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1201733 PAZOPANIB HYDROCHLORIDE 15309 10446 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR TAZAROTENE TAZAROTENE 15610529 15311 10447 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Flavonoid derivative 1 15313 10448 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR antagonist 178104004 BIRINAPANT 15314 10449 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ALPHA-NAPHTHOFLAVONE ALPHA-NAPHTHOFLAVONE 15316 10450 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZASERINE AZASERINE 15318 10451 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE EPZ004777 27535106 15319 10452 DPP8 54878 DRUGGABLE GENOME, PROTEASE, ENZYME Thiomorpholine derivative 1 15323 10453 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ONO-5129 15324 10454 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR RHAMNETIN RHAMNETIN 15326 10455 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DESOXYCORTICOSTERONE PIVALATE 15327 10456 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESCULIN ESCULIN 15329 10457 MAPT 4137 DRUGGABLE GENOME 7,8,2'-TRIHYDROXYFLAVONE CHEMBL244707 15330 10458 TNNC1 7134 DRUGGABLE GENOME Levosimendan LEVOSIMENDAN 15331 10459 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Cisplatin CISPLATIN 15333 10460 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SODIUM DIMETHYLCARBAMODITHIOATE SODIUM DIMETHYLCARBAMODITHIOATE 15334 10461 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE GDC-0941 PICTILISIB 28119489 15335 10462 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tacrine-phenothiazine hybrid derivative 1 15336 10463 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE BEPRIDIL BEPRIDIL 15339 10464 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GNF-PF-4337 CHEMBL277148 15340 10465 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DOCUSATE SODIUM DOCUSATE SODIUM 15341 10466 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545365 ALTIRATINIB 15343 10467 TSPO 706 DRUGGABLE GENOME PMID27599163-Compound-82 15345 10468 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METHYLDOPA (RACEMIC) METHYLDOPA (RACEMIC) 15346 10469 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652098 15347 10470 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SNS-314 SNS-314 15348 10471 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR LOVASTATIN LOVASTATIN 15349 10472 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CID 4101591 CHEMBL428789 15350 10473 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE ENMD-1198 15351 10474 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE GSK3052230 FP-1039 23536011 15352 10475 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE BERKELEYACETAL C BERKELEYACETAL C 17970594 15354 10476 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DN24-02 15355 10477 MARCHF8 220972 ENZYME Aflunov 15356 10478 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE BUCINDOLOL BUCINDOLOL 15360 10479 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201653 INSULIN ZINC SUSP PURIFIED PORK 15363 10480 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR ALISERTIB ALISERTIB 15365 10481 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR OXYTETRACYCLINE OXYTETRACYCLINE 15366 10482 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ANTIPARASITIC 16381664 15368 10483 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME febuxostat FEBUXOSTAT 27798726 15369 10484 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MORPHINE MORPHINE 15371 10485 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ACETAMINOPHEN ACETAMINOPHEN 2242029 15372 10486 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545234 15373 10487 RGS4 5999 DRUGGABLE GENOME METHYLDOPA (RACEMIC) METHYLDOPA (RACEMIC) 15374 10488 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-67436 CHEMBL1331995 15376 10489 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME Anti-CEA CAR-T cells 15378 10490 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ZAFIRLUKAST ZAFIRLUKAST 15379 10491 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL592445 GEDATOLISIB 15380 10492 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3545178 CERALASERTIB 15382 10493 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE Fruquintinib FRUQUINTINIB 15386 10494 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE doxorubicin DOXORUBICIN 15387 10495 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 theophylline THEOPHYLLINE 15388 10496 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1370561 AMINOPHYLLINE 15389 10497 HTT 3064 DRUGGABLE GENOME LEFLUNOMIDE LEFLUNOMIDE 15390 10498 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE QUINALIZARIN QUINALIZARIN 15391 10499 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW300657X GW300657X 15392 10500 CEL 1056 CELL SURFACE, DRUGGABLE GENOME, ENZYME ACTINOMYCIN D 2016288 15394 10501 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Fused triazoloamino-phenyl analog 1 15396 10502 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL112 ACETAMINOPHEN 15397 10503 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Gefitinib GEFITINIB 17463250,24165158,23542356,27612490 15398 10504 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 381744920 15399 10505 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL2107832 PIMASERTIB 15400 10506 RORB 6096 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, KINASE US9598431, 5 15402 10507 BAZ2B 29994 NA NALIDIXIC ACID NALIDIXIC ACID 15403 10508 CSF1 1435 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Emactuzumab EMACTUZUMAB 15404 10509 PTGS2 5743 DRUGGABLE GENOME, ENZYME Tenoxicam TENOXICAM 15405 10510 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-125000 CHEMBL579742 15406 10511 DPP9 91039 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 363894186 TALABOSTAT 15407 10512 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL FELODIPINE FELODIPINE 15408 10513 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ASPIRIN ASPIRIN 15200494 15409 10514 LANCL2 55915 NA 384403642 15410 10515 TUBB2B 347733 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 15411 10516 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL494089 GSK-690693 15412 10517 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 3-(N-PHENETHYLSULFAMOYL)BENZOIC ACID CHEMBL1871992 15414 10518 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR N-quinolin-benzene sulphonamide derivative 2 15415 10519 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE VATALANIB VATALANIB 15417 10520 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-319347A GSK-319347A 15418 10521 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL325041 BORTEZOMIB 15422 10522 ALOX15B 247 DRUGGABLE GENOME, ENZYME NSC-632536 CHEMBL1367933 15423 10523 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME ENTRECTINIB ENTRECTINIB 15424 10524 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE methotrexate METHOTREXATE 22016816,21317831,21606946 15425 10525 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ANTIESTROGEN 11306479 15426 10526 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME MAXY-G34 15427 10527 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME GENISTEIN GENISTEIN 15428 10528 ARID1A 8289 CLINICALLY ACTIONABLE SORAFENIB SORAFENIB 29113912 15429 10529 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE loratadine LORATADINE 18695978 15431 10530 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME leucovorin LEUCOVORIN 16115875 15432 10531 NDUFA10 4705 ENZYME inhibitor CHEMBL3545135 NV-128 15433 10532 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENOL PHENOL 15434 10533 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MT-3995 MT-3995 15435 10534 FZD6 8323 CELL SURFACE, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651914 15436 10535 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650701 15438 10536 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR OBETICHOLIC ACID 15440 10537 GUSB 2990 DRUGGABLE GENOME, ENZYME PerioPatch 15441 10538 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER OXALIPLATIN OXALIPLATIN 24957073 15443 10539 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE ERLOTINIB ERLOTINIB 31027687 15445 10540 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIENESTROL DIENESTROL 15446 10541 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor AMG900 AMG-900 15448 10542 ATAD5 79915 NA N-PHENETHYL-NICOTINAMIDE CHEMBL309848 15449 10543 PADI3 51702 ENZYME, DRUGGABLE GENOME O-F-AMIDINE CHEMBL1910970 21882827 15452 10544 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR Saracatinib SARACATINIB 26802156 15453 10545 PTBP1 5725 DRUGGABLE GENOME GNF-PF-4418 CHEMBL604321 15454 10546 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME UC-857993 25825487 15456 10547 NDUFA12 55967 ENZYME inhibitor CHEMBL3545135 NV-128 15457 10548 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMITRIPTYLINE AMITRIPTYLINE 22931300 15458 10549 TUBB 203068 DRUGGABLE GENOME ABI-011 15459 10550 PTPRD 5789 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE US9340574, 7 15460 10551 GMNN 51053 DRUGGABLE GENOME DIGOXIN DIGOXIN 15461 10552 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE docetaxel DOCETAXEL 21151855 15462 10553 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33l 15463 10554 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE BENZBROMARONE BENZBROMARONE 15465 10555 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Aminopyridine derivative 1 15466 10556 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TENIPOSIDE TENIPOSIDE 15467 10557 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORMADINONE CHLORMADINONE 15468 10558 CBX1 10951 NA OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 15469 10559 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650869 QUETIAPINE 15470 10560 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE CALCITRIOL CALCITRIOL 3139763 15472 10561 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme12-1 15473 10562 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Rucaparib RUCAPARIB 28148839 15476 10563 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUSILAZOLE FLUSILAZOLE 15478 10564 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor 178103252 SELEGILINE 15480 10565 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY PREDNISONE PREDNISONE 2745931 15481 10566 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISOPIMPINELLIN ISOPIMPINELLIN 15483 10567 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PMID28048944-Compound-6 15484 10568 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Mosapride MOSAPRIDE 15486 10569 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125756 CHEMBL536599 15487 10570 CD276 80381 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME antibody 340590220 ENOBLITUZUMAB 15488 10571 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CHLOROPYRAMINE CHLOROPYRAMINE 15489 10572 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IV-23D1 CHEMBL1094675 20371180 15490 10573 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID27744724-Compound-26 15491 10574 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME C5A 8348695 15492 10575 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE HYPOXANTHINE HYPOXANTHINE 3528863 15493 10576 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR 6-BROMOTRYPTOPHANARGININE CHEMBL401607 18271554 15494 10577 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PX-866 SONOLISIB 15496 10578 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-26 15497 10579 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-71 15498 10580 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL1946170 REGORAFENIB 15499 10581 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650699 15500 10582 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR BOVINE CARTILAGE 12525389 15503 10583 ALOX15 246 ENZYME, DRUGGABLE GENOME DALBERGIONE, 4-METHOXY-4'-HYDROXY- DALBERGIONE, 4-METHOXY-4'-HYDROXY- 15506 10584 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-7 15508 10585 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME inhibitor 178103314 15509 10586 EYA2 2139 DNA REPAIR DNDI1417099 CHEMBL1565444 15511 10587 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BUPARLISIB HYDROCHLORIDE 15512 10588 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 1225609 CHEMBL444376 15513 10589 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE sitamaquine SITAMAQUINE 15514 10590 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME KRP-104 BISEGLIPTIN 15515 10591 PAPPA 5069 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE TRANSFORMING GROWTH FACTOR 12817760 15516 10592 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL AZIETOMIDATE AZIETOMIDATE 16884293 15517 10593 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME VX-680 TOZASERTIB 15519 10594 DGAT2 84649 ENZYME PMID25470667-Compound-roselipins 15520 10595 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PINDOLOL PINDOLOL 2903243 15521 10596 ATAD5 79915 NA TCMDC-125738 CHEMBL527585 15522 10597 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DAIDZEIN DAIDZEIN 15523 10598 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL3707355 AZD8108 15524 10599 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID26161698-Compound-17 15525 10600 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1200933 HEXAFLUORENIUM BROMIDE 15526 10601 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AZD-1080 AZD-1080 15528 10602 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PANITUMUMAB PANITUMUMAB 28783719,19001320,25673644,26687137,23325582,31515458,29431699 15529 10603 DDO 8528 DRUGGABLE GENOME topotecan TOPOTECAN 24444404 15533 10604 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE DNDI1417467 CHEMBL1997335 15536 10605 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 178100973 15537 10606 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AMINOQUINURIDE AMINOQUINURIDE 15538 10607 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2107760 NEBENTAN 15540 10608 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHA-767491 CHEMBL225519 15542 10609 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL193 NIFEDIPINE 15543 10610 PSPH 5723 ENZYME l-methionine METHIONINE 24651765 15544 10611 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME CAR-T cells targeting Mucl 15545 10612 ALDH7A1 501 ENZYME, DRUGGABLE GENOME M-518101 PEFCALCITOL 15546 10613 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIMETHYLPHENYLPIPERAZINIUM DIMETHYLPHENYLPIPERAZINIUM 15548 10614 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE METHYLCURCUMIN METHYLCURCUMIN 25753330 15549 10615 PTGS1 5742 ENZYME, DRUGGABLE GENOME DERSALAZINE DERSALAZINE 15550 10616 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 8425178 15551 10617 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545368 PANOBINOSTAT LACTATE 15552 10618 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIBUTYLCHLOROSTANNANE TRIBUTYLCHLOROSTANNANE 15553 10619 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE HEPTACHLOR HEPTACHLOR 15556 10620 MPHOSPH8 54737 NA MITOXANTRONE MITOXANTRONE 15557 10621 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE palbociclib PALBOCICLIB 15558 10622 BACH1 571 DNA REPAIR, TRANSCRIPTION FACTOR isoniazid ISONIAZID 22341855,29036176 15560 10623 UGT2B7 7364 DRUGGABLE GENOME fluvastatin FLUVASTATIN 15561 10624 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-40 15562 10625 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Pegvisomant PEGVISOMANT 15563 10626 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1200984 AMLODIPINE MALEATE 15564 10627 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME JNJ-7706621 JNJ-7706621 21106455 15565 10628 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR QUINOXYFEN QUINOXYFEN 15566 10629 LIPF 8513 ENZYME, DRUGGABLE GENOME Cetilistat CETILISTAT 15567 10630 CBX1 10951 NA NSC-699479 CHEMBL1701915 15568 10631 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE alpelisib ALPELISIB 15569 10632 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Thiazolidinedione THIAZOLIDINEDIONE 15570 10633 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CEPHALOTHIN CEPHALOTHIN 15571 10634 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE dexamethasone DEXAMETHASONE 15573 10635 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR gemcitabine GEMCITABINE 31616045 15574 10636 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME FolateImmune 15575 10637 BAZ2B 29994 NA CHLORPROMAZINE HYDROCHLORIDE CHLORPROMAZINE HYDROCHLORIDE 15576 10638 ADAM10 102 ENZYME, CELL SURFACE, TRANSPORTER, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE inhibitor 348353646 15577 10639 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200443 MERETHOXYLLINE PROCAINE 15578 10640 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1743087 VEDOLIZUMAB 15579 10641 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL MIDAZOLAM MIDAZOLAM 15580 10642 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER QUINALIZARIN QUINALIZARIN 15581 10643 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AZTREONAM AZTREONAM 22931300 15582 10644 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL646 TRIAZOLAM 15583 10645 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NAFAMOSTAT NAFAMOSTAT 15584 10646 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545285 XL-999 15586 10647 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME PREMETREXED 15587 10648 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 178102318 KW-2449 15589 10649 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyrimidine derivative 10 15590 10650 RABGAP1L 9910 NA ethanol ALCOHOL 15591 10651 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PANITUMUMAB PANITUMUMAB 29196463,24653627,26888827,28287083 15592 10652 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE BIL010t 15593 10653 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER DNDI1417599 CHEMBL2094833 15595 10654 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 135651065 SPIRONOLACTONE 15596 10655 AKR1C3 8644 ENZYME, DRUGGABLE GENOME Beta-naphthylacetic acids derivative 1 15597 10656 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PSAMMAPLIN A PSAMMAPLIN A 25884112 15598 10657 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE ENTRECTINIB ENTRECTINIB 15599 10658 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID2350207 CHEMBL259615 15600 10659 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 252827451 SAR-260301 15601 10660 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME BERKELEYACETAL A BERKELEYACETAL A 17970594 15603 10661 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE 6,6-fused nitrogenous heterocyclic compound 3 15605 10662 WNK2 65268 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565802 15606 10663 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 7 15607 10664 CRBN 51185 ENZYME, DRUG RESISTANCE inhibitor CHEMBL468 THALIDOMIDE 15611 10665 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3218576 COPANLISIB 15612 10666 GAA 2548 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1561 MIGLITOL 15615 10667 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PONATINIB PONATINIB 22238366,26179511,24771645 15620 10668 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 223365885 DOTHIEPIN 15624 10669 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MESALAMINE MESALAMINE 15625 10670 PTGES 9536 DRUGGABLE GENOME, ENZYME Piperidine carboxamide derivative 1 15626 10671 BCHE 590 DRUGGABLE GENOME, ENZYME Quinazoline alkaloid derivative 1 15628 10672 AKR1C1 1645 DRUGGABLE GENOME, ENZYME ESTRONE ESTRONE 3859707 15630 10673 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLUMAZENIL FLUMAZENIL 15631 10674 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Peptide analog 53 15635 10675 KRT17 3872 NA IFN 7516473 15636 10676 CTH 1491 ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 27779248 15637 10677 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Benzamide derivative 11 15639 10678 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL2178577 AZD-5363 15640 10679 TK2 7084 KINASE, ENZYME, DRUGGABLE GENOME DDC ZALCITABINE 14659972 15642 10680 ALOX5 240 DRUGGABLE GENOME, ENZYME ABT-761 ATRELEUTON 15643 10681 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor GDC-0980 APITOLISIB 15644 10682 MAP3K13 9175 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL290352 CEP-1347 15646 10683 MAPT 4137 DRUGGABLE GENOME 3,8'-BIAPIGENIN CHEMBL515252 15647 10684 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR JNK-401 15648 10685 TUBB3 10381 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 15650 10686 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 249565705 TIPIFARNIB 15652 10687 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME MYRICETIN MYRICETIN 15653 10688 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MENADIONE MENADIONE 15654 10689 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR LINOLENIC ACID LINOLENIC ACID 15655 10690 DUSP3 1845 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE LOMOFUNGIN LOMOFUNGIN 15657 10691 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME PROTEASOME INHIBITOR 15890091 15658 10692 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR modulator CHEMBL2105694 TELAPRISTONE ACETATE 15659 10693 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 15662 10694 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE BGB-324 BEMCENTINIB 15663 10695 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 15664 10696 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR TEW-7197 VACTOSERTIB 15665 10697 MAOB 4129 DRUGGABLE GENOME, ENZYME 3,4-Dihydroxybenzaldehyde 15667 10698 CBX1 10951 NA AG-808 CHEMBL68534 15670 10699 MAPT 4137 DRUGGABLE GENOME PD-169316 PD-169316 15673 10700 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100325 15675 10701 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135651122 15677 10702 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SELUMETINIB SELUMETINIB 23200175,19029981,25199829,21985784,26125448,28492898,22392911 15678 10703 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor 223366042 CAPIVASERTIB 15679 10704 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NANDROLONE NANDROLONE 15680 10705 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 385612249 15682 10706 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-139459 CHEMBL86464 15683 10707 POLI 11201 DNA REPAIR DNDI1416969 CHEMBL1453126 15684 10708 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 249565819 15685 10709 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SB-216763 SB-216763 15686 10710 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRETINOIN TRETINOIN 15692 10711 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE RU 486 7627771 15694 10712 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AG-538 CHEMBL56393 15695 10713 KCNT2 343450 ION CHANNEL, DRUGGABLE GENOME activator 135650269 15697 10714 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL876 MECLOFENAMATE SODIUM 15703 10715 GAA 2548 DRUGGABLE GENOME, ENZYME MORIN MORIN 15704 10716 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 178103494 IBRUTINIB 15705 10717 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME U-74389G MALEATE CHEMBL1256186 15706 10718 GMNN 51053 DRUGGABLE GENOME CORONOPILIN CORONOPILIN 15708 10719 PSMB9 5698 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL451887 CARFILZOMIB 15709 10720 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PAZOPANIB PAZOPANIB 15710 10721 GAA 2548 DRUGGABLE GENOME, ENZYME AM-404 CHEMBL39878 15711 10722 RGS4 5999 DRUGGABLE GENOME inhibitor 249565573 CHEMBL1917204 15712 10723 RPS6KA6 27330 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME US10081632, Compound 25 15713 10724 CD37 951 DRUGGABLE GENOME BI-836826 15714 10725 BAZ2B 29994 NA GNF-PF-321 CHEMBL581044 15716 10726 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME SB-220025 SB-220025 15717 10727 ALDH1A2 8854 DRUGGABLE GENOME, ENZYME atenolol ATENOLOL 29097388 15718 10728 GCH1 2643 ENZYME ProSavin 15720 10729 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME ESTAZOLAM ESTAZOLAM 15721 10730 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102559 NINTEDANIB 15722 10731 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR PROTEASOME INHIBITOR 11509005 15723 10732 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME inhibitor 252827482 15724 10733 PDE7B 27115 DRUGGABLE GENOME, ENZYME inhibitor 178101846 15725 10734 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TANSHINONE IIA SULFONATE TANSHINONE IIA SULFONATE 15726 10735 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE CYC-116 CYC-116 15727 10736 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL NG2-73 ADIPIPLON 15729 10737 GMNN 51053 DRUGGABLE GENOME TCMDC-124576 CHEMBL579420 15730 10738 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650030 BUFOTENINE 15731 10739 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AMIODARONE AMIODARONE 22931300 15732 10740 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565739 AZD-6482 15733 10741 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE 5,8,11,14-EICOSATETRAYNOIC ACID CHEMBL458328 15734 10742 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME 4-AMINO-[1,2]NAPHTHOQUINONE 4-AMINO-[1,2]NAPHTHOQUINONE 15735 10743 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-35 15736 10744 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CYC-116 CYC-116 15737 10745 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE sufentanil SUFENTANIL 31773688 15740 10746 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PF-573228 27793840 15742 10747 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME LGD-1550 15744 10748 POLK 51426 DNA REPAIR, ENZYME TCMDC-123912 CHEMBL106525 15746 10749 F3 2152 DRUGGABLE GENOME, CELL SURFACE ALT-836 15747 10750 PANX1 24145 ION CHANNEL inhibitor 178100972 CARBENOXOLONE 15748 10751 IRS1 3667 KINASE, CLINICALLY ACTIONABLE fluorouracil FLUOROURACIL 15750 10752 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR BUTYRYLHYDROXAMIC ACID BUTYRYLHYDROXAMIC ACID 21874153 15751 10753 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE ATR KINASE INHIBITOR BAY1895344 15752 10754 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE FADROZOLE FADROZOLE 18256205 15753 10755 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME CENISERTIB CENISERTIB 15759 10756 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Sorafenib SORAFENIB 25900027 15760 10757 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE TAMATINIB R-406 15761 10758 MAPT 4137 DRUGGABLE GENOME AG-370 CHEMBL59150 15762 10759 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Talazoparib TALAZOPARIB 23881923 15763 10760 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL3039518 BATEFENTEROL 15764 10761 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER idarubicin IDARUBICIN 25558979,20938465,25567217,16331627 15766 10762 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NICLOSAMIDE NICLOSAMIDE 15767 10763 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RG7112 RO-5045337 26459177 15768 10764 ABCC9 10060 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER CHEMBL2105160 NAMINIDIL 15770 10765 UCP2 7351 TRANSPORTER, DRUGGABLE GENOME INTRALIPID SOYBEAN OIL 10868951 15772 10766 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR LYC-55716 15773 10767 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Cediranib CEDIRANIB 22238366,25589496 15775 10768 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE antibody MAPATUMUMAB MAPATUMUMAB 15778 10769 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3545006 PWT-33587 15779 10770 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-4 15780 10771 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR FENRETINIDE FENRETINIDE 15782 10772 MST1 4485 PROTEASE, KINASE, DRUGGABLE GENOME RETINOIC ACID 9886825 15784 10773 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL2107386 VORAPAXAR SULFATE 15785 10774 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME OLPRINONE OLPRINONE 15786 10775 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE VINCRISTINE SULFATE VINCRISTINE SULFATE 15788 10776 GABBR2 9568 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL301742 ARBACLOFEN 15789 10777 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME METHYLDOPA (RACEMIC) METHYLDOPA (RACEMIC) 15790 10778 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PALMITOYL-CARNITINE PALMITOYL-CARNITINE 15791 10779 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE Rinfabate RINFABATE 15792 10780 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX antagonist 135650003 15793 10781 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CHEMBL1257 ENFLURANE 15794 10782 MAOB 4129 DRUGGABLE GENOME, ENZYME Tranylcypromine TRANYLCYPROMINE 15796 10783 MPHOSPH8 54737 NA AMSACRINE HYDROCHLORIDE AMSACRINE HYDROCHLORIDE 15798 10784 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE QUININE ETHYLCARBONATE QUININE ETHYLCARBONATE 15799 10785 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER prednisone PREDNISONE 12175731,25637052 15805 10786 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1672627 LAS101057 15806 10787 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE ALZT-OP1 15807 10788 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OMEPRAZOLE OMEPRAZOLE 15808 10789 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL 1,2,4-triazole derivative 3 15809 10790 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME 681640 CHEMBL379975 15810 10791 CSK 1445 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor 223365983 RIVOCERANIB 15812 10792 SRP19 6728 NA paroxetine PAROXETINE 22795047 15814 10793 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-12 15815 10794 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE CHLOROTHIAZIDE CHLOROTHIAZIDE 15816 10795 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BAY-11-7085 BAY-11-7085 15817 10796 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor BGJ398 INFIGRATINIB 15818 10797 GMNN 51053 DRUGGABLE GENOME DNDI1417383 CHEMBL2094665 15820 10798 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Cyclophosphamide CYCLOPHOSPHAMIDE 15822 10799 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE SOLANEZUMAB SOLANEZUMAB 15824 10800 GHRL 51738 DRUGGABLE GENOME Unacylated ghrelin 15825 10801 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME AZD3293 LANABECESTAT 15826 10802 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METHYLDOPA METHYLDOPA 15827 10803 KDM1B 221656 DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING, ENZYME PMID27019002-Compound-48 15829 10804 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALLETHRIN ALLETHRIN 15832 10805 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-29 15833 10806 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CEDIRANIB CEDIRANIB 15834 10807 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM BROMIDE 15836 10808 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALITRETINOIN ALITRETINOIN 15837 10809 TMEM97 27346 NA Isoindoline derivative 3 15838 10810 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Denosumab DENOSUMAB 27322743 15839 10811 HSPA4 3308 NA KETANSERIN KETANSERIN 9864262 15841 10812 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HARMINE HARMINE 15842 10813 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1316 CARPROFEN 15843 10814 POR 5447 ENZYME, DRUGGABLE GENOME cyclosporine CYCLOSPORINE 29135906,24658827,24061445 15844 10815 ALOX15 246 ENZYME, DRUGGABLE GENOME DIPYRONE SODIUM DIPYRONE SODIUM 15845 10816 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-2272 CHEMBL601757 15846 10817 TARDBP 23435 TUMOR SUPPRESSOR TCMDC-124746 CHEMBL524407 15848 10818 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE Fostamatinib disodium 15849 10819 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR DAUNORUBICIN DAUNORUBICIN 22260166 15852 10820 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Oxazolyl methylthiothiazole derivative 1 15853 10821 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL AZIETOMIDATE AZIETOMIDATE 16884293 15854 10822 PMAIP1 5366 CLINICALLY ACTIONABLE BORTEZOMIB BORTEZOMIB 16024631 15855 10823 TOP2B 7155 DRUGGABLE GENOME, ENZYME RTA 744 15856 10824 GMNN 51053 DRUGGABLE GENOME GNF-PF-254 CHEMBL461579 15859 10825 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652004 15861 10826 RGS12 6002 DRUGGABLE GENOME SANGUINARIUM SANGUINARIUM 15862 10827 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME KALOPANAX-SAPONIN F METHYL ESTER CHEMBL1834951 21889336 15863 10828 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200968 HYDROCORTISONE SODIUM PHOSPHATE 15864 10829 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Debio 0932 15865 10830 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 2,6-DIMETHOXYQUINONE 2,6-DIMETHOXYQUINONE 15866 10831 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZM-449829 CHEMBL154580 15868 10832 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE RABEPRAZOLE RABEPRAZOLE 16815316 15869 10833 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ATOSIBAN ATOSIBAN 15870 10834 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist 310264689 CHEMBL201013 15871 10835 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Lapatinib LAPATINIB 20179222,27595477,18413839,27197158,27140927,26270481,27108243,22908275,24971884,22586653,27760111,26296355,18774637,27450453,27900369,23948973,27026198,23940356,24868024,26245675,19786658,22046346,23220880,25435280,26432108,26487584,25221644,27697991,26243863,25238247,26628478,26920887 15872 10836 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor 328083472 15873 10837 MAP2K6 5608 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE, TUMOR SUPPRESSOR inhibitor SELUMETINIB SELUMETINIB 15874 10838 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BN-DF-037 15875 10839 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651390 15877 10840 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NEFAZODONE HYDROCHLORIDE NEFAZODONE HYDROCHLORIDE 15878 10841 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE MK-1775 ADAVOSERTIB 27998224 15879 10842 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-L1 15880 10843 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1516 OLMESARTAN 15881 10844 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-138263 CHEMBL535307 15882 10845 CXCL8 3576 DRUGGABLE GENOME RETINAL RETINAL 15885 10846 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME ADINAZOLAM ADINAZOLAM 15888 10847 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1768 BETHANECHOL CHLORIDE 15889 10848 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 252827367 OZANIMOD 15890 10849 PSME3 10197 NA inhibitor BORTEZOMIB BORTEZOMIB 15891 10850 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Ryzodeq 15893 10851 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135650611 15894 10852 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651550 15896 10853 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE antibody 178103956 BLINATUMOMAB 15897 10854 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SEW-03621 CHEMBL1271059 15898 10855 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9422240, 1-282 15900 10856 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR captopril CAPTOPRIL 19286758 15901 10857 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Regorafenib REGORAFENIB 15902 10858 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Binimetinib BINIMETINIB 26544513 15903 10859 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200705 HYDROXYAMPHETAMINE HYDROBROMIDE 15904 10860 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ALSTERPAULLONE ALSTERPAULLONE 15905 10861 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 252827533 15907 10862 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ARISTOLACTONE ARISTOLACTONE 15908 10863 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME inhibitor 404859124 15909 10864 NGFR 4804 CELL SURFACE, DRUGGABLE GENOME CXB909 15910 10865 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CINOLAZEPAM CINOLAZEPAM 15911 10866 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER MURUCOIDIN V MURUCOIDIN V 22148475 15912 10867 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PROTOAPIGENONE PROTOAPIGENONE 15915 10868 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Valproate 15917 10869 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL452 CLONAZEPAM 15918 10870 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME LCAR-B38M CAR-T Cell 15919 10871 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL289351 FOSBRETABULIN DISODIUM 15920 10872 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051798 BELINOSTAT 15922 10873 BAZ2B 29994 NA TANSHINONE IIA TANSHINONE IIA 15923 10874 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 15924 10875 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure1-Aphanamixoid A 15925 10876 GMNN 51053 DRUGGABLE GENOME QUINAPRIL HYDROCHLORIDE QUINAPRIL HYDROCHLORIDE 15926 10877 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ERYTHROPOIETIN EPOETIN BETA 15816864 15927 10878 ATXN2 6311 NA LASALOCID A SODIUM LASALOCID A SODIUM 15929 10879 GLO1 2739 ENZYME, DRUGGABLE GENOME 2-(4-METHOXYBENZAMIDO)BENZOIC ACID CHEMBL1701911 21669529 15930 10880 GHRL 51738 DRUGGABLE GENOME RISPERIDONE RISPERIDONE 18480685 15933 10881 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NCX116 15935 10882 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ITRAZOLE ITRACONAZOLE 15936 10883 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME temozolomide TEMOZOLOMIDE 24444404 15938 10884 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GNF-PF-5411 CHEMBL15134 15940 10885 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PYRITHIONE ZINC PYRITHIONE ZINC 15941 10886 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE cisplatin CISPLATIN 21605004,29662106,27995989,20634689,19159907,19307503 15942 10887 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE DOVITINIB DOVITINIB 15943 10888 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-131 15946 10889 COQ2 27235 ENZYME atorvastatin ATORVASTATIN 20347093 15947 10890 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Lapatinib LAPATINIB 27595477 15948 10891 MAPT 4137 DRUGGABLE GENOME 3,4-DICHLOROISOCOUMARIN CHEMBL24983 15949 10892 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-MTC-427 15951 10893 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 1-HYDROXY-6-(4-HYDROXY-PHENYL)-1-PHENYL-HEXAN-3-ONE (ENANTIOMERIC MIX) 1-HYDROXY-6-(4-HYDROXY-PHENYL)-1-PHENYL-HEXAN-3-ONE (ENANTIOMERIC MIX) 20430632 15954 10894 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME ADM 10422567 15956 10895 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C16 15960 10896 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIDODECYL-DIMETHYL-AMMONIUM BROMIDE CHEMBL332670 15961 10897 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor SIROLIMUS SIROLIMUS 15962 10898 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 178101984 15963 10899 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 178103820 NEBIVOLOL 15965 10900 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PROGESTERONE PROGESTERONE 15966 10901 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 363894210 PANULISIB 15967 10902 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 135651284 TROPISETRON 15968 10903 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-30 15970 10904 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE WORTMANNIN WORTMANNIN 10318860,7559410,8955143 15971 10905 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME JUGLONE JUGLONE 15973 10906 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-K1 15976 10907 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ZIRAM ZIRAM 15977 10908 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (S)-FELODIPINE (S)-FELODIPINE 15978 10909 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE inhibitor 329968448 15979 10910 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135649939 AMITRIPTYLINE 15980 10911 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME VBY- 036 15981 10912 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ROTTLERIN ROTTLERIN 15982 10913 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650086 15984 10914 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TCMDC-124422 CHEMBL527620 15985 10915 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Avelumab AVELUMAB 15988 10916 ATAD5 79915 NA 8-PHENOXYCAFFEINE CHEMBL1529697 15989 10917 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE antibody 223366081 EMIBETUZUMAB 15990 10918 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER DIMETHYL SULFOXIDE 8762455 15991 10919 BAZ2B 29994 NA FLUMEQUINE FLUMEQUINE 15992 10920 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 5-FLUOROURIDINE CHEMBL54918 15993 10921 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NEBIVOLOL NEBIVOLOL 15995 10922 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PMID29671355-Compound-67 15996 10923 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE CHEMBL2109402 MM-121 15998 10924 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor TANDUTINIB TANDUTINIB 15999 10925 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NSC-9037 CHEMBL1451216 16000 10926 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2-MORPHOLINOETHYL 1-PHENYLCYCLOHEXANECARBOXYLATE CHEMBL305881 16001 10927 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565617 RIVICICLIB 16002 10928 BAG6 7917 NA carbamazepine CARBAMAZEPINE 16538176 16004 10929 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor LAPATINIB LAPATINIB 16005 10930 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE VERMISTATIN VERMISTATIN 22295871 16006 10931 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE EOSIN_Y EOSIN_Y 22889313 16008 10932 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1201099 CODEINE PHOSPHATE 16009 10933 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor EVEROLIMUS EVEROLIMUS 16011 10934 ATXN2 6311 NA TCMDC-123713 CHEMBL586135 16012 10935 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Gemcitabine GEMCITABINE 16014 10936 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME DNDI1417467 CHEMBL1997335 16016 10937 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE Brinzolamide BRINZOLAMIDE 16017 10938 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1237061 PITAVASTATIN CALCIUM 16018 10939 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME GSK2141795 UPROSERTIB 24265152 16020 10940 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SP-600125 SP-600125 16021 10941 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL blocker 178101137 16022 10942 HSPB2 3316 KINASE MTX METHOTREXATE 15519494 16023 10943 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME PMID27539678-Compound-13 16026 10944 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Tricyclic pyrrolopyridine compound 1 16027 10945 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MIANSERIN MIANSERIN 16028 10946 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200395 ORPHENADRINE CITRATE 16029 10947 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GARCINONE E GARCINONE E 16031 10948 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MAPROTILINE HYDROCHLORIDE MAPROTILINE HYDROCHLORIDE 16032 10949 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Roscovitine derivative 1 16034 10950 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR AZAKENPAULLONE AZAKENPAULLONE 16035 10951 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-25 16036 10952 SLC27A4 10999 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 252827468 16038 10953 POLK 51426 DNA REPAIR, ENZYME 4-AMINOPHENOL 4-AMINOPHENOL 16039 10954 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME INS-19 16040 10955 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 1245272 CHEMBL408850 16041 10956 BAZ2B 29994 NA E324 E324 16042 10957 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE PERIFOSINE PERIFOSINE 16043 10958 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GALLIC ACID METHYL ESTER GALLIC ACID METHYL ESTER 16044 10959 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXANDROLONE OXANDROLONE 16046 10960 ATXN2 6311 NA BW-723C86 CHEMBL1255834 16047 10961 GPT 2875 ENZYME PROTEASE INHIBITOR 9769871 16048 10962 PTGS1 5742 ENZYME, DRUGGABLE GENOME CURCUMIN PYRAZOLE CURCUMIN PYRAZOLE 24920381 16049 10963 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NITROXOLINE NITROXOLINE 16050 10964 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1611 PHENYTOIN SODIUM 16051 10965 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER GARDENIN GARDENIN 16052 10966 PTK6 5753 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, ENZYME inhibitor 315661136 16053 10967 KMO 8564 DRUGGABLE GENOME, ENZYME Cyclopropane 1-carboxylic acid derivative 2 16054 10968 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 6 16056 10969 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER 3-((2-PHENETHYLPHENOXY)METHYL)PYRIDINE CHEMBL217425 18257545 16057 10970 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CARBETAPENTANE CITRATE CARBETAPENTANE CITRATE 16058 10971 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE hydroxychloroquine HYDROXYCHLOROQUINE 18322994 16059 10972 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32r 16061 10973 CD276 80381 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME N/A 16062 10974 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL3545004 PL-225B 16063 10975 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL501 AMPHETAMINE SULFATE 16064 10976 BRCA2 675 CLINICALLY ACTIONABLE BMN673 16066 10977 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 363894181 16067 10978 FST 10468 DRUGGABLE GENOME TUMOR NECROSIS FACTOR 17436000 16068 10979 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PROPYLPARABEN PROPYLPARABEN 16071 10980 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-155 16073 10981 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE carbamazepine CARBAMAZEPINE 11294926 16074 10982 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-1654 CHEMBL602776 16076 10983 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Squalamine SQUALAMINE 16077 10984 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3545248 DS-7423 16078 10985 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (S)-3,5-DIHYDROXYPHENYLGLYCINE CHEMBL39221 16079 10986 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE Curcumin CURCUMIN 16081 10987 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-348401 CHEMBL515505 16082 10988 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE everolimus EVEROLIMUS 16083 10989 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor CHEMBL3544911 PREXASERTIB 16084 10990 MAOB 4129 DRUGGABLE GENOME, ENZYME EUGENOL EUGENOL 16085 10991 GLA 2717 ENZYME, DRUGGABLE GENOME migalastat MIGALASTAT 16087 10992 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME pitavastatin PITAVASTATIN 15159445,16595711,20175818,23007012 16088 10993 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BISPECIFIC ANTIBODY 11280736 16089 10994 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE PD-98059 CHEMBL35482 15613028 16091 10995 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 135650153 16092 10996 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-2559 CHEMBL583584 16095 10997 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE GNF-2 CHEMBL483847 16415863 16097 10998 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 328083484 16099 10999 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL967 TEMAZEPAM 16101 11000 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 252166827 16103 11001 APC 324 CLINICALLY ACTIONABLE Niclosamide NICLOSAMIDE 21531761 16104 11002 NUAK1 9891 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 315661259 16105 11003 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE atezolizumab ATEZOLIZUMAB 16106 11004 UCP2 7351 TRANSPORTER, DRUGGABLE GENOME BRL49653 9299560 16110 11005 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamide derivative 24 16112 11006 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE M3541 16113 11007 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-41 16114 11008 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FORMESTANE FORMESTANE 16115 11009 PLA2G7 7941 DRUGGABLE GENOME, ENZYME inhibitor 354702268 16117 11010 HEBP1 50865 DRUGGABLE GENOME Pyridyl compound 1 16119 11011 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GARDENIN GARDENIN 16121 11012 VSIR 64115 DRUGGABLE GENOME, CLINICALLY ACTIONABLE CA-170 16122 11013 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PI3K/BET INHIBITOR LY294002 26490311 16123 11014 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME ALN-TTRsc 16124 11015 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CEDIRANIB CEDIRANIB 16126 11016 EGR2 1959 TRANSCRIPTION FACTOR RETINOIC ACID 1361214 16128 11017 ATXN2 6311 NA ALPHA-SOLANINE CHEMBL1392894 16129 11018 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Decitabine DECITABINE 24077826 16130 11019 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545244 ALLITINIB 16131 11020 UGT2B7 7364 DRUGGABLE GENOME simvastatin SIMVASTATIN 16132 11021 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING SODIUM SELENITE SODIUM SELENITE 16133 11022 PTGS2 5743 DRUGGABLE GENOME, ENZYME Carbamate derivative 2 16135 11023 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-103 16136 11024 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor PAZOPANIB PAZOPANIB 16138 11025 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CAMPTOTHECIN CAMPTOTHECIN 24529870,19783447,15509164,20155916,22867019,24099994,25913198,20494586,25240093,25003995,21388138,22647222,26216018,21600681,21095131,23920485,21823606,22867097,20942490,26312433,11000035,19386396,24103429,23603616,23849207,25909279,25282261,25815139,23987476,24094433,19691293,22329436,19715319,1324981,23202849,25799376,17827007,20630766,25244612,9632354,25626146,23321564,22503207,17276690,24502276,25317694 16142 11026 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 374883848 16143 11027 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME MB-12066 LAPACHONE 16144 11028 KEAP1 9817 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor CHEMBL1762621 BARDOXOLONE METHYL 16145 11029 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR TUBERATOLIDE A TUBERATOLIDE A 21142112 16146 11030 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 178102429 16147 11031 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER NBI-98854 VALBENAZINE TOSYLATE 16148 11032 ADAM12 8038 NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178103981 ILOMASTAT 16150 11033 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME VU0080241 CHEMBL477396 16151 11034 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AZD9056 AZD9056 16152 11035 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HEXACHLOROPHENE HEXACHLOROPHENE 16153 11036 HTT 3064 DRUGGABLE GENOME NITROXOLINE NITROXOLINE 16154 11037 GAA 2548 DRUGGABLE GENOME, ENZYME TERAZOSIN HYDROCHLORIDE TERAZOSIN HYDROCHLORIDE 16156 11038 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE pravastatin PRAVASTATIN 17047488 16158 11039 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-92 16161 11040 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL628 PENTOXIFYLLINE 16162 11041 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR 2-METHOXYESTRADIOL 2-METHOXYESTRADIOL 18292194 16163 11042 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE GNF-PF-5159 CHEMBL1493528 16166 11043 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Rosiglitazone XR 16167 11044 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-254 CHEMBL461579 16168 11045 HMOX2 3163 ENZYME STANNSOPORFIN STANNSOPORFIN 16170 11046 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PHLORETIN PHLORETIN 16171 11047 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BENZOPHENONE BENZOPHENONE 16172 11048 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME activator CHEMBL266510 FLINDOKALNER 16173 11049 CD55 1604 DRUGGABLE GENOME, CELL SURFACE PD-98059 CHEMBL35482 11528371 16174 11050 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Vistusertib VISTUSERTIB 26359452 16175 11051 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME interferon beta-1a 27020477 16177 11052 MIA 8190 GROWTH FACTOR, DRUGGABLE GENOME TGFBETA1 16845326 16179 11053 IGF1 3479 GROWTH FACTOR, HORMONE ACTIVITY, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE inhibitor CHEMBL2109355 DUSIGITUMAB 16180 11054 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PH-011685 CHEMBL126804 16181 11055 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TRIPELENNAMINE TRIPELENNAMINE 16183 11056 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-67746 CHEMBL333177 16188 11057 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR URACIL URACIL 17076658 16189 11058 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BENSERAZIDE BENSERAZIDE 16190 11059 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051807 SCRIPTAID 16192 11060 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 4 16193 11061 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE IL-3 8910323 16194 11062 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SULINDAC SULINDAC 22931300 16195 11063 GSTT1 2952 DRUGGABLE GENOME BPDE 11731429,10607731 16197 11064 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 16198 11065 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL1200721 ESTRAMUSTINE PHOSPHATE SODIUM 16199 11066 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CL-329167 CL-329167 16200 11067 BMPR1A 657 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 252166689 16201 11068 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200974 CARBINOXAMINE MALEATE 16202 11069 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 249565617 RIVICICLIB 16203 11070 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ALCAFTADINE ALCAFTADINE 16204 11071 SLC25A5 292 DRUGGABLE GENOME, TRANSPORTER CLODRONATE CLODRONIC ACID 16205 11072 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL2110732 DACOMITINIB 16206 11073 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor 178101507 PENTOSTATIN 16207 11074 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PHENANTHROLINE PHENANTHROLINE 16208 11075 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR CHEMOKINES 15059845 16209 11076 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PSD-506 16210 11077 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CETUXIMAB CETUXIMAB 19001320,19603018,31566309,28363909,26989027,19571295,22281684,28972961,19603024,22180495,27729313,20619739,31515458 16212 11078 ATAD5 79915 NA 6-BROMOFLAVONE 6-BROMOFLAVONE 16214 11079 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SAPRISARTAN SAPRISARTAN 16215 11080 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME OSI-632 OSI-632 16216 11081 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL1094 FELBAMATE 16217 11082 SDC2 6383 CELL SURFACE, DRUGGABLE GENOME HEPARAN SULFATE 8642635 16218 11083 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR THIPHENAMIL THIPHENAMIL 16219 11084 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1201014 PREDNISOLONE SODIUM PHOSPHATE 16220 11085 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CR845 DIFELIKEFALIN 16221 11086 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BCG BCG VACCINE 17028812 16224 11087 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-4803 CHEMBL585240 16226 11088 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR sumatriptan SUMATRIPTAN 25096645 16227 11089 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR antagonist 223366043 16229 11090 RHOB 388 NA TRIMETHYL-[3-(TETRADECANE-1-SULFONYLAMINO)-PROPYL]-AMMONIUM IODIDE TRIMETHYL-[3-(TETRADECANE-1-SULFONYLAMINO)-PROPYL]-AMMONIUM IODIDE 24095759 16231 11091 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774822-Compound-Figure8Example5 16232 11092 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651314 16233 11093 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DINOTERB DINOTERB 16235 11094 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE N/A 16236 11095 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX PIROCTONE PIROCTONE 16237 11096 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-A1 16239 11097 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KINASE INHIBITOR 17307797 16240 11098 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE ISIS 113715 16241 11099 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LEVOTHYROXINE LEVOTHYROXINE 16242 11100 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE GM-CSF/IL-3 FUSION PROTEIN 1713254 16243 11101 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SB-220025 SB-220025 16245 11102 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor 178102591 16247 11103 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE MK-1903 16254 11104 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649988 BETHANECHOL 16255 11105 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SNS-314 SNS-314 16256 11106 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Tarafenacin TARAFENACIN 16257 11107 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE PREXASERTIB PREXASERTIB 28490518 16259 11108 BAZ2B 29994 NA SJ000032159 CHEMBL591361 16261 11109 KMT2C 58508 ENZYME, CLINICALLY ACTIONABLE, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, DRUG RESISTANCE EXEMESTANE EXEMESTANE 29755131 16264 11110 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL402548 DANUSERTIB 16266 11111 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER CISPLATIN CISPLATIN 9270026 16267 11112 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051804 RESMINOSTAT 16268 11113 HBB 3043 DRUGGABLE GENOME, ENZYME AZATHIOPRINE AZATHIOPRINE 16269 11114 RAB9A 9367 ENZYME, DRUGGABLE GENOME SU-4312 CHEMBL328710 16272 11115 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 363894209 PAMAPIMOD 16274 11116 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME E324 E324 16276 11117 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL563 FLURBIPROFEN 16278 11118 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 16280 11119 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ANTIDEPRESSANTS 12614997 16283 11120 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME bosentan BOSENTAN 17496208 16284 11121 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR US9006244, E1 16285 11122 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Panitumumab PANITUMUMAB 16286 11123 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME AMITRIPTYLINE AMITRIPTYLINE 16287 11124 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103875 TERAZOSIN 16289 11125 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-43 16290 11126 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-3323 CHEMBL1270169 16293 11127 POLK 51426 DNA REPAIR, ENZYME NSC-36398 CHEMBL483206 16294 11128 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR GANETESPIB GANETESPIB 16295 11129 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 223366147 ORANTINIB 16297 11130 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TOZASERTIB TOZASERTIB 16299 11131 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Imidazo bicyclic iminium derivative 2 16300 11132 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE BMS-754807 BMS-754807 19778024 16301 11133 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565869 CEP-11981 16302 11134 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 223366203 RONICICLIB 16303 11135 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Avrina 16304 11136 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 249565843 16305 11137 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 16306 11138 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DICYCLOHEXYLCARBODIIMIDE DICYCLOHEXYLCARBODIIMIDE 16307 11139 PDE3A 5139 ENZYME, DRUGGABLE GENOME Org-30029 16308 11140 RACGAP1 29127 NA BENZOTHIAZOLE-2,6-DIAMINE CHEMBL328540 16309 11141 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OLMESARTAN OLMESARTAN 16310 11142 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 315661135 16312 11143 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR 2-PYRIDYLCARBOXALDEHYDE P-BROMOBENZOYLHYDRAZONE CHEMBL400912 16313 11144 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PIPERIDINE-2,3-DICARBOXYLIC ACID CHEMBL431504 16314 11145 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR HORMONE THERAPY 24185512 16315 11146 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SULCONAZOLE NITRATE SULCONAZOLE NITRATE 16317 11147 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE SJ000196127 CHEMBL605084 16318 11148 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 26 16319 11149 IL18 3606 DRUGGABLE GENOME POLYPHENOL 16143535 16321 11150 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DEXAMETHASONE DEXAMETHASONE 7664296 16322 11151 TGFBR2 7048 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME agonist 178101755 16323 11152 HLA-DRB5 3127 DRUGGABLE GENOME, CLINICALLY ACTIONABLE 1D09C3 1D09C3 16324 11153 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-Figure6C 16325 11154 CA9 768 DRUGGABLE GENOME, ENZYME Girentuximab GIRENTUXIMAB 16326 11155 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 L-THREO-BENZYLOXY ASPARTATE CHEMBL79140 16327 11156 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CAMPTOTHECIN CAMPTOTHECIN 16329 11157 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR QUINPIROLE QUINPIROLE 16330 11158 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME DEXANABINOL DEXANABINOL 16331 11159 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1200825 METHADONE HYDROCHLORIDE 16332 11160 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE PD-194035 CHEMBL415893 10386941 16333 11161 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE agonist 135651492 GLYCINE 16335 11162 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME PALBOCICLIB PALBOCICLIB 16336 11163 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE inhibitor 178103112 16337 11164 PRMT5 10419 ENZYME, METHYL TRANSFERASE inhibitor 336446913 16340 11165 ERAP1 51752 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103847 TOSEDOSTAT 16344 11166 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ZAMIFENACIN ZAMIFENACIN 16347 11167 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL484785 CRISABOROLE 16348 11168 IL11 3589 DRUGGABLE GENOME, KINASE, GROWTH FACTOR 5-FLUOROURACIL FLUOROURACIL 1832057 16350 11169 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CARVEDILOL CARVEDILOL 16352 11170 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-45 16353 11171 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor 354702241 16354 11172 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1709 SERTRALINE HYDROCHLORIDE 16355 11173 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE JSM 6427 16356 11174 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME ENOXOLONE ENOXOLONE 24461294 16358 11175 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE RG-1530 RG-1530 16360 11176 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR IRETOL IRETOL 16363 11177 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-3996 CHEMBL584458 16365 11178 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PHENACYL CHLORIDE PHENACYL CHLORIDE 16366 11179 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 KHELLIN KHELLIN 16367 11180 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME CANDOXATRIL CANDOXATRIL 16368 11181 XRCC1 7515 CLINICALLY ACTIONABLE ALPHA-TOCOPHEROL VITAMIN E 12618330 16369 11182 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GSK2334470 CHEMBL1765740 28416483 16373 11183 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1691 BETAXOLOL HYDROCHLORIDE 16374 11184 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME ANASTROZOLE ANASTROZOLE 11983488 16375 11185 PDE4A 5141 DRUGGABLE GENOME, ENZYME ONO-6126 16376 11186 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE ivacaftor / lumacaftor 24973281,29126871,29451946,28606620,27298017,29327948,28325531,27334259 16377 11187 TARDBP 23435 TUMOR SUPPRESSOR NSC-95397 CHEMBL429095 16378 11188 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-3716 CHEMBL609606 16379 11189 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE N'-(2-HYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE SALINAZID 16380 11190 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE Cerdulatinib CERDULATINIB 16381 11191 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX NICOTINE NICOTINE 12111438,11979430 16382 11192 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME phenytoin PHENYTOIN 24915025 16383 11193 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE SORAFENIB SORAFENIB 16384 11194 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE FLUORODEOXYURIDINE FLOXURIDINE 17177846 16386 11195 KDM4A 9682 DRUGGABLE GENOME, ENZYME IMIDAZOLE-4-ACETIC ACID HCL CHEMBL1256325 16387 11196 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178101923 ACETAMINOPHEN 16390 11197 PPOX 5498 DRUGGABLE GENOME, ENZYME Aminolevulinic Acid Hydrochloride 16391 11198 PRMT6 55170 ENZYME, METHYL TRANSFERASE inhibitor 178103616 16393 11199 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BROMODICHLOROACETIC ACID BROMODICHLOROACETIC ACID 16394 11200 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL1201752 IXABEPILONE 16395 11201 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CHLORPROPAMIDE CHLORPROPAMIDE 22931300 16397 11202 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME VORINOSTAT VORINOSTAT 16398 11203 HMOX1 3162 ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE NEUROTROPHIC FACTOR 16298686 16399 11204 SULT2A1 6822 DRUGGABLE GENOME EMATE EMATE 16400 11205 SLC29A4 222962 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 252166690 16401 11206 GSTT1 2952 DRUGGABLE GENOME ERYTHROPOIETIN EPOETIN BETA 15595630 16402 11207 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PUROMYCIN PUROMYCIN 11866936 16403 11208 ALDH1A1 216 DRUGGABLE GENOME, ENZYME EUGENOL EUGENOL 16406 11209 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME carboplatin CARBOPLATIN 26194361 16407 11210 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Tricyclic isoxazoloquinazoline derivative 3 16408 11211 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-65 16409 11212 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME MINAPRINE MINAPRINE 16410 11213 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TORSEMIDE TORSEMIDE 22931300 16411 11214 MIA 8190 GROWTH FACTOR, DRUGGABLE GENOME TRP-1 15760338 16412 11215 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-124266 CHEMBL124006 16414 11216 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BRIMONIDINE BRIMONIDINE 16416 11217 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR RG7741 23594139 16417 11218 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TAMSULOSIN TAMSULOSIN 16419 11219 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ANTHRALIN ANTHRALIN 16420 11220 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER THIORIDAZINE HYDROCHLORIDE THIORIDAZINE HYDROCHLORIDE 16423 11221 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROPACHLOR PROPACHLOR 16424 11222 BAZ2B 29994 NA DNDI1417623 CHEMBL2002849 16426 11223 TUBB2B 347733 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 16427 11224 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GUANFACINE HYDROCHLORIDE GUANFACINE HYDROCHLORIDE 16429 11225 RAB9A 9367 ENZYME, DRUGGABLE GENOME SJ000150791 CHEMBL600572 16430 11226 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 223366204 COPANLISIB 16432 11227 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417905 CHEMBL1449731 16433 11228 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME JNJ-26483327 JNJ-26483327 16434 11229 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Crenezumab CRENEZUMAB 16436 11230 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DOXYCYCLINE DOXYCYCLINE 16437 11231 PRKAA2 5563 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME metformin METFORMIN 22722338 16439 11232 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CALCIMYCIN CALCIMYCIN 16440 11233 ATXN2 6311 NA NSC-693571 CHEMBL1287983 16441 11234 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 252827520 DUBERMATINIB 16442 11235 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME SIROLIMUS SIROLIMUS 16444 11236 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Dezocine DEZOCINE 16445 11237 ACKR3 57007 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135652600 16446 11238 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrazolopyridine derivative 3 16447 11239 PADI3 51702 ENZYME, DRUGGABLE GENOME inhibitor 252166884 16448 11240 SETD7 80854 ENZYME, METHYL TRANSFERASE SINEFUNGIN SINEFUNGIN 23981144 16449 11241 DHFR 1719 DRUGGABLE GENOME, ENZYME Leucovorin Calcium 16450 11242 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DEOXIEPINEPHRINE DEOXIEPINEPHRINE 16451 11243 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor PANOBINOSTAT PANOBINOSTAT 16453 11244 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Sym013 16454 11245 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE dimercaprol DIMERCAPROL 417891 16455 11246 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE SIROLIMUS SIROLIMUS 23171796 16456 11247 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-3792 CHEMBL582983 16459 11248 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME nicotine NICOTINE 19644963 16460 11249 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 16462 11250 AQP4 361 ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME TOPIRAMATE TOPIRAMATE 18572411 16463 11251 BCHE 590 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL636 RIVASTIGMINE 16465 11252 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TACRINE TACRINE 22931300 16466 11253 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR DNDI1417086 CHEMBL1224755 16467 11254 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 178102608 IC261 16470 11255 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE INS-117548 16472 11256 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 354702215 16476 11257 ATAD5 79915 NA NIFEDIPINE NIFEDIPINE 16477 11258 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME GTP-004 16480 11259 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Isoflavone derivative 1 16481 11260 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Imidazo[1,2-b]pyridazine derivative 3 16482 11261 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CINOLAZEPAM CINOLAZEPAM 16483 11262 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 178102327 PHA-665752 16485 11263 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE AZD-1152-HQPA AZD-1152-HQPA 16486 11264 DHFR 1719 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3244648 METHOTREXATE SODIUM 16488 11265 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL1237099 DOXACURIUM CHLORIDE 16489 11266 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PF-477736 PF-00477736 26140595 16490 11267 TNFSF10 8743 DRUGGABLE GENOME DA-3607 16491 11268 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME SB-220025 SB-220025 16492 11269 SMN2 6607 DRUGGABLE GENOME 2-PYRIDYLKETONE BENZOYL HYDRAZONE CHEMBL252151 16494 11270 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ILORASERTIB ILORASERTIB 16495 11271 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 135651882 16496 11272 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Pyrrolidine derivative 9 16497 11273 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME caffeine CAFFEINE 9334205,11525881,29344738 16498 11274 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME ELLAGIC ACID ELLAGIC ACID 16500 11275 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME GSK618334 16501 11276 TOLLIP 54472 KINASE acetylcysteine ACETYLCYSTEINE 16502 11277 COP1 64326 CLINICALLY ACTIONABLE, ENZYME Flecainide FLECAINIDE 16503 11278 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE FOLIC ACID 14608078 16507 11279 RAB9A 9367 ENZYME, DRUGGABLE GENOME DINALINE DINALINE 16509 11280 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 178102290 AT-7519 16511 11281 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME FLUDARABINE FLUDARABINE 12040435 16512 11282 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME vernakalant VERNAKALANT 16513 11283 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ONO-4053 16514 11284 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651289 16515 11285 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME HYDROCORTISONE HYDROCORTISONE 1712816 16516 11286 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY MK-8521 16517 11287 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PHENOTHIAZINE PHENOTHIAZINE 16518 11288 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CLOXYQUIN CLOXYQUIN 16519 11289 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ALFUZOSIN ALFUZOSIN 16520 11290 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Erdafitinib ERDAFITINIB 16522 11291 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GENISTEIN GENISTEIN 16526 11292 PDE5A 8654 ENZYME, DRUGGABLE GENOME UK-371800 CHEMBL460293 16527 11293 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE TELATINIB TELATINIB 16528 11294 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL24778 SILODOSIN 16530 11295 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR METHYLPREDNISOLONE METHYLPREDNISOLONE 16532 11296 PDE3A 5139 ENZYME, DRUGGABLE GENOME BEMORADAN BEMORADAN 16534 11297 MT1H 4496 NA GLUCOCORTICOID 11713267 16535 11298 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME HOMIDIUM BROMIDE HOMIDIUM BROMIDE 16539 11299 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE IL-9 9261146 16540 11300 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651731 16541 11301 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1702 ATOMOXETINE HYDROCHLORIDE 16543 11302 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 6 16544 11303 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 2-(P-HYDROXYBENZYL)PRODIGIOSIN CHEMBL578220 18922034 16545 11304 POLK 51426 DNA REPAIR, ENZYME ENOXOLONE ENOXOLONE 16547 11305 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor GIVINOSTAT GIVINOSTAT 16548 11306 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 223365981 FALNIDAMOL 16549 11307 ATXN2 6311 NA SJ000160630 CHEMBL591404 16552 11308 ATXN2 6311 NA (E)-DIBENZYLIDENEACETONE CHEMBL17201 16553 11309 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652254 16555 11310 POLI 11201 DNA REPAIR LORNOXICAM LORNOXICAM 16556 11311 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 363894199 16557 11312 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 3 16559 11313 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MICONAZOLE NITRATE MICONAZOLE NITRATE 16560 11314 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 363894217 VORUCICLIB 16561 11315 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE RALOXIFENE RALOXIFENE 14533013 16565 11316 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Imatinib IMATINIB 16566 11317 COP1 64326 CLINICALLY ACTIONABLE, ENZYME Procainamide PROCAINAMIDE 16569 11318 TK1 7083 ENZYME, KINASE, DRUGGABLE GENOME Radiosensitizer gene therapy 16570 11319 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CYTOKINES 11839503 16571 11320 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLAVONE FLAVONE 16572 11321 PDE10A 10846 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL628 PENTOXIFYLLINE 16573 11322 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME ondansetron ONDANSETRON 21247998 16575 11323 TAC1 6863 DRUGGABLE GENOME GOSSYPOL GOSSYPOL 2887120 16577 11324 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 178103534 TAZAROTENE 16578 11325 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200334 MORICIZINE HYDROCHLORIDE 16580 11326 NT5C 30833 ENZYME lamivudine LAMIVUDINE 16582 11327 ATF2 1386 TRANSCRIPTION FACTOR GLUCOCORTICOID 17525285 16583 11328 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 329968432 16584 11329 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649910 16585 11330 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AZATHIOPRINE AZATHIOPRINE 22931300 16586 11331 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 178102554 16588 11332 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PHENOXYBENZAMINE HYDROCHLORIDE PHENOXYBENZAMINE HYDROCHLORIDE 16590 11333 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME OLEIC ACID OLEIC ACID 16591 11334 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME pitavastatin PITAVASTATIN 27839692 16592 11335 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE antibody TRASTUZUMAB TRASTUZUMAB 16593 11336 DNER 92737 NA Tetra-hydro-quinoline derivative 3 16594 11337 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL3545349 EVT-101 16595 11338 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MRL24 16597 11339 NOS1 4842 DRUGGABLE GENOME, ENZYME MUSTARD 8917686 16598 11340 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE antisense oligonucleotide OBLIMERSON 16599 11341 GSTM1 2944 DRUGGABLE GENOME, ENZYME busulfan BUSULFAN 23677058 16601 11342 TUBB4B 10383 DRUGGABLE GENOME MEBENDAZOLE MEBENDAZOLE 16602 11343 FAAH 2166 ENZYME, DRUGGABLE GENOME Ketoheterocycle derivative 4 16604 11344 HPRT1 3251 DRUGGABLE GENOME, ENZYME Mycophenolic Acid 16606 11345 MAPT 4137 DRUGGABLE GENOME AROMATICIN AROMATICIN 16607 11346 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ISOPROTERENOL ISOPROTERENOL 16608 11347 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Paclitaxel PACLITAXEL 22784709 16609 11348 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME celecoxib CELECOXIB 22336956 16612 11349 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-3641 CHEMBL599098 16614 11350 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL OCINAPLON OCINAPLON 16615 11351 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200449 TRIAMCINOLONE DIACETATE 16616 11352 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SULFASALAZINE SULFASALAZINE 16619 11353 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME DS-7423 DS-7423 16620 11354 ALOX15 246 ENZYME, DRUGGABLE GENOME LANSOPRAZOLE LANSOPRAZOLE 16621 11355 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE HPP-851 16624 11356 GJA1 2697 ION CHANNEL BLEOMYCIN BLEOMYCIN 16600115 16625 11357 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE BMS-387032 BMS-387032 16627 11358 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME Imatinib IMATINIB 16629 11359 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE FP-1039 FP-1039 16632 11360 TOP1MT 116447 DRUGGABLE GENOME, ENZYME LE-SN38 16633 11361 TUBA1B 10376 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 16635 11362 PSMD12 5718 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 16636 11363 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1200900 16637 11364 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR IMIPENEM CILASTATIN SODIUM 7933537 16638 11365 PLD1 5337 ENZYME, DRUGGABLE GENOME US9127005, P2B 16639 11366 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 3-oxo-2,3-dihydro-1H-indazole-4-carboxamide derivative 5 16641 11367 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650785 OXYMETAZOLINE 16642 11368 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE THUNBERGINOL E THUNBERGINOL E 16643 11369 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 887167 CHEMBL260342 16644 11370 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 repaglinide REPAGLINIDE 16647 11371 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME CID 94381 CHEMBL374632 16648 11372 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TCMDC-124317 CHEMBL586937 16650 11373 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL603469 LESTAURTINIB 16651 11374 TOP2B 7155 DRUGGABLE GENOME, ENZYME DOXORUBICIN DOXORUBICIN 16653 11375 ADAMTS1 9510 ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE inhibitor 252166863 16654 11376 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR DHEA PRASTERONE 15501480 16656 11377 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1889140 ROPIVACAINE HYDROCHLORIDE 16657 11378 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Trilaciclib TRILACICLIB 16660 11379 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HAPLAMINE HAPLAMINE 16662 11380 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-747270 CHEMBL594772 16663 11381 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 252827524 16664 11382 ALPL 249 ENZYME, DRUGGABLE GENOME Levamisole LEVAMISOLE 16666 11383 GUCY2C 2984 DRUGGABLE GENOME, KINASE agonist 374883898 DOLCANATIDE 16667 11384 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME BAICALEIN BAICALEIN 16668 11385 PSMA8 143471 DRUGGABLE GENOME, PROTEASE BORTEZOMIB BORTEZOMIB 24524217 16669 11386 GMNN 51053 DRUGGABLE GENOME NIFEDIPINE NIFEDIPINE 16670 11387 HMGCR 3156 ENZYME, DRUGGABLE GENOME Teriflunomide TERIFLUNOMIDE 16672 11388 XRCC1 7515 CLINICALLY ACTIONABLE PLATINUM PLATINUM 17925548 16673 11389 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 252166576 ITACITINIB 16675 11390 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME 4-(4-AMINOPHENYL)BUTANOIC ACID CHEMBL1650245 24044874 16677 11391 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER IODOACETAMIDE IODOACETAMIDE 16678 11392 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 16679 11393 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PONATINIB PONATINIB 23190221,24236021,25349473 16682 11394 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000029259 CHEMBL592558 16683 11395 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 381118805 16685 11396 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR KEPONE KEPONE 16687 11397 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1684984 PA-799 16688 11398 SLC9A3 6550 DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE, EXCHANGER AZD1722 16690 11399 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE BB 0223767 16691 11400 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL blocker 135652708 PICROTOXININ 16693 11401 GNA11 2767 CLINICALLY ACTIONABLE CGM097 CGM-097 27507190 16694 11402 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-31 16695 11403 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR CETUXIMAB CETUXIMAB 26644315 16697 11404 PRKAB1 5564 ENZYME, KINASE, DRUGGABLE GENOME METFORMIN METFORMIN 16699 11405 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PROTRIPTYLINE PROTRIPTYLINE 16700 11406 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL274654 ORANTINIB 16702 11407 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE JNJ-7706621 JNJ-7706621 16703 11408 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 doxepin DOXEPIN 12360109 16704 11409 PTGS2 5743 DRUGGABLE GENOME, ENZYME SULFASALAZINE SULFASALAZINE 16706 11410 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR CARBOPLATIN CARBOPLATIN 12499281 16707 11411 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-317605 CHEMBL1312050 16710 11412 TDO2 6999 ENZYME, DRUGGABLE GENOME PMID29473428-Compound-76 16711 11413 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE HEXACHLOROPHENE HEXACHLOROPHENE 16712 11414 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR BDBM50158794 16714 11415 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE LAPATINIB LAPATINIB 25691057,21840482 16715 11416 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GS 6201 GS 6201 16716 11417 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 252827414 16717 11418 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL2103852 CROLIBULIN 16719 11419 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649710 16722 11420 TYMP 1890 GROWTH FACTOR, DRUGGABLE GENOME fluorouracil FLUOROURACIL 24167597 16723 11421 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME morphine MORPHINE 19523031,8351162,17986163 16724 11422 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL970 HALAZEPAM 16725 11423 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CCT241161 25500121,15294323,17210691 16726 11424 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Gallamine Triethiodide 16727 11425 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME MIFEPRISTONE MIFEPRISTONE 9052414 16728 11426 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUDIOXONIL FLUDIOXONIL 16729 11427 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Crystalline anhydrous toluene derivative 1 16730 11428 SRP19 6728 NA citalopram CITALOPRAM 22795047 16735 11429 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ABT-737 ABT 737 21468686 16737 11430 KDM4A 9682 DRUGGABLE GENOME, ENZYME METHACYCLINE HYDROCHLORIDE METHACYCLINE HYDROCHLORIDE 16738 11431 BAZ2B 29994 NA DNDI1417055 CHEMBL1486366 16739 11432 GMNN 51053 DRUGGABLE GENOME ESTRADIOL BENZOATE ESTRADIOL BENZOATE 16741 11433 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE docetaxel DOCETAXEL 21636554 16743 11434 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 135649967 ASOPRISNIL 16744 11435 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL112 ACETAMINOPHEN 16745 11436 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING NSC-155693 CHEMBL68096 16746 11437 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor 315661124 ERDAFITINIB 16747 11438 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DIHYDROERGOTAMINE DIHYDROERGOTAMINE 16748 11439 EYA2 2139 DNA REPAIR IMATINIB IMATINIB 16749 11440 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME DELAVIRDINE DELAVIRDINE 21189339 16750 11441 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PMID29671355-Compound-25 16752 11442 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE SORAFENIB SORAFENIB 16755 11443 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BICALUTAMIDE BICALUTAMIDE 20381361,23017882,21050768,22175694 16756 11444 HTT 3064 DRUGGABLE GENOME Tractinostat 16757 11445 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PAPAVERINE PAPAVERINE 16761 11446 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102715 16762 11447 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Thioureidobutyronitrile 4-ISOTHIOUREIDOBUTYRONITRILE 16763 11448 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US8524917, 10 16765 11449 H19 283120 CLINICALLY ACTIONABLE Platinum compounds 26729200 16766 11450 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 249565654 XL-019 16768 11451 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ERGOCRYPTINE ERGOCRYPTINE 16770 11452 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TAXIFOLIN TAXIFOLIN 16772 11453 PTGS1 5742 ENZYME, DRUGGABLE GENOME Balsalazide BALSALAZIDE 16773 11454 PPP2R5D 5528 PROTEIN PHOSPHATASE, ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 16774 11455 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565590 CHEMBL1236539 16775 11456 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201563 INTERFERON BETA-1B 16776 11457 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PAZOPANIB PAZOPANIB 16778 11458 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1118 DESVENLAFAXINE 16779 11459 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Cyclic cyanoethypypazole derivative 1 16781 11460 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME partial agonist CHEMBL3545230 APIMOSTINEL 16784 11461 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2107803 AVOSENTAN 16785 11462 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE FASUDIL FASUDIL 16786 11463 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PANOBINOSTAT PANOBINOSTAT 16787 11464 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AG-527 CHEMBL258767 16791 11465 PSMB7 5695 DRUGGABLE GENOME, PROTEASE inhibitor CARFILZOMIB CARFILZOMIB 16792 11466 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR 17-BETA ESTRADIOL 16793 11467 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist CHEMBL547 ISOTRETINOIN 16794 11468 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME GEFITINIB GEFITINIB 16988945 16795 11469 SLC39A8 64116 TRANSPORTER ethanol ALCOHOL 32451486 16798 11470 DPEP1 1800 PROTEASE, DRUGGABLE GENOME, ENZYME CILASTATIN CILASTATIN 16799 11471 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Sitagliptin SITAGLIPTIN 16800 11472 SMN1 6606 DRUGGABLE GENOME METHYL ROBUSTONE METHYL ROBUSTONE 16801 11473 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CINOLAZEPAM CINOLAZEPAM 16803 11474 CFLAR 8837 DRUG RESISTANCE, DRUGGABLE GENOME, PROTEASE DEHYDROEQUOL IDRONOXIL 16805 11475 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BMS-182874 BMS-182874 16807 11476 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR palonosetron PALONOSETRON 29177570 16808 11477 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DAUNORUBICIN DAUNORUBICIN 16809 11478 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BAZEDOXIFENE ACETATE BAZEDOXIFENE ACETATE 16810 11479 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE RETEPLASE RETEPLASE 16811 11480 CBX1 10951 NA TCMDC-124518 CHEMBL527584 16812 11481 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BW-28C51 CHEMBL140020 16814 11482 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CANNABINOL CANNABINOL 16815 11483 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE CO-TRIMOXAZOLE CO-TRIMOXAZOLE 46571 16816 11484 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME imatinib IMATINIB 24123600,30713339,18981009,24322003 16817 11485 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL738 THIOPENTAL SODIUM 16819 11486 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TOXYLOXANTHONE C TOXYLOXANTHONE C 16820 11487 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME HTS-05058 CHEMBL261692 16823 11488 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME KERACYANIN KERACYANIN 17360708 16826 11489 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE Interferon Alfa-2b, Recombinant 16827 11490 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2364612 LATANOPROSTENE BUNOD 16828 11491 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CHLORDANE CHLORDANE 16830 11492 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CROCIN CROCIN 16833 11493 KIF11 3832 DRUGGABLE GENOME ARQ-621 16836 11494 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-135810 CHEMBL1605629 16837 11495 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME PMID27774824-Compound-Figure11Example1up 16838 11496 KDM4A 9682 DRUGGABLE GENOME, ENZYME HEXACHLOROPHENE HEXACHLOROPHENE 16840 11497 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-L3 16841 11498 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME RG-1530 RG-1530 16842 11499 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE Vitamin B-complex, Incl. Combinations 27035272,27520898,31058543 16847 11500 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650520 BEXAROTENE 16848 11501 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME PMA 8503863 16849 11502 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE EMD-1204831 EMD-1204831 16851 11503 GMNN 51053 DRUGGABLE GENOME BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE 16852 11504 POLB 5423 DNA REPAIR, DRUGGABLE GENOME EMODIN EMODIN 16854 11505 TSPO 706 DRUGGABLE GENOME CLORAZEPATE CLORAZEPIC ACID 16855 11506 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135650656 16856 11507 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME ISOSILYBIN B ISOSILYBIN B 23401473 16858 11508 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 384403641 RG-1530 16859 11509 CTH 1491 ENZYME inhibitor 178101828 16860 11510 MPI 4351 ENZYME, DRUGGABLE GENOME EBSELEN EBSELEN 16861 11511 POLK 51426 DNA REPAIR, ENZYME CEFIXIME CEFIXIME 16862 11512 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545245 BAY-1082439 16863 11513 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor TRAMETINIB TRAMETINIB 16864 11514 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1201759 BEPOTASTINE BESYLATE 16865 11515 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE inhibitor 252166826 16866 11516 NDUFAF1 51103 NA inhibitor CHEMBL3545135 NV-128 16867 11517 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PRN1371 16870 11518 GMNN 51053 DRUGGABLE GENOME DIPYRIDAMOLE DIPYRIDAMOLE 16871 11519 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SKF-83959 CHEMBL520992 16872 11520 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME RHENIUM-186 HYDROXYETHYLIDENE DIPHOSPHONATE 12087455 16873 11521 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR SOTRASTAURIN SOTRASTAURIN 16874 11522 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE CID 94381 CHEMBL374632 16875 11523 ALOX15B 247 DRUGGABLE GENOME, ENZYME DIHYDROXIDINE DIHYDROXIDINE 16876 11524 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Sumatriptan SUMATRIPTAN 16878 11525 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL MIDAZOLAM MIDAZOLAM 16881 11526 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor DASATINIB DASATINIB 16882 11527 SHMT1 6470 ENZYME methotrexate METHOTREXATE 20386493,18322994,15797993,22838948,18368069 16883 11528 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE INTERFERON GAMMA 7559588 16885 11529 BRCA2 675 CLINICALLY ACTIONABLE rucaparib RUCAPARIB 16886 11530 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE Lidocaine LIDOCAINE 16888 11531 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor 348353679 16890 11532 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE TG100-115 TG100-115 17685602 16891 11533 ATXN2 6311 NA BAS03450373 CHEMBL1576310 16892 11534 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME METHACYCLINE HYDROCHLORIDE METHACYCLINE HYDROCHLORIDE 16893 11535 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2219421 RECILISIB 16894 11536 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME GARLIC GARLIC 12125104 16896 11537 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY ALL-TRANS-RETINOIC ACID 10946899 16897 11538 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME GOSSYPOL GOSSYPOL 19555126 16898 11539 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME BDBM50173330 16900 11540 ABAT 18 DRUGGABLE GENOME, ENZYME Pyridoxal Phosphate 16902 11541 PADI3 51702 ENZYME, DRUGGABLE GENOME inhibitor 252166885 16903 11542 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME ALISERTIB ALISERTIB 16904 11543 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 178103458 VORINOSTAT 16905 11544 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR INDOLE-3-BUTYRIC ACID INDOLE-3-BUTYRIC ACID 16906 11545 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 16907 11546 MAPT 4137 DRUGGABLE GENOME MANGOSTIN MANGOSTIN 16909 11547 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME MEDRYSONE MEDRYSONE 16910 11548 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Olcegepant OLCEGEPANT 16911 11549 TNFRSF18 8784 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME 178101765 16912 11550 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Mafenide MAFENIDE 16914 11551 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist 135651455 16915 11552 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR RALOXIFENE RALOXIFENE 20659801 16916 11553 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 385612218 16917 11554 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY PB-1023 16918 11555 DHCR7 1717 ENZYME, DRUGGABLE GENOME cholic acid 16919 11556 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-49 16920 11557 BAZ2B 29994 NA NSC-353263 CHEMBL1383812 16921 11558 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1201468 ESTROGENS, ESTERIFIED 16922 11559 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME GSK-1004723 GSK-1004723 16923 11560 ALDH3A1 218 DRUGGABLE GENOME, ENZYME fluorouracil FLUOROURACIL 16924 11561 BAZ2B 29994 NA SJ000117451 CHEMBL592123 16926 11562 PSMD3 5709 NA inhibitor CHEMBL451887 CARFILZOMIB 16927 11563 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 381118852 16928 11564 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL2109460 SCH-708980 16931 11565 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CID 4101591 CHEMBL428789 16932 11566 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CLOFENOXYDE CLOFENOXYDE 16934 11567 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Radiotherapy 25589492 16935 11568 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 178103556 16936 11569 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME WORTMANNIN WORTMANNIN 10464177 16937 11570 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor HESPERADIN HESPERADIN 19035792 16938 11571 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650989 16939 11572 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 328083520 ESFLURBIPROFEN 16940 11573 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Benzamide derivative 7 16943 11574 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2016054807Example1 16945 11575 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME DU-176b EDOXABAN TOSYLATE 16946 11576 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE VANDETANIB VANDETANIB 16947 11577 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CAPECITABINE CAPECITABINE 19571295,22180495 16949 11578 ALOX15 246 ENZYME, DRUGGABLE GENOME GBR-12935 CHEMBL26320 16951 11579 BCL2A1 597 DRUGGABLE GENOME Apogossypolone 16953 11580 MAPT 4137 DRUGGABLE GENOME 2,5-BIS(4-MORPHOLINOSTYRYL)PYRAZINE CHEMBL2181041 22913544 16954 11581 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CASODEX CASODEX 15754350 16955 11582 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR BAS 02077837 CHEMBL1485809 16956 11583 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CATECHIN CATECHIN 16957 11584 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME DOVITINIB DOVITINIB 16958 11585 UBE2N 7334 ENZYME, DRUGGABLE GENOME HYDROXYSTILBAMIDINE ISETHIONATE HYDROXYSTILBAMIDINE ISETHIONATE 16959 11586 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PARBENDAZOLE PARBENDAZOLE 16961 11587 CAMK1D 57118 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME losartan LOSARTAN 25410890 16962 11588 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME 5,6,7-TRIBROMOISATIN CHEMBL376616 17088067 16963 11589 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4864 CHEMBL583558 16965 11590 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-106547 CHEMBL223575 16967 11591 EEF2 1938 DRUGGABLE GENOME, KINASE inhibitor CHEMBL1201550 DENILEUKIN DIFTITOX 16968 11592 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CICLOSPORIN CYCLOSPORINE 12673034 16969 11593 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Mirabegron MIRABEGRON 16970 11594 FGB 2244 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, FIBRINOGEN, DRUGGABLE GENOME HAEMATOXYLIN HAEMATOXYLIN 16971 11595 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DNDI1417413 CHEMBL1343568 16972 11596 TXNRD1 7296 DRUGGABLE GENOME Golden phosphorous acetyletic compound 2 16976 11597 TGFA 7039 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME panitumumab PANITUMUMAB 16978 11598 KDM4A 9682 DRUGGABLE GENOME, ENZYME DOPAMINE HYDROCHLORIDE DOPAMINE HYDROCHLORIDE 16980 11599 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ILORASERTIB ILORASERTIB 16981 11600 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-663284 CHEMBL337173 16983 11601 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE NSAID 10025882 16984 11602 GAPDH 2597 DRUGGABLE GENOME, ENZYME NSC-119911 CHEMBL502775 16985 11603 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-Fomula2 16987 11604 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CRIZOTINIB CRIZOTINIB 12460923,9826708,1104268,17483355,25157968,10417759,11750879 16988 11605 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME Diaryl amine derivative 4 16990 11606 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL TEMAZEPAM TEMAZEPAM 16991 11607 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ALVIMOPAN ALVIMOPAN 16992 11608 ATAD5 79915 NA N6-PHENYLADENOSINE N6-PHENYLADENOSINE 16993 11609 ALOX5 240 DRUGGABLE GENOME, ENZYME FPL-62064 16994 11610 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125784 CHEMBL581574 16996 11611 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure1-Sarcaboside B 16997 11612 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Lapatinib LAPATINIB 16999 11613 MAPT 4137 DRUGGABLE GENOME OXOGLAUCINE OXOGLAUCINE 17000 11614 PTGS2 5743 DRUGGABLE GENOME, ENZYME Ketoprofen KETOPROFEN 17001 11615 EYA2 2139 DNA REPAIR SJ000114740 CHEMBL592068 17003 11616 CDH1 999 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Erlotinib ERLOTINIB 26251290 17005 11617 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RIMSULFURON RIMSULFURON 17006 11618 TUBA1C 84790 DRUGGABLE GENOME CHEMBL2103826 DAVUNETIDE 17007 11619 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR AT-406 AT-406 25520882 17008 11620 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR TYROSINE KINASE INHIBITORS 15289348 17009 11621 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER INGENOL MEBUTATE 17014 11622 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 315661328 17016 11623 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME modafinil MODAFINIL 17018 11624 HTT 3064 DRUGGABLE GENOME CS-00028 17019 11625 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR TOZASERTIB TOZASERTIB 17021 11626 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRICHLORFON TRICHLORFON 17022 11627 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE GNF-PF-4068 CHEMBL584668 17027 11628 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 363894210 PANULISIB 17029 11629 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178103795 MEPERIDINE 17031 11630 SMN1 6606 DRUGGABLE GENOME 7,3'-DIMETHOXYFLAVONE 7,3'-DIMETHOXYFLAVONE 17033 11631 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2218917 CEVIMELINE HYDROCHLORIDE 17034 11632 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Benzene sulfonamide derivative 9 17035 11633 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PU-AD 17037 11634 TUBA4A 7277 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 17038 11635 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE E-10030 PEGPLERANIB SODIUM 17040 11636 KDM5C 8242 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 310264759 17041 11637 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649751 17044 11638 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME MILTIRONE MILTIRONE 26339922 17045 11639 PTGS1 5742 ENZYME, DRUGGABLE GENOME BROMFENAC BROMFENAC 17046 11640 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 375973265 17047 11641 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE METHIMAZOLE METHIMAZOLE 8491516 17049 11642 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME LCAR-B4822M CAR-T Cell 17051 11643 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME L-744,832 9515813 17052 11644 ABCB4 5244 TRANSPORTER, DRUGGABLE GENOME, ENZYME, ABC TRANSPORTER VINBLASTINE VINBLASTINE 7918493 17053 11645 CYBA 1535 TRANSPORTER simvastatin SIMVASTATIN 15936011 17057 11646 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME lusutrombopag LUSUTROMBOPAG 17061 11647 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME NVP-BSK805 27075627,22271575 17062 11648 CXCL2 2920 DRUGGABLE GENOME IL-13 16439363 17063 11649 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649955 17066 11650 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR palbociclib PALBOCICLIB 17067 11651 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 252166789 17068 11652 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565823 17069 11653 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHR-3996 NANATINOSTAT 17070 11654 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DYCLONINE DYCLONINE 17071 11655 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME DOXORUBICIN DOXORUBICIN 16211302 17072 11656 MAPT 4137 DRUGGABLE GENOME TANSHINONE IIA TANSHINONE IIA 17076 11657 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651880 RELAXIN 17079 11658 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME HISPIDIN HISPIDIN 17081 11659 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Enzoxazolinone sulfonamide derivative 1 17082 11660 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PF-562271 PF-00562271 17083 11661 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME CP-101,606 17084 11662 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR MGCD-0103 MOCETINOSTAT 17085 11663 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200495 HYDROCORTISONE SODIUM SUCCINATE 17088 11664 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR E-GUGGULSTERONE E-GUGGULSTERONE 17090 11665 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME CARBARIL CARBARIL 17091 11666 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Reolysin PELAREOREP 26156229,24798549 17092 11667 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652008 17097 11668 PTGS1 5742 ENZYME, DRUGGABLE GENOME ThermoProfen 17098 11669 KDM4A 9682 DRUGGABLE GENOME, ENZYME PHYSODIC ACID PHYSODIC ACID 17102 11670 GAA 2548 DRUGGABLE GENOME, ENZYME BENZAMIL BENZAMIL 17104 11671 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MELPHALAN MELPHALAN 17105 11672 ESRRG 2104 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135649823 17107 11673 RGS4 5999 DRUGGABLE GENOME EBSELEN EBSELEN 17109 11674 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL3545158 PEXIDARTINIB 17110 11675 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE BMS-754807 BMS-754807 17111 11676 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 17112 11677 COL2A1 1280 DRUGGABLE GENOME COLLAGENASE COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 17113 11678 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PRAVASTATIN PRAVASTATIN 15616150 17115 11679 ATXN2 6311 NA SJ000294102 CHEMBL607309 17116 11680 PFKFB3 5209 ENZYME, KINASE inhibitor 381118835 17117 11681 RGS4 5999 DRUGGABLE GENOME LUZINDOLE LUZINDOLE 17118 11682 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME 3-phenyl isoquinolin-1(2H) derivative 1 17119 11683 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING BELINOSTAT BELINOSTAT 17120 11684 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ZM-336372 CHEMBL186526 17122 11685 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 11 17123 11686 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR AVOBENZONE AVOBENZONE 17124 11687 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLOROTHALONIL CHLOROTHALONIL 17125 11688 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 178103520 17128 11689 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE GLPG0187 GLPG-0187 17129 11690 ALOX15B 247 DRUGGABLE GENOME, ENZYME PSEUDOEPHEDRINE PSEUDOEPHEDRINE 17131 11691 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE chlorpheniramine CHLORPHENIRAMINE 18695978 17132 11692 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 tolterodine TOLTERODINE 17134 11693 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor REGORAFENIB REGORAFENIB 17135 11694 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL FELODIPINE FELODIPINE 17136 11695 MPHOSPH8 54737 NA LEVODOPA LEVODOPA 17137 11696 TUBA1B 10376 DRUGGABLE GENOME CHEMBL2105643 FOSBRETABULIN TROMETHAMINE 17139 11697 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE NAX014 26168818 17140 11698 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME AG-1879 CHEMBL406845 19447617,16509573 17144 11699 PLOD1 5351 ENZYME, DRUGGABLE GENOME Ascorbate 17145 11700 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME COLCHICINE COLCHICINE 22931300 17146 11701 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 385612234 17147 11702 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME CEFOTAXIME SODIUM CEFOTAXIME SODIUM 17150 11703 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME Warfarin WARFARIN 17151 11704 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME RU-24969 RU-24969 17152 11705 KDM1A 23028 DRUGGABLE GENOME, ENZYME, CELL SURFACE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING 2-[N-(PHTHALIMIDO)]ETHYL CARBAMIMIDOTHIOATE HCL CHEMBL2182009 22876979 17153 11706 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE blocker CHEMBL3545169 AZD1305 17154 11707 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist 315661198 17157 11708 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ZIRAM ZIRAM 17159 11709 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE simvastatin SIMVASTATIN 25493567 17160 11710 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EMETINE DIHYDROCHLORIDE EMETINE HYDROCHLORIDE 17164 11711 GAA 2548 DRUGGABLE GENOME, ENZYME APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 17165 11712 PMP22 5376 DRUGGABLE GENOME, TRANSPORTER PROGESTERONE PROGESTERONE 9751213 17166 11713 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE FLUOROURACIL FLUOROURACIL 12237773 17169 11714 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-11 17170 11715 PTGS2 5743 DRUGGABLE GENOME, ENZYME Phenylbutazone PHENYLBUTAZONE 17171 11716 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist CHEMBL3545210 SR16234 17173 11717 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565629 SOTRASTAURIN 17174 11718 BMPR1A 657 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 249565800 17175 11719 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL608533 MIDOSTAURIN 17177 11720 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME MIV-701 17179 11721 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME FELBAMATE FELBAMATE 17181 11722 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 187051762 GLYCOPYRROLATE 17184 11723 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PHENOLPHTHALEIN PHENOLPHTHALEIN 17185 11724 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME IMMUNOSUPPRESSIVE 16914544 17187 11725 MMP11 4320 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166865 17190 11726 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME GSK-269962A GSK-269962A 17192 11727 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Aldosterone ALDOSTERONE 17193 11728 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME IL-12 10229872 17195 11729 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX BAY 61-3606 22237022 17196 11730 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BUPARLISIB HYDROCHLORIDE 17197 11731 ALOX15 246 ENZYME, DRUGGABLE GENOME MYRICETIN MYRICETIN 17198 11732 RAPGEF3 10411 ENZYME ISOQUINOLINE-1,3(2H,4H)-DIONE CHEMBL1210769 17199 11733 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor 404859118 17200 11734 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Ibritumomab IBRITUMOMAB TIUXETAN 17201 11735 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME OSI-632 OSI-632 17202 11736 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NORHARMANE NORHARMANE 17205 11737 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIBUTYLDICHLOROSTANNANE DIBUTYLDICHLOROSTANNANE 17206 11738 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME AGI-6780 23558173 17208 11739 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Cetuximab CETUXIMAB 17209 11740 IL23A 51561 DRUGGABLE GENOME inhibitor CHEMBL1742995 BRIAKINUMAB 17210 11741 CDK17 5128 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR inhibitor CHEMBL1230607 PHA-793887 17211 11742 MT1F 4494 NA DEXAMETHASONE DEXAMETHASONE 3342021 17213 11743 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ACTB1003 17215 11744 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LJM716 ELGEMTUMAB 28539475 17216 11745 ACVR1B 91 SERINE THREONINE KINASE, CELL SURFACE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 223366128 GALUNISERTIB 17217 11746 SLC2A3 6515 DRUGGABLE GENOME, TRANSPORTER RESVERATROL RESVERATROL 11277764 17218 11747 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME aspirin ASPIRIN 21449675 17219 11748 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BETA-LAPACHONE LAPACHONE 17220 11749 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE brivanib BRIVANIB 20124951 17222 11750 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE IRINOTECAN IRINOTECAN 17224 11751 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR antagonist 223366065 CHEMBL504559 17226 11752 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ISOFLUPREDONE ACETATE ISOFLUPREDONE ACETATE 17227 11753 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9340511, 7 17228 11754 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE 6-METHYLMERCAPTOPURINE RIBOSIDE 10102 17229 11755 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135650010 17230 11756 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651037 SERTINDOLE 17233 11757 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME deferasirox DEFERASIROX 28346059,27193993,27043265 17238 11758 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER NSC-228155 CHEMBL505670 17243 11759 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545205 INCB-40093 17244 11760 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX RIBOCICLIB RIBOCICLIB 29236940 17245 11761 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CANCER DRUG 16319987 17246 11762 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME OPHIOBOLIN O OPHIOBOLIN O 22130129 17247 11763 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUOCINONIDE FLUOCINONIDE 17248 11764 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER teniposide TENIPOSIDE 17249 11765 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE MEK INHIBITOR PD0325901 24141786 17250 11766 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE Urokinase UROKINASE 17251 11767 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR TRIBUTYLCHLOROSTANNANE TRIBUTYLCHLOROSTANNANE 17253 11768 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor HESPERADIN HESPERADIN 19035792 17257 11769 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MM-121 MM-121 17258 11770 RAPGEF3 10411 ENZYME LUTEOLIN LUTEOLIN 17259 11771 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PYRILAMINE PYRILAMINE 17260 11772 TNC 3371 DRUGGABLE GENOME, FIBRINOGEN NEURADIAB 17262 11773 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 178103992 CARFILZOMIB 17263 11774 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PHENYLGLYOXAL PHENYLGLYOXAL 17266 11775 KMT5A 387893 ENZYME inhibitor 178102575 17267 11776 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PENICILLIOL B PENICILLIOL B 19223184 17268 11777 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-2298 CHEMBL578905 17269 11778 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID25656651-Compound-33b 17270 11779 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 17271 11780 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NATEGLINIDE NATEGLINIDE 22931300 17272 11781 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME NM-3 17274 11782 SRD5A1 6715 DRUGGABLE GENOME LEVONORGESTREL LEVONORGESTREL 17277 11783 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PYROGALLOL PYROGALLOL 17278 11784 PDF 64146 DRUGGABLE GENOME PREMETREXED 17279 11785 IL13RA2 3598 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME AER001,AEROVANT 17280 11786 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor SORAFENIB SORAFENIB 17282 11787 NDUFV2 4729 ENZYME inhibitor CHEMBL3545320 ME-344 17285 11788 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE oxazepam OXAZEPAM 17286 11789 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PG-490-88 17287 11790 KCNJ5 3762 TRANSPORTER, ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME activator 135652743 17288 11791 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME META-SIRTINOL CHEMBL200762 23189967 17289 11792 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651319 17290 11793 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565856 17291 11794 CBX1 10951 NA SU-4312 CHEMBL328710 17292 11795 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PD-0166285 PD-0166285 17293 11796 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR SP-600125 SP-600125 17294 11797 KCNT2 343450 ION CHANNEL, DRUGGABLE GENOME blocker 53801073 CLOFILIUM 17298 11798 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102054 17299 11799 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME TCMDC-125185 CHEMBL580819 17301 11800 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Saracatinib SARACATINIB 27231123,26725216 17302 11801 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1201148 MEPREDNISONE 17303 11802 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CARMUSTINE CARMUSTINE 11070098 17305 11803 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650394 17309 11804 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FLOXURIDINE FLOXURIDINE 22931300 17311 11805 MAP3K1 4214 CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME paclitaxel PACLITAXEL 21636554 17312 11806 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENYTOIN PHENYTOIN 17313 11807 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2107312 ARBACLOFEN PLACARBIL 17314 11808 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CHEMBL2108583 CINTREDEKIN BESUDOTOX 17316 11809 PROZ 8858 PROTEASE, DRUGGABLE GENOME MENADIONE MENADIONE 17317 11810 RGS4 5999 DRUGGABLE GENOME SCH-23390 SCH-23390 17318 11811 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CANDESARTAN CILEXETIL CANDESARTAN CILEXETIL 17319 11812 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PD-404182 CHEMBL595227 17320 11813 GMNN 51053 DRUGGABLE GENOME SJ000024939 CHEMBL590691 17321 11814 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor TANDUTINIB TANDUTINIB 17322 11815 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TRIDIHEXETHYL TRIDIHEXETHYL 17323 11816 MAOA 4128 DRUGGABLE GENOME, ENZYME Tarnylcypromine derivative 2 17324 11817 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 249565602 17326 11818 PLD2 5338 ENZYME, DRUGGABLE GENOME activator 135651531 17327 11819 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TOLTERODINE TOLTERODINE 17330 11820 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME INTERLEUKIN-1-BETA 8677009 17331 11821 GFRA1 2674 KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE PYM50028 17333 11822 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TYRPHOSTIN 23 TYRPHOSTIN 23 17334 11823 RAB9A 9367 ENZYME, DRUGGABLE GENOME TCMDC-123748 CHEMBL530609 17335 11824 KMO 8564 DRUGGABLE GENOME, ENZYME Aryl pyrimidine derivative 9 17336 11825 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OLANZAPINE OLANZAPINE 17339 11826 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE E-3810 RABEPRAZOLE SODIUM 17340 11827 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Spironolactone SPIRONOLACTONE 17342 11828 ATXN2 6311 NA GNF-PF-254 CHEMBL461579 17343 11829 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor 249565884 A-443654 17344 11830 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (S)-AMPA (S)-AMPA 17349 11831 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201180 DICLOFENAC EPOLAMINE 17350 11832 BAZ2B 29994 NA GNF-PF-2755 CHEMBL600738 17351 11833 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL856 PRIMIDONE 17352 11834 MALAT1 378938 NA Cilobradine CILOBRADINE 17354 11835 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 252827525 17357 11836 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUNISOLIDE FLUNISOLIDE 17358 11837 PRMT5 10419 ENZYME, METHYL TRANSFERASE inhibitor 252166500 17360 11838 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 315661214 17361 11839 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ESTRADIOL ESTRADIOL 20659801,16520733,19561619 17362 11840 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR CURCUMIN CURCUMIN 17617388,18420184 17363 11841 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME BUDIODARONE BUDIODARONE 17364 11842 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME hmg coa reductase inhibitors 21795085 17365 11843 HPD 3242 ENZYME, DRUGGABLE GENOME NITISINONE NITISINONE 17367 11844 IL23R 149233 KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE celecoxib CELECOXIB 23778325 17368 11845 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PHENAZOPYRIDINE HYDROCHLORIDE PHENAZOPYRIDINE HYDROCHLORIDE 17370 11846 HTT 3064 DRUGGABLE GENOME TERAZOSIN TERAZOSIN 17371 11847 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GLAFENINE GLAFENINE 22931300 17372 11848 NOS2 4843 DRUGGABLE GENOME, ENZYME ibuprofen IBUPROFEN 25502615 17373 11849 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 lopinavir LOPINAVIR 27142945,24950369 17374 11850 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE PX-478 PX-478 17376 11851 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DIMENHYDRINATE DIMENHYDRINATE 17379 11852 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PT005 17380 11853 ADRM1 11047 ENZYME BORTEZOMIB BORTEZOMIB 24524217 17381 11854 GMNN 51053 DRUGGABLE GENOME GNF-PF-1654 CHEMBL602776 17382 11855 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CUCURBITACIN B CUCURBITACIN B 17383 11856 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650160 DARIFENACIN 17385 11857 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR TRICHOSTATIN TRICHOSTATIN 21055848,16921367,19966789,19385600 17386 11858 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME inhibitor CHEMBL3137331 DEFACTINIB 17392 11859 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE S63845 27760111 17393 11860 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor BELINOSTAT BELINOSTAT 17394 11861 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE AZACITIDINE AZACITIDINE 17396 11862 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL1615025 TAK-733 17397 11863 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-44 17398 11864 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR methamphetamine METHAMPHETAMINE 24279859,28692418,26401760 17400 11865 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AG-1288 CHEMBL166486 17404 11866 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR CRYPTOCHINONE A CRYPTOCHINONE A 25127166 17405 11867 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 318164802 17406 11868 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE methotrexate METHOTREXATE 27217051,24241962,29791011,23069858,25502615,23222202,21317831,18381794 17407 11869 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ALOE VERA GEL 9834927 17409 11870 HEXB 3074 ENZYME OMEPRAZOLE OMEPRAZOLE 9593221 17410 11871 ALOX15 246 ENZYME, DRUGGABLE GENOME 3',4'-DIHYDROXYFLAVONE CHEMBL222556 17412 11872 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR MIBEFRADIL MIBEFRADIL 17415 11873 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE OLAPARIB OLAPARIB 28454547,25144364,26650448 17417 11874 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BAY-11-7085 BAY-11-7085 17418 11875 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE 7-azaindole derivative 5 17419 11876 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME CENISERTIB CENISERTIB 17421 11877 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Carbamide derivative 13 17422 11878 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 135651125 17424 11879 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3559672 RAUWOLFIA SERPENTINA 17425 11880 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652292 SEGLITIDE 17427 11881 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIMETHENAMID DIMETHENAMID 17430 11882 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor PAZOPANIB PAZOPANIB 17431 11883 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor 249565817 17432 11884 PIPSL 266971 KINASE inhibitor CARFILZOMIB CARFILZOMIB 17433 11885 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102409 17434 11886 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PF-429242 CHEMBL233611 17583500 17435 11887 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE FLT3L 15102482 17436 11888 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME CI-1040 CI-1040 17437 11889 UBR1 197131 ENZYME DEXAMETHASONE DEXAMETHASONE 17264220 17439 11890 TNFAIP3 7128 PROTEASE, ENZYME, CLINICALLY ACTIONABLE, KINASE Tumor necrosis factor alpha (TNF-alpha) inhibitors 24776844,30653751 17440 11891 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Crizotinib CRIZOTINIB 25971938,27149990,26438783 17441 11892 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135650384 IMIPRAMINE 17442 11893 ATAD5 79915 NA DNDI1417181 CHEMBL1537417 17444 11894 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-16 17445 11895 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR AG-1879 CHEMBL406845 17446 11896 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME REC-01 17447 11897 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE PMID29130358-Compound-Figure17(10) 17448 11898 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Biomed 101 17450 11899 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GSK-269962A GSK-269962A 17451 11900 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR CGTG-102 17452 11901 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651494 17453 11902 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DIETHYLSTILBESTROL DIPROPIONATE DIETHYLSTILBESTROL DIPROPIONATE 17454 11903 PTGS2 5743 DRUGGABLE GENOME, ENZYME ETODOLAC ETODOLAC 17455 11904 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ZD1694 RALTITREXED 10785598 17456 11905 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SGI110 17458 11906 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GNF-PF-1969 CHEMBL601364 17459 11907 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 363894200 TENELIGLIPTIN 17460 11908 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201022 PHENAZOPYRIDINE HYDROCHLORIDE 17461 11909 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1417254 CHEMBL2094567 17462 11910 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DOCEBENONE DOCEBENONE 17464 11911 AKR1C3 8644 ENZYME, DRUGGABLE GENOME N-(benzimidazolylcarbonyl)-piperidine derivative 1 17465 11912 MVD 4597 DRUGGABLE GENOME, ENZYME inhibitor 249565674 17466 11913 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DESIPRAMINE DESIPRAMINE 17467 11914 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME KETOTIFEN KETOTIFEN 17468 11915 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PALBOCICLIB PALBOCICLIB 24417566 17469 11916 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102241 17471 11917 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor BKM120 BUPARLISIB 17472 11918 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BAICALEIN BAICALEIN 17473 11919 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL2103879 GANETESPIB 17477 11920 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 2',4'-DIHYDROXYCHALCONE 2',4'-DIHYDROXYCHALCONE 17478 11921 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR docetaxel DOCETAXEL 17479 11922 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TEBUFENOZIDE TEBUFENOZIDE 17480 11923 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor CHEMBL1090771 AVAGACESTAT 17481 11924 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MITOGEN-ACTIVATED PROTEIN KINASE KINASE INHIBITOR 25952648,29386539 17482 11925 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME NSD-788 17487 11926 TRPV2 51393 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE activator 178100971 CANNABIDIOL 17488 11927 POLI 11201 DNA REPAIR STREPTONIGRIN STREPTONIGRIN 17489 11928 BAZ2B 29994 NA THIETHYLPERAZINE MALATE THIETHYLPERAZINE MALATE 17490 11929 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 178103840 PHENELZINE 17491 11930 TPBG 7162 CELL SURFACE, DRUGGABLE GENOME CHEMBL2108248 ANATUMOMAB MAFENATOX 17492 11931 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ISOFLAVONES 16780800 17493 11932 ATAD5 79915 NA VANOXERINE VANOXERINE 17494 11933 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE TRANEXAMIC ACID 17495 11934 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-125086 CHEMBL532504 17496 11935 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 252827400 VS-4718 17497 11936 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 381744923 17499 11937 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME tiotropium TIOTROPIUM 17500 11938 EREG 2069 KINASE, GROWTH FACTOR, DRUGGABLE GENOME cetuximab CETUXIMAB 17502 11939 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL QUAZEPAM QUAZEPAM 17503 11940 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER DNDI1417076 CHEMBL1526167 17504 11941 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ZEARALENONE ZEARALENONE 17505 11942 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR losartan LOSARTAN 15743363,10594793,20436376 17506 11943 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DOCONEXENT DOCONEXENT 17508 11944 AMPD1 270 DRUGGABLE GENOME, ENZYME methotrexate METHOTREXATE 20386493,27217051,29520081,16947783,27992285 17510 11945 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE KW-2149 9402313 17511 11946 NT5C3A 51251 ENZYME cytarabine CYTARABINE 25000516 17512 11947 ATXN2 6311 NA CAMPTOTHECIN CAMPTOTHECIN 17513 11948 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Trastuzumab TRASTUZUMAB 17514 11949 PRKCH 5583 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565629 SOTRASTAURIN 17515 11950 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME IMGN-853 MIRVETUXIMAB SORAVTANSINE 17517 11951 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-47 17518 11952 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR LEVONORGESTREL LEVONORGESTREL 17519 11953 PDE4D 5144 DRUGGABLE GENOME, ENZYME AN-2898 17521 11954 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME blocker 135651562 SPERMINE 17522 11955 POLK 51426 DNA REPAIR, ENZYME PROSTAGLANDIN B1 PROSTAGLANDIN B1 17523 11956 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200790 METHYPRYLON 17525 11957 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Pyrrolidine carboxamide derivative 1 17526 11958 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR carboplatin CARBOPLATIN 31616045 17527 11959 CXCL8 3576 DRUGGABLE GENOME EMODIN EMODIN 17528 11960 ATAD5 79915 NA MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 17530 11961 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TrasGEX 17531 11962 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BN-AA-003-NY 17534 11963 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor 178101910 MILRINONE 17536 11964 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BKM120 BUPARLISIB 28108151 17537 11965 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BIPHENYL BIPHENYL 17538 11966 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 348353651 17539 11967 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL1946170 REGORAFENIB 17540 11968 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PHA-665752 PHA-665752 18077425 17542 11969 XYLT2 64132 ENZYME carboplatin CARBOPLATIN 31616045 17543 11970 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR DOPAMINE HYDROCHLORIDE DOPAMINE HYDROCHLORIDE 17547 11971 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME TAMATINIB R-406 17548 11972 CDC25C 995 KINASE, PROTEIN PHOSPHATASE, DRUGGABLE GENOME CDDP CISPLATIN 9743457 17550 11973 PRSS3 5646 ENZYME, PROTEASE, DRUGGABLE GENOME CYANOPEPTOLIN S CYANOPEPTOLIN S 17551 11974 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650686 17552 11975 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME PIROXICAM PIROXICAM 9090444 17554 11976 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME NS1 27820802 17555 11977 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 3-CHLOROEVODIAMINE CHEMBL2171782 22867019 17558 11978 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZAMETHIPHOS AZAMETHIPHOS 17559 11979 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME THIOGUANOSINE THIOGUANOSINE 17561 11980 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE olaparib OLAPARIB 17563 11981 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE TAK-593 TAK-593 17565 11982 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FLUNISOLIDE FLUNISOLIDE 22931300 17566 11983 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Pyrimidine analogues 12209976,28950804,24923815,30858516,23603345,16115930,27122156,31382864,22490566,9470816,18600527,26603945,18443386,17700593,17165084,17000685,19530960,26794347,19795123,12360106,19473056,9439663,29845393,26099996,26216193,27864592,17121937,18299612,28295243,15132136,20819423,27995989,16151913,15017333,24817302,30114658,29846282,9323575,29134491,17203168,11895907,32378051,25677447,17064846,20385995,25796495,26265035,17417073,30723313,17848752,23930673,20665215,26804652,29239269,28929491,11350878,11555601,23942539,18452418,27454530,25410891,16361556,21077799,10803677,29889674,14635116,11156223,26846104,21498394,19858398,10071185,23585145 17567 11984 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107647 LANICEMINE 17568 11985 PROS1 5627 DRUGGABLE GENOME Lusutrombopag LUSUTROMBOPAG 17570 11986 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MICHLER'S KETONE MICHLER'S KETONE 17571 11987 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR SR 16234 17572 11988 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE FANCHININ FANCHININ 17574 11989 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100355 ZAFIRLUKAST 17575 11990 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DINOSEB DINOSEB 17578 11991 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor 178102589 17579 11992 HSPB1 3315 DRUGGABLE GENOME CYCLOFENIL CYCLOFENIL 17581 11993 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE GNF-PF-1947 CHEMBL585591 17582 11994 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE MEDI-575 TOVETUMAB 17583 11995 CAMLG 819 NA CYCLOSPORINE A 17584 11996 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE 879325-11-8 17585 11997 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Bevacizumab + Erlotinib 17586 11998 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PF-562271 PF-00562271 17587 11999 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL1721885 SU-014813 17588 12000 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME S-NITROSOGLUTATHIONE S-NITROSOGLUTATHIONE 17590 12001 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER CSA CYCLOSPORINE 11189941 17591 12002 CA5A 763 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL18 ETHOXZOLAMIDE 17592 12003 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE TP-0903 DUBERMATINIB 17593 12004 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE antagonist 178100871 VORAPAXAR 17595 12005 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TRANSPLATIN TRANSPLATIN 17597 12006 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CYCLOSPORINE CYCLOSPORINE 21348461,24720452,17964170,11754602,23017888,24992153 17598 12007 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DISULFIRAM DISULFIRAM 17599 12008 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VIRAL VECTOR 10811480 17603 12009 HTT 3064 DRUGGABLE GENOME Pracinostat PRACINOSTAT 17604 12010 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE VAPBGCRAUJRZPO-UHFFFAOYSA-N 17606 12011 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9409892, 59 17607 12012 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 178102324 NILOTINIB 17610 12013 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 328083495 17611 12014 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLURANDRENOLIDE FLURANDRENOLIDE 17614 12015 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102708 17615 12016 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Diaryl amine derivative 1 17618 12017 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL1569 AMANTADINE HYDROCHLORIDE 17619 12018 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NONOXYNOL 9 NONOXYNOL 9 17620 12019 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 4-HYDROXYBENZALDEHYDE PHENYLHYDRAZONE CHEMBL224032 17621 12020 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103521 17622 12021 TSPO 706 DRUGGABLE GENOME METRONIDAZOLE METRONIDAZOLE 1320691 17623 12022 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 17624 12023 PPP3CA 5530 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Voclosporin VOCLOSPORIN 17625 12024 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 348353622 17626 12025 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR KAEMPFEROL KAEMPFEROL 17627 12026 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Pyridine derivative 21 17629 12027 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE URSODEOXYCHOLIC ACID 9141420 17631 12028 GMNN 51053 DRUGGABLE GENOME CALANOLIDE A CALANOLIDE A 17632 12029 BAZ2B 29994 NA NSC-102742 CHEMBL1519374 17633 12030 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051798 BELINOSTAT 17635 12031 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL3545025 INSM-18 17636 12032 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE Anti-GPC3 CAR T 17637 12033 TSPO 706 DRUGGABLE GENOME Imidazo[1,2-b]pyridazine acetamide derivative 2 17638 12034 RGS4 5999 DRUGGABLE GENOME quetiapine QUETIAPINE 17640 12035 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ANTI-CD3 ANTIBODY 7517362 17641 12036 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALCIPOTRIOL CALCIPOTRIOL 17642 12037 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME SAM-6 17643 12038 PSMC3 5702 NA inhibitor BORTEZOMIB BORTEZOMIB 17644 12039 SPP1 6696 DRUGGABLE GENOME WORTMANNIN WORTMANNIN 14703434 17645 12040 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL998 LORATADINE 17646 12041 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1879463 DACTOLISIB 17647 12042 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 252166565 17648 12043 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME PLATINUM COMPOUND 26057002 17652 12044 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 4-NITROANILINE 4-NITROANILINE 17654 12045 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BGB-283 LIFIRAFENIB 17655 12046 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652553 17656 12047 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEXAMETHASONE DEXAMETHASONE 22931300 17657 12048 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Dacomitinib DACOMITINIB 17658 12049 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-122400 CHEMBL2059067 22524450 17659 12050 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PERFLUOROOCTYLBROMIDE PERFLUBRON 8399771 17660 12051 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME allosteric modulator 223365961 COBIMETINIB 17663 12052 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 223366040 17664 12053 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AMANTADINE HYDROCHLORIDE AMANTADINE HYDROCHLORIDE 17667 12054 TNFRSF11B 4982 DRUGGABLE GENOME EPINEPHRINE EPINEPHRINE 11239501 17670 12055 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME BI-505 BI-505 17673 12056 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Bortezomib BORTEZOMIB 28151717 17676 12057 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BEZ235 DACTOLISIB 17677 12058 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Antibodie derivative 9 17680 12059 ALOX15B 247 DRUGGABLE GENOME, ENZYME 4-TERT-BUTYLCATECHOL CHEMBL220845 17681 12060 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-155693 CHEMBL68096 17682 12061 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME PMID26161698-Compound-18 17683 12062 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR GENISTEIN GENISTEIN 17684 12063 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE olanzapine OLANZAPINE 23559402 17689 12064 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 328083526 CITARINOSTAT 17690 12065 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME ISOQUINOLINE-1,3(2H,4H)-DIONE CHEMBL1210769 17692 12066 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE PHENAMIL METHANESULFONATE PHENAMIL METHANESULFONATE 17693 12067 ALOX15 246 ENZYME, DRUGGABLE GENOME OLEOYL DOPAMINE OLEOYL DOPAMINE 17694 12068 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE REL-8ALPHA-TIGLOYLOXYHIRSUTINOLIDE CHEMBL2062862 26331426 17695 12069 P4HA1 5033 DRUGGABLE GENOME, ENZYME PYRIDINE-2,5-DICARBOXYLIC ACID PYRIDINE-2,5-DICARBOXYLIC ACID 26022078 17696 12070 HTT 3064 DRUGGABLE GENOME CG-200745 CG-200745 17697 12071 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1234354 PF-04691502 17699 12072 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 381744916 17701 12073 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM BROMIDE 17702 12074 SLC22A11 55867 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 252827456 CEPHALOTHIN 17703 12075 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 381744997 REPOTRECTINIB 17704 12076 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ML-10302 CHEMBL286136 17706 12077 PML 5371 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GEMTUZUMAB OZOGAMICIN 15187030 17707 12078 MLH1 4292 CLINICALLY ACTIONABLE, DRUGGABLE GENOME KU60648 28224663 17708 12079 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200334 MORICIZINE HYDROCHLORIDE 17709 12080 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Fluticasone FLUTICASONE 17711 12081 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL411907 SONOLISIB 17712 12082 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX IL-1 7688736,15063754 17713 12083 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR CSA CYCLOSPORINE 15494209 17714 12084 KCNH8 131096 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL113461 TEDISAMIL 17716 12085 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DYCLONINE DYCLONINE 17720 12086 PTGS2 5743 DRUGGABLE GENOME, ENZYME ketoprofen patch 17722 12087 KMO 8564 DRUGGABLE GENOME, ENZYME Isoxazoles and isoxazoline derivative 1 17724 12088 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DIPHYLLIN DIPHYLLIN 17726 12089 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BDBM50080563 17727 12090 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 6-3'-DIMETHYLFLAVONE CHEMBL137498 17728 12091 EML4 27436 CLINICALLY ACTIONABLE, KINASE Sirolimus SIROLIMUS 21613408 17729 12092 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 17730 12093 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417784 CHEMBL1504762 17734 12094 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE RECOMBINANT STEM CELL FACTOR 10432289 17735 12095 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000040829 CHEMBL589711 17736 12096 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TAM 11306479 17737 12097 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Meclizine MECLIZINE 17738 12098 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMPHOTERICIN B AMPHOTERICIN B 22931300 17739 12099 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW612286X GW612286X 17742 12100 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-WO2013082253 32 17743 12101 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME atazanavir ATAZANAVIR 17745 12102 PSMD6 9861 NA CARFILZOMIB CARFILZOMIB 24524217 17747 12103 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID28270010-Compound-Figure21-b 17748 12104 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor CHEMBL1421 DASATINIB 17749 12105 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201828 ECULIZUMAB 17750 12106 SGK1 6446 SERINE THREONINE KINASE, KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME, DRUG RESISTANCE SALINE SODIUM CHLORIDE 16924469 17752 12107 MARCKSL1 65108 KINASE IL-6 11483670 17753 12108 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME 7-NITROINDAZOLE 7-NITROINDAZOLE 17756 12109 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Cisplatin CISPLATIN 28148839 17757 12110 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DIPHEMANIL METHYLSULFATE 17758 12111 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SJ000168197 CHEMBL590670 17760 12112 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PX-866 SONOLISIB 17761 12113 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Sulfaphenazole SULFAPHENAZOLE 17762 12114 ALOX15B 247 DRUGGABLE GENOME, ENZYME PROTOPORPHYRIN PROTOPORPHYRIN 17764 12115 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME FLURAZEPAM FLURAZEPAM 17766 12116 CCL2 6347 DRUGGABLE GENOME RS-504393 17767 12117 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME 20(S)-PROTOPANAXADIOL CHEMBL375563 17261067 17769 12118 FABP1 2168 DRUGGABLE GENOME FENOFIBRIC ACID 17771 12119 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME GIVINOSTAT GIVINOSTAT 17773 12120 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652674 CABERGOLINE 17774 12121 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Radiotherapy 27196762 17777 12122 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CARBETOCIN CARBETOCIN 17781 12123 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE GUTTIFERONE K GUTTIFERONE K 17782 12124 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Isoproterenol ISOPROTERENOL 17784 12125 GBA 2629 DRUGGABLE GENOME, ENZYME CHLORHEXIDINE CHLORHEXIDINE 17785 12126 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 178101464 EMPAGLIFLOZIN 17786 12127 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROCHLORPERAZINE EDISYLATE PROCHLORPERAZINE EDISYLATE 17787 12128 HTT 3064 DRUGGABLE GENOME CGP-60474 CHEMBL300389 17790 12129 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE IRINOTECAN IRINOTECAN 20628391 17791 12130 PAK6 56924 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 310264718 PF-03758309 17792 12131 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102294 BI-2536 17793 12132 TARDBP 23435 TUMOR SUPPRESSOR 1-O-ACETYLGEOPYXIN A CHEMBL1902074 17794 12133 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE BUTAPROST BUTAPROST 17795 12134 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-33 17798 12135 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE agonist CHEMBL1201556 BECAPLERMIN 17799 12136 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME GDC-0349 RG-7603 17800 12137 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 384403681 17801 12138 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 17802 12139 POLK 51426 DNA REPAIR, ENZYME 7,8-DIHYDROXYFLAVONE 7,8-DIHYDROXYFLAVONE 17804 12140 HDAC11 79885 DRUGGABLE GENOME, ENZYME VORINOSTAT VORINOSTAT 19344175,19966789,26211462,23622981,22260166,20491440,21548582,19084294 17807 12141 PTGS1 5742 ENZYME, DRUGGABLE GENOME FLURBIPROFEN FLURBIPROFEN 17808 12142 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BEZAFIBRATE BEZAFIBRATE 17809 12143 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR VEMURAFENIB VEMURAFENIB 24265153,21383288 17810 12144 ATP1A2 477 ENZYME, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME olanzapine OLANZAPINE 17813 12145 FGG 2266 DRUGGABLE GENOME, FIBRINOGEN, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE eptifibatide EPTIFIBATIDE 20938371 17814 12146 PGC 5225 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166834 17818 12147 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 328083464 17819 12148 HBB 3043 DRUGGABLE GENOME, ENZYME MERCAPTOPURINE MERCAPTOPURINE 17820 12149 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE curcumin CURCUMIN 27007499 17821 12150 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ARC029 17822 12151 POLA1 5422 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, DNA REPAIR FLUDARABINE FLUDARABINE 17823 12152 FBP1 2203 DRUGGABLE GENOME, ENZYME MB07803 MB-07803 17824 12153 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HAEMATOXYLIN HAEMATOXYLIN 17825 12154 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FENBUTATIN OXIDE FENBUTATIN OXIDE 17827 12155 ACKR3 57007 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135651708 17830 12156 MAN2C1 4123 DRUGGABLE GENOME M-0011 17835 12157 POLB 5423 DNA REPAIR, DRUGGABLE GENOME DEPHOSTATIN DEPHOSTATIN 17837 12158 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SJ000001592 CHEMBL591834 17839 12159 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME FP-1097 17840 12160 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TIMOLOL TIMOLOL 17841 12161 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CEFUROXIME CEFUROXIME 22166395 17842 12162 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME (S)-FLUOXETINE CHEMBL1169388 17843 12163 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE inhibitor 178103929 ABT-384 17847 12164 NGFR 4804 CELL SURFACE, DRUGGABLE GENOME 178101573 17848 12165 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME glatiramer acetate 22111603 17850 12166 BAZ2B 29994 NA NSC-9037 CHEMBL1451216 17851 12167 ATAD5 79915 NA THUNBERGINOL E THUNBERGINOL E 17852 12168 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL105442 CI-1040 17853 12169 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE carboplatin CARBOPLATIN 17855 12170 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TCMDC-125110 CHEMBL580816 17856 12171 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102338 SU-014813 17857 12172 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor 178103840 PHENELZINE 17859 12173 ALOX5AP 241 DRUGGABLE GENOME AM-103 17860 12174 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR 6,4'-DIMETHOXYFLAVONE 6,4'-DIMETHOXYFLAVONE 17861 12175 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652115 17862 12176 MAPT 4137 DRUGGABLE GENOME DIMETHYL 2-(2-NITROBENZYLIDENE)MALONATE CHEMBL1569494 17863 12177 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178103952 PALBOCICLIB 17864 12178 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISONIAZID ISONIAZID 17866 12179 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Benzamide derivative 8 17867 12180 MDH2 4191 NA EXPECTORANT 15225672 17868 12181 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor CHEMBL1980297 ILORASERTIB 17869 12182 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR LJN452 TROPIFEXOR 17870 12183 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FENTANYL FENTANYL 17987285 17873 12184 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER TCMDC-123769 CHEMBL534353 17874 12185 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GRINIMIBINE GRINIMIBINE 17876 12186 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Isoquinoline sulfonyl derivative 3 17877 12187 KDM7A 80853 ENZYME inhibitor 178103604 17878 12188 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LORATADINE LORATADINE 17879 12189 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE RG-1530 RG-1530 17883 12190 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR 681640 CHEMBL379975 17884 12191 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 17888 12192 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650785 OXYMETAZOLINE 17890 12193 IL7R 3575 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PF-06342674 17891 12194 GAA 2548 DRUGGABLE GENOME, ENZYME PURPUROGALLIN PURPUROGALLIN 17892 12195 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL193240 ROFLUMILAST 17893 12196 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME (RS)-ROSCOVITINE (RS)-ROSCOVITINE 17896 12197 MAPT 4137 DRUGGABLE GENOME 5-NITRO-2-PHENYLPROPYLAMINOBENZOIC ACID [NPPB] 5-NITRO-2-PHENYLPROPYLAMINOBENZOIC ACID [NPPB] 17898 12198 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME acetaminophen ACETAMINOPHEN 19219744,11095574,26049587,19308365,17564651 17899 12199 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE Indole-based analog 3 17900 12200 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Egonol compound 1 17901 12201 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL1096380 PLINABULIN 17903 12202 TH 7054 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200862 METYROSINE 17904 12203 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME DESMEDIPHAM DESMEDIPHAM 17906 12204 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 384403667 17908 12205 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FIIN-2 28034880 17911 12206 XRCC5 7520 KINASE CISPLATIN CISPLATIN 15944802 17912 12207 ANGPT1 284 KINASE, DRUGGABLE GENOME, FIBRINOGEN TREBANINIB 17913 12208 HASPIN 83903 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 252827442 SGI-1776 17915 12209 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 Curcumin CURCUMIN 17916 12210 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NOSCAPINE NOSCAPINE 17917 12211 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME PYRIDINE PYRIDINE 17918 12212 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR INTERFERON ALPHA-2B 10022737 17921 12213 LIPC 3990 ENZYME, PHOSPHOLIPASE, LIPASE, DRUGGABLE GENOME pravastatin PRAVASTATIN 16103896,16115483 17923 12214 TUBB4B 10383 DRUGGABLE GENOME CHEMBL2304041 SAGOPILONE 17924 12215 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME RO-137410 CHEMBL275311 17927 12216 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER TCMDC-125784 CHEMBL581574 17929 12217 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200891 OXYPHENCYCLIMINE HYDROCHLORIDE 17930 12218 GATA2 2624 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX N/A 22147895,22533337,22271902,22814295,25241285,23521373,21892162 17931 12219 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-123762 CHEMBL547483 17932 12220 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE NIC5-15 METHYLINOSITOL 17933 12221 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565885 17934 12222 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1963681 AVANAFIL 17935 12223 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME MNU 12960407 17936 12224 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NICLOSAMIDE NICLOSAMIDE 17937 12225 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME IRINOTECAN IRINOTECAN 28783719,19603018,26687137,26989027,19603024,22180495,27729313 17940 12226 RORA 6095 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE agonist 135651223 T091317 17941 12227 CLDN18 51208 KINASE, DRUGGABLE GENOME antibody 315661285 ZOLBETUXIMAB 17942 12228 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW642138X GW642138X 17943 12229 EIF5A 1984 NA SNS01-T 17944 12230 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417013 CHEMBL1452227 17945 12231 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ESOXYBUTYNIN ESOXYBUTYNIN 17946 12232 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL blocker 178101103 PICROTIN 17947 12233 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Celastrol CELASTROL 17950 12234 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Vistusertib VISTUSERTIB 17951 12235 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-J2 17952 12236 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1200624 ETHYNODIOL DIACETATE 17953 12237 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PANITUMUMAB PANITUMUMAB 17954 12238 CXCL8 3576 DRUGGABLE GENOME BROXURIDINE BROXURIDINE 17956 12239 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651574 LEVOTHYROXINE SODIUM 17957 12240 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-1654 CHEMBL602776 17958 12241 PSMA4 5685 DRUGGABLE GENOME, PROTEASE CARFILZOMIB CARFILZOMIB 24524217 17962 12242 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Plerixafor PLERIXAFOR 17963 12243 GUCY1B1 2983 DRUGGABLE GENOME activator CHEMBL1200689 NITRIC OXIDE 17964 12244 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178103847 PIROXICAM 17965 12245 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 178103272 17966 12246 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE COBIMETINIB COBIMETINIB 30835257 17968 12247 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SUFORAPHANE ISOSELENOCYANATE SUFORAPHANE ISOSELENOCYANATE 20304643 17970 12248 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-48300 CHEMBL1091971 17972 12249 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 9-NITRO-ANTHRACENE CHEMBL166112 17974 12250 CLK1 1195 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 17975 12251 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE BIFONAZOLE BIFONAZOLE 17976 12252 ATAD5 79915 NA TCMDC-125195 CHEMBL531709 17978 12253 PRKAB2 5565 KINASE, ENZYME SAPONARIN SAPONARIN 26471090 17979 12254 BCL2L2 599 CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL443684 NAVITOCLAX 17981 12255 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME 3-(6-allyloxy-2-naphthyl)-1-(4-piperidylmethyl)pyrazolo[3,4-d]pyrimidin-4-amine 17982 12256 MAPT 4137 DRUGGABLE GENOME GNF-PF-3716 CHEMBL609606 17983 12257 KDM4A 9682 DRUGGABLE GENOME, ENZYME N-METHYLHISTAMINE DIHYDROCHLORIDE N-METHYLHISTAMINE DIHYDROCHLORIDE 17984 12258 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR pegaspargase PEGASPARGASE 24141364 17986 12259 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BUFEXAMAC BUFEXAMAC 17987 12260 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME CMI-392 17989 12261 CFL1 1072 KINASE SERTRALINE SERTRALINE 16680159 17990 12262 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 178102572 17991 12263 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NSC-95397 CHEMBL429095 17992 12264 QPRT 23475 ENZYME ARI-3037MO 17993 12265 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE PHA-767491 CHEMBL225519 17995 12266 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor REGORAFENIB REGORAFENIB 17996 12267 NOS1 4842 DRUGGABLE GENOME, ENZYME ANTI-ULCER AGENT 8809208 17998 12268 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Sodium Sulfate 17999 12269 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME US9024044, 3 18000 12270 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME BKM120 BUPARLISIB 26544513 18003 12271 ALOX15 246 ENZYME, DRUGGABLE GENOME IRIGENOL IRIGENOL 18006 12272 HTT 3064 DRUGGABLE GENOME DIPYRITHIONE DIPYRITHIONE 18011 12273 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-2100 CHEMBL576175 18012 12274 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL30219 METHOHEXITAL SODIUM 18013 12275 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME [3H]-PHORBOL 12,13-DIBUTYRATE CHEMBL27768 24794745 18014 12276 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CLENBUTEROL HYDROCHLORIDE CLENBUTEROL HYDROCHLORIDE 18015 12277 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR N,N'-DIPHENYL-GUANIDINE CHEMBL77675 18018 12278 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR S-555739 ASAPIPRANT 18020 12279 HP 3240 DRUGGABLE GENOME, PROTEASE, ENZYME 17 BETA-ESTRADIOL 2078644 18024 12280 POLI 11201 DNA REPAIR PROTOPORPHYRIN PROTOPORPHYRIN 18025 12281 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME 2-PAM derivative 1 18026 12282 BAZ2B 29994 NA SLAZINIC ACID SLAZINIC ACID 18027 12283 POLR3G 10622 NA nevirapine NEVIRAPINE 21810746 18028 12284 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor TOZASERTIB TOZASERTIB 18029 12285 ARSA 410 DRUGGABLE GENOME, ENZYME SQ-22536 CHEMBL64239 18030 12286 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Alteplase ALTEPLASE 18031 12287 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL107 COLCHICINE 18036 12288 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE BIBW 2992 18037 12289 GGCX 2677 DRUGGABLE GENOME, ENZYME ANISINDIONE ANISINDIONE 18038 12290 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE OMEPRAZOLE OMEPRAZOLE 16570509 18041 12291 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor HESPERADIN HESPERADIN 19035792 18042 12292 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Zemab 22069744 18043 12293 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor NINTEDANIB NINTEDANIB 18044 12294 PGP 283871 NA DOCETAXEL DOCETAXEL 18045 12295 RGS4 5999 DRUGGABLE GENOME inhibitor 252827385 18047 12296 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3276 CHEMBL582081 18049 12297 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PLERIXAFOR PLERIXAFOR 18050 12298 SLC1A2 6506 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE inhibitor 178101294 18051 12299 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYPROTERONE ACETATE 26000489 18053 12300 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR INDINAVIR INDINAVIR 10479132 18054 12301 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE DAUNOMYCIN DAUNORUBICIN 2967076 18055 12302 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID29757691-Compound-2a-i 18056 12303 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 16787583 18057 12304 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-73 18058 12305 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme25-4 18061 12306 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR RG-1530 RG-1530 18062 12307 CA2 760 DRUGGABLE GENOME, ENZYME TRICHLORMETHIAZIDE TRICHLORMETHIAZIDE 18063 12308 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BENZPHETAMINE BENZPHETAMINE 18064 12309 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MMV666022 CHEMBL599100 18065 12310 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TENATOPRAZOLE TENATOPRAZOLE 18067 12311 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 336446957 18068 12312 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 6ALPHA-HYDROXYESTRADIOL CHEMBL1432305 18069 12313 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME AZIETOMIDATE AZIETOMIDATE 16884293 18071 12314 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE CLORGILINE CLORGILINE 18073 12315 SMN1 6606 DRUGGABLE GENOME 6,4'-DIMETHOXYFLAVONE 6,4'-DIMETHOXYFLAVONE 18074 12316 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8921389, 123 18075 12317 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651059 CAPESEROD 18077 12318 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-19 18078 12319 PAH 5053 DRUGGABLE GENOME, ENZYME inhibitor 178101924 FENCLONINE 18079 12320 JUNB 3726 TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR INSULIN INSULIN 8264634 18081 12321 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME hydromorphone HYDROMORPHONE 17986163 18082 12322 KDM1A 23028 DRUGGABLE GENOME, ENZYME, CELL SURFACE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING inhibitor 249565921 18083 12323 MOCS1 4337 ENZYME ALXN1101 18084 12324 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE CHIR-99021 CHIR-99021 18086 12325 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200694 SEVOFLURANE 18087 12326 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LORACARBEF HYDRATE LORACARBEF 18088 12327 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX EMETINE HYDROCHLORIDE EMETINE HYDROCHLORIDE 18089 12328 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PF-562271 PF-00562271 18091 12329 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PRECLINICAL 26619011,19657110,20736745,19075190,21576590,16291983,19255327,23414587,18390968,21107323,17384584,23515407,2278970,20406486,20179705,2674680,16273091,19773371,23569304,22761467,18948947,21829508,24370118,3122217,16434492,23076151,26821351,23614898,25157968,20619739,21305640,12460918,17699718,23538902,20130576,8120410,22407852,23406027,20149136,21729679 18093 12330 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIBUTYLTIN-OXIDE TRIBUTYLTIN-OXIDE 18094 12331 FMO3 2328 ENZYME, DRUGGABLE GENOME tamoxifen TAMOXIFEN 23962908 18095 12332 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NSC-69187 CHEMBL19954 18096 12333 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER LICARIN A LICARIN A 18097 12334 HTT 3064 DRUGGABLE GENOME CT-200 18098 12335 HSPB1 3315 DRUGGABLE GENOME VITAMIN C 12473058 18099 12336 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR BUTYRYLHYDROXAMIC ACID BUTYRYLHYDROXAMIC ACID 21874153 18100 12337 APOC3 345 ENZYME, DRUGGABLE GENOME ISIS-APOCIIIRx 18102 12338 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE LINIFANIB LINIFANIB 18107 12339 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650720 18108 12340 PSMD11 5717 KINASE BORTEZOMIB BORTEZOMIB 24524217 18110 12341 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL3544940 G1T28-1 18112 12342 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 187051793 GIVINOSTAT 18114 12343 FCGR2A 2212 CLINICALLY ACTIONABLE, DRUGGABLE GENOME adalimumab ADALIMUMAB 25823785,24667440,24048425,27044681 18115 12344 RPS6KA5 9252 DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor 249565811 18116 12345 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE BDBM50080408 18118 12346 GMNN 51053 DRUGGABLE GENOME HALOPERIDOL HALOPERIDOL 18121 12347 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME SALICYLANILIDE SALICYLANILIDE 18122 12348 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE paclitaxel PACLITAXEL 21636554 18123 12349 ALDH1A1 216 DRUGGABLE GENOME, ENZYME OXYTETRACYCLINE HYDROCHLORIDE OXYTETRACYCLINE HYDROCHLORIDE 18124 12350 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-36 18126 12351 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652100 18127 12352 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PHENACYL CHLORIDE PHENACYL CHLORIDE 18129 12353 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102652 18130 12354 PTGS2 5743 DRUGGABLE GENOME, ENZYME SALICYLIC ACID 18131 12355 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE COCAINE COCAINE 18132 12356 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR STANOLONE STANOLONE 18134 12357 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 8-GERANYLOXY PSORALEN CHEMBL1412710 18135 12358 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME SP-600125 SP-600125 18136 12359 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE GEFITINIB GEFITINIB 18137 12360 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 18138 12361 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL2133806 JNJ-38877605 18141 12362 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DASATINIB DASATINIB 18142 12363 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE INCB62079 18145 12364 PSMA3 5684 PROTEASE, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 24524217 18147 12365 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE TACROLIMUS TACROLIMUS 18149 12366 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 363894160 OZAGREL 18151 12367 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PATULIN PATULIN 18152 12368 ATAD5 79915 NA DNDI1417032 CHEMBL1523974 18153 12369 IPO13 9670 NA MKC-1 ENMD-981693 18154 12370 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Lapatinib LAPATINIB 19718025 18155 12371 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-67 CHEMBL578512 18156 12372 ATXN2 6311 NA GNF-PF-4418 CHEMBL604321 18158 12373 KDM4A 9682 DRUGGABLE GENOME, ENZYME PMID27019002-Compound-21c 18159 12374 ABHD12 26090 ENZYME, DRUGGABLE GENOME, PHOSPHOLIPASE inhibitor 178101960 ORLISTAT 18160 12375 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL501867 VINCRISTINE SULFATE 18161 12376 CYB5R3 1727 DRUGGABLE GENOME, ENZYME sodium nitrite 18163 12377 LNPEP 4012 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, TRANSPORTER, PROTEASE US10023583, Example 13 18165 12378 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR HEPARIN HEPARIN 7794926 18167 12379 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME TAE-684 TAE-684 18168 12380 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME PMID29130358-Compound-Figure16(9a) 18170 12381 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Ex vivo adenosine deaminase-transduced hematopoietic stem cell therapy 18171 12382 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BKM120 BUPARLISIB 27307593 18173 12383 MAP3K10 4294 SERINE THREONINE KINASE, ENZYME, KINASE, DRUGGABLE GENOME DOVITINIB DOVITINIB 18174 12384 PTPRS 5802 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE, CLINICALLY ACTIONABLE inhibitor 252827507 18175 12385 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 328083485 OSI-930 18177 12386 TUBB 203068 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 18178 12387 PIP4K2A 5305 ENZYME, KINASE CB7969312 CHEMBL599255 18179 12388 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR LDE225 SONIDEGIB 18180 12389 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 dapsone DAPSONE 9187528 18182 12390 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE BIMOSIAMOSE BIMOSIAMOSE 18183 12391 RAB9A 9367 ENZYME, DRUGGABLE GENOME AMLEXANOX AMLEXANOX 18186 12392 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SAPRISARTAN SAPRISARTAN 18187 12393 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME DIMETHENAMID DIMETHENAMID 18188 12394 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW621970X GW621970X 18189 12395 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PIM447 18191 12396 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL691 ETHINYL ESTRADIOL 18192 12397 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 acetaminophen ACETAMINOPHEN 19219744,23462933,8659683,26049587,18695978,11866476,9548799 18195 12398 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME activator CHEMBL748 PRALIDOXIME CHLORIDE 18196 12399 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE AZD6738 CERALASERTIB 26563132,26517239 18198 12400 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE LECANORIC ACID LECANORIC ACID 18199 12401 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METFORMIN HYDROCHLORIDE METFORMIN HYDROCHLORIDE 18200 12402 PDE4D 5144 DRUGGABLE GENOME, ENZYME GSK-356278 GSK-356278 18201 12403 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CHLORPROMAZINE CHLORPROMAZINE 18203 12404 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1620 DIPHENHYDRAMINE HYDROCHLORIDE 18204 12405 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SB-216763 SB-216763 25467150,20708937,20030405 18207 12406 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Paclitaxel PACLITAXEL 18208 12407 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125310 CHEMBL582030 18209 12408 S100A12 6283 DRUGGABLE GENOME, KINASE MTX METHOTREXATE 15077313 18210 12409 MAP3K9 4293 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565853 CEP-1347 18211 12410 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME CENISERTIB CENISERTIB 18212 12411 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125620 CHEMBL530291 18216 12412 PDE3A 5139 ENZYME, DRUGGABLE GENOME THEOPHYLLINE THEOPHYLLINE 18217 12413 CFL1 1072 KINASE ROTENONE ROTENONE 16680159 18219 12414 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME agonist 178100889 18220 12415 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME ILORASERTIB ILORASERTIB 18221 12416 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651134 18222 12417 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ENDRIN ENDRIN 18223 12418 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Pyrrolo-pyrrolone derivative 1 18224 12419 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER TDR77403 CHEMBL1534035 18227 12420 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL FLURAZEPAM FLURAZEPAM 18230 12421 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE CYC116 18231 12422 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1339 VARDENAFIL HYDROCHLORIDE 18232 12423 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY PYRAZOLE PYRAZOLE 6992153 18233 12424 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME BISLEUCONOTHINE A BISLEUCONOTHINE A 26176165 18235 12425 HMGCR 3156 ENZYME, DRUGGABLE GENOME Aspirin ASPIRIN 18236 12426 PSMD12 5718 NA inhibitor BORTEZOMIB BORTEZOMIB 18237 12427 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR (+)-ISOBICYCLOGERMACRENAL CHEMBL2333548 18238 12428 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody 249565770 NECITUMUMAB 18240 12429 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ondansetron ONDANSETRON 9187528 18241 12430 BRCA2 675 CLINICALLY ACTIONABLE NU1025 15829966 18243 12431 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Ruxolitinib RUXOLITINIB 24398328,21926964,22271575,24251790,21393331,26472029 18247 12432 PSMD6 9861 NA inhibitor CHEMBL325041 BORTEZOMIB 18248 12433 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE Oxcarbazepine OXCARBAZEPINE 18249 12434 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME GLPG0974 GLPG-0974 18250 12435 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200382 BEPRIDIL HYDROCHLORIDE 18251 12436 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME WEDELOLACTONE WEDELOLACTONE 18252 12437 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CLONAZEPAM CLONAZEPAM 18259 12438 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHYSTICIN METHYSTICIN 18261 12439 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL24 ATENOLOL 18262 12440 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201558 INTERFERON ALFA-2B 18265 12441 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE allosteric modulator 178102544 18266 12442 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-31 18267 12443 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR PLERIXAFOR PLERIXAFOR 18270 12444 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ROSE BENGAL ROSE BENGAL 18271 12445 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BEZAFIBRATE BEZAFIBRATE 18276 12446 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-69 18277 12447 TNNC1 7134 DRUGGABLE GENOME LEVOSIMENDAN LEVOSIMENDAN 18278 12448 ALDH1A1 216 DRUGGABLE GENOME, ENZYME E319 E319 18279 12449 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Mapracorat MAPRACORAT 18281 12450 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DIGOXIN DIGOXIN 18282 12451 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ATRA TRETINOIN 18048326 18284 12452 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE CEP-5214 CEP-5214 14640546 18285 12453 XDH 7498 DRUGGABLE GENOME, ENZYME Azole benzene derivative 2 18288 12454 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SHP099 27362227 18290 12455 E2F1 1869 TRANSCRIPTION FACTOR LARGAZOLE LARGAZOLE 18291 12456 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL296468 BMS-387032 18292 12457 CXCL8 3576 DRUGGABLE GENOME HARMINE HYDROCHLORIDE HARMINE HYDROCHLORIDE 18293 12458 YWHAG 7532 DRUGGABLE GENOME, KINASE DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 18294 12459 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102336 BOSUTINIB 18295 12460 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME PMID29130358-Compound-Figure16(9b) 18298 12461 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE Drug 2849330 18302 12462 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE TKM-APOB 18304 12463 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE antagonist CHEMBL1743030 ICRUCUMAB 18305 12464 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Dextrothyroxine Sodium 18307 12465 FLCN 201163 CLINICALLY ACTIONABLE EVEROLIMUS EVEROLIMUS 23995526 18308 12466 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 6 18309 12467 MAPT 4137 DRUGGABLE GENOME Davunetide intranasal spray 18310 12468 EYA2 2139 DNA REPAIR DIACEREIN DIACEREIN 18311 12469 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR FLUOXETINE FLUOXETINE 9228186 18312 12470 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650754 OCAPERIDONE 18313 12471 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE allosteric modulator 252166706 REPARIXIN 18314 12472 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR MYRICETIN MYRICETIN 18315 12473 COL18A1 80781 DRUGGABLE GENOME ASPIRIN ASPIRIN 11353854 18316 12474 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AZITHROMYCIN AZITHROMYCIN 22931300 18317 12475 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL940 GABAPENTIN 18319 12476 ALOX15 246 ENZYME, DRUGGABLE GENOME INAMRINONE INAMRINONE 18320 12477 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 135650845 PROPYLPYRAZOLETRIOL 18321 12478 GAA 2548 DRUGGABLE GENOME, ENZYME PHLORETIN PHLORETIN 18322 12479 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE PACLITAXEL PACLITAXEL 26096845 18323 12480 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649960 18324 12481 CA2 760 DRUGGABLE GENOME, ENZYME Chlorothiazide CHLOROTHIAZIDE 18327 12482 HMGCR 3156 ENZYME, DRUGGABLE GENOME PMID27537201-Compound-Figure13c 18328 12483 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE (20S,21S)-FLUOROCAMPTOTHECIN (20S,21S)-FLUOROCAMPTOTHECIN 24069881 18329 12484 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME partial agonist CHEMBL3545230 APIMOSTINEL 18330 12485 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200606 MEXILETINE HYDROCHLORIDE 18331 12486 GMNN 51053 DRUGGABLE GENOME CEPHALOCHROMIN CEPHALOCHROMIN 18333 12487 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor SF1126 18334 12488 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR GEMFIBROZIL GEMFIBROZIL 17823123 18335 12489 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565729 18336 12490 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CHLOPHEDIANOL CHLOPHEDIANOL 18339 12491 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE etanercept ETANERCEPT 20309874,23007924 18340 12492 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CAROTENOIDS 15309450 18341 12493 GMNN 51053 DRUGGABLE GENOME AMIODARONE HYDROCHLORIDE AMIODARONE HYDROCHLORIDE 18343 12494 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL antagonist CHEMBL14935 TEZAMPANEL 18345 12495 PDE5A 8654 ENZYME, DRUGGABLE GENOME VARDENAFIL VARDENAFIL 18346 12496 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME afutuzumab OBINUTUZUMAB 24795454 18347 12497 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 3R14S-OCHRATOXIN A 3R14S-OCHRATOXIN A 18348 12498 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 indinavir INDINAVIR 9187528 18349 12499 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME DASATINIB DASATINIB 18350 12500 NDUFS5 4725 ENZYME inhibitor CHEMBL3545320 ME-344 18352 12501 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE GW441756X GW441756X 18353 12502 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Nelipepimut S 18354 12503 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUTOLANIL FLUTOLANIL 18355 12504 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL1237099 DOXACURIUM CHLORIDE 18357 12505 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Acyl piperidine derivative 1 18361 12506 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME KB07 CHEMBL373822 17181166 18362 12507 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 310264691 18363 12508 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 187051798 BELINOSTAT 18365 12509 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE CEPHALOTHIN CEPHALOTHIN 18366 12510 KCNC3 3748 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL113461 TEDISAMIL 18368 12511 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C23 18370 12512 UGT1A10 54575 DRUGGABLE GENOME, ENZYME oxcarbazepine OXCARBAZEPINE 27900402 18371 12513 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DISULFIRAM DISULFIRAM 18373 12514 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR ARSENIC TRIOXIDE 25759020 18374 12515 IRS1 3667 KINASE, CLINICALLY ACTIONABLE GLIMEPIRIDE GLIMEPIRIDE 15710354 18375 12516 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME FEXOFENADINE FEXOFENADINE 18376 12517 TH 7054 ENZYME, DRUGGABLE GENOME IFN 8724983 18377 12518 TH 7054 ENZYME, DRUGGABLE GENOME DOXYCYCLINE DOXYCYCLINE 15585109 18378 12519 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-3125 CHEMBL534288 18381 12520 PTGS2 5743 DRUGGABLE GENOME, ENZYME SULINDAC SULINDAC 18382 12521 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Dinaciclib DINACICLIB 27550941,25931518 18383 12522 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 252166637 RELENOPRIDE 18384 12523 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHYL ROBUSTONE METHYL ROBUSTONE 18385 12524 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE ERYTHROPOIETIN EPOETIN BETA 11023508 18386 12525 EYA2 2139 DNA REPAIR CLOFAZIMINE CLOFAZIMINE 18387 12526 ATAD5 79915 NA GNF-PF-78 CHEMBL579318 18389 12527 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 7,12-DIMETHYL-BENZO[A]ANTHRACENE CHEMBL329673 18392 12528 TDO2 6999 ENZYME, DRUGGABLE GENOME TCDD 7716779 18394 12529 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR 4-(4-AMINOPHENYL)BUTANOIC ACID CHEMBL1650245 24044874 18396 12530 GGCX 2677 DRUGGABLE GENOME, ENZYME ANISINDIONE ANISINDIONE 18398 12531 MAOB 4129 DRUGGABLE GENOME, ENZYME PF9601N 18400 12532 IFNGR2 3460 CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist CHEMBL1201564 INTERFERON GAMMA-1B 18401 12533 ATXN2 6311 NA PYRONIN Y PYRONIN Y 18402 12534 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CETUXIMAB CETUXIMAB 19603024,20619739,19223544,28424201 18403 12535 HTT 3064 DRUGGABLE GENOME SHP-141 REMETINOSTAT 18404 12536 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME enasidenib ENASIDENIB 18405 12537 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NBQX NBQX 18406 12538 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RAPAMYCIN SIROLIMUS 16651424 18407 12539 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME NILE RED NILE RED 18408 12540 KLKB1 3818 DRUGGABLE GENOME, PROTEASE, ENZYME KVD001 18409 12541 THBD 7056 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME LEVOTHYROXINE LEVOTHYROXINE 14763909 18410 12542 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651741 18411 12543 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TCMDC-123634 CHEMBL530499 18413 12544 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 187051816 CHEMBL2153434 18414 12545 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE ALN-VSP 18415 12546 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650109 CLOBENPROPIT 18417 12547 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME AZD-1152-HQPA AZD-1152-HQPA 18419 12548 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL3545078 PF-03814735 18420 12549 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL2105635 DAVALINTIDE 18422 12550 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 lesinurad LESINURAD 18423 12551 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE vincristine VINCRISTINE 18424 12552 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE Crofelemer CROFELEMER 18425 12553 UCP2 7351 TRANSPORTER, DRUGGABLE GENOME HEPARIN HEPARIN 10868951 18426 12554 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200446 TRIPELENNAMINE HYDROCHLORIDE 18427 12555 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Human prothrombin complex concentrate 18428 12556 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 363894216 TUCATINIB 18429 12557 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650982 18430 12558 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103458 VORINOSTAT 18431 12559 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1201139 MEGESTROL ACETATE 18432 12560 TUBB 203068 DRUGGABLE GENOME CHEMBL2105643 FOSBRETABULIN TROMETHAMINE 18433 12561 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE KU004 26437915 18434 12562 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-124356 CHEMBL22062 18435 12563 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR HAEMATOXYLIN HAEMATOXYLIN 18436 12564 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 135651333 CHEMBL189753 18437 12565 PTGS2 5743 DRUGGABLE GENOME, ENZYME PMID29130358-Compound-LonimacranthoideVI 18438 12566 GMNN 51053 DRUGGABLE GENOME MMV006389 CHEMBL586000 18441 12567 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 363894224 HENATINIB 18443 12568 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME O,O'-DIMETHYLCAFFEIC ACID O,O'-DIMETHYLCAFFEIC ACID 18445 12569 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AZD6738 CERALASERTIB 26563132,28062704 18446 12570 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-317605 CHEMBL1312050 18450 12571 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AGI-5198 23558169,26363012,28148839 18451 12572 EYA2 2139 DNA REPAIR GNF-PF-67 CHEMBL578512 18452 12573 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 381118862 18453 12574 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE GDC-0068 IPATASERTIB 18454 12575 SMN2 6607 DRUGGABLE GENOME GNF-PF-1211 CHEMBL600968 18457 12576 MAOA 4128 DRUGGABLE GENOME, ENZYME Secondary and tertiary (hetero)arylamide derivative 2 18459 12577 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 QUINALIZARIN QUINALIZARIN 18462 12578 RORA 6095 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE agonist 135651457 CHOLESTEROL 18463 12579 CDA 978 ENZYME, DRUGGABLE GENOME CYTARABINE CYTARABINE 12008078 18466 12580 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 363894130 TANZISERTIB 18467 12581 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE 2'-AMINO-3'-METHOXYFLAVONE 18349105 18468 12582 IFNG 3458 DRUGGABLE GENOME SURAMIN SURAMIN 1899122 18471 12583 IL1B 3553 KINASE, DRUGGABLE GENOME risedronate RISEDRONIC ACID 16257277 18473 12584 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649920 ALNIDITAN 18474 12585 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE doxorubicin DOXORUBICIN 539595 18475 12586 SF3B1 23451 CLINICALLY ACTIONABLE Spliceostatin A 25424858 18476 12587 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LERCANIDIPINE HYDROCHLORIDE LERCANIDIPINE HYDROCHLORIDE 18477 12588 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME GNF-PF-1919 CHEMBL576409 18478 12589 KDM4A 9682 DRUGGABLE GENOME, ENZYME Selenium compound 2 18479 12590 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Cyclohexane carboxamide derivative 3 18480 12591 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME HYDROXYZINE PAMOATE HYDROXYZINE PAMOATE 18481 12592 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE AC1LE05K 18483 12593 LTC4S 4056 ENZYME, DRUGGABLE GENOME inhibitor 385612238 18484 12594 IL1B 3553 KINASE, DRUGGABLE GENOME Celastrol CELASTROL 18485 12595 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor MK0752 18487 12596 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Pazopanib + Tyverb/Tykerb 18488 12597 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME TRIAZOLAM TRIAZOLAM 18490 12598 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME LAMIVUDINE LAMIVUDINE 15309715 18492 12599 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 310264733 FIMEPINOSTAT 18493 12600 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME KAI-1455 18497 12601 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE RESVERATROL RESVERATROL 11008129 18500 12602 PPCDC 60490 ENZYME gemcitabine GEMCITABINE 18501 12603 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZOXAMIDE ZOXAMIDE 18502 12604 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SB-203580 SB-203580 18504 12605 DHFR 1719 DRUGGABLE GENOME, ENZYME PEMETREXED PEMETREXED 18507 12606 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Beta-phe compound 3 18508 12607 FXR2 9513 NA methylphenidate METHYLPHENIDATE 29382897 18509 12608 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME radiotherapy 25054431 18510 12609 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 178102101 18513 12610 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE STX-0119 CHEMBL1687979 18514 12611 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE TILUDRONATE TILUDRONIC ACID 18515 12612 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545248 DS-7423 18516 12613 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200395 ORPHENADRINE CITRATE 18517 12614 GATM 2628 ENZYME, TRANSPORTER simvastatin SIMVASTATIN 18519 12615 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102549 18520 12616 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BENZALKONIUM CHLORIDE BENZALKONIUM CHLORIDE 18521 12617 GPI 2821 ENZYME, GROWTH FACTOR, DRUGGABLE GENOME 6-AN 10884030 18522 12618 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 26194362 18523 12619 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DICHLOROTRIPHENYLBISMUTHANE DICHLOROTRIPHENYLBISMUTHANE 18524 12620 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 7-Vanillyl alcohol 18525 12621 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-4791 CHEMBL583555 18526 12622 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE CVBT-141H 18527 12623 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR RV-GM-CSF 10880241 18528 12624 APOE 348 DRUGGABLE GENOME VITAMIN E 12076219 18529 12625 PSMC6 5706 NA BORTEZOMIB BORTEZOMIB 24524217 18531 12626 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ACTINOMYCIN D 9494516 18532 12627 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL ARC029 18533 12628 MALT1 10892 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE inhibitor 354702255 MEPAZINE 18535 12629 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Cholecalciferol CHOLECALCIFEROL 18537 12630 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 diazepam DIAZEPAM 9187528 18538 12631 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Triazolo-pyrazinone derivative 1 18543 12632 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FOSFONET FOSFONET 18544 12633 POLI 11201 DNA REPAIR MITONAFIDE MITONAFIDE 18546 12634 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER p53-SLP vaccine 21328579,19621448 18547 12635 DHODH 1723 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL973 TERIFLUNOMIDE 18548 12636 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PENTACHLOROPHENOL PENTACHLOROPHENOL 18549 12637 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME taxanes 26194361 18551 12638 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650065 18556 12639 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SCLAREOL SCLAREOL 18557 12640 PSENEN 55851 DRUGGABLE GENOME LY-411575 CHEMBL392068 23181502,19443228 18558 12641 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Desloratadine DESLORATADINE 18559 12642 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE JTT-654 18561 12643 GMNN 51053 DRUGGABLE GENOME TCMDC-124395 CHEMBL534047 18562 12644 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-18 18563 12645 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Isoxazole derivative 1 18564 12646 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PF-562271 PF-00562271 18565 12647 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME 7,8,2'-TRIHYDROXYFLAVONE CHEMBL244707 18567 12648 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME ErepoXen 18568 12649 RRM2 6241 DRUGGABLE GENOME, ENZYME CALAA-01 18570 12650 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1258517 PKI-179 18571 12651 BARD1 580 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR APITOLISIB APITOLISIB 28389374 18572 12652 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL GABOXADOL GABOXADOL 18573 12653 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL3545381 PLX-7486 18575 12654 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Imidazo[1,2-b]pyridazine derivative 1 18576 12655 HLA-DRB5 3127 DRUGGABLE GENOME, CLINICALLY ACTIONABLE clozapine CLOZAPINE 11146763 18577 12656 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR everolimus EVEROLIMUS 18579 12657 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2012135799 43(1.5) 18580 12658 MPHOSPH8 54737 NA METHYLDOPA (RACEMIC) METHYLDOPA (RACEMIC) 18582 12659 HTT 3064 DRUGGABLE GENOME ARTEMISIN ARTEMISIN 18583 12660 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE RO5126766 26438159 18584 12661 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALACHLOR ALACHLOR 18585 12662 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRADIOL PHOSPHATE ESTRADIOL PHOSPHATE 18587 12663 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME IFN 15634924,15657875 18588 12664 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL87992 ESLICARBAZEPINE ACETATE 18589 12665 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Indazole derivative 1 18590 12666 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GDC-0032 TASELISIB 25172762,26333383 18591 12667 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DAPIPRAZOLE DAPIPRAZOLE 18592 12668 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL944 CHLOROPROCAINE HYDROCHLORIDE 18594 12669 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME Selective serotonin reuptake inhibitors 24930681,22086748,19204908,17414739,28639488 18596 12670 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RS-100329 CHEMBL56331 18597 12671 BAZ2B 29994 NA NAFTOPIDIL DIHYDROCHLORIDE NAFTOPIDIL DIHYDROCHLORIDE 18598 12672 MPHOSPH8 54737 NA PIMOZIDE PIMOZIDE 18599 12673 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE nicorandil NICORANDIL 18602 12674 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Sapitinib SAPITINIB 24886365 18603 12675 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33g 18604 12676 CYP20A1 57404 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME MBC 9347928 18605 12677 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR DAPHNORIN DAPHNORIN 18606 12678 MAGEA3 4102 ENZYME, DRUGGABLE GENOME vaccine EP-2101 18607 12679 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Cevimeline CEVIMELINE 18608 12680 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME BMS-387032 BMS-387032 18609 12681 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR TACEDINALINE TACEDINALINE 18692397 18610 12682 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE HAEMATOXYLIN HAEMATOXYLIN 18611 12683 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650342 GSK-9578 18612 12684 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME OSI-632 OSI-632 18613 12685 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 INDOMETHACIN INDOMETHACIN 22931300 18615 12686 CBX1 10951 NA MYRICETIN MYRICETIN 18616 12687 GMNN 51053 DRUGGABLE GENOME DYCLONINE DYCLONINE 18617 12688 HPN 3249 DRUGGABLE GENOME, PROTEASE, CELL SURFACE N-Methyl-D-aspartic acid 18619 12689 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME YM-264 18620 12690 PSENEN 55851 DRUGGABLE GENOME inhibitor PF03084014 18623 12691 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2103736 FENOPROFEN CALCIUM 18624 12692 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE asparaginase ASPARAGINASE 18625 12693 FTO 79068 ENZYME azathioprine AZATHIOPRINE 27558924 18627 12694 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist CHEMBL3545016 CLASCOTERONE 18628 12695 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER NELFINAVIR NELFINAVIR 17664327 18630 12696 ATAD5 79915 NA GNF-PF-710 CHEMBL596839 18632 12697 NR1D1 9572 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME agonist 310264681 SR9011 18633 12698 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME HOMIDIUM HOMIDIUM 18634 12699 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 amiodarone AMIODARONE 9187528 18635 12700 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER nefazodone NEFAZODONE 21449676 18638 12701 CCND2 894 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE BAY1000394 18641 12702 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE GLISOFLAVONE GLISOFLAVONE 20724155 18642 12703 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE AZD-8055 AZD-8055 23375793 18644 12704 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100418 18647 12705 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE HYDROCORTISONE HYDROCORTISONE 2395837 18648 12706 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 17 18649 12707 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor BYL719 ALPELISIB 18650 12708 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PANITUMUMAB PANITUMUMAB 22270724 18651 12709 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PHA-767491 CHEMBL225519 18652 12710 LTC4S 4056 ENZYME, DRUGGABLE GENOME US20160326143, 3 18657 12711 XDH 7498 DRUGGABLE GENOME, ENZYME NITROFURANTOIN NITROFURANTOIN 6297496 18658 12712 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 223365982 AC-480 18660 12713 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ETHANOL ALCOHOL 10092515 18661 12714 HBB 3043 DRUGGABLE GENOME, ENZYME NSC-348401 CHEMBL515505 18663 12715 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 178102681 WORTMANNIN 18664 12716 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor MK0752 18668 12717 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLOFIBRATE CLOFIBRATE 22931300 18670 12718 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MUSCLE RELAXANT 9918604 18671 12719 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BINIMETINIB BINIMETINIB 31566309,29573941 18672 12720 MAPT 4137 DRUGGABLE GENOME DEHYDROVARIABILIN DEHYDROVARIABILIN 18675 12721 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200694 SEVOFLURANE 18678 12722 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE METHOTREXATE METHOTREXATE 14512390 18679 12723 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PMID29130358-Compound-Figure18(14) 18680 12724 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Tariquidar TARIQUIDAR 18682 12725 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR US9073931, E2 18683 12726 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor PD-0332991 PALBOCICLIB 18684 12727 KDM4A 9682 DRUGGABLE GENOME, ENZYME CHLOROXINE CHLOROXINE 18687 12728 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRITON X TRITON X 18688 12729 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ticlopidine TICLOPIDINE 17339877 18689 12730 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE TYRPHOSTIN A9 TYRPHOSTIN A9 18692 12731 TUBB2B 347733 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 18693 12732 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE MODIFIED IFN-ALPHA 18695 12733 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 385612248 18696 12734 TUBB 203068 DRUGGABLE GENOME Plinabulin PLINABULIN 18697 12735 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME LY3023414 SAMOTOLISIB 18700 12736 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE S-110 18701 12737 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Paricalcitol PARICALCITOL 18702 12738 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE PF-04840082 18704 12739 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 2-(4-HYDROXYBENZYLIDENE)MALONONITRILE CHEMBL305695 18705 12740 MAPK7 5598 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TG02, SB1317 18706 12741 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR ASCORBIC ACID 12520757 18707 12742 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-747270 CHEMBL594772 18709 12743 PDF 64146 DRUGGABLE GENOME Proguanil CHLOROGUANIDE 18710 12744 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 328083477 18711 12745 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103403 BRINZOLAMIDE 18712 12746 SLC25A4 291 DRUGGABLE GENOME, TRANSPORTER Clodronate CLODRONIC ACID 18713 12747 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Amelubant AMELUBANT 18714 12748 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ELLAGIC ACID ELLAGIC ACID 18715 12749 ATAD5 79915 NA MMV020651 CHEMBL549216 18716 12750 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GAMOLENIC ACID GAMOLENIC ACID 18718 12751 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME MLN-8054 MLN-8054 18719 12752 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME CATECHIN CATECHIN 18722 12753 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW786460X GW786460X 18725 12754 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AM-461 AM-461 18728 12755 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ALISERTIB ALISERTIB 18730 12756 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 354702216 LODOXAMIDE 18731 12757 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor GDC-0980 APITOLISIB 18732 12758 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-95397 CHEMBL429095 18733 12759 CHST3 9469 DRUGGABLE GENOME, ENZYME thalidomide THALIDOMIDE 20038957 18734 12760 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE YU238259 26116172 18736 12761 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103686 ALFUZOSIN 18739 12762 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Oxeglitazar OXEGLITAZAR 18740 12763 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Amidopyrazole derivative 2 18741 12764 PTGS2 5743 DRUGGABLE GENOME, ENZYME CELECOXIB CELECOXIB 18742 12765 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BRUCINE BRUCINE 18743 12766 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565805 18745 12767 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE montelukast MONTELUKAST 18746 12768 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE LOXO-101 LAROTRECTINIB 18749 12769 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE modulator CHEMBL189475 LADARIXIN 18750 12770 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE VX-970 BERZOSERTIB 18751 12771 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE CAPECITABINE CAPECITABINE 18752 12772 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SORAFENIB TOSYLATE SORAFENIB TOSYLATE 18753 12773 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEFUROXIME SODIUM CEFUROXIME SODIUM 18754 12774 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Irinotecan IRINOTECAN 25567130 18755 12775 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PF-05280586 18756 12776 KDM4A 9682 DRUGGABLE GENOME, ENZYME ACID BLUE 129 ACID BLUE 129 18758 12777 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RETINYLRETINOATE RETINYLRETINOATE 18511283 18759 12778 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist 178100903 18761 12779 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ISOFLUPREDONE ACETATE ISOFLUPREDONE ACETATE 18766 12780 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME EFAVIRENZ EFAVIRENZ 21189339 18770 12781 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Tricyclic compound 11 18771 12782 GMNN 51053 DRUGGABLE GENOME RESERPINE RESERPINE 18773 12783 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SNS-314 SNS-314 18774 12784 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor MK2206 MK-2206 18775 12785 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LAUROGUADINE LAUROGUADINE 18776 12786 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME efavirenz EFAVIRENZ 24729586 18778 12787 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TERBUTALINE TERBUTALINE 18779 12788 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME TCMDC-124356 CHEMBL22062 18780 12789 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor 328083477 18782 12790 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ALRESTATIN ALRESTATIN 18783 12791 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RETINOL RETINOL 18511283 18784 12792 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL483158 ALISERTIB 18785 12793 CDK10 8558 DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL488436 AZD-5438 18786 12794 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME IODOPHTHALEIN IODOPHTHALEIN 18787 12795 ATAD5 79915 NA 7,12-DIMETHYL-BENZO[A]ANTHRACENE CHEMBL329673 18789 12796 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Olaparib OLAPARIB 18790 12797 MAPKAPK5 8550 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 363894142 18791 12798 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28117607-Compound-6 18792 12799 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor AUY922 18793 12800 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE MELPHALAN MELPHALAN 9031449 18795 12801 PSMD6 9861 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 18797 12802 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME LY-2090314 LY-2090314 18798 12803 GBA 2629 DRUGGABLE GENOME, ENZYME DNDI1417773 CHEMBL1379900 18800 12804 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ELLIPTECINE ELLIPTECINE 18802 12805 MAPT 4137 DRUGGABLE GENOME METHYSERGIDE MALEATE 18803 12806 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE AMG 900 18807 12807 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 363894215 TAFETINIB 18808 12808 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 249565632 AT-9283 18809 12809 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER lopinavir LOPINAVIR 23996099 18810 12810 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ASTEMIZOLE ASTEMIZOLE 18811 12811 POLK 51426 DNA REPAIR, ENZYME OXYTETRACYCLINE OXYTETRACYCLINE 18818 12812 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME TGX-221 26577700,26137449 18819 12813 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME ARRY-162 BINIMETINIB 18822 12814 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME cetuximab CETUXIMAB 26438111 18823 12815 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE N/A 18824 12816 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CBT-1 18827 12817 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 178102318 KW-2449 18829 12818 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR INTERLEUKIN-1 9352015 18830 12819 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TROGLITAZONE TROGLITAZONE 22931300 18831 12820 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-78 CHEMBL579318 18833 12821 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME MILTIRONE MILTIRONE 26339922 18834 12822 AREG 374 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE cetuximab CETUXIMAB 23959273 18835 12823 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CHRYSOERIOL CHRYSOERIOL 25190466 18837 12824 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ETHACRIDINE ETHACRIDINE 18838 12825 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Demcizumab DEMCIZUMAB 26855149 18839 12826 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME fluvastatin FLUVASTATIN 18840 12827 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PF-04217903 PF-04217903 18841 12828 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL18 ETHOXZOLAMIDE 18843 12829 SLC1A3 6507 TRANSPORTER, DRUGGABLE GENOME, CELL SURFACE 178101255 18844 12830 CCL28 56477 DRUGGABLE GENOME ANTISERUM 15681819 18845 12831 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor OLAPARIB OLAPARIB 18846 12832 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyrrolo-pyrimidine derivative 1 18847 12833 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ACEPROMETAZINE ACEPROMETAZINE 18848 12834 MPHOSPH8 54737 NA SR-2640 SR-2640 18849 12835 MICU1 10367 TRANSPORTER ALD-403 EPTINEZUMAB 18850 12836 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE MARIMASTAT MARIMASTAT 18851 12837 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BOLDINE BOLDINE 18852 12838 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CTLA4-IG ABATACEPT 9758890 18853 12839 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33h 18855 12840 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LEVONORGESTREL LEVONORGESTREL 18857 12841 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SORAFENIB SORAFENIB 18858 12842 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme12-2 18860 12843 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME CENISERTIB CENISERTIB 18861 12844 CD59 966 DRUGGABLE GENOME, CELL SURFACE, KINASE MBL 17113913 18862 12845 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DICYCLOHEXYLCARBODIIMIDE DICYCLOHEXYLCARBODIIMIDE 18865 12846 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-D2 18867 12847 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor RETASPIMYCIN RETASPIMYCIN 18868 12848 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650862 18870 12849 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AD-CD154 15914559 18871 12850 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PROTUBOXEPIN A PROTUBOXEPIN A 22595423 18872 12851 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 HYDROXYZINE HYDROXYZINE 22931300 18873 12852 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE C-RAF ANTISENSE OLIGONUCLEOTIDE 18874 12853 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DIGITOXIN DIGITOXIN 18879 12854 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME SSR-126517E 18880 12855 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL2108061 VOLOCIXIMAB 18882 12856 PTGES 9536 DRUGGABLE GENOME, ENZYME AAD-2004 18886 12857 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-21 18889 12858 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BI-87E7 CHEMBL523200 18890 12859 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ELLAGIC ACID ELLAGIC ACID 18893 12860 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DIPHEMANIL METHYLSULFATE 18894 12861 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Crizotinib CRIZOTINIB 25264305,25667280 18896 12862 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GEFITINIB GEFITINIB 18897 12863 NOS2 4843 DRUGGABLE GENOME, ENZYME VEGF 10928051 18898 12864 HKDC1 80201 DRUGGABLE GENOME, KINASE DNDI1417874 CHEMBL1865517 18900 12865 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL2364639 VALBENAZINE 18901 12866 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NIZOFENONE NIZOFENONE 18902 12867 F5 2153 DRUGGABLE GENOME Eltrombopag ELTROMBOPAG 18903 12868 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME MORIN MORIN 18905 12869 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PD173074 27179038,23908597,24122810,26036639,22869148 18906 12870 DDX43 55510 DRUG RESISTANCE MEK INHIBITOR PD0325901 24899684 18907 12871 PDK3 5165 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE CPI-613 18909 12872 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL98 VORINOSTAT 18911 12873 HBB 3043 DRUGGABLE GENOME, ENZYME FLUOROURACIL FLUOROURACIL 18912 12874 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OCTYL_GALLATE OCTYL_GALLATE 18915 12875 CRYZ 1429 ENZYME, DRUGGABLE GENOME 2'-HYDROXYCHALCONE 2'-HYDROXYCHALCONE 20639112 18916 12876 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE TROGLITAZONE TROGLITAZONE 11947963 18917 12877 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Brivanib BRIVANIB 22238366 18921 12878 FCGR2A 2212 CLINICALLY ACTIONABLE, DRUGGABLE GENOME SM-101 VALZIFLOCEPT 18924 12879 PSMB4 5692 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL451887 CARFILZOMIB 18927 12880 GLS 2744 ENZYME NAFCILLIN SODIUM NAFCILLIN SODIUM 18930 12881 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE PROGESTIN PROGESTERONE 11590147 18931 12882 TNFRSF4 7293 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE antibody 315661320 VONLEROLIZUMAB 18932 12883 GMNN 51053 DRUGGABLE GENOME GLYCYROL GLYCYROL 18933 12884 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR Ace Inhibitors, Plain 14643574 18934 12885 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ROFECOXIB ROFECOXIB 16707021 18936 12886 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Troplasminogen alfa 18937 12887 MVK 4598 KINASE, ENZYME inhibitor 135651486 FARNESOL 18939 12888 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PECTOLINARIGENIN PECTOLINARIGENIN 18940 12889 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR R0-93877 18942 12890 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME ENALAPRIL ENALAPRIL 10712274 18943 12891 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RS-100329 CHEMBL56331 18945 12892 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CH5132799 PA-799 21558396 18947 12893 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BETULIN BETULIN 11754608 18948 12894 PSMD6 9861 NA inhibitor CARFILZOMIB CARFILZOMIB 18950 12895 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL verapamil VERAPAMIL 20031608 18953 12896 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 2,2,3,3,4,4,5,5,6,6,7,7,8,8,9,9,9-HEPTADECAFLUORO-NONANOIC ACID CHEMBL426404 18954 12897 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE OPB-31121 18955 12898 FAAH 2166 ENZYME, DRUGGABLE GENOME Tetra-hydro-naphthalene derivative 3 18956 12899 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME 4-CHLOROBENZOHYDROXAMIC ACID CHEMBL569419 25937017 18958 12900 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR irinotecan IRINOTECAN 18959 12901 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR ISOPROTERENOL ISOPROTERENOL 9730867 18964 12902 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME DACTOLISIB DACTOLISIB 18965 12903 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 252827404 18966 12904 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CINOLAZEPAM CINOLAZEPAM 18967 12905 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE LOXO-195 SELITRECTINIB 18968 12906 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US10149841, Compound 9 18969 12907 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE 8ALPHA-HYDROXYHIRSUTINOLIDE CHEMBL2062863 26331426 18970 12908 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Temozolomide TEMOZOLOMIDE 25910950 18972 12909 PCSK5 5125 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178103178 18974 12910 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051797 APICIDIN 18975 12911 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AMG 232 25567130 18977 12912 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE ICA-105665 18978 12913 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE OPB-51602 18979 12914 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 U-0126 U-0126 18980 12915 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LAS-101057 LAS101057 18981 12916 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 249565649 ROCILETINIB 18982 12917 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BAS-8770931 CHEMBL515495 19179076 18983 12918 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 336446933 18984 12919 KDM4A 9682 DRUGGABLE GENOME, ENZYME GERONTOXANTHONE H GERONTOXANTHONE H 18985 12920 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 LEUCINE LEUCINE 22931300 18986 12921 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME POL-6326 POL6326 18987 12922 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DESOGESTREL DESOGESTREL 18988 12923 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor BUPARLISIB HYDROCHLORIDE 18989 12924 VEGFC 7424 GROWTH FACTOR, TRANSPORTER, DRUGGABLE GENOME BEVACIZUMAB BEVACIZUMAB 18990 12925 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme21Left 18991 12926 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME PYRONIN Y PYRONIN Y 18992 12927 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PROTOPORPHYRIN PROTOPORPHYRIN 9267885 18993 12928 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE IGF-1R antibody 27196767 18995 12929 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2107979 PEXELIZUMAB 18996 12930 GNA13 10672 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR oxaliplatin OXALIPLATIN 24444404 19000 12931 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2,4,6-TRIBROMOPHENOL CHEMBL220087 19002 12932 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME ELMIRON ELMIRON 17071199 19003 12933 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ADRIAMYCIN ADRIAMYCIN 8162589 19004 12934 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 178102328 PI-103 19006 12935 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME HEMATIDE PEGINESATIDE 19008 12936 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 178102572 19009 12937 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR INSULIN INSULIN 8945471,8712800 19010 12938 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Triazolo-pyrimidinedione derivative 1 19011 12939 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102714 19013 12940 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PEG-3350 19016 12941 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE antibody APOMAB APOMAB 19017 12942 ALPI 248 DRUGGABLE GENOME, ENZYME NSC-353720 CHEMBL1408276 19018 12943 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE FLAVOPIRIDOL ALVOCIDIB 14767524 19020 12944 GMNN 51053 DRUGGABLE GENOME FEPRAZONE FEPRAZONE 19021 12945 UGT1A6 54578 ENZYME, DRUGGABLE GENOME phenytoin PHENYTOIN 26049587 19022 12946 RGS4 5999 DRUGGABLE GENOME CISPLATIN CISPLATIN 19024 12947 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Amidopyrazole derivative 1 19025 12948 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545381 PLX-7486 19026 12949 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 4'-METHOXYFLAVONE 4'-METHOXYFLAVONE 19027 12950 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME VRT11E 24265153 19028 12951 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME blocker 135650220 ECONAZOLE 19029 12952 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200802 TALBUTAL 19030 12953 PTGS1 5742 ENZYME, DRUGGABLE GENOME TENOXICAM TENOXICAM 19032 12954 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TRIETHYLENETHIOPHOSPHORAMIDE 12058967 19034 12955 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME ENTRECTINIB ENTRECTINIB 19035 12956 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL simvastatin SIMVASTATIN 27839692,25753936 19036 12957 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ANTIDEPRESSANT 7901780 19038 12958 TSPO 706 DRUGGABLE GENOME Estazolam ESTAZOLAM 19039 12959 TRPM6 140803 ION CHANNEL, DRUGGABLE GENOME, ENZYME, TRANSPORTER, KINASE, SERINE THREONINE KINASE blocker 135652746 19041 12960 BAZ2B 29994 NA NSC-228155 CHEMBL505670 19042 12961 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR 5'-DEOXY-5-FLUOROURIDINE 12408764 19043 12962 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE YUANHUADINE YUANHUADINE 21916433 19044 12963 TUBB 203068 DRUGGABLE GENOME CHEMBL2108628 PACLITAXEL POLIGLUMEX 19046 12964 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102818 19047 12965 VEGFB 7423 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR VEGF-2 19049 12966 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR YM-358 CHEMBL347610 19050 12967 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE ILORASERTIB ILORASERTIB 19051 12968 HEBP1 50865 DRUGGABLE GENOME inhibitor CHEMBL1762621 BARDOXOLONE METHYL 19052 12969 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME 178101640 REGRAMOSTIM 19053 12970 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SGM-1019 19054 12971 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CLOTIAZEPAM CLOTIAZEPAM 19056 12972 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENOFIBRATE FENOFIBRATE 19057 12973 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME METHADONE METHADONE 22685215 19062 12974 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME inhibitor 375973226 19063 12975 SQSTM1 8878 SERINE THREONINE KINASE IMX-942 DUSQUETIDE 19064 12976 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774824-Compound-Figure11Example1up 19065 12977 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ARZOXIFENE ARZOXIFENE 19066 12978 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL601719 CRIZOTINIB 19067 12979 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor NINTEDANIB NINTEDANIB 19068 12980 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE CHEMBL1743078 TEPLIZUMAB 19069 12981 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 249565855 19070 12982 ALPL 249 ENZYME, DRUGGABLE GENOME THUNBERGINOL B THUNBERGINOL B 19073 12983 IL1B 3553 KINASE, DRUGGABLE GENOME rabeprazole RABEPRAZOLE 16815316,21054464,14638340 19074 12984 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE Thyrotropin THYROTROPIN 19075 12985 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL646 TRIAZOLAM 19077 12986 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME simvastatin SIMVASTATIN 27839692 19078 12987 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME VALPROIC ACID VALPROIC ACID 18294844,16921367,25304896 19079 12988 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417111 CHEMBL2094456 19080 12989 TAGLN 6876 NA 5-AZACYTIDINE AZACITIDINE 14662021 19081 12990 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 APIGENIN APIGENIN 19082 12991 KLK7 5650 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252166691 19083 12992 PDE8A 5151 DRUGGABLE GENOME, ENZYME inhibitor 178101509 DIPYRIDAMOLE 19084 12993 TXNRD1 7296 DRUGGABLE GENOME Palmarumycin derivative 2 19086 12994 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME etoposide ETOPOSIDE 12969965 19087 12995 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUNISOLIDE FLUNISOLIDE 19088 12996 FARP2 9855 NA methylphenidate METHYLPHENIDATE 29382897 19092 12997 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-180246 CHEMBL484640 19094 12998 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PURPUROGALLIN PURPUROGALLIN 19095 12999 IL1B 3553 KINASE, DRUGGABLE GENOME ARA-C 7523795 19096 13000 GLS 2744 ENZYME NSC-37642 CHEMBL1707907 19097 13001 GMNN 51053 DRUGGABLE GENOME LYCOPENE LYCOPENE 19098 13002 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME Pyridinone compound 1 19099 13003 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME R-1487 R-1487 19101 13004 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR XL888 XL-888 19104 13005 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE CISPLATIN CISPLATIN 3337743 19105 13006 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GALLIC ACID GALLIC ACID 19106 13007 MUC5AC 4586 DRUGGABLE GENOME KLS-0611 19107 13008 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-52 19108 13009 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE N6-2-PHENYLETHYLADENOSINE CHEMBL1257013 19109 13010 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE CI-1040 CI-1040 19111 13011 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR DIFLUFENICAN DIFLUFENICAN 19112 13012 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 4-Carboxamido-isoindolinone derivative 3 19115 13013 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 384403640 19116 13014 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE PD-0166285 PD-0166285 19117 13015 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL539423 SPARSENTAN 19118 13016 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GW7647 GW7647 19119 13017 MID1 4281 ENZYME, B30_2 SPRY DOMAIN, DRUGGABLE GENOME SUN-N8075 19120 13018 KEAP1 9817 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 252827430 19123 13019 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MESALAMINE MESALAMINE 19124 13020 ACTG1 71 NA vincristine VINCRISTINE 19126 13021 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ZEARALENONE ZEARALENONE 19128 13022 POLK 51426 DNA REPAIR, ENZYME ERYTHROSINE ERYTHROSINE 19129 13023 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C21 19130 13024 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Trastuzumab TRASTUZUMAB 19134 13025 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL445813 AT-7519 19135 13026 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME VORINOSTAT VORINOSTAT 19344175,19966789,26211462,23622981,22260166,18381238,20491440,21548582,19084294 19138 13027 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALC-0061 19139 13028 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE pemetrexed PEMETREXED 29662106,24732178,20634689,19307503 19140 13029 DROSHA 29102 NA cyclophosphamide CYCLOPHOSPHAMIDE 24614921 19143 13030 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 19144 13031 ALOX15 246 ENZYME, DRUGGABLE GENOME POMIFERIN POMIFERIN 19145 13032 CXCL8 3576 DRUGGABLE GENOME CIDOFOVIR CIDOFOVIR 10630964 19146 13033 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 2,3,4'-TRIHYDROXY-4-METHOXYBENZOPHENONE 2,3,4'-TRIHYDROXY-4-METHOXYBENZOPHENONE 19147 13034 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3544935 XL-418 19150 13035 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 340590226 OLECLUMAB 19151 13036 LPAR2 9170 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 135651509 19152 13037 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 315661268 19153 13038 MAPT 4137 DRUGGABLE GENOME IODOPHTHALEIN IODOPHTHALEIN 19154 13039 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE ACP-001 ACP-001 19156 13040 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Vemurafenib VEMURAFENIB 24265153,24265152,27196754,27048951 19157 13041 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 9 19158 13042 PGA3 643834 PROTEASE, DRUGGABLE GENOME, ENZYME SUCRALFATE SUCRALFATE 19159 13043 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 223366206 INFIGRATINIB 19160 13044 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR SLAZINIC ACID SLAZINIC ACID 19161 13045 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Afatinib AFATINIB 28274957,26545934,27044931,24971884,22325357,27923043,25589492,23775486,28363995,23578997,26964772,23948973,28167203,25370464,26243863,21617858 19162 13046 RACGAP1 29127 NA NSC-699479 CHEMBL1701915 19165 13047 TSPO 706 DRUGGABLE GENOME Bidentate pyrazolopyrimidine acetamide analog 2 19166 13048 MAPT 4137 DRUGGABLE GENOME LAPACHOL LAPACHOL 19167 13049 FMO3 2328 ENZYME, DRUGGABLE GENOME daunorubicin DAUNORUBICIN 25119182 19168 13050 STK10 6793 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 381118815 19169 13051 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLOBENPROPIT CLOBENPROPIT 19171 13052 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NINTEDANIB NINTEDANIB 19172 13053 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CGP-7930 CHEMBL1256697 19173 13054 CCR7 1236 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR agonist 178100552 19175 13055 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Pyrido[1,2-a]indole-1.-carboxylic acid analog 7 19176 13056 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Alpha-adrenoreceptor antagonists 19177 13057 KDM4A 9682 DRUGGABLE GENOME, ENZYME METHIOTHEPIN MESYLATE METHIOTHEPIN MESYLATE 19180 13058 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor 318164849 CDP840 19181 13059 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545385 WX-037 19182 13060 TNFRSF4 7293 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE GBR 830 19183 13061 SULT1A3 6818 DRUGGABLE GENOME, ENZYME tramadol TRAMADOL 19184 13062 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GEFITINIB GEFITINIB 19185 13063 GBA 2629 DRUGGABLE GENOME, ENZYME GNF-PF-2094 CHEMBL578928 19186 13064 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PHYSOSTIGMINE PHYSOSTIGMINE 19187 13065 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker 135650352 CHEMBL298475 19188 13066 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-19 19192 13067 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SB-220025 SB-220025 19194 13068 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor VORINOSTAT VORINOSTAT 19196 13069 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE clavulanate CLAVULANIC ACID 30664875 19197 13070 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME ISOLATED SOY PROTEIN 11125428 19201 13071 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE OPIOID 16450289 19202 13072 NFKBIA 4792 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME 6-METHOXYCOMAPARVIN 5-METHYL ETHER CHEMBL256967 18088098 19203 13073 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Vemurafenib VEMURAFENIB 24265152 19205 13074 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-348401 CHEMBL515505 19206 13075 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20120264760C81 19208 13076 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR FASUDIL FASUDIL 19211 13077 TMEM97 27346 NA Piperazinyl methyl quinazolinone derivative 1 19214 13078 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE RANITIDINE RANITIDINE 10383521 19215 13079 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1096 AMLEXANOX 19216 13080 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AG-99 CHEMBL296407 19217 13081 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE ABT-263 NAVITOCLAX 19220 13082 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME TF0023 19222 13083 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LORATADINE LORATADINE 19223 13084 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE JNJ-7706621 JNJ-7706621 19225 13085 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 19227 13086 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLOFIBRIC ACID CLOFIBRIC ACID 19228 13087 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME 5-NITRO-2-PHENYLPROPYLAMINOBENZOIC ACID [NPPB] 5-NITRO-2-PHENYLPROPYLAMINOBENZOIC ACID [NPPB] 19229 13088 FAAH 2166 ENZYME, DRUGGABLE GENOME Azetidine urea derivative 2 19230 13089 GMNN 51053 DRUGGABLE GENOME GNF-PF-3876 CHEMBL596631 19232 13090 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417268 CHEMBL1517542 19233 13091 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ASIMADOLINE ASIMADOLINE 19234 13092 ACVR1B 91 SERINE THREONINE KINASE, CELL SURFACE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE US10030004, Compound 11a 19235 13093 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-172614 CHEMBL1317506 19237 13094 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME QUERCETIN DIHYDRATE QUERCETIN DIHYDRATE 19238 13095 ATAD5 79915 NA MICHLER'S KETONE MICHLER'S KETONE 19240 13096 SDC1 6382 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CART-138 cells 19241 13097 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3314 CHEMBL582287 19242 13098 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR VEGF 11018037,12114504 19243 13099 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 315661253 19244 13100 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-37 19247 13101 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Dovitinib DOVITINIB 22238366,23175443,24325461,27932416,28034880,25589496 19249 13102 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME REL-CARINATIN C CHEMBL2332127 19250 13103 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME DIHYDROTANSHINONE I DIHYDROTANSHINONE I 26339922 19251 13104 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417055 CHEMBL1486366 19253 13105 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE PONEZUMAB PONEZUMAB 19254 13106 IMPA1 3612 ENZYME, DRUGGABLE GENOME inhibitor 178101897 19255 13107 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DINOSEB DINOSEB 19256 13108 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PP-121 26483207 19257 13109 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR 6R-SENECIONYLCHAPARRIN CHEMBL564009 19199792 19258 13110 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor MK2206 MK-2206 19260 13111 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651410 CHEMBL1767409 19261 13112 DMD 1756 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Ataluren ATALUREN 19262 13113 ADCY9 115 KINASE, ENZYME, DRUGGABLE GENOME dalcetrapib DALCETRAPIB 25583994 19263 13114 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME PF-562271 PF-00562271 19264 13115 CYB5R1 51706 DRUGGABLE GENOME metoclopramide METOCLOPRAMIDE 19267 13116 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Cetuximab CETUXIMAB 28783719,25714871,28363909,26208524,26287849,22270724,22281684,25838391,27312529,26916115,27002107,24523613 19271 13117 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME DOVITINIB DOVITINIB 19272 13118 CDK10 8558 DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL1230607 PHA-793887 19274 13119 POLK 51426 DNA REPAIR, ENZYME PENICILLIOL A PENICILLIOL A 19223184 19275 13120 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER ANTIVIRAL 12105214 19276 13121 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE RINDOPEPIMUT RINDOPEPIMUT 25586468 19277 13122 KDM4A 9682 DRUGGABLE GENOME, ENZYME OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 19278 13123 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE OLAPARIB OLAPARIB 19279 13124 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-67 19282 13125 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Cenestin CENESTIN 19283 13126 POLK 51426 DNA REPAIR, ENZYME DEXKETOPROFEN DEXKETOPROFEN 19284 13127 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE rosuvastatin ROSUVASTATIN 30100615 19285 13128 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AGROCLAVINE AGROCLAVINE 19286 13129 TSC22D3 1831 NA HYDROCORTISONE HYDROCORTISONE 15728202 19288 13130 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor BIBW 2992 19290 13131 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Peptide analog 50 19291 13132 MBL2 4153 DRUGGABLE GENOME, CELL SURFACE DANAZOL DANAZOL 12076401 19293 13133 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME BUPIVACAINE BUPIVACAINE 10838161 19295 13134 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 8606853 19296 13135 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ISTRADEFYLLINE ISTRADEFYLLINE 19297 13136 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR leucovorin LEUCOVORIN 24141364 19299 13137 NPR3 4883 DRUGGABLE GENOME antagonist 178101571 19302 13138 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102578 19303 13139 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME 178101283 19306 13140 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME ARUNCIN B ARUNCIN B 22197393 19308 13141 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIETHYLCARBAMAZINE CITRATE DIETHYLCARBAMAZINE CITRATE 19309 13142 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200771 TRIDIHEXETHYL CHLORIDE 19310 13143 CBL 867 KINASE, ENZYME, CLINICALLY ACTIONABLE DASATINIB DASATINIB 23696637 19311 13144 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651417 19312 13145 HTT 3064 DRUGGABLE GENOME DNDI1417941 CHEMBL2095095 19313 13146 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 328083460 19314 13147 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER colchicine COLCHICINE 25876828 19316 13148 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Semuloparin SEMULOPARIN 19317 13149 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME DIPHOSPHONATE 3923787 19318 13150 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DIETHYLSTILBESTROL DIETHYLSTILBESTROL 19320 13151 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME FLUORANTHEN-3-YLAMINE CHEMBL103583 19321 13152 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 18221820 19322 13153 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GLYBURIDE GLYBURIDE 19324 13154 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2-METHYL-5,7,8-TRIMETHOXYISOFLAVONE 2-METHYL-5,7,8-TRIMETHOXYISOFLAVONE 19325 13155 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE Peptide analog 57 19327 13156 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX BREFELDIN A BREFELDIN A 19329 13157 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 178102514 REGORAFENIB 19331 13158 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PROPRANOLOL PROPRANOLOL 22931300 19333 13159 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE CHEMOSENSITIZER 15503311 19336 13160 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor LY2835219 ABEMACICLIB 19337 13161 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR olanzapine OLANZAPINE 24595507 19338 13162 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 2-ARACHIDONOYLGLYCEROL 2-ARACHIDONOYLGLYCEROL 19339 13163 USP1 7398 DNA REPAIR, PROTEASE, ENZYME (+)-ALPHA-TOCOPHERYL SUCCINATE (+)-ALPHA-TOCOPHERYL SUCCINATE 19340 13164 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME SUNITINIB SUNITINIB 19341 13165 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE 6-HYDROXYFLAVONE 6-HYDROXYFLAVONE 19342 13166 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 650707 CHEMBL408653 19343 13167 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GNF-PF-5114 CHEMBL601952 19344 13168 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Bis-aminopyrimidine derivative 1 19345 13169 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody 178103470 IPILIMUMAB 19346 13170 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME HORMONES 16099855 19347 13171 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME PMID28594589-Compound-TABLE3C14 19349 13172 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME PF-06826647 19350 13173 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 315661333 BIIB021 19351 13174 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BROMAMINIC ACID BROMAMINIC ACID 19353 13175 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE DESLANOSIDE DESLANOSIDE 19354 13176 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME verubecestat VERUBECESTAT 19355 13177 GMNN 51053 DRUGGABLE GENOME LENPERONE LENPERONE 19357 13178 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Research programme: peroxisome proliferator-activated receptor gamma agonist, Omeros 19358 13179 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PMID27376512-Compound-Figure3CM 19359 13180 RGS4 5999 DRUGGABLE GENOME PYRROLIDINE DITHIOCARBAMATE PYRROLIDINE DITHIOCARBAMATE 19362 13181 CLK3 1198 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, TYROSINE KINASE HARMINE HARMINE 22998443 19366 13182 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIFLUMIZOLE TRIFLUMIZOLE 19367 13183 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME NATALIZUMAB NATALIZUMAB 19369 13184 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-miR-155-5p 19373 13185 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CATECHIN CATECHIN 19374 13186 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME NORETHISTERONE ACETATE 11915588 19375 13187 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DICHLON DICHLON 19377 13188 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201729 DRONEDARONE HYDROCHLORIDE 19378 13189 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR AMSACRINE HYDROCHLORIDE AMSACRINE HYDROCHLORIDE 19379 13190 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 363894130 TANZISERTIB 19380 13191 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Pyridoxal Phosphate 19382 13192 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545112 ME-401 19384 13193 VAC14 55697 KINASE docetaxel DOCETAXEL 19385 13194 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 223365930 LEVORPHANOL 19386 13195 GLS 2744 ENZYME CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 19388 13196 ABCA4 24 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME StarGen 19389 13197 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE osimertinib OSIMERTINIB 19391 13198 MAPT 4137 DRUGGABLE GENOME TETROQUINONE TETROQUINONE 19394 13199 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 178102671 19395 13200 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CLIOXANIDE CLIOXANIDE 19397 13201 AQP1 358 ION CHANNEL, DRUGGABLE GENOME CARBONIC ANHYDRASE INHIBITOR 14704128 19398 13202 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PACLITAXEL PACLITAXEL 19400 13203 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102720 19402 13204 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE IRIGINOL HEXAACEATATE IRIGINOL HEXAACEATATE 19403 13205 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE APIGENIN APIGENIN 19405 13206 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor PX-866 SONOLISIB 19406 13207 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE US9156852, 38 19407 13208 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 3,4-DICHLOROISOCOUMARIN CHEMBL24983 19408 13209 POLB 5423 DNA REPAIR, DRUGGABLE GENOME QUINACRINE DIHYDROCHLORIDE QUINACRINE DIHYDROCHLORIDE 19410 13210 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE MOTESANIB MOTESANIB 19411 13211 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL3545418 BMS-779788 19412 13212 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIMETHYL YELLOW DIMETHYL YELLOW 19413 13213 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 363894201 TENALISIB 19414 13214 SMN1 6606 DRUGGABLE GENOME AG1295 AG1295 19415 13215 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4-METHYLENE-5BETA-HYDROPEROXYOVATODIOLIDE CHEMBL471694 26178912 19416 13216 SMARCA4 6597 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING TOZASERTIB TOZASERTIB 28102363 19418 13217 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE Peptide analog 58 19419 13218 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CCT128930 CHEMBL263664 21191045 19421 13219 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME AG-494 CHEMBL56731 19422 13220 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PYRIDOSTIGMINE PYRIDOSTIGMINE 19423 13221 GMNN 51053 DRUGGABLE GENOME GEDUNIN GEDUNIN 19424 13222 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102639 19428 13223 HSPG2 3339 KINASE, DRUGGABLE GENOME antipsychotics 21808285 19430 13224 MAOB 4129 DRUGGABLE GENOME, ENZYME 8-[3-(TRIFLUOROMETHYL)PHENOXYMETHYL]CAFFEINE CHEMBL2088303 22705191 19431 13225 MAOB 4129 DRUGGABLE GENOME, ENZYME 4-Hydroxy-2,5-dimethyl-3(2H)-furanone 19432 13226 RACGAP1 29127 NA SJ000264145 CHEMBL590675 19434 13227 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-228155 CHEMBL505670 19435 13228 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DNDI1417221 CHEMBL1459280 19438 13229 EZH1 2145 METHYL TRANSFERASE, ENZYME inhibitor 249565920 19441 13230 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GARLIC GARLIC 16351512 19442 13231 TH 7054 ENZYME, DRUGGABLE GENOME INDOMETHACIN INDOMETHACIN 12646303 19444 13232 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3545322 PANULISIB 19446 13233 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200478 DYCLONINE HYDROCHLORIDE 19448 13234 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE KU-0060648 CHEMBL1086377 23855836 19449 13235 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROMETHAZINE PROMETHAZINE 19450 13236 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PKC412 MIDOSTAURIN 11719451 19451 13237 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CHEMBL1257 ENFLURANE 19452 13238 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL1743075 TABALUMAB 19453 13239 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545052 FIMEPINOSTAT 19454 13240 TRH 7200 DRUGGABLE GENOME 6-AMINONICOTINAMIDE 6-AMINONICOTINAMIDE 6240361 19456 13241 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME DNDI1417467 CHEMBL1997335 19457 13242 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 404859136 19458 13243 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE FRM-0962 19460 13244 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 223366170 NS-018 19461 13245 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE JSM 6427 19462 13246 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TYROSINE KINASE INHIBITORS 15811957 19464 13247 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MONTELUKAST MONTELUKAST 22931300 19465 13248 NUP50 10762 NA teniposide TENIPOSIDE 24444404 19466 13249 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER GLUFOSFAMIDE GLUFOSFAMIDE 19467 13250 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE AR-A014418 CHEMBL259850 19468 13251 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PIPENZOLATE PIPENZOLATE 19469 13252 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 223366123 BARICITINIB 19471 13253 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor PIVANEX AN-9 19473 13254 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RACLOPRIDE RACLOPRIDE 19474 13255 UGCG 7357 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1029 MIGLUSTAT 19475 13256 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER GNF-PF-910 CHEMBL585408 19476 13257 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME INDOPROFEN INDOPROFEN 19478 13258 NDUFS1 4719 ENZYME inhibitor CHEMBL3545320 ME-344 19479 13259 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE L-ASPARAGINASE ASPARAGINASE 9264396 19480 13260 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-3257 CHEMBL601768 19481 13261 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Deflazacort DEFLAZACORT 19483 13262 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102597 19485 13263 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE PMID26882240-Compound-2 19487 13264 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PF-2413873 19489 13265 BAZ2B 29994 NA TDR78834 CHEMBL1507526 19490 13266 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CETALKONIUM CHLORIDE CETALKONIUM CHLORIDE 19491 13267 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL1230609 FORETINIB 19492 13268 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ETHAVERINE ETHAVERINE 19493 13269 ATXN2 6311 NA CUCURBITACIN B CUCURBITACIN B 19494 13270 ICA1 3382 NA tramadol TRAMADOL 30971809 19496 13271 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102334 19497 13272 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NILUTAMIDE NILUTAMIDE 26000489 19498 13273 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SNS-314 SNS-314 19501 13274 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ENMD-2076 ENMD-2076 19503 13275 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-Figure5aVIII 19504 13276 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE IMMUNOSTIMULANT 10483872 19505 13277 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker 178100954 19506 13278 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL HALAZEPAM HALAZEPAM 19507 13279 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME clopidogrel CLOPIDOGREL 24971633 19508 13280 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-348401 CHEMBL515505 19511 13281 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Levocetirizine dihydrochloride 19512 13282 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DARIFENACIN DARIFENACIN 19513 13283 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-asCEBP-2HPE 19516 13284 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL3707400 INDANTADOL 19517 13285 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE P7170 PANULISIB 25700704 19518 13286 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE EMETINE EMETINE 15974627 19520 13287 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 249565801 19521 13288 CGA 1081 DRUGGABLE GENOME, HORMONE ACTIVITY 4-{([(4'-CHLOROPHENYL)AMINO]CARBONYLAMINO)}BENZENESULFONAMIDE CHEMBL1446150 19522 13289 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME 1-(biphenyl-4-yl-methyl)-1H-imidazole derivative 1 19524 13290 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME C 82 19526 13291 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 prednisolone PREDNISOLONE 9187528 19527 13292 ABHD6 57406 PHOSPHOLIPASE, ENZYME inhibitor 381744927 19528 13293 ATXN2 6311 NA PROADIFEN HYDROCHLORIDE PROADIFEN HYDROCHLORIDE 19529 13294 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL501867 VINCRISTINE SULFATE 19532 13295 PSMA7 5688 PROTEASE, DRUGGABLE GENOME inhibitor CARFILZOMIB CARFILZOMIB 19533 13296 ALPL 249 ENZYME, DRUGGABLE GENOME CID 646303 CHEMBL505807 19534 13297 GDF15 9518 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR NSAIDS 15509713 19535 13298 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 405560501 19536 13299 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME HINOKITIOL HINOKITIOL 19538 13300 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 5-FU FLUOROURACIL 12904931 19539 13301 ATAD5 79915 NA (R)-PIA (R)-PIA 19541 13302 EIF4E 1977 DRUGGABLE GENOME LY2275796 19544 13303 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1889140 ROPIVACAINE HYDROCHLORIDE 19545 13304 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME GR-127935 GR-127935 19546 13305 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME RG7388 IDASANUTLIN 19548 13306 POU5F1 5460 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE phenytoin PHENYTOIN 19549 13307 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 178102337 SORAFENIB 19551 13308 TCF7L2 6934 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR hydrochlorothiazide HYDROCHLOROTHIAZIDE 19552 13309 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE MASITINIB MASITINIB 19553 13310 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR DISTAMYCIN 9161031 19554 13311 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GUAIFENESIN GUAIFENESIN 22931300 19555 13312 AIFM1 9131 DRUGGABLE GENOME CYCLOSPORIN A 12787063 19558 13313 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AP-7 AP-7 19559 13314 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DROPERIDOL DROPERIDOL 19560 13315 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Virexxa 19561 13316 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1200745 OXPRENOLOL HYDROCHLORIDE 19562 13317 CGA 1081 DRUGGABLE GENOME, HORMONE ACTIVITY CIS-DIAMMINEDICHLOROPLATINUM 6181870 19563 13318 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PF-562271 PF-00562271 19564 13319 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 alprazolam ALPRAZOLAM 32112986 19566 13320 BAZ2B 29994 NA N-2-NAPHTHYLIMIDODICARBONIMIDIC DIAMIDE CHEMBL43078 19567 13321 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL FLUDIAZEPAM FLUDIAZEPAM 19569 13322 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650384 IMIPRAMINE 19570 13323 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME NS1 27820802 19571 13324 ATAD5 79915 NA CGP-60474 CHEMBL300389 19573 13325 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 REL-CISAPRIDE REL-CISAPRIDE 22931300 19575 13326 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Bortezomib BORTEZOMIB 28151717 19576 13327 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NSC-69187 CHEMBL19954 19578 13328 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE XL820 19579 13329 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1201165 QUINESTROL 19580 13330 TNNC1 7134 DRUGGABLE GENOME LEVOSIMENDAN LEVOSIMENDAN 19581 13331 TUBB2A 7280 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 19583 13332 MPHOSPH8 54737 NA CEFOTAXIME SODIUM CEFOTAXIME SODIUM 19587 13333 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-640556 CHEMBL1983317 21074425 19591 13334 FAAH 2166 ENZYME, DRUGGABLE GENOME Pyrrolidinyl urea derivative 1 19592 13335 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651630 19593 13336 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650697 19595 13337 MAPT 4137 DRUGGABLE GENOME LY-83583 CHEMBL312487 19597 13338 MAPT 4137 DRUGGABLE GENOME PURPURIN PURPURIN 19598 13339 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON BETA 19599 13340 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MK-8745 22293494 19600 13341 RRM2B 50484 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL1096882 FLUDARABINE PHOSPHATE 19602 13342 EPRS1 2058 DRUGGABLE GENOME, ENZYME HT-100 HALOFUGINONE 19603 13343 CD55 1604 DRUGGABLE GENOME, CELL SURFACE PAT-SC1 19604 13344 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID27744724-Compound-10 19606 13345 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE VALPROIC ACID 9098922 19607 13346 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor XL228 XL-228 19608 13347 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE agonist CHEMBL1201717 MECASERMIN RINFABATE 19609 13348 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME BITHIONOL BITHIONOL 19610 13349 DUOX2 50506 TRANSPORTER, ENZYME, DRUGGABLE GENOME, CELL SURFACE inhibitor 363894227 19611 13350 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2218894 FLUVASTATIN SODIUM 19612 13351 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CURCUMIN CURCUMIN 25753330 19613 13352 NOS1 4842 DRUGGABLE GENOME, ENZYME CLARITHROMYCIN CLARITHROMYCIN 14730107 19614 13353 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR NIFEDIPINE NIFEDIPINE 19615 13354 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME NSC-228155 CHEMBL505670 19616 13355 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DIOXYBENZONE DIOXYBENZONE 19618 13356 HSPA4 3308 NA CYTARABINE CYTARABINE 12530536 19619 13357 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR E1501 E1501 19620 13358 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417995 CHEMBL1439833 19622 13359 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE AOD9604 19623 13360 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DOVITINIB DOVITINIB 19624 13361 GMNN 51053 DRUGGABLE GENOME SJ000147784 CHEMBL590186 19625 13362 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1201120 REMIFENTANIL HYDROCHLORIDE 19626 13363 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE DEOXYURIDINE MONOPHOSPHATE DEOXYURIDINE MONOPHOSPHATE 6434741 19627 13364 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 249565596 FILGOTINIB 19628 13365 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 10-(4-PYRIDYL)CAMPTOTHECIN HCL CHEMBL1762594 21333532 19629 13366 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor 178101880 19631 13367 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE SP-600125 SP-600125 19632 13368 UGT2B10 7365 DRUGGABLE GENOME nicotine NICOTINE 18300939,17909004,24192532 19634 13369 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR EI1 28135235 19635 13370 MAPT 4137 DRUGGABLE GENOME PD-404182 CHEMBL595227 19637 13371 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ADL5945 BEVENOPRAN 19639 13372 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME hmg coa reductase inhibitors 19641 13373 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator CHEMBL1201414 TINZAPARIN SODIUM 19643 13374 ACP5 54 ENZYME, DRUGGABLE GENOME STREPTOZOTOCIN STREPTOZOCIN 14640894 19645 13375 POLI 11201 DNA REPAIR CHARTREUSIN CHARTREUSIN 19646 13376 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL454 BUTALBITAL 19647 13377 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE DACOMITINIB DACOMITINIB 19651 13378 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AKB-6548 VADADUSTAT 19653 13379 RGS4 5999 DRUGGABLE GENOME inhibitor 252827379 19654 13380 ABCC9 10060 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER allosteric modulator 252827466 19655 13381 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ARQ-501 LAPACHONE 19656 13382 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE carbidopa CARBIDOPA 12083967 19657 13383 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Aminotriazolopyridine derivative 1 19659 13384 ST14 6768 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 252166696 19660 13385 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE DASATINIB DASATINIB 26703895,29133777 19661 13386 COL15A1 1306 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 19664 13387 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 404859109 19666 13388 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR cabozantinib CABOZANTINIB 27370605 19669 13389 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IPA-3 CHEMBL472940 19670 13390 PTGS1 5742 ENZYME, DRUGGABLE GENOME EXO-230 24303153 19671 13391 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1558 PRAZOSIN HYDROCHLORIDE 19672 13392 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR BML-210 CHEMBL324053 16921367 19673 13393 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME AMG 386 19675 13394 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHOSALONE PHOSALONE 19676 13395 KDM4A 9682 DRUGGABLE GENOME, ENZYME GLICLAZIDE GLICLAZIDE 19679 13396 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOMATINE TOMATINE 19682 13397 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLOROPHACINONE CHLOROPHACINONE 19685 13398 TPM3 7170 KINASE, CLINICALLY ACTIONABLE EPINEPHRINE EPINEPHRINE 18172836 19687 13399 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Vinorelbine VINORELBINE 27992451,24742739 19688 13400 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 223366128 GALUNISERTIB 19689 13401 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-711237 CHEMBL408732 19691 13402 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER AV 133 19692 13403 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ENDOSULFAN SULFATE ENDOSULFAN SULFATE 19693 13404 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125840 CHEMBL475813 19696 13405 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE CVBT-141B 19699 13406 MAPT 4137 DRUGGABLE GENOME GNF-PF-372 CHEMBL580155 19700 13407 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME CER-522 19701 13408 RAPGEF3 10411 ENZYME IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 19703 13409 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE DINOPROSTONE DINOPROSTONE 19704 13410 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ORTHOTOLIDINE ORTHOTOLIDINE 19705 13411 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME 681640 CHEMBL379975 19710 13412 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE 2,2-dimethylbenzopyran derivative 2 19713 13413 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 187051843 LASOFOXIFENE 19714 13414 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PHENOBARBITAL PHENOBARBITAL 16928449 19716 13415 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Phthalazine ketone derivative 3 19717 13416 GJA1 2697 ION CHANNEL CARVEDILOL CARVEDILOL 16448880 19718 13417 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PROPACHLOR PROPACHLOR 19719 13418 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PMID28460551-Compound-1 19720 13419 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32f 19721 13420 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor CHEMBL494089 GSK-690693 19722 13421 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A1 19723 13422 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME agonist 178101632 FILGRASTIM 19724 13423 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME TCMDC-125758 CHEMBL546797 19725 13424 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1200418 DOBUTAMINE HYDROCHLORIDE 19727 13425 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649656 19729 13426 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SIROLIMUS SIROLIMUS 19730 13427 PTGS1 5742 ENZYME, DRUGGABLE GENOME ASPIRIN ASPIRIN 19732 13428 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE rasburicase RASBURICASE 17387701,23989394,20196170,28370399,23209099,24787449,27119769,12075750,24372186,20701405,12942574,23860572,29290749,24750455,2019023,25988058,22573495,26033222,9369411,19654083,16204390,22190578,18561168,22015451,24915143,25115783 19733 13429 PRKCH 5583 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL3545332 CEP-2563 19734 13430 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME FLUOXASTROBIN FLUOXASTROBIN 19736 13431 KDM4A 9682 DRUGGABLE GENOME, ENZYME ENALAPRIL MALEATE ENALAPRIL MALEATE 19737 13432 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 2-MERCAPTOBENZOTHIAZOLE 2-MERCAPTOBENZOTHIAZOLE 19738 13433 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651262 TIFLUADOM 19739 13434 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME THIOLACTOMYCIN THIOLACTOMYCIN 19742 13435 POLI 11201 DNA REPAIR EMODIC ACID EMODIC ACID 19744 13436 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CARMUSTINE CARMUSTINE 22931300 19745 13437 NOS2 4843 DRUGGABLE GENOME, ENZYME Curcumin CURCUMIN 19746 13438 SMN2 6607 DRUGGABLE GENOME 2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE CHEMBL502774 19747 13439 TLR7 51284 DRUGGABLE GENOME IMIQUIMOD IMIQUIMOD 19748 13440 ORM2 5005 DRUGGABLE GENOME docetaxel DOCETAXEL 24619498 19749 13441 SPP1 6696 DRUGGABLE GENOME IMMUNOSUPPRESSANT 15978615 19750 13442 IL17RA 23765 DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 27670766 19751 13443 CXCL8 3576 DRUGGABLE GENOME DICYCLOHEXYLCARBODIIMIDE DICYCLOHEXYLCARBODIIMIDE 19753 13444 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL593430 ATAGABALIN 19754 13445 INPP5D 3635 DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE activator 315661324 ROSIPTOR 19756 13446 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 249565596 FILGOTINIB 19757 13447 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE EP4-R antagonist 19759 13448 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RETINYL ACETATE RETINYL ACETATE 19760 13449 UBE2N 7334 ENZYME, DRUGGABLE GENOME ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 19761 13450 POLB 5423 DNA REPAIR, DRUGGABLE GENOME LIOTHYRONINE SODIUM LIOTHYRONINE SODIUM 19763 13451 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METOPROLOL TARTRATE 19765 13452 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE RG-1530 RG-1530 19766 13453 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor BELINOSTAT BELINOSTAT 19767 13454 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE MTOR KINASE INHIBITOR PP242 21358673 19768 13455 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIHYDROXYBERGAMOTTIN DIHYDROXYBERGAMOTTIN 21393461 19772 13456 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME BORTEZOMIB BORTEZOMIB 24524217 19773 13457 PSMD4 5710 NA inhibitor CHEMBL451887 CARFILZOMIB 19774 13458 TARDBP 23435 TUMOR SUPPRESSOR OLEOYL DOPAMINE OLEOYL DOPAMINE 19775 13459 DGAT1 8694 ENZYME, DRUGGABLE GENOME Hesperetin HESPERETIN 19777 13460 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME AMD-070 MAVORIXAFOR 19780 13461 CES1 1066 DRUGGABLE GENOME, ENZYME 2-oxo-clopidogrel 23275066 19781 13462 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME TW-37 CHEMBL217354 25665005 19783 13463 HNRNPA1 3178 DRUGGABLE GENOME CAMPTOTHECIN CAMPTOTHECIN 22071521 19784 13464 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 4-HYDROXYFLAVONOL CHEMBL272682 19785 13465 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME inhibitor REGORAFENIB REGORAFENIB 19788 13466 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR 6-HYDROXYDOPAMINE 16890350 19789 13467 RGMA 56963 CELL SURFACE, KINASE Elezanumab ELEZANUMAB 19791 13468 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651424 ACETYLCHOLINE 19792 13469 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Beta-phe compound 1 19794 13470 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL408513 BELINOSTAT 19795 13471 AAK1 22848 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME inhibitor 223366123 BARICITINIB 19796 13472 ATXN2 6311 NA MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 19797 13473 RGS4 5999 DRUGGABLE GENOME IODOACETAMIDE IODOACETAMIDE 19798 13474 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR ANTI-VEGF MONOCLONAL ANTIBODY 28103578 19801 13475 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RO-137410 CHEMBL275311 19803 13476 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR (E)-DIBENZYLIDENEACETONE CHEMBL17201 19804 13477 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME TCMDC-123598 CHEMBL547269 19805 13478 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Osimertinib OSIMERTINIB 25870145 19806 13479 GSTM1 2944 DRUGGABLE GENOME, ENZYME NITROGLYCERIN NITROGLYCERIN 2110160 19808 13480 CCR6 1235 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR TRAIL 12176034 19809 13481 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-123951 CHEMBL587849 19810 13482 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE 4SCAR19 and 4SCAR123 19811 13483 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor GIVINOSTAT GIVINOSTAT 19812 13484 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ADJUVANT 10873087,9816327 19813 13485 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Neratinib NERATINIB 20479403,17085664,25948633,26206867,25931286,21325073 19814 13486 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME IMIDACLOPRID IMIDACLOPRID 19815 13487 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TCMDC-123713 CHEMBL586135 19817 13488 SFTPA1 653509 DRUGGABLE GENOME RECOMBINANT HUMAN KERATINOCYTE GROWTH FACTOR 12740217 19818 13489 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SB-681323 DILMAPIMOD 19819 13490 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE LITHOCHOLIC ACID LITHOCHOLIC ACID 19820 13491 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CARBAZOLE CARBAZOLE 19822 13492 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE KU-60019 25870146 19823 13493 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1256 ISOFLURANE 19824 13494 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME bortezomib BORTEZOMIB 22541434 19826 13495 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565834 19828 13496 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Bis-aminopyrimidine derivative 1 19829 13497 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME SSR-128428 19830 13498 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME mipomersen MIPOMERSEN 19831 13499 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ETHOPROPAZINE HYDROCHLORIDE ETHOPROPAZINE HYDROCHLORIDE 19832 13500 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR HAEMATOXYLIN HAEMATOXYLIN 19836 13501 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 363894169 SEPETAPROST 19837 13502 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 178103761 FENOFIBRATE 19838 13503 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE LY-411575 CHEMBL392068 23181502,19443228 19839 13504 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME TESTOSTERONE UNDECANOATE 14555326 19840 13505 FGF1 2246 CLINICALLY ACTIONABLE, GROWTH FACTOR, DRUGGABLE GENOME PENTOSAN POLYSULFATE 19841 13506 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8921389, 2 19842 13507 ALOX15 246 ENZYME, DRUGGABLE GENOME L-755507 L-755507 19843 13508 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VERAPAMIL VERAPAMIL 3566185 19844 13509 MAOB 4129 DRUGGABLE GENOME, ENZYME LEVODOPA LEVODOPA 7867755 19845 13510 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor PKI-587 GEDATOLISIB 19848 13511 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE SNS-314 SNS-314 19849 13512 ATXN2 6311 NA FLUOXETINE HYDROCHLORIDE FLUOXETINE HYDROCHLORIDE 19850 13513 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178103955 RIBOCICLIB 19853 13514 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE GNF-PF-254 CHEMBL461579 19857 13515 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1200724 PSEUDOEPHEDRINE HYDROCHLORIDE 19859 13516 BCHE 590 DRUGGABLE GENOME, ENZYME PMID29757691-Compound-8a 19860 13517 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NU-2058 CHEMBL269881 19861 13518 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME TG02, SB1317 19862 13519 HPRT1 3251 DRUGGABLE GENOME, ENZYME mycophenolic acid 19863 13520 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GNF-PF-5159 CHEMBL1493528 19864 13521 SMN1 6606 DRUGGABLE GENOME DEHYDROVARIABILIN DEHYDROVARIABILIN 19868 13522 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178101952 19869 13523 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Pyrazolo[4,3-c]pyridine derivative 2 19870 13524 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Rivoglitazone RIVOGLITAZONE 19871 13525 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR JNJ-7706621 JNJ-7706621 19876 13526 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-3418 CHEMBL582099 19877 13527 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ANISOTROPINE METHYLBROMIDE 19880 13528 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker 178101078 19881 13529 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20120264760C88 19883 13530 XRCC1 7515 CLINICALLY ACTIONABLE CISPLATIN CISPLATIN 16875718 19884 13531 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AZINPHOS-ETHYL AZINPHOS-ETHYL 19885 13532 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE Ivacaftor IVACAFTOR 19887 13533 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Temsirolimus TEMSIROLIMUS 27016228 19888 13534 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR METHYLISOTHIOCYANATE METHYLISOTHIOCYANATE 19889 13535 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 178103533 DEXTROTHYROXINE 19890 13536 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Pyrimidine derivative 21 19892 13537 DNER 92737 NA Isoxazole-based bicyclic compound 6 19893 13538 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRICLOCARBAN TRICLOCARBAN 19895 13539 POLK 51426 DNA REPAIR, ENZYME LEVONORDEFRIN LEVONORDEFRIN 19896 13540 CALU 813 DRUGGABLE GENOME acenocoumarol ACENOCOUMAROL 17596133,29479633 19898 13541 BAZ2B 29994 NA PYRAZINOIC ACID PYRAZINOIC ACID 19900 13542 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME brexpiprazole BREXPIPRAZOLE 19901 13543 CBX1 10951 NA RALOXIFENE RALOXIFENE 19902 13544 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME IODOACETAMIDE IODOACETAMIDE 19904 13545 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 252827523 CEBRANOPADOL 19906 13546 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Fused aromatic compound 1 19907 13547 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR GO-6976 GO-6976 19910 13548 GMNN 51053 DRUGGABLE GENOME VANDETANIB VANDETANIB 19911 13549 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE QUERCETIN QUERCETIN 22212721 19912 13550 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME BMS-345541 BMS-345541 19913 13551 TOP2B 7155 DRUGGABLE GENOME, ENZYME doxorubicin DOXORUBICIN 21048526 19914 13552 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ATROPINE ATROPINE 15315164 19918 13553 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROGESTIN PROGESTERONE 10713180 19920 13554 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417309 CHEMBL1341830 19921 13555 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER MMV666022 CHEMBL599100 19924 13556 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME MK2206 MK-2206 21289267 19925 13557 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 315661176 19926 13558 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Ambrisentan AMBRISENTAN 19927 13559 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME QUAZEPAM QUAZEPAM 19928 13560 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX modulator CHEMBL146506 MOFAROTENE 19930 13561 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-2947 CHEMBL581677 19932 13562 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE ADOZELESIN ADOZELESIN 10933811 19933 13563 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SB-203186 CHEMBL1255781 19934 13564 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE MINODRONATE 19935 13565 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR SJ000044511 CHEMBL592124 19937 13566 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME DIMIRACETAM DIMIRACETAM 19938 13567 NQO2 4835 DRUGGABLE GENOME, ENZYME NSC-640353 CHEMBL1288253 21074425 19940 13568 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME VEGLIN 19946 13569 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME ALPHA INTERFERON CETUXIMAB 2016633 19947 13570 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TS-1 24982373 19949 13571 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Busulfan BUSULFAN 19953 13572 HBB 3043 DRUGGABLE GENOME, ENZYME 5-FLUOROURIDINE CHEMBL54918 19954 13573 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE TCN-P 19955 13574 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor BGJ398 INFIGRATINIB 19956 13575 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650385 IMMEPIP 19957 13576 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALPHOSTIN C CALPHOSTIN C 19958 13577 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME DESOXIMETASONE DESOXIMETASONE 19959 13578 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ROSMARINIC ACID ROSMARINIC ACID 19960 13579 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Ascorbic Acid 19962 13580 NCL 4691 NA Itarnafloxin QUARFLOXIN 21455236 19963 13581 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR CRA-024781 ABEXINOSTAT 19964 13582 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor 315661124 ERDAFITINIB 19967 13583 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ARRY-614 PEXMETINIB 19968 13584 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE QUERCETIN QUERCETIN 16149735 19969 13585 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 23622981 19970 13586 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32f 19971 13587 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Treprostinil TREPROSTINIL 19972 13588 CGA 1081 DRUGGABLE GENOME, HORMONE ACTIVITY TUMOR NECROSIS FACTOR 9764349,10788437 19974 13589 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor LAPATINIB LAPATINIB 19975 13590 MTTP 4547 DRUGGABLE GENOME LOMITAPIDE LOMITAPIDE 19978 13591 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW300660X GW300660X 19979 13592 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR inhibitor ZD4054 19980 13593 DHFR 1719 DRUGGABLE GENOME, ENZYME inhibitor 178101517 METHOTREXATE 19981 13594 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Quinolinyl pyrazinyl urea derivative 1 19984 13595 GMNN 51053 DRUGGABLE GENOME NSC-695801 CHEMBL461193 19985 13596 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102338 SU-014813 19986 13597 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR L-PHENYLALANINE PHENYLALANINE 19987 13598 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PYRITHIONE SODIUM PYRITHIONE SODIUM 19988 13599 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX TAZAROTENE TAZAROTENE 19989 13600 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GW1929 CHEMBL434063 19990 13601 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (R)-PINOCEMBRIN (R)-PINOCEMBRIN 19991 13602 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME DEMECARIUM BROMIDE 19992 13603 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME DIFLUBENZURON DIFLUBENZURON 19994 13604 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PRAVASTATIN PRAVASTATIN 17615423 19995 13605 PDE8B 8622 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL628 PENTOXIFYLLINE 19996 13606 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200578 THEOPHYLLINE SODIUM GLYCINATE 19998 13607 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Vapitadine VAPITADINE 19999 13608 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545298 AZD-6918 20000 13609 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE DNDI1417484 CHEMBL1308677 20001 13610 CBX1 10951 NA TYRPHOSTIN AG-835 CHEMBL261557 20004 13611 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 187051799 DACINOSTAT 20005 13612 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL41355 EZOGABINE 20008 13613 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME BMS-387032 BMS-387032 20010 13614 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE DIGOXIN DIGOXIN 20011 13615 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Rosiglitazone + metformin 20013 13616 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Olaparib OLAPARIB 26546619,20609467,27454287,25193512,25366685,22172724 20014 13617 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL967 TEMAZEPAM 20015 13618 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GNF-PF-2267 CHEMBL601764 20016 13619 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PD-404182 CHEMBL595227 20017 13620 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NIACIN NIACIN 22931300 20018 13621 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR CORTISOL HYDROCORTISONE 7895901 20019 13622 MPHOSPH8 54737 NA CAPSAZEPINE CAPSAZEPINE 20020 13623 XDH 7498 DRUGGABLE GENOME, ENZYME inhibitor 178103401 ALLOPURINOL 20021 13624 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE VITAMIN B2 VITAMIN B2 20022 13625 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME STREPTOZOTOCIN STREPTOZOCIN 7664670 20023 13626 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-15 20025 13627 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135651082 20026 13628 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME OXYTETRACYCLINE OXYTETRACYCLINE 20028 13629 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR OXCARBAZEPINE OXCARBAZEPINE 20030 13630 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL1742994 BRENTUXIMAB VEDOTIN 20031 13631 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE RUCAPARIB RUCAPARIB 20032 13632 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Tolazamide TOLAZAMIDE 20033 13633 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PRACINOSTAT PRACINOSTAT 20034 13634 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-asCEBP-1HPE 20035 13635 LNPEP 4012 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, TRANSPORTER, PROTEASE US10059720, Example 84 20036 13636 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051823 20037 13637 IL1A 3552 CELL SURFACE, DRUGGABLE GENOME RILONACEPT RILONACEPT 20038 13638 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AZILSARTAN AZILSARTAN 20039 13639 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DITHIAZANINE IODIDE DITHIAZANINE IODIDE 20042 13640 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME NSC-19063 CHEMBL1310138 20043 13641 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME AMATUXIMAB AMATUXIMAB 20044 13642 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE GENISTEIN GENISTEIN 12124395 20045 13643 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE CEDIRANIB CEDIRANIB 20046 13644 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE VX-680 TOZASERTIB 20047 13645 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME SODIUM PHENYLBUTYRATE 16246228 20048 13646 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL451 CHLORDIAZEPOXIDE 20049 13647 TOP2B 7155 DRUGGABLE GENOME, ENZYME GPX-150D 20050 13648 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TOLFENAMIC ACID TOLFENAMIC ACID 20051 13649 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR 1-hydroxyl-3,5-bis(4-hydroxylstyryl)benzene derivative 2 20052 13650 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME LINIFANIB LINIFANIB 20057 13651 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TAZOBACTAM SODIUM TAZOBACTAM SODIUM 20058 13652 CSNK2A2 1459 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME, TRANSCRIPTION FACTOR inhibitor 249565806 SILMITASERTIB 20059 13653 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL nimodipine NIMODIPINE 19205682 20060 13654 F5 2153 DRUGGABLE GENOME DROTRECOGIN ALFA 20061 13655 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE RO4929097 RG-4733 27154916 20062 13656 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE DICHLOROPHEN DICHLOROPHEN 20063 13657 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME antagonist 178103271 20064 13658 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE INDOCATE INDOCATE 20067 13659 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist CHEMBL3545294 DAROLUTAMIDE 20068 13660 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Pyrazolo[1,5-a]-1,3,5-triazine derivative 1 20069 13661 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FISETIN FISETIN 20070 13662 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIAZEPAM DIAZEPAM 20072 13663 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME AZD-1775 ADAVOSERTIB 20073 13664 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR antagonist 381118897 20074 13665 HEBP1 50865 DRUGGABLE GENOME Benzo[d]oxazole derivative 2 20075 13666 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3544988 DAPRODUSTAT 20076 13667 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CLIOQUINOL CLIOQUINOL 20077 13668 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME ROTENONE ROTENONE 16680159 20078 13669 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME trametinib TRAMETINIB 20079 13670 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME FLUMETHASONE PIVALATE 20081 13671 TPM3 7170 KINASE, CLINICALLY ACTIONABLE AMINOGLYCOSIDES 15164360 20082 13672 KCNS3 3790 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL113461 TEDISAMIL 20083 13673 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor GDC-0941 PICTILISIB 20087 13674 GMNN 51053 DRUGGABLE GENOME SANTIN SANTIN 20088 13675 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE SAMIDOPRHAN 20089 13676 IL1B 3553 KINASE, DRUGGABLE GENOME lansoprazole LANSOPRAZOLE 16815316,21054464,14638340 20091 13677 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE TAK-715 TAK-715 20092 13678 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TENIPOSIDE TENIPOSIDE 9426516 20093 13679 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MIANSERIN HYDROCHLORIDE MIANSERIN HYDROCHLORIDE 20095 13680 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 249565844 20096 13681 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DNDI1417309 CHEMBL1341830 20099 13682 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody 252166509 SERIBANTUMAB 20102 13683 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME AG-024322 AG-24322 20103 13684 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3545322 PANULISIB 20104 13685 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor HESPERADIN HESPERADIN 19035792 20108 13686 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 135649930 TAMIBAROTENE 20109 13687 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR inhibitor 178103606 20110 13688 TXNRD1 7296 DRUGGABLE GENOME 4-aryl quinol derivative 2 20112 13689 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE Cisplatin CISPLATIN 22753594 20114 13690 SMN2 6607 DRUGGABLE GENOME DNDI1417548 CHEMBL2094789 20115 13691 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL2107339 ESMIRTAZAPINE MALEATE 20118 13692 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR BITHIONOL BITHIONOL 20120 13693 RAPGEF3 10411 ENZYME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 20121 13694 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 249565874 20125 13695 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Imatinib IMATINIB 20127 13696 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PROTOPORPHYRIN DISODIUM PROTOPORPHYRIN DISODIUM 20128 13697 NAPRT 93100 NA GNE-617 24097869 20129 13698 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL1200993 GALLAMINE TRIETHIODIDE 20130 13699 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 1 20131 13700 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE THALIDOMIDE THALIDOMIDE 15457133 20133 13701 SMN2 6607 DRUGGABLE GENOME N-HISTIDYL-2-AMINONAPHTHALENE (BETANA) N-HISTIDYL-2-AMINONAPHTHALENE (BETANA) 20135 13702 GLS 2744 ENZYME PURPUROGALLIN PURPUROGALLIN 20137 13703 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME JNJ-7706621 JNJ-7706621 20138 13704 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BETAMETHASONE BUTYRATE PROPIONATE BETAMETHASONE BUTYRATE PROPIONATE 20139 13705 ESRRG 2104 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650300 GENISTEIN 20140 13706 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GW0742 CHEMBL38508 20142 13707 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME TAE226 26090892 20143 13708 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE Propylthiouracil PROPYLTHIOURACIL 20144 13709 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650023 BRL-15,572 20145 13710 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Panitumumab PANITUMUMAB 26644315 20147 13711 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE THIOMERSAL THIMEROSAL 20148 13712 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME MG-132 MG-132 24321833 20149 13713 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL944 CHLOROPROCAINE HYDROCHLORIDE 20150 13714 SERPINA6 866 DRUGGABLE GENOME, PROTEASE INHIBITOR CICLESONIDE CICLESONIDE 20153 13715 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ERLOTINIB ERLOTINIB 20154 13716 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME clozapine CLOZAPINE 9587740,26876947,2222133 20155 13717 ABAT 18 DRUGGABLE GENOME, ENZYME DIVALPROEX SODIUM 20158 13718 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TARENFLURBIL TARENFLURBIL 20159 13719 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ACTINONIN ACTINONIN 20160 13720 SLC22A3 6581 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER catecholamines 20859243 20161 13721 HDAC11 79885 DRUGGABLE GENOME, ENZYME PHENYLBUTANOIC ACID PHENYLBUTANOIC ACID 24044874 20162 13722 PARP3 10039 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR inhibitor 252166678 20163 13723 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE MSC2363318A MSC-2363318A 20164 13724 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME MOCETINOSTAT MOCETINOSTAT 23829483,26287310 20165 13725 ENPP2 5168 ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING NSC-12188 CHEMBL1089321 20349977 20166 13726 TGFB2 7042 GROWTH FACTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BELAGENPUMATUCEL-L BELAGENPUMATUCEL-L 20168 13727 ALOX15 246 ENZYME, DRUGGABLE GENOME inhibitor 252827409 20169 13728 S100A8 6279 DRUGGABLE GENOME, KINASE, ENZYME MTX METHOTREXATE 14722212 20170 13729 POLI 11201 DNA REPAIR AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 20173 13730 GMNN 51053 DRUGGABLE GENOME CLOFENOXYDE CLOFENOXYDE 20175 13731 PDE4A 5141 DRUGGABLE GENOME, ENZYME DIPYRIDAMOLE DIPYRIDAMOLE 20176 13732 BAZ2B 29994 NA GNF-PF-5149 CHEMBL600309 20177 13733 TNFRSF1A 7132 CELL SURFACE, DRUGGABLE GENOME UVB 9754576 20178 13734 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RABEPRAZOLE SODIUM RABEPRAZOLE SODIUM 20179 13735 PEBP4 157310 DRUGGABLE GENOME methylphenidate METHYLPHENIDATE 29382897 20180 13736 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL190 THEOPHYLLINE 20181 13737 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32m 20182 13738 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR CENISERTIB CENISERTIB 20184 13739 EDAR 10913 DRUGGABLE GENOME 178102765 20186 13740 MAOB 4129 DRUGGABLE GENOME, ENZYME Tetra-hydro-oxazolopyridine derivative 2 20190 13741 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TAK-491 AZILSARTAN MEDOXOMIL 20191 13742 BAZ2B 29994 NA GNF-PF-2671 CHEMBL578878 20192 13743 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW809897X GW809897X 20193 13744 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DNDI1417523 CHEMBL598663 20194 13745 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME 2-AMINO-ANTHRAQUINONE CHEMBL84685 20195 13746 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CYCLOOXYGENASE INHIBITOR 2054945 20197 13747 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651165 20198 13748 NDUFA3 4696 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 20199 13749 POLK 51426 DNA REPAIR, ENZYME MORIN MORIN 20200 13750 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME DNDI1417467 CHEMBL1997335 20204 13751 APOBEC3B 9582 ENZYME corticosteroids 30697902 20206 13752 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200819 ARTICAINE HYDROCHLORIDE 20211 13753 NOS1 4842 DRUGGABLE GENOME, ENZYME TESTOSTERONE TESTOSTERONE 7515189 20213 13754 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME allosteric modulator 310264717 20214 13755 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 135651725 20215 13756 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME DISULFIRAM DISULFIRAM 20216 13757 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PMID29130358-Compound-Figure16(9a) 20217 13758 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLEMASTINE CLEMASTINE 22931300 20218 13759 TOP2B 7155 DRUGGABLE GENOME, ENZYME Dexrazoxane DEXRAZOXANE 20220 13760 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PREDNICARBATE PREDNICARBATE 20221 13761 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 318164813 20222 13762 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamate derivative 14 20223 13763 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME CERITINIB CERITINIB 23837797 20224 13764 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME LAM-001 20227 13765 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL NITRAZEPAM NITRAZEPAM 20228 13766 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GSK2126458 OMIPALISIB 20229 13767 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE MLN0128 SAPANISERTIB 26272063,27974663 20233 13768 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3,7-DIMETHOXYFLAVONE 3,7-DIMETHOXYFLAVONE 20234 13769 GET1 7485 NA methylphenidate METHYLPHENIDATE 29382897 20235 13770 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE UROKINASE UROKINASE 20237 13771 POLI 11201 DNA REPAIR GAMOLENIC ACID GAMOLENIC ACID 20238 13772 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GATIFLOXACIN GATIFLOXACIN 20240 13773 MAPT 4137 DRUGGABLE GENOME GEFITINIB GEFITINIB 20242 13774 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL DSP-2230 DSP-2230 20243 13775 LPAR2 9170 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 178100857 20244 13776 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE atenolol ATENOLOL 16027735 20245 13777 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2336071 SIPONIMOD 20246 13778 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Desoxycorticosterone Pivalate 20247 13779 MVK 4598 KINASE, ENZYME alendronate ALENDRONIC ACID 25223561 20248 13780 RUNX3 864 TRANSCRIPTION FACTOR LEUCOVORIN LEUCOVORIN 17372756 20249 13781 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 328083470 20250 13782 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 4 20252 13783 TBC1D32 221322 KINASE Bisphosphonates 20254 13784 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CISPLATIN CISPLATIN 20255 13785 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 178102323 MLN-8054 20256 13786 DHFR 1719 DRUGGABLE GENOME, ENZYME FOLIC ACID 10956384 20257 13787 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME CEPHALOSPORINS 8774083 20259 13788 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ESTROGEN ESTROGEN 20260 13789 LTBR 4055 DRUGGABLE GENOME 178101763 20261 13790 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100764 20262 13791 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 336446940 20263 13792 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor GSK2126458 OMIPALISIB 20266 13793 POLB 5423 DNA REPAIR, DRUGGABLE GENOME METHACYCLINE HYDROCHLORIDE METHACYCLINE HYDROCHLORIDE 20267 13794 SEM1 7979 NA inhibitor CHEMBL451887 CARFILZOMIB 20268 13795 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-31 20269 13796 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-348401 CHEMBL515505 20270 13797 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYCLOHEXIMIDE CYCLOHEXIMIDE 20272 13798 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR THEONELLASTEROL F THEONELLASTEROL F 21428459 20273 13799 TSPO 706 DRUGGABLE GENOME PMID27599163-Compound-52 20274 13800 IFNG 3458 DRUGGABLE GENOME MONOCLONAL ANTIBODY 17-1A 2121912 20275 13801 TPBG 7162 CELL SURFACE, DRUGGABLE GENOME PF-06263507 PF-06263507 20276 13802 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor CHEMBL3137349 BOCOCIZUMAB 20277 13803 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GSK321 26436839 20279 13804 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 178100746 20280 13805 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE SP-600125 SP-600125 20281 13806 UGT2B7 7364 DRUGGABLE GENOME morphine MORPHINE 17724700,25340733,24703092,16580900,12185559,28063968,31607718 20282 13807 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR 1-hydroxyl-3,5-bis(4-hydroxylstyryl)benzene derivative 4 20283 13808 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME 4-(4-AMINOPHENYL)BUTANOIC ACID CHEMBL1650245 24044874 20284 13809 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist,antagonist 135649800 AFIMOXIFENE 20285 13810 THY1 7070 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE HEL 6186895 20287 13811 RBP4 5950 DRUGGABLE GENOME FENRETINIDE FENRETINIDE 21591606 20288 13812 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME PEXIDARTINIB PEXIDARTINIB 28759044 20289 13813 ATAD5 79915 NA CANTHARIDIC_ACID CANTHARIDIC_ACID 20290 13814 GMNN 51053 DRUGGABLE GENOME DIACYLGLYCEROL KINASE INHIBITOR II DIACYLGLYCEROL KINASE INHIBITOR II 20291 13815 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRYPTANTHRIN TRYPTANTHRIN 20299 13816 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Vandetanib VANDETANIB 25910950 20300 13817 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-693571 CHEMBL1287983 20301 13818 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GW441756X GW441756X 20302 13819 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME KC706 20303 13820 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR IBI-20089 20305 13821 PDE4B 5142 DRUGGABLE GENOME, ENZYME Piclamilast PICLAMILAST 20306 13822 RAB9A 9367 ENZYME, DRUGGABLE GENOME 3,6-DIPHENYL-[1,2,4,5]TETRAZINE CHEMBL17784 20309 13823 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LAROPIPRANT LAROPIPRANT 20310 13824 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE CEFOPERAZONE CEFOPERAZONE 22166395 20311 13825 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL450 METHARBITAL 20314 13826 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME MB-CART20.1 20316 13827 KAT2B 8850 ENZYME, DRUGGABLE GENOME ANACARDIC ACID 20655754 20317 13828 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER irinotecan IRINOTECAN 27845419 20319 13829 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR US10174026, Example 2 20320 13830 TSPO 706 DRUGGABLE GENOME Chlormezanone CHLORMEZANONE 20322 13831 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX A-443654 A-443654 20324 13832 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALPHA-TERTHIENYL ALPHA-TERTHIENYL 20326 13833 CYP27B1 1594 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 252827515 CHEMBL255088 20328 13834 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE Interferon alfa-n1 20329 13835 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE FULVESTRANT FULVESTRANT 27252418 20331 13836 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME KH064 20333 13837 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 384403646 20335 13838 ITPR3 3710 ION CHANNEL, DRUGGABLE GENOME activator 135652731 20339 13839 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SJ000089001 CHEMBL591618 20341 13840 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TOZASERTIB TOZASERTIB 20345 13841 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME CYC-116 CYC-116 20347 13842 POLK 51426 DNA REPAIR, ENZYME 2-AMINOPHENOXAZINONE CHEMBL146710 20348 13843 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ARACHIDONOYL DOPAMINE ARACHIDONOYL DOPAMINE 20352 13844 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 363894185 20354 13845 SIRT5 23408 ENZYME GNF-PF-1720 CHEMBL578329 20355 13846 MARCKSL1 65108 KINASE PMA 8596017 20356 13847 CES1 1066 DRUGGABLE GENOME, ENZYME Eldacimibe ELDACIMIBE 20357 13848 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME TCMDC-123713 CHEMBL586135 20360 13849 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME dolutegravir DOLUTEGRAVIR 28858994 20361 13850 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL377300 BRIVANIB 20362 13851 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650226 ETHYLKETOCYCLAZOCINE 20363 13852 PCSK6 5046 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE inhibitor 178103178 20369 13853 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SANGUINARIUM SANGUINARIUM 20370 13854 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BKM120 BUPARLISIB 20371 13855 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR VIGABATRIN VIGABATRIN 20372 13856 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor AZD4547 20373 13857 GAA 2548 DRUGGABLE GENOME, ENZYME CASTANOSPERMINE CASTANOSPERMINE 20374 13858 RGS4 5999 DRUGGABLE GENOME 3,4-METHYLENEDIOXYB-NITROSTYRENE CHEMBL596380 20375 13859 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR NORETHISTERONE ACETATE 12385861 20376 13860 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME 2,3,4,4'-TETRAMETHOXYBIPHENYL 2,3,4,4'-TETRAMETHOXYBIPHENYL 20378 13861 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FF-284 25169980 20380 13862 RACGAP1 29127 NA EQUILIN EQUILIN 20382 13863 MAPT 4137 DRUGGABLE GENOME MYRICETIN MYRICETIN 20384 13864 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (R,S)-IFENPRODIL (R,S)-IFENPRODIL 20385 13865 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME SPH-1285 20386 13866 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NALOXONE HYDROCHLORIDE NALOXONE HYDROCHLORIDE 20387 13867 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker 53801055 20388 13868 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antibody MDX-1105 BMS-936559 20389 13869 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-15 20390 13870 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME IFN 7507709,8081556 20391 13871 BAZ2B 29994 NA IDEBENONE IDEBENONE 20393 13872 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE allosteric modulator 178102433 20394 13873 CBX1 10951 NA APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 20397 13874 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER Sulfinpyrazone SULFINPYRAZONE 20398 13875 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-725317 CHEMBL260417 20399 13876 RGS4 5999 DRUGGABLE GENOME NS-398 NS-398 20400 13877 MKNK1 8569 SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 178101606 DORSOMORPHIN 20401 13878 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE NAQUOTINIB NAQUOTINIB 29386539 20402 13879 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROMETHAZINE PROMETHAZINE 20403 13880 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME APOCIDEINE APOCIDEINE 20404 13881 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IDEBENONE IDEBENONE 20406 13882 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SANGUINARINE SULFATE SANGUINARINE SULFATE 20408 13883 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR FISPEMIFENE FISPEMIFENE 20410 13884 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE BCG BCG VACCINE 11441103,15213127 20411 13885 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MC-3001 20413 13886 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE vitamin c 11418378,1138591 20414 13887 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL552212 LEXIBULIN 20415 13888 HTT 3064 DRUGGABLE GENOME DITHIAZANINE DITHIAZANINE 20416 13889 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME RG-1530 RG-1530 20417 13890 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR letrozole LETROZOLE 26536870 20418 13891 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MOMETASONE FUROATE MOMETASONE FUROATE 20419 13892 USP1 7398 DNA REPAIR, PROTEASE, ENZYME OLEIC ACID OLEIC ACID 20420 13893 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NARATRIPTAN NARATRIPTAN 20421 13894 PDF 64146 DRUGGABLE GENOME Chlorproguanil CHLORPROGUANIL 20422 13895 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR CG-0070 20425 13896 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME THALIDOMIDE THALIDOMIDE 12515619 20426 13897 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE FILGRASTIM FILGRASTIM 16549824 20427 13898 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL2140408 AMG-900 20428 13899 BAZ2B 29994 NA HESPERIDIN HESPERIDIN 20432 13900 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ERGOCRISTINE ERGOCRISTINE 20433 13901 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649684 20434 13902 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650005 20435 13903 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 8-MOP METHOXSALEN 17003103 20436 13904 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33e 20437 13905 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE PMID27539678-Compound-8 20439 13906 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TOLTERODINE TOLTERODINE 20440 13907 BAZ2B 29994 NA AG-527 CHEMBL258767 20441 13908 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE LINIFANIB LINIFANIB 20442 13909 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 acetaminophen ACETAMINOPHEN 26049587,11866476,9548799 20444 13910 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE CHEMBL457504 20445 13911 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Bexarotene BEXAROTENE 20446 13912 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 249565718 CHEMBL573107 20447 13913 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME CANTHARIDIC_ACID CANTHARIDIC_ACID 20448 13914 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 363894161 20450 13915 POLK 51426 DNA REPAIR, ENZYME GAMOLENIC ACID GAMOLENIC ACID 20452 13916 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PHENOBARBITAL PHENOBARBITAL 22931300 20453 13917 XDH 7498 DRUGGABLE GENOME, ENZYME Fused heterocyclic compound 7 20454 13918 ATAD5 79915 NA TCMDC-123808 CHEMBL546493 20456 13919 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-60340 CHEMBL1534034 20457 13920 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME PMID27998201-Compound-19 20458 13921 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 20460 13922 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE VELIPARIB VELIPARIB 20461 13923 CD3D 915 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE CATUMAXOMAB CATUMAXOMAB 20462 13924 POLI 11201 DNA REPAIR NAVITOCLAX NAVITOCLAX 20463 13925 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL blocker 178100875 PICROTOXIN 20464 13926 RACGAP1 29127 NA MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 20465 13927 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE 178101323 20466 13928 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200382 BEPRIDIL HYDROCHLORIDE 20467 13929 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER ETOPOSIDE ETOPOSIDE 9472114,7671247 20469 13930 TSPO 706 DRUGGABLE GENOME Imidazopyridine derivative 1 20470 13931 ABCB4 5244 TRANSPORTER, DRUGGABLE GENOME, ENZYME, ABC TRANSPORTER Ortataxel ORTATAXEL 20471 13932 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-21 20475 13933 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME KO-143 CHEMBL488910 24304387,22266779,24611893 20476 13934 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 363894209 PAMAPIMOD 20479 13935 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ALKS 33 20480 13936 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ILORASERTIB ILORASERTIB 20482 13937 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Isoflavone derivative 9 20483 13938 PTGS1 5742 ENZYME, DRUGGABLE GENOME IBUPROFEN IBUPROFEN 20485 13939 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME SOTRASTAURIN SOTRASTAURIN 20487 13940 MGAT2 4247 ENZYME Dihydropyrimidinone derivative 4 20488 13941 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor AMUVATINIB AMUVATINIB 20489 13942 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE CHEMBL457504 20493 13943 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 354702223 NECROSTATIN 20497 13944 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX PARTHENOLIDE PARTHENOLIDE 25190466 20498 13945 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ELLAGIC ACID ELLAGIC ACID 20499 13946 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyridopyrimidinone derivative 3 20500 13947 SLC38A1 81539 TRANSPORTER 178101263 20501 13948 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PROMAZINE PROMAZINE 20502 13949 FFAR4 338557 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102223 20503 13950 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE PD-0166285 PD-0166285 20504 13951 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PYRAZOLOACRIDINE PYRAZOLOACRIDINE 19501511 20505 13952 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor PD 0332991 20506 13953 C1S 716 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252166820 20508 13954 CCL21 6366 DRUGGABLE GENOME HEPARIN HEPARIN 11286540 20509 13955 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Carbamazepine CARBAMAZEPINE 20512 13956 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHIR-265 RAF-265 20514 13957 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR inhibitor CRIZOTINIB CRIZOTINIB 20515 13958 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE CHEMBL3833373 AVELUMAB 20516 13959 MAPT 4137 DRUGGABLE GENOME ARISTOLOCHIC ACID ARISTOLOCHIC ACID 20517 13960 IL1B 3553 KINASE, DRUGGABLE GENOME OFLOXACIN OFLOXACIN 3260587 20521 13961 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-402083 CHEMBL1546228 20523 13962 PTGS1 5742 ENZYME, DRUGGABLE GENOME KETOPROFEN KETOPROFEN 20524 13963 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE LY3164530 LY-3164530 20525 13964 CRBN 51185 ENZYME, DRUG RESISTANCE 178103899 THALIDOMIDE 20526 13965 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TETROQUINONE TETROQUINONE 20528 13966 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody 249565679 SARILUMAB 20529 13967 IFNG 3458 DRUGGABLE GENOME BLEOMYCIN BLEOMYCIN 8556994 20531 13968 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME AMSACRINE AMSACRINE 20534 13969 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME simeprevir SIMEPREVIR 20535 13970 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor AT9283 AT-9283 20536 13971 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 328083462 20538 13972 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME ISRAPAFANT ISRAPAFANT 20541 13973 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200342 PARAMETHASONE ACETATE 20542 13974 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102737 20544 13975 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR GW-870086-X 20545 13976 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME PD-98059 CHEMBL35482 15385570 20549 13977 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody NIMOTUZUMAB NIMOTUZUMAB 20554 13978 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651625 VASOPRESSIN 20555 13979 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL3545075 LAROTRECTINIB 20556 13980 ATAD5 79915 NA GNF-PF-3037 CHEMBL600336 20557 13981 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHELERYTHRINE CHELERYTHRINE 20560 13982 ATAD5 79915 NA DIPYRIDAMOLE DIPYRIDAMOLE 20561 13983 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME inhibitor COBIMETINIB COBIMETINIB 20562 13984 PAK3 5063 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 310264720 20563 13985 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NEFAZODONE HYDROCHLORIDE NEFAZODONE HYDROCHLORIDE 20565 13986 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME erlotinib ERLOTINIB 20567 13987 TSPO 706 DRUGGABLE GENOME Benzodiazepine derivative 1 20568 13988 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR 7-azaindole derivative 2 20569 13989 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor BI2536 20570 13990 HMGCR 3156 ENZYME, DRUGGABLE GENOME hmg coa reductase inhibitors 17563401,18815589,18332269,16103896,18261733,15199031,20403997 20571 13991 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 flunitrazepam FLUNITRAZEPAM 20574 13992 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DROSPIRENONE DROSPIRENONE 20577 13993 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE ERY974 ERY-974 20578 13994 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL3545238 CS-8080 20579 13995 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TCMDC-123713 CHEMBL586135 20580 13996 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ALFUZOSIN ALFUZOSIN 20581 13997 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 178102582 20582 13998 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE PHENTOLAMINE PHENTOLAMINE 10381893 20583 13999 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200819 ARTICAINE HYDROCHLORIDE 20584 14000 SRP19 6728 NA sertraline SERTRALINE 22795047 20586 14001 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID27744724-Compound-21 20587 14002 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Erlotinib ERLOTINIB 27659046 20588 14003 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PHENSERINE PHENSERINE 20589 14004 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE partial agonist CHEMBL3545408 NALTALIMIDE 20592 14005 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL865 VALDECOXIB 20593 14006 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178101914 NAPROXEN 20595 14007 PICK1 9463 KINASE, TRANSPORTER methamphetamine METHAMPHETAMINE 17606663 20596 14008 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 135650039 20597 14009 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE allosteric modulator 178101052 20598 14010 DYRK2 8445 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 249565807 20599 14011 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE alfentanil ALFENTANIL 16906017,19605407 20600 14012 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL969 PRAZEPAM 20602 14013 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME 178101729 20604 14014 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 363894135 MERESTINIB 20606 14015 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR LITHOCHOLIC ACID LITHOCHOLIC ACID 20607 14016 POLB 5423 DNA REPAIR, DRUGGABLE GENOME (+)-TAXIFOLIN (+)-TAXIFOLIN 20608 14017 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (R)-PINOCEMBRIN (R)-PINOCEMBRIN 20610 14018 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 quinine QUININE 9187528 20612 14019 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME CYC065 CYC-065 20613 14020 ALOX15B 247 DRUGGABLE GENOME, ENZYME JUGLONE JUGLONE 20614 14021 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME CEFADROXIL CEFADROXIL 8774083 20615 14022 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NORGESTREL NORGESTREL 20616 14023 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME AZD-1775 ADAVOSERTIB 20619 14024 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR QUINALDINE BLUE QUINALDINE BLUE 20620 14025 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Phenylbutyrate PHENYLBUTANOIC ACID 20621 14026 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Afatinib AFATINIB 26341921,27338794,25870145 20622 14027 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-1030061A GSK-1030061A 20623 14028 SLC12A6 9990 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 178101310 20624 14029 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SILIBININ SILIBININ 20625 14030 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Darifenacin DARIFENACIN 20626 14031 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8829193, 2 20627 14032 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BETA-LAPACHONE LAPACHONE 20630 14033 GAL 51083 DRUGGABLE GENOME CORTISOL HYDROCORTISONE 17982695 20631 14034 BRDT 676 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE PMID26924192-Compound-103 20632 14035 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TRIMEPRAZINE TARTRATE TRIMEPRAZINE TARTRATE 20634 14036 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE TOREMIFENE TOREMIFENE 8262671 20635 14037 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER W-198 20636 14038 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GLYCINE GLYCINE 22931300 20637 14039 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE US9156852, 1 20639 14040 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ARISTOYUNNOLIN A ARISTOYUNNOLIN A 20640 14041 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRIADIMENOL TRIADIMENOL 20641 14042 GAA 2548 DRUGGABLE GENOME, ENZYME 2-HYDROXYESTRADIOL CHEMBL467987 20644 14043 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE GEMCITABINE GEMCITABINE 28577946 20645 14044 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-9037 CHEMBL1451216 20646 14045 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inducer VADIMEZAN VADIMEZAN 20647 14046 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PURPURIN PURPURIN 20648 14047 GMNN 51053 DRUGGABLE GENOME GITOXIN GITOXIN 20649 14048 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME opioids 17986163 20650 14049 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE N/A 20652 14050 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650400 20653 14051 IL1B 3553 KINASE, DRUGGABLE GENOME CORTISOL HYDROCORTISONE 2162889 20654 14052 GAA 2548 DRUGGABLE GENOME, ENZYME IMINOSTILBENE IMINOSTILBENE 20655 14053 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME FICLATUZUMAB FICLATUZUMAB 20657 14054 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1113 AMOXAPINE 20659 14055 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-4659 CHEMBL584442 20660 14056 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE inhibitor CHEMBL2108184 CROFELEMER 20661 14057 SLC28A1 9154 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ADENOSINE ADENOSINE 23388705 20662 14058 IL1B 3553 KINASE, DRUGGABLE GENOME MAPK INHIBITORS 11382751 20663 14059 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TCMDC-123764 CHEMBL533226 20664 14060 EYA2 2139 DNA REPAIR DIMETHYL YELLOW DIMETHYL YELLOW 20667 14061 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649931 20668 14062 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TESTOSTERONE TESTOSTERONE 22931300 20669 14063 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-317605 CHEMBL1312050 20671 14064 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LINOLENIC ACID LINOLENIC ACID 20672 14065 LOXL2 4017 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL2109667 SIMTUZUMAB 20673 14066 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR inhibitor 178103428 HYDROXYUREA 20674 14067 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ATROPINE ATROPINE 2128054 20675 14068 MAPT 4137 DRUGGABLE GENOME SARCOLYSIN SARCOLYSIN 20676 14069 TAT 6898 ENZYME ALBUMIN ALBUMIN HUMAN 6127852 20677 14070 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 315661304 RAVOXERTINIB 20679 14071 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 374883876 20680 14072 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME BROMAZEPAM BROMAZEPAM 20681 14073 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32t 20682 14074 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUOXYMESTERONE FLUOXYMESTERONE 20684 14075 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1356607 NOREPINEPHRINE BITARTRATE 20685 14076 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE VEMURAFENIB VEMURAFENIB 24265152 20687 14077 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-699479 CHEMBL1701915 20688 14078 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME HYDRALAZINE HYDRALAZINE 20689 14079 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 178101445 20691 14080 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE GNF-PF-4353 CHEMBL527307 20693 14081 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 20694 14082 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178101606 DORSOMORPHIN 20696 14083 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX THIOINOSINE THIOINOSINE 20697 14084 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE JNJ-63709178 20698 14085 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME trametinib TRAMETINIB 20699 14086 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LYCOPENE LYCOPENE 11437362 20700 14087 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYCLOPHOSPHAMIDE HYDRATE CYCLOPHOSPHAMIDE 20701 14088 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR GIVINOSTAT GIVINOSTAT 20702 14089 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NIFEDIPINE NIFEDIPINE 17655375 20703 14090 PTGS2 5743 DRUGGABLE GENOME, ENZYME OXAPROZIN OXAPROZIN 20704 14091 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178103587 MOCETINOSTAT 20705 14092 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Capecitabine CAPECITABINE 20706 14093 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL1739 METOCURINE IODIDE 20708 14094 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Carbamide derivative 23 20711 14095 MMP7 4316 NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 178103078 DOXYCYCLINE 20712 14096 PSMA1 5682 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL325041 BORTEZOMIB 20713 14097 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103121 20714 14098 GMNN 51053 DRUGGABLE GENOME EPOXYCYTOCHALASIN H EPOXYCYTOCHALASIN H 20715 14099 HSPA4 3308 NA POH 17024970 20716 14100 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE antibody 310264712 MM-111 20718 14101 BAZ2B 29994 NA DNDI1417601 CHEMBL1503729 20719 14102 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SORAFENIB SORAFENIB 20720 14103 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 gemtuzumab ozogamicin 22584460 20722 14104 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Pentostatin PENTOSTATIN 20724 14105 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PANOBINOSTAT PANOBINOSTAT 24694055 20725 14106 MAPT 4137 DRUGGABLE GENOME GNF-PF-3012 CHEMBL582715 20726 14107 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME desipramine DESIPRAMINE 9918137,8422746,20531370,10895986,1346258,15252821,14652703,14716707,6488689,18359183,14520122,8867869,9049581,8181196,8941025,17721180,3533565,3356084,17667959,15115913,12360109,14646691,15205367,27440861,11682257,16024198,3769385,16361630,17008819,23486447,10460069,9585799,16871470,11417443 20727 14108 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE GLPG0187 GLPG-0187 20728 14109 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-18 20729 14110 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 178100440 CHEMBL500272 20731 14111 CHKA 1119 ENZYME, KINASE TCD-717 TCD-717 20732 14112 VDAC3 7419 KINASE OLESOXIME OLESOXIME 20733 14113 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME 5,8,11,14-EICOSATETRAYNOIC ACID CHEMBL458328 20734 14114 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AZITHROMYCIN AZITHROMYCIN 22931300 20735 14115 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DNDI1417086 CHEMBL1224755 20736 14116 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME IMIPRAMINE HYDROCHLORIDE IMIPRAMINE HYDROCHLORIDE 20737 14117 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR ETANERCEPT ETANERCEPT 12906870 20738 14118 RAB9A 9367 ENZYME, DRUGGABLE GENOME 4'-HYDROXYPHENYL-BENZO[D]THIAZOLE CHEMBL47875 20739 14119 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545055 INK-1117 20740 14120 USP1 7398 DNA REPAIR, PROTEASE, ENZYME NSC-95397 CHEMBL429095 20741 14121 PAK3 5063 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 310264719 20743 14122 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PHENYLBUTYRATE PHENYLBUTANOIC ACID 10696460 20744 14123 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Indoline derivative 8 20745 14124 HMOX1 3162 ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE HORMONES 16214137 20746 14125 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ETHYL ANTHRANILATE ETHYL ANTHRANILATE 20747 14126 GMNN 51053 DRUGGABLE GENOME PENTACHLOROPHENOL PENTACHLOROPHENOL 20748 14127 HINT1 3094 NA nicotine NICOTINE 17978999 20749 14128 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SELENIUM 12577306 20750 14129 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 135651447 20752 14130 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor CHEMBL27759 ENTINOSTAT 20753 14131 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MIRISTALKONIUM CHLORIDE MIRISTALKONIUM CHLORIDE 20754 14132 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON BETA 20755 14133 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHYLPREDNISOLONE SODIUM SUCCINATE METHYLPREDNISOLONE SODIUM SUCCINATE 20757 14134 POLI 11201 DNA REPAIR CEFSULODIN SODIUM CEFSULODIN SODIUM 20758 14135 BAZ2A 11176 ENZYME inhibitor 252166772 20759 14136 PTGS2 5743 DRUGGABLE GENOME, ENZYME ibuprofen IBUPROFEN 25502615,16678543,19602986 20760 14137 BAZ2B 29994 NA MIFEPRISTONE MIFEPRISTONE 20761 14138 CBX1 10951 NA N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 20762 14139 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE METHYLNALTREXONE METHYLNALTREXONE 20763 14140 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR METHYLBENZETHONIUM CHLORIDE METHYLBENZETHONIUM CHLORIDE 20764 14141 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE docetaxel DOCETAXEL 30071039 20765 14142 GGCX 2677 DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 20767 14143 CDH3 1001 DRUGGABLE GENOME PF-3732010 20769 14144 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME CAP-232 20770 14145 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 135650518 20771 14146 PKN1 5585 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 135652717 STAUROSPORINE 20772 14147 KAT2B 8850 ENZYME, DRUGGABLE GENOME inhibitor 252166597 20773 14148 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102485 IRALUKAST 20774 14149 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIMETHYL GAMBOGATE DIMETHYL GAMBOGATE 20775 14150 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME METHYLDOPA (RACEMIC) METHYLDOPA (RACEMIC) 20777 14151 ALPL 249 ENZYME, DRUGGABLE GENOME TYRPHOSTIN 23 TYRPHOSTIN 23 20778 14152 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GF-109203 GF-109203 20779 14153 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME volatile anesthetics 30136624 20780 14154 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER LAMIVUDINE LAMIVUDINE 12218384 20781 14155 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR N/A 20782 14156 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-4283 CHEMBL606166 20783 14157 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME P32/98 20784 14158 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-1737 CHEMBL531710 20785 14159 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ENTINOSTAT ENTINOSTAT 19966789,20491440 20787 14160 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME TESTOSTERONE TESTOSTERONE 1764091 20788 14161 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Binimetinib BINIMETINIB 20790 14162 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Sapanisertib SAPANISERTIB 25261369 20792 14163 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR PMID26924192-Compound-104 20794 14164 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR JQEZ5 27135738 20795 14165 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PAROXETINE HYDROCHLORIDE PAROXETINE HYDROCHLORIDE 20796 14166 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200819 ARTICAINE HYDROCHLORIDE 20797 14167 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist 135649903 20798 14168 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE GLIPIZIDE GLIPIZIDE 8043894 20799 14169 DMD 1756 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME WVE-210201 20800 14170 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE IL-2 ALDESLEUKIN 10229082 20801 14171 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON BETA-1B 20803 14172 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ISOBOLDINE ISOBOLDINE 20805 14173 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME JNJ-7706621 JNJ-7706621 20808 14174 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE DOCETAXEL DOCETAXEL 16969094 20810 14175 TH 7054 ENZYME, DRUGGABLE GENOME ANTIESTROGEN 11223814 20811 14176 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545428 CHIAURANIB 20812 14177 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR THEONELLASTEROL C THEONELLASTEROL C 21428459 20813 14178 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Indoline derivative 15 20814 14179 ATAD5 79915 NA GNF-PF-4046 CHEMBL600090 20817 14180 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL2110725 VINFLUNINE 20818 14181 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY TGFBETA1 10770487,10194419 20820 14182 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1200973 ESTRADIOL CYPIONATE 20821 14183 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR emapalumab EMAPALUMAB 20823 14184 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor 405560268 LINEZOLID 20825 14185 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A8 20826 14186 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 328083478 20827 14187 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LAS38096 CHEMBL375293 20828 14188 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 7 20829 14189 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 3-((2,4-DICHLOROPHENYLTHIO)METHYL)BENZOATE CHEMBL1923999 22047606 20830 14190 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 178103383 20831 14191 PPID 5481 DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING, KINASE US8901295, F673 20835 14192 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1711 ISOPROTERENOL HYDROCHLORIDE 20836 14193 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AEE788 AEE-788 19147750 20837 14194 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME estradiol / progesterone 20838 14195 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 223365913 20839 14196 METAP2 10988 ENZYME, DRUGGABLE GENOME, KINASE, PROTEASE BELORANIB BELORANIB 20840 14197 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1100 PARAMETHADIONE 20841 14198 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Trametinib TRAMETINIB 20842 14199 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 381118839 REVEFENACIN 20843 14200 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE BRONCHODILATOR 15806595 20844 14201 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE JNJ-42756493 ERDAFITINIB 28341788 20845 14202 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME inhibitor 135649695 20846 14203 NOS2 4843 DRUGGABLE GENOME, ENZYME inhibitor 178101915 20847 14204 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME WORTMANNIN WORTMANNIN 9603913 20848 14205 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 17 BETA-ESTRADIOL 1315250 20850 14206 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME NFX 12756268 20851 14207 PRKAB2 5565 KINASE, ENZYME allosteric modulator 252827478 20855 14208 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME KAEMPFERITRIN KAEMPFERITRIN 22014228 20858 14209 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ORTATAXEL ORTATAXEL 20859 14210 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER CDDP CISPLATIN 11372415 20860 14211 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHLORANIL CHLORANIL 20861 14212 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL ritodrine RITODRINE 28391406 20862 14213 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME Cobimetinib COBIMETINIB 20863 14214 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 20864 14215 CDK17 5128 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR inhibitor CHEMBL488436 AZD-5438 20865 14216 PRKAG2 51422 ENZYME, KINASE METFORMIN METFORMIN 26471090 20867 14217 COMT 1312 DRUGGABLE GENOME, ENZYME nicotine NICOTINE 18192898,22695756,26555332,11927842,16395295 20869 14218 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME INCOMPLETE FREUNDS ADJUVANT 11768621 20870 14219 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C2 20872 14220 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102234 20873 14221 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NALBUPHINE NALBUPHINE 20874 14222 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME GNF-PF-308 CHEMBL600334 20875 14223 PREP 5550 PROTEASE, ENZYME, DRUGGABLE GENOME STZ STREPTOZOCIN 8190911 20876 14224 PSMC3 5702 NA inhibitor CARFILZOMIB CARFILZOMIB 20877 14225 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor CHEMBL2105721 NIVOCASAN 20878 14226 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ACITRETIN ACITRETIN 20879 14227 DNER 92737 NA Isoxazole-based bicyclic compound 18 20880 14228 POLK 51426 DNA REPAIR, ENZYME CARMINOMYCIN CARUBICIN 20881 14229 GMNN 51053 DRUGGABLE GENOME SJ000032152 CHEMBL590665 20882 14230 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME inhibitor 135652074 20883 14231 GLS 2744 ENZYME LOMOFUNGIN LOMOFUNGIN 20884 14232 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME FLUPIRTINE FLUPIRTINE 20885 14233 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-16 20887 14234 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1-NAPHTHOL 1-NAPHTHOL 20888 14235 F7 2155 ENZYME, DRUGGABLE GENOME, PROTEASE Factor viia 20889 14236 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME BGT226 BGT-226 20890 14237 ATP2C1 27032 ENZYME, TRANSPORTER, DRUGGABLE GENOME ENFLURANE ENFLURANE 20891 14238 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-3996 CHEMBL584458 20893 14239 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SULINDAC SULINDAC 20894 14240 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL3545328 XL-019 20895 14241 RGS4 5999 DRUGGABLE GENOME GNF-PF-1969 CHEMBL601364 20897 14242 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE PLX4720 PLX-4720 24504448 20898 14243 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BROMOENOL LACTONE BROMOENOL LACTONE 20900 14244 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME TOZASERTIB TOZASERTIB 20901 14245 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-36 20902 14246 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE GRNVAC1 20903 14247 POLG 5428 ENZYME divalproex sodium 20906 14248 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor CHEMBL494089 GSK-690693 20907 14249 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE MAHANINE MAHANINE 20184324 20908 14250 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE positive modulator CHEMBL1255840 NEBOGLAMINE 20909 14251 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE AFM-13 20911 14252 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist 178100653 20912 14253 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist 178100667 20913 14254 REG3A 5068 DRUGGABLE GENOME HIP-2B 20914 14255 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AFATINIB AFATINIB 19122144,22325357,26296355,26559459,30096481,22418700,25370464,26596672 20915 14256 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME ACACETIN ACACETIN 20916 14257 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE GSK2110183 AFURESERTIB 20917 14258 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SLAZINIC ACID SLAZINIC ACID 20920 14259 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER DEXTROAMPHETAMINE DEXTROAMPHETAMINE 20921 14260 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 310264781 ADL-5747 20922 14261 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR Pyrrolo-pyrrolone derivative 1 20923 14262 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CART-EGFR 20924 14263 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME SUBEROHYDROXAMIC ACID SUBEROHYDROXAMIC ACID 16921367 20925 14264 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GW7647 GW7647 20926 14265 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1631540 GSK163090 20927 14266 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ETHACRIDINE LACTATE ETHACRIDINE LACTATE 20928 14267 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DHM25 26237138 20929 14268 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1018 DIENESTROL 20930 14269 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME SP-600125 SP-600125 23634759 20931 14270 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL1879463 DACTOLISIB 20932 14271 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE PHA-767491 CHEMBL225519 20933 14272 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 315661176 20934 14273 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DNDI1417827 CHEMBL1363249 20935 14274 POLK 51426 DNA REPAIR, ENZYME OXYTETRACYCLINE HYDROCHLORIDE OXYTETRACYCLINE HYDROCHLORIDE 20936 14275 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DIETHYLSTILBESTROL DIETHYLSTILBESTROL 26408814 20938 14276 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE PICTILISIB PICTILISIB 20939 14277 MAOA 4128 DRUGGABLE GENOME, ENZYME HARMINE HARMINE 20941 14278 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE LACTULOSE LACTULOSE 11226652 20942 14279 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CHEMBL681 ETOMIDATE 20947 14280 SLC22A5 6584 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PROPIONYL-L-CARNITINE 20950 14281 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SULFISOXAZOLE SULFISOXAZOLE 20952 14282 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL3545044 LUMATEPERONE 20954 14283 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-56 20956 14284 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BETAXOLOL BETAXOLOL 20957 14285 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE PKI-590 20958 14286 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 249565787 VACTOSERTIB 20959 14287 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME 2,3,7,8-TETRACHLORODIBENZO-P-DIOXIN 2,3,7,8-TETRACHLORODIBENZO-P-DIOXIN 14684315 20960 14288 TXK 7294 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 249565828 20961 14289 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER ENOXOLONE ENOXOLONE 24461294 20962 14290 ACLY 47 ENZYME, DRUGGABLE GENOME ETC-1002 BEMPEDOIC ACID 20964 14291 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME XANTHONE XANTHONE 20965 14292 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME agonist CHEMBL2107866 PEGINESATIDE 20966 14293 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ECONAZOLE NITRATE ECONAZOLE NITRATE 20967 14294 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME BTT-1023 TIMOLUMAB 20968 14295 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Drug 2881078 20969 14296 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Metformin METFORMIN 26363012 20973 14297 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Tolterodine TOLTERODINE 20974 14298 ALOX15 246 ENZYME, DRUGGABLE GENOME CADMIUM ACETATE CADMIUM ACETATE 20975 14299 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE LY3023414 SAMOTOLISIB 20976 14300 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CANRENOATE POTASSIUM CANRENOATE POTASSIUM 20977 14301 PYGL 5836 DRUGGABLE GENOME, ENZYME PSN357 20978 14302 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX AMINOQUINOL AMINOQUINOL 20980 14303 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 381118805 20981 14304 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME QUERCETIN QUERCETIN 15741050 20983 14305 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GUTHION GUTHION 20985 14306 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL812 PYRIDOSTIGMINE BROMIDE 20988 14307 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ALPHA-NAPHTHOFLAVONE ALPHA-NAPHTHOFLAVONE 20989 14308 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL87992 ESLICARBAZEPINE ACETATE 20990 14309 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-28 20992 14310 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR REVERSETRIIODOTHYRONINE REVERSETRIIODOTHYRONINE 20993 14311 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON BETA-1A 20995 14312 COMT 1312 DRUGGABLE GENOME, ENZYME lithium LITHIUM 20996 14313 PTBP1 5725 DRUGGABLE GENOME SJ000154295 CHEMBL578502 20997 14314 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME SMT-D002 20999 14315 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DINOPROSTONE DINOPROSTONE 25701254 21001 14316 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR 7-O-METHYLCRYPTOCHINONE B 7-O-METHYLCRYPTOCHINONE B 25127166 21003 14317 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 53801005 21004 14318 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME ACY-1215 RICOLINOSTAT 21006 14319 UGT1A6 54578 ENZYME, DRUGGABLE GENOME methotrexate METHOTREXATE 29791011 21007 14320 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 8 21008 14321 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME MLN-8054 MLN-8054 21010 14322 CBX1 10951 NA SB-415286 CHEMBL322970 21011 14323 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ATALUREN ATALUREN 21014 14324 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GRAMINE GRAMINE 21017 14325 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE azathioprine AZATHIOPRINE 26332308 21023 14326 ALB 213 TRANSPORTER, DRUGGABLE GENOME PHENYLBUTAZONE PHENYLBUTAZONE 20869876 21028 14327 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER antipsychotics 27272046 21030 14328 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 178103204 NATALIZUMAB 21031 14329 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-24 21032 14330 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 223366044 21033 14331 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE BMS-777607 BMS-777607 21035 14332 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-45a 21037 14333 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 381744974 POLYGODIAL 21038 14334 PLD2 5338 ENZYME, DRUGGABLE GENOME inhibitor 178101970 21039 14335 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE AG-494 CHEMBL56731 21040 14336 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 bleomycin BLEOMYCIN 21043 14337 POLI 11201 DNA REPAIR FLUPIRTINE MALEATE FLUPIRTINE MALEATE 21044 14338 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE lomitapide LOMITAPIDE 21045 14339 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME INDOLE-3-CARBINOL INDOLE-3-CARBINOL 15611077 21047 14340 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ISOPROTERENOL ISOPROTERENOL 21048 14341 SOS1 6654 KINASE 385612239 21049 14342 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor MGCD265 GLESATINIB 21052 14343 ATXN2 6311 NA ANGUSTIBALIN ANGUSTIBALIN 21054 14344 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 1-AMINOCYCLOHEXANECARBOXYLIC ACID CHEMBL559934 21055 14345 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE antagonist EZN-2968 21056 14346 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DEPHOSTATIN DEPHOSTATIN 21057 14347 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody ROBATUMUMAB ROBATUMUMAB 21058 14348 ALOX5 240 DRUGGABLE GENOME, ENZYME PTC299 21059 14349 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE AMEDIPLASE AMEDIPLASE 21060 14350 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE REGN-727 ALIROCUMAB 21061 14351 CA2 760 DRUGGABLE GENOME, ENZYME COUMATE 21062 14352 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100463 DABUZALGRON 21064 14353 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME CIANIDANOL CIANIDANOL 21067 14354 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE BRYOSTATIN-1 10918054 21068 14355 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 10 21071 14356 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200989 ALCLOMETASONE DIPROPIONATE 21072 14357 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL24828 VANDETANIB 21075 14358 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650465 L-165461 21076 14359 PSMD7 5713 PROTEASE BORTEZOMIB BORTEZOMIB 24524217 21077 14360 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR EED226 28135235 21080 14361 RACGAP1 29127 NA HYDROXYSTILBAMIDINE ISETHIONATE HYDROXYSTILBAMIDINE ISETHIONATE 21082 14362 HBEGF 1839 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME cetuximab CETUXIMAB 21085 14363 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Amlexanox AMLEXANOX 21086 14364 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING ANTHRACENE-9-CARBOXYLIC ACID ANTHRACENE-9-CARBOXYLIC ACID 21087 14365 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-22 21089 14366 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TUBERCIDIN TUBERCIDIN 21090 14367 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR VER 50589 21091 14368 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR escitalopram ESCITALOPRAM 19641488 21092 14369 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AFATINIB AFATINIB 21093 14370 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Heterocyclic-fused piperazine derivative 1 21094 14371 EYA2 2139 DNA REPAIR DIOTYROSINE DIOTYROSINE 21095 14372 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650814 ALPROSTADIL 21096 14373 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ALSTERPAULLONE ALSTERPAULLONE 21098 14374 ATAD5 79915 NA TCMDC-123764 CHEMBL533226 21102 14375 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Pembrolizumab PEMBROLIZUMAB 28039262 21103 14376 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor PF-04217903 PF-04217903 21104 14377 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545365 ALTIRATINIB 21106 14378 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME URSOLIC ACID URSOLIC ACID 19534471 21107 14379 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 2,6-DIMETHOXYQUINONE 2,6-DIMETHOXYQUINONE 21109 14380 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 imipramine IMIPRAMINE 9187528 21110 14381 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER DELAVIRDINE DELAVIRDINE 17172311 21111 14382 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE AG-1879 CHEMBL406845 21112 14383 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 21116 14384 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PI-3065 24919154 21118 14385 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SJ000059272 CHEMBL592369 21119 14386 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-1947 CHEMBL585591 21120 14387 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL741 LAMOTRIGINE 21121 14388 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CUMENE HYDROPEROXIDE CUMENE HYDROPEROXIDE 21122 14389 GLS 2744 ENZYME 4-AMINOPHENOL 4-AMINOPHENOL 21123 14390 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL HX-100 21124 14391 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-6 21125 14392 PSMB10 5699 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL2103884 OPROZOMIB 21126 14393 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME inhibitor 249565916 21129 14394 APOE 348 DRUGGABLE GENOME ritonavir RITONAVIR 17700364,15809899 21130 14395 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ZOLANTIDINE ZOLANTIDINE 21131 14396 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE carbamazepine CARBAMAZEPINE 21449672,22630058,22188362,20216337,21738081,25155934,22256867,23697249,24567120,21799461,23252947 21132 14397 IL7R 3575 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME antibody 340590234 21134 14398 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE LAPATINIB LAPATINIB 25305330,24355130 21136 14399 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL BROMAZEPAM BROMAZEPAM 21138 14400 MAP2K3 5606 KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE WX-554 WX-554 21139 14401 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565693 21141 14402 KDM4A 9682 DRUGGABLE GENOME, ENZYME EBSELEN EBSELEN 21144 14403 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL598797 CUDC-101 21145 14404 ALOX15B 247 DRUGGABLE GENOME, ENZYME PHENOTHIAZINE PHENOTHIAZINE 21147 14405 FGF1 2246 CLINICALLY ACTIONABLE, GROWTH FACTOR, DRUGGABLE GENOME PENTOSAN POLYSULFATE 21149 14406 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR AST-487 AST-487 21150 14407 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR HEPARAN SULFATE 1331122 21151 14408 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUMETHASONE PIVALATE 21152 14409 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME M-CSF CILMOSTIM 10770207 21154 14410 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ANG1005 ANG1005 21155 14411 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE DIAZOXIDE DIAZOXIDE 14499880 21157 14412 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NARINGIN NARINGIN 21159 14413 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME TAMATINIB R-406 21161 14414 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR TCMDC-124530 CHEMBL582593 21162 14415 AKR1B1 231 DRUGGABLE GENOME, ENZYME ARI-809 21164 14416 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2016054807Example112 21166 14417 GLS 2744 ENZYME 2',3,4-TRIHYDROXYCHALCONE CHEMBL339587 21168 14418 MAPT 4137 DRUGGABLE GENOME GNF-PF-3537 CHEMBL601110 21171 14419 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ISOCONAZOLE ISOCONAZOLE 21172 14420 COL1A2 1278 DRUGGABLE GENOME COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 21174 14421 ICA1 3382 NA o-desmethyl-tramadol 30971809 21175 14422 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME desloratadine DESLORATADINE 31406237 21177 14423 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME sulfasalazine SULFASALAZINE 25872459,24394199,28322941,18167504 21178 14424 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AZAKENPAULLONE AZAKENPAULLONE 21179 14425 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR GEFITINIB GEFITINIB 21180 14426 FAP 2191 PROTEASE, CELL SURFACE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME RG7461 21182 14427 MAPT 4137 DRUGGABLE GENOME GF-109203 GF-109203 21183 14428 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 23622981 21185 14429 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TANESPIMYCIN TANESPIMYCIN 21187 14430 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MENADIONE MENADIONE 21191 14431 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 249565775 21193 14432 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME 681640 CHEMBL379975 21194 14433 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE bisoprolol fumarate / perindopril arginine 21195 14434 BCL2L11 10018 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR 22426421 21197 14435 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DEXAMETHASONE DEXAMETHASONE 22931300 21198 14436 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME 2,6-DIMETHOXYQUINONE 2,6-DIMETHOXYQUINONE 21200 14437 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor CHEMBL1201605 DACLIZUMAB 21201 14438 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VALPROIC ACID VALPROIC ACID 18294844,16921367,25304896 21202 14439 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME PMA 10586059 21204 14440 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IDARUBICIN IDARUBICIN 21205 14441 RAB9A 9367 ENZYME, DRUGGABLE GENOME PECTOLINARIGENIN PECTOLINARIGENIN 21206 14442 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Everolimus EVEROLIMUS 23629727 21207 14443 ALDH1A1 216 DRUGGABLE GENOME, ENZYME EBSELEN EBSELEN 21212 14444 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650675 21213 14445 PTGS2 5743 DRUGGABLE GENOME, ENZYME FENOPROFEN FENOPROFEN 21216 14446 VKORC1 79001 DRUGGABLE GENOME, ENZYME PHENPROCOUMON PHENPROCOUMON 21219 14447 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME inhibitor 336446965 21222 14448 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE MT-110 21224 14449 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE GO-6976 GO-6976 21225 14450 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE LIOTHYRONINE SODIUM LIOTHYRONINE SODIUM 21227 14451 CSK 1445 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE 936563-93-8 21230 14452 SH2B3 10019 CLINICALLY ACTIONABLE, KINASE candesartan CANDESARTAN 31327267 21231 14453 CBR1 873 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME N6022 N6022 21232 14454 ATXN1L 342371 DRUG RESISTANCE TRAMETINIB TRAMETINIB 28178529 21235 14455 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 328083501 21237 14456 PRKAB1 5564 ENZYME, KINASE, DRUGGABLE GENOME PROPYLTHIOURACIL PROPYLTHIOURACIL 12433937 21238 14457 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE 178101758 21240 14458 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2218898 BARUSIBAN 21242 14459 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR GNF-PF-2307 CHEMBL421088 21243 14460 AOAH 313 ENZYME, DRUGGABLE GENOME inhibitor 252166807 21248 14461 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CSL-362-AML 21249 14462 GRB2 2885 NA HEREGULIN 11175341 21250 14463 RCSD1 92241 NA IMATINIB IMATINIB 27125982 21251 14464 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 23 21252 14465 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US9682991, 2 21253 14466 IMPDH2 3615 DRUGGABLE GENOME, ENZYME cyclosporine CYCLOSPORINE 21996196,19770842,18444945,19617864,22960765 21254 14467 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE XL-499 21256 14468 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BARDOXOLONE METHYL BARDOXOLONE METHYL 21258 14469 GMNN 51053 DRUGGABLE GENOME PROSULTIAMINE PROSULTIAMINE 21259 14470 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Phenytoin PHENYTOIN 21260 14471 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE PRT6207 24419749 21261 14472 CBX1 10951 NA 3,4-DICHLOROISOCOUMARIN CHEMBL24983 21263 14473 BAZ2B 29994 NA GNF-PF-1295 CHEMBL579837 21265 14474 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 178102556 AZD-1480 21266 14475 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 315661147 21267 14476 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME dabrafenib DABRAFENIB 21268 14477 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 10-IODOEVODIAMINE CHEMBL2171807 22867019 21269 14478 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR modulator CHEMBL3545047 BMS-852927 21270 14479 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BENZO(K)FLUORANTHENE BENZO(K)FLUORANTHENE 21271 14480 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SULFAPHENAZOLE SULFAPHENAZOLE 22931300 21274 14481 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 21275 14482 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103310 FLUTICASONE 21276 14483 GMNN 51053 DRUGGABLE GENOME METHYL DEOXYCHOLATE METHYL DEOXYCHOLATE 21277 14484 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BUPRENORPHINE HYDROCHLORIDE BUPRENORPHINE HYDROCHLORIDE 21278 14485 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE ACI-24 24148220 21279 14486 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME RG-1530 RG-1530 21280 14487 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL1042 CHOLECALCIFEROL 21281 14488 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135651957 21282 14489 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 385612249 21283 14490 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME OPC-14523 21284 14491 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR xenobiotics 11942593 21285 14492 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME APG-101 ASUNERCEPT 21286 14493 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 381744991 21287 14494 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DANAZOL DANAZOL 21289 14495 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR PF-562271 PF-00562271 21290 14496 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME TETRADECYLTHIOACETIC ACID TETRADECYLTHIOACETIC ACID 21291 14497 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR METHYL PARATHIONE METHYL PARATHIONE 21292 14498 BCHE 590 DRUGGABLE GENOME, ENZYME ISOFLUROPHATE ISOFLUROPHATE 21295 14499 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME PF-04965842 ABROCITINIB 21298 14500 SLCO3A1 28232 TRANSPORTER, DRUGGABLE GENOME 178101458 21299 14501 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR DOXYCYCLINE DOXYCYCLINE 16202406,15728539 21300 14502 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US9580418, Example 8 21301 14503 TUBB2A 7280 DRUGGABLE GENOME ALB109564(A) 21302 14504 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 21303 14505 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 375973251 21307 14506 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME BTT-1023 TIMOLUMAB 21308 14507 XPO1 7514 CLINICALLY ACTIONABLE, KINASE Eltanexor oral 21309 14508 TXNRD1 7296 DRUGGABLE GENOME Triazole gold complexe 3 21310 14509 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL411 DIETHYLSTILBESTROL 21312 14510 PSMB3 5691 PROTEASE, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 24524217 21313 14511 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200420 MIDAZOLAM HYDROCHLORIDE 21314 14512 PSMA1 5682 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL2103884 OPROZOMIB 21316 14513 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE MITOXANTRONE MITOXANTRONE 11751483 21318 14514 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BROQUINALDOL BROQUINALDOL 21319 14515 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist,antagonist 135650065 21321 14516 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ACTINOMYCIN D 10899924 21323 14517 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL1201023 ORPHENADRINE HYDROCHLORIDE 21328 14518 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE CHEMBL1743053 OTELIXIZUMAB 21329 14519 ATXN2 6311 NA MAPROTILINE MAPROTILINE 21330 14520 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-96 21331 14521 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist 135650994 21332 14522 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CAPSAICIN CAPSAICIN 21333 14523 NOTCH2 4853 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE antibody 252166663 TAREXTUMAB 21335 14524 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4ALPHA-HYDROPEROXY-5-ENOVATODIOLIDE CHEMBL512307 26178912 21336 14525 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-377852 CHEMBL1466186 21337 14526 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ETHYL 2,4,6-TRIHYDROXYBENZOATE CHEMBL2204435 22579484 21341 14527 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SOFALCONE SOFALCONE 21342 14528 TRH 7200 DRUGGABLE GENOME PHENYTOIN PHENYTOIN 6262046 21344 14529 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TRIFLUPROMAZINE HYDROCHLORIDE TRIFLUPROMAZINE HYDROCHLORIDE 21345 14530 SDHB 6390 ENZYME, CLINICALLY ACTIONABLE ANTIBIOTIC ANTIBIOTIC 6277242 21349 14531 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME EPO EPOETIN ALFA 17112829 21350 14532 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TRASTUZUMAB TRASTUZUMAB 18089830 21352 14533 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 328083499 SNS-314 21354 14534 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE LYS-6KAKT1 21355 14535 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PYRVINIUM PAMOATE PYRVINIUM PAMOATE 21356 14536 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CARBOPLATIN CARBOPLATIN 11157479 21357 14537 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545026 FAMITINIB 21361 14538 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME DNDI1417884 CHEMBL1346025 21362 14539 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE TAMATINIB R-406 21364 14540 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Antivirals for treatment of HIV infections, combinations 22162992 21365 14541 POLB 5423 DNA REPAIR, DRUGGABLE GENOME HISPIDIN HISPIDIN 21366 14542 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE INSULIN INSULIN 8826975 21367 14543 S100B 6285 DRUGGABLE GENOME, KINASE STREPTOZOTOCIN STREPTOZOCIN 14583344 21368 14544 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3545208 AZD3161 21370 14545 GMNN 51053 DRUGGABLE GENOME BUFOGENIN BUFOGENIN 21372 14546 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Glutethimide GLUTETHIMIDE 21373 14547 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BINIMETINIB BINIMETINIB 24588908,28284557,29245078,26987942,26821351 21376 14548 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME antagonist AT-406 AT-406 21377 14549 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor HESPERADIN HESPERADIN 19035792 21378 14550 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE LAK 2007574 21379 14551 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME GW843682X GW843682X 21381 14552 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ribociclib RIBOCICLIB 21382 14553 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GARCINONE E GARCINONE E 21383 14554 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 4SC-202 DOMATINOSTAT 21384 14555 HLA-DPA1 3113 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE peginterferon alfa-2b 26387494 21385 14556 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor NMS1286937 21386 14557 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE JNJ-7706621 JNJ-7706621 21387 14558 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX Trifarotene TRIFAROTENE 21390 14559 RGS4 5999 DRUGGABLE GENOME GW7074 CHEMBL72365 21393 14560 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR carvedilol CARVEDILOL 15864115,20643254,15861037,16815314,20352314,12709726,12921807,15735607,18075464,12844134,22617224,17496726,14534524,21311897,14502278,27643874,20235788 21394 14561 POLB 5423 DNA REPAIR, DRUGGABLE GENOME MMV006513 CHEMBL585622 21395 14562 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME gemcitabine GEMCITABINE 22441531 21396 14563 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor CHEMBL3137318 TALAZOPARIB TOSYLATE 21397 14564 FAAH 2166 ENZYME, DRUGGABLE GENOME Boronic acid derivative 2 21398 14565 SMARCB1 6598 CLINICALLY ACTIONABLE Alvocidib ALVOCIDIB 18223228 21399 14566 PSMB10 5699 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 21401 14567 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650408 21403 14568 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME etoposide ETOPOSIDE 26663398 21404 14569 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME OLEOYL DOPAMINE OLEOYL DOPAMINE 21406 14570 GLA 2717 ENZYME, DRUGGABLE GENOME Anamorelin ANAMORELIN 21407 14571 TNC 3371 DRUGGABLE GENOME, FIBRINOGEN CHEMBL2109582 81C6 131I 21408 14572 PSMD4 5710 NA inhibitor CHEMBL325041 BORTEZOMIB 21409 14573 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 178102555 JNJ-7706621 21413 14574 DHFR 1719 DRUGGABLE GENOME, ENZYME PEMETREXED PEMETREXED 21414 14575 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE ENTRECTINIB ENTRECTINIB 21418 14576 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 354702239 21419 14577 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-2301 CHEMBL578061 21422 14578 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR SCRIPTAID SCRIPTAID 19966789 21423 14579 KCNT2 343450 ION CHANNEL, DRUGGABLE GENOME inhibitor 135650820 21424 14580 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650624 MORPHINE 21425 14581 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE JWH-015 CHEMBL306764 21428 14582 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650519 21429 14583 TUBB2A 7280 DRUGGABLE GENOME COLCHICINE COLCHICINE 21430 14584 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL552212 LEXIBULIN 21433 14585 KDM6A 7403 ENZYME, CLINICALLY ACTIONABLE inhibitor 310264759 21435 14586 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201168 ISOCARBOXAZID 21436 14587 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE TOZASERTIB TOZASERTIB 21437 14588 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-31 21438 14589 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652253 21439 14590 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 384403666 21440 14591 PCNA 5111 NA ATX-101 DEOXYCHOLIC ACID 21441 14592 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ASN007 21442 14593 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 21443 14594 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE BUPRENORPHINE BUPRENORPHINE 21444 14595 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SALINE SODIUM CHLORIDE 12907413 21445 14596 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME IRINOTECAN IRINOTECAN 20619739,21575616 21446 14597 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 310264693 ACALABRUTINIB 21447 14598 CDC42BPA 8476 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TAE-684 TAE-684 21449 14599 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME PMID27774824-Compound-Figure11Example1up 21450 14600 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PYRACLOSTROBIN PYRACLOSTROBIN 21451 14601 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE TTP-814 21452 14602 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 21453 14603 TSPO 706 DRUGGABLE GENOME Benzothiazepine analog 6 21454 14604 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME sunitinib SUNITINIB 22948895 21455 14605 EPHB3 2049 DRUGGABLE GENOME, TYROSINE KINASE, KINASE inhibitor CHEMBL24828 VANDETANIB 21456 14606 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE carvedilol CARVEDILOL 15861037,20352314,21599570,12835612 21458 14607 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE INTOPLICINE INTOPLICINE 21459 14608 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SJ000071821 CHEMBL589924 21461 14609 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE ENMD-2076 ENMD-2076 21462 14610 ALOX15 246 ENZYME, DRUGGABLE GENOME SANGUINARINE SULFATE SANGUINARINE SULFATE 21464 14611 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER VEGF 11720743,15579019 21465 14612 HDAC11 79885 DRUGGABLE GENOME, ENZYME PMID29671355-Compound-43 21466 14613 GPER1 2852 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR antagonist 178103094 21467 14614 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME MYRICETIN MYRICETIN 21469 14615 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE BEPRIDIL BEPRIDIL 21470 14616 CPA2 1358 PROTEASE, ENZYME, DRUGGABLE GENOME asparaginase ASPARAGINASE 27114598 21471 14617 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME KANZONOL X KANZONOL X 20022509 21472 14618 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR R-ETODOLAC 21474 14619 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME CS-7017 EFATUTAZONE HYDROCHLORIDE 21475 14620 GLA 2717 ENZYME, DRUGGABLE GENOME L-GLUTAMIC ACID, N-PHTHALOYL CHEMBL1256390 21476 14621 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000113257 CHEMBL528694 21478 14622 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SOTRASTAURIN SOTRASTAURIN 21480 14623 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545168 IMD-1041 21481 14624 KDM4A 9682 DRUGGABLE GENOME, ENZYME THIETHYLPERAZINE MALATE THIETHYLPERAZINE MALATE 21482 14625 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 375973251 21483 14626 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PIFITHRIN-MU CHEMBL1241268 16862141 21488 14627 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33j 21490 14628 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 405560192 21492 14629 SMARCB1 6598 CLINICALLY ACTIONABLE Tazemetostat TAZEMETOSTAT 26360609,23620515 21495 14630 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PENTOXIFYLLINE PENTOXIFYLLINE 21496 14631 CEACAM1 634 KINASE, CELL SURFACE, DRUGGABLE GENOME RETINOID 8609714 21497 14632 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-42 21498 14633 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650834 21499 14634 PPID 5481 DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING, KINASE SCY-635 SCY 635 21500 14635 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 L-162313 CHEMBL288174 21501 14636 HTT 3064 DRUGGABLE GENOME JNJ-26481585 QUISINOSTAT 21502 14637 POLK 51426 DNA REPAIR, ENZYME ARACHIDONOYL GABA ARACHIDONOYL GABA 21504 14638 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE (+/-)-HYDNOCARPIN CHEMBL91638 24018191 21505 14639 APH1B 83464 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL1090771 AVAGACESTAT 21506 14640 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME QUINALIZARIN QUINALIZARIN 21508 14641 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE GO-6976 GO-6976 21511 14642 ALOX15 246 ENZYME, DRUGGABLE GENOME Imidazole derivative 11 21512 14643 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME TANDUTINIB TANDUTINIB 21513 14644 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ANTHRACENE-9-CARBOXYLIC ACID ANTHRACENE-9-CARBOXYLIC ACID 21517 14645 APC 324 CLINICALLY ACTIONABLE iCRT-14 21393571 21519 14646 SMN2 6607 DRUGGABLE GENOME NSC-234945 CHEMBL260311 21521 14647 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME PMID28270010-Compound-Figure24-b 21522 14648 TUBA3C 7278 DRUGGABLE GENOME ABT-751 ABT-751 25468039 21523 14649 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TERFENADINE TERFENADINE 21524 14650 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME APTIGANEL APTIGANEL 21525 14651 SMN1 6606 DRUGGABLE GENOME FORMONONETIN FORMONONETIN 21528 14652 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE US8614253, 32-5 21530 14653 ALOX15 246 ENZYME, DRUGGABLE GENOME EBSELEN EBSELEN 21531 14654 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic-carboxamide derivative 2 21533 14655 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME METHDILAZINE METHDILAZINE 21535 14656 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BAICALEIN BAICALEIN 21536 14657 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME GOSSYPOL GOSSYPOL 21537 14658 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL HALAZEPAM HALAZEPAM 21538 14659 TNFRSF1A 7132 CELL SURFACE, DRUGGABLE GENOME CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 9894568 21539 14660 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 374883888 21541 14661 GJB4 127534 ION CHANNEL inhibitor 135652731 21542 14662 PREP 5550 PROTEASE, ENZYME, DRUGGABLE GENOME S-17092-1 21544 14663 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051826 21545 14664 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME CYC-116 CYC-116 21546 14665 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE RETEPLASE RETEPLASE 21547 14666 PTGS2 5743 DRUGGABLE GENOME, ENZYME CIMICOXIB CIMICOXIB 21549 14667 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR LINOLENIC ACID LINOLENIC ACID 21550 14668 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR docetaxel DOCETAXEL 24193570 21551 14669 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051803 21553 14670 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR MLN-8054 MLN-8054 21555 14671 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL270190 ALVIMOPAN 21556 14672 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2',3,4-TRIHYDROXYCHALCONE CHEMBL339587 21559 14673 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME BENZOHYDROXAMATE BENZOHYDROXAMATE 23368884,25937017 21560 14674 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9216972, 61 21561 14675 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GRAMINE GRAMINE 21564 14676 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-74429 CHEMBL1269022 21565 14677 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Ro 31-7453 21566 14678 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE HOMIDIUM BROMIDE HOMIDIUM BROMIDE 21570 14679 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Bevacizumab BEVACIZUMAB 27893038,23940356,21216929,25363205 21571 14680 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME DEMETHYLWEDELOLACTONE DEMETHYLWEDELOLACTONE 22926226 21572 14681 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Selective serotonin reuptake inhibitors 24930681 21574 14682 KNG1 3827 DRUGGABLE GENOME, PROTEASE INHIBITOR hormonal contraceptives for systemic use 28750087 21575 14683 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649703 21577 14684 CBX1 10951 NA NSC-228155 CHEMBL505670 21578 14685 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650858 PROPRANOLOL 21580 14686 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201662 DESIRUDIN 21581 14687 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME MYCOPHENOLATE MOFETIL 11750393 21582 14688 ATAD5 79915 NA CYCLOASPEPTIDE A CYCLOASPEPTIDE A 21583 14689 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Benzothiazepine analog 11 21585 14690 TUBB 203068 DRUGGABLE GENOME T-607 21589 14691 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650558 LY-510929 21592 14692 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME DOVITINIB DOVITINIB 21593 14693 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER propafenone PROPAFENONE 21597 14694 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME GABOXADOL GABOXADOL 21600 14695 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1280 VERAPAMIL HYDROCHLORIDE 21601 14696 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200914 TAMSULOSIN HYDROCHLORIDE 21603 14697 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-US20130053382 35(1-11) 21604 14698 CA12 771 DRUGGABLE GENOME COUMATE 21605 14699 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650083 21608 14700 DBP 1628 TRANSCRIPTION FACTOR ALBUMIN ALBUMIN HUMAN 2331750 21610 14701 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4237 CHEMBL600701 21613 14702 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GA201 IMGATUZUMAB 23209031 21614 14703 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ILORASERTIB ILORASERTIB 21617 14704 CD27 939 PROTEASE INHIBITOR, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME N/A 21618 14705 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Alkylating Agents 25545243,24533712,11160862,21479364,10208650,21946896,18511948 21620 14706 HTT 3064 DRUGGABLE GENOME LAURYL ISOQUINOLINIUM LAURYL ISOQUINOLINIUM 21621 14707 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME desmethyl clomipramine 28470111 21622 14708 ALB 213 TRANSPORTER, DRUGGABLE GENOME EPIGALLOCATECHIN EPIGALLOCATECHIN 20598557 21623 14709 SLC15A1 6564 DRUGGABLE GENOME, TRANSPORTER hmg coa reductase inhibitors 21624 14710 IRS2 8660 KINASE, CLINICALLY ACTIONABLE DEXAMETHASONE DEXAMETHASONE 16943575 21625 14711 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR NORSTICTIC ACID NORSTICTIC ACID 21627 14712 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME UCN-01 UCN-01 15255949 21628 14713 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Peptide analog 48 21629 14714 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-107 CHEMBL578675 21630 14715 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 249565749 21631 14716 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1201831 CERTOLIZUMAB PEGOL 21633 14717 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME evodiamine EVODIAMINE 21647174 21635 14718 POLI 11201 DNA REPAIR 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 21636 14719 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 LOVASTATIN LOVASTATIN 22931300 21637 14720 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LEUPROLIDE LEUPROLIDE 29211833 21638 14721 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME (S)-FLUOXETINE CHEMBL1169388 21640 14722 EPHX1 2052 ENZYME, DRUGGABLE GENOME phenytoin PHENYTOIN 19952982 21641 14723 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MENADIONE MENADIONE 21642 14724 PTK6 5753 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, ENZYME TAE-684 TAE-684 21643 14725 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 fluoxetine FLUOXETINE 21645 14726 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BENZYL ISOTHIOCYANATE BENZYL ISOTHIOCYANATE 21646 14727 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE Sirolimus SIROLIMUS 20142330 21647 14728 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE TAMATINIB R-406 21648 14729 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR GNF-PF-1947 CHEMBL585591 21649 14730 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE inhibitor 178103128 21650 14731 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 21651 14732 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651426 ADENOSINE 21653 14733 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE FLUFENAMIC ACID FLUFENAMIC ACID 21654 14734 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CLIOQUINOL CLIOQUINOL 21657 14735 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650806 21658 14736 SDHB 6390 ENZYME, CLINICALLY ACTIONABLE CORTICOSTEROIDS 1537729 21659 14737 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 21662 14738 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME FLUOXETINE FLUOXETINE 21663 14739 ALPI 248 DRUGGABLE GENOME, ENZYME AG-538 CHEMBL56393 21665 14740 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3876 CHEMBL596631 21666 14741 USP1 7398 DNA REPAIR, PROTEASE, ENZYME NSC-693571 CHEMBL1287983 21668 14742 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL1908397 KW-2449 21669 14743 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE sibutramine SIBUTRAMINE 18695978 21670 14744 LAMA5 3911 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 21674 14745 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200996 MEPHENTERMINE SULFATE 21675 14746 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE ALSTERPAULLONE ALSTERPAULLONE 21676 14747 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor AUY922 21678 14748 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE Selumetinib SELUMETINIB 22550165 21681 14749 HSPA4 3308 NA CISPLATIN CISPLATIN 11478701 21682 14750 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL3707400 INDANTADOL 21684 14751 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER tetracycline TETRACYCLINE 21685 14752 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE LINIFANIB LINIFANIB 21686 14753 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051805 QUISINOSTAT 21687 14754 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8669361, 105 21688 14755 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE ANTITHROMBIN 21690 14756 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE SORAFENIB SORAFENIB 22357254,17699867,19461405 21691 14757 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE EGFR TYROSINE KINASE INHIBITOR 12576461 21692 14758 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY BETHANECHOL CHLORIDE 449696 21693 14759 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR MEFENAMIC ACID MEFENAMIC ACID 21694 14760 NOS1 4842 DRUGGABLE GENOME, ENZYME POLYESTRADIOL PHOSPHATE 10096401 21695 14761 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SJ000295151 CHEMBL590660 21696 14762 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER propofol PROPOFOL 29755652 21697 14763 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE LAS 100977 21698 14764 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE DOVITINIB DOVITINIB 21699 14765 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME RETIGABINE EZOGABINE 21703 14766 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TEBUFENOZIDE TEBUFENOZIDE 21704 14767 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR SEMAPIMOD SEMAPIMOD 21705 14768 GMNN 51053 DRUGGABLE GENOME CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 21706 14769 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1200585 OXYMETHOLONE 21707 14770 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 405560388 21709 14771 ACAT1 38 ENZYME ATR-01 21711 14772 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME TYRPHOSTIN 23 TYRPHOSTIN 23 21713 14773 MVK 4598 KINASE, ENZYME inhibitor 135651580 21715 14774 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME HOMIDIUM BROMIDE HOMIDIUM BROMIDE 21717 14775 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME ELTROMBOPAG ELTROMBOPAG 21422191 21723 14776 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor AT9283 AT-9283 21724 14777 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Enzalutamide ENZALUTAMIDE 25544636 21725 14778 PSMD11 5717 KINASE inhibitor CHEMBL3545432 IXAZOMIB CITRATE 21726 14779 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIHYDROGAMBOGIC ACID DIHYDROGAMBOGIC ACID 21727 14780 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALCITRIOL CALCITRIOL 22285943,19309155,24818857,20452225,20883026 21730 14781 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TECHTOCHRYSIN TECHTOCHRYSIN 21731 14782 RGS12 6002 DRUGGABLE GENOME MMV009085 CHEMBL581225 21732 14783 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 135652717 STAUROSPORINE 21733 14784 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1879463 DACTOLISIB 21736 14785 DYNC2H1 79659 CLINICALLY ACTIONABLE Platinum compounds 21118971 21737 14786 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 249565684 21738 14787 CRBN 51185 ENZYME, DRUG RESISTANCE 178103903 LENALIDOMIDE 21739 14788 CD69 969 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ANTITUMOR ANTIBIOTICS 11811939 21740 14789 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650783 21743 14790 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME inhibitor 178103148 21744 14791 GMNN 51053 DRUGGABLE GENOME DNDI1417548 CHEMBL2094789 21745 14792 ALOX15 246 ENZYME, DRUGGABLE GENOME CHAULMOOGRIC ACID, ETHYL ESTER CHAULMOOGRIC ACID, ETHYL ESTER 21746 14793 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ANDROSTENEDIOL ANDROSTENEDIOL 21747 14794 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor TEMSIROLIMUS TEMSIROLIMUS 21748 14795 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE Pyrimidopyridazinone derivative 1 21749 14796 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE PF-562271 PF-00562271 21751 14797 PSMA6 5687 PROTEASE, DRUGGABLE GENOME inhibitor CARFILZOMIB CARFILZOMIB 21752 14798 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR INOC-005 21753 14799 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZOXYSTROBIN AZOXYSTROBIN 21754 14800 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR Diamidothiazole derivative 1 21755 14801 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor CHEMBL3545332 CEP-2563 21760 14802 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DIPHENYLENEIODONIUM DIPHENYLENEIODONIUM 21763 14803 PRKCH 5583 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE BRYOSTATIN-1 21764 14804 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME dabrafenib DABRAFENIB 27023328 21766 14805 GMNN 51053 DRUGGABLE GENOME AROMATICIN AROMATICIN 21767 14806 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME PYRONIN Y PYRONIN Y 21769 14807 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CYC-116 CYC-116 21773 14808 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME AR-A014418 CHEMBL259850 21774 14809 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME CLOMIPHENE CITRATE 12012626 21775 14810 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-124022 CHEMBL548017 21776 14811 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CAPSAICIN CAPSAICIN 21777 14812 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HC-Toxin 21778 14813 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Imidazo[4,5-c]pyridine derivative 1 21779 14814 ATXN2 6311 NA SJ000012773 CHEMBL589715 21780 14815 CXCL8 3576 DRUGGABLE GENOME sunitinib SUNITINIB 26387812 21782 14816 EIF4E 1977 DRUGGABLE GENOME MTOR INHIBITOR 15190216 21783 14817 USP1 7398 DNA REPAIR, PROTEASE, ENZYME HEXYLRESORCINOL HEXYLRESORCINOL 21785 14818 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor MGCD265 GLESATINIB 21786 14819 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER doxycycline DOXYCYCLINE 21787 14820 PPP3CA 5530 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Tacrolimus TACROLIMUS 21789 14821 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Telcagepant TELCAGEPANT 21790 14822 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 6-O-BENZYLGUANINE 6-O-BENZYLGUANINE 21792 14823 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor GSK2636771 GSK-2636771 21793 14824 PTPRS 5802 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE, CLINICALLY ACTIONABLE Etidronic acid 21795 14825 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Imatinib IMATINIB 18795925,15790786,21689725,26316776,27370604,24317392,25673643,26687836,15236194,15201427,27980106,12481435,25015329,28611108,19861435,25594040,21969494,28196207,24419427,25003536,23567324,25239608,19812602,20372153,12374669,18751412,16954519,16015387,16462496,16751810,23582185,27777285,28334365 21798 14826 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX KAEMPFEROL KAEMPFEROL 25190466 21800 14827 SMN2 6607 DRUGGABLE GENOME PICEATANNOL PICEATANNOL 21802 14828 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL ETOMIDATE ETOMIDATE 16884293 21803 14829 POLI 11201 DNA REPAIR NSC-133896 CHEMBL512908 21805 14830 PLTP 5360 DRUGGABLE GENOME ALPHA-TOCOPHEROL VITAMIN E 15576481,10224231 21807 14831 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 amitriptyline AMITRIPTYLINE 9187528 21808 14832 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DUAL IGF-1R/INSR INHIBITOR BMS-754807 25527633 21809 14833 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CA19-9 ANTIGEN 1394194 21810 14834 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR ARDEPARIN 21812 14835 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME vaccine RAS PEPTIDE CANCER VACCINE 21813 14836 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BROTIZOLAM BROTIZOLAM 21814 14837 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2011000295210 21815 14838 TMEM97 27346 NA Benzamide derivative 10 21817 14839 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-3 21818 14840 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE AZD6482 AZD-6482 26504226,23674493,26577700 21820 14841 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE DIGITOXIN DIGITOXIN 21821 14842 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4-AMINOPHENOL 4-AMINOPHENOL 21823 14843 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Aryl pyrimidine derivative 1 21825 14844 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 381744995 SELITRECTINIB 21826 14845 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TIRATRICOL TIRATRICOL 21828 14846 PLCB1 23236 ENZYME, DRUGGABLE GENOME, PHOSPHOLIPASE Selective serotonin reuptake inhibitors 25649181 21829 14847 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL598797 CUDC-101 21830 14848 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL2165191 AZD-6482 21831 14849 GJA1 2697 ION CHANNEL inhibitor 178100972 CARBENOXOLONE 21833 14850 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Conjugated 3-(indolyl)-and 3-(azaindolyl)-4-arylmaleimide compound 1 21835 14851 SCNN1A 6337 DRUGGABLE GENOME, ION CHANNEL TRIAMTERENE TRIAMTERENE 21836 14852 PTGS2 5743 DRUGGABLE GENOME, ENZYME NAPROXEN ETEMESIL 21837 14853 IRF2 3660 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IFN 16241857,16533423 21840 14854 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL Ethchlorvynol ETHCHLORVYNOL 21841 14855 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AZEPEXOLE AZEPEXOLE 21842 14856 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 223366033 21843 14857 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE lamivudine LAMIVUDINE 21845 14858 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DINALINE DINALINE 21846 14859 MKNK1 8569 SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 178102632 21847 14860 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME 1,2,4-triazolo[1,5a]pyridine derivative 1 21848 14861 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BLEOMYCIN BLEOMYCIN 11489978 21849 14862 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME BAS03450373 CHEMBL1576310 21850 14863 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-G5 21851 14864 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE AXITINIB AXITINIB 21853 14865 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651289 21854 14866 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ALVESPIMYCIN ALVESPIMYCIN 21855 14867 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME JNJ-7706621 JNJ-7706621 21856 14868 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-28 21857 14869 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PHOSPHATIDYLINOSITIDE 3-KINASE INHIBITOR 25002028 21858 14870 TMEM97 27346 NA Isoindoline derivative 5 21859 14871 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 249565704 LONAFARNIB 21860 14872 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER Deutetrabenazine DEUTETRABENAZINE 21861 14873 VKORC1 79001 DRUGGABLE GENOME, ENZYME ACENOCOUMAROL ACENOCOUMAROL 21865 14874 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TCMDC-125317 CHEMBL528373 21868 14875 SLC15A1 6564 DRUGGABLE GENOME, TRANSPORTER inhibitor 178101414 21869 14876 DGAT1 8694 ENZYME, DRUGGABLE GENOME LCQ908 21871 14877 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 363894197 CT-7001 21874 14878 CBX1 10951 NA EMODIN EMODIN 21875 14879 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR STROPHANTHIDIN ACETATE STROPHANTHIDIN ACETATE 21876 14880 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3707249 ASM-024 21877 14881 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PI-CLONIDINE PI-CLONIDINE 21880 14882 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 5-DEMETHYLNOBILETIN 5-DEMETHYLNOBILETIN 21882 14883 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE PD-332991 21883 14884 S100A4 6275 NA SP-MET-1 21884 14885 USP1 7398 DNA REPAIR, PROTEASE, ENZYME MESALAMINE MESALAMINE 21885 14886 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-139459 CHEMBL86464 21887 14887 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR DABRAFENIB DABRAFENIB 24265155 21888 14888 FZD1 8321 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, KINASE GNF-PF-3411 CHEMBL593726 23453073 21889 14889 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR GTI-2501 21890 14890 RIPK3 11035 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 384403666 21891 14891 SPP1 6696 DRUGGABLE GENOME RETINOIC ACID 9224725 21893 14892 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Triazole derivative 4 21898 14893 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR trastuzumab TRASTUZUMAB 21899 14894 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OXYCODONE OXYCODONE 21902 14895 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Triciribine TRICIRIBINE 20644979 21903 14896 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CISPLATIN CISPLATIN 12438277 21904 14897 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NEFAZODONE NEFAZODONE 21905 14898 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME BML-210 CHEMBL324053 16921367 21906 14899 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 340590228 ROVELIZUMAB 21907 14900 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR atenolol ATENOLOL 11593098,14700505 21908 14901 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MEPERIDINE MEPERIDINE 21909 14902 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME LINIFANIB LINIFANIB 21911 14903 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL738 THIOPENTAL SODIUM 21912 14904 USP1 7398 DNA REPAIR, PROTEASE, ENZYME AMBAZONE AMBAZONE 21913 14905 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ROSE BENGAL ROSE BENGAL 21914 14906 TOP2B 7155 DRUGGABLE GENOME, ENZYME Liposomal encapsulated doxorubicin (LED) 21915 14907 ATAD5 79915 NA STREPTONIGRIN STREPTONIGRIN 21917 14908 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIMETHYL FUMARATE DIMETHYL FUMARATE 23647822 21918 14909 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PKI-179 PKI-179 20797855 21920 14910 OGA 10724 ENZYME, DRUGGABLE GENOME MK 8719 21921 14911 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Pyrazolopyridine derivative 5 21922 14912 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW627512B GW627512B 21923 14913 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE sorafenib SORAFENIB 22912756,28362716 21926 14914 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SAQUINAVIR MESYLATE SAQUINAVIR MESYLATE 21928 14915 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PROGESTERONE PROGESTERONE 15350188 21929 14916 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME THIETHYLPERAZINE THIETHYLPERAZINE 21930 14917 COL5A1 1289 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 21932 14918 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102479 CHEMBL196779 21933 14919 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE FLOXURIDINE FLOXURIDINE 21934 14920 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Antroquinonol ANTROQUINONOL 21935 14921 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME INSULIN ASPART 21936 14922 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE DEMETHYLWEDELOLACTONE DEMETHYLWEDELOLACTONE 22926226 21937 14923 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NOVIFLUMURON NOVIFLUMURON 21938 14924 SYP 6855 TRANSPORTER DIMETHYL SULFOXIDE 2512391 21939 14925 HTT 3064 DRUGGABLE GENOME OBP-801 OBP-801 21941 14926 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor BGJ398 INFIGRATINIB 21942 14927 UGCG 7357 ENZYME, DRUGGABLE GENOME MIGLUSTAT MIGLUSTAT 21943 14928 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Cetuximab CETUXIMAB 23729478 21944 14929 PTGS2 5743 DRUGGABLE GENOME, ENZYME valdecoxib VALDECOXIB 19602986 21945 14930 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-61 21946 14931 APC 324 CLINICALLY ACTIONABLE CCT031374 20610623 21947 14932 BRDT 676 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE inhibitor 187051813 21948 14933 BRCA2 675 CLINICALLY ACTIONABLE AZD2461 27550455 21951 14934 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE EOTAXIN 11358986 21953 14935 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BI-87E7 CHEMBL523200 21954 14936 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE THONZONIUM BROMIDE THONZONIUM BROMIDE 21956 14937 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FERROUS SULFATE FERROUS SULFATE 22931300 21957 14938 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME cyclophosphamide CYCLOPHOSPHAMIDE 19786980,25008867,21362365,22188361,20568049 21958 14939 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178101060 21959 14940 DHRS9 10170 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE SESQUITERPENE O-BENZOQUINONE CHEMBL517425 19188072 21960 14941 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING STICTIC ACID STICTIC ACID 21961 14942 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME KENPAULLONE KENPAULLONE 21962 14943 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME TOSITUMOMAB TOSITUMOMAB 21963 14944 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR CIRAZOLINE CIRAZOLINE 21964 14945 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-P6 21965 14946 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PMID27376512-Compound-MTC-427 21969 14947 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545006 PWT-33587 21970 14948 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHRYSIN CHRYSIN 19592245 21971 14949 ATAD5 79915 NA CID 94381 CHEMBL374632 21972 14950 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor GDC-0068 IPATASERTIB 21975 14951 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651573 LIOTHYRONINE SODIUM 21976 14952 RACGAP1 29127 NA XAMOTEROL FUMARATE XAMOTEROL FUMARATE 21977 14953 GAA 2548 DRUGGABLE GENOME, ENZYME BMN-701 REVEGLUCOSIDASE ALFA 21978 14954 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE APC-100 APC-100 21979 14955 GBA 2629 DRUGGABLE GENOME, ENZYME ISOLIQUIRITIGENIN ISOLIQUIRITIGENIN 21982 14956 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL796 METHYLPHENIDATE 21983 14957 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL valproic acid 23407051 21984 14958 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200464 PROPARACAINE HYDROCHLORIDE 21985 14959 MGLL 11343 DRUGGABLE GENOME, ENZYME Pyrazole derivative 83 21988 14960 GAA 2548 DRUGGABLE GENOME, ENZYME ALFUZOSIN ALFUZOSIN 21992 14961 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL23261 DARUSENTAN 21995 14962 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 flibanserin FLIBANSERIN 21996 14963 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 21997 14964 XDH 7498 DRUGGABLE GENOME, ENZYME POLYPHENOL 12694877 21998 14965 GMNN 51053 DRUGGABLE GENOME 3,4-DICHLOROISOCOUMARIN CHEMBL24983 21999 14966 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR TAK-733 TAK-733 22000 14967 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AMG 232 25567130,26162687 22001 14968 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME CER-001 22002 14969 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE Cyclolignan picropodophyllin 22003 14970 NCOA1 8648 ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 22005 14971 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE ILORASERTIB ILORASERTIB 22006 14972 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650057 CARVEDILOL 22007 14973 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyrrolo-pyrimidine derivative 8 22009 14974 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR BELINOSTAT BELINOSTAT 25937017 22012 14975 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER TANGERETIN TANGERETIN 22015 14976 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CEDIRANIB CEDIRANIB 22017 14977 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CLOSANTEL CLOSANTEL 22018 14978 POLK 51426 DNA REPAIR, ENZYME LOMOFUNGIN LOMOFUNGIN 22019 14979 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE COLFORSIN COLFORSIN 22020 14980 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 22021 14981 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102334 22023 14982 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE cisplatin CISPLATIN 22024 14983 XDH 7498 DRUGGABLE GENOME, ENZYME OXYPURINOL OXYPURINOL 22026 14984 METAP1 23173 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL2103847 TOSEDOSTAT 22028 14985 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR fenofibrate FENOFIBRATE 15608561 22029 14986 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 223365983 RIVOCERANIB 22030 14987 CSF1 1435 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RG7155 22031 14988 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME blocker 135652746 22033 14989 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DNDI1417171 CHEMBL1438389 22034 14990 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Ponatinib PONATINIB 22035 14991 POLB 5423 DNA REPAIR, DRUGGABLE GENOME MYRICETIN MYRICETIN 22037 14992 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1752 DYPHYLLINE 22038 14993 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist CHEMBL1908373 ONAPRISTONE 22039 14994 TNFRSF1B 7133 DRUGGABLE GENOME ACTINOMYCIN D 11125300 22040 14995 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 178102314 IMATINIB 22042 14996 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ANISOCOUMARIN H ANISOCOUMARIN H 22043 14997 ATXN1L 342371 DRUG RESISTANCE VEMURAFENIB VEMURAFENIB 28178529 22044 14998 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LOSARTAN LOSARTAN 22045 14999 XDH 7498 DRUGGABLE GENOME, ENZYME Azole benzene derivative 3 22046 15000 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE CAMPTOTHECIN CAMPTOTHECIN 8938795 22048 15001 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c][1,2,4]benzotriazine derivative 3 22049 15002 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PHENSERINE PHENSERINE 22050 15003 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Peptidomimetic analog 2 22051 15004 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MECLOFENAMATE SODIUM MECLOFENAMATE SODIUM 22052 15005 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL87992 ESLICARBAZEPINE ACETATE 22053 15006 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 22054 15007 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME R-flurbiprofen 22056 15008 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545366 VOXTALISIB 22058 15009 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 HESPERETIN HESPERETIN 22060 15010 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR Chenodiol CHENODIOL 22061 15011 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-4068 CHEMBL584668 22063 15012 POLK 51426 DNA REPAIR, ENZYME 4-BENZAMIDOPHENYLSTIBONIC ACID CHEMBL1726814 22065 15013 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 310264780 22066 15014 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE N6-METHYLADENOSINE CHEMBL383144 22067 15015 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE formoterol FORMOTEROL 22068 15016 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BAY80-6946 COPANLISIB 22069 15017 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650278 FLUSPIRILENE 22073 15018 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 381118891 22074 15019 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 178101018 22075 15020 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 53801089 HYDROCORTISONE 22076 15021 KMO 8564 DRUGGABLE GENOME, ENZYME Benzene sulfonamide derivative 2 22078 15022 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL2107762 NERISPIRDINE 22080 15023 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL1201748 CABAZITAXEL 22082 15024 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BYL719 ALPELISIB 22084 15025 SGMS2 166929 KINASE, ENZYME inhibitor 375973242 22089 15026 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME LAK 3489774 22090 15027 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545396 BMS-690514 22092 15028 GAA 2548 DRUGGABLE GENOME, ENZYME HONOKIOL HONOKIOL 22094 15029 MPHOSPH8 54737 NA MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 22095 15030 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1522 ESZOPICLONE 22096 15031 GC 2638 DRUGGABLE GENOME VITAMIN D 761406 22097 15032 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178101336 22099 15033 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL544665 FINGOLIMOD HYDROCHLORIDE 22100 15034 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME CAPTOPRIL CAPTOPRIL 2864479 22105 15035 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Carboplatin-Taxol Regimen 22106 15036 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX PD-98059 CHEMBL35482 15385570 22107 15037 ATAD5 79915 NA GNF-PF-4590 CHEMBL529361 22108 15038 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Tyverb/Tykerb 22109 15039 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BUTYLATED HYDROXYTOLUENE BUTYLATED HYDROXYTOLUENE 22931300 22110 15040 NAAA 27163 ENZYME, DRUGGABLE GENOME inhibitor 315661261 22111 15041 IL1B 3553 KINASE, DRUGGABLE GENOME CEFACLOR CEFACLOR 3260587 22113 15042 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000032159 CHEMBL591361 22114 15043 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DIENESTROL DIENESTROL 22115 15044 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102641 22117 15045 CMKLR1 1240 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CCX832 22118 15046 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 6-10 22123 15047 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE BKM120 BUPARLISIB 22124 15048 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL254219 DIGITOXIN 22125 15049 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ISOQUINE ISOQUINE 22127 15050 SMN1 6606 DRUGGABLE GENOME PHENYLBUTYRATE PHENYLBUTANOIC ACID 14560316 22129 15051 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL628 PENTOXIFYLLINE 22130 15052 HTT 3064 DRUGGABLE GENOME Aniline derivative 1 22131 15053 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL3545252 DOCETAXEL 22135 15054 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER RITONAVIR RITONAVIR 11745741 22136 15055 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PALBOCICLIB PALBOCICLIB 22137 15056 TNFSF13 8741 DRUGGABLE GENOME Atacicept ATACICEPT 22138 15057 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2108887 AFELIMOMAB 22139 15058 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME FENRETINIDE FENRETINIDE 22142 15059 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 695758 CHEMBL260028 22143 15060 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE fluorouracil FLUOROURACIL 24980946 22144 15061 NDUFAB1 4706 NA inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 22145 15062 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3265032 ENTOSPLETINIB 22146 15063 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 387065608 22147 15064 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200461 MIDODRINE HYDROCHLORIDE 22148 15065 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Tricyclic isoxazoloquinazoline derivative 1 22150 15066 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE JUGLONE JUGLONE 22152 15067 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE glipizide GLIPIZIDE 22154 15068 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME 2-O, 3-O DESULFATED HEPARIN 22155 15069 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102251 CHEMBL375293 22156 15070 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE IROFULVEN IROFULVEN 17229870 22157 15071 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE PALBOCICLIB PALBOCICLIB 24417566 22159 15072 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-159 CHEMBL599924 22160 15073 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX 4-AMINOPHENOL 4-AMINOPHENOL 22163 15074 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE MK2206 MK-2206 22166 15075 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-137788 CHEMBL587564 22167 15076 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Rogaratinib ROGARATINIB 22168 15077 PTGS1 5742 ENZYME, DRUGGABLE GENOME Salsalate SALSALATE 22169 15078 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PENBUTOLOL PENBUTOLOL 22170 15079 PIKFYVE 200576 SERINE THREONINE KINASE, ENZYME, KINASE LAM-002 22171 15080 ACAT1 38 ENZYME inhibitor 381118860 22172 15081 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 135650300 GENISTEIN 22173 15082 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Carbamazepine CARBAMAZEPINE 22174 15083 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TELMISARTAN TELMISARTAN 22176 15084 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Cetirizine CETIRIZINE 22177 15085 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER EPIRUBICIN EPIRUBICIN 15161039 22178 15086 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NICLOSAMIDE NICLOSAMIDE 22179 15087 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 381118815 22182 15088 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 22183 15089 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLOTIAZEPAM CLOTIAZEPAM 22184 15090 NTS 4922 DRUGGABLE GENOME NORETHISTERONE NORETHINDRONE 11495683 22186 15091 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME SAR245409 VOXTALISIB 22189 15092 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME GW441756X GW441756X 22190 15093 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE IDEBENONE IDEBENONE 22191 15094 FAAH 2166 ENZYME, DRUGGABLE GENOME Azole derivative 5 22192 15095 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545133 JNJ-26483327 22193 15096 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME Mesothelin-targeted T cells 22194 15097 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR CHONDROITIN SULFATE 10959709 22197 15098 GUCY1B1 2983 DRUGGABLE GENOME RIOCIGUAT RIOCIGUAT 22198 15099 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME DEQUALINIUM DEQUALINIUM 22201 15100 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MINERAL OIL 14741172 22202 15101 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Ajmalicine 22203 15102 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER OC144-093 22206 15103 CD38 952 CELL SURFACE, DRUGGABLE GENOME MOR-202 22207 15104 TUBB6 84617 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 22209 15105 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545212 AMG-337 22210 15106 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME 6-METHOXYCOMAPARVIN CHEMBL401565 18088098 22211 15107 CSNK1G3 1456 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME TAK-715 TAK-715 22212 15108 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER methylphenidate METHYLPHENIDATE 23771192 22214 15109 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME PMID25468267-Compound-46 22218 15110 MUC16 94025 DRUGGABLE GENOME opioids 22222 15111 ATXN2 6311 NA VANOXERINE VANOXERINE 22227 15112 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME PENTABROMOPHENOL PENTABROMOPHENOL 22229 15113 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Afatinib AFATINIB 22230 15114 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BENZHYDRYL 4-HYDROXYBENZOATE CHEMBL2071180 22647217 22231 15115 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE GEMCITABINE GEMCITABINE 12684687 22232 15116 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE DOVITINIB DOVITINIB 22233 15117 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE ENMD-2076 ENMD-2076 22234 15118 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE TUMOR NECROSIS FACTOR 14764603 22235 15119 CRP 1401 DRUGGABLE GENOME adalimumab ADALIMUMAB 27096233 22236 15120 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ENDOSULFAN ENDOSULFAN 22237 15121 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYLDOPA METHYLDOPA 22239 15122 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME RUCAPARIB RUCAPARIB 22240 15123 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR SELECTIVE ESTROGEN RECEPTOR MODULATOR 11901050 22241 15124 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 348353622 22242 15125 CA1 759 DRUGGABLE GENOME, ENZYME Methazolamide METHAZOLAMIDE 22243 15126 MAPT 4137 DRUGGABLE GENOME HOMIDIUM BROMIDE HOMIDIUM BROMIDE 22244 15127 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ACETANILIDE ACETANILIDE 22245 15128 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR inhibitor 381744997 REPOTRECTINIB 22246 15129 GMNN 51053 DRUGGABLE GENOME DESOGESTREL DESOGESTREL 22247 15130 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NICERGOLINE NICERGOLINE 22248 15131 TUBA1A 7846 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 22249 15132 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ribavirin RIBAVIRIN 23360626,12873589 22250 15133 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE GNF-PF-2272 CHEMBL601757 22252 15134 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL538943 VINORELBINE TARTRATE 22253 15135 POLI 11201 DNA REPAIR 2-AMINOPHENOXAZINONE CHEMBL146710 22254 15136 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178104008 MILNACIPRAN 22256 15137 ADRM1 11047 ENZYME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 22257 15138 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME CLOZAPINE CLOZAPINE 15659539 22260 15139 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MEPHENTERMINE MEPHENTERMINE 22261 15140 PSMB6 5694 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CARFILZOMIB CARFILZOMIB 22262 15141 TUBA1C 84790 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 22263 15142 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHOXYCHLOR METHOXYCHLOR 22264 15143 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Bicyclic heteroaryl benzamide derivative 8 22266 15144 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL OXAZEPAM OXAZEPAM 22267 15145 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME PROTEIN PHOSPHATASE INHIBITOR 12952980 22268 15146 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME FLAVONE FLAVONE 22269 15147 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 rucaparib RUCAPARIB 22270 15148 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NAFTIDROFURYL NAFTIDROFURYL 22271 15149 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CA-4948 22273 15150 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE SEROTONIN SEROTONIN 22274 15151 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-26 22275 15152 MAOB 4129 DRUGGABLE GENOME, ENZYME Coumarin/resveratrol hybrid derivative 2 22276 15153 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor 178103944 APREMILAST 22277 15154 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 178102645 22279 15155 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 3-METHOXY-MORPHANIN HCL CHEMBL1257022 22280 15156 CASP2 835 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL197672 EMRICASAN 22281 15157 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL2178422 RIMEGEPANT 22282 15158 ALOX5 240 DRUGGABLE GENOME, ENZYME MECLOFENAMIC ACID 22284 15159 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE STREPTOKINASE STREPTOKINASE 22286 15160 XDH 7498 DRUGGABLE GENOME, ENZYME CHINESE HERBS 3007357 22287 15161 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Five membered heterocyclic benzamide derivative 1 22288 15162 BAZ2B 29994 NA GNF-PF-4542 CHEMBL585999 22289 15163 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AMINACRINE HYDROCHLORIDE AMINACRINE HYDROCHLORIDE 22290 15164 CENPE 1062 KINASE inhibitor GSK-923295 22291 15165 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZD5363 CAPIVASERTIB 26351323,26931343,28376212,28489509 22292 15166 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2103884 OPROZOMIB 22293 15167 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Travoprost TRAVOPROST 22294 15168 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME LINIFANIB LINIFANIB 22295 15169 POLK 51426 DNA REPAIR, ENZYME 2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE 2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE 22296 15170 CAPN1 823 PROTEASE, DRUGGABLE GENOME, ENZYME Undecylenic acid derivative 1 22298 15171 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 252166682 22303 15172 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201013 OLSALAZINE SODIUM 22306 15173 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR IL-6 10994633 22307 15174 COL4A4 1286 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 22308 15175 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME MLN-8054 MLN-8054 22309 15176 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 diclofenac DICLOFENAC 15861034 22311 15177 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TESTOSTERONE TESTOSTERONE 22312 15178 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME IDM-2101 22313 15179 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3218576 COPANLISIB 22314 15180 ATXN2 6311 NA CHLORPROMAZINE HYDROCHLORIDE CHLORPROMAZINE HYDROCHLORIDE 22315 15181 KDM5B 10765 ENZYME inhibitor 310264759 22317 15182 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IVA AESCULIOSIDE IVA 20371180 22318 15183 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME TRIAZOLAM TRIAZOLAM 22319 15184 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME DEXANABINOL DEXANABINOL 22320 15185 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor CHEMBL3545157 TIDEGLUSIB 22321 15186 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME Anti-meso-CAR vector transduced T cells 22322 15187 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-F2 22323 15188 CASP8 841 DRUGGABLE GENOME, PROTEASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 252166828 22324 15189 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CETUXIMAB CETUXIMAB 22586653,26296355,28223103 22326 15190 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CADMIUM ACETATE CADMIUM ACETATE 22327 15191 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 178101641 22328 15192 POLB 5423 DNA REPAIR, DRUGGABLE GENOME PHLORETIN PHLORETIN 22329 15193 ELAVL1 1994 DRUGGABLE GENOME DHT ANDROSTANOLONE 11356683 22330 15194 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE trastuzumab TRASTUZUMAB 30071039 22331 15195 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1317721 CHEMBL1385558 22332 15196 AK2 204 ENZYME, KINASE tenofovir TENOFOVIR 22335 15197 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2011799419010 22337 15198 HTT 3064 DRUGGABLE GENOME DNDI1417995 CHEMBL1439833 22341 15199 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201611 INSULIN LISPRO PROTAMINE RECOMBINANT 22342 15200 MAPT 4137 DRUGGABLE GENOME SLAZINIC ACID SLAZINIC ACID 22343 15201 DPP8 54878 DRUGGABLE GENOME, PROTEASE, ENZYME Thiomorpholine derivative 2 22344 15202 RRM2 6241 DRUGGABLE GENOME, ENZYME LY-2334737 LY-2334737 22345 15203 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TYRPHOSTIN 23 TYRPHOSTIN 23 22346 15204 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ALPHA-TOCOPHEROL VITAMIN E 15158075 22347 15205 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME NEFAZODONE NEFAZODONE 22349 15206 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-1644 CHEMBL600734 22350 15207 UCHL1 7345 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166861 22351 15208 QRFPR 84109 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 329968382 22352 15209 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000029642 CHEMBL591126 22354 15210 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME FIRATEGRAST FIRATEGRAST 22356 15211 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-O2 22359 15212 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CHEMBL407 FLUMAZENIL 22360 15213 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE 22361 15214 SH2D5 400745 NA gemcitabine GEMCITABINE 22838950 22363 15215 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL450 METHARBITAL 22365 15216 TLR7 51284 DRUGGABLE GENOME DV1179 22366 15217 ENG 2022 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antibody 315661183 CAROTUXIMAB 22367 15218 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE APC-100 APC-100 22369 15219 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME TCMDC-124356 CHEMBL22062 22370 15220 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DECITABINE DECITABINE 25968887 22371 15221 NOS1 4842 DRUGGABLE GENOME, ENZYME DIETHYLDITHIOCARBAMIC ACID 9154347 22374 15222 GMNN 51053 DRUGGABLE GENOME OLEIC ACID OLEIC ACID 22375 15223 SMN2 6607 DRUGGABLE GENOME NSC-116702 CHEMBL1477383 22377 15224 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200425 PARGYLINE HYDROCHLORIDE 22378 15225 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PROTOPORPHYRIN PROTOPORPHYRIN 22379 15226 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PGF2alpha 22382 15227 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE SR13668 SR-13668 22385 15228 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1068 OXCARBAZEPINE 22386 15229 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 22387 15230 GMNN 51053 DRUGGABLE GENOME SJ000113257 CHEMBL528694 22388 15231 F5 2153 DRUGGABLE GENOME hormonal contraceptives for systemic use 11532625,16113779,15208046,15946211,12869355,16301339,9459317,10073976,15467059,11859850,10943572,12069454,16769590,12138364,14551147,7968118 22389 15232 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 381118861 22390 15233 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PROCATEROL HYDROCHLORIDE PROCATEROL HYDROCHLORIDE 22392 15234 TMEM97 27346 NA Piperazinyl norbenzomorphane compound 1 22393 15235 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING VALPROIC ACID VALPROIC ACID 18294844,16921367,25304896 22394 15236 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER tamoxifen TAMOXIFEN 22396 15237 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LETROZOLE LETROZOLE 22398 15238 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL antagonist 135649951 22400 15239 GAPDH 2597 DRUGGABLE GENOME, ENZYME BISPHOSPHONATES 8518293 22401 15240 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME cisplatin CISPLATIN 16875718 22403 15241 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 315661214 22405 15242 CD52 1043 DRUGGABLE GENOME antibody ALEMTUZUMAB ALEMTUZUMAB 22406 15243 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME BETA-LAPACHONE LAPACHONE 22407 15244 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME IL-6 9187131 22408 15245 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DIMETHYL GAMBOGATE DIMETHYL GAMBOGATE 22409 15246 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL738 THIOPENTAL SODIUM 22410 15247 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME SJ000071854 CHEMBL602127 22411 15248 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MERCAPTOPURINE MERCAPTOPURINE 22414 15249 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 aspirin ASPIRIN 26517138,20833683 22416 15250 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE VACCINE 12007880 22417 15251 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME OXAZEPAM OXAZEPAM 22419 15252 TUBB4B 10383 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 22420 15253 SLC12A2 6558 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE BUMETANIDE BUMETANIDE 22421 15254 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 249565807 22423 15255 NOS1 4842 DRUGGABLE GENOME, ENZYME THIOURACIL THIOURACIL 10967532 22424 15256 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Pyrazole derivative 65 22425 15257 PPP2R5D 5528 PROTEIN PHOSPHATASE, ENZYME fluorouracil FLUOROURACIL 22426 15258 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE epirubicin EPIRUBICIN 24599932,24958282 22428 15259 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE oxaliplatin OXALIPLATIN 18245544,17700593,29845393,27864592,20819423,29134491,25331073,20385995,27557140,24980946,23407049 22432 15260 MPHOSPH8 54737 NA 2-(ALPHA-NAPHTHOYL)ETHYLTRIMETHYLAMMONIUM IODIDE CHEMBL1255936 22434 15261 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME GW441756X GW441756X 22435 15262 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL448 PENTOBARBITAL 22437 15263 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme4Upper 22438 15264 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Isoquinoline sulfonamide derivative 1 22440 15265 BAZ2B 29994 NA SJ000113211 CHEMBL602927 22441 15266 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BUTONATE BUTONATE 22443 15267 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649991 22444 15268 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Savolitinib SAVOLITINIB 22445 15269 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CINNAMALDEHYDE CINNAMALDEHYDE 22448 15270 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-102 22450 15271 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MMV085203 CHEMBL586031 22451 15272 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER mercaptopurine MERCAPTOPURINE 20393862 22452 15273 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOLYLFLUANID TOLYLFLUANID 22453 15274 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME HORMONES 8779894 22454 15275 MYB 4602 CLINICALLY ACTIONABLE 12-O-TETRADECANOYLPHORBOL-13-ACETATE 12354938 22455 15276 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME PD-98059 CHEMBL35482 22456 15277 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME DIETHYL-2-TETRADECYLIDENEMALONATE CHEMBL257748 21292492 22457 15278 CD38 952 CELL SURFACE, DRUGGABLE GENOME antibody 178103967 DARATUMUMAB 22458 15279 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 sunitinib SUNITINIB 17825686,24566734 22460 15280 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MICONAZOLE MICONAZOLE 22461 15281 MAOB 4129 DRUGGABLE GENOME, ENZYME Lazabemide analog 1 22462 15282 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CHEMOKINES 15840024 22463 15283 SLC23A2 9962 TRANSPORTER Vitamin C 22466 15284 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE RALTITREXED RALTITREXED 22467 15285 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-30 22469 15286 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 granisetron GRANISETRON 9187528 22470 15287 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ADRIAMYCIN ADRIAMYCIN 1363885,11069027 22474 15288 DNAJB1 3337 NA HSP70 15047721,16533811,15115283 22475 15289 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR INOSITOL INOSITOL 8013389 22476 15290 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PILOCARPINE PILOCARPINE 22477 15291 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-18 22479 15292 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BERGAPTOL BERGAPTOL 22480 15293 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200334 MORICIZINE HYDROCHLORIDE 22482 15294 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME 3R14S-OCHRATOXIN A 3R14S-OCHRATOXIN A 22483 15295 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 363894216 TUCATINIB 22484 15296 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE QUERCETIN QUERCETIN 22485 15297 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201631 INSULIN 22486 15298 CBX1 10951 NA THIORIDAZINE THIORIDAZINE 22487 15299 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IODOFORM IODOFORM 22488 15300 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 178102309 PICTILISIB 22490 15301 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE hmg coa reductase inhibitors 22491 15302 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SOTRASTAURIN SOTRASTAURIN 22492 15303 SLC16A1 6566 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 404859052 22493 15304 SMN1 6606 DRUGGABLE GENOME PD-98059 CHEMBL35482 22494 15305 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL PHENACEMIDE PHENACEMIDE 22495 15306 RAPGEF3 10411 ENZYME 2,4-DIHYDROXYBENZOPHENONE 2,4-DIHYDROXYBENZOPHENONE 22497 15307 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 178101892 22498 15308 IL11 3589 DRUGGABLE GENOME, KINASE, GROWTH FACTOR ANTISENSE OLIGONUCLEOTIDES 8427997 22499 15309 RACGAP1 29127 NA 4,4'-THIODIANILINE 4,4'-THIODIANILINE 22500 15310 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 252166577 PRACINOSTAT 22501 15311 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PENICILLIOL A PENICILLIOL A 19223184 22503 15312 MAPT 4137 DRUGGABLE GENOME 2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE 2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE 22504 15313 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR QUININE QUININE 22505 15314 SMN1 6606 DRUGGABLE GENOME RESVERATROL RESVERATROL 22506 15315 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PROTEASOME INHIBITOR 15147973 22507 15316 LOXL2 4017 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 385612244 22508 15317 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 22509 15318 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor 249565645 MK-2461 22510 15319 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 315661259 22511 15320 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Carbamide derivative 15 22512 15321 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME DHEA PRASTERONE 17102100 22513 15322 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CIPROFLOXACIN CIPROFLOXACIN 22931300 22515 15323 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650137 22517 15324 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PI3-KINASE INHIBITORS 12606824 22519 15325 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor PF03084014 22520 15326 EREG 2069 KINASE, GROWTH FACTOR, DRUGGABLE GENOME CETUXIMAB CETUXIMAB 23374602 22522 15327 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR SP-600125 SP-600125 22523 15328 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME OXALIPLATIN OXALIPLATIN 12072547 22526 15329 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE blocker CHEMBL2107762 NERISPIRDINE 22529 15330 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FIPEXIDE HYDROCHLORIDE FIPEXIDE HYDROCHLORIDE 22530 15331 XDH 7498 DRUGGABLE GENOME, ENZYME CARVEDILOL CARVEDILOL 15853634 22531 15332 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TRIADIMEFON TRIADIMEFON 22532 15333 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE cryptotanshinone CRYPTOTANSHINONE 23957426 22533 15334 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545194 LGH-447 22535 15335 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE adalimumab ADALIMUMAB 20309874,23007924 22537 15336 PTPRD 5789 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE pioglitazone PIOGLITAZONE 22538 15337 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GW8510 CHEMBL1276446 22539 15338 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ACRIFLAVINE CHLORIDE ACRIFLAVINE 22541 15339 BAZ2B 29994 NA L-750667 CHEMBL1256738 22543 15340 GALNT2 2590 DRUGGABLE GENOME atenolol ATENOLOL 22546 15341 GMNN 51053 DRUGGABLE GENOME SJ000044511 CHEMBL592124 22547 15342 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER cytarabine CYTARABINE 25558979,20938465,25567217,16331627 22548 15343 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIFLUOPERAZINE TRIFLUOPERAZINE 26372073 22549 15344 TUSC2 11334 NA Fus-1 tumor suppressor gene therapy - nanoparticle formulation 22551 15345 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BERGAPTOL BERGAPTOL 22554 15346 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME VX-702 VX-702 22555 15347 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652674 CABERGOLINE 22556 15348 IL11 3589 DRUGGABLE GENOME, KINASE, GROWTH FACTOR escitalopram ESCITALOPRAM 23142150 22557 15349 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102292 CEDIRANIB 22558 15350 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1762621 BARDOXOLONE METHYL 22560 15351 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ALVOCIDIB ALVOCIDIB 22561 15352 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL PF-05089771 PF-05089771 22562 15353 CBX1 10951 NA ETHOPROPAZINE ETHOPROPAZINE 22564 15354 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE antagonist CHEMBL1743051 ONARTUZUMAB 22566 15355 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE BEPRIDIL BEPRIDIL 22567 15356 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE AZD9291 OSIMERTINIB 27694386,27393507,27252416 22568 15357 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME EMETINE HYDROCHLORIDE EMETINE HYDROCHLORIDE 22569 15358 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Pyrrolo-pyrrolone derivative 2 22571 15359 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist 252166530 VENETOCLAX 22573 15360 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PREDNISOLONE PREDNISOLONE 12673034 22574 15361 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 indomethacin INDOMETHACIN 12876643 22575 15362 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL3707402 PF-06372865 22576 15363 APCS 325 TRANSPORTER, DRUGGABLE GENOME GSK-2315698 MIRIDESAP 26225229 22577 15364 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650756 OLANZAPINE 22578 15365 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GNF-PF-793 CHEMBL604311 22579 15366 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE ELSAMICIN A 14529449 22581 15367 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000157363 CHEMBL590947 22582 15368 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102325 PAZOPANIB 22583 15369 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE ACE INHIBITOR 12215475,8622594 22584 15370 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor XL-765 VOXTALISIB 22585 15371 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME JNJ-7706621 JNJ-7706621 22587 15372 CXCL8 3576 DRUGGABLE GENOME DIPYRIDAMOLE DIPYRIDAMOLE 10660968 22588 15373 PADI2 11240 ENZYME O-F-AMIDINE CHEMBL1910970 21882827 22589 15374 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR MESALAMINE MESALAMINE 15887108 22591 15375 GMNN 51053 DRUGGABLE GENOME LERCANIDIPINE LERCANIDIPINE 22592 15376 HBB 3043 DRUGGABLE GENOME, ENZYME Hemoglobin raffimer 22593 15377 VKORC1 79001 DRUGGABLE GENOME, ENZYME inhibitor 178103414 DICUMAROL 22594 15378 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME ARI-2243 21106865 22596 15379 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME DARBEPOETIN ALFA 22597 15380 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE antibody 387065587 JNJ-61186372 22599 15381 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIPYRITHIONE DIPYRITHIONE 22600 15382 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 249565873 22601 15383 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL931 HALOTHANE 22602 15384 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NOMIFENSINE NOMIFENSINE 22605 15385 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DIENOCHLOR DIENOCHLOR 22606 15386 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE Andecaliximab ANDECALIXIMAB 22607 15387 PTPN6 5777 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TOFACITINIB TOFACITINIB 24978112 22608 15388 TNKS2 80351 DRUGGABLE GENOME, ENZYME inhibitor 404859119 22613 15389 SMN2 6607 DRUGGABLE GENOME CID 1245272 CHEMBL408850 22616 15390 GMNN 51053 DRUGGABLE GENOME 5-NITRO-[1,10]PHENANTHROLINE CHEMBL101815 22618 15391 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Panitumumab PANITUMUMAB 22620 15392 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 178103893 VARDENAFIL 22621 15393 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Benzimidazole derivative 7 22623 15394 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 178102292 CEDIRANIB 22624 15395 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL403989 TG100-801 22625 15396 MPHOSPH8 54737 NA HISPIDIN HISPIDIN 22627 15397 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 336446944 22628 15398 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER fexofenadine FEXOFENADINE 11503014 22629 15399 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GW1929 CHEMBL434063 22630 15400 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE HELENALIN HELENALIN 22633 15401 SLCO2A1 6578 TRANSPORTER, DRUGGABLE GENOME PMID26099857-Compound-WO2011037610Formula(I) 22634 15402 BCHE 590 DRUGGABLE GENOME, ENZYME cocaine COCAINE 24312228 22635 15403 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE NSC-675972 CHEMBL1379243 22212721 22636 15404 CD7 924 DRUGGABLE GENOME CD7.CAR/28zeta CAR T cells 22637 15405 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR DABRAFENIB DABRAFENIB 24265153,25673644 22638 15406 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ketoprofen KETOPROFEN 25989235 22639 15407 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649959 AMMONIUM TRICHLOROTELLURATE 22640 15408 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR GDC-0152 GDC-0152 22643 15409 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 252827366 GILTERITINIB 22644 15410 MAPT 4137 DRUGGABLE GENOME 2-BENZOYL-5-METHOXYBENZOQUINONE 2-BENZOYL-5-METHOXYBENZOQUINONE 22646 15411 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GNF-PF-4085 CHEMBL528181 22649 15412 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME MERSALYL MERSALYL 22656 15413 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR XL888 XL-888 22657 15414 HLA-DQA1 3117 CLINICALLY ACTIONABLE mercaptopurine MERCAPTOPURINE 25217962 22659 15415 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME CARVEDILOL CARVEDILOL 16759520,12973927 22661 15416 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME activator 363894230 22663 15417 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GUTHION GUTHION 22666 15418 GMNN 51053 DRUGGABLE GENOME FLUNARIZINE DIHYDROCHLORIDE FLUNARIZINE DIHYDROCHLORIDE 22667 15419 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650061 BARDOXOLONE 22668 15420 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-30 22669 15421 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME GNF-PF-4665 CHEMBL601744 22671 15422 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR BAY-613606 CHEMBL541400 22672 15423 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 2-PHENYLACETYLAMINOBENZOTHIAZOLE CHEMBL1405979 22673 15424 GJB4 127534 ION CHANNEL inhibitor 135650269 22676 15425 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME isoflurane ISOFLURANE 25989378,12411786,26951757,8828983,19919814,17710899,7829078,9334205,21965348,11063719,10823104,20681998,25611019,19648156,25256590,12220451,11668625,23736090,14500992,9066328,14641996,18945287,25960145,7889656,11575529,18212565,16284304,8602662,18306019,28326467,11928716,18502356,10352931,12151923,11525881,17122579,16917943,8220422,10700782,16163667,17226826,9389851,16732128,16835904,11448278,29101530,9450902,7547049,23628358,9543323,24361844,26994242,12208234,15448513,16621918,21455645,11553045,12124989,19020143,19191329,27918309,8220423,12059893,10612851,16732084,10793526,27382027,15108991,12709367,12123492,26381711,25268394,28063098,11493496,12434264,12411788,19685112,25735680,8902717,29608462,27663056,7751854,8012359,9520251,15731587,15210166,1510267,10888602,22030266,25466363,17483490,28403410,12237752,1774074,17081152,18564801,10484775,21282829,16244001,7586638,19191333,25086907,7633940,17667581,12883402,19346234,1354642,22415532 22678 15426 MAPT 4137 DRUGGABLE GENOME GNF-PF-2414 CHEMBL601353 22679 15427 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING GO-Y015 CHEMBL477052 21504179 22680 15428 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178103844 PHENYLBUTAZONE 22681 15429 SPTBN1 6711 NA ABT-413 22682 15430 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR GP100 16968820 22684 15431 PBK 55872 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, ENZYME inhibitor 223366144 22686 15432 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME cisplatin CISPLATIN 19786980,22188361,17409936,15254763,31666714,25592234 22687 15433 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor VATALANIB VATALANIB 22688 15434 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME MITOGEN-ACTIVATED PROTEIN KINASE KINASE INHIBITOR 26996308,31580757 22690 15435 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135650200 22691 15436 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME CART-Muc1 cells 22693 15437 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME BELINOSTAT BELINOSTAT 25937017 22694 15438 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650426 22696 15439 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-747268 CHEMBL595911 22698 15440 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545196 PD-0166285 22701 15441 CASP4 837 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166854 22702 15442 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME nivolumab NIVOLUMAB 22704 15443 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Pelitinib PELITINIB 22707 15444 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor 135650453 KETANSERIN 22711 15445 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor REFAMETINIB REFAMETINIB 22713 15446 SLC15A2 6565 TRANSPORTER, DRUGGABLE GENOME 178101375 22714 15447 BRCA2 675 CLINICALLY ACTIONABLE Rucaparib RUCAPARIB 22715 15448 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME METHOTREXATE METHOTREXATE 22716 15449 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33d 22718 15450 GRK2 156 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 249565822 BALANOL 22719 15451 ATXN2 6311 NA HYCANTHONE HYCANTHONE 22721 15452 ALPI 248 DRUGGABLE GENOME, ENZYME GNF-PF-1947 CHEMBL585591 22723 15453 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL3039530 ABEDITEROL 22724 15454 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PMID29130358-Compound-Figure11(3) 22726 15455 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME prasugrel PRASUGREL 21828263 22727 15456 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY RETINOIC ACID 11563543 22728 15457 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE Berberine BERBERINE 22729 15458 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME IMATINIB IMATINIB 22730 15459 RAPGEF3 10411 ENZYME RAFOXANIDE RAFOXANIDE 22731 15460 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TCMDC-124224 CHEMBL580421 22733 15461 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 375973222 22734 15462 COMT 1312 DRUGGABLE GENOME, ENZYME sumatriptan SUMATRIPTAN 25096645 22736 15463 PBRM1 55193 CLINICALLY ACTIONABLE ATEZOLIZUMAB ATEZOLIZUMAB 29301960 22737 15464 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL462018 TRICIRIBINE PHOSPHATE 22739 15465 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GEDUNIN GEDUNIN 25756299 22740 15466 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565686 BX-795 22743 15467 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor CHEMBL3545085 XL-228 22744 15468 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME TRICHOSTATIN TRICHOSTATIN 21055848,16921367,19966789,19385600 22747 15469 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CEFAMANDOLE CEFAMANDOLE 22166395 22748 15470 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 354702275 22749 15471 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor CHEMBL3544964 RAVOXERTINIB 22752 15472 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIPYRIDYL DIPYRIDYL 22754 15473 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LATANOPROST LATANOPROST 22755 15474 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE MTOR INHIBITOR 20085938 22756 15475 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE XL147 PILARALISIB 23948973 22757 15476 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME IMATINIB MESYLATE 15805252 22758 15477 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor AXITINIB AXITINIB 22760 15478 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME ILORASERTIB ILORASERTIB 22761 15479 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR N-quinolin-benzene sulphonamide derivative 3 22763 15480 ATAD5 79915 NA PHENANTHROLINE PHENANTHROLINE 22764 15481 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX R547 17121911 22767 15482 LIMK2 3985 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565797 22768 15483 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-693571 CHEMBL1287983 22769 15484 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Niravoline NIRAVOLINE 22770 15485 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR FE-202767 FE 202767 22771 15486 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270010-Compound-Figure5-1 22772 15487 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME TYRPHOSTIN 47 TYRPHOSTIN 47 22773 15488 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor RO 4929097 22775 15489 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 KARANJIN KARANJIN 22777 15490 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL3545351 AV-101 22780 15491 CD248 57124 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2109397 ONTUXIZUMAB 22781 15492 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CHIR-99021 CHIR-99021 22782 15493 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TCMDC-123869 CHEMBL546597 22783 15494 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE N/A 22785 15495 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody MEHD7945A DULIGOTUZUMAB 22786 15496 PAH 5053 DRUGGABLE GENOME, ENZYME carbocisteine CARBOCYSTEINE 19036622 22787 15497 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-186 CHEMBL601140 22788 15498 IMPDH2 3615 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL866 MYCOPHENOLIC ACID 22789 15499 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME LEVODOPA LEVODOPA 22790 15500 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL1201152 NALMEFENE HYDROCHLORIDE 22791 15501 CD276 80381 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME MGD009 22792 15502 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER progesterone PROGESTERONE 22793 15503 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR CYC-116 CYC-116 22794 15504 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Six-membered heterocyclic benzamide derivative 5 22795 15505 TUBB6 84617 DRUGGABLE GENOME CHEMBL2304041 SAGOPILONE 22796 15506 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME BMS-345541 BMS-345541 18702457 22797 15507 CYP27A1 1593 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 inhibitor 252827515 CHEMBL255088 22798 15508 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-586581A GSK-586581A 22799 15509 SMN2 6607 DRUGGABLE GENOME JNJ-16259685 CHEMBL174588 22800 15510 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BEZ235 DACTOLISIB 26272063 22801 15511 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1201486 QUINIDINE POLYGALACTURONATE 22802 15512 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL PRAZEPAM PRAZEPAM 22803 15513 PPME1 51400 ENZYME, DRUGGABLE GENOME inhibitor 252166809 22804 15514 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME STREPTOZOTOCIN STREPTOZOCIN 12403787 22805 15515 GAA 2548 DRUGGABLE GENOME, ENZYME Deoxynojirimycin DUVOGLUSTAT 22806 15516 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW580509X GW580509X 22807 15517 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ZIPRASIDONE ZIPRASIDONE 22808 15518 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 249565863 22809 15519 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SOFALCONE SOFALCONE 22813 15520 PTGES 9536 DRUGGABLE GENOME, ENZYME Betais-sulfonylamino derivative 1 22814 15521 SRD5A1 6715 DRUGGABLE GENOME DUTASTERIDE DUTASTERIDE 22815 15522 UBE2N 7334 ENZYME, DRUGGABLE GENOME GNF-PF-3286 CHEMBL581880 22816 15523 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AKTI-1/2 18725974 22817 15524 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 22(S)-HYDROXYCHOLESTEROL CHEMBL1243244 24480357,24268541 22818 15525 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 404859029 22819 15526 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE MASITINIB MASITINIB 22821 15527 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE IC261 IC261 20350806 22825 15528 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE inhibitor CHEMBL2107856 IMETELSTAT 22826 15529 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE docetaxel DOCETAXEL 23963862 22827 15530 IFIT2 3433 CLINICALLY ACTIONABLE IFN 12433283 22828 15531 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL289351 FOSBRETABULIN DISODIUM 22830 15532 TFF3 7033 DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 25900183 22831 15533 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CEDIRANIB CEDIRANIB 22832 15534 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DIPYRIDAMOLE DIPYRIDAMOLE 22833 15535 PML 5371 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRETINOIN TRETINOIN 21505136,8674046,21613260,23670176,11704842,30289902 22834 15536 TNFAIP3 7128 PROTEASE, ENZYME, CLINICALLY ACTIONABLE, KINASE ustekinumab USTEKINUMAB 27564082,23521149 22836 15537 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Idelalisib IDELALISIB 26137449 22838 15538 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE INTERLEUKINS 2538824 22841 15539 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE DASATINIB DASATINIB 22842 15540 ABCA1 19 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL608 PROBUCOL 22843 15541 GMNN 51053 DRUGGABLE GENOME CHRYSEN-6-YLAMINE CHEMBL313154 22845 15542 CBR1 873 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME doxorubicinol 19016765 22846 15543 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME MAPROTILINE MAPROTILINE 22847 15544 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME THYROXINE THYROXINE 10452218 22848 15545 TCIM 56892 NA ANTIANGIOGENIC 15289477 22851 15546 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CID 1540545 CHEMBL259784 22852 15547 KDM4A 9682 DRUGGABLE GENOME, ENZYME 4-HYDROXYDERRICIN CHEMBL458094 22853 15548 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PD-404182 CHEMBL595227 22854 15549 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 385612170 KZR-616 22856 15550 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyridine derivative 1 22857 15551 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME L-765314 L-765314 22858 15552 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 22859 15553 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ALLITRIDIN ALLITRIDIN 22860 15554 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 249565634 BGT-226 22861 15555 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102925 AURANOFIN 22862 15556 OPLAH 26873 ENZYME MELPHALAN MELPHALAN 9751079 22863 15557 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NUTLIN-3 NUTLIN-3 21058726,26288684,24268795,19928922 22864 15558 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 315661104 NAVOXIMOD 22868 15559 CBX1 10951 NA NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 22869 15560 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 22870 15561 GMNN 51053 DRUGGABLE GENOME HEXACHLOROPHENE HEXACHLOROPHENE 22872 15562 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417601 CHEMBL1503729 22873 15563 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor AFATINIB AFATINIB 22875 15564 IGFBP1 3484 DRUGGABLE GENOME STZ STREPTOZOCIN 1713293,7589849 22879 15565 ALDH1A1 216 DRUGGABLE GENOME, ENZYME OBTUSAQUINONE OBTUSAQUINONE 22880 15566 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME GDC-0623 RG-7420 22882 15567 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 328083484 22884 15568 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR TETRACYCLINE TETRACYCLINE 22885 15569 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PX-866 SONOLISIB 22886 15570 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 348353622 22887 15571 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650344 22890 15572 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE CYC-116 CYC-116 22893 15573 MAPKAP1 79109 KINASE inhibitor OSI-027 OSI-027 22894 15574 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor AZD4547 22895 15575 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103528 22898 15576 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652583 22899 15577 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Imidazo [1,2-a]pyridine compound 1 22900 15578 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME blocker 381744985 22901 15579 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Bis-aminopyrimidine derivative 4 22902 15580 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4798 CHEMBL584635 22903 15581 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER DESFERRIOXAMINE DEFEROXAMINE 12514119 22905 15582 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENBUCONAZOLE FENBUCONAZOLE 22907 15583 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE INTERFERON GAMMA 1557656 22908 15584 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Gefitinib GEFITINIB 26936917 22909 15585 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE AP-301-IH 22910 15586 LIPC 3990 ENZYME, PHOSPHOLIPASE, LIPASE, DRUGGABLE GENOME fluvastatin FLUVASTATIN 16103896 22911 15587 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIETHYLCARBAMAZINE CITRATE DIETHYLCARBAMAZINE CITRATE 22913 15588 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME SP-600125 SP-600125 22914 15589 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE TAMATINIB R-406 22916 15590 PSMA5 5686 PROTEASE, DRUGGABLE GENOME CARFILZOMIB CARFILZOMIB 24524217 22917 15591 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist 249565878 PATIDEGIB 22918 15592 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME antibody FICLATUZUMAB FICLATUZUMAB 22919 15593 CASP2 835 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166828 22920 15594 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Cyclopropyl-spiro piperidine derivative 1 22921 15595 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE R763 22922 15596 BAZ2B 29994 NA TCMDC-123650 CHEMBL580727 22926 15597 ACVR2B 93 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME antagonist CHEMBL3137353 BIMAGRUMAB 22927 15598 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL antagonist CHEMBL220492 TOPIRAMATE 22928 15599 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE TAMATINIB R-406 22930 15600 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Cabozantinib CABOZANTINIB 27694386,27825638 22931 15601 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE PROPOXYPHENE PROPOXYPHENE 22932 15602 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LAUROGUADINE LAUROGUADINE 22933 15603 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE CORDYCEPIN CORDYCEPIN 24283924 22934 15604 CRBN 51185 ENZYME, DRUG RESISTANCE 178103920 POMALIDOMIDE 22935 15605 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR UCN-01 UCN-01 22936 15606 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135650977 ALBUTEROL 22939 15607 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135652694 22941 15608 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME METHOXYCHLOR METHOXYCHLOR 22945 15609 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ISOPROTERENOL ISOPROTERENOL 22948 15610 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Lapatinib LAPATINIB 27595477,20215545,23917401,18199554 22949 15611 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Indoline derivative 21 22950 15612 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR partial agonist CHEMBL2108144 TENELIXIMAB 22951 15613 POLK 51426 DNA REPAIR, ENZYME 3',4'-DIHYDROXYFLAVONE CHEMBL222556 22956 15614 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651066 SPIROXATRINE 22958 15615 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME OTX-015 BIRABRESIB 22960 15616 PAH 5053 DRUGGABLE GENOME, ENZYME Pegvaliase PEGVALIASE 22962 15617 MYD88 4615 CLINICALLY ACTIONABLE IMO-8400 BAZLITORAN 22963 15618 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX antagonist 178100886 22964 15619 TARDBP 23435 TUMOR SUPPRESSOR 2',3'-DIDEOXYADENOSINE CHEMBL23094 22965 15620 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE IBRUTINIB IBRUTINIB 28830912 22966 15621 MAOB 4129 DRUGGABLE GENOME, ENZYME Tarnylcypromine derivative 2 22969 15622 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200654 BENOXINATE HYDROCHLORIDE 22970 15623 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL19019 NALTREXONE 22971 15624 RAPGEF3 10411 ENZYME 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 22972 15625 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SOBUZOXANE SOBUZOXANE 22973 15626 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR PROMETHAZINE HYDROCHLORIDE PROMETHAZINE HYDROCHLORIDE 22974 15627 TRH 7200 DRUGGABLE GENOME KPS-0373 ROVATIRELIN 22975 15628 HTT 3064 DRUGGABLE GENOME GNF-PF-1702 CHEMBL600313 22976 15629 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-2657 CHEMBL578944 22978 15630 ABCC9 10060 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER Tolbutamide TOLBUTAMIDE 22979 15631 GAA 2548 DRUGGABLE GENOME, ENZYME DUVOGLUSTAT DUVOGLUSTAT 22980 15632 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MIFEPRISTONE MIFEPRISTONE 22981 15633 PSMD12 5718 NA inhibitor CARFILZOMIB CARFILZOMIB 22983 15634 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR PHA-848125AC MILCICLIB MALEATE 23347136 22984 15635 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Bis-aminopyrimidine derivative 4 22985 15636 MPHOSPH8 54737 NA AG-34 CHEMBL80155 22986 15637 APBA1 320 NA PHENAZINE-2,3-DIAMINE CHEMBL274921 22989 15638 GPR12 2835 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CYCLOCITRINOL CYCLOCITRINOL 18656987 22990 15639 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE 2,4-DIACETYL PHLOROGLUCINOL CHEMBL276139 22992 15640 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 22993 15641 PSMC4 5704 NA CARFILZOMIB CARFILZOMIB 24524217 22994 15642 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME UNBS3157 CHEMBL244268 17658777 22995 15643 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL411907 SONOLISIB 22996 15644 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE INDINAVIR SULFATE INDINAVIR SULFATE 22997 15645 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE erlotinib ERLOTINIB 22998 15646 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-MTC-433 23001 15647 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 178103529 23002 15648 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME doxorubicin DOXORUBICIN 11956086 23003 15649 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CRIZOTINIB CRIZOTINIB 23004 15650 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417097 CHEMBL1531222 23005 15651 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE inhibitor 252827503 CGS-27023A 23006 15652 BAZ2B 29994 NA AG-528 CHEMBL56542 23007 15653 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-125480 CHEMBL546257 23009 15654 NOD1 10392 CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 178101718 23010 15655 HMBS 3145 ENZYME P-9808 23012 15656 PSMD2 5708 NA inhibitor CARFILZOMIB CARFILZOMIB 23013 15657 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME pravastatin PRAVASTATIN 27839692 23015 15658 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1706 NAPHAZOLINE HYDROCHLORIDE 23017 15659 GSTM1 2944 DRUGGABLE GENOME, ENZYME XANTHOPHYLLS 15355982 23018 15660 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Vemurafenib VEMURAFENIB 26343583,28514312 23019 15661 PSMD7 5713 PROTEASE inhibitor CARFILZOMIB CARFILZOMIB 23022 15662 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Benzimidazole derivative 6 23024 15663 COMT 1312 DRUGGABLE GENOME, ENZYME Selective serotonin reuptake inhibitors 24930681 23026 15664 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DOXAZOSIN DOXAZOSIN 23027 15665 HSPA4 3308 NA DDC ZALCITABINE 10591146 23029 15666 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME lofexidine LOFEXIDINE 23031 15667 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Pyridine derivative 20 23033 15668 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3544999 SAMOTOLISIB 23035 15669 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Sunitinib SUNITINIB 26864210,23455880 23037 15670 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER lamivudine LAMIVUDINE 23996099 23039 15671 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR TUBERATOLIDE B TUBERATOLIDE B 21142112 23040 15672 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 135651398 23041 15673 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DEXBROMPHENIRAMINE DEXBROMPHENIRAMINE 23042 15674 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME KETOCONAZOLE KETOCONAZOLE 17518356 23043 15675 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 23045 15676 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER hmg coa reductase inhibitors 24595600 23046 15677 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ORYZALIN ORYZALIN 23047 15678 CEACAM1 634 KINASE, CELL SURFACE, DRUGGABLE GENOME RETINOIC ACID 15364113 23049 15679 HMMR 3161 KINASE, CELL SURFACE, DRUGGABLE GENOME epirubicin EPIRUBICIN 23050 15680 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-36 23051 15681 FGF19 9965 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR FISOGATINIB 31575541 23052 15682 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ALTENUSIN ALTENUSIN 23053 15683 TH 7054 ENZYME, DRUGGABLE GENOME METYROSINE METYROSINE 23055 15684 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL565612 SOTRASTAURIN 23056 15685 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C1 23057 15686 KDM4A 9682 DRUGGABLE GENOME, ENZYME PIROXICAM PIROXICAM 23058 15687 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor SB939 23060 15688 HTT 3064 DRUGGABLE GENOME CHLOROXINE CHLOROXINE 23061 15689 MAOA 4128 DRUGGABLE GENOME, ENZYME 8-[(3-TRIFLUOROMETHYL)BENZYLOXY]CAFFEINE CHEMBL602466 20093036 23062 15690 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 354702299 ALVESPIMYCIN 23063 15691 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 348353621 PYROTINIB 23064 15692 CD37 951 DRUGGABLE GENOME antibody 374883838 OTLERTUZUMAB 23066 15693 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR GNF-PF-4029 CHEMBL596633 23067 15694 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 650707 CHEMBL408653 23068 15695 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW642125X GW642125X 23069 15696 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102759 23070 15697 IMPDH1 3614 ENZYME, DRUGGABLE GENOME inhibitor 178103448 RIBAVIRIN 23071 15698 SCTR 6344 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME SECRETIN SECRETIN 23072 15699 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 381744915 23073 15700 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Imatinib IMATINIB 22323597 23075 15701 POLI 11201 DNA REPAIR CEFOTETAN CEFOTETAN 23078 15702 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME METHYLERGONOVINE METHYLERGONOVINE 23079 15703 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OXYMETHOLONE OXYMETHOLONE 23080 15704 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 363894217 VORUCICLIB 23081 15705 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE allosteric modulator 328083529 MIRANSERTIB 23082 15706 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 223366076 23083 15707 MAPT 4137 DRUGGABLE GENOME S-166659 CHEMBL252417 23084 15708 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROADIFEN HYDROCHLORIDE PROADIFEN HYDROCHLORIDE 23085 15709 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-2307 CHEMBL421088 23086 15710 ALOX15 246 ENZYME, DRUGGABLE GENOME 4-TERT-BUTYLCATECHOL CHEMBL220845 23087 15711 GMNN 51053 DRUGGABLE GENOME TRIPARANOL TRIPARANOL 23088 15712 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102445 TREPROSTINIL 23090 15713 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 385612210 23091 15714 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PACLITAXEL PACLITAXEL 16467099 23092 15715 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor BGJ398 INFIGRATINIB 23093 15716 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 bleomycin BLEOMYCIN 23094 15717 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE MEPENZOLATE MEPENZOLATE 23096 15718 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE BERKELEYTRIONE BERKELEYTRIONE 17970594 23098 15719 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650510 23099 15720 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Carbamide derivative 10 23100 15721 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651592 23102 15722 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR HYDROMORPHONE HYDROMORPHONE 23103 15723 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ORCIPRENALINE METAPROTERENOL 23104 15724 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME SJ000113972 CHEMBL591137 23105 15725 ENO2 2026 CELL SURFACE INDOMETHACIN INDOMETHACIN 12711954 23107 15726 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME FASUDIL FASUDIL 23108 15727 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 5-FU FLUOROURACIL 16421754,15538739,11501504 23109 15728 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME ADJUVANT 17301541 23110 15729 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000044511 CHEMBL592124 23111 15730 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DAIDZEIN DAIDZEIN 23112 15731 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME PMID28270010-Compound-Figure5-1 23113 15732 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 135650356 CHEMBL497392 23116 15733 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHR-3996 NANATINOSTAT 23121 15734 HEBP1 50865 DRUGGABLE GENOME 1-phenyl-1,3,4-triazole derivative 1 23122 15735 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32n 23123 15736 ALPL 249 ENZYME, DRUGGABLE GENOME DNDI1417523 CHEMBL598663 23125 15737 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE TIAGABINE TIAGABINE 23126 15738 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE (-)-OLEOCANTHAL (-)-OLEOCANTHAL 23403296 23128 15739 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-67 CHEMBL578512 23130 15740 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR SANGUINARIUM CHLORIDE SANGUINARIUM CHLORIDE 23131 15741 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IV-23E CHEMBL1094674 20371180 23132 15742 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TRAVOPROST TRAVOPROST 23133 15743 PRMT1 3276 ENZYME, METHYL TRANSFERASE inhibitor 310264736 23138 15744 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Pyrrolo-pyrrolone derivative 3 23140 15745 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Torkinib 21358673 23141 15746 SMN2 6607 DRUGGABLE GENOME CID 887167 CHEMBL260342 23142 15747 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-44 23143 15748 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AT-7867 24978597,20423992 23144 15749 CD248 57124 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE MORAB-004 ONTUXIZUMAB 23145 15750 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565794 23146 15751 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME inhibitor 178103235 23149 15752 EIF2AK2 5610 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR IFN ALPHA-2B 17501760 23151 15753 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Benzonaphthyridine derivative 2 23152 15754 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651044 23153 15755 ACSS2 55902 ENZYME, TRANSCRIPTION FACTOR docetaxel DOCETAXEL 21636554 23154 15756 BRCA2 675 CLINICALLY ACTIONABLE Radiotherapy 28062704,26116172 23155 15757 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LABETALOL LABETALOL 22931300 23156 15758 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 3 23157 15759 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Metoprolol METOPROLOL 23158 15760 POLK 51426 DNA REPAIR, ENZYME CHARTREUSIN CHARTREUSIN 23160 15761 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE TRAMETINIB TRAMETINIB 29127119 23161 15762 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR VIA-3196 RESMETIROM 23162 15763 SMN2 6607 DRUGGABLE GENOME HYDRALAZINE HYDROCHLORIDE HYDRALAZINE HYDROCHLORIDE 23164 15764 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR E6201 E-6201 24448821 23165 15765 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CEDIRANIB CEDIRANIB 23167 15766 PDE4D 5144 DRUGGABLE GENOME, ENZYME LIRIMILAST LIRIMILAST 23168 15767 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE HM-78136B 23169 15768 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 2-CHLOROADENOSINE CHEMBL285819 23170 15769 CDC42BPA 8476 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PF-562271 PF-00562271 23171 15770 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE DEGUELIN DEGUELIN 23172 15771 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody CETUXIMAB CETUXIMAB 23173 15772 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor CHEMBL3707266 RIBOCICLIB SUCCINATE 23175 15773 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BEXAROTENE BEXAROTENE 23177 15774 TARDBP 23435 TUMOR SUPPRESSOR FORMESTANE FORMESTANE 23178 15775 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ZK-thiazolidinone 23179 15776 RGS4 5999 DRUGGABLE GENOME HELENALIN HELENALIN 23181 15777 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE XL-820 XL-820 23182 15778 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545076 LY-2584702 23183 15779 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651258 THIOPERAMIDE 23185 15780 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME VEMURAFENIB VEMURAFENIB 23186 15781 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ALISERTIB ALISERTIB 23187 15782 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CARBOQUONE CARBOQUONE 23190 15783 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER azathioprine AZATHIOPRINE 20393862 23191 15784 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Afatinib AFATINIB 23192 15785 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RN-1 26837761 23193 15786 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR AFIMOXIFENE AFIMOXIFENE 23200 15787 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TANESPIMYCIN TANESPIMYCIN 23202 15788 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYPROTERONE CYPROTERONE 23204 15789 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LANSOPRAZOLE LANSOPRAZOLE 23205 15790 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-22 23206 15791 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AZD4547 23207 15792 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE LY-294002 LY-294002 17562705,22212721 23208 15793 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PACLITAXEL PACLITAXEL 16289636 23210 15794 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103420 ETHOXZOLAMIDE 23211 15795 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE SNS-314 SNS-314 23212 15796 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME RG-1530 RG-1530 23213 15797 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AMILORIDE AMILORIDE 23214 15798 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR FENOLDOPAM MESYLATE FENOLDOPAM MESYLATE 23217 15799 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRITON X TRITON X 23219 15800 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID25991433-Compound-P5 23220 15801 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR JNK INHIBITOR VIII CHEMBL210618 23221 15802 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR CEPHALOTHIN SODIUM CEPHALOTHIN SODIUM 23222 15803 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GF-109203 GF-109203 23223 15804 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE BAY-613606 CHEMBL541400 23226 15805 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 23227 15806 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-69 23228 15807 IL1RN 3557 DRUGGABLE GENOME AC-201 DIACEREIN 23229 15808 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METHOTRIMEPRAZINE LEVOMEPROMAZINE 23230 15809 GMNN 51053 DRUGGABLE GENOME PRAZOSIN HYDROCHLORIDE PRAZOSIN HYDROCHLORIDE 23231 15810 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME GLPG-0634 FILGOTINIB 23232 15811 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR GW5074 CHEMBL1794051 20030343 23233 15812 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR TERFENADINE TERFENADINE 8836342 23234 15813 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135651365 23236 15814 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME VX-745 NEFLAMAPIMOD 23237 15815 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SB-415286 CHEMBL322970 23240 15816 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PROPYLPYRAZOLETRIOL PROPYLPYRAZOLETRIOL 23244 15817 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR antagonist CHEMBL3545391 ORG-34517 23245 15818 POLK 51426 DNA REPAIR, ENZYME PRAZOSIN HYDROCHLORIDE PRAZOSIN HYDROCHLORIDE 23246 15819 PTGES 9536 DRUGGABLE GENOME, ENZYME Imidazopyridine derivative 7 23248 15820 CD74 972 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE antibody 252166479 MILATUZUMAB 23249 15821 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR M-0004 23250 15822 HTT 3064 DRUGGABLE GENOME GNF-PF-1399 CHEMBL578504 23251 15823 GJA1 2697 ION CHANNEL PROTEASE INHIBITOR 15870950 23252 15824 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MK-1775 ADAVOSERTIB 24791855 23253 15825 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-742864 CHEMBL103080 23255 15826 SMN2 6607 DRUGGABLE GENOME DNDI1417268 CHEMBL1517542 23258 15827 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE ORAL CONTRACEPTIVE 8392873,12388132 23260 15828 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650784 OXYBUTYNIN 23261 15829 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE phenobarbital PHENOBARBITAL 23262 15830 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER DNDI1417254 CHEMBL2094567 23263 15831 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Abemaciclib ABEMACICLIB 27217383 23264 15832 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178100700 23266 15833 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE HUMAX-EGFR ZALUTUMUMAB 23267 15834 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ECADOTRIL ECADOTRIL 23270 15835 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER FLAVOKAWAIN A FLAVOKAWAIN A 22112540 23272 15836 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME 3TC LAMIVUDINE 17538878 23274 15837 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1615835 MUPARFOSTAT 23275 15838 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE ORTERONEL ORTERONEL 23277 15839 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROPARGITE PROPARGITE 23278 15840 AQP1 358 ION CHANNEL, DRUGGABLE GENOME inhibitor 178101032 23279 15841 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SE-METHYLSELENOCYSTEINE METHYLSELENOCYSTEINE 23282 15842 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Carboplatin CARBOPLATIN 28514312 23283 15843 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR LAUROGUADINE LAUROGUADINE 23284 15844 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME NAPHTHOQUINONE NAPHTHOQUINONE 16699520 23285 15845 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Ponatinib PONATINIB 26270481 23288 15846 ORAI1 84876 TRANSCRIPTION FACTOR, ION CHANNEL, TRANSPORTER blocker 381118797 23290 15847 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MICONAZOLE MICONAZOLE 23291 15848 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE THIOTHIXENE THIOTHIXENE 23292 15849 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE DNDI1417080 CHEMBL1498652 23294 15850 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL PHENETHYLISOTHIOCYANATE PHENETHYLISOTHIOCYANATE 26263397 23295 15851 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Geminally-substituted cyanoethylpypazolo pyridone derivative 1 23296 15852 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 2,6-DIMETHOXYQUINONE 2,6-DIMETHOXYQUINONE 23298 15853 HMGCR 3156 ENZYME, DRUGGABLE GENOME PITAVASTATIN CALCIUM 23299 15854 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C25 23300 15855 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 6-11 23301 15856 BRD9 65980 ENZYME inhibitor 310264731 23303 15857 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE erlotinib ERLOTINIB 23304 15858 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TAMOXIFEN TAMOXIFEN 23307 15859 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 252827436 23308 15860 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL3545252 DOCETAXEL 23310 15861 KCNJ5 3762 TRANSPORTER, ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker 135650721 23311 15862 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178100903 23312 15863 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565865 23314 15864 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME INDOMETHACIN INDOMETHACIN 9090444 23316 15865 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE LY2780301 28750271 23317 15866 XDH 7498 DRUGGABLE GENOME, ENZYME Cyclic pyranopterin monophosphate 23319 15867 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SKF-89626 CHEMBL284609 23320 15868 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Afatinib AFATINIB 26916115 23321 15869 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-2671 CHEMBL578878 23322 15870 ALOX15 246 ENZYME, DRUGGABLE GENOME GAVESTINEL SODIUM GAVESTINEL SODIUM 23323 15871 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME ROMIDEPSIN ROMIDEPSIN 23324 15872 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Alicaforsen ALICAFORSEN 23326 15873 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-26 23327 15874 HEBP1 50865 DRUGGABLE GENOME Benzo[d]oxazole derivative 4 23329 15875 TANC1 85461 CLINICALLY ACTIONABLE radiotherapy 24974847 23330 15876 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator CHEMBL3545292 QBW251 23331 15877 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 178101695 23332 15878 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GLPG-0492 GLPG0492 23333 15879 POLI 11201 DNA REPAIR NSC-60340 CHEMBL1534034 23335 15880 SERPINA6 866 DRUGGABLE GENOME, PROTEASE INHIBITOR Alclometasone ALCLOMETASONE 23337 15881 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ETHANOL ALCOHOL 15258586 23338 15882 EPHX2 2053 DRUGGABLE GENOME, ENZYME 6BIO 6BIO 24697244 23340 15883 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PROSTAGLANDIN A2 PROSTAGLANDIN A2 23341 15884 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL79 LIDOCAINE 23342 15885 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103690 AMLEXANOX 23343 15886 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE antibody 249565938 ANIFROLUMAB 23345 15887 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Pyridine derivative 20 23346 15888 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1726 NISOLDIPINE 23347 15889 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 381118806 ACALISIB 23349 15890 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MMV396678 CHEMBL1459149 23350 15891 SI 6476 DRUGGABLE GENOME, ENZYME TOTAL PARENTERAL NUTRITION 10712262 23351 15892 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Upadacitinib UPADACITINIB 23352 15893 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ENCLOMIPHENE CITRATE ENCLOMIPHENE CITRATE 23353 15894 GAA 2548 DRUGGABLE GENOME, ENZYME GNF-PF-372 CHEMBL580155 23354 15895 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER ACID BLUE 129 ACID BLUE 129 23355 15896 POLI 11201 DNA REPAIR ACRIFLAVINE CHLORIDE ACRIFLAVINE 23356 15897 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 249565659 CHEMBL411274 23359 15898 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178103351 CHEMBL2171124 23360 15899 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor IMATINIB IMATINIB 23361 15900 DDC 1644 ENZYME, DRUGGABLE GENOME inhibitor 178101809 23362 15901 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 252827462 RITONAVIR 23364 15902 XRCC1 7515 CLINICALLY ACTIONABLE fluorouracil FLUOROURACIL 23314736 23365 15903 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RITANSERIN RITANSERIN 23366 15904 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Neratinib NERATINIB 23371 15905 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE fentanyl FENTANYL 23372 15906 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 23373 15907 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TCMDC-124479 CHEMBL587259 23375 15908 ATAD5 79915 NA 1,4-BIS(2,6-DIFLUOROPHENYLSULFONYL)PIPERAZINE CHEMBL1093369 23377 15909 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR MONOCILLIN I MONOCILLIN I 16499313 23378 15910 PTPRG 5793 PROTEIN PHOSPHATASE, DRUGGABLE GENOME inhibitor 252827488 23380 15911 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CHLOROXINE CHLOROXINE 23381 15912 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33g 23382 15913 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Benzothiazine derivative 1 23384 15914 AKR1B1 231 DRUGGABLE GENOME, ENZYME Celiprolol hcl 23385 15915 FKBP5 2289 DRUGGABLE GENOME citalopram CITALOPRAM 18597649,21449676,20709156,19676097,15565110,23733030,17467808 23387 15916 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME inhibitor 223366150 23391 15917 KDM5B 10765 ENZYME inhibitor 178103605 23392 15918 TARDBP 23435 TUMOR SUPPRESSOR DICLOFENAC SODIUM DICLOFENAC SODIUM 23393 15919 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE DOXORUBICIN DOXORUBICIN 23394 15920 XRCC5 7520 KINASE TRIBUTYRIN TRIBUTYRIN 16000590 23396 15921 MAPT 4137 DRUGGABLE GENOME PHOSMET PHOSMET 23397 15922 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Dabrafenib DABRAFENIB 22608338,27659046,25370473,27797976,27255157,28268064,24265153,28512244,27770002,26732095,27500726,27523909,26811525,27048246,25265492,22735384,27697975,22389471,26392102,28784858,24885690,28891408,27312529,27080216,24265154 23398 15923 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1201607 NATALIZUMAB 23399 15924 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-27 23401 15925 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GNF-PF-2950 CHEMBL602807 23402 15926 POLI 11201 DNA REPAIR LUTEOLIN LUTEOLIN 23403 15927 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL NITRAZEPAM NITRAZEPAM 23404 15928 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME HuCART-meso cells 23405 15929 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME DIHYDROXANTHOHUMOL DIHYDROXANTHOHUMOL 23406 15930 TOP2B 7155 DRUGGABLE GENOME, ENZYME INNO-206 ALDOXORUBICIN 23407 15931 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-STYRYL-QUINOLINE CHEMBL127579 23408 15932 TPCN2 219931 ION CHANNEL, DRUGGABLE GENOME activator 178100233 23409 15933 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CARMINE CARMINE 23412 15934 DPEP1 1800 PROTEASE, DRUGGABLE GENOME, ENZYME Cilastatin CILASTATIN 23413 15935 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3545334 AVE8134 23414 15936 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650245 ETONITAZENE 23417 15937 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FUROXAN FUROXAN 23419 15938 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR L-DOPA LEVODOPA 16139809 23421 15939 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ATHRAQUINONES A ATHRAQUINONES A 23422 15940 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENAMIDONE FENAMIDONE 23423 15941 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OLANZAPINE OLANZAPINE 23424 15942 ITGA1 3672 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE SAN-300 SAN-300 23425 15943 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME rosiglitazone ROSIGLITAZONE 27271184 23426 15944 CA2 760 DRUGGABLE GENOME, ENZYME CHLOROTHIAZIDE CHLOROTHIAZIDE 23428 15945 KDM4A 9682 DRUGGABLE GENOME, ENZYME INDOCYANINE GREEN SODIUM INDOCYANINE GREEN 23430 15946 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Beta blocking agents, selective 23431 15947 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 135652069 23432 15948 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL2103836 IMAGABALIN 23436 15949 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor PAZOPANIB PAZOPANIB 23437 15950 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PD-153035 CHEMBL29197 23438 15951 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME DOVITINIB DOVITINIB 23439 15952 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AZ960 24398328 23441 15953 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME mirabegron MIRABEGRON 23445 15954 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PF-04449913 GLASDEGIB 23447 15955 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE CHEMBL457504 23448 15956 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIETHYLSTILBESTROL DIETHYLSTILBESTROL 23449 15957 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE phenobarbital PHENOBARBITAL 26049587 23450 15958 SLC15A1 6564 DRUGGABLE GENOME, TRANSPORTER 178101319 23451 15959 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR RO4927350 21705440 23452 15960 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME GSK2118436 DABRAFENIB 23454 15961 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ritonavir RITONAVIR 25923589 23455 15962 NOS2 4843 DRUGGABLE GENOME, ENZYME DIAZOXIDE DIAZOXIDE 12856829 23456 15963 MAOA 4128 DRUGGABLE GENOME, ENZYME TRANYLCYPROMINE TRANYLCYPROMINE 23457 15964 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE IL-1 23458 15965 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166854 23459 15966 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME ISOQUINOLINE-1,3(2H,4H)-DIONE CHEMBL1210769 23461 15967 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GOSSYPOL GOSSYPOL 23462 15968 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL ALPRAZOLAM ALPRAZOLAM 23463 15969 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Thiazolopyridine derivative 1 23464 15970 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE DOVITINIB DOVITINIB 22238366,26619011,18552176,23908597,23002168 23466 15971 E2F1 1869 TRANSCRIPTION FACTOR VASOPRESSIN VASOPRESSIN 12063292 23467 15972 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHENYTOIN PHENYTOIN 22931300 23470 15973 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PREDNISOLONE HEMISUCCINATE PREDNISOLONE HEMISUCCINATE 23471 15974 TOP2B 7155 DRUGGABLE GENOME, ENZYME Mitoxantrone MITOXANTRONE 23472 15975 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL2103744 MORPHINE SULFATE 23473 15976 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ETAZOLATE ETAZOLATE 23474 15977 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE BOSUTINIB BOSUTINIB 14745431,15256422,23676790,11853795,20697894,12623848,19466505,20367437,17114651,18828913,15381060,21895409,21489624,11964322,24456693,18615627,25157968,14559829,21605905,21562040,21505103,19652056,12399961 23476 15978 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR inhibitor 252166598 23477 15979 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor PI-103 PI-103 23479 15980 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 135651435 TRETINOIN 23480 15981 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 178102659 23482 15982 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Estradiol valerate/dienogest 23483 15983 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200443 MERETHOXYLLINE PROCAINE 23484 15984 TXNRD1 7296 DRUGGABLE GENOME Acyl oxymethyl acrylamide ester derivative 1 23487 15985 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AMITRAZ AMITRAZ 23488 15986 BAZ2B 29994 NA DIPYRIDYL DIPYRIDYL 23489 15987 KDM4A 9682 DRUGGABLE GENOME, ENZYME BIFONAZOLE BIFONAZOLE 23491 15988 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PEG-SN38 23492 15989 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER YW3-56 25612620 23493 15990 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 318164845 ABEDITEROL 23494 15991 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-19063 CHEMBL1310138 23496 15992 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 223366186 23497 15993 ALDH1L1 10840 DRUGGABLE GENOME l-methionine METHIONINE 24651765 23499 15994 MAP2K5 5607 KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME WX-554 WX-554 23500 15995 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000018300 CHEMBL590927 23501 15996 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME PMID27998201-Compound-22 23502 15997 GMNN 51053 DRUGGABLE GENOME CURCUMIN CURCUMIN 23503 15998 POLK 51426 DNA REPAIR, ENZYME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 23504 15999 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650630 23505 16000 FST 10468 DRUGGABLE GENOME KINASE INHIBITOR 16854407 23506 16001 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME panitumumab PANITUMUMAB 26438111 23509 16002 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME SR-123781A 23510 16003 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE CENISERTIB CENISERTIB 23512 16004 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME PMID27539678-Compound-16 23513 16005 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOPOTECAN TOPOTECAN 21440338 23514 16006 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME TACRINE TACRINE 23517 16007 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE antibody 178101741 PERTUZUMAB 23518 16008 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2105659 VARESPLADIB METHYL 23519 16009 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER paroxetine PAROXETINE 24192121,18215618,21449676,26704739,22641028 23521 16010 BAZ2B 29994 NA DAZOXIBEN HYDROCHLORIDE DAZOXIBEN HYDROCHLORIDE 23522 16011 NUDT15 55270 ENZYME, CLINICALLY ACTIONABLE Mercaptopurine MERCAPTOPURINE 23523 16012 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE KAMEBANIN KAMEBANIN 23524 16013 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SULPIRIDE SULPIRIDE 22931300 23525 16014 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME FLURAZEPAM FLURAZEPAM 23526 16015 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GNF-PF-5159 CHEMBL1493528 23527 16016 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE GDC-0941 PICTILISIB 27604488 23528 16017 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL NITRAZEPAM NITRAZEPAM 23530 16018 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NKTR-181 OXYCODEGOL 23531 16019 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-70 23532 16020 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR A-007 SIVIFENE 23534 16021 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE CUCURBITACIN E CUCURBITACIN E 20347305 23535 16022 PER1 5187 TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE MORPHINE MORPHINE 15977398 23536 16023 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PIOGLITAZONE PIOGLITAZONE 23539 16024 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor 363894147 MK-0873 23541 16025 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor 328083492 CERALASERTIB 23542 16026 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor 178101944 ROLIPRAM 23543 16027 COMT 1312 DRUGGABLE GENOME, ENZYME Drugs used in nicotine dependence 26555332 23544 16028 GSTM1 2944 DRUGGABLE GENOME, ENZYME PREDNISONE PREDNISONE 11186134 23545 16029 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE mycophenolate mofetil 22765258,16198654,18946804,22210424,20565459 23546 16030 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-16 23549 16031 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE DERAZANTINIB DERAZANTINIB 30420614,27627808 23550 16032 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL918 PHENACEMIDE 23553 16033 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 1,5-di-substituted pyridine derivative 1 23555 16034 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FENHEXAMID FENHEXAMID 23558 16035 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME MYRICETIN MYRICETIN 23560 16036 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DITHIODIMORPHOLINE DITHIODIMORPHOLINE 23562 16037 TNFRSF1A 7132 CELL SURFACE, DRUGGABLE GENOME infliximab INFLIXIMAB 22480748 23563 16038 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE PROTEIN KINASE INHIBITOR 9473774 23564 16039 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102667 23565 16040 TMEM97 27346 NA Benzamide derivative 2 23566 16041 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE APAP ACETAMINOPHEN 17188792 23567 16042 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME PRI-724 PRI-724 23568 16043 ITGA2 3673 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE E7820 E-7820 23570 16044 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME INSULIN INSULIN 23571 16045 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR SB-202190 SB-202190 22951114 23572 16046 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9340511, 2 23573 16047 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING BUPROPION HYDROCHLORIDE BUPROPION HYDROCHLORIDE 23574 16048 ABAT 18 DRUGGABLE GENOME, ENZYME inhibitor 178101523 VIGABATRIN 23576 16049 GCLM 2730 ENZYME H2O2 7615092 23578 16050 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135651256 23579 16051 ATAD5 79915 NA APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 23580 16052 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CURCUMIN CURCUMIN 15090070 23581 16053 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-127133 CHEMBL1172911 23582 16054 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 385612201 23583 16055 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Eletriptan ELETRIPTAN 23585 16056 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE trazodone TRAZODONE 18695978 23587 16057 GSTM1 2944 DRUGGABLE GENOME, ENZYME paclitaxel PACLITAXEL 26803611 23593 16058 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE tretinoin TRETINOIN 18695978 23594 16059 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650421 23596 16060 ATXN2 6311 NA TCMDC-124176 CHEMBL588038 23597 16061 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR BRYOSTATIN-1 23600 16062 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR EPALRESTAT EPALRESTAT 23601 16063 GJB5 2709 ION CHANNEL inhibitor 178101095 OCTANOL 23603 16064 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor SORAFENIB SORAFENIB 23608 16065 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME BMS-345541 BMS-345541 23609 16066 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MESTRANOL MESTRANOL 23610 16067 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR R(+)-BUTYLINDAZONE CHEMBL1256719 23611 16068 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME VALACYCLOVIR VALACYCLOVIR 24185376 23612 16069 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CAPTAN CAPTAN 23614 16070 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR atenolol ATENOLOL 15864115,20643254,15861037,16815314,20352314,12709726,12921807,15735607,18075464,12844134,22617224,11787477,17496726,14534524,21311897,14502278,20235788 23615 16071 LIPC 3990 ENZYME, PHOSPHOLIPASE, LIPASE, DRUGGABLE GENOME HEMOCLAR PENTOSAN POLYSULFATE SODIUM 2433786 23616 16072 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-693571 CHEMBL1287983 23618 16073 HTT 3064 DRUGGABLE GENOME MECETRONIUM MECETRONIUM 23619 16074 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE VINORELBIN DITARTRATE VINORELBINE TARTRATE 23620 16075 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ISATIN ISATIN 23621 16076 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PF-4455242 23622 16077 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 178102336 BOSUTINIB 23623 16078 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME EPINEPHRINE EPINEPHRINE 23624 16079 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE THEAFLAVINS 11591714 23625 16080 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME GLUCOCORTICOID 8968045 23628 16081 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL NIFEDIPINE NIFEDIPINE 23629 16082 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME Other general anesthetics 30136624 23631 16083 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2218887 23633 16084 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-3407 CHEMBL602990 23634 16085 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME IMIPRAMINE IMIPRAMINE 23635 16086 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL PHENOBARBITAL PHENOBARBITAL 23638 16087 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE TROGLITAZONE TROGLITAZONE 14764597 23639 16088 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102594 23640 16089 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME AMINODIMETHOXYQUINAZOLINYLPIPERAZINE AMINODIMETHOXYQUINAZOLINYLPIPERAZINE 23643 16090 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CFZ533 ISCALIMAB 23644 16091 PCNA 5111 NA VIT-100 23645 16092 TNFRSF1A 7132 CELL SURFACE, DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 22480748,24776844,25311255 23646 16093 ASGR1 432 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME AMG 529 23648 16094 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565884 A-443654 23649 16095 ALOX15 246 ENZYME, DRUGGABLE GENOME AM-404 CHEMBL39878 23651 16096 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PEITC 16921492 23652 16097 GMNN 51053 DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 23654 16098 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 249565940 AVOSENTAN 23655 16099 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE HEXACHLOROPHENE HEXACHLOROPHENE 23656 16100 FGA 2243 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, FIBRINOGEN ANISTREPLASE ANISTREPLASE 23657 16101 PTGS2 5743 DRUGGABLE GENOME, ENZYME VB-201 VB-201 23660 16102 F7 2155 ENZYME, DRUGGABLE GENOME, PROTEASE Recombinant factor VIIa PEGylated liposomal 23661 16103 TSPO 706 DRUGGABLE GENOME Isoquinoline carboxamide derivative 1 23663 16104 FNTA 2339 ENZYME, DRUGGABLE GENOME inhibitor TIPIFARNIB TIPIFARNIB 23665 16105 SCTR 6344 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1201488 SECRETIN SYNTHETIC HUMAN 23666 16106 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545299 BMS-698769 23667 16107 SLAMF7 57823 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor CHEMBL1743010 ELOTUZUMAB 23668 16108 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Gimatecan GIMATECAN 23670 16109 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PRN1109 23671 16110 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL1743070 SILTUXIMAB 23672 16111 CYBA 1535 TRANSPORTER idarubicin IDARUBICIN 19448608,28485375,16330681,25823784 23673 16112 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL271227 ABIRATERONE ACETATE 23674 16113 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Cobimetinib COBIMETINIB 22084396,25265494,28649441 23676 16114 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor RO 4929097 23678 16115 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 23679 16116 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200705 HYDROXYAMPHETAMINE HYDROBROMIDE 23680 16117 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650047 CALCIPOTRIOL 23681 16118 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Olaparib OLAPARIB 28363999 23682 16119 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Enzalutamide ENZALUTAMIDE 23683 16120 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SAR405838 SAR-405838 25145672,27550999,27765850 23684 16121 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX CID 1245272 CHEMBL408850 23686 16122 TXNRD1 7296 DRUGGABLE GENOME 4-aryl quinol derivative 1 23687 16123 CD27 939 PROTEASE INHIBITOR, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CDX-1127 VARLILUMAB 23692 16124 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR TGF-BETA 2 9272212 23694 16125 EPHA7 2045 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 381118815 23696 16126 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL408513 BELINOSTAT 23697 16127 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649706 23698 16128 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CURCUMIN CURCUMIN 25753330 23699 16129 COMT 1312 DRUGGABLE GENOME, ENZYME BIA 3-202 23700 16130 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME (S)-5-IODOWILLARDIINE CHEMBL121915 23703 16131 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 405560506 23705 16132 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SOTRASTAURIN SOTRASTAURIN 23706 16133 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Ritodrine RITODRINE 23707 16134 HMOX2 3163 ENZYME MORPHINE MORPHINE 14580950,10686338 23708 16135 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Altiratinib ALTIRATINIB 26285778,26965451,24362531 23709 16136 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL activator 135651381 23710 16137 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-31884 CHEMBL74644 23711 16138 LGR4 55366 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100589 23712 16139 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PF-477736 PF-00477736 26140595 23713 16140 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 23714 16141 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Debio1347 DEBIO-1347 23716 16142 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME 9cUAB-30 23719 16143 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565840 23720 16144 ATXN2 6311 NA FENRETINIDE FENRETINIDE 23721 16145 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL1201752 IXABEPILONE 23722 16146 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-10 23723 16147 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THIOPROPERAZINE MESYLATE THIOPROPERAZINE MESYLATE 23725 16148 CARM1 10498 ENZYME, METHYL TRANSFERASE, DRUGGABLE GENOME EOSIN EOSIN 18348515 23726 16149 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PREDNISONE PREDNISONE 22931300 23728 16150 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME peginterferon alfa-2b 21572301 23730 16151 PTGS2 5743 DRUGGABLE GENOME, ENZYME activator 381744924 23732 16152 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-34 23733 16153 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE Opioid anesthetics 30136624 23736 16154 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-136 23737 16155 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28270021-Compound-WO2015042088Example4 23738 16156 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ERGOLOID MESYLATE 23739 16157 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Zolmitriptan ZOLMITRIPTAN 23740 16158 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE IONOMYCIN IONOMYCIN 1701176 23741 16159 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ARQ-087 DERAZANTINIB 23742 16160 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-125293 CHEMBL548629 23743 16161 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIPHENYLENEIODONIUM DIPHENYLENEIODONIUM 23744 16162 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL ESTAZOLAM ESTAZOLAM 23745 16163 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME RUXOLITINIB RUXOLITINIB 26258521 23746 16164 GLS 2744 ENZYME PMID30273516-Compound-39 23749 16165 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE PMA 10679127 23750 16166 TOP2B 7155 DRUGGABLE GENOME, ENZYME Daniquidone DANIQUIDONE 23751 16167 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR THIORIDAZINE THIORIDAZINE 23752 16168 UGT1A6 54578 ENZYME, DRUGGABLE GENOME phenobarbital PHENOBARBITAL 26049587 23754 16169 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER THUNBERGINOL B THUNBERGINOL B 23756 16170 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL289228 TIPIFARNIB 23758 16171 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 proguanil CHLOROGUANIDE 9187528 23760 16172 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 23761 16173 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE COBALT 9144774 23762 16174 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PHOSMET PHOSMET 23764 16175 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL allosteric modulator 178100984 23765 16176 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL495 ALPROSTADIL 23766 16177 PTGS2 5743 DRUGGABLE GENOME, ENZYME MESALAZINE MESALAMINE 23767 16178 VCAM1 7412 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PHORBOL MYRISTATE ACETATE 7678355 23768 16179 CP 1356 DRUGGABLE GENOME, ENZYME CELL SURFACE ANTIGEN 9242695 23770 16180 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 387065613 23772 16181 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Ponatinib PONATINIB 27338794 23773 16182 CDK11B 984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3544942 RONICICLIB 23775 16183 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135651325 23776 16184 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL698 TETRACAINE 23779 16185 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GNF-PF-4945 CHEMBL585628 23780 16186 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL3182444 MK-5108 23781 16187 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-123713 CHEMBL586135 23782 16188 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AG-490 CHEMBL56543 23783 16189 ALOX15 246 ENZYME, DRUGGABLE GENOME (+)-EPITAXIFOLIN (+)-EPITAXIFOLIN 23784 16190 PDE4B 5142 DRUGGABLE GENOME, ENZYME CAFFEINE CAFFEINE 23785 16191 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650474 23786 16192 CCR6 1235 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE CHEMBL114544 23794 16193 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PARAOXON PARAOXON 23796 16194 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME AZ8010 22869148 23797 16195 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Amitriptyline AMITRIPTYLINE 23800 16196 RBFOX1 54715 NA antineoplastic agents 25823661 23801 16197 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor CHEMBL2041933 AZD-7762 23802 16198 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651088 23803 16199 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565739 AZD-6482 23804 16200 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE SF1126 23805 16201 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE BMS-299897 CHEMBL247471 23806 16202 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME EP217609 23808 16203 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135652140 23812 16204 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor CHEMBL1213490 ROMIDEPSIN 23813 16205 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565784 LY-2874455 23815 16206 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 381118914 23816 16207 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEMETON S DEMETON S 23818 16208 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME carboplatin CARBOPLATIN 21636554 23819 16209 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL2110814 DELUCEMINE 23820 16210 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PIFITHRIN-ALPHA CHEMBL198759 16862141 23822 16211 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102570 23823 16212 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PROSTAGLANDIN A2 PROSTAGLANDIN A2 23824 16213 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PTHRP 12417254 23825 16214 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME inhibitor PD 0325901 23826 16215 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor SARACATINIB SARACATINIB 23829 16216 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME DNDI1417156 CHEMBL1504679 23830 16217 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 25-HYDROXYCHOLECALCIFEROL CALCIFEDIOL 23831 16218 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 5,7-DIHYDROXYISOFLAVONE 5,7-DIHYDROXYISOFLAVONE 23832 16219 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FLUPHENAZINE HYDROCHLORIDE FLUPHENAZINE HYDROCHLORIDE 23833 16220 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE GEFITINIB GEFITINIB 23835 16221 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GEFITINIB GEFITINIB 23993328,19969465,20151670 23836 16222 ATXN2 6311 NA TCMDC-123927 CHEMBL531268 23837 16223 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL539423 SPARSENTAN 23838 16224 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-O3 23840 16225 CDC25C 995 KINASE, PROTEIN PHOSPHATASE, DRUGGABLE GENOME QUERCETIN QUERCETIN 11488465 23844 16226 GAPDH 2597 DRUGGABLE GENOME, ENZYME NSC-95397 CHEMBL429095 23845 16227 ATAD5 79915 NA SJ000113257 CHEMBL528694 23846 16228 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178103995 LINSITINIB 23847 16229 RAPGEF3 10411 ENZYME TANSHINONE I TANSHINONE I 23848 16230 GBA 2629 DRUGGABLE GENOME, ENZYME EBSELEN EBSELEN 23849 16231 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ONO-7475 23850 16232 PLCE1 51196 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME hydrochlorothiazide HYDROCHLOROTHIAZIDE 31327267 23852 16233 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SF1126 23853 16234 DHFR 1719 DRUGGABLE GENOME, ENZYME TCMDC-124296 CHEMBL22148 25984755 23854 16235 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENDILINE HYDROCHLORIDE FENDILINE HYDROCHLORIDE 23855 16236 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME MANNITOL MANNITOL 11471882 23856 16237 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER BISANTRENE BISANTRENE 9816258 23857 16238 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651611 23858 16239 CREB1 1385 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR lithium LITHIUM 24885933 23859 16240 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR antidepressants 22965830,21338649,23733030,23619509,19236730,29748862,20016225 23862 16241 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 374883851 23863 16242 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650788 23864 16243 MUTYH 4595 DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 24533712 23866 16244 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME SILIBININ SILIBININ 23401473 23867 16245 UBE2N 7334 ENZYME, DRUGGABLE GENOME TCMDC-124022 CHEMBL548017 23870 16246 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AMSACRINE AMSACRINE 23874 16247 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE XL228 XL-228 23875 16248 ALOX5 240 DRUGGABLE GENOME, ENZYME Flobufen 23876 16249 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BROMODIOLONE BROMODIOLONE 23877 16250 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PICTILISIB PICTILISIB 23360348 23879 16251 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR latanoprost LATANOPROST 27336732,25339146,17467803 23880 16252 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NXN-188 23881 16253 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor GSK2126458 OMIPALISIB 23882 16254 NFKBIA 4792 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME DEMETHYLWEDELOLACTONE DEMETHYLWEDELOLACTONE 22926226 23883 16255 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417300 CHEMBL1401091 23884 16256 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135649890 ACIPIMOX 23886 16257 IFNGR1 3459 DRUGGABLE GENOME, CLINICALLY ACTIONABLE INDOLE-3-CARBINOL INDOLE-3-CARBINOL 14988219 23887 16258 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GUTHION GUTHION 23890 16259 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BW-373U86 CHEMBL25230 23891 16260 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Larotrectinib LAROTRECTINIB 23892 16261 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL501867 VINCRISTINE SULFATE 23895 16262 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL501867 VINCRISTINE SULFATE 23897 16263 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL2107869 INSULIN DEGLUDEC 23898 16264 BRCA2 675 CLINICALLY ACTIONABLE Olaparib OLAPARIB 26510020,26546619,20609467,25366685,26116172,21097693 23899 16265 PTGS1 5742 ENZYME, DRUGGABLE GENOME GINGER GINGER 14693173 23901 16266 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1201103 METHOXAMINE HYDROCHLORIDE 23902 16267 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR BCG BCG VACCINE 14742634 23904 16268 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GNF-PF-3889 CHEMBL598270 23906 16269 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR TRANSFORMING GROWTH FACTOR 11746354 23909 16270 RNPEPL1 57140 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL2103847 TOSEDOSTAT 23913 16271 BAZ2B 29994 NA TCMDC-125066 CHEMBL533577 23914 16272 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE ANTISERUM 16482517 23917 16273 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR BISPHOSPHONATES 15590626 23918 16274 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist CHEMBL1276308 MIFEPRISTONE 23920 16275 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME ALSTERPAULLONE ALSTERPAULLONE 23921 16276 BMP2 650 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR METHYL 4-AMINOBENZOATE CHEMBL1927048 22041064 23923 16277 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME AMINACRINE HYDROCHLORIDE AMINACRINE HYDROCHLORIDE 23924 16278 MAGEA3 4102 ENZYME, DRUGGABLE GENOME GL-0817 BIROPEPIMUT-S 23925 16279 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 670282 CHEMBL260213 23926 16280 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor BMS-599626 AC-480 23930 16281 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ADECATUMUMAB ADECATUMUMAB 23931 16282 CBX1 10951 NA SB-202190 SB-202190 23933 16283 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1159650 CLOBETASOL PROPIONATE 23934 16284 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-Table1Example16 23935 16285 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR SNS-314 SNS-314 23937 16286 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Aminooxazole carboxamide derivative 1 23939 16287 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE CHEMBL114544 23940 16288 IL18 3606 DRUGGABLE GENOME Iboctadekin IBOCTADEKIN 23941 16289 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE MACROPHAGE COLONY STIMULATING FACTOR 3877730 23942 16290 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CLORAZEPATE CLORAZEPIC ACID 23943 16291 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CLOTIAZEPAM CLOTIAZEPAM 23944 16292 BAZ2B 29994 NA STILONIUM IODIDE STILONIUM IODIDE 23945 16293 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE PLX9486 23946 16294 GLA 2717 ENZYME, DRUGGABLE GENOME Migalastat MIGALASTAT 23948 16295 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MECHLORETHAMINE HYDROCHLORIDE MECHLORETHAMINE HYDROCHLORIDE 23949 16296 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody BIIB022 23950 16297 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL CHLORZOXAZONE CHLORZOXAZONE 23951 16298 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-2335 CHEMBL601146 23952 16299 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MIRIPIRIUM CHLORIDE MIRIPIRIUM CHLORIDE 23953 16300 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TAE-684 TAE-684 23954 16301 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR ESTRAMUSTINE ESTRAMUSTINE 23956 16302 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ISOPROPANOL ISOPROPYL ALCOHOL 6409434 23957 16303 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102561 BOHEMINE 23958 16304 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PYRITHIONE PYRITHIONE 23959 16305 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GSK2334470 CHEMBL1765740 27451907 23963 16306 ATAD5 79915 NA AURIN AURIN 23965 16307 CDC42 998 DRUGGABLE GENOME SECRAMINE B SECRAMINE B 16408091 23966 16308 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor AS703569 CENISERTIB 23967 16309 TUBB 203068 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 23968 16310 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 178101606 DORSOMORPHIN 23969 16311 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE IODOPHTHALEIN IODOPHTHALEIN 23970 16312 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-4832 CHEMBL601137 23971 16313 HMOX1 3162 ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE SELENIUM 12751798 23972 16314 PTK6 5753 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, ENZYME OSI-632 OSI-632 23973 16315 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME efavirenz / emtricitabine / tenofovir disoproxil 23975 16316 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Scopolamine SCOPOLAMINE 23976 16317 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME DARBEPOETIN ALFA 23977 16318 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE ANTI-CTLA-4 MONOCLONAL ANTIBODY 25970248 23981 16319 COP1 64326 CLINICALLY ACTIONABLE, ENZYME Quinine QUININE 23982 16320 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650232 ENPROSTIL 23983 16321 F11 2160 DRUGGABLE GENOME, PROTEASE, ENZYME DEXTRAN SULFATE 12968031 23984 16322 MAP3K5 4217 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565756 23987 16323 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565738 23988 16324 CBX1 10951 NA GNF-PF-1969 CHEMBL601364 23989 16325 DCBLD1 285761 NA cisplatin CISPLATIN 23478653 23990 16326 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR RETINOIC ACID 10809758 23992 16327 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor CHR-3996 NANATINOSTAT 23993 16328 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR NORGESTREL NORGESTREL 23995 16329 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 252166731 RO-5028442 23996 16330 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME CID 94381 CHEMBL374632 23999 16331 KDM4A 9682 DRUGGABLE GENOME, ENZYME ORPHENADRINE CITRATE ORPHENADRINE CITRATE 24001 16332 XRCC1 7515 CLINICALLY ACTIONABLE DOCETAXEL DOCETAXEL 19157633 24002 16333 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL1201179 LAPATINIB DITOSYLATE 24003 16334 TARDBP 23435 TUMOR SUPPRESSOR SQ-22536 CHEMBL64239 24004 16335 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME Ridaforolimus RIDAFOROLIMUS 24006 16336 ALDH1A1 216 DRUGGABLE GENOME, ENZYME THYROXINE THYROXINE 24007 16337 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GNF-PF-5510 CHEMBL578741 24008 16338 PSMA2 5683 DRUGGABLE GENOME, PROTEASE BORTEZOMIB BORTEZOMIB 24524217 24009 16339 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME curcumin CURCUMIN 25587128 24010 16340 TDP2 51567 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GNF-PF-4418 CHEMBL604321 24011 16341 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200790 METHYPRYLON 24013 16342 GMNN 51053 DRUGGABLE GENOME 4,4'-BIPYRIDINE CHEMBL1374568 24014 16343 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 20 24015 16344 NOS1 4842 DRUGGABLE GENOME, ENZYME IL-1RA ANAKINRA 9206098 24016 16345 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME EPHEDRINE SULFATE EPHEDRINE SULFATE 24018 16346 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051793 GIVINOSTAT 24019 16347 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE HESPERIDIN HESPERIDIN 24020 16348 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 178102597 24021 16349 TNFRSF4 7293 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Anti-OX40 mab 24022 16350 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ALITRETIONINE 24024 16351 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME inhibitor 223366192 RELACATIB 24025 16352 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist CHEMBL1201515 PEGVISOMANT 24027 16353 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MIANSERIN MIANSERIN 18033297 24029 16354 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME AZD-1775 ADAVOSERTIB 24033 16355 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GALLAMINE GALLAMINE 24034 16356 CALR 811 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME RETINOIC ACID 9013706 24035 16357 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE PMID28460551-Compound-6 24036 16358 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME NICLOSAMIDE NICLOSAMIDE 24037 16359 SLC1A5 6510 TRANSPORTER inhibitor 178101229 BENZYLCYSTEINE 24039 16360 CCL11 6356 DRUGGABLE GENOME TNF-ALPHA 15972682 24040 16361 HMGCR 3156 ENZYME, DRUGGABLE GENOME XZK-monascus 24041 16362 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178101961 THIORPHAN 24042 16363 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FP-1039 FP-1039 23226697 24044 16364 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Benzimidazole and imadazopyridine carboximidamide compound 2 24045 16365 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL FLURAZEPAM FLURAZEPAM 24046 16366 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME INTERLEUKIN-1 12421568 24048 16367 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 336446949 24049 16368 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE RADIATION THERAPY 26589432 24050 16369 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PANOBINOSTAT PANOBINOSTAT 24051 16370 GAA 2548 DRUGGABLE GENOME, ENZYME OLANZAPINE OLANZAPINE 24052 16371 PTGS1 5742 ENZYME, DRUGGABLE GENOME TENOXICAM TENOXICAM 24053 16372 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Panitumumab PANITUMUMAB 22797062 24054 16373 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-4579 CHEMBL584626 24055 16374 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PF-05212384 GEDATOLISIB 24056 16375 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENOXYBENZAMINE PHENOXYBENZAMINE 24057 16376 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR SULFURETIN SULFURETIN 24058 16377 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE LY-2090314 LY-2090314 24059 16378 FST 10468 DRUGGABLE GENOME INDOMETHACIN INDOMETHACIN 15941869 24060 16379 TNFRSF9 3604 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE PF-05082566 UTOMILUMAB 24061 16380 OAT 4942 ENZYME, DRUGGABLE GENOME GABACULINE GABACULINE 26288681 24063 16381 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 893238 CHEMBL473735 24065 16382 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 5-CARBOXAMIDOTRYPTAMINE MALEATE CHEMBL1256863 24066 16383 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE ORPHENADRINE ORPHENADRINE 24069 16384 ATAD5 79915 NA SHINJULACTONE B SHINJULACTONE B 24071 16385 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE MODIFIED IFN-BETA 24072 16386 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PHENYLBUTANOIC ACID PHENYLBUTANOIC ACID 24044874 24073 16387 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME ALPRAZOLAM ALPRAZOLAM 22137933 24075 16388 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE KENPAULLONE KENPAULLONE 24076 16389 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR METHYLENE BLUE METHYLENE BLUE 24078 16390 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody PANITUMUMAB PANITUMUMAB 24079 16391 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE N/A 24081 16392 COMT 1312 DRUGGABLE GENOME, ENZYME paroxetine PAROXETINE 18989660 24083 16393 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GOSSYPOL GOSSYPOL 24084 16394 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CLOTIAZEPAM CLOTIAZEPAM 24087 16395 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651591 DIQUAFOSOL 24089 16396 FANCC 2176 CLINICALLY ACTIONABLE, DNA REPAIR CISPLATIN CISPLATIN 16243825 24090 16397 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650258 FENTANYL 24091 16398 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1201160 RITODRINE HYDROCHLORIDE 24092 16399 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor PALBOCICLIB PALBOCICLIB 24093 16400 POLK 51426 DNA REPAIR, ENZYME FLUORESCEIN FLUORESCEIN 24094 16401 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE BUCINDOLOL BUCINDOLOL 24098 16402 PAK2 5062 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 310264720 24099 16403 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651300 24100 16404 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE INDOMETHACIN INDOMETHACIN 11950807 24102 16405 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RU 486 1302037 24104 16406 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BROXYQUINOLINE BROXYQUINOLINE 24105 16407 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLOMIPRAMINE CLOMIPRAMINE 24106 16408 CBX1 10951 NA PYRONIN Y PYRONIN Y 24107 16409 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 223366042 CAPIVASERTIB 24111 16410 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Phenylpropionic acid derivative 1 24112 16411 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565617 RIVICICLIB 24113 16412 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Five membered heterocyclic benzamide derivative 3 24114 16413 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker 178100816 MECAMYLAMINE 24115 16414 GNA11 2767 CLINICALLY ACTIONABLE SELUMETINIB SELUMETINIB 26619011,2549426,22808163,24141786,21083380,21444680,25157968,1328859,22733540 24116 16415 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DAIDZEIN DAIDZEIN 24117 16416 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649889 ACIFRAN 24118 16417 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHLOROXINE CHLOROXINE 24119 16418 GLIPR1 11010 NA AdRTVP-1 24120 16419 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102726 24121 16420 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FENCLONINE FENCLONINE 24124 16421 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Piperidine derivative 6 24125 16422 RACGAP1 29127 NA BENZIDINE BENZIDINE 24126 16423 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE ALISERTIB ALISERTIB 24127 16424 PLA2G10 8399 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME inhibitor 252827445 24129 16425 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE VANDETANIB VANDETANIB 24130 16426 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DICHLORODIMETHYLSTANNANE DICHLORODIMETHYLSTANNANE 24131 16427 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME DAUNORUBICIN DAUNORUBICIN 22260166 24133 16428 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE Romiplostim ROMIPLOSTIM 24134 16429 GMNN 51053 DRUGGABLE GENOME FLUOROSALAN FLUOROSALAN 24137 16430 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TROPOLONE TROPOLONE 24138 16431 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201538 INSULIN LISPRO 24141 16432 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE BMS-986189 24142 16433 PDE3A 5139 ENZYME, DRUGGABLE GENOME opioids 24143 16434 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE activator 135652752 24146 16435 CA12 771 DRUGGABLE GENOME Curcumin CURCUMIN 24149 16436 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103106 CANDOXATRIL 24150 16437 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL1628502 GABAPENTIN ENACARBIL 24152 16438 MAPT 4137 DRUGGABLE GENOME NSC-11437 CHEMBL1814509 24154 16439 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE JNJ-26483327 JNJ-26483327 24155 16440 CASP8 841 DRUGGABLE GENOME, PROTEASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 178101978 24156 16441 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 24158 16442 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME VINORELBINE VINORELBINE 11720482 24159 16443 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Premarin/Trimegestone 20838656 24160 16444 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201557 INTERFERON ALFACON-1 24162 16445 POLI 11201 DNA REPAIR TCMDC-125180 CHEMBL586163 24164 16446 FXYD2 486 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL254219 DIGITOXIN 24166 16447 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR Macrocycle derivative 14 24167 16448 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Vilaprisan VILAPRISAN 24169 16449 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650101 24170 16450 SV2A 9900 DRUGGABLE GENOME, TRANSPORTER LEVETIRACETAM LEVETIRACETAM 24171 16451 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE FX-007 24172 16452 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 363894217 VORUCICLIB 24175 16453 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201142 RASAGILINE MESYLATE 24176 16454 BAZ2B 29994 NA N,N'-DIPHENYL-P-PHENYLENEDIAMINE N,N'-DIPHENYL-P-PHENYLENEDIAMINE 24177 16455 COP1 64326 CLINICALLY ACTIONABLE, ENZYME Tocainide TOCAINIDE 24178 16456 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PYROGALLOL RED PYROGALLOL RED 24181 16457 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor BEZ235 DACTOLISIB 24182 16458 IGF2BP2 10644 NA repaglinide REPAGLINIDE 24184 16459 RPSA 3921 NA PMID25747044-Compound-miRNA 24185 16460 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE LEVOMEPROMAZINE MALEATE LEVOMEPROMAZINE MALEATE 24187 16461 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE LM-CD45 24188 16462 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ESTRAMUSTINE ESTRAMUSTINE 24189 16463 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME RG-1530 RG-1530 24190 16464 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME TAMATINIB R-406 24191 16465 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR Trametinib TRAMETINIB 26487278 24192 16466 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY PREDNISOLONE PREDNISOLONE 3427792,8636270 24193 16467 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Trametinib TRAMETINIB 26343583,28783719,27760111,22805292,27488531,27500726,28514312,22389471,22983396,28179366 24195 16468 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME TANDUTINIB TANDUTINIB 24196 16469 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL105060 DNK333 24198 16470 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565832 24199 16471 MAP3K7 6885 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565754 24200 16472 GMNN 51053 DRUGGABLE GENOME 3,5 DIBROMOTYROSINE DIBROMOTYROSINE 24201 16473 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DNDI1417467 CHEMBL1997335 24203 16474 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR KC706 24204 16475 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Fludarabine FLUDARABINE 24205 16476 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Saracatinib SARACATINIB 23242808 24206 16477 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE OXPRENOLOL OXPRENOLOL 24207 16478 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR MORIN MORIN 24209 16479 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor MGCD265 GLESATINIB 24210 16480 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CNTO 148 24211 16481 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (S)-ISRADIPINE (S)-ISRADIPINE 24212 16482 MPHOSPH8 54737 NA TETRADECYLTHIOACETIC ACID TETRADECYLTHIOACETIC ACID 24213 16483 HP 3240 DRUGGABLE GENOME, PROTEASE, ENZYME PYRIDOXINE PYRIDOXINE 6935482 24214 16484 ALDH1A1 216 DRUGGABLE GENOME, ENZYME EMODIC ACID EMODIC ACID 24215 16485 PSIP1 11168 CLINICALLY ACTIONABLE US9132129, Cpd002 24217 16486 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Doxil DOXIL 21216929 24218 16487 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TCMDC-123781 CHEMBL581194 24219 16488 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE DURVALUMAB DURVALUMAB 28472902 24220 16489 PGF 5228 GROWTH FACTOR, DRUGGABLE GENOME inhibitor CHEMBL1742982 AFLIBERCEPT 24221 16490 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL3545105 POL6326 24222 16491 BRCA2 675 CLINICALLY ACTIONABLE Cyclophosphamide CYCLOPHOSPHAMIDE 25589624 24224 16492 MAPT 4137 DRUGGABLE GENOME WORTMANNIN WORTMANNIN 24225 16493 CD44 960 DRUGGABLE GENOME, CELL SURFACE MPA PROGESTERONE 11605071 24226 16494 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE vincristine VINCRISTINE 24227 16495 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TCMDC-124224 CHEMBL580421 24228 16496 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE SAR-100842 25593637 24229 16497 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-34 24230 16498 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DIETHYLSTILBESTROL DIETHYLSTILBESTROL 24231 16499 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GOSSYPETIN GOSSYPETIN 25190466 24233 16500 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ANESTHETICS 16738805 24234 16501 CA1 759 DRUGGABLE GENOME, ENZYME SULFAMIDE SULFAMIDE 24235 16502 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ESTRADIOL ESTRADIOL 22931300 24236 16503 ITPR1 3708 ION CHANNEL, KINASE, DRUGGABLE GENOME, TRANSPORTER activator 135652731 24239 16504 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CURCUMIN CURCUMIN 24240 16505 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178103273 KETOROLAC 24241 16506 MAPT 4137 DRUGGABLE GENOME NSC-102742 CHEMBL1519374 24242 16507 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 IPRONIAZID IPRONIAZID 22931300 24244 16508 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE BMS-599626 AC-480 24246 16509 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE IMC-3G3 OLARATUMAB 24247 16510 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TYRPHOSTIN AG-835 CHEMBL261557 24248 16511 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE MI-503 27535106 24251 16512 GMNN 51053 DRUGGABLE GENOME CRYPTOTANSHINONE CRYPTOTANSHINONE 24254 16513 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME terbinafine TERBINAFINE 24255 16514 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME RHEIN RHEIN 24256 16515 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME ALVOCIDIB ALVOCIDIB 24259 16516 NDUFA4L2 56901 NA inhibitor CHEMBL3545135 NV-128 24260 16517 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor BELINOSTAT BELINOSTAT 24261 16518 MAOB 4129 DRUGGABLE GENOME, ENZYME SAFINAMIDE SAFINAMIDE 23631427,24560738 24263 16519 AREG 374 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE CRIZOTINIB CRIZOTINIB 21791641 24265 16520 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR TAMOXIFEN TAMOXIFEN 24266 16521 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME BVI-007 24267 16522 BAZ2B 29994 NA LOBARIC ACID LOBARIC ACID 24268 16523 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2103858 NARONAPRIDE 24269 16524 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE CENISERTIB CENISERTIB 24270 16525 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 zidovudine ZIDOVUDINE 22960662,9187528 24273 16526 NME2 4831 KINASE zidovudine ZIDOVUDINE 22960662 24276 16527 PTGS2 5743 DRUGGABLE GENOME, ENZYME E163 E163 10075763 24283 16528 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE AT-7519 AT-7519 24284 16529 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102547 24285 16530 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650416 24286 16531 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 249565716 24287 16532 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GW1929 CHEMBL434063 24289 16533 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME FLUNARIZINE FLUNARIZINE 24290 16534 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 178102666 24293 16535 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor SF1126 24294 16536 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102735 24295 16537 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL270995 BRIVANIB ALANINATE 24298 16538 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FISETIN FISETIN 24302 16539 BAZ2B 29994 NA GNF-PF-2947 CHEMBL581677 24305 16540 PIGF 5281 DRUGGABLE GENOME antibody ZALTRAP ZALTRAP 24306 16541 DNER 92737 NA Isoxazole-based bicyclic compound 1 24308 16542 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR Guggulsterone GUGGULSTERONE 24310 16543 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650583 METHIMEPIP 24312 16544 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR FLUPIRTINE MALEATE FLUPIRTINE MALEATE 24314 16545 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3544983 TESEVATINIB 24315 16546 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102570 24316 16547 UGT1A10 54575 DRUGGABLE GENOME, ENZYME allopurinol ALLOPURINOL 27798726 24317 16548 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR SLAZINIC ACID SLAZINIC ACID 24318 16549 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor AS703569 CENISERTIB 24319 16550 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 15193230 24320 16551 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME AMBUNOL AMBUNOL 24321 16552 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR SJ000014858 CHEMBL591628 24322 16553 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MERCURIC CHLORIDE MERCURIC CHLORIDE 24323 16554 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor DASATINIB DASATINIB 24324 16555 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 249565898 24330 16556 GLS 2744 ENZYME CEFSULODIN SODIUM CEFSULODIN SODIUM 24331 16557 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE CID 5330286 24332 16558 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME AZD-1080 AZD-1080 24333 16559 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Aryl sulphoxide imine derivative 1 24334 16560 POLK 51426 DNA REPAIR, ENZYME CEFOTAXIME SODIUM CEFOTAXIME SODIUM 24335 16561 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL608533 MIDOSTAURIN 24337 16562 LGMN 5641 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 252166833 24338 16563 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME PF-562271 PF-00562271 24340 16564 PPAT 5471 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200400 AZATHIOPRINE SODIUM 24342 16565 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178101056 24343 16566 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY AMIODARONE AMIODARONE 8778159 24344 16567 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE DITHIAZANINE IODIDE DITHIAZANINE IODIDE 24345 16568 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LINIFANIB LINIFANIB 24347 16569 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUOXYMESTERONE FLUOXYMESTERONE 24348 16570 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIPHENYL PHOSPHATE TRIPHENYL PHOSPHATE 24349 16571 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL1773 CAPECITABINE 24350 16572 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor 404859153 24351 16573 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL608533 MIDOSTAURIN 24354 16574 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE MC-2001 24356 16575 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE SUNITINIB SUNITINIB 16638875,18955458,22261812,25239608,22439647,26772734 24357 16576 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME NORTRIPTYLINE NORTRIPTYLINE 24358 16577 SDC1 6382 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CD138 CAR T cells 24359 16578 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 178103784 LEVALLORPHAN 24363 16579 HOXA9 3205 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE G-CSF FILGRASTIM 11687616 24364 16580 GMNN 51053 DRUGGABLE GENOME TDR77593 CHEMBL1510164 24365 16581 ATAD5 79915 NA GNF-PF-1813 CHEMBL577662 24368 16582 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL inhibitor 178101216 ISRADIPINE 24369 16583 CBX1 10951 NA FLUSPIRILENE FLUSPIRILENE 24371 16584 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE cyclophosphamide CYCLOPHOSPHAMIDE 24599932,24958282 24373 16585 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE LYSINE LYSINE 27875625 24374 16586 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-18 24376 16587 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-377852 CHEMBL1466186 24378 16588 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 178103584 24379 16589 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL2107762 NERISPIRDINE 24381 16590 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE IMATINIB IMATINIB 24382 16591 POLI 11201 DNA REPAIR MONTELUKAST SODIUM MONTELUKAST SODIUM 24383 16592 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL1201733 PAZOPANIB HYDROCHLORIDE 24384 16593 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1200367 ECHOTHIOPHATE IODIDE 24385 16594 MAP3K7 6885 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 348353615 24386 16595 VAMP2 6844 DRUGGABLE GENOME PMA 17196367 24387 16596 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL574737 UCN-01 24389 16597 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PD-153035 CHEMBL29197 17681471 24390 16598 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IIIE AESCULIOSIDE IIIE 20371180 24391 16599 ITPA 3704 ENZYME mercaptopurine MERCAPTOPURINE 26237184,18685564,21395650 24394 16600 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CELASTROL CELASTROL 25756299 24395 16601 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME busulfan BUSULFAN 24396 16602 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HYDROXYZINE HYDROXYZINE 22931300 24398 16603 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Vandetanib VANDETANIB 25910950 24399 16604 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CIANIDANOL CIANIDANOL 24400 16605 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Veliparib VELIPARIB 26801247,25824335,25589624,26842236 24402 16606 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102264 24403 16607 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 HYCANTHONE HYCANTHONE 22931300 24404 16608 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME activator 135651219 SURAMIN 24405 16609 DUSP1 1843 PROTEIN PHOSPHATASE, KINASE, DRUGGABLE GENOME Avastin+/-Tarceva 24406 16610 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME COMBRETASTATIN A4 COMBRETASTATIN A4 22982122 24407 16611 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME IL-1 15084582 24408 16612 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-6 24409 16613 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor AZD8330 24410 16614 MAPT 4137 DRUGGABLE GENOME CYSTAMINE DIHYDROCHLORIDE CYSTAMINE DIHYDROCHLORIDE 24411 16615 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CHLOROTHALONIL CHLOROTHALONIL 24412 16616 ATAD5 79915 NA DNDI1417215 CHEMBL1390650 24413 16617 TJP1 7082 KINASE, TRANSCRIPTION FACTOR DEXAMETHASONE DEXAMETHASONE 8206910 24414 16618 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL FOSPROPOFOL FOSPROPOFOL 24415 16619 ATXN2 6311 NA CLOTRIMAZOLE CLOTRIMAZOLE 24417 16620 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor AXITINIB AXITINIB 24418 16621 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CART-HER-2 24419 16622 PI4KA 5297 DRUGGABLE GENOME, ENZYME, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE BYL719 ALPELISIB 24420 16623 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DITHIAZANINE DITHIAZANINE 24421 16624 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 384403641 RG-1530 24424 16625 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE MRK-003 25104330 24427 16626 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME allosteric modulator 178103908 ETAZOLATE 24428 16627 CXCL8 3576 DRUGGABLE GENOME ENDOSULFAN ENDOSULFAN 24431 16628 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROGABIDE PROGABIDE 24432 16629 QPCT 25797 ENZYME, PROTEASE, DRUGGABLE GENOME PQ-912 24403873 24433 16630 ATAD5 79915 NA DNDI1417031 CHEMBL1333049 24434 16631 TGFBR3 7049 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME BFGF 1556106 24436 16632 DHFR 1719 DRUGGABLE GENOME, ENZYME SULFASALAZINE SULFASALAZINE 22555 24437 16633 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE activator CHEMBL2108147 STREPTOKINASE 24439 16634 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME Altiratinib ALTIRATINIB 24443 16635 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR TRIVALENT INFLUENZA VACCINE 12409329 24444 16636 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ATHRAQUINONES A ATHRAQUINONES A 24445 16637 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE capecitabine CAPECITABINE 24980946 24447 16638 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL107 COLCHICINE 24449 16639 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR DIGOXIN DIGOXIN 12691286 24450 16640 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 249565825 24451 16641 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PF-562271 PF-00562271 24452 16642 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR INSULIN INSULIN 11956149 24453 16643 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor AZD8931 SAPITINIB 24454 16644 COL4A2 1284 DRUGGABLE GENOME NLG919 NAVOXIMOD 24455 16645 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE inhibitor 348353652 24456 16646 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR BGP-15 24457 16647 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE A66 23674493,21668414 24458 16648 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-124353 CHEMBL529918 24460 16649 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR KENPAULLONE KENPAULLONE 24461 16650 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545147 IMD-2560 24462 16651 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE nitrous oxide 18580170 24464 16652 POLK 51426 DNA REPAIR, ENZYME ASTERRIC ACID ASTERRIC ACID 24465 16653 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor TAK-733 TAK-733 24466 16654 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME Enasidenib ENASIDENIB 24467 16655 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417263 CHEMBL1431115 24468 16656 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 178101238 24470 16657 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ribavirin RIBAVIRIN 23360626 24471 16658 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 135651567 24472 16659 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1234354 PF-04691502 24473 16660 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100357 24474 16661 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRICLOSAN TRICLOSAN 24475 16662 PRKAA2 5563 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME METFORMIN HYDROCHLORIDE 24477 16663 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Triazolo-pyridine derivative 1 24478 16664 CBX1 10951 NA PAPAVERINE PAPAVERINE 24479 16665 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor 363894146 24480 16666 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE FULVESTRANT FULVESTRANT 31091374 24482 16667 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME 6-THIOGUANINE THIOGUANINE 1207869 24484 16668 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE MK-5108 MK-5108 24486 16669 KDM4A 9682 DRUGGABLE GENOME, ENZYME ENCLOMIPHENE ENCLOMIPHENE 24487 16670 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TOLCAPONE TOLCAPONE 24490 16671 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651190 24491 16672 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE TANDUTINIB TANDUTINIB 24492 16673 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Navitoclax NAVITOCLAX 26474387 24494 16674 PTGES 9536 DRUGGABLE GENOME, ENZYME inhibitor 348353668 24495 16675 TUBB6 84617 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 24496 16676 HSPA4 3308 NA PKC412 MIDOSTAURIN 17032922 24497 16677 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE eszopiclone ESZOPICLONE 18695978 24498 16678 NDUFS5 4725 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 24499 16679 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 329968451 SOLABEGRON 24501 16680 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MEPENZOLATE MEPENZOLATE 24503 16681 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Volitinib SAVOLITINIB 24504 16682 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME QUINOXALINE-2-CARBOXYLIC ACID CHEMBL151797 24506 16683 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135649895 24507 16684 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OXYBUTYNIN OXYBUTYNIN 24511 16685 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 carbamazepine CARBAMAZEPINE 21738081,26574235,9187528,25495409,26421491,23252947 24514 16686 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL1683544 ERIBULIN MESYLATE 24518 16687 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR THUNBERGINOL B THUNBERGINOL B 24519 16688 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 53801089 HYDROCORTISONE 24520 16689 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR QUINOXYFEN QUINOXYFEN 24522 16690 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CHEMBL407 FLUMAZENIL 24523 16691 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LY2874455 LY-2874455 23175443,28034880,21900693 24524 16692 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HYCANTHONE HYCANTHONE 24525 16693 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor 363894172 24526 16694 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor REGORAFENIB REGORAFENIB 24527 16695 MBNL1 4154 DRUGGABLE GENOME LOMOFUNGIN LOMOFUNGIN 24529 16696 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY ETHER ETHER 9721940 24531 16697 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL MC-1 24532 16698 PSMC4 5704 NA inhibitor CARFILZOMIB CARFILZOMIB 24533 16699 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178101606 DORSOMORPHIN 24534 16700 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ABAMECTIN ABAMECTIN 24536 16701 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ATORVASTATIN ATORVASTATIN 16796407 24537 16702 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1200611 24539 16703 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AIR645 24540 16704 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CARVEDILOL CARVEDILOL 24541 16705 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CHEMBL3039540 ADUCANUMAB 24542 16706 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE AMILORIDE AMILORIDE 24543 16707 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-215505 CHEMBL2110371 24544 16708 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE NIVOLUMAB NIVOLUMAB 26918451,26086854,28472902 24545 16709 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE PD-0325901 PD-0325901 26936919 24547 16710 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PD173074 22837387,22869148,25589496 24549 16711 GSTT1 2952 DRUGGABLE GENOME troglitazone TROGLITAZONE 12732844 24550 16712 LATS2 26524 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565889 24551 16713 FGB 2244 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, FIBRINOGEN, DRUGGABLE GENOME eptifibatide EPTIFIBATIDE 20938371 24552 16714 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IIA AESCULIOSIDE IIA 20371180 24553 16715 PRKG1 5592 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565578 IPATASERTIB 24554 16716 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIACEREIN DIACEREIN 24555 16717 SGPL1 8879 ENZYME, DRUGGABLE GENOME LX2931 LX-2931 24556 16718 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1700 SOTALOL HYDROCHLORIDE 24557 16719 POLI 11201 DNA REPAIR MORIN MORIN 24558 16720 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME KENPAULLONE KENPAULLONE 24559 16721 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Pertuzumab PERTUZUMAB 24561 16722 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE AZD4547 24562 16723 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Canertinib CANERTINIB 16843263 24563 16724 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR US10022354, Example 151 24565 16725 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OXYMETAZOLINE OXYMETAZOLINE 24566 16726 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PLICAMYCIN PLICAMYCIN 22931300 24571 16727 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME activator 252166700 24572 16728 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR Selumetinib SELUMETINIB 26676756 24573 16729 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651031 SCOPOLAMINE 24574 16730 CYB5R3 1727 DRUGGABLE GENOME, ENZYME isosorbide mononitrate 24577 16731 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME GW843682X GW843682X 24578 16732 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DIETHYL-2-PENTADECYLIDENEMALONATE CHEMBL404916 21292492 24582 16733 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE ILORASERTIB ILORASERTIB 24583 16734 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GDC-0980 APITOLISIB 25673820,21998291 24584 16735 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE tenofovir TENOFOVIR 31619748,19400747,25485598,26535588,26807589,26287941,17083032 24585 16736 KDM4A 9682 DRUGGABLE GENOME, ENZYME CLOXYQUIN CLOXYQUIN 24586 16737 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE OT-730 24587 16738 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE BAPINEUZUMAB BAPINEUZUMAB 24589 16739 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Efalizumab EFALIZUMAB 24590 16740 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GSK2982772 24591 16741 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE RIBOCICLIB RIBOCICLIB 29408328 24593 16742 LRRC59 55379 NA MELAGATRAN MELAGATRAN 22494098 24594 16743 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CID 3241312 CHEMBL265715 24595 16744 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR Gerilimzumab 24596 16745 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR INK-1117 INK-1117 24597 16746 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE NIFLUMIC ACID 24599 16747 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OXATOMIDE OXATOMIDE 24600 16748 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor SOPHORETIN QUERCETIN 24601 16749 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CAPMATINIB CAPMATINIB 25971938,32877583 24602 16750 PDE3A 5139 ENZYME, DRUGGABLE GENOME RPL-554 24604 16751 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MRL20 24605 16752 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MORIN MORIN 24606 16753 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE ALK2 INHIBITOR LDN-193189 24705252 24608 16754 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Irinotecan IRINOTECAN 24609 16755 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLOBAZAM CLOBAZAM 24613 16756 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PF-00610355 PF-00610355 24614 16757 HTT 3064 DRUGGABLE GENOME ITF2357 GIVINOSTAT 24615 16758 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME corticosteroids 24307847 24616 16759 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PHENYLBUTANOIC ACID PHENYLBUTANOIC ACID 24044874 24617 16760 AMACR 23600 ENZYME cholic acid 24618 16761 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LANSOPRAZOLE LANSOPRAZOLE 24619 16762 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME irinotecan IRINOTECAN 28395759 24620 16763 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 trimethadione TRIMETHADIONE 9187528 24621 16764 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR TAMATINIB R-406 24622 16765 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRADIOL PROPIONATE ESTRADIOL PROPIONATE 24623 16766 ARSA 410 DRUGGABLE GENOME, ENZYME PIRENPERONE PIRENPERONE 24624 16767 TMEM97 27346 NA antagonist 178103294 24625 16768 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9187437, 24 24626 16769 GMNN 51053 DRUGGABLE GENOME FLUSPIRILENE FLUSPIRILENE 24627 16770 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME allosteric modulator 249565604 BINIMETINIB 24628 16771 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 223366208 BMS-690514 24630 16772 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BYL719 ALPELISIB 24631 16773 AKR1C3 8644 ENZYME, DRUGGABLE GENOME N-(naphthylamino)-benzoate derivative 1 24632 16774 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL772 RESERPINE 24633 16775 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL552212 LEXIBULIN 24634 16776 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417080 CHEMBL1498652 24635 16777 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201754 RUFINAMIDE 24636 16778 XDH 7498 DRUGGABLE GENOME, ENZYME ALLOPURINOL ALLOPURINOL 24638 16779 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BUTAMBEN BUTAMBEN 24639 16780 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR DIOTYROSINE DIOTYROSINE 24640 16781 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 1-NAPHTHYLISOTHIOCYANATE 1-NAPHTHYLISOTHIOCYANATE 24641 16782 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE IBRUTINIB IBRUTINIB 25222877 24643 16783 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL452 CLONAZEPAM 24644 16784 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 252166594 VS-5584 24646 16785 TUBB2A 7280 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 24647 16786 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 24649 16787 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE SUNITINIB SUNITINIB 24650 16788 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650507 24651 16789 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PLX-5622 PLX-5622 22294205 24653 16790 KDM4A 9682 DRUGGABLE GENOME, ENZYME SALICYLALDEHYDE THIOSEMICARBAZONE SALICYLALDEHYDE THIOSEMICARBAZONE 24654 16791 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Pyrimidine derivative 30 24656 16792 PTGS2 5743 DRUGGABLE GENOME, ENZYME SUPROFEN SUPROFEN 24657 16793 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 310264719 24658 16794 PDHX 8050 KINASE AUTOANTIGEN 8464876 24660 16795 UGCG 7357 ENZYME, DRUGGABLE GENOME ADRIAMYCIN ADRIAMYCIN 10702281 24661 16796 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2015042088Example4 24663 16797 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GW441756X GW441756X 24664 16798 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SULFAPHENAZOLE SULFAPHENAZOLE 22931300 24665 16799 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL1200567 DOXYCYCLINE HYCLATE 24666 16800 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE docetaxel DOCETAXEL 23963862 24667 16801 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-4516 CHEMBL586029 24669 16802 NGFR 4804 CELL SURFACE, DRUGGABLE GENOME Voclosporin VOCLOSPORIN 24670 16803 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MITOMYCIN MITOMYCIN 14514923 24671 16804 MAPT 4137 DRUGGABLE GENOME PTEROSTILBENE PTEROSTILBENE 24672 16805 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE AVX-470 24673 16806 ATP5F1E 514 TRANSPORTER certolizumab pegol 26307125 24675 16807 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME CANDESARTAN CILEXETIL 10029562 24677 16808 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME inhibitor 384403652 24678 16809 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 135651355 ZAPRINAST 24679 16810 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SUMATRIPTAN SUMATRIPTAN 24680 16811 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PRX-105 24682 16812 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TDR77135 CHEMBL1529479 24683 16813 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR BIOCHANIN BIOCHANIN 24684 16814 SIK3 23387 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 178102336 BOSUTINIB 24685 16815 GLS 2744 ENZYME 6-DIAZO-5-OXO-L-NORLEUCINE 6-DIAZO-5-OXO-L-NORLEUCINE 7867599 24687 16816 BAZ2B 29994 NA SJ000147784 CHEMBL590186 24688 16817 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PYRAZINAMIDE PYRAZINAMIDE 22931300 24689 16818 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SANGUINARIUM SANGUINARIUM 24690 16819 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-123598 CHEMBL547269 24691 16820 ATXN2 6311 NA GERONTOXANTHONE H GERONTOXANTHONE H 24692 16821 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-15 24693 16822 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor CHEMBL3039517 RABUSERTIB 24694 16823 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME FLUVOXAMINE FLUVOXAMINE 24696 16824 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135651127 24697 16825 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SOBUZOXANE SOBUZOXANE 24698 16826 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME MP-0112 ABICIPAR PEGOL 24700 16827 HDAC11 79885 DRUGGABLE GENOME, ENZYME RESMINOSTAT RESMINOSTAT 24701 16828 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE 24702 16829 BAZ2B 29994 NA TCMDC-125738 CHEMBL527585 24703 16830 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102306 FORETINIB 24704 16831 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE METAPHIT METHANESULFONATE METAPHIT METHANESULFONATE 24708 16832 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE agonist 178101033 24709 16833 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565645 MK-2461 24710 16834 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 135651433 ALLICIN 24712 16835 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE SULFINPYRAZONE SULFINPYRAZONE 24713 16836 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL2010872 CEP-11981 24715 16837 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE PROTHYMOSIN ALPHA 7798593 24716 16838 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE ISOBOLDINE ISOBOLDINE 24717 16839 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651511 24718 16840 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE INOSITOL INOSITOL 8063863 24719 16841 RACGAP1 29127 NA NSC-130813 CHEMBL463783 24720 16842 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565629 SOTRASTAURIN 24721 16843 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GSK-4112 GSK-4112 23656296 24725 16844 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME GUTHION GUTHION 24726 16845 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Olaparib OLAPARIB 24727 16846 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650520 BEXAROTENE 24728 16847 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUTAMIDE FLUTAMIDE 24730 16848 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker 135651438 ANANDAMIDE 24731 16849 NDUFB6 4712 ENZYME inhibitor CHEMBL3545320 ME-344 24733 16850 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 178102612 24734 16851 TNFRSF1A 7132 CELL SURFACE, DRUGGABLE GENOME 178101767 24735 16852 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL1946170 REGORAFENIB 24736 16853 RAB9A 9367 ENZYME, DRUGGABLE GENOME DROMETRIZOLE DROMETRIZOLE 24737 16854 SMAD2 4087 KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DEMETHOXYCURCUMIN DEMETHOXYCURCUMIN 23145932 24738 16855 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 310264675 CUDC-101 24740 16856 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-124381 CHEMBL579919 24742 16857 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor PD 0325901 24744 16858 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME DOXORUBICIN DOXORUBICIN 7927909 24747 16859 BAZ2B 29994 NA 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 24748 16860 USP1 7398 DNA REPAIR, PROTEASE, ENZYME LAPACHOL LAPACHOL 24749 16861 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR RAMIPRIL RAMIPRIL 15128880 24751 16862 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor SOPHORETIN QUERCETIN 24753 16863 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Tri-substituted urea derivative 2 24754 16864 SHMT1 6470 ENZYME bevacizumab BEVACIZUMAB 22044939 24756 16865 NOS1 4842 DRUGGABLE GENOME, ENZYME ACETAZOLAMIDE ACETAZOLAMIDE 11711216 24758 16866 PTGS1 5742 ENZYME, DRUGGABLE GENOME ACETYLSALICYLIC ACID 24762 16867 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME Roscovitine derivative 1 24763 16868 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PF-00477736 PF-00477736 22713237 24764 16869 POLI 11201 DNA REPAIR NSC-61836 CHEMBL521171 24765 16870 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR VATALANIB VATALANIB 24766 16871 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DOXYLAMINE DOXYLAMINE 24769 16872 USP1 7398 DNA REPAIR, PROTEASE, ENZYME BETA-LAPACHONE LAPACHONE 24771 16873 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SULINDAC SULINDAC 23434637 24772 16874 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 24774 16875 UGDH 7358 ENZYME ACETYLSALICYLIC ACID 8014943 24775 16876 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CLOFARABINE CLOFARABINE 24776 16877 SLC29A4 222962 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 135650270 FLUOXETINE 24778 16878 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 249565688 CHEMBL1765740 24779 16879 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000067611 CHEMBL602126 24780 16880 TYMP 1890 GROWTH FACTOR, DRUGGABLE GENOME capecitabine CAPECITABINE 24167597 24782 16881 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PREDNISONE PREDNISONE 22931300 24783 16882 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000111875 CHEMBL590949 24785 16883 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL BROMAZEPAM BROMAZEPAM 24786 16884 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antagonist CHEMBL1743064 ROBATUMUMAB 24788 16885 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE CISPLATIN CISPLATIN 12543810,11350408 24789 16886 SGSH 6448 DRUGGABLE GENOME, ENZYME HGT-1410 N-SULFOGLUCOSAMINE SULFOHYDROLASE RECOMBINANT 24790 16887 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE MK-2461 MK-2461 24791 16888 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ABX-0401 24792 16889 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DILTIAZEM DILTIAZEM 22931300,21393461 24793 16890 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME CT84.66 24796 16891 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 135649903 24797 16892 POLK 51426 DNA REPAIR, ENZYME EPINEPHRINE EPINEPHRINE 24798 16893 FNTA 2339 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL289228 TIPIFARNIB 24800 16894 CTSA 5476 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 223366200 TELAPREVIR 24802 16895 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CP-195543 CP-195543 24803 16896 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEPHALEXIN CEPHALEXIN 24804 16897 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE MGBG MITOGUAZONE 3528175 24805 16898 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GO-6976 GO-6976 24806 16899 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME VENETOCLAX VENETOCLAX 30725494 24807 16900 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565869 CEP-11981 24809 16901 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200517 DIHYDROERGOTAMINE MESYLATE 24810 16902 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AMG 900 24091768 24811 16903 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650397 N-METHYLHISTAMINE 24813 16904 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE EPO EPOETIN ALFA 8910323 24814 16905 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652267 24815 16906 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VORINOSTAT VORINOSTAT 24816 16907 CDC37 11140 KINASE SODIUM MOLYBDATE SODIUM MOLYBDATE 21486005 24817 16908 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 384403645 24818 16909 FST 10468 DRUGGABLE GENOME FREUNDS ADJUVANT 10734405 24820 16910 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125587 CHEMBL532160 24821 16911 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL575448 BMS-754807 24822 16912 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1201061 LEVALBUTEROL HYDROCHLORIDE 24823 16913 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER AMITRIPTYLINE HYDROCHLORIDE AMITRIPTYLINE HYDROCHLORIDE 24824 16914 DRAM1 55332 NA CISPLATIN CISPLATIN 15940259 24825 16915 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HER2-specific CAR T cell 24826 16916 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE fluorouracil FLUOROURACIL 24827 16917 ASS1 445 ENZYME, DRUG RESISTANCE CHLOROQUINE CHLOROQUINE 27735949 24829 16918 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME INSULIN DETEMIR 24830 16919 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ASCORBIC ACID 15050748 24832 16920 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Anti-CD20-CAR vector-transduced autologous T cells 24833 16921 GLS 2744 ENZYME PMID30273516-Compound-41 24834 16922 SERPINA6 866 DRUGGABLE GENOME, PROTEASE INHIBITOR I-vation 24836 16923 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 24838 16924 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 1225609 CHEMBL444376 24839 16925 MPHOSPH8 54737 NA CYSTAMINE DIHYDROCHLORIDE CYSTAMINE DIHYDROCHLORIDE 24840 16926 IGF1 3479 GROWTH FACTOR, HORMONE ACTIVITY, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE NNZ-2566 24841 16927 NDUFA4 4697 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545320 ME-344 24842 16928 MMP14 4323 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252827503 CGS-27023A 24843 16929 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CLEVIDIPINE CLEVIDIPINE 24845 16930 PTGS2 5743 DRUGGABLE GENOME, ENZYME HYDROXYCHLOROQUINE HYDROXYCHLOROQUINE 14963695 24847 16931 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SELUMETINIB SELUMETINIB 22425996 24848 16932 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR LY2606368 24851 16933 DYRK4 8798 ENZYME, KINASE, DRUGGABLE GENOME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 249565847 24852 16934 IL15RA 3601 DRUGGABLE GENOME, CELL SURFACE agonist 178101678 INTERLEUKIN 15, RECOMBINANT NON-GLYCOSYLATED 24853 16935 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE TALAZOPARIB TALAZOPARIB 28242752 24854 16936 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME LY-294002 LY-294002 17562705 24855 16937 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE Indazolyl-thiadiazolamine derivative 1 24857 16938 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US8975409, Example 13 24858 16939 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-1813 CHEMBL577662 24859 16940 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR LOBARIC ACID LOBARIC ACID 24861 16941 PRKAB1 5564 ENZYME, KINASE, DRUGGABLE GENOME SAPONARIN SAPONARIN 26471090 24862 16942 PADI2 11240 ENZYME STREPTONIGRIN STREPTONIGRIN 24440480 24864 16943 HTT 3064 DRUGGABLE GENOME TCMDC-125620 CHEMBL530291 24866 16944 COL18A1 80781 DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 16651433 24867 16945 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL428690 ALVOCIDIB 24868 16946 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Mirvetuximab soravtansine 24869 16947 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Methotrexate METHOTREXATE 24870 16948 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2326966 SF-1126 24872 16949 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DIOXYBENZONE DIOXYBENZONE 24873 16950 CBR1 873 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME fluorouracil FLUOROURACIL 24876 16951 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME TRASTUZUMAB TRASTUZUMAB 23204226 24877 16952 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE DOVITINIB DOVITINIB 24878 16953 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE (S)-DRF-1042 24883 16954 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NISOLDIPINE NISOLDIPINE 22931300 24884 16955 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Methanesulfonyl fluoride 24885 16956 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PF-05212384 GEDATOLISIB 24888 16957 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR pertuzumab PERTUZUMAB 24889 16958 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME TYROSINE KINASE INHIBITOR 15324351 24890 16959 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3348923 MLN-2480 24891 16960 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME BELACTOSIN A BELACTOSIN A 23547757 24892 16961 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CUDC-907 FIMEPINOSTAT 22693356 24894 16962 CXCL2 2920 DRUGGABLE GENOME CYCLOSPORIN A 7490125 24895 16963 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201557 INTERFERON ALFACON-1 24896 16964 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3545385 WX-037 24897 16965 VDAC2 7417 NA OLESOXIME OLESOXIME 24898 16966 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Trametinib TRAMETINIB 28783719,26036643,26582713,27312529 24899 16967 MAPT 4137 DRUGGABLE GENOME GNF-PF-3350 CHEMBL600747 24900 16968 IRS1 3667 KINASE, CLINICALLY ACTIONABLE DHEA PRASTERONE 15501480 24901 16969 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR QUINOLINIC ACID QUINOLINIC ACID 24902 16970 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DNDI1417195 CHEMBL1303948 24903 16971 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE INCB054828 PEMIGATINIB 24905 16972 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-1 24906 16973 GAA 2548 DRUGGABLE GENOME, ENZYME DOXAZOSIN MESYLATE DOXAZOSIN MESYLATE 24907 16974 MAPT 4137 DRUGGABLE GENOME SR-2640 SR-2640 24908 16975 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GUTHION GUTHION 24909 16976 TXK 7294 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 24911 16977 COMT 1312 DRUGGABLE GENOME, ENZYME inhibitor 178103260 ENTACAPONE 24912 16978 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 310264754 OMIPALISIB 24913 16979 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 178102045 24914 16980 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE COUMARIN-3-CARBOXYLIC ACID COUMARIN-3-CARBOXYLIC ACID 24915 16981 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FIIN-01 23175443,20338520 24916 16982 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 178102555 JNJ-7706621 24917 16983 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE NALOXONE METHIODIDE NALOXONE METHIODIDE 24919 16984 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DICLAZURIL DICLAZURIL 24921 16985 HLA-DRA 3122 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE PEMBROLIZUMAB PEMBROLIZUMAB 26822383 24922 16986 CLK1 1195 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor 249565842 24925 16987 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GNF-PF-3947 CHEMBL584508 24926 16988 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651129 24927 16989 KCNH8 131096 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL2107762 NERISPIRDINE 24930 16990 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME DAUNORUBICIN DAUNORUBICIN 22260166 24931 16991 MARCHF8 220972 ENZYME Live attenuated influenza vaccine 24932 16992 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyrrolo-pyrimidine derivative 11 24934 16993 MAPT 4137 DRUGGABLE GENOME PURPUROGALLIN PURPUROGALLIN 24935 16994 UGT2B15 7366 DRUGGABLE GENOME lorazepam LORAZEPAM 15961980 24936 16995 NOS1 4842 DRUGGABLE GENOME, ENZYME fluorouracil FLUOROURACIL 24937 16996 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TG100-115 TG100-115 17685602 24939 16997 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME KGP94 24940 16998 GMNN 51053 DRUGGABLE GENOME TCMDC-125185 CHEMBL580819 24941 16999 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX TRETINOIN TRETINOIN 24944 17000 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIAMCINOLONE TRIAMCINOLONE 24945 17001 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PSEUDOEPHEDRINE PSEUDOEPHEDRINE 24946 17002 PGP 283871 NA PACLITAXEL PACLITAXEL 24947 17003 BAZ2B 29994 NA 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 24949 17004 ATXN2 6311 NA GNF-PF-2272 CHEMBL601757 24950 17005 APBA1 320 NA GNF-PF-3464 CHEMBL602213 24952 17006 MAPT 4137 DRUGGABLE GENOME CAPSAZEPINE CAPSAZEPINE 24953 17007 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL1201748 CABAZITAXEL 24955 17008 POLB 5423 DNA REPAIR, DRUGGABLE GENOME 5,8,11,14-EICOSATETRAYNOIC ACID CHEMBL458328 24957 17009 TAC1 6863 DRUGGABLE GENOME SULINDAC SULINDAC 1707646 24958 17010 TMPRSS11D 9407 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166870 24959 17011 HTT 3064 DRUGGABLE GENOME ACRIFLAVINE CHLORIDE ACRIFLAVINE 24960 17012 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE antibody 178103957 CATUMAXOMAB 24961 17013 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BITHIONOLATE SODIUM BITHIONOLATE SODIUM 24962 17014 RAB9A 9367 ENZYME, DRUGGABLE GENOME LANSOPRAZOLE LANSOPRAZOLE 24964 17015 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 249565869 CEP-11981 24967 17016 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolo[3,2-c]pyridine derivative 1 24968 17017 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR CISPLATIN CISPLATIN 11163512,9772291,10810335,9703867 24970 17018 CD52 1043 DRUGGABLE GENOME CAMPATH ALEMTUZUMAB 8981930 24971 17019 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME inhibitor 249565699 CHEMBL322970 24973 17020 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 381118861 24975 17021 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL blocker 375973238 24977 17022 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME THAPSIGARGIN THAPSIGARGIN 24980 17023 CBR3 874 ENZYME, DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, CLINICALLY ACTIONABLE daunorubicin DAUNORUBICIN 20007405 24982 17024 RCE1 9986 ENZYME, PROTEASE, DRUGGABLE GENOME NSC-37136 CHEMBL1370674 24983 17025 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 381118905 24984 17026 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR HUMAN CHORIONIC GONADOTROPIN 15242988 24988 17027 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME OXYTETRACYCLINE OXYTETRACYCLINE 24989 17028 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME NICLOSAMIDE NICLOSAMIDE 24990 17029 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 178103299 TACRINE 24991 17030 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE OXALIPLATIN OXALIPLATIN 16187112 24992 17031 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME indacaterol INDACATEROL 24994 17032 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME HSP70 11133992 24995 17033 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 2-(PHENOXYMETHYL)BENZOTHIAZOLE 2-(PHENOXYMETHYL)BENZOTHIAZOLE 24998 17034 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3348923 MLN-2480 24999 17035 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL797 PHENSUXIMIDE 25000 17036 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME HEPARIN HEPARIN 25001 17037 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME NICLOSAMIDE NICLOSAMIDE 25002 17038 IFNGR1 3459 DRUGGABLE GENOME, CLINICALLY ACTIONABLE INTERFERON GAMMA-1B 25007 17039 ALOX15B 247 DRUGGABLE GENOME, ENZYME EMBELIN EMBELIN 25009 17040 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-638080 CHEMBL136344 25011 17041 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE THALIDOMIDE THALIDOMIDE 25013 17042 CA1 759 DRUGGABLE GENOME, ENZYME COUMATE 25014 17043 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FASUDIL FASUDIL 25016 17044 ALOX15B 247 DRUGGABLE GENOME, ENZYME LINOLENIC ACID LINOLENIC ACID 25018 17045 CBX1 10951 NA DIZOCILPINE DIZOCILPINE 25019 17046 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TRemelimumab + MEDI0562 25020 17047 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TAMOXIFEN CITRATE TAMOXIFEN CITRATE 25023 17048 MPHOSPH8 54737 NA AG-494 CHEMBL56731 25024 17049 PTGS2 5743 DRUGGABLE GENOME, ENZYME TENOXICAM TENOXICAM 25025 17050 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME DINACICLIB DINACICLIB 25026 17051 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME agonist CHEMBL3707402 PF-06372865 25027 17052 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SJ000029642 CHEMBL591126 25029 17053 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Obatoclax OBATOCLAX 22460902 25030 17054 ATAD5 79915 NA KENPAULLONE KENPAULLONE 25031 17055 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL ETOMIDATE ETOMIDATE 16884293,20704351 25032 17056 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ANTIMYCIN A ANTIMYCIN A 25033 17057 POLI 11201 DNA REPAIR NSC-107022 CHEMBL1601846 25034 17058 USP1 7398 DNA REPAIR, PROTEASE, ENZYME NSC-102742 CHEMBL1519374 25035 17059 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 387065580 25036 17060 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEFOTETAN CEFOTETAN 25040 17061 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME ALPELISIB ALPELISIB 28363909 25044 17062 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-20 25045 17063 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200802 TALBUTAL 25046 17064 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Ambenonium AMBENONIUM 25047 17065 KDM4A 9682 DRUGGABLE GENOME, ENZYME SALSOLINOL HYDROBROMIDE SALSOLINOL HYDROBROMIDE 25048 17066 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PROSTAGLANDIN B1 PROSTAGLANDIN B1 25049 17067 KDM4A 9682 DRUGGABLE GENOME, ENZYME TOLAZAMIDE TOLAZAMIDE 25050 17068 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE POLY I:C 15315972 25051 17069 FAP 2191 PROTEASE, CELL SURFACE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 252166764 25052 17070 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor PX-866 SONOLISIB 25053 17071 CYBB 1536 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME, ENZYME APIGENIN APIGENIN 23786520 25054 17072 KDM4A 9682 DRUGGABLE GENOME, ENZYME CLOSANTEL CLOSANTEL 25055 17073 CXCL8 3576 DRUGGABLE GENOME TOCOPHEROL ACETATE 15150308 25056 17074 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZOMEPIRAC SODIUM ZOMEPIRAC SODIUM 25057 17075 BCHE 590 DRUGGABLE GENOME, ENZYME PMID29757691-Compound-8d 25058 17076 DNER 92737 NA Quinazolinone derivative 3 25059 17077 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor HESPERADIN HESPERADIN 19035792 25060 17078 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE STREPTOZOTOCIN STREPTOZOCIN 15616011 25063 17079 ATAD5 79915 NA DNDI1417701 CHEMBL1326164 25066 17080 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIPHENADIONE DIPHENADIONE 25067 17081 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE TAE-684 TAE-684 25068 17082 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200395 ORPHENADRINE CITRATE 25069 17083 CPT2 1376 DRUGGABLE GENOME PERHEXILINE PERHEXILINE 25072 17084 CSRNP3 80034 NA Bisphosphonates 25076 17085 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR AR-42 AR-42 25077 17086 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE ETHYLNITROSOUREA 9330624 25078 17087 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 178100448 25079 17088 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ABY-025 25080 17089 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PALBOCICLIB PALBOCICLIB 25082 17090 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 381744922 SC-560 25084 17091 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200898 25085 17092 PTGS1 5742 ENZYME, DRUGGABLE GENOME SULINDAC SULINDAC 25087 17093 BRCA2 675 CLINICALLY ACTIONABLE VX-970 BERZOSERTIB 25089 17094 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrrolo-pyridone derivative 3 25090 17095 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL haloperidol HALOPERIDOL 27023437 25094 17096 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE CYC-116 CYC-116 25095 17097 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor HTS-466284 CHEMBL261454 19035792 25096 17098 TARDBP 23435 TUMOR SUPPRESSOR 2-(2'-METHOXYPHENYL)-1H-INDOLE 2-(2'-METHOXYPHENYL)-1H-INDOLE 25098 17099 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL108 CARBAMAZEPINE 25099 17100 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20100022547C83 25100 17101 HMGCR 3156 ENZYME, DRUGGABLE GENOME LOVASTATIN LOVASTATIN 25101 17102 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE JUGLONE JUGLONE 25102 17103 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor CHEMBL300138 ENZASTAURIN 25104 17104 IMPDH2 3615 DRUGGABLE GENOME, ENZYME Urea and carbamate bioisostere derivative 1 25106 17105 DMD 1756 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Golodirsen GOLODIRSEN 25108 17106 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 249565922 25111 17107 GSTM1 2944 DRUGGABLE GENOME, ENZYME DICUMAROL DICUMAROL 15044619 25112 17108 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE OXALIPLATIN OXALIPLATIN 10098743 25113 17109 BRCA2 675 CLINICALLY ACTIONABLE TALAZOPARIB TALAZOPARIB 28242752 25114 17110 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 385612186 25116 17111 TGFBR2 7048 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME TGF-BR2 mab 25117 17112 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE inhibitor 223366028 AZD-4017 25118 17113 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 25121 17114 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE EUPALININ A EUPALININ A 17980607 25123 17115 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE 7,3',4'-TRIMETHOXYISOFLAVONE CHEMBL273891 25126 17116 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL3707225 GSK2798745 25127 17117 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor CHEMBL220492 TOPIRAMATE 25130 17118 COL27A1 85301 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 25132 17119 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME VANDETANIB VANDETANIB 25134 17120 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME SEN-196 25135 17121 UGT2B15 7366 DRUGGABLE GENOME sipoglitazar SIPOGLITAZAR 22960998,23444281 25138 17122 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 178102533 25139 17123 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor SF1126 25140 17124 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE CATUMAXOMAB CATUMAXOMAB 25142 17125 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME SELENIUM 2035236 25143 17126 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3039525 GOLVATINIB 25144 17127 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-61 25145 17128 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL1852688 INFIGRATINIB 25146 17129 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME PF-562271 PF-00562271 25147 17130 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR OXYTETRACYCLINE OXYTETRACYCLINE 25148 17131 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEXAMETHASONE DEXAMETHASONE 15870285 25149 17132 RPS6KA4 8986 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, ENZYME inhibitor 252827421 25150 17133 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Gemcitabine GEMCITABINE 25151 17134 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUACIZINE FLUACIZINE 25152 17135 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE Cerulenin CERULENIN 25154 17136 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker 178100950 AMANTADINE 25157 17137 SMN1 6606 DRUGGABLE GENOME PIFITHRIN-ALPHA CHEMBL198759 25160 17138 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-52 25161 17139 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE alprazolam ALPRAZOLAM 18695978 25162 17140 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LECANORIC ACID LECANORIC ACID 25163 17141 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 25167 17142 IGFBP1 3484 DRUGGABLE GENOME ETHANOL ALCOHOL 11894976 25169 17143 CA9 768 DRUGGABLE GENOME, ENZYME celecoxib CELECOXIB 22336956 25170 17144 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MERCAPTOPURINE MERCAPTOPURINE 25171 17145 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME (RS)-ROSCOVITINE (RS)-ROSCOVITINE 25172 17146 HSPB2 3316 KINASE ANTINEOPLASTIC 11174852 25175 17147 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650064 CETIRIZINE 25176 17148 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ibrutinib IBRUTINIB 25178 17149 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE (R)-DIHYDRONIPHATENONE B CHEMBL1946449 22148427 25179 17150 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1689 TOLAZOLINE HYDROCHLORIDE 25180 17151 GALNT18 374378 NA tocilizumab TOCILIZUMAB 27339827 25181 17152 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Nandrolone NANDROLONE 25182 17153 RGS4 5999 DRUGGABLE GENOME BRIMONIDINE BRIMONIDINE 25184 17154 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME CNS-5161 CNS-5161 25185 17155 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL venlafaxine VENLAFAXINE 23394390 25186 17156 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PACLITAXEL PACLITAXEL 15657900 25187 17157 COMT 1312 DRUGGABLE GENOME, ENZYME CGP-28014 25188 17158 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102615 25190 17159 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE hydrocodone HYDROCODONE 18695978 25191 17160 MAP3K9 4293 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565786 25192 17161 NOS1 4842 DRUGGABLE GENOME, ENZYME GREEN TEA EXTRACT 15820752 25193 17162 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE HER2 INHIBITOR CP-724,714 24685132 25195 17163 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545285 XL-999 25196 17164 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652307 25197 17165 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Ro 31-7453 25198 17166 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 381744922 SC-560 25200 17167 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME EMEDASTINE EMEDASTINE 25201 17168 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 252827462 RITONAVIR 25202 17169 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3-AMINOBENZAMIDE 3-AMINOBENZAMIDE 25203 17170 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor AS703569 CENISERTIB 25204 17171 BCHE 590 DRUGGABLE GENOME, ENZYME DEMECARIUM BROMIDE 25205 17172 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE INSM-18 INSM-18 25206 17173 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Alpelisib ALPELISIB 27659046 25207 17174 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A6 25211 17175 SLC15A2 6565 TRANSPORTER, DRUGGABLE GENOME 178101319 25212 17176 MAP2K6 5608 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE, TUMOR SUPPRESSOR inhibitor GDC-0973 COBIMETINIB 25213 17177 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME E324 E324 25214 17178 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 25216 17179 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 25217 17180 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE BAY-613606 CHEMBL541400 25218 17181 GLO1 2739 ENZYME, DRUGGABLE GENOME N-METHYLFORMAMIDE 3480403 25219 17182 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2010127754 25221 17183 ALOX15B 247 DRUGGABLE GENOME, ENZYME HYPERICIN HYPERICIN 25223 17184 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CAPTAN CAPTAN 25224 17185 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL285674 ESTAZOLAM 25229 17186 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME BAS03450373 CHEMBL1576310 25230 17187 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE LUTEOLIN LUTEOLIN 21265555 25231 17188 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME SJ000071854 CHEMBL602127 25232 17189 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE TAMATINIB R-406 25234 17190 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR P1446A-05 VORUCICLIB 25236 17191 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE DX-2802 25237 17192 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL2108677 PEGINTERFERON BETA-1A 25238 17193 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME Selective BACE 1 inhibitor 25241 17194 KDM4A 9682 DRUGGABLE GENOME, ENZYME TDR78109 CHEMBL1304363 25242 17195 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL3545017 GTX-758 25243 17196 KCNC3 3748 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 25244 17197 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TAMOXIFEN TAMOXIFEN 22931300 25245 17198 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE LY3015014 FROVOCIMAB 25246 17199 PSMC4 5704 NA inhibitor CHEMBL2103884 OPROZOMIB 25247 17200 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL1908376 SEOCALCITOL 25248 17201 GMNN 51053 DRUGGABLE GENOME EMETINE HYDROCHLORIDE EMETINE HYDROCHLORIDE 25249 17202 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650554 EGLUMEGAD 25251 17203 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL ADINAZOLAM ADINAZOLAM 25253 17204 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 249565861 25254 17205 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR antagonist GDC0917 25255 17206 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR KF-17837 CHEMBL27508 25257 17207 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR AR-42 AR-42 25258 17208 FABP1 2168 DRUGGABLE GENOME fenofibrate FENOFIBRATE 15249972 25259 17209 HTT 3064 DRUGGABLE GENOME THIOMERSAL THIMEROSAL 25261 17210 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Cisplatin CISPLATIN 27040853 25262 17211 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME MVA-BN 25264 17212 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor GDC-0941 PICTILISIB 25265 17213 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1088752 LOSMAPIMOD 25266 17214 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 328083454 HARMINE 25267 17215 DNER 92737 NA Isoxazole-based bicyclic compound 15 25268 17216 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 25269 17217 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AM580 CHEMBL69367 25270 17218 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME CARFILZOMIB CARFILZOMIB 25271 17219 POLK 51426 DNA REPAIR, ENZYME CIMETIDINE CIMETIDINE 25272 17220 ALOX15B 247 DRUGGABLE GENOME, ENZYME SANGUINARINE SULFATE SANGUINARINE SULFATE 25273 17221 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Farletuzumab FARLETUZUMAB 25274 17222 MAPT 4137 DRUGGABLE GENOME QUINALIZARIN QUINALIZARIN 25275 17223 MAOB 4129 DRUGGABLE GENOME, ENZYME Tetra-hydro-oxazolopyridine derivative 1 25277 17224 SREBF1 6720 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR hmg coa reductase inhibitors 24329191 25279 17225 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE IDH305 25282 17226 TXNRD1 7296 DRUGGABLE GENOME 4-aryl quinol derivative 3 25283 17227 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RIMEXOLONE RIMEXOLONE 25284 17228 GMNN 51053 DRUGGABLE GENOME LOFEPRAMINE LOFEPRAMINE 25285 17229 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ZSTK474 25286 17230 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-2A, RECOMBINANT 25287 17231 CA1 759 DRUGGABLE GENOME, ENZYME ETHOXZOLAMIDE ETHOXZOLAMIDE 25288 17232 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL MENTHOL MENTHOL 25289 17233 RAB9A 9367 ENZYME, DRUGGABLE GENOME INDOPROFEN INDOPROFEN 25290 17234 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE TRANSFORMING GROWTH FACTOR 9403612 25292 17235 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TYRPHOSTIN AG 879 15526167 25293 17236 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 178100444 25294 17237 ITGB5 3693 CELL SURFACE, DRUGGABLE GENOME inhibitor CILENGITIDE CILENGITIDE 25295 17238 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME BI 2536 25296 17239 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE TAXANE COMPOUND 21920589 25299 17240 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME QUERCETIN QUERCETIN 1478066 25302 17241 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME SILYDIANIN SILYDIANIN 23401473 25303 17242 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LE-SN38 25304 17243 SMN2 6607 DRUGGABLE GENOME GNF-PF-516 CHEMBL602970 25305 17244 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CSA CYCLOSPORINE 10609555 25306 17245 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME EQUINE CHORIONIC GONADOTROPIN 16885537 25307 17246 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DIENESTROL DIENESTROL 25308 17247 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 252166781 MAVORIXAFOR 25309 17248 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135651219 SURAMIN 25310 17249 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL568 OXAZEPAM 25311 17250 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-50 25312 17251 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ARRY-380 TUCATINIB 25313 17252 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR VALPROIC ACID VALPROIC ACID 18294844,16921367,25304896 25315 17253 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE epirubicin EPIRUBICIN 25316 17254 ERAP1 51752 PROTEASE, ENZYME, DRUGGABLE GENOME UMBELLIFERONE UMBELLIFERONE 25319 17255 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR irbesartan IRBESARTAN 11593098,15614026,14700505 25320 17256 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 387065600 25321 17257 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR U-50488 METHANE SULFONATE U-50488 METHANE SULFONATE 25323 17258 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650680 NALBUPHINE 25324 17259 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000002502 CHEMBL591630 25325 17260 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE NYSTATIN NYSTATIN 11593015 25326 17261 ABAT 18 DRUGGABLE GENOME, ENZYME CPP -15 25329 17262 POLI 11201 DNA REPAIR METHACYCLINE HYDROCHLORIDE METHACYCLINE HYDROCHLORIDE 25330 17263 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-61 25331 17264 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE ETOPOSIDE ETOPOSIDE 22364746 25332 17265 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 53801033 25333 17266 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE METHYLNALTREXONE BROMIDE 25334 17267 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR etoposide ETOPOSIDE 25336 17268 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MONTELUKAST MONTELUKAST 22931300 25337 17269 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE DOVITINIB DOVITINIB 25339 17270 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHENACYL CHLORIDE PHENACYL CHLORIDE 25340 17271 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 178102312 25341 17272 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME Anti-mesothelin CAR T Cells 25342 17273 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20120264760C83 25343 17274 APC 324 CLINICALLY ACTIONABLE TRIIODOTHYRONINE LIOTHYRONINE SODIUM 12856637 25345 17275 TUBB 203068 DRUGGABLE GENOME inhibitor 135650118 COLCHICINE 25346 17276 VKORC1L1 154807 DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 25347 17277 FZD7 8324 G PROTEIN COUPLED RECEPTOR, KINASE OMP-18R5 VANTICTUMAB 25348 17278 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE inhibitor 178101880 25351 17279 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL781 MAZINDOL 25352 17280 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 178103387 TOSITUMOMAB 25353 17281 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE MNU 16616109 25354 17282 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 178102535 25355 17283 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL969 PRAZEPAM 25356 17284 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER maprotiline MAPROTILINE 25357 17285 GATA2 2624 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX BORTEZOMIB BORTEZOMIB 22541434 25359 17286 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Dovitinib DOVITINIB 22238366,23658459,27315356,17698633 25360 17287 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR RETINOID 15020266 25361 17288 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PDC-41 25362 17289 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYDROXYPROGESTERONE CAPROATE HYDROXYPROGESTERONE CAPROATE 25363 17290 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417601 CHEMBL1503729 25364 17291 PSMC4 5704 NA inhibitor BORTEZOMIB BORTEZOMIB 25365 17292 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NORDEFRIN NORDEFRIN 25366 17293 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor PKI-587 GEDATOLISIB 25368 17294 HTT 3064 DRUGGABLE GENOME TRICLOCARBAN TRICLOCARBAN 25369 17295 FAAH 2166 ENZYME, DRUGGABLE GENOME Tetra-hydro-naphthyridine derivative 1 25370 17296 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME LINIFANIB LINIFANIB 25371 17297 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME gemcitabine GEMCITABINE 25374 17298 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIMETHYLPHENYLPIPERAZINIUM IODIDE DIMETHYLPHENYLPIPERAZINIUM IODIDE 25376 17299 EED 8726 ENZYME, CLINICALLY ACTIONABLE ASTEMIZOLE ASTEMIZOLE 25369470 25377 17300 MAPT 4137 DRUGGABLE GENOME ARACHIDONIC ACID ARACHIDONIC ACID 25378 17301 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL1687 TUBOCURARINE CHLORIDE 25381 17302 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SURAMIN SURAMIN 25382 17303 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR UNC1999 27135738 25383 17304 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135650431 ISOPROTERENOL 25385 17305 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AZD-1080 AZD-1080 25386 17306 NCAM1 4684 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CHEMBL1743037 LORVOTUZUMAB MERTANSINE 25390 17307 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE NSC-95397 CHEMBL429095 25392 17308 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR inhibitor CHEMBL325424 ALEPLASININ 25393 17309 PSENEN 55851 DRUGGABLE GENOME inhibitor MK0752 25394 17310 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1200541 AMBENONIUM CHLORIDE 25399 17311 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-56 25400 17312 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HER2 CAR-T cells 28426845,28710747,25800760,28284008 25401 17313 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL237500 LINAGLIPTIN 25402 17314 BCL6 604 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE inhibitor 348353630 25403 17315 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME valproic acid 23407051 25404 17316 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE Crizotinib CRIZOTINIB 28476735 25405 17317 KEAP1 9817 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING 135650061 BARDOXOLONE 25406 17318 TP53AIP1 63970 NA epirubicin EPIRUBICIN 25407 17319 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR SIGNAL TRANSDUCTION INHIBITORS 16926049 25408 17320 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-3 25409 17321 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Benzodihydroisofuran derivative 3 25410 17322 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 363894144 GW-406381 25411 17323 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY 5-AZACYTIDINE AZACITIDINE 2476239 25412 17324 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TOPOTECAN HYDROCHLORIDE TOPOTECAN HYDROCHLORIDE 25413 17325 NOX4 50507 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 363894226 25417 17326 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME antagonist BIRINAPANT BIRINAPANT 25419 17327 IGFBP4 3487 DRUGGABLE GENOME PMSG 9258879 25420 17328 COL3A1 1281 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 25421 17329 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 178102936 LINAGLIPTIN 25423 17330 PRKAA2 5563 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME METFORMIN METFORMIN 26471090 25424 17331 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CRYPTOTANSHINONE CRYPTOTANSHINONE 25425 17332 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME TCMDC-125385 CHEMBL586628 25426 17333 PRKCH 5583 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE BRYOSTATIN BRYOSTATIN 25427 17334 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 POMIFERIN POMIFERIN 25431 17335 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE LORGLUMIDE SODIUM LORGLUMIDE SODIUM 25434 17336 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL1200549 RAPACURONIUM BROMIDE 25435 17337 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamide derivative 25 25436 17338 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 25437 17339 CPN1 1369 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252166856 25438 17340 POLI 11201 DNA REPAIR TCMDC-123912 CHEMBL106525 25440 17341 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9187437, 38 25441 17342 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3545276 CP-778875 25443 17343 ATXN2 6311 NA CLOFOCTOL CLOFOCTOL 25445 17344 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GSK2830371 25658463 25446 17345 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE MTX METHOTREXATE 12972956 25447 17346 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200447 25448 17347 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417072 CHEMBL1310701 25449 17348 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BEXAROTENE BEXAROTENE 25450 17349 EYA2 2139 DNA REPAIR MORIN MORIN 25452 17350 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE ANDROGRAPHOLIDE ANDROGRAPHOLIDE 22026410 25453 17351 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 brivaracetam BRIVARACETAM 25454 17352 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PMID28048944-Compound-4 25455 17353 PAK2 5062 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565812 25456 17354 RAB27A 5873 ENZYME inhibitor 328083519 25458 17355 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE CISPLATIN CISPLATIN 16982732 25461 17356 MAOA 4128 DRUGGABLE GENOME, ENZYME TRYPTAMINE TRYPTAMINE 25462 17357 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE LOVASTATIN LOVASTATIN 25463 17358 MAPT 4137 DRUGGABLE GENOME 2,6-DIMETHOXYQUINONE 2,6-DIMETHOXYQUINONE 25464 17359 SCNN1A 6337 DRUGGABLE GENOME, ION CHANNEL GS-9411 25465 17360 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY MORPHINE MORPHINE 6993188 25466 17361 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 5-METHOXY DMT OXALATE CHEMBL1256920 25467 17362 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME PHENOBARBITAL PHENOBARBITAL 14977870 25469 17363 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR VITAMIN K 12053098 25470 17364 IFNG 3458 DRUGGABLE GENOME CISPLATIN CISPLATIN 8044830 25475 17365 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR ISOFLAVONES 15195125 25476 17366 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME BMS-387032 BMS-387032 25478 17367 HSPA4 3308 NA AG-707 25479 17368 BAZ2B 29994 NA SJ000029642 CHEMBL591126 25480 17369 PTGIS 5740 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME PHENYLBUTAZONE PHENYLBUTAZONE 25481 17370 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ethosuximide ETHOSUXIMIDE 9187528 25482 17371 HTT 3064 DRUGGABLE GENOME DITHIAZANINE IODIDE DITHIAZANINE IODIDE 25484 17372 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PURPUROGALLIN PURPUROGALLIN 25487 17373 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3716 CHEMBL609606 25488 17374 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE RALOXIFENE RALOXIFENE 11901050 25489 17375 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Piperidine derivative 4 25491 17376 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL3545349 EVT-101 25492 17377 PTGS1 5742 ENZYME, DRUGGABLE GENOME aspirin ASPIRIN 20938371,16493486,22940005 25493 17378 TUBA1C 84790 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 25495 17379 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL1207366 GW468816 25496 17380 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 348353656 SOLCITINIB 25498 17381 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR CHLORAMPHENICOL CHLORAMPHENICOL 9931456 25499 17382 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Indazole derivative 3 25500 17383 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MECYSTEINE HYDROCHLORIDE MECYSTEINE HYDROCHLORIDE 25501 17384 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ROSE BENGAL ROSE BENGAL 25502 17385 POLI 11201 DNA REPAIR GNF-PF-3145 CHEMBL579761 25504 17386 SLC12A5 57468 DRUGGABLE GENOME, TRANSPORTER BUMETANIDE BUMETANIDE 25505 17387 MAP2K3 5606 KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE inhibitor MEK162 BINIMETINIB 25506 17388 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLONIDINE CLONIDINE 25511 17389 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135650279 FLUVASTATIN 25512 17390 GMNN 51053 DRUGGABLE GENOME SJ000119988 CHEMBL589694 25515 17391 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME TAMOXIFEN TAMOXIFEN 7532467 25516 17392 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE SIROLIMUS SIROLIMUS 15647370 25517 17393 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME JNJ-7706621 JNJ-7706621 25518 17394 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TRAFERMIN TRAFERMIN 25519 17395 HBB 3043 DRUGGABLE GENOME, ENZYME CAMPTOTHECIN CAMPTOTHECIN 25520 17396 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR ALPHA-TOCOPHEROL VITAMIN E 15271854 25521 17397 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE HGS-TR2J 25524 17398 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CLOTIAZEPAM CLOTIAZEPAM 25525 17399 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME SB-220025 SB-220025 25526 17400 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GW7074 CHEMBL72365 25527 17401 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 25528 17402 TUBA4A 7277 DRUGGABLE GENOME CHEMBL2105643 FOSBRETABULIN TROMETHAMINE 25529 17403 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE CH-5132799 PA-799 25530 17404 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Platinum compounds 23510626 25531 17405 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650836 25535 17406 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HARMOL HYDROCHLORIDE HARMOL HYDROCHLORIDE 25537 17407 PSMB10 5699 PROTEASE, DRUGGABLE GENOME inhibitor CARFILZOMIB CARFILZOMIB 25538 17408 PTGS2 5743 DRUGGABLE GENOME, ENZYME ACETYLSALICYLIC ACID 25539 17409 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-30 25540 17410 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME fluorouracil FLUOROURACIL 16875718 25541 17411 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE 178101574 25542 17412 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TETRANITROMETHANE TETRANITROMETHANE 25545 17413 MSMB 4477 DRUGGABLE GENOME, CLINICALLY ACTIONABLE Tigapotide TIGAPOTIDE 25546 17414 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME NAVEGLITAZAR NAVEGLITAZAR 25547 17415 TUBB6 84617 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 25549 17416 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL605 PROCAINAMIDE HYDROCHLORIDE 25550 17417 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor SUNITINIB SUNITINIB 25551 17418 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME PSAMMAPLIN A PSAMMAPLIN A 21215647 25554 17419 NOS2 4843 DRUGGABLE GENOME, ENZYME LT-1951 25555 17420 PDE4A 5141 DRUGGABLE GENOME, ENZYME Arofylline AROFYLLINE 25557 17421 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LANSOPRAZOLE SULFIDE LANSOPRAZOLE SULFIDE 25560 17422 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor MLN 8237 ALISERTIB 25561 17423 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME STAUROSPORINE STAUROSPORINE 17255535 25564 17424 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 6ALPHA-METHYLPREDNISOLONE ACETATE METHYLPREDNISOLONE ACETATE 25565 17425 RPS2 6187 NA FGF3 16263090 25566 17426 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MEK162 BINIMETINIB 24569456 25568 17427 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 315661187 CHEMBL119054 25570 17428 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TYRPHOSTIN 23 TYRPHOSTIN 23 25572 17429 NAAA 27163 ENZYME, DRUGGABLE GENOME inhibitor 381118831 25573 17430 CDC42 998 DRUGGABLE GENOME SECRAMINE A SECRAMINE A 16408091 25574 17431 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650704 25575 17432 IL11 3589 DRUGGABLE GENOME, KINASE, GROWTH FACTOR BFGF 12063288 25577 17433 HTT 3064 DRUGGABLE GENOME IPRIFLAVONE IPRIFLAVONE 25579 17434 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SAQUINAVIR MESYLATE SAQUINAVIR MESYLATE 25580 17435 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BENZYLACETONE BENZYLACETONE 25581 17436 KCNJ3 3760 EXTERNAL SIDE OF PLASMA MEMBRANE, ION CHANNEL, DRUGGABLE GENOME blocker 223366037 25582 17437 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DODECYL GALLATE DODECYL GALLATE 25583 17438 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178101914 NAPROXEN 25584 17439 CXCL8 3576 DRUGGABLE GENOME RECOMBINANT HUMAN IL-4 11228246 25585 17440 ATXN2 6311 NA SJ000113107 CHEMBL589245 25586 17441 TUBB 203068 DRUGGABLE GENOME Liposomal encapsulated paclitaxel (LEP) 25587 17442 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652196 ICATIBANT 25588 17443 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR INDOMETHACIN INDOMETHACIN 9357777 25590 17444 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545133 JNJ-26483327 25592 17445 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Copanlisib COPANLISIB 24170767 25593 17446 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR 3R14S-OCHRATOXIN A 3R14S-OCHRATOXIN A 25594 17447 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR ARRY-797 ARRY-797 25600 17448 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL1614 DESLANOSIDE 25601 17449 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME PD-404182 CHEMBL595227 25602 17450 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LIRANAFTATE LIRANAFTATE 25603 17451 UBE2T 29089 ENZYME, DNA REPAIR, CLINICALLY ACTIONABLE MK-2206 MK-2206 25604 17452 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME DACTINOMYCIN DACTINOMYCIN 25606 17453 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DIPHENADIONE DIPHENADIONE 25608 17454 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER Reserpine RESERPINE 25610 17455 SPP1 6696 DRUGGABLE GENOME CHONDROITIN SULFATE 12118914 25613 17456 SGK1 6446 SERINE THREONINE KINASE, KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 405067332 25616 17457 BAZ2B 29994 NA CLOSANTEL CLOSANTEL 25617 17458 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-4803 CHEMBL585240 25618 17459 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR ISORHAMNETIN ISORHAMNETIN 25190466 25619 17460 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 23622981 25621 17461 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER valganciclovir VALGANCICLOVIR 27402191 25622 17462 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR HMN-214 HMN-214 25156567 25623 17463 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor 315661148 ENOXIMONE 25624 17464 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME 681640 CHEMBL379975 25626 17465 TARDBP 23435 TUMOR SUPPRESSOR ADENINE ADENINE 25629 17466 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135651327 25630 17467 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE SPC/ENZ2968 25631 17468 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR CYPROTERONE ACETATE CYPROTERONE ACETATE 25632 17469 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SAR-156597 ROMILKIMAB 25633 17470 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor AZD5363 CAPIVASERTIB 25638 17471 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR URSOLIC ACID URSOLIC ACID 19716700 25639 17472 NFKBIB 4793 TRANSCRIPTION FACTOR, KINASE gefitinib GEFITINIB 31664190 25640 17473 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 363894206 ALLITINIB 25641 17474 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE TCMDC-125758 CHEMBL546797 25644 17475 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE F200 25647 17476 MAPT 4137 DRUGGABLE GENOME HTS-05056 CHEMBL196814 25649 17477 PTGS1 5742 ENZYME, DRUGGABLE GENOME IBUPROFEN IBUPROFEN 23651359 25653 17478 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME NSC-95397 CHEMBL429095 25654 17479 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-27 25655 17480 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 2-BENZOYL-5-METHOXYBENZOQUINONE 2-BENZOYL-5-METHOXYBENZOQUINONE 25656 17481 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME hmg coa reductase inhibitors 25657 17482 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Benzodihydroisofuran derivative 4 25658 17483 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1879463 DACTOLISIB 25659 17484 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME KENPAULLONE KENPAULLONE 25662 17485 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MGCD516 SITRAVATINIB 25663 17486 SLC7A11 23657 TRANSPORTER, DRUGGABLE GENOME, CELL SURFACE RILUZOLE RILUZOLE 25664 17487 GSTM1 2944 DRUGGABLE GENOME, ENZYME TROGLITAZONE TROGLITAZONE 12732844 25665 17488 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PONATINIB PONATINIB 22238366,26574622,24550739 25666 17489 SMARCB1 6598 CLINICALLY ACTIONABLE Tazemetostat TAZEMETOSTAT 25667 17490 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE codeine CODEINE 25752520 25668 17491 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GW441756X GW441756X 25669 17492 WIF1 11197 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE Platinum compounds 24980784 25671 17493 HSPB1 3315 DRUGGABLE GENOME 4,6-DICHLORORESORCINOL CHEMBL2332783 25672 17494 DGAT1 8694 ENZYME, DRUGGABLE GENOME Lactam derivative 1 25673 17495 PSMD12 5718 NA CARFILZOMIB CARFILZOMIB 24524217 25674 17496 FBXW7 55294 DNA REPAIR, CLINICALLY ACTIONABLE Vorinostat VORINOSTAT 23274910 25677 17497 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CKD602 25678 17498 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650814 ALPROSTADIL 25680 17499 POLK 51426 DNA REPAIR, ENZYME PENTAMIDINE ISETHIONATE PENTAMIDINE ISETHIONATE 25682 17500 SRP19 6728 NA fluoxetine FLUOXETINE 22795047 25686 17501 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1120 BISMUTH SUBSALICYLATE 25688 17502 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME 1207456-01-6 25690 17503 H2AW 92815 NA ANTISERUM 11006266 25691 17504 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME JNJ-7706621 JNJ-7706621 25693 17505 MGLL 11343 DRUGGABLE GENOME, ENZYME Piperazine carbamic compound 5 25695 17506 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE CHEMBL2108029 ERTUMAXOMAB 25696 17507 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650350 HIMBACINE 25697 17508 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TCMDC-125518 CHEMBL587772 25698 17509 COQ8B 79934 KINASE, DRUGGABLE GENOME, ENZYME, TRANSPORTER Immunoglobulins 21987091 25699 17510 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME escitalopram ESCITALOPRAM 25701 17511 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AR-42 AR-42 25702 17512 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32i 25706 17513 ALOX15 246 ENZYME, DRUGGABLE GENOME AG-537 CHEMBL67535 25710 17514 DNER 92737 NA Isoxazole-based bicyclic compound 17 25715 17515 F11 2160 DRUGGABLE GENOME, PROTEASE, ENZYME hormonal contraceptives for systemic use 28750087 25716 17516 PAEP 5047 DRUGGABLE GENOME CYPROTERONE ACETATE 1388220 25717 17517 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1405 ESTRONE 25718 17518 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME OXAZEPAM OXAZEPAM 25719 17519 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL PICROTOXIN PICROTOXIN 25721 17520 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME RETUSIN RETUSIN 23851114 25722 17521 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1236962 OMIPALISIB 25723 17522 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Diphenhydramine DIPHENHYDRAMINE 25725 17523 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ISONIPECOTIC ACID ISONIPECOTIC ACID 25038482 25726 17524 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME THIOMERSAL THIMEROSAL 25728 17525 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Talazoparib TALAZOPARIB 28148839 25729 17526 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME mycophenolic acid 25163792 25732 17527 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PF-562271 PF-00562271 25733 17528 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3833344 GANCOTAMAB 25734 17529 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METILDIGOXIN METILDIGOXIN 25735 17530 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2010077680 481 25736 17531 ABAT 18 DRUGGABLE GENOME, ENZYME 4-hydroxybenzaldehyde 4-HYDROXYBENZALDEHYDE 25737 17532 GAA 2548 DRUGGABLE GENOME, ENZYME 5-HYDROXYINDOLE CHEMBL404923 25738 17533 HSPA4 3308 NA PUROMYCIN PUROMYCIN 3170555,3664499,1986403 25739 17534 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE PODOFILOX PODOFILOX 25741 17535 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 25742 17536 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565909 25743 17537 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CADMIUM DICHLORIDE CADMIUM DICHLORIDE 25745 17538 PSMD4 5710 NA inhibitor CARFILZOMIB CARFILZOMIB 25746 17539 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL METHARBITAL METHARBITAL 25748 17540 RCE1 9986 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252166757 25749 17541 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METHYLERGONOVINE METHYLERGONOVINE 25751 17542 RAB9A 9367 ENZYME, DRUGGABLE GENOME 3-(4'-HYDROXYPHENYL)COUMARIN CHEMBL71271 25752 17543 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody 404859059 TEPROTUMUMAB 25753 17544 MCAM 4162 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME antibody 354702277 25754 17545 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL3544947 BURAPITANT 25755 17546 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SUFENTANIL SUFENTANIL 25757 17547 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE CEP-11981 CEP-11981 22148921 25758 17548 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME SSR-240612 17618300 25759 17549 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Aromatic bicyclic compound 1 25760 17550 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CARBAMAZEPINE CARBAMAZEPINE 25761 17551 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR fulvestrant FULVESTRANT 25762 17552 KDM4A 9682 DRUGGABLE GENOME, ENZYME THIOINOSINE THIOINOSINE 25763 17553 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DNA VACCINE 15382049 25764 17554 POLB 5423 DNA REPAIR, DRUGGABLE GENOME DEQUALINIUM CHLORIDE DEQUALINIUM CHLORIDE 25765 17555 NOS1 4842 DRUGGABLE GENOME, ENZYME CAFFEINE CAFFEINE 15556151 25766 17556 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-26 25768 17557 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2-HYDROXYPHENAZINE 5,10-DIOXIDE CHEMBL179611 25769 17558 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor NINTEDANIB NINTEDANIB 25770 17559 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 KAEMPFEROL KAEMPFEROL 25771 17560 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME GEDATOLISIB GEDATOLISIB 20166697 25773 17561 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 252166844 25774 17562 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME fluvastatin FLUVASTATIN 25775 17563 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME DOVITINIB DOVITINIB 25776 17564 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651566 25779 17565 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 2-ARACHIDONOYLGLYCEROL 2-ARACHIDONOYLGLYCEROL 25783 17566 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AG-881 25785 17567 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-739452 CHEMBL408564 25787 17568 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ETONOGESTREL ETONOGESTREL 25789 17569 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4384 CHEMBL602763 25790 17570 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-5134 CHEMBL602969 25792 17571 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE PF-03084014 NIROGACESTAT 26202948,25564152,23868008 25795 17572 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1473 FLUTICASONE PROPIONATE 25796 17573 PFKFB3 5209 ENZYME, KINASE INGAP peptide 15492571 25798 17574 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-55 25799 17575 IGFBP1 3484 DRUGGABLE GENOME OCTREOTIDE OCTREOTIDE 9512248,7525123 25801 17576 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 381118841 25804 17577 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 178102430 25806 17578 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ALSTERPAULLONE ALSTERPAULLONE 25807 17579 ATXN2 6311 NA CHELERYTHRINE CHELERYTHRINE 25808 17580 GMNN 51053 DRUGGABLE GENOME 25-HYDROXYCHOLECALCIFEROL CALCIFEDIOL 25811 17581 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-107022 CHEMBL1601846 25813 17582 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TAM 18539158 25814 17583 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME AZD6244, ARRY-142886 25816 17584 INPP1 3628 ENZYME LITHIUM LITHIUM 16787706 25818 17585 DGAT1 8694 ENZYME, DRUGGABLE GENOME amidepsines 25819 17586 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme25-2 25820 17587 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME N-phenyl-pyrimidin-4-amine derivative 1 25821 17588 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ALSTERPAULLONE ALSTERPAULLONE 25822 17589 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME RWJ-671818 CHEMBL1083499 25823 17590 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PEMETREXED PEMETREXED 21879757 25824 17591 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PMID29130358-Compound-LonimacranthoideVII 25825 17592 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME AZELASTINE AZELASTINE 25826 17593 GMNN 51053 DRUGGABLE GENOME ISOCONAZOLE ISOCONAZOLE 25827 17594 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 375973232 ABIVERTINIB 25828 17595 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME RUTAECARPINE RUTAECARPINE 25830 17596 BAZ2B 29994 NA SERTACONAZOLE NITRATE SERTACONAZOLE NITRATE 25833 17597 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor ROMIDEPSIN ROMIDEPSIN 25834 17598 GMNN 51053 DRUGGABLE GENOME GNF-PF-159 CHEMBL599924 25836 17599 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1200402 AMLODIPINE BESYLATE 25837 17600 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE antagonist 252166530 VENETOCLAX 25838 17601 ATXN2 6311 NA CUDRAFLAVONE B CUDRAFLAVONE B 25841 17602 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 8 25842 17603 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 5-HYDROXYINDOLACETIC ACID CHEMBL395915 25843 17604 SMN1 6606 DRUGGABLE GENOME ACLARUBICIN ACLARUBICIN 11734549 25845 17605 RAPGEF5 9771 NA antidepressants 25846 17606 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3',4'-DIMETHOXYFLAVONE 3',4'-DIMETHOXYFLAVONE 25847 17607 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650821 25849 17608 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME N-ETHYLMALEIMIDE N-ETHYLMALEIMIDE 25850 17609 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme9EHT6840 25851 17610 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR antidepressants 18794724 25852 17611 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE FOSTAMATINIB FOSTAMATINIB 25853 17612 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL428690 ALVOCIDIB 25856 17613 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor 178103911 25859 17614 PRMT5 10419 ENZYME, METHYL TRANSFERASE inhibitor 310264735 25860 17615 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Levalbuterol LEVOSALBUTAMOL 25861 17616 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DESERPIDINE DESERPIDINE 25862 17617 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORDANE CHLORDANE 25863 17618 NAT1 9 ENZYME, DRUGGABLE GENOME cotinine COTININE 25864 17619 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1096 AMLEXANOX 25865 17620 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLARITHROMYCIN CLARITHROMYCIN 22931300 25866 17621 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL428647 PACLITAXEL 25867 17622 KLK2 3817 PROTEASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 252166692 25868 17623 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 249565692 25869 17624 CBX1 10951 NA 3,4-METHYLENEDIOXYB-NITROSTYRENE CHEMBL596380 25870 17625 GMNN 51053 DRUGGABLE GENOME HALOPROGIN HALOPROGIN 25871 17626 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE LATREPIRDINE LATREPIRDINE 25873 17627 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ICI-199,441 ICI-199,441 25878 17628 PREP 5550 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 252166765 25879 17629 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GW441756X GW441756X 25880 17630 GHRL 51738 DRUGGABLE GENOME Relamorelin RELAMORELIN 25882 17631 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ICOSAPENT ICOSAPENT 25883 17632 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor TELATINIB TELATINIB 25884 17633 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR Irinotecan IRINOTECAN 26936505 25885 17634 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ALVOCIDIB ALVOCIDIB 25886 17635 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR belimumab BELIMUMAB 25887 17636 POLI 11201 DNA REPAIR IRSOGLADINE MALEATE IRSOGLADINE MALEATE 25889 17637 PMVK 10654 ENZYME, KINASE inhibitor 135651554 25890 17638 DOT1L 84444 CLINICALLY ACTIONABLE, DNA REPAIR, METHYL TRANSFERASE, DRUGGABLE GENOME, ENZYME candesartan CANDESARTAN 31327267 25892 17639 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME FLUORESCEIN FLUORESCEIN 25893 17640 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DOFETILIDE DOFETILIDE 22931300 25895 17641 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE S-49076 23804704 25897 17642 BAZ2B 29994 NA PROCHLORPERAZINE MALEATE PROCHLORPERAZINE MALEATE 25898 17643 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER bromperidol BROMPERIDOL 25900 17644 NDUFA4L2 56901 NA inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 25901 17645 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-102029 CHEMBL74913 25902 17646 FAAH 2166 ENZYME, DRUGGABLE GENOME Pyrazole derivative 83 25903 17647 IFNG 3458 DRUGGABLE GENOME MELATONIN MELATONIN 7722866 25904 17648 TLR7 51284 DRUGGABLE GENOME 852 25906 17649 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PERHEXILINE MALEATE PERHEXILINE MALEATE 25907 17650 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 223366124 PACRITINIB 25910 17651 GAL 51083 DRUGGABLE GENOME opioids 25912 17652 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GNF-PF-4668 CHEMBL584860 25913 17653 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX LGD-1550 25914 17654 GMNN 51053 DRUGGABLE GENOME ACRIDONE ACRIDONE 25915 17655 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME Darbepoetin alfa 25916 17656 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING SERTRALINE SERTRALINE 16680159 25918 17657 STXBP2 6813 NA emapalumab EMAPALUMAB 25919 17658 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor DINACICLIB DINACICLIB 25920 17659 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BIFONAZOLE BIFONAZOLE 25922 17660 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE 3-PHENYLUMBELLIFERONE CHEMBL153505 25923 17661 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000260214 CHEMBL602740 25924 17662 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME LIDOFLAZINE LIDOFLAZINE 25925 17663 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TRIACETYLRESVERATROL TRIACETYLRESVERATROL 25926 17664 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200434 OXTRIPHYLLINE 25927 17665 SFTPA1 653509 DRUGGABLE GENOME AMIODARONE AMIODARONE 11597911 25928 17666 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PRACINOSTAT PRACINOSTAT 25929 17667 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE PAZOPANI 25930 17668 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SPD-557 REVEXEPRIDE 25931 17669 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ARBIDOL UMIFENOVIR 25933 17670 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651887 CHEMBL442494 25936 17671 POLK 51426 DNA REPAIR, ENZYME ACETOSIDE ACETOSIDE 25937 17672 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME activator 381744978 25938 17673 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME LESTAURTINIB LESTAURTINIB 25939 17674 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME YOHIMBINE YOHIMBINE 25940 17675 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR SYNTHETIC CONJUGATED ESTROGENS 25942 17676 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PMID26666870-Compound-16 25943 17677 DGAT1 8694 ENZYME, DRUGGABLE GENOME Azole derivative 7 25944 17678 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME SCH-1359113 25945 17679 DIABLO 56616 NA RESVERATROL RESVERATROL 15837718,15469386 25946 17680 TRAF1 7185 NA adalimumab ADALIMUMAB 23007924 25947 17681 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NORADRENALINE NOREPINEPHRINE BITARTRATE 25948 17682 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist 252166705 NAVARIXIN 25950 17683 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX OXYQUINOLINE OXYQUINOLINE 25951 17684 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME SPERMIDINE SPERMIDINE 25952 17685 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE EPINEPHRINE EPINEPHRINE 12376414 25953 17686 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor GIVINOSTAT GIVINOSTAT 25955 17687 RRAS2 22800 NA tamoxifen TAMOXIFEN 19047159 25956 17688 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIPHENYLPYRALINE DIPHENYLPYRALINE 25957 17689 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist CHEMBL1201620 SOMATREM 25958 17690 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR FAMCICLOVIR FAMCICLOVIR 10522033 25959 17691 SMN1 6606 DRUGGABLE GENOME DNDI1417268 CHEMBL1517542 25960 17692 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor PF03084014 25961 17693 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE CENISERTIB CENISERTIB 25962 17694 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CARBOXYMETHOXYLAMINE CARBOXYMETHOXYLAMINE 25963 17695 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Veliparib VELIPARIB 26779812 25966 17696 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Dimethindene DIMETHINDENE 25967 17697 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER rituximab RITUXIMAB 25637052 25969 17698 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PAPAVEROLINE PAPAVEROLINE 25970 17699 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE NAKIJIQUINONES H NAKIJIQUINONES H 18676149 25971 17700 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Xanthine/amino piperidine compound 1 25972 17701 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MANGOSTIN MANGOSTIN 25973 17702 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-46080 CHEMBL1331754 22524450 25975 17703 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 bupropion BUPROPION 26132489 25977 17704 COL6A3 1293 DRUGGABLE GENOME, PROTEASE INHIBITOR CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 25979 17705 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME inhibitor CHEMBL2108678 NESVACUMAB 25981 17706 ALOX15B 247 DRUGGABLE GENOME, ENZYME O-DEMETHYLATED ADAPALENE O-DEMETHYLATED ADAPALENE 25982 17707 ALOX15 246 ENZYME, DRUGGABLE GENOME E324 E324 25984 17708 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650807 25985 17709 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE MPA PROGESTERONE 16123159 25988 17710 SLC6A19 340024 DRUGGABLE GENOME, TRANSPORTER inhibitor 223365936 BENZATROPINE 25990 17711 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 25991 17712 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CART-20 cells 25992 17713 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME MLN-8054 MLN-8054 25993 17714 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME ethinyl estradiol / norelgestromin 25994 17715 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Betamethasone Valerate 25995 17716 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DESMEDIPHAM DESMEDIPHAM 25998 17717 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PMID29334795-Compound-61 25999 17718 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME RIBOCICLIB RIBOCICLIB 26987942 26000 17719 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME AW-01208 CHEMBL560532 19631549 26001 17720 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER GO-Y034 CHEMBL595816 22112540 26005 17721 NDUFA4 4697 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545135 NV-128 26006 17722 GMNN 51053 DRUGGABLE GENOME GW282974X GW282974X 26007 17723 HSPA8 3312 TUMOR SUPPRESSOR ACETAMINOPHEN ACETAMINOPHEN 15010265 26008 17724 GAL 51083 DRUGGABLE GENOME mirtazapine MIRTAZAPINE 26009 17725 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 315661215 26011 17726 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BCMA-specific CAR-expressing T Lymphocytes 26013 17727 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BML-210 CHEMBL324053 16921367 26015 17728 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME JUGLONE JUGLONE 26016 17729 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-E4 26017 17730 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Venetoclax VENETOCLAX 27974663 26018 17731 TXN 7295 DRUGGABLE GENOME, THIOREDOXIN GAMBOGENIC ACID GAMBOGENIC ACID 22663155 26020 17732 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102707 26021 17733 PNP 4860 ENZYME, DRUGGABLE GENOME BCX-3408 ULODESINE 26022 17734 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME IBRITUMOMAB IBRITUMOMAB TIUXETAN 26024 17735 XDH 7498 DRUGGABLE GENOME, ENZYME METHYLENE BLUE 2855011 26026 17736 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-65a 26027 17737 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALCIMYCIN CALCIMYCIN 26028 17738 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME Dasatinib DASATINIB 26030 17739 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE NSC-95397 CHEMBL429095 26031 17740 PTGS1 5742 ENZYME, DRUGGABLE GENOME NAPROXEN NAPROXEN 26032 17741 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE CARBOPLATIN CARBOPLATIN 26033 17742 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME flupenthixol E-FLUPENTIXOL 27992301 26034 17743 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Fluorouracil FLUOROURACIL 27626067,26637369 26035 17744 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor RIDAFOROLIMUS RIDAFOROLIMUS 26036 17745 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE IRIGINOL HEXAACEATATE IRIGINOL HEXAACEATATE 26037 17746 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ARQ 087 26038 17747 TSPO 706 DRUGGABLE GENOME 11C-PBR-28 26039 17748 TARDBP 23435 TUMOR SUPPRESSOR SJ000260212 CHEMBL607138 26040 17749 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME DOVITINIB DOVITINIB 26041 17750 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 223366202 AXL-1717 26043 17751 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME PIFEXOLE PIFEXOLE 26044 17752 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE NORDIHYDROGUAIARETIC ACID 2122915 26045 17753 ADH1C 126 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1308 FOMEPIZOLE 26046 17754 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR L-NOREPINEPHRINE L-NOREPINEPHRINE 26047 17755 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR efavirenz EFAVIRENZ 24819158 26048 17756 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME simvastatin acid 28350522,29469964,25446771,26367500 26049 17757 FKBP5 2289 DRUGGABLE GENOME clozapine CLOZAPINE 25751398 26050 17758 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL232943 MK0686 26053 17759 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3707380 RG6029 26054 17760 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 252166612 OMARIGLIPTIN 26055 17761 POLB 5423 DNA REPAIR, DRUGGABLE GENOME 9-AMINOCAMPTOTHECIN 9-AMINOCAMPTOTHECIN 26056 17762 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CAR-20/19-T Cells 26057 17763 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Tricyclic heterocycle derivative 5 26059 17764 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650904 RITANSERIN 26060 17765 COMT 1312 DRUGGABLE GENOME, ENZYME Antiinflammatory agents, non-steroids 25096645 26061 17766 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-95397 CHEMBL429095 26062 17767 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SNS-032 BMS-387032 26063 17768 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE TCMDC-125758 CHEMBL546797 26064 17769 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME unspecified IGF-1R antibody 26577700 26065 17770 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Estriol ESTRIOL 26066 17771 PML 5371 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE arsenic trioxide 24433361 26067 17772 KDM1B 221656 DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING, ENZYME PMID27019002-Compound-47 26069 17773 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME KOPARIN KOPARIN 26070 17774 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME LCZ696 LCZ696 26071 17775 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PYROGALLOL RED PYROGALLOL RED 26072 17776 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME NITROGLYCERIN NITROGLYCERIN 16612556 26073 17777 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SURAMIN SURAMIN 26074 17778 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2105729 DABRAFENIB MESYLATE 26075 17779 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 187051806 26076 17780 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE Z160 Z160 19815411 26077 17781 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME RGH-896 RADIPRODIL 26079 17782 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE BMS-695735 CHEMBL459729 26080 17783 IL13RA2 3598 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CHEMBL2108583 CINTREDEKIN BESUDOTOX 26081 17784 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ENMD-2076 ENMD-2076 26082 17785 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL488436 AZD-5438 26083 17786 TF 7018 CELL SURFACE, DRUGGABLE GENOME adalimumab ADALIMUMAB 27115882 26084 17787 RGS4 5999 DRUGGABLE GENOME inhibitor 252827387 26086 17788 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 310264695 CC-223 26089 17789 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-54 26090 17790 MAOA 4128 DRUGGABLE GENOME, ENZYME Schiff base compound 1 26092 17791 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE inhibitor 135652717 STAUROSPORINE 26093 17792 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BENZYL NICOTINATE BENZYL NICOTINATE 26094 17793 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor X-82 X-82 26098 17794 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL3545240 CLX-0921 26100 17795 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME Pfizer 4 26101 17796 KDM4A 9682 DRUGGABLE GENOME, ENZYME TETRYDAMINE TETRYDAMINE 26102 17797 ATAD5 79915 NA 2-(4-METHOXYPHENYL)BENZO[D]THIAZOLE CHEMBL460508 26103 17798 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 THIOPENTAL SODIUM THIOPENTAL SODIUM 26104 17799 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME CP-868596 CRENOLANIB 26105 17800 SMN1 6606 DRUGGABLE GENOME 2-(4-METHOXYPHENYL)BENZO[D]THIAZOLE CHEMBL460508 26106 17801 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE Peptide analog 60 26108 17802 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Tricyclic heterocycle derivative 5 26109 17803 TUBB2A 7280 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 26110 17804 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200341 INDECAINIDE HYDROCHLORIDE 26112 17805 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PONATINIB PONATINIB 20513156 26116 17806 DNER 92737 NA Isoxazole-based bicyclic compound 19 26117 17807 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR PMID25980951-Compound-27 26120 17808 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 26121 17809 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR WORTMANNIN WORTMANNIN 26123 17810 KDM4A 9682 DRUGGABLE GENOME, ENZYME BUTOCONAZOLE NITRATE BUTOCONAZOLE NITRATE 26124 17811 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NSC-66209 CHEMBL175266 26125 17812 ACP1 52 ENZYME, DRUGGABLE GENOME, PROTEIN PHOSPHATASE GNF-PF-3542 CHEMBL598477 26126 17813 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Avelumab AVELUMAB 26127 17814 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody ZALUTUMUMAB ZALUTUMUMAB 26128 17815 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor SB939 26133 17816 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR DNDI1417086 CHEMBL1224755 26136 17817 NEDD4L 23327 ENZYME citalopram CITALOPRAM 23809733 26137 17818 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GEFITINIB GEFITINIB 26140 17819 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652043 26141 17820 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IIIC AESCULIOSIDE IIIC 20371180 26144 17821 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Quinoxaline derivative 4 26145 17822 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PENTACHLORONITROBENZENE PENTACHLORONITROBENZENE 26146 17823 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SB-220025 SB-220025 26147 17824 PTGES 9536 DRUGGABLE GENOME, ENZYME TRANSFORMING GROWTH FACTOR 16572115 26148 17825 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME DX-8951F EXATECAN MESYLATE 11802813 26149 17826 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR INDIUM CHLORIDE INDIUM CHLORIDE 26150 17827 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32c 26151 17828 KCNK5 8645 ION CHANNEL, DRUGGABLE GENOME blocker 135650872 QUINIDINE 26152 17829 KLK1 3816 PROTEASE, DRUGGABLE GENOME, ENZYME ECALLANTIDE ECALLANTIDE 26153 17830 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIPYRITHIONE DIPYRITHIONE 26154 17831 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650248 26155 17832 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-125814 CHEMBL533082 26157 17833 CCL2 6347 DRUGGABLE GENOME MCP-1 26158 17834 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME PF-562271 PF-00562271 26159 17835 HMGCR 3156 ENZYME, DRUGGABLE GENOME ROSUVASTATIN ROSUVASTATIN 26160 17836 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR INDOMETHACIN INDOMETHACIN 16956981 26161 17837 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Ponatinib PONATINIB 26270481 26163 17838 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CER-002 CER-002 20393155 26164 17839 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME cariprazine CARIPRAZINE 26165 17840 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE Conatumumab CONATUMUMAB 26166 17841 TSPO 706 DRUGGABLE GENOME Cinolazepam CINOLAZEPAM 26167 17842 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102777 SC-41390 26168 17843 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor BORTEZOMIB BORTEZOMIB 26170 17844 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545399 R-112 26173 17845 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL1980297 ILORASERTIB 26174 17846 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME VANDETANIB VANDETANIB 26175 17847 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RS-17053 CHEMBL88272 26176 17848 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME FOSPROPOFOL FOSPROPOFOL 26177 17849 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE BECAPLERMIN BECAPLERMIN 26179 17850 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 223366077 RGB-286638 26180 17851 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME PMID29130358-Compound-Figure18(14) 26181 17852 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor NERATINIB NERATINIB 26183 17853 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE ERDAFITINIB ERDAFITINIB 26324363,31340094 26184 17854 MARK1 4139 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 26185 17855 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PROPYLPYRAZOLETRIOL PROPYLPYRAZOLETRIOL 26186 17856 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE varlitinib VARLITINIB 26191 17857 POLK 51426 DNA REPAIR, ENZYME 2,3-DIHYDROXY-4-METHOXY-4'-ETHOXYBENZOPHENONE 2,3-DIHYDROXY-4-METHOXY-4'-ETHOXYBENZOPHENONE 26193 17858 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ANTI-CD20 ANTIBODY 11830481 26194 17859 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LAPATINIB LAPATINIB 25305330,24355130 26195 17860 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor VORINOSTAT VORINOSTAT 26196 17861 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Finerenone FINERENONE 26197 17862 KDM4A 9682 DRUGGABLE GENOME, ENZYME 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 26198 17863 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 178100411 26199 17864 ALOX15B 247 DRUGGABLE GENOME, ENZYME RHODOMYRTOXIN B RHODOMYRTOXIN B 26200 17865 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BERBERINE BERBERINE 26201 17866 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL1952329 SGI-1776 26203 17867 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CNTO-95 INTETUMUMAB 26204 17868 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Carbamide derivative 6 26205 17869 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200948 TRIMIPRAMINE MALEATE 26206 17870 POLK 51426 DNA REPAIR, ENZYME FLAVANOMAREIN FLAVANOMAREIN 26207 17871 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE UH-232 CHEMBL278751 26208 17872 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Namitecan NAMITECAN 26209 17873 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PF-562271 PF-00562271 26210 17874 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL2096626 26211 17875 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX ALITRETIONINE 26212 17876 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Olaparib OLAPARIB 28148839 26213 17877 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 354702224 26214 17878 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HYDRALAZINE HYDROCHLORIDE HYDRALAZINE HYDROCHLORIDE 26215 17879 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ramucirumab RAMUCIRUMAB 26216 17880 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR CNF1010 TANESPIMYCIN 26217 17881 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 310264777 26218 17882 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZO[B]TRIPHENYLENE BENZO[B]TRIPHENYLENE 26219 17883 HSPA4 3308 NA ARSENIC TRIOXIDE 11678611 26221 17884 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CEDIRANIB CEDIRANIB 26222 17885 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545144 TAS-115 26223 17886 AQP4 361 ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ETHOXZOLAMIDE ETHOXZOLAMIDE 18572411 26225 17887 XDH 7498 DRUGGABLE GENOME, ENZYME GLUCOCORTICOID 8920983 26226 17888 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME activator 135650748 26227 17889 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-8 26228 17890 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR CORT 108297 26229 17891 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME MASITINIB MASITINIB 26231 17892 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 363894217 VORUCICLIB 26232 17893 KCNC2 3747 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL113461 TEDISAMIL 26233 17894 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RESERPINE RESERPINE 26235 17895 IL1B 3553 KINASE, DRUGGABLE GENOME clodronate CLODRONIC ACID 16257277 26236 17896 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE antipsychotics 17976958 26237 17897 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME DACTOLISIB DACTOLISIB 26238 17898 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-69187 CHEMBL19954 26241 17899 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME AG-1879 CHEMBL406845 26242 17900 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALITRETINOIN ALITRETINOIN 21489804,25057340,7807131 26244 17901 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME ALSTERPAULLONE ALSTERPAULLONE 26245 17902 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME N-METHOXYCARBONYLMETHYL-OXALAMIC ACID METHYL ESTER CHEMBL92309 19359167 26246 17903 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR PF-562271 PF-00562271 26248 17904 CEBPA 1050 TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE N/A 20038735,26601784,19171880,22814295,25241285,23521373 26249 17905 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MG-132 MG-132 26250 17906 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PROTEASOME INHIBITOR 18298552 26251 17907 GHRL 51738 DRUGGABLE GENOME ARD-07 MACIMORELIN 26252 17908 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TEROXIRONE TEROXIRONE 26253 17909 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3545341 SAR-407899 26254 17910 MAST3 23031 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 252827499 26256 17911 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-91 26257 17912 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 tolterodine TOLTERODINE 26259 17913 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651427 ADENOSINE DIPHOSPHATE 26260 17914 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER amisulpride AMISULPRIDE 29443543 26262 17915 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE VERAPAMIL VERAPAMIL 9579573 26266 17916 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE inhibitor 178102653 SIROLIMUS 26267 17917 SLC28A2 9153 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME gemcitabine GEMCITABINE 18538445,20665488 26269 17918 CBX1 10951 NA GNF-PF-5007 CHEMBL1989853 26271 17919 CDH17 1015 TRANSPORTER, CELL SURFACE TCDD 12054747 26272 17920 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL49642 INDIBULIN 26274 17921 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME 4-BENZAMIDOPHENYLSTIBONIC ACID CHEMBL1726814 26275 17922 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME REGN1979 ODRONEXTAMAB 26276 17923 CBX1 10951 NA GNF-PF-5134 CHEMBL602969 26277 17924 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID25991433-Compound-P1 26279 17925 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178103501 PRUNETIN 26281 17926 CYP24A1 1591 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME CTA018 LUNACALCIPOL 26282 17927 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Pemetrexed PEMETREXED 27876675 26284 17928 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BETAMETHASONE SODIUM PHOSPHATE BETAMETHASONE SODIUM PHOSPHATE 26286 17929 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CYC-116 CYC-116 20462263 26287 17930 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650728 26288 17931 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LEAD DIACETATE TRIHYDRATE LEAD DIACETATE TRIHYDRATE 26289 17932 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor 178103250 BEFLOXATONE 26291 17933 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME TACEDINALINE TACEDINALINE 18692397 26292 17934 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE HORMONES 8119934 26294 17935 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-US20120277229 40(1.2) 26297 17936 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME AG-537 CHEMBL67535 26300 17937 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NAPHTHALENE-1,2-DIOL CHEMBL204543 24997687 26301 17938 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR DNDI1417080 CHEMBL1498652 26303 17939 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE TCMDC-125785 CHEMBL588525 26305 17940 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE inhibitor 354702208 26306 17941 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Pyridinone carboxamide derivative 1 26308 17942 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652214 26309 17943 KCNH6 81033 DRUGGABLE GENOME, ION CHANNEL inhibitor 223366024 26311 17944 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102563 26312 17945 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL646 TRIAZOLAM 26313 17946 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565691 CHEMBL1086377 26314 17947 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME 5-AZACYTIDINE AZACITIDINE 9801800 26317 17948 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR THEOPHYLLINE THEOPHYLLINE 26318 17949 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME APICIDIN APICIDIN 19705846 26319 17950 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR SL-0101 CHEMBL240954 26320 17951 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR SILYMARIN SILYBIN A 15103051 26321 17952 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME Azetidine derivative 2 26322 17953 EML4 27436 CLINICALLY ACTIONABLE, KINASE AZD3463 27009859 26324 17954 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ANTI-DIABETIC AGENT 15207658 26328 17955 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE zoledronate ZOLEDRONIC ACID 21196316 26330 17956 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME bucillamine BUCILLAMINE 26332 17957 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL1201129 DECITABINE 26333 17958 EHMT1 79813 ENZYME, DRUGGABLE GENOME inhibitor 249565918 26334 17959 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME blocker 318164837 26336 17960 TANC2 26115 NA calcium channel blockers 24192120 26337 17961 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201563 INTERFERON BETA-1B 26338 17962 COMT 1312 DRUGGABLE GENOME, ENZYME Methyldopa METHYLDOPA 26340 17963 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR ALISERTIB ALISERTIB 26342 17964 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TRASTUZUMAB TRASTUZUMAB 26619011,22908275,25157968,23220880,16397024,26243863 26344 17965 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR ARA-C 8819077,8450676 26345 17966 CRABP2 1382 NA RETINOID 12153175 26346 17967 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650236 EPROSARTAN 26348 17968 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE VX-970 BERZOSERTIB 28363999 26351 17969 DHFR 1719 DRUGGABLE GENOME, ENZYME PRALATREXATE PRALATREXATE 26352 17970 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Panitumumab PANITUMUMAB 26354 17971 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GALANGIN GALANGIN 26355 17972 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR METHYLERGONOVINE METHYLERGONOVINE 26357 17973 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE inhibitor SOPHORETIN QUERCETIN 26362 17974 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER rifampin RIFAMPIN 26363 17975 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 252827527 26365 17976 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME RETINOIC ACID 9392425 26366 17977 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SJ000007704 CHEMBL589469 26368 17978 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SCOPOLETIN SCOPOLETIN 26369 17979 IL1B 3553 KINASE, DRUGGABLE GENOME Platinum compounds 27498158 26375 17980 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PROGESTERONE PROGESTERONE 18665217 26377 17981 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 178102328 PI-103 26378 17982 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CHEMBL681 ETOMIDATE 26380 17983 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE MAGNESIUM SULFATE 16384608 26382 17984 MAPT 4137 DRUGGABLE GENOME RHAMNETIN RHAMNETIN 26384 17985 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Desogestrel DESOGESTREL 26385 17986 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE FENAMIC ACID FENAMIC ACID 20038108 26386 17987 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 178101919 26387 17988 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME BETUNOLIC ACID BETUNOLIC ACID 26390 17989 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649900 OTENZEPAD 26392 17990 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BETAMETHASONE DIPROPIONATE BETAMETHASONE DIPROPIONATE 26393 17991 HTT 3064 DRUGGABLE GENOME PYRITHIONE ZINC PYRITHIONE ZINC 26395 17992 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR R-1487 R-1487 26398 17993 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-5478 CHEMBL586982 26399 17994 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AR-67 AR-67 26400 17995 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 385612186 26401 17996 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ALISERTIB ALISERTIB 26402 17997 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545402 XL-820 26405 17998 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR COMPLETE FREUND'S ADJUVANT 16288729 26406 17999 CA12 771 DRUGGABLE GENOME FERULIC ACID 26408 18000 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NIHYDRAZONE NIHYDRAZONE 26410 18001 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME COAGULATION FACTOR VIIA 26412 18002 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME MITHRAMYCIN PLICAMYCIN 17124180 26413 18003 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650159 26414 18004 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 387065600 26415 18005 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ELLAGIC ACID ELLAGIC ACID 26416 18006 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-18 26417 18007 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZAFIRLUKAST ZAFIRLUKAST 26418 18008 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-G1 26420 18009 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 404859129 26423 18010 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE IMATINIB IMATINIB 26424 18011 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME DICLOFENAC DICLOFENAC 9090444 26425 18012 SCD 6319 DRUGGABLE GENOME, ENZYME COLCHICINE COLCHICINE 6148915 26426 18013 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-60340 CHEMBL1534034 26427 18014 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE IMATINIB IMATINIB 20537386,26758680,19075254,27125982,15930265,16775234,24367893,12623848,18191450,25686603,25207766,22371878,12476305,15194504 26428 18015 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME NCX 1510 26429 18016 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME COLESTIPOL HYDROCHLORIDE 2642754 26430 18017 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MITOBRONITOL MITOBRONITOL 26431 18018 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3545249 GLPG-0555 26432 18019 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Afatinib AFATINIB 27207775 26434 18020 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ROTENONE ROTENONE 26435 18021 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE ANTIESTROGEN 16682955 26437 18022 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 2-BROMO-HEXADECANOIC ACID CHEMBL118417 26438 18023 HTT 3064 DRUGGABLE GENOME GNF-PF-3286 CHEMBL581880 26440 18024 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 178100451 26443 18025 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE PMID26882240-Compound-14 26445 18026 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 11 26446 18027 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZ-TAK1 27655129 26448 18028 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ESCULETIN ESCULETIN 26449 18029 TLR7 51284 DRUGGABLE GENOME agonist 315661110 26450 18030 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102305 DASATINIB 26451 18031 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Bicyclic hexapeptide derivative 2 26452 18032 MUC2 4583 DRUGGABLE GENOME 5-FU FLUOROURACIL 14576935 26453 18033 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 178102626 26455 18034 TSPO 706 DRUGGABLE GENOME Alprazolam ALPRAZOLAM 26456 18035 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AMSACRINE AMSACRINE 22931300 26457 18036 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE BMS-690514 BMS-690514 26458 18037 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR KAVAIN KAVAIN 26459 18038 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL antagonist 329968408 26460 18039 TNK1 8711 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor TOZASERTIB TOZASERTIB 19035792 26461 18040 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Ralinepag RALINEPAG 26462 18041 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE VELIPARIB VELIPARIB 29338080 26464 18042 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL967 TEMAZEPAM 26465 18043 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL1567 SUNITINIB MALATE 26467 18044 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200597 ETIDOCAINE HYDROCHLORIDE 26470 18045 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BROMCRESOL GREEN BROMCRESOL GREEN 26471 18046 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE TEMSIROLIMUS TEMSIROLIMUS 26472 18047 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme11 26474 18048 HPD 3242 ENZYME, DRUGGABLE GENOME 6-HYDROXYDOPAMINE 18495353 26475 18049 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100465 26476 18050 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE VE-822 BERZOSERTIB 26477 18051 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PURPURIN PURPURIN 26478 18052 KCNA7 3743 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL113461 TEDISAMIL 26479 18053 FAAH 2166 ENZYME, DRUGGABLE GENOME Ketoheterocycle derivative 2 26481 18054 FZD6 8323 CELL SURFACE, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651915 26483 18055 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme21Right 26484 18056 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME UVB 14962109 26485 18057 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FENAMIC ACID FENAMIC ACID 26486 18058 SMARCA4 6597 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING ABEMACICLIB ABEMACICLIB 30718512,30718506 26487 18059 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-123916 CHEMBL493863 26488 18060 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200703 CHLORDIAZEPOXIDE HYDROCHLORIDE 26489 18061 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE LITHIUM LITHIUM 16300803 26490 18062 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NSC-117271 CHEMBL287689 26491 18063 HBB 3043 DRUGGABLE GENOME, ENZYME ELLAGIC ACID ELLAGIC ACID 26492 18064 KDM4A 9682 DRUGGABLE GENOME, ENZYME CINTAZONE CINTAZONE 26494 18065 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 363894185 26495 18066 TSPO 706 DRUGGABLE GENOME LORAZEPAM LORAZEPAM 26496 18067 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TAM 8388708 26498 18068 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 4-HYDROXYBENZALDEHYDE PHENYLHYDRAZONE CHEMBL224032 26499 18069 TRPC4 7223 ION CHANNEL, KINASE, DRUGGABLE GENOME, CELL SURFACE blocker 135651058 26500 18070 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 zidovudine ZIDOVUDINE 22960662 26501 18071 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 363894217 VORUCICLIB 26502 18072 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR DIOSMIN DIOSMIN 26503 18073 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652514 26507 18074 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135652148 ENDOMORPHIN-1 26509 18075 PARP11 57097 DRUGGABLE GENOME antidepressants 26510 18076 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SCRIPTAID SCRIPTAID 19966789 26513 18077 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME PROGESTIN PROGESTERONE 1831804 26515 18078 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DIETHYLTOLUAMIDE DIETHYLTOLUAMIDE 26516 18079 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 clozapine CLOZAPINE 23297297 26517 18080 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROPRANOLOL PROPRANOLOL 2903243 26518 18081 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BAY1125976 27699769 26520 18082 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID30259754-Compound-Px-102 26521 18083 TOP2B 7155 DRUGGABLE GENOME, ENZYME XB-947 10518594 26522 18084 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Bremelanotide BREMELANOTIDE 26523 18085 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE PALIFERMIN PALIFERMIN 26524 18086 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE OBATOCLAX OBATOCLAX 26525 18087 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TCMDC-124518 CHEMBL527584 26526 18088 PGD 5226 ENZYME, DRUGGABLE GENOME GHRP-2 26528 18089 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMA 10777098,8946678 26530 18090 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHYCLOTHIAZIDE METHYCLOTHIAZIDE 26531 18091 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME Anti-CEA-CAR T 26532 18092 VCAM1 7412 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME AGI-1067, SUCCINOBUCOL 26533 18093 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER 5-FU FLUOROURACIL 16892554 26534 18094 INHBE 83729 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME GNRH GONADORELIN ACETATE 8756531 26535 18095 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME Clonidine CLONIDINE 26536 18096 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 2,7-BIS[3-(DIETHYLAMINO)PROPIONAMIDO]ANTHRAQUINONE CHEMBL91163 18571928 26537 18097 EPHB4 2050 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE XL647 TESEVATINIB 26538 18098 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER ABT-702 CHEMBL66089 26539 18099 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Alectinib ALECTINIB 28476735 26541 18100 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE PALIFERMIN PALIFERMIN 26542 18101 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ENTRECTINIB ENTRECTINIB 32315394 26544 18102 POLB 5423 DNA REPAIR, DRUGGABLE GENOME LASALOCID A SODIUM LASALOCID A SODIUM 26545 18103 F5 2153 DRUGGABLE GENOME inhibitor CHEMBL2109065 DROTRECOGIN ALFA (ACTIVATED) 26546 18104 POLB 5423 DNA REPAIR, DRUGGABLE GENOME PICEID PICEID 26548 18105 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE ISOPROPANOL ISOPROPYL ALCOHOL 6409434 26549 18106 PLD2 5338 ENZYME, DRUGGABLE GENOME inhibitor 252827440 26551 18107 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CY-208243 CHEMBL313737 26553 18108 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME TAMATINIB R-406 26554 18109 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Anti-IP10 26555 18110 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ADJUVANT 15567937 26556 18111 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE LEPIRUDIN LEPIRUDIN 16038707 26558 18112 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME SIB-1893 CHEMBL88612 26559 18113 KDM4A 9682 DRUGGABLE GENOME, ENZYME NCG-C00094421-01 CHEMBL553503 26561 18114 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3201 CHEMBL581872 26564 18115 MMP7 4316 NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor CHEMBL1200567 DOXYCYCLINE HYCLATE 26565 18116 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE RUCAPARIB RUCAPARIB 26566 18117 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TAE-684 TAE-684 26569 18118 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE aspirin ASPIRIN 17184645,16458133,16675000,11723016,16493486,10704169,11054089,15840736,10459913,16153930,23834376,22028352,20138334,16581111 26570 18119 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE CHEMBL457504 26571 18120 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME METHYLDOPA METHYLDOPA 22931300 26572 18121 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SAQUINAVIR MESYLATE SAQUINAVIR MESYLATE 26573 18122 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ISOETHARINE MESYLATE ISOETHARINE MESYLATE 26575 18123 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MLN2480 26576 18124 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200584 AMINOSALICYLATE POTASSIUM 26578 18125 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CLIOQUINOL CLIOQUINOL 26579 18126 DDC 1644 ENZYME, DRUGGABLE GENOME CARBIDOPA CARBIDOPA 26580 18127 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Certoparin sodium 26581 18128 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ROCAGLAMIDE ROCAGLAMIDE 26583 18129 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Carboxamide derivative 9 26584 18130 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME IPRATROPIUM IPRATROPIUM 26585 18131 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER latanoprost LATANOPROST 25339146 26589 18132 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamate derivative 11 26590 18133 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Sirolimus SIROLIMUS 15647370,26882569,28514312,19029981,17376864 26591 18134 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL411907 SONOLISIB 26593 18135 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NOSCAPINE NOSCAPINE 26594 18136 PON1 5444 ENZYME, TRANSPORTER, DRUGGABLE GENOME oxaliplatin OXALIPLATIN 26595 18137 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LINIFANIB LINIFANIB 26596 18138 TYMP 1890 GROWTH FACTOR, DRUGGABLE GENOME inhibitor CHEMBL65375 TIPIRACIL HYDROCHLORIDE 26597 18139 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652582 26598 18140 PTGES 9536 DRUGGABLE GENOME, ENZYME 6BIO 6BIO 24697244 26599 18141 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102576 CHELERYTHRINE 26600 18142 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 249565843 26603 18143 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OXENDOLONE OXENDOLONE 26605 18144 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652024 26606 18145 PTPN6 5777 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-87877 CHEMBL472004 26608 18146 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME activator 135652736 26609 18147 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ARUNDINE ARUNDINE 26610 18148 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL2103743 TOFACITINIB CITRATE 26613 18149 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 178100751 26614 18150 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SANGUINARINE SULFATE SANGUINARINE SULFATE 26615 18151 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000069305 CHEMBL603739 26616 18152 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE CEDIRANIB CEDIRANIB 26618 18153 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME TECADENOSON TECADENOSON 23388705 26619 18154 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER unspecified IGF-1R antibody 27196767 26622 18155 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE INCB13739 26623 18156 ATP5F1D 513 TRANSPORTER DESFLURANE DESFLURANE 26624 18157 COL1A1 1277 CLINICALLY ACTIONABLE, DRUGGABLE GENOME valproic acid 26727275 26625 18158 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PYRROLIDINE DITHIOCARBAMATE PYRROLIDINE DITHIOCARBAMATE 26626 18159 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-63 26627 18160 MT-RNR1 4549 KINASE neomycin NEOMYCIN 18830133,16875663,9164619,19682603,16631122,21495045,16458854,12031626,16375862,9831149,17637808,22475488,11857751,27397648,9779807,7689389,20111055,9111378,27427311,17698030,11313749,20416460,16168391,24703164,9950117,21504270,11174059,8285309,18790089,15917167,20353758,16955413,16380089,14699607,17999439,14755216,17341440,19376484,15708009,25515069,15555598,11079536,17434445 26628 18161 CDH17 1015 TRANSPORTER, CELL SURFACE DEXAMETHASONE DEXAMETHASONE 10760957 26629 18162 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME LY2886721 LY-2886721 26630 18163 ALB 213 TRANSPORTER, DRUGGABLE GENOME Iodipamide IODIPAMIDE 26631 18164 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor ARQ736 26632 18165 AKR1B1 231 DRUGGABLE GENOME, ENZYME URACIL URACIL 9057855 26635 18166 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000044511 CHEMBL592124 26636 18167 TSPO 706 DRUGGABLE GENOME Aryl oxyanilide derivative 3 26639 18168 SMN1 6606 DRUGGABLE GENOME CID 752709 CHEMBL429335 26640 18169 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DASATINIB DASATINIB 26641 18170 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LANSOPRAZOLE LANSOPRAZOLE 26642 18171 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PI-103 PI-103 26644 18172 KIF11 3832 DRUGGABLE GENOME Ispinesib ISPINESIB 26645 18173 PRSS3 5646 ENZYME, PROTEASE, DRUGGABLE GENOME DERMOLASTIN 26646 18174 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR bisoprolol BISOPROLOL 15861037,16325050 26648 18175 ATXN2 6311 NA AFIMOXIFENE AFIMOXIFENE 26650 18176 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CARMINE CARMINE 26651 18177 BARD1 580 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR carboplatin CARBOPLATIN 30071039 26652 18178 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102540 26655 18179 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME ZM-447439 CHEMBL202721 26656 18180 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TRIAMTERENE TRIAMTERENE 26657 18181 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME ESTAZOLAM ESTAZOLAM 26658 18182 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CHEMBL2108576 BAPINEUZUMAB 26659 18183 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650529 26660 18184 HMGCR 3156 ENZYME, DRUGGABLE GENOME LOVASTATIN LOVASTATIN 26661 18185 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE EPIGALLOCATECHIN GALLATE 11936850 26662 18186 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME KHK2455 26663 18187 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME sulfamethoxazole / trimethoprim 26086150 26666 18188 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 385612208 26667 18189 ITPR1 3708 ION CHANNEL, KINASE, DRUGGABLE GENOME, TRANSPORTER antagonist 135652750 26668 18190 ATAD5 79915 NA CID 5310801 CHEMBL260451 26669 18191 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650509 26670 18192 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE 178101647 26673 18193 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME PMID27998201-Compound-9 26674 18194 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR Indole-based analog 14 26675 18195 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME MK-1775 ADAVOSERTIB 26678 18196 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102679 TIVOZANIB 26683 18197 NOS1 4842 DRUGGABLE GENOME, ENZYME NSAID 11837731 26684 18198 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR LY2940680 26685 18199 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MIDODRINE MIDODRINE 22931300 26686 18200 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 318164840 26687 18201 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DNA VACCINE 16751417 26688 18202 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE ALISERTIB ALISERTIB 26689 18203 IL1B 3553 KINASE, DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 24776844,28696418 26691 18204 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZD4547 27338794 26694 18205 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565902 NORHARMANE 26695 18206 CDK13 8621 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 375973251 26696 18207 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE (RS)-ROSCOVITINE (RS)-ROSCOVITINE 26697 18208 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 5-AZA-2-DEOXYCYTIDINE 14559817 26698 18209 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE RIGOSERTIB RIGOSERTIB 26701 18210 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL58323 ERLOSAMIDE 26704 18211 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR ADRIAMYCIN ADRIAMYCIN 15707569 26705 18212 MGLL 11343 DRUGGABLE GENOME, ENZYME URB597 URB-597 19232787 26706 18213 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISOKOBUSONE ISOKOBUSONE 26707 18214 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545115 ASCIMINIB 26708 18215 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CHIR-99021 CHIR-99021 26712 18216 POLB 5423 DNA REPAIR, DRUGGABLE GENOME LUTEOLIN LUTEOLIN 26713 18217 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ADCT-502 26714 18218 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR GALLIUM NITRATE 8381250 26718 18219 CXCL8 3576 DRUGGABLE GENOME MBL 12900342 26721 18220 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MEFENAMIC ACID MEFENAMIC ACID 22931300 26723 18221 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SP-600125 SP-600125 26726 18222 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2,3,4,6-TETRACHLORO-PHENOL CHEMBL320361 26729 18223 TSPO 706 DRUGGABLE GENOME Imidazopyridine acetamide analog 4 26732 18224 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL403989 TG100-801 26733 18225 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME enalapril ENALAPRIL 16627748 26734 18226 APC 324 CLINICALLY ACTIONABLE PKF118-310 14749129 26735 18227 ANO1 55107 ION CHANNEL blocker 178101041 26736 18228 EML4 27436 CLINICALLY ACTIONABLE, KINASE Crizotinib CRIZOTINIB 26775591,27009859,22277784,20979469,22235099,28476735,27354483,27432227,25228534,26698910,21613408,26554404,23344087,21791641,27780853,24675041 26737 18229 POLK 51426 DNA REPAIR, ENZYME NOREPINEPHRINE NOREPINEPHRINE 26739 18230 KMO 8564 DRUGGABLE GENOME, ENZYME Aryl pyrimidine derivative 3 26740 18231 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME JNJ-7706621 JNJ-7706621 26741 18232 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE H-1152 26742 18233 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME CHEMBL395091 ESKETAMINE 26745 18234 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor POZIOTINIB POZIOTINIB 26746 18235 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3545151 CC-223 26747 18236 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CARBAMAZEPINE CARBAMAZEPINE 15565432 26748 18237 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR MEDI5117 COR-001 26749 18238 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE antibody 252166668 OTELIXIZUMAB 26750 18239 F12 2161 DRUGGABLE GENOME, ENZYME, PROTEASE BORTEZOMIB BORTEZOMIB 20875739 26751 18240 TUBB4B 10383 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 26753 18241 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZM-39923 HCL CHEMBL538798 26754 18242 PLD1 5337 ENZYME, DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 12237338 26755 18243 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR LORLATINIB LORLATINIB 25733882,30171048,27401242 26756 18244 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor CHEMBL3545022 ULIXERTINIB 26759 18245 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 223366149 PH-797804 26760 18246 POLK 51426 DNA REPAIR, ENZYME 2,3,4'-TRIHYDROXY-4-METHOXYBENZOPHENONE 2,3,4'-TRIHYDROXY-4-METHOXYBENZOPHENONE 26762 18247 PSMD12 5718 NA inhibitor CHEMBL2103884 OPROZOMIB 26763 18248 MPHOSPH8 54737 NA D-DOPA CHEMBL211670 26764 18249 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CARTEOLOL CARTEOLOL 2903243 26768 18250 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor GDC-0980 APITOLISIB 26770 18251 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PEN-221 26771 18252 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 3-FLUOROEVODIAMINE CHEMBL2171781 22867019 26772 18253 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME activator 53801066 26773 18254 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME amprenavir AMPRENAVIR 26774 18255 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Leucovorin LEUCOVORIN 28784859,27626067,26432108 26775 18256 SMN1 6606 DRUGGABLE GENOME CID 867101 CHEMBL406557 26778 18257 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE IT-141 7-ETHYL-10-HYDROXYCAMPTOTHECIN 26781 18258 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME DNDI1417467 CHEMBL1997335 26782 18259 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE THIOGUANINE THIOGUANINE 26783 18260 PDE4B 5142 DRUGGABLE GENOME, ENZYME PAPAVERINE PAPAVERINE 26785 18261 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR GANODERIC ACID TR GANODERIC ACID TR 22014750 26786 18262 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor BMS-599626 AC-480 26787 18263 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650932 26789 18264 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME MOCETINOSTAT MOCETINOSTAT 23829483,26287310 26790 18265 HTT 3064 DRUGGABLE GENOME TCMDC-125310 CHEMBL582030 26791 18266 TAOK3 51347 DNA REPAIR, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME opioids 30031856 26792 18267 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ISOXSUPRINE ISOXSUPRINE 26793 18268 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME AG-538 CHEMBL56393 26794 18269 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 315661266 26797 18270 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100494 DARUSENTAN 26798 18271 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE buspirone BUSPIRONE 18695978 26799 18272 EPHB2 2048 KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME KO-947 26801 18273 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TYRPHOSTIN A9 TYRPHOSTIN A9 26802 18274 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME sorafenib SORAFENIB 20124951 26803 18275 EML4 27436 CLINICALLY ACTIONABLE, KINASE Alectinib ALECTINIB 27009859,28476735,25393796,26849637,27432227,26682573,25228534,21575866,26698910,23344087 26807 18276 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE STREPTOZOTOCIN STREPTOZOCIN 9394952 26808 18277 POLK 51426 DNA REPAIR, ENZYME REVERSETRIIODOTHYRONINE REVERSETRIIODOTHYRONINE 26809 18278 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor ALVOCIDIB ALVOCIDIB 26810 18279 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR RESVERATROL RESVERATROL 26811 18280 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor 249565722 26812 18281 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL1234354 PF-04691502 26814 18282 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME PMID27828716-Compound-15 26815 18283 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650773 CHEMBL296908 26816 18284 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME E-3810 RABEPRAZOLE SODIUM 26819 18285 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651547 26820 18286 POLK 51426 DNA REPAIR, ENZYME NORDEFRIN NORDEFRIN 26822 18287 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 O-DEMETHYLATED ADAPALENE O-DEMETHYLATED ADAPALENE 26823 18288 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME DINACICLIB DINACICLIB 26824 18289 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545085 XL-228 26826 18290 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ISOETHARINE ISOETHARINE 26827 18291 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650410 IPRATROPIUM 26828 18292 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL101253 VATALANIB 26829 18293 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 178100944 26831 18294 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178102310 26832 18295 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SULFAPHENAZOLE SULFAPHENAZOLE 26833 18296 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DNDI1417400 CHEMBL1362503 26834 18297 RACGAP1 29127 NA FLUORANTHEN-3-YLAMINE CHEMBL103583 26835 18298 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CGP-7930 CHEMBL1256697 26836 18299 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME inhibitor 135650390 INDOMETHACIN 26837 18300 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME GEFITINIB GEFITINIB 26840 18301 DYRK4 8798 ENZYME, KINASE, DRUGGABLE GENOME, TYROSINE KINASE, SERINE THREONINE KINASE TAMATINIB R-406 26841 18302 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor SOPHORETIN QUERCETIN 26842 18303 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antibody VITAXIN ETARACIZUMAB 26844 18304 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201023 ORPHENADRINE HYDROCHLORIDE 26845 18305 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417215 CHEMBL1390650 26846 18306 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Flutamide FLUTAMIDE 26847 18307 STEAP1 26872 TRANSPORTER, DRUGGABLE GENOME RG7450 VANDORTUZUMAB VEDOTIN 24424355 26848 18308 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL1683544 ERIBULIN MESYLATE 26849 18309 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor BELINOSTAT BELINOSTAT 26850 18310 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE blocker 178100974 26853 18311 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME PMID29130358-Compound-Figure10(2a) 26854 18312 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Balixafortide BALIXAFORTIDE 26855 18313 ENOSF1 55556 ENZYME capecitabine CAPECITABINE 17549067,27995989,20714149,27001118,23263912,28347776 26857 18314 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1698 BUPROPION HYDROCHLORIDE 26858 18315 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE ORLISTAT ORLISTAT 26861 18316 KRT6A 3853 NA TD101 26862 18317 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 363894188 26863 18318 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 348353623 26864 18319 IL23A 51561 DRUGGABLE GENOME CNTO 1275 26865 18320 TOP2B 7155 DRUGGABLE GENOME, ENZYME Pefloxacin PEFLOXACIN 26866 18321 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody AV-203 AV-203 26867 18322 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Rogaratinib ROGARATINIB 26868 18323 TRIM24 8805 ENZYME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE 387065618 26869 18324 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME MITOXANTRONE MITOXANTRONE 26870 18325 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE OTSSP167 26871 18326 ORAI2 80228 ION CHANNEL blocker 381118797 26873 18327 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE cisplatin CISPLATIN 21636554 26874 18328 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649715 26876 18329 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ELLIPTECINE ELLIPTECINE 26877 18330 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Panitumumab PANITUMUMAB 26878 18331 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE TRICHLORMETHIAZIDE TRICHLORMETHIAZIDE 26879 18332 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME GSK-2256098 GSK-2256098 26880 18333 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE BORTEZOMIB BORTEZOMIB 20875739 26881 18334 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL ANAVEX 2-73 26883 18335 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 178102323 MLN-8054 26884 18336 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652562 26885 18337 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE ARSENIC TRIOXIDE 16285558 26886 18338 AKR1B1 231 DRUGGABLE GENOME, ENZYME M-16209 26887 18339 TUBA3C 7278 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 26890 18340 PTGS1 5742 ENZYME, DRUGGABLE GENOME BROMFENAC BROMFENAC 26891 18341 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-33 26894 18342 SMN1 6606 DRUGGABLE GENOME DNDI1417701 CHEMBL1326164 26895 18343 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE Anifrolumab ANIFROLUMAB 26897 18344 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME ACRIFLAVINE CHLORIDE ACRIFLAVINE 26898 18345 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CLOTRIMAZOLE CLOTRIMAZOLE 26900 18346 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 310264697 UMBRALISIB 26901 18347 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Anti-MUC1 CAR-T cells 26903 18348 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist 404859012 26907 18349 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL TEMAZEPAM TEMAZEPAM 26912 18350 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 8 26913 18351 GMNN 51053 DRUGGABLE GENOME GNF-PF-3955 CHEMBL605747 26914 18352 CEL 1056 CELL SURFACE, DRUGGABLE GENOME, ENZYME GENISTEIN GENISTEIN 10600647 26916 18353 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DALFAMPRIDINE DALFAMPRIDINE 26917 18354 HDAC11 79885 DRUGGABLE GENOME, ENZYME MGCD-0103 MOCETINOSTAT 26918 18355 COMT 1312 DRUGGABLE GENOME, ENZYME cisplatin CISPLATIN 19898482,28445188,23820299,25141953,24642735,23588304,28448657,28560854,25551397 26919 18356 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BRL-54443 CHEMBL1256797 26920 18357 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL SAFINAMIDE SAFINAMIDE 26921 18358 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Pyrido[1,2-a]indole-1.-carboxylic acid analog 1 26922 18359 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ANTIBIOTIC ANTIBIOTIC 10634213 26924 18360 BAZ2B 29994 NA MERCAPTOPURINE MERCAPTOPURINE 26926 18361 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor GDC-0980 APITOLISIB 26928 18362 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER OFLOXACIN OFLOXACIN 10817732 26929 18363 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR LY2603618 26930 18364 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME AMG 172 26931 18365 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Pyridine derivative 19 26933 18366 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER TAXOL C TAXOL C 16289636 26934 18367 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL587723 AEE-788 26935 18368 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651246 TERGURIDE 26936 18369 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL1908391 MASITINIB 26937 18370 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DROSPIRENONE DROSPIRENONE 26938 18371 CSNK1G3 1456 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME CENISERTIB CENISERTIB 26939 18372 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR EMETINE HYDROCHLORIDE EMETINE HYDROCHLORIDE 26940 18373 GMNN 51053 DRUGGABLE GENOME PERPHENAZINE PERPHENAZINE 26942 18374 F5 2153 DRUGGABLE GENOME THROMBIN THROMBIN 26943 18375 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE SNS-314 SNS-314 26944 18376 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME Patisiran PATISIRAN 26945 18377 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME DNDI1417132 CHEMBL1492017 26946 18378 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ARQ 087 26948 18379 INPP5D 3635 DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE TURNAGAINOLIDE B TURNAGAINOLIDE B 21539394 26950 18380 TARDBP 23435 TUMOR SUPPRESSOR PAXILLINE PAXILLINE 26953 18381 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 26954 18382 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 3R14S-OCHRATOXIN A 3R14S-OCHRATOXIN A 26956 18383 GRK2 156 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, G PROTEIN COUPLED RECEPTOR, ENZYME US9493490, E 26958 18384 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ATRACTYLENOLIDE I ATRACTYLENOLIDE I 22365756 26960 18385 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE ILORASERTIB ILORASERTIB 26961 18386 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME LINURON LINURON 26963 18387 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MIDODRINE MIDODRINE 26964 18388 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor 178103557 SEMAGACESTAT 26965 18389 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4-AMINO-[1,2]NAPHTHOQUINONE 4-AMINO-[1,2]NAPHTHOQUINONE 26966 18390 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 385612197 26968 18391 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHINOMETHIONAT CHINOMETHIONAT 26969 18392 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Mizolastine MIZOLASTINE 26970 18393 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME Labetuzumab I-131 26971 18394 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR crizotinib CRIZOTINIB 26972 18395 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 26973 18396 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Erlotinib ERLOTINIB 27694386,27803065,24101053 26974 18397 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE TAMATINIB R-406 25222877 26977 18398 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 315661328 26979 18399 MAOB 4129 DRUGGABLE GENOME, ENZYME Cyclic peptide derivative 1 26982 18400 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CARBACHOL CARBACHOL 26983 18401 PDE3A 5139 ENZYME, DRUGGABLE GENOME Olprinone OLPRINONE 26984 18402 CBX1 10951 NA NSC-693571 CHEMBL1287983 26985 18403 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DIHYDROERGOTAMINE DIHYDROERGOTAMINE 26986 18404 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL activator 178101088 26987 18405 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SEMAPIMOD SEMAPIMOD 26988 18406 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BKM120 BUPARLISIB 27307593,24265152 26989 18407 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR S-METOLACHLOR S-METOLACHLOR 26990 18408 IL18 3606 DRUGGABLE GENOME COLCHICINE COLCHICINE 15281431 26991 18409 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL NG2-73 ADIPIPLON 26993 18410 TSPO 706 DRUGGABLE GENOME Bidentate pyrazolopyrimidine acetamide analog 4 26994 18411 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650431 ISOPROTERENOL 26995 18412 CD38 952 CELL SURFACE, DRUGGABLE GENOME antibody 252827377 ISATUXIMAB 26996 18413 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 187051794 26998 18414 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER lansoprazole LANSOPRAZOLE 17190370 27000 18415 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE 9-CIS-RETINOIC ACID 12063559 27001 18416 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR cladribine CLADRIBINE 24024897 27003 18417 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL2219422 AFURESERTIB 27005 18418 E2F1 1869 TRANSCRIPTION FACTOR URSODEOXYCHOLIC ACID 15222754 27007 18419 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125298 CHEMBL581152 27008 18420 BMPR1A 657 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 249565835 27009 18421 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL276711 SEMAXANIB 27010 18422 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9707205, 40 27011 18423 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-1947 CHEMBL585591 27012 18424 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125539 CHEMBL533388 27014 18425 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE N-ACETYLGLUCOSAMINE THIAZOLINE CHEMBL257158 20822912 27016 18426 NOTCH3 4854 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor RO4929097 RG-4733 27017 18427 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651424 ACETYLCHOLINE 27020 18428 ATAD5 79915 NA DNDI1417614 CHEMBL1567571 27021 18429 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Benzodihydroisofuran derivative 1 27022 18430 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GW405833 CHEMBL73711 27023 18431 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR TOPOISOMERASE INHIBITORS 1727386 27024 18432 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LY-674 LY-518674 27026 18433 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR carboplatin CARBOPLATIN 19786980,22188361,18347182,21902499,25069034,21057378,29662106,19362955,27498158,21262916,22026922,22329723 27027 18434 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE agonist CHEMBL2107846 DULANERMIN 27028 18435 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR ANTI-ANGIOGENIC AGENTS 15578913 27029 18436 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME ZYDPLA 1 27030 18437 TUBA1C 84790 DRUGGABLE GENOME CHEMBL2108628 PACLITAXEL POLIGLUMEX 27031 18438 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE triamterene TRIAMTERENE 23788015 27032 18439 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME EPO EPOETIN ALFA 9310190 27033 18440 RAMP1 10267 DRUGGABLE GENOME, CELL SURFACE PRAMLINTIDE PRAMLINTIDE 27038 18441 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TRYPTOPHAN TRYPTOPHAN 27040 18442 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME VER-49009 CHEMBL365617 27042 18443 PDE3B 5140 ENZYME, DRUGGABLE GENOME NM-702 27043 18444 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR CAMPTOTHECIN CAMPTOTHECIN 12464623 27044 18445 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 381744939 27045 18446 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-A8 27046 18447 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR AZORUBINE AZORUBINE 27049 18448 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE DASATINIB DASATINIB 22328973,23932362,18938156 27050 18449 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR STAUROSPORINE STAUROSPORINE 15053922 27051 18450 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Aryl alkanolamine derivative 2 27053 18451 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 coumarin COUMARIN 11394901,16679388,10544257,14583682,10923861,9827545,27339126,16041240,15900015,12325023,12844137,9409631,21521021,15993850,11779172,2322567,11278503,11038160 27054 18452 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OLANZAPINE OLANZAPINE 27056 18453 HSPB1 3315 DRUGGABLE GENOME MOMETASONE FUROATE MOMETASONE FUROATE 27057 18454 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METCONAZOLE METCONAZOLE 27058 18455 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OSM-S-55 CHEMBL1363033 27060 18456 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1200782 DEXTROAMPHETAMINE ADIPATE 27061 18457 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME ICA-17043 SENICAPOC 27062 18458 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GW501516 GW501516 27066 18459 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 249565808 27067 18460 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR Siltuximab SILTUXIMAB 27071 18461 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL475251 R-406 27073 18462 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ATORVASTATIN ATORVASTATIN 10559511 27075 18463 POLK 51426 DNA REPAIR, ENZYME PROTOPORPHYRIN DISODIUM PROTOPORPHYRIN DISODIUM 27079 18464 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565799 27081 18465 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody RO5083945 IMGATUZUMAB 27084 18466 TOP2B 7155 DRUGGABLE GENOME, ENZYME ETOPOSIDE ETOPOSIDE 16309315,25945730,26264845,22364746 27085 18467 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565889 27086 18468 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME RG-1530 RG-1530 27087 18469 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR TESTOSTERONE PROPIONATE TESTOSTERONE PROPIONATE 27088 18470 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SILICON PHTHALOCYANINE 4 11121139 27090 18471 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR epinephrine EPINEPHRINE 27091 18472 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE RX-0201 ARCHEXIN 27092 18473 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE activator 135651519 27094 18474 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE HYPOXANTHINE HYPOXANTHINE 16611376 27095 18475 IMPDH1 3614 ENZYME, DRUGGABLE GENOME mycophenolic acid 24220207 27097 18476 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DIPHENYLPYRALINE DIPHENYLPYRALINE 27098 18477 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE 2-Methoxyestradiol 2-METHOXYESTRADIOL 27100 18478 REV3L 5980 DRUGGABLE GENOME, DNA DIRECTED RNA POLYMERASE fluorouracil FLUOROURACIL 27101 18479 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIAMIDE DIAMIDE 27104 18480 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MIDODRINE MIDODRINE 27105 18481 DHODH 1723 DRUGGABLE GENOME, ENZYME leflunomide LEFLUNOMIDE 19207032 27106 18482 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL704 MESALAMINE 27107 18483 GAA 2548 DRUGGABLE GENOME, ENZYME MIGLITOL MIGLITOL 23106358 27109 18484 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYDROXYFLUTAMIDE HYDROXYFLUTAMIDE 27110 18485 SLC38A3 10991 TRANSPORTER 178101351 27111 18486 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE NSAIDS 11813903 27112 18487 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME IPRODIONE IPRODIONE 27114 18488 POLK 51426 DNA REPAIR, ENZYME QUINALIZARIN QUINALIZARIN 27115 18489 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3',5-DIHYDROXYFLAVONE CHEMBL502242 27117 18490 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL598797 CUDC-101 27119 18491 ATXN2 6311 NA DEPHOSTATIN DEPHOSTATIN 27121 18492 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TRETINOIN TRETINOIN 27122 18493 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME GLYCOPEG-GCSF 27123 18494 EIF2AK1 27102 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565848 27124 18495 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR TAMATINIB R-406 27127 18496 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor SONIDEGIB SONIDEGIB 27128 18497 PNP 4860 ENZYME, DRUGGABLE GENOME 2'3'-Dideoxyinosine 27129 18498 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ofatumumab OFATUMUMAB 27131 18499 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200392 DOXYLAMINE SUCCINATE 27132 18500 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME TOFACITINIB TOFACITINIB 26258521 27133 18501 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR DORAMAPIMOD DORAMAPIMOD 27134 18502 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1544 LIOTHYRONINE 27135 18503 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME encorafenib ENCORAFENIB 27137 18504 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE CATECHOL CATECHOL 27139 18505 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor PX-866 SONOLISIB 27140 18506 CA2 760 DRUGGABLE GENOME, ENZYME BRINZOLAMIDE BRINZOLAMIDE 27141 18507 ECE2 9718 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252166873 27143 18508 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 135651285 27144 18509 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DESIPRAMINE DESIPRAMINE 27145 18510 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor 249565618 27147 18511 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL3707249 ASM-024 27148 18512 P2RX4 5025 ION CHANNEL, DRUGGABLE GENOME antagonist 336446929 27149 18513 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PF-562271 PF-00562271 27151 18514 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL ALPRAZOLAM ALPRAZOLAM 27152 18515 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 4-HYDROXYEVODIAMINE CHEMBL2171794 22867019 27153 18516 GMNN 51053 DRUGGABLE GENOME TCMDC-124552 CHEMBL547245 27154 18517 DHFR 1719 DRUGGABLE GENOME, ENZYME 4-HYDROPEROXYCYCLOPHOSPHAMIDE PERFOSFAMIDE 11162315 27155 18518 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE PLX4720 PLX-4720 26351322 27156 18519 CDKN2D 1032 KINASE 5-AZA-2'-DEOXYCYTIDINE 11753657 27157 18520 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME MMV009085 CHEMBL581225 27160 18521 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-123868 CHEMBL548615 27161 18522 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME KRAS G12C INHIBITOR MRTX849 27162 18523 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650678 NADOLOL 27163 18524 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METRIBUZIN METRIBUZIN 27164 18525 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE ILORASERTIB ILORASERTIB 27167 18526 DDAH1 23576 ENZYME inhibitor 252827487 27169 18527 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE FSA2 27172 18528 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING CARBOXYMETHYL-TRIMETHYL-ARSONIUM CARBOXYMETHYL-TRIMETHYL-ARSONIUM 27173 18529 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-601364 CHEMBL1270061 22524450 27175 18530 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR BECLOMETHASONE DIPROPIONATE 9230235 27176 18531 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545285 XL-999 27178 18532 PRKCH 5583 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL494089 GSK-690693 27179 18533 PDE4D 5144 DRUGGABLE GENOME, ENZYME allosteric modulator 385612211 BPN-14770 27180 18534 BMPR1A 657 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 249565801 27182 18535 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 363894211 PEXMETINIB 27183 18536 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE FAS LIGAND 10729215 27184 18537 ATXN2 6311 NA TCMDC-124317 CHEMBL586937 27185 18538 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178102325 PAZOPANIB 27186 18539 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BUSPIRONE BUSPIRONE 27187 18540 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-36398 CHEMBL483206 27188 18541 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR US10174026, Example 99 27189 18542 KEAP1 9817 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor CHEMBL2107333 DIMETHYL FUMARATE 27190 18543 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME Enasidenib ENASIDENIB 28588020,28193778 27191 18544 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3544942 RONICICLIB 27193 18545 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HEXYLRESORCINOL HEXYLRESORCINOL 27195 18546 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR POLYPHENOL 16463383 27196 18547 ATXN2 6311 NA TUBERCIDIN TUBERCIDIN 27197 18548 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000154295 CHEMBL578502 27200 18549 ATAD5 79915 NA CID 649849 CHEMBL405914 27201 18550 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 387065576 27203 18551 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MODUFOLIN ARFOLITIXORIN 27204 18552 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TRASTUZUMAB EMTANSINE 27205 18553 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE TD-1211 AXELOPRAN 27208 18554 USP1 7398 DNA REPAIR, PROTEASE, ENZYME STREPTONIGRIN STREPTONIGRIN 27209 18555 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CSP-1103 27211 18556 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE NITROGEN MUSTARD 12753603 27212 18557 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OKADAIC ACID OKADAIC ACID 22608922 27213 18558 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE SOTRASTAURIN SOTRASTAURIN 27216 18559 TXNRD1 7296 DRUGGABLE GENOME Terpyridineplatinum(II) complexe 1 27217 18560 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1070 NABUMETONE 27218 18561 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE trastuzumab TRASTUZUMAB 18347005,21109570 27219 18562 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor AZD4547 27220 18563 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BROMODIPHENHYDRAMINE BROMODIPHENHYDRAMINE 27221 18564 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MECAMYLAMINE MECAMYLAMINE 22931300 27223 18565 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME L-GLUTAMATE GLUTAMIC ACID 27224 18566 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor 354702259 FUTIBATINIB 27226 18567 ALPI 248 DRUGGABLE GENOME, ENZYME HAEMATOXYLIN HAEMATOXYLIN 27227 18568 MIF 4282 DRUGGABLE GENOME, CELL SURFACE Anti-MIF antibodies 22238348 27228 18569 PDE7A 5150 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200875 FLAVOXATE HYDROCHLORIDE 27229 18570 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME PD-0166285 PD-0166285 27230 18571 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DEOXYVASICINONE DEOXYVASICINONE 27231 18572 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL3544906 BENZPHETAMINE HYDROCHLORIDE 27232 18573 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Phenytoin PHENYTOIN 27233 18574 HDAC11 79885 DRUGGABLE GENOME, ENZYME 2-ENE-VALPROATE CHEMBL117487 17566732 27237 18575 MDM4 4194 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, DRUGGABLE GENOME ALRN-6924 27238 18576 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE AKT INHIBITOR MK2206 23888070,22180495 27240 18577 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3-FORMYLINDOLE 3-FORMYLINDOLE 25458499 27243 18578 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME AT-406 AT-406 21443232 27245 18579 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE PMID27539678-Compound-3 27246 18580 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Cisapride CISAPRIDE 27248 18581 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 REL-CISAPRIDE REL-CISAPRIDE 22931300 27250 18582 KDM4A 9682 DRUGGABLE GENOME, ENZYME QUISQUALATE QUISQUALATE 27251 18583 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE HEREGULIN 16847284 27254 18584 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PENICILLIN V BENZATHINE PENICILLIN V BENZATHINE 27255 18585 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 27257 18586 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR EPROSARTAN EPROSARTAN 27259 18587 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-3467 CHEMBL601774 27260 18588 GMNN 51053 DRUGGABLE GENOME FENDILINE HYDROCHLORIDE FENDILINE HYDROCHLORIDE 27261 18589 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HARMINE HYDROCHLORIDE HARMINE HYDROCHLORIDE 27263 18590 NDUFS3 4722 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545135 NV-128 27264 18591 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200437 QUINIDINE GLUCONATE 27266 18592 BAZ2B 29994 NA TCMDC-123868 CHEMBL548615 27268 18593 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR VITAMIN E 1505665 27269 18594 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Isoquinoline 1,3-dione derivative 1 27270 18595 MPHOSPH8 54737 NA SB-415286 CHEMBL322970 27272 18596 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE Imatinib IMATINIB 27273 18597 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL750 ZONISAMIDE 27275 18598 GMNN 51053 DRUGGABLE GENOME CLOFOCTOL CLOFOCTOL 27276 18599 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE Flecainide FLECAINIDE 27277 18600 GMNN 51053 DRUGGABLE GENOME GEFITINIB GEFITINIB 27278 18601 COL4A1 1282 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 27279 18602 BAZ2B 29994 NA SJ000124275 CHEMBL602150 27280 18603 ST14 6768 ENZYME, DRUGGABLE GENOME, PROTEASE US8569313, Inhibitor 19 27281 18604 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLORHEXIDINE DIACETATE CHLORHEXIDINE DIACETATE 27282 18605 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Antazoline ANTAZOLINE 27283 18606 MAPT 4137 DRUGGABLE GENOME XANTHOANGELOL XANTHOANGELOL 27285 18607 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-13 27286 18608 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL agonist 178101063 27287 18609 ACE2 59272 ENZYME, TRANSPORTER, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, CELL SURFACE, PROTEASE GL1001 ORE-1001 27288 18610 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE HYPERBARIC OXYGEN 15589527 27290 18611 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME TYRPHOSTIN 23 TYRPHOSTIN 23 27291 18612 TSPYL2 64061 NA BROMODEOXYURIDINE 11395479 27292 18613 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME umeclidinium / vilanterol 27293 18614 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME ENASIDENIB ENASIDENIB 28588020,28193778 27296 18615 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 prasugrel PRASUGREL 21828263 27298 18616 SCNN1G 6340 ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE amiloride AMILORIDE 23788015 27299 18617 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ARI-3037MO 27300 18618 ATAD5 79915 NA CP-55940 CP-55940 27301 18619 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME 178101255 27303 18620 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME AR-42 AR-42 27304 18621 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 27305 18622 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 6 27306 18623 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CM-2236 27307 18624 HSPB6 126393 NA AZX-100 AZX-100 27308 18625 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME AST-487 AST-487 27309 18626 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE CHEMOTHERAPY 32068648 27311 18627 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TYRPHOSTIN 1 TYRPHOSTIN 1 27312 18628 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR docetaxel DOCETAXEL 27314 18629 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 27315 18630 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE montelukast MONTELUKAST 18695978 27316 18631 ALOX15B 247 DRUGGABLE GENOME, ENZYME BITHIONOLATE SODIUM BITHIONOLATE SODIUM 27317 18632 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE SP-600125 SP-600125 27318 18633 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Cobimetinib COBIMETINIB 26566875 27319 18634 SGK1 6446 SERINE THREONINE KINASE, KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565720 27320 18635 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE CENISERTIB CENISERTIB 27321 18636 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER terfenadine TERFENADINE 27322 18637 KDM4A 9682 DRUGGABLE GENOME, ENZYME BAS-8770957 CHEMBL500812 27324 18638 HSPB2 3316 KINASE IL-10 INTERLEUKIN-10 11034403 27325 18639 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PROPAZINE PROPAZINE 27326 18640 ABAT 18 DRUGGABLE GENOME, ENZYME L-Alanine L-ALANINE 27327 18641 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 178103525 FLUTAMIDE 27328 18642 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL GABAPENTIN GABAPENTIN 27329 18643 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME PARAPLATIN CARBOPLATIN 27330 18644 NR1D2 9975 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 310264683 27332 18645 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ALEGLITAZAR ALEGLITAZAR 27333 18646 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651298 27335 18647 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME AMPICILLIN TRIHYDRATE AMPICILLIN TRIHYDRATE 27336 18648 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL931 HALOTHANE 27337 18649 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Buparlisib BUPARLISIB 27340 18650 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME DACINOSTAT DACINOSTAT 17956988 27341 18651 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LABETALOL LABETALOL 27342 18652 ALOX5 240 DRUGGABLE GENOME, ENZYME CMI-392 27343 18653 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 667285 CHEMBL267160 27344 18654 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 223366213 RIDAFOROLIMUS 27345 18655 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor PD 0325901 27347 18656 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NEFAZODONE NEFAZODONE 27348 18657 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL329123 ETALOCIB 27350 18658 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE BMS-754807 BMS-754807 19778024 27351 18659 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SJ000044511 CHEMBL592124 27352 18660 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650727 27353 18661 POLB 5423 DNA REPAIR, DRUGGABLE GENOME PINAFIDE PINAFIDE 27354 18662 HK2 3099 ENZYME, KINASE VDA-1102 topical ointment 27355 18663 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ACETAMINOPHEN ACETAMINOPHEN 22931300 27356 18664 TH 7054 ENZYME, DRUGGABLE GENOME METYROSINE METYROSINE 27357 18665 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME N-(4-FLUOROBENZYLCARBAMOTHIOYL)BENZAMIDE CHEMBL1545737 27358 18666 CACNA2D3 55799 ION CHANNEL, DRUGGABLE GENOME celecoxib CELECOXIB 22336956 27359 18667 NEK4 6787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GW441756X GW441756X 27360 18668 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Tasosartan TASOSARTAN 27361 18669 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER amitriptyline AMITRIPTYLINE 24192121,18215618,26704739,22641028 27362 18670 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER LIM-0705 QUERCETIN-3'-O-PHOSPHATE 27364 18671 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR GSK-269962A GSK-269962A 27365 18672 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102225 27367 18673 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR APIGENIN APIGENIN 27368 18674 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GEFITINIB GEFITINIB 27371 18675 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL49642 INDIBULIN 27372 18676 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649789 27373 18677 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME AMD070 MAVORIXAFOR 19640718 27375 18678 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE JNJ-7706621 JNJ-7706621 27376 18679 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE G1T38 LEROCICLIB 27378 18680 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000044511 CHEMBL592124 27379 18681 IDS 3423 ENZYME, DRUGGABLE GENOME IDURONATE-2 SULFATASE 27381 18682 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CRYPTOTANSHINONE CRYPTOTANSHINONE 27382 18683 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE antibody MM-111 MM-111 27384 18684 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BEVACIZUMAB BEVACIZUMAB 23828442 27386 18685 MTRR 4552 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME folic acid 22926161 27387 18686 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TCMDC-123927 CHEMBL531268 27388 18687 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FLUOXETINE FLUOXETINE 22931300 27389 18688 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME 681640 CHEMBL379975 27390 18689 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR warfarin WARFARIN 29298995 27391 18690 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-64 27393 18691 GSTM1 2944 DRUGGABLE GENOME, ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 27785604 27395 18692 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PD173074 22837387,27535980 27396 18693 VKORC1 79001 DRUGGABLE GENOME, ENZYME inhibitor 178103459 WARFARIN 27397 18694 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME DIHYDREXIDINE DIHYDREXIDINE 27399 18695 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor 223366040 27400 18696 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DOBUTAMINE DOBUTAMINE 27401 18697 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1963502 PKI-166 27402 18698 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE MEFENAMIC ACID MEFENAMIC ACID 27403 18699 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GSK2141795 UPROSERTIB 27404 18700 SMYD2 56950 ENZYME, METHYL TRANSFERASE inhibitor 178103600 27406 18701 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PACHYRRIZINE PACHYRRIZINE 27409 18702 MAPT 4137 DRUGGABLE GENOME RACEPINEPHRINE RACEPINEPHRINE 27411 18703 ATAD5 79915 NA GELDANAMYCIN GELDANAMYCIN 27412 18704 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 1302037 27413 18705 SLC1A2 6506 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE 178101410 27415 18706 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL572878 TOZASERTIB 27418 18707 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE Imidamide derivative 1 27420 18708 NUMA1 4926 CLINICALLY ACTIONABLE calcium channel blockers 24192120 27422 18709 GUCY2C 2984 DRUGGABLE GENOME, KINASE SP-333 DOLCANATIDE 27423 18710 ALOX15 246 ENZYME, DRUGGABLE GENOME ETHOPROPAZINE HYDROCHLORIDE ETHOPROPAZINE HYDROCHLORIDE 27424 18711 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor PI-103 PI-103 27425 18712 ABCB11 8647 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CHOLIC ACID CHOLIC ACID 22464344 27426 18713 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME C646 26603525 27427 18714 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PHTHALIC ACID PHTHALIC ACID 27432 18715 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-AMINO-ANTHRAQUINONE CHEMBL84685 27433 18716 GAA 2548 DRUGGABLE GENOME, ENZYME PROTOCATECHUIC ACID PROTOCATECHUIC ACID 27434 18717 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX FLUDARABINE FLUDARABINE 27436 18718 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor PAZOPANIB PAZOPANIB 27438 18719 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Tamibarotene TAMIBAROTENE 27439 18720 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PARAROSANILINE PARAROSANILINE 27442 18721 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-61 27443 18722 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 27444 18723 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID25991433-Compound-J3 27445 18724 MAPKAPK5 8550 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565858 27446 18725 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE 27447 18726 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME P276-00 RIVICICLIB 27448 18727 NPTXR 23467 NA NNZ-2566 27450 18728 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Platinum compounds 29662106 27451 18729 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE AZD0156 AZD-0156 27452 18730 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID28048944-Compound-3 27453 18731 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE PREDNISOLONE PREDNISOLONE 2079995 27454 18732 GSTM1 2944 DRUGGABLE GENOME, ENZYME SULFORAPHANE SULFORAPHANE 16332662 27455 18733 CBX1 10951 NA GNF-PF-1319 CHEMBL235891 27456 18734 IMPDH1 3614 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1456 MYCOPHENOLATE MOFETIL 27457 18735 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ribavirin RIBAVIRIN 20812847 27458 18736 UTRN 7402 NA ENZYME INHIBITOR 15639474 27459 18737 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 381118818 27460 18738 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IRIGINOL HEXAACEATATE IRIGINOL HEXAACEATATE 27461 18739 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CELECOXIB CELECOXIB 27462 18740 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME MAPK INHIBITORS 16170570 27463 18741 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE M2698 MSC-2363318A 27464 18742 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FERROUS SULFATE FERROUS SULFATE 22931300 27468 18743 TARDBP 23435 TUMOR SUPPRESSOR RILUZOLE RILUZOLE 27469 18744 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CD40L 10940895 27470 18745 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PENBUTOLOL PENBUTOLOL 27471 18746 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME E6201 E-6201 24448821,23039341 27472 18747 HTT 3064 DRUGGABLE GENOME OXOPURPUREINE OXOPURPUREINE 27473 18748 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE trametinib TRAMETINIB 27475 18749 PDE10A 10846 ENZYME, DRUGGABLE GENOME Pyrido[3,2-e][1,2,4]triazolo[4,3-a]pyrazine derivative 2 27476 18750 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1963683 TAFLUPROST 27478 18751 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Pyrazolopyridines and imidazopyridine derivative 1 27480 18752 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME inhibitor 404859110 27482 18753 MGA 23269 TRANSCRIPTION FACTOR inhibitor CHEMBL1566 ACARBOSE 27483 18754 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 9-AMINOCAMPTOTHECIN 9-AMINOCAMPTOTHECIN 27484 18755 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651435 TRETINOIN 27485 18756 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL544665 FINGOLIMOD HYDROCHLORIDE 27486 18757 BSG 682 DRUGGABLE GENOME, TRANSPORTER [131I]-Metuximab injection 27487 18758 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME DASATINIB DASATINIB 27488 18759 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME NITRAZEPAM NITRAZEPAM 27489 18760 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CAMPTOTHECIN CAMPTOTHECIN 9918583 27490 18761 PTP4A1 7803 DRUGGABLE GENOME, PROTEIN PHOSPHATASE HALOFUGINONE HALOFUGINONE 16508789 27491 18762 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TOZASERTIB TOZASERTIB 27493 18763 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HESPERETIN HESPERETIN 27494 18764 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649966 27499 18765 KCNJ5 3762 TRANSPORTER, ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME phorbol 12-myristate 13-acetate 27502 18766 ATAD5 79915 NA TCMDC-123951 CHEMBL587849 27503 18767 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE CENISERTIB CENISERTIB 27504 18768 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BENZQUINAMIDE BENZQUINAMIDE 27505 18769 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Dipeptide analog 2 27506 18770 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE pioglitazone PIOGLITAZONE 18695978 27507 18771 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NVP-AUY922 LUMINESPIB 25313505 27508 18772 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200841 PROCAINE HYDROCHLORIDE 27510 18773 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE 2'H,4H-[2,8'-BICHROMEN]-4-ONE 2'H,4H-[2,8'-BICHROMEN]-4-ONE 23600958 27512 18774 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor DANUSERTIB DANUSERTIB 27513 18775 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME GW441756X GW441756X 27514 18776 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KETOCONAZOLE KETOCONAZOLE 27515 18777 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-124317 CHEMBL586937 27517 18778 FST 10468 DRUGGABLE GENOME INHIBINS 10864854 27518 18779 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649827 CHEMBL185951 27520 18780 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME IRX-5183 NRX195183 27522 18781 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL1614713 CC-401 27523 18782 MPHOSPH8 54737 NA EMODIN EMODIN 27524 18783 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 381118864 27526 18784 USP1 7398 DNA REPAIR, PROTEASE, ENZYME LONCHOCARPIC ACID LONCHOCARPIC ACID 27527 18785 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TCMDC-125195 CHEMBL531709 27528 18786 CDKN2D 1032 KINASE IL-4 8760794,14657870 27530 18787 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Nefazodone NEFAZODONE 27531 18788 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-278538 CHEMBL275200 27532 18789 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR MARIJUANA 15857384 27533 18790 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME NSC-234945 CHEMBL260311 27534 18791 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE MDX-1100 ELDELUMAB 27535 18792 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor VELIPARIB VELIPARIB 27536 18793 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Pyrazolodihydropyridine derivative 1 27537 18794 HBB 3043 DRUGGABLE GENOME, ENZYME GBT440 VOXELOTOR 27538 18795 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Phenylpropylamine derivative 2 27539 18796 RAB9A 9367 ENZYME, DRUGGABLE GENOME NSC-636948 CHEMBL1998001 27540 18797 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE GS-5745 ANDECALIXIMAB 27541 18798 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Sodium pyruvate 27543 18799 GMNN 51053 DRUGGABLE GENOME GNF-PF-2383 CHEMBL578915 27545 18800 TUBB 203068 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 27546 18801 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 340590269 27547 18802 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LOPINAVIR LOPINAVIR 27548 18803 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ERGOCALCIFEROL ERGOCALCIFEROL 27550 18804 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SU-11274 CHEMBL261641 17595299 27551 18805 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178103973 NIMESULIDE 27552 18806 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EFAVIRENZ EFAVIRENZ 27553 18807 GMNN 51053 DRUGGABLE GENOME MICHLER'S KETONE MICHLER'S KETONE 27555 18808 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME THYMOSIN BETA-4 27556 18809 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545332 CEP-2563 27558 18810 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135650664 27560 18811 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SR-2640 SR-2640 27561 18812 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIALLYLDISULFIDE DIALLYLDISULFIDE 27563 18813 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Vistusertib VISTUSERTIB 25805799 27568 18814 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 318164806 GSK-1521498 27569 18815 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor 354702261 27571 18816 BAZ2B 29994 NA TRIFLUOPERAZINE HYDROCHLORIDE TRIFLUOPERAZINE HYDROCHLORIDE 27572 18817 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Chlorobenzamide derivative 2 27574 18818 POLI 11201 DNA REPAIR INDIGOTINDISULFONATE INDIGOTINDISULFONATE 27575 18819 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE IONIS-PTP1BRX 27576 18820 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL940 GABAPENTIN 27577 18821 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR BUMETANIDE BUMETANIDE 11807827 27585 18822 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BETANECHOL 27586 18823 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRIPARANOL TRIPARANOL 27588 18824 RACGAP1 29127 NA 3-(PHENYLAMINO)PHENOL CHEMBL1523215 27589 18825 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178100905 27590 18826 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 695758 CHEMBL260028 27592 18827 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME PMID27998201-Compound-5 27594 18828 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE Pyrimido[4,5-d] pyrimidines and pyrido[4,3-d] pyrimidine derivative 1 27595 18829 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545150 AZM-475271 27598 18830 GJA3 2700 ION CHANNEL, TRANSPORTER inhibitor 178101095 OCTANOL 27601 18831 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor BMS-690514 BMS-690514 27602 18832 PTGS1 5742 ENZYME, DRUGGABLE GENOME SUPROFEN SUPROFEN 27603 18833 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME DNDI1417957 CHEMBL1570199 27604 18834 PDE7A 5150 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL628 PENTOXIFYLLINE 27605 18835 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PREDNISONE PREDNISONE 27606 18836 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME AST-487 AST-487 27607 18837 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR EGCG EPIGALOCATECHIN GALLATE 17987129 27610 18838 HEXA 3073 DRUGGABLE GENOME, ENZYME THIOCORALINE THIOCORALINE 27612 18839 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER simeprevir SIMEPREVIR 27613 18840 MAPT 4137 DRUGGABLE GENOME NITAZOXANIDE NITAZOXANIDE 27614 18841 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ELLAGIC ACID ELLAGIC ACID 27615 18842 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DISULFIRAM DISULFIRAM 27616 18843 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Alpelisib ALPELISIB 27974663,27126994,27451907 27617 18844 APBA1 320 NA NSC-50654 CHEMBL1372046 27618 18845 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIFORINE TRIFORINE 27619 18846 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE RX-0201 ARCHEXIN 27621 18847 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR DIMERCAPROL DIMERCAPROL 27624 18848 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR 10-METHOXYLRUTAECARPINE CHEMBL85826 27625 18849 GLS 2744 ENZYME AMPICILLIN AMPICILLIN 27626 18850 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor PD-0332991 PALBOCICLIB 27628 18851 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3039564 IRINOTECAN SUCROSOFATE 27629 18852 SLC12A8 84561 TRANSPORTER, DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 26194362 27632 18853 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER LOBELINE LOBELINE 27634 18854 GMNN 51053 DRUGGABLE GENOME P-CYANOCHALCONE CHEMBL445153 27635 18855 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE DASATINIB DASATINIB 27636 18856 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125140 CHEMBL525106 27638 18857 ITPR1 3708 ION CHANNEL, KINASE, DRUGGABLE GENOME, TRANSPORTER activator 178100946 27639 18858 EIF2AK4 440275 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME olanzapine OLANZAPINE 24751813 27641 18859 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME BLZ-945 27646 18860 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 27647 18861 MAOB 4129 DRUGGABLE GENOME, ENZYME TRYPTAMINE TRYPTAMINE 27651 18862 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME ALSTERPAULLONE ALSTERPAULLONE 27653 18863 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102643 27655 18864 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3544942 RONICICLIB 27656 18865 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PD-0166285 PD-0166285 27657 18866 DTYMK 1841 KINASE 5-FU FLUOROURACIL 15067352 27660 18867 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE SB-203580 SB-203580 27663 18868 EML4 27436 CLINICALLY ACTIONABLE, KINASE AUY922 26698910 27664 18869 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME GP39 7843250 27665 18870 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR GP-120 9878821 27667 18871 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor INIPARIB INIPARIB 27668 18872 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1241153 IBUPROFEN SODIUM 27669 18873 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Unii-I92MU0V408 27670 18874 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE POSIPHEN PHENSERINE, (+)- 27671 18875 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ILORASERTIB ILORASERTIB 27672 18876 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR GNF-PF-4078 CHEMBL584883 27673 18877 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE KTN0073-IgG2 27550450 27674 18878 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR ILORASERTIB ILORASERTIB 27675 18879 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565894 27676 18880 GAA 2548 DRUGGABLE GENOME, ENZYME GZ402666 27677 18881 PLD1 5337 ENZYME, DRUGGABLE GENOME ML272 27679 18882 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ISOFLAVONES 11435074 27682 18883 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Steroid derivative 1 27683 18884 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MRS-2220 CHEMBL74121 27684 18885 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417420 CHEMBL1546223 27685 18886 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE modulator CHEMBL190083 TARENFLURBIL 27686 18887 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME antagonist GDC0917 27689 18888 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 27691 18889 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE SENNOSIDE B SENNOSIDE B 27694 18890 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE CHRYSIN CHRYSIN 23600958 27695 18891 SLC33A1 9197 TRANSPORTER US8592431, 457 27696 18892 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Cyanomethyl pypazole carboxamide derivative 1 27697 18893 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-23 27699 18894 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL622 ETODOLAC 27700 18895 RABEP1 9135 CLINICALLY ACTIONABLE, GROWTH FACTOR valproic acid 28694205 27701 18896 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME JB991 27702 18897 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE CLEMIZOLE CLEMIZOLE 27703 18898 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PAROXETINE HYDROCHLORIDE PAROXETINE HYDROCHLORIDE 27707 18899 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IOBENGUANE IOBENGUANE 27709 18900 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135651043 SIBUTRAMINE 27710 18901 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME SALINE SODIUM CHLORIDE 15641688 27711 18902 GMNN 51053 DRUGGABLE GENOME THIRAM THIRAM 27712 18903 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL2104927 FIGOPITANT 27713 18904 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HOMIDIUM BROMIDE HOMIDIUM BROMIDE 27714 18905 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL ZONISAMIDE ZONISAMIDE 27715 18906 SMN1 6606 DRUGGABLE GENOME 2-ETHYLANTHRAQUINONE CHEMBL42355 27717 18907 IL23A 51561 DRUGGABLE GENOME AMG-139 BRAZIKUMAB 27718 18908 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME APG-1252 27719 18909 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE PD 153035 9096655 27722 18910 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR ARRY-797 ARRY-797 27723 18911 ETS2 2114 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TK216 27724 18912 MAPT 4137 DRUGGABLE GENOME BERBERINE CHLORIDE BERBERINE CHLORIDE 27727 18913 FAAH 2166 ENZYME, DRUGGABLE GENOME Piperazine urea derivative 2 27729 18914 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE SJ000024553 CHEMBL589238 27730 18915 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE TRAMADOL TRAMADOL 27732 18916 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME H2O2 12729926 27733 18917 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Iodine I 131-6-Beta-Iodomethyl-19-Norcholesterol 27734 18918 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OXYPHENCYCLIMINE OXYPHENCYCLIMINE 27735 18919 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 310264777 27736 18920 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL MENTHOL MENTHOL 27739 18921 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RESVERATROL RESVERATROL 27740 18922 APOE 348 DRUGGABLE GENOME TRIAMCINOLONE TRIAMCINOLONE 9150415 27741 18923 TLR7 51284 DRUGGABLE GENOME IMIQUIMOD IMIQUIMOD 27742 18924 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-119915 CHEMBL1481974 27744 18925 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE FLUORESCEIN DIPHOSPHATE FLUORESCEIN DIPHOSPHATE 21482108 27745 18926 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME PMID28270010-Compound-Figure5-2 27746 18927 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Anti-PD-L1 ATEZOLIZUMAB 27748 18928 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIBUTYLTIN-OXIDE TRIBUTYLTIN-OXIDE 27749 18929 GMNN 51053 DRUGGABLE GENOME DNQX DNQX 27751 18930 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AMCINAFIDE AMCINAFIDE 27752 18931 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME LOBARIC ACID LOBARIC ACID 27753 18932 KDM4A 9682 DRUGGABLE GENOME, ENZYME Disulfiram analog 1 27754 18933 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME MGCD-0103 MOCETINOSTAT 27755 18934 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565633 DACTOLISIB 27756 18935 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SUBEROHYDROXAMIC ACID SUBEROHYDROXAMIC ACID 16921367 27758 18936 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME AMORFRUTIN A AMORFRUTIN A 27759 18937 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Paclitaxel PACLITAXEL 25637314,25833835 27760 18938 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PROTOAPIGENONE PROTOAPIGENONE 27761 18939 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BIS(PIPERIDINYLTHIOCARBONYL)DISULFIDE BIS(PIPERIDINYLTHIOCARBONYL)DISULFIDE 27762 18940 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652286 27763 18941 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Clotrimazole CLOTRIMAZOLE 27766 18942 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652673 BUPRENORPHINE 27768 18943 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DAPHNETIN DAPHNETIN 27770 18944 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL ISRADIPINE ISRADIPINE 27772 18945 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 LINEZOLID LINEZOLID 24044938 27773 18946 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1201178 LISDEXAMFETAMINE DIMESYLATE 27775 18947 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 27778 18948 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 COBALT 8577819 27779 18949 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CI-1040 CI-1040 27780 18950 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Aerovant 27781 18951 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME TRIMIPRAMINE TRIMIPRAMINE 27782 18952 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 9 27784 18953 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GNF-PF-2686 CHEMBL578276 27785 18954 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLUDIOXONIL FLUDIOXONIL 27788 18955 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178100245 ETORICOXIB 27789 18956 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-3418 CHEMBL582099 27791 18957 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING BENZO[B]FLUORANTHENE BENZO[B]FLUORANTHENE 27793 18958 BRCA2 675 CLINICALLY ACTIONABLE POL I INHIBITOR CX5461 28211448 27794 18959 BAZ2B 29994 NA LIOTHYRONINE SODIUM LIOTHYRONINE SODIUM 27795 18960 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR E324 E324 27796 18961 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR XANTHOHUMOL XANTHOHUMOL 22111577 27798 18962 GMNN 51053 DRUGGABLE GENOME PIMETHIXENE MALEATE PIMETHIXENE MALEATE 27800 18963 BAZ2B 29994 NA PIROXICAM PIROXICAM 27801 18964 NOS1 4842 DRUGGABLE GENOME, ENZYME RAPAMYCIN SIROLIMUS 16408196 27802 18965 PRKCH 5583 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL565612 SOTRASTAURIN 27804 18966 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650927 ROSIGLITAZONE 27808 18967 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201666 LEPIRUDIN 27809 18968 TARDBP 23435 TUMOR SUPPRESSOR DIMETHYL 2-(2-NITROBENZYLIDENE)MALONATE CHEMBL1569494 27810 18969 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR XL518 COBIMETINIB 27811 18970 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE CAR-GPC3 T cells 27812 18971 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE QUIFENADINE QUIFENADINE 27815 18972 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME ELLIPTECINE ELLIPTECINE 27816 18973 PPIA 5478 DRUGGABLE GENOME, ENZYME inhibitor 135652074 27817 18974 NQO2 4835 DRUGGABLE GENOME, ENZYME DABIGATRAN DABIGATRAN 22494098 27819 18975 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102731 27820 18976 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TRAZODONE TRAZODONE 27822 18977 TMEM167A 153339 NA radiotherapy 28796378 27823 18978 DNER 92737 NA Tetra-hydro-quinoline derivative 4 27825 18979 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE Vorapaxar VORAPAXAR 27826 18980 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 348353617 CEVIMELINE 27828 18981 TMEM97 27346 NA PMID30185082-Compound-63 27830 18982 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE 4-N-BENZYLCYTOSINE CHEMBL2063052 22854677 27831 18983 RACGAP1 29127 NA VU001171 CHEMBL515763 27833 18984 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME TEMOZOLOMIDE TEMOZOLOMIDE 15486188 27835 18985 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A1 27836 18986 CA1 759 DRUGGABLE GENOME, ENZYME ETHOXZOLAMIDE ETHOXZOLAMIDE 27838 18987 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL TRIAZOLAM TRIAZOLAM 27839 18988 EPHB4 2050 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor XL647 TESEVATINIB 27841 18989 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Lenvatinib LENVATINIB 26169970 27842 18990 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER adefovir dipivoxil 27843 18991 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650850 PREDNISOLONE 27844 18992 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-17 27846 18993 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Romidepsin ROMIDEPSIN 27847 18994 CLCN7 1186 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER blocker 178100996 27850 18995 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BAS 01152706 CHEMBL2002487 27851 18996 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR EMETINE HYDROCHLORIDE EMETINE HYDROCHLORIDE 27852 18997 PSME1 5720 NA inhibitor BORTEZOMIB BORTEZOMIB 27853 18998 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PYRIMETHAMINE PYRIMETHAMINE 25984755 27854 18999 RIPK3 11035 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 178102513 PONATINIB 27855 19000 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200472 QUAZEPAM 27856 19001 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE imatinib IMATINIB 28762371 27858 19002 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650894 RENZAPRIDE 27860 19003 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME FLUORESCEIN FLUORESCEIN 27861 19004 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PENTAMIDINE DIISETHIONATE PENTAMIDINE ISETHIONATE 27862 19005 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ARBACLOFEN ARBACLOFEN 27863 19006 POLB 5423 DNA REPAIR, DRUGGABLE GENOME 3,5 DIBROMOTYROSINE DIBROMOTYROSINE 27864 19007 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER cimetidine CIMETIDINE 27865 19008 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ENILCONAZOLE ENILCONAZOLE 27866 19009 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 223366038 LESOGABERAN 27867 19010 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME SUBEROHYDROXAMIC ACID SUBEROHYDROXAMIC ACID 16921367 27869 19011 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Pheniramine PHENIRAMINE 27870 19012 ABCB11 8647 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CYCLOSPORINE CYCLOSPORINE 23129211 27871 19013 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE CHEMBL1714 KETAMINE HYDROCHLORIDE 27872 19014 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2-(ALPHA-NAPHTHOYL)ETHYLTRIMETHYLAMMONIUM IODIDE CHEMBL1255936 27873 19015 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 sevoflurane SEVOFLURANE 9187528 27874 19016 UBE2N 7334 ENZYME, DRUGGABLE GENOME RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 27875 19017 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PROGESTERONE PROGESTERONE 27876 19018 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SCH772984 27312529 27877 19019 CTH 1491 ENZYME AKOS003197197 27878 19020 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL506871 VELIPARIB 27879 19021 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 L-755507 L-755507 27880 19022 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-83217 CHEMBL120806 27881 19023 CP 1356 DRUGGABLE GENOME, ENZYME PENICILLAMINE PENICILLAMINE 11721763 27882 19024 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MERCAPTOPURINE MERCAPTOPURINE 22931300 27883 19025 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-70 27884 19026 CCL5 6352 CELL SURFACE, ENZYME, KINASE, DRUGGABLE GENOME NI-0701 27886 19027 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ERYTHROSINE ERYTHROSINE 27887 19028 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DOCEBENONE DOCEBENONE 27888 19029 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BUTYRYLHYDROXAMIC ACID BUTYRYLHYDROXAMIC ACID 21874153 27891 19030 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Ribociclib Succinate 27892 19031 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE PEGINTERFERON ALFA-2A 27893 19032 ICAM3 3385 DRUGGABLE GENOME VITAMIN D 10891379 27894 19033 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME RABEPRAZOLE RABEPRAZOLE 27896 19034 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-348401 CHEMBL515505 27897 19035 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-735465 CHEMBL261440 27899 19036 RGS4 5999 DRUGGABLE GENOME 5,4'-DIHYDROXYFLAVONE CHEMBL484662 27900 19037 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUTORPHANOL BUTORPHANOL 27901 19038 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMINOPURVALANOL AMINOPURVALANOL 27902 19039 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL3545073 AMA0076 27904 19040 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Aromatic and heteroaryl compound 1 27906 19041 POLI 11201 DNA REPAIR NSC-74859 CHEMBL477936 27908 19042 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE CI-1040 CI-1040 27821489 27909 19043 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Fluorinated donepezil derivative 1 27911 19044 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE amiloride AMILORIDE 23788015 27912 19045 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 19 27914 19046 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 315661095 27916 19047 MTTP 4547 DRUGGABLE GENOME Granotapide GRANOTAPIDE 27918 19048 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME pamidronate PAMIDRONIC ACID 18594024 27920 19049 RRM2 6241 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1750 CLOFARABINE 27921 19050 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 178103637 27923 19051 EPHX1 2052 ENZYME, DRUGGABLE GENOME phenprocoumon PHENPROCOUMON 21057703 27925 19052 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME PMID25468267-Compound-55 27926 19053 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PHENSERINE PHENSERINE 27927 19054 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME SILYBIN B SILYBIN B 23401473 27928 19055 AKR1B10 57016 DRUGGABLE GENOME, ENZYME TOLRESTAT TOLRESTAT 21561086 27929 19056 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RS-39604 CHEMBL66114 27930 19057 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Doxil DOXIL 16243804 27933 19058 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL OXAZEPAM OXAZEPAM 27935 19059 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRICLOSAN TRICLOSAN 27937 19060 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE FUTIBATINIB FUTIBATINIB 31109923 27938 19061 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE EGFR/IGFR tandem adnectin 27939 19062 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650387 IMPROGAN 27940 19063 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PENCONAZOLE PENCONAZOLE 27942 19064 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BEXAROTENE BEXAROTENE 27943 19065 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK711701A GSK-711701A 27945 19066 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AZD4547 26351320,23082000,27550940,22837387,26936917,27179038,27535980,28108151,26359452 27946 19067 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ULIPRISTAL ULIPRISTAL 27947 19068 BAZ2B 29994 NA DNDI1318477 CHEMBL428064 27948 19069 CCR6 1235 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR SJ000044511 CHEMBL592124 27950 19070 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CLOBETASOL PROPIONATE 11555673 27951 19071 POLK 51426 DNA REPAIR, ENZYME TYRPHOSTIN 25 TYRPHOSTIN 25 27952 19072 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR METHANANDAMIDE METHANANDAMIDE 27954 19073 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR BYL719 ALPELISIB 27312529 27955 19074 SMN2 6607 DRUGGABLE GENOME NITAZOXANIDE NITAZOXANIDE 27956 19075 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL THIOCOLCHICOSIDE THIOCOLCHICOSIDE 27957 19076 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE GSK933776A 24255592 27958 19077 ACADM 34 ENZYME HORMONES 9164869 27959 19078 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103502 BENZOLAMIDE 27960 19079 GART 2618 ENZYME, DRUGGABLE GENOME PEMETREXED PEMETREXED 27961 19080 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX PLUMBAGIN PLUMBAGIN 22483392 27962 19081 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME ABT-737 ABT 737 22386982,22747598 27963 19082 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Pyrazolo[1,5-a]-1,3,5-triazine derivative 1 27965 19083 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 310264780 27966 19084 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201729 DRONEDARONE HYDROCHLORIDE 27968 19085 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL193240 ROFLUMILAST 27970 19086 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE CYC-116 CYC-116 27971 19087 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor 249565694 CHIR-99021 27972 19088 PTGIS 5740 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 252827453 27975 19089 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565581 AFURESERTIB 27976 19090 NPC1L1 29881 DRUGGABLE GENOME, TRANSPORTER pravastatin PRAVASTATIN 19752398 27977 19091 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE COPTIS 9875508 27978 19092 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER EMTRICITABINE EMTRICITABINE 17172311 27979 19093 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME ASP-015K PEFICITINIB 27980 19094 ATAD5 79915 NA SJ000082805 CHEMBL531043 27981 19095 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CTCE-9908 CTCE-9908 27982 19096 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 178103354 27983 19097 KDM4A 9682 DRUGGABLE GENOME, ENZYME 2-HYDROXYESTRADIOL CHEMBL467987 27987 19098 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE 7-azaindole derivative 4 27988 19099 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME N,N'-DIPHENYL-GUANIDINE CHEMBL77675 27990 19100 POLI 11201 DNA REPAIR AMINACRINE HYDROCHLORIDE AMINACRINE HYDROCHLORIDE 27992 19101 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200798 TRAZODONE HYDROCHLORIDE 27994 19102 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE JNJ-7706621 JNJ-7706621 27996 19103 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME LINIFANIB LINIFANIB 27998 19104 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CB-03-01 CLASCOTERONE 27999 19105 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME PAZOPANIB PAZOPANIB 28001 19106 COMT 1312 DRUGGABLE GENOME, ENZYME TOLCAPONE TOLCAPONE 28002 19107 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RESACTIN A RESACTIN A 28004 19108 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 178103269 28006 19109 PDE4B 5142 DRUGGABLE GENOME, ENZYME Ronomilast 28007 19110 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103704 BIPERIDEN 28009 19111 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLORMIDAZOLE CHLORMIDAZOLE 28011 19112 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1416917 CHEMBL1335833 28012 19113 MMP14 4323 PROTEASE, DRUGGABLE GENOME, ENZYME CARMINIC ACID CARMINIC ACID 28014 19114 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ILORASERTIB ILORASERTIB 28015 19115 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE NSC-95397 CHEMBL429095 28017 19116 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 252827367 OZANIMOD 28018 19117 TSPO 706 DRUGGABLE GENOME Fludiazepam FLUDIAZEPAM 28019 19118 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Anti-N3pG-Abeta antibody 28020 19119 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE fentanyl FENTANYL 26771271,30281924 28022 19120 CCNA2 890 DRUGGABLE GENOME, KINASE ETHINYL ESTRADIOL 9806355 28023 19121 METAP2 10988 ENZYME, DRUGGABLE GENOME, KINASE, PROTEASE Beloranib BELORANIB 28024 19122 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME METHOTRIMEPRAZINE LEVOMEPROMAZINE 28025 19123 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-59 28026 19124 BCAR1 9564 KINASE celecoxib CELECOXIB 22336956 28027 19125 MAPK6 5597 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE sorafenib SORAFENIB 20124951 28028 19126 UBE2N 7334 ENZYME, DRUGGABLE GENOME METHYLBENZETHONIUM CHLORIDE METHYLBENZETHONIUM CHLORIDE 28029 19127 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 252166846 28030 19128 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME CID 1245272 CHEMBL408850 28031 19129 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID25656651-Compound-34c 28032 19130 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Tucatinib TUCATINIB 28053022 28033 19131 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 28034 19132 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE TIROFIBAN TIROFIBAN 28035 19133 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX SJ000128325 CHEMBL602718 28036 19134 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-119915 CHEMBL1481974 28040 19135 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor CHEMBL1980297 ILORASERTIB 28041 19136 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR PROPRANOLOL PROPRANOLOL 12691286 28042 19137 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650508 28043 19138 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 VALPROIC ACID VALPROIC ACID 22931300 28044 19139 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR THUNBERGINOL A THUNBERGINOL A 28047 19140 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ROSIGLITAZONE MALEATE ROSIGLITAZONE MALEATE 28049 19141 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LAK 10431685 28051 19142 CDK12 51755 KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR, SERINE THREONINE KINASE inhibitor 375973251 28054 19143 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE LY3023414 SAMOTOLISIB 27439478 28055 19144 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE Biphenyl carboxylic acid derivative 1 28057 19145 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX RUTIN RUTIN 25496805 28059 19146 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 318164813 28060 19147 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE LUMACAFTOR LUMACAFTOR 26041577 28062 19148 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALPHA 28063 19149 NGFR 4804 CELL SURFACE, DRUGGABLE GENOME LM11A-31 28064 19150 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor CHEMBL932 DIPYRIDAMOLE 28066 19151 ALOX15 246 ENZYME, DRUGGABLE GENOME BISABOLOL BISABOLOL 28068 19152 GP6 51206 CELL SURFACE, KINASE PR-15 28071 19153 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor PKI-587 GEDATOLISIB 28072 19154 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PRAVASTATIN PRAVASTATIN 8312689 28073 19155 ATAD5 79915 NA TYRPHOSTIN AG-1478 TYRPHOSTIN AG-1478 28081 19156 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE diuretics 22543981 28083 19157 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 385612199 DAROLUTAMIDE 28084 19158 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor VATALANIB VATALANIB 28086 19159 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 28087 19160 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RIBAVIRIN RIBAVIRIN 28090 19161 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 vinblastine VINBLASTINE 9187528 28092 19162 TK1 7083 ENZYME, KINASE, DRUGGABLE GENOME TK-DLI 28093 19163 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PYRACLOSTROBIN PYRACLOSTROBIN 28094 19164 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 223366147 ORANTINIB 28096 19165 ALDH3A1 218 DRUGGABLE GENOME, ENZYME ANTABUSE ANTABUSE 7907815 28097 19166 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE OXALIPLATIN OXALIPLATIN 25788273 28098 19167 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ALSTERPAULLONE ALSTERPAULLONE 28099 19168 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE allosteric modulator 315661298 28100 19169 PDE4B 5142 DRUGGABLE GENOME, ENZYME AN-2898 28101 19170 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CLOBAZAM CLOBAZAM 28102 19171 MAT1A 4143 ENZYME, DRUGGABLE GENOME ANTISENSE OLIGONUCLEOTIDES 9537246 28106 19172 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124328 CHEMBL532143 28107 19173 SFN 2810 DRUGGABLE GENOME IMATINIB IMATINIB 21962576 28108 19174 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE blocker 178101019 28109 19175 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CD20-CART 28110 19176 ATAD5 79915 NA CID 893238 CHEMBL473735 28111 19177 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103658 FLUOROMETHOLONE 28112 19178 PTGES 9536 DRUGGABLE GENOME, ENZYME PMID28627961-Compound-22 28114 19179 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Imidazole derivative 8 28115 19180 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ALPROSTADIL ALPROSTADIL 28119 19181 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME vancomycin VANCOMYCIN 32439433 28120 19182 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652041 28121 19183 H2AX 3014 NA TESTOSTERONE TESTOSTERONE 8810267 28122 19184 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 381118809 28124 19185 LTF 4057 CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, PROTEASE Talactoferrin TALACTOFERRIN ALFA 28125 19186 PSMB9 5698 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL2103884 OPROZOMIB 28126 19187 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE PF-562271 PF-00562271 28127 19188 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200472 QUAZEPAM 28128 19189 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Oxetane 3,3-dicarboxamide compound 2 28130 19190 HLA-DQA1 3117 CLINICALLY ACTIONABLE interferon beta-1b 21502966 28131 19191 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME BENZOFURAN BENZOFURAN 28133 19192 AKR1B1 231 DRUGGABLE GENOME, ENZYME Ranirestat RANIRESTAT 28135 19193 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE esomeprazole ESOMEPRAZOLE 18695978 28136 19194 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX KAEMPFERIDE KAEMPFERIDE 25190466 28137 19195 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME PMID25468267-Compound-47 28139 19196 NR1D1 9572 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME GSK-4112 GSK-4112 23656296 28142 19197 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AURIN AURIN 28148 19198 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MERCURIC CHLORIDE MERCURIC CHLORIDE 28149 19199 GLS 2744 ENZYME MYRICETIN MYRICETIN 28150 19200 RPS6KA2 6196 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME BI-D1870 CHEMBL573107 28151 19201 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AMG 337 27196782,26432108 28152 19202 MAPT 4137 DRUGGABLE GENOME GNF-PF-1295 CHEMBL579837 28153 19203 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-2559 CHEMBL583584 28154 19204 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Endoxifen ENDOXIFEN 28155 19205 POLB 5423 DNA REPAIR, DRUGGABLE GENOME METHYLDOPA (RACEMIC) METHYLDOPA (RACEMIC) 28157 19206 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE NANAOMYCIN NANAOMYCIN 28158 19207 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME RISEDRONIC ACID RISEDRONIC ACID 28159 19208 NOTCH2 4853 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE inhibitor RO4929097 RG-4733 28160 19209 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TCMDC-123951 CHEMBL587849 28161 19210 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor SELUMETINIB SELUMETINIB 28162 19211 POLK 51426 DNA REPAIR, ENZYME L-NOREPINEPHRINE L-NOREPINEPHRINE 28164 19212 KCNH8 131096 DRUGGABLE GENOME, ION CHANNEL blocker 135652729 28166 19213 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651259 THIORIDAZINE 28169 19214 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MELPHALAN MELPHALAN 28170 19215 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 348353617 CEVIMELINE 28171 19216 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135649824 MESALAMINE 28173 19217 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE CP-339818 CP-339818 28174 19218 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Momelotinib MOMELOTINIB 24398328,21926964 28175 19219 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 178100879 28177 19220 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SB-431542 SB-431542 28178 19221 POR 5447 ENZYME, DRUGGABLE GENOME zidovudine ZIDOVUDINE 22960662 28179 19222 BAZ2B 29994 NA SJ000089001 CHEMBL591618 28180 19223 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-19063 CHEMBL1310138 28182 19224 ATP1A2 477 ENZYME, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME inhibitor CHEMBL3545057 ACETYLDIGITOXIN 28183 19225 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 329968373 28185 19226 BAZ2B 29994 NA GNF-PF-2491 CHEMBL577851 28187 19227 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CINOBUFOTALIN CINOBUFOTALIN 28189 19228 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIRIBEDIL PIRIBEDIL 28190 19229 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GNF-PF-3023 CHEMBL535331 28192 19230 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL377300 BRIVANIB 28193 19231 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROMETHAZINE PROMETHAZINE 28194 19232 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME AG-1879 CHEMBL406845 28195 19233 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR inhibitor 252827512 CHEMBL481422 28197 19234 EPHX1 2052 ENZYME, DRUGGABLE GENOME AR9281 AR9281 28198 19235 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR PROMAZINE HYDROCHLORIDE PROMAZINE HYDROCHLORIDE 28199 19236 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor GSK2636771 GSK-2636771 28201 19237 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE DACTOLISIB DACTOLISIB 28202 19238 HBB 3043 DRUGGABLE GENOME, ENZYME NSC-119236 CHEMBL458765 28204 19239 TOP2B 7155 DRUGGABLE GENOME, ENZYME Pixantrone PIXANTRONE 28205 19240 KDM4A 9682 DRUGGABLE GENOME, ENZYME 2',3,4-TRIHYDROXYCHALCONE CHEMBL339587 28206 19241 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE omeprazole OMEPRAZOLE 18695978 28207 19242 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C15 28208 19243 ATAD2 29028 NUCLEAR HORMONE RECEPTOR, ENZYME inhibitor 252166841 28209 19244 GCLM 2730 ENZYME CAROTENOID 15657364 28211 19245 CBX1 10951 NA CEFOTAXIME CEFOTAXIME 28212 19246 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE FDG FLUDEOXYGLUCOSE-F18 7884509,12900743 28214 19247 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 178101843 28215 19248 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DNDI1417025 CHEMBL1320453 28216 19249 EGLN2 112398 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2338329 ROXADUSTAT 28218 19250 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE PRT062607 28219 19251 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL315985 ESLICARBAZEPINE 28220 19252 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR CUDC-427 GDC-0917 28221 19253 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 sertraline SERTRALINE 9187528 28222 19254 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SJ000044511 CHEMBL592124 28223 19255 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR peginterferon alfa-2b 28224 19256 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TYRPHOSTIN 23 TYRPHOSTIN 23 28225 19257 PDE4A 5141 DRUGGABLE GENOME, ENZYME DENBUFYLLINE DENBUFYLLINE 28226 19258 GSTM1 2944 DRUGGABLE GENOME, ENZYME UVB 12083949 28227 19259 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER MS-209 10049760 28228 19260 TARDBP 23435 TUMOR SUPPRESSOR EPIANDROSTERONE EPIANDROSTERONE 28229 19261 HR 55806 NUCLEAR HORMONE RECEPTOR Repirinast REPIRINAST 28230 19262 POLK 51426 DNA REPAIR, ENZYME FURAMIDINE FURAMIDINE 28231 19263 KDM6B 23135 ENZYME inhibitor 310264759 28232 19264 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 28233 19265 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-44 28234 19266 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME (-)-GRACILIOETHER B CHEMBL2178596 22934537 28236 19267 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR RIZATRIPTAN RIZATRIPTAN 28237 19268 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SANGUINARINE SULFATE SANGUINARINE SULFATE 28238 19269 IKBKG 8517 KINASE, DRUGGABLE GENOME artesunate ARTESUNATE 28241 19270 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PYRIDOSTIGMINE PYRIDOSTIGMINE 22931300 28242 19271 GUCY1B1 2983 DRUGGABLE GENOME activator CHEMBL6622 ISOSORBIDE DINITRATE 28243 19272 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ETOPOSIDE ETOPOSIDE 9389690 28244 19273 ABAT 18 DRUGGABLE GENOME, ENZYME TIAGABINE TIAGABINE 28245 19274 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE GNF-PF-159 CHEMBL599924 28246 19275 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME RESVERATROL RESVERATROL 28247 19276 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Monoaryl-1,2-diamine derivative 1 28248 19277 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NIFUROXAZIDE NIFUROXAZIDE 28250 19278 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 328083527 BAY-1161909 28251 19279 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MECLIZINE MECLIZINE 22931300 28252 19280 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME conjugated estrogens 11477075 28253 19281 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GS-9820 ACALISIB 28254 19282 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000147784 CHEMBL590186 28255 19283 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100765 VALSARTAN 28257 19284 APC 324 CLINICALLY ACTIONABLE Binimetinib BINIMETINIB 26206338 28258 19285 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE nalidixic acid 4190560 28259 19286 DHODH 1723 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL960 LEFLUNOMIDE 28260 19287 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TRETINOIN TRETINOIN 28262 19288 TOP2B 7155 DRUGGABLE GENOME, ENZYME F-14512 28264 19289 CST5 1473 PROTEASE INHIBITOR, DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 28268 19290 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE EGFR antibody 27196767 28269 19291 TOP2B 7155 DRUGGABLE GENOME, ENZYME GSK2140944 GEPOTIDACIN 28271 19292 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor GDC-0973 COBIMETINIB 28272 19293 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135650814 ALPROSTADIL 28273 19294 PTGS1 5742 ENZYME, DRUGGABLE GENOME ACETAMINOPHEN ACETAMINOPHEN 19053765 28274 19295 TUBB3 10381 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 28275 19296 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME fluvastatin FLUVASTATIN 28277 19297 HSPA4 3308 NA Enkastim-ev 28279 19298 UMPS 7372 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE fluorouracil FLUOROURACIL 20647221,16818689 28282 19299 PDE4D 5144 DRUGGABLE GENOME, ENZYME Ronomilast 28283 19300 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE N-ETHYL-N-NITROSOUREA 12838503 28284 19301 ALOX15 246 ENZYME, DRUGGABLE GENOME allosteric modulator 315661226 28286 19302 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyrrolo-pyridine derivative 1 28288 19303 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ANGUSTIBALIN ANGUSTIBALIN 28290 19304 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28270010-Compound-Figure5-1 28293 19305 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649768 28294 19306 ATAD5 79915 NA SULFURETIN SULFURETIN 28295 19307 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TDR78277 CHEMBL1308346 28297 19308 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE VORAPAXAR VORAPAXAR 28299 19309 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 7A-METHYL-19-NORTESTOSTERONE,MENT 28301 19310 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME INSULIN GLULISINE 28303 19311 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE FASUDIL FASUDIL 28305 19312 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME RG-1530 RG-1530 28306 19313 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR antagonist AT-406 AT-406 28307 19314 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PHA-767491 CHEMBL225519 28308 19315 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TEMSIROLIMUS TEMSIROLIMUS 28310 19316 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Trastuzumab TRASTUZUMAB 17936563,21676217,26759238,24470511,28784859,27140927,27108243,26880266,26296355,23801166,26469692,24691421,24606768,24982373,20728210,17679724,27626067,23948973,28167203,23940356,24742739,28539475,26245675,19874578,23220880,21558396,25370464,26432108,24300914,27697991,26243863 28312 19317 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE SUNITINIB SUNITINIB 19861435,21969494,23375402,22357254 28314 19318 PSMD2 5708 NA inhibitor CHEMBL325041 BORTEZOMIB 28315 19319 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102240 FK453 28316 19320 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CARFILZOMIB CARFILZOMIB 28317 19321 RPS6KA5 9252 DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE GSK-269962A GSK-269962A 28318 19322 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME antidepressants 28320 19323 PDE3B 5140 ENZYME, DRUGGABLE GENOME US9388139, 12 28321 19324 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE warfarin WARFARIN 28322 19325 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID29757691-Compound-2a 28323 19326 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ACTH CORTICOTROPIN 11956163 28324 19327 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME 5-AZACYTIDINE AZACITIDINE 7511991 28327 19328 DYNC2H1 79659 CLINICALLY ACTIONABLE etoposide ETOPOSIDE 21118971 28328 19329 SCG5 6447 CLINICALLY ACTIONABLE, DRUGGABLE GENOME TGFBETA1 14709802 28330 19330 ALOX15 246 ENZYME, DRUGGABLE GENOME DAPHNETIN DAPHNETIN 28332 19331 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR JUGLONE JUGLONE 28333 19332 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 328083511 TARLOXOTINIB 28334 19333 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178102747 28335 19334 NDUFB10 4716 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 28338 19335 AQP1 358 ION CHANNEL, DRUGGABLE GENOME inhibitor 178100948 28339 19336 KMT2C 58508 ENZYME, CLINICALLY ACTIONABLE, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, DRUG RESISTANCE LETROZOLE LETROZOLE 29755131 28340 19337 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME TPCK TPCK 28341 19338 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER clopidogrel CLOPIDOGREL 26362473,24262617,24762860,28135763,17112805,21831410,28914344,25060201,28378058,20801498,27380588,25542807,19106083,25850030,23726091,23364775,22045970,23056288,22940005,21806387,24535487,28358842,28589365,25430046,20650435,21918510,23150151,29397568,20801494,22723959,22190063,22028352,22285300,22990067,22624833 28342 19339 TUBB4B 10383 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 28343 19340 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE GEMCITABINE GEMCITABINE 23390248 28345 19341 SLC28A1 9154 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE zidovudine ZIDOVUDINE 22960662 28347 19342 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 7,8,2'-TRIHYDROXYFLAVONE CHEMBL244707 28348 19343 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PIRETANIDE PIRETANIDE 28350 19344 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL2105759 BARICITINIB 28352 19345 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME PF-562271 PF-00562271 28354 19346 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TCMDC-125602 CHEMBL580183 28356 19347 GNL3 26354 NA epirubicin EPIRUBICIN 28357 19348 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PF-562271 PF-00562271 28359 19349 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor TAK-733 TAK-733 28360 19350 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE N/A 28361 19351 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Anti-CD19 and Anti-CD20 CAR-T Cells 28362 19352 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TCMDC-124377 CHEMBL531269 28363 19353 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Panobinostat PANOBINOSTAT 22693356,19490892,26725216 28364 19354 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME IMATINIB IMATINIB 28366 19355 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL NITRAZEPAM NITRAZEPAM 28367 19356 CTSC 1075 ENZYME, DRUGGABLE GENOME, PROTEASE CALCIUM GLUCONATE 18822840 28368 19357 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE Lumefantrine LUMEFANTRINE 28370 19358 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE BMS-754807 BMS-754807 21148487 28371 19359 GJB5 2709 ION CHANNEL inhibitor 178100972 CARBENOXOLONE 28375 19360 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME KARANJIN KARANJIN 28376 19361 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ondansetron ONDANSETRON 21596874 28377 19362 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE ANISTREPLASE ANISTREPLASE 28380 19363 TXNRD1 7296 DRUGGABLE GENOME Palmarumycin derivative 3 28381 19364 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE K-756 27196752 28382 19365 NDUFAF4 29078 NA inhibitor CHEMBL3545135 NV-128 28383 19366 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL448 PENTOBARBITAL 28384 19367 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR DOXORUBICIN DOXORUBICIN 16905201 28385 19368 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE 681640 CHEMBL379975 28387 19369 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor PONATINIB PONATINIB 28388 19370 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME NSC-71033 CHEMBL116548 28389 19371 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 10-METHOXYLRUTAECARPINE CHEMBL85826 28390 19372 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 11 28391 19373 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TOLONIUM CHLORIDE TOLONIUM CHLORIDE 28392 19374 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TORSEMIDE TORSEMIDE 22931300 28393 19375 AXIN1 8312 CLINICALLY ACTIONABLE, KINASE (+/-)-HYDNOCARPIN CHEMBL91638 24018191 28397 19376 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545083 RGB-286638 28399 19377 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1201066 VENLAFAXINE HYDROCHLORIDE 28400 19378 KIF11 3832 DRUGGABLE GENOME 4SC-205 28402 19379 RGS4 5999 DRUGGABLE GENOME BEMESETRON BEMESETRON 28403 19380 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BRONOPOL BRONOPOL 28404 19381 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Phenylpropylamine derivative 4 28405 19382 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor DABRAFENIB MESYLATE 28406 19383 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME cetuximab CETUXIMAB 26812186,22537608,26162609,25183481,23071293,22734028,23324806,26371285,27897268,25210463,26438111,20978259,23090619,24727325 28407 19384 RGS4 5999 DRUGGABLE GENOME RS-16566 CHEMBL145725 28408 19385 TNKS 8658 DRUGGABLE GENOME, ENZYME PMID27841036-Compound-37 28409 19386 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 187051823 28410 19387 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 16 28411 19388 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 187051818 28412 19389 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME NITRAZEPAM NITRAZEPAM 28415 19390 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OBE-101 19300572 28417 19391 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE TAE-684 TAE-684 28418 19392 DIABLO 56616 NA TRAIL 10950947,12941843,15137068,12670926 28419 19393 TJP1 7082 KINASE, TRANSCRIPTION FACTOR GENISTEIN GENISTEIN 10330056 28420 19394 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CO1686 27252416 28424 19395 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL2109431 LENZILUMAB 28425 19396 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MEDROXYPROGESTERONE ACETATE MEDROXYPROGESTERONE ACETATE 28427 19397 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 249565658 CHEMBL259026 28428 19398 TUBB 203068 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 28429 19399 VDAC2 7417 NA TCDD 17998243 28432 19400 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR METHYLENE BLUE CHLORIDE HYDRATE METHYLENE BLUE 28433 19401 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE RETINOIC ACID 10950817 28434 19402 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE CODEINE CODEINE 28437 19403 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 18 28438 19404 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR TRICHOSTATIN TRICHOSTATIN 21055848,16921367,19966789,19385600,24074025 28440 19405 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE atorvastatin ATORVASTATIN 18997459 28441 19406 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Pregnenolone PREGNENOLONE 28444 19407 TSPO 706 DRUGGABLE GENOME Benzothiazepine analog 5 28445 19408 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CYC-116 CYC-116 20462263 28446 19409 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE GSK-269962A GSK-269962A 28447 19410 NOS1 4842 DRUGGABLE GENOME, ENZYME RESINIFERATOXIN RESINIFERATOXIN 8595209 28448 19411 FURIN 5045 ENZYME, PROTEASE, CELL SURFACE, DRUGGABLE GENOME US9266828, E 28449 19412 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-1211 CHEMBL600968 28450 19413 PLAUR 5329 DRUGGABLE GENOME, ENZYME, CELL SURFACE G-CSF FILGRASTIM 15747404 28452 19414 TXNRD1 7296 DRUGGABLE GENOME Metal complex derivative 2 28453 19415 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME 178101458 28457 19416 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649682 28458 19417 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178103994 DACOMITINIB 28459 19418 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DANAZOL DANAZOL 28460 19419 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DICYCLOMINE DICYCLOMINE 28461 19420 MAP3K1 4214 CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 223366167 E-6201 28464 19421 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565760 28465 19422 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SBI-0640726 20531415,26603897 28466 19423 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ING-1 ING-1 28467 19424 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL3545207 EVENAMIDE 28468 19425 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000071821 CHEMBL589924 28470 19426 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor 252166503 SAFINAMIDE 28471 19427 ICAM3 3385 DRUGGABLE GENOME inhibitor CHEMBL2109481 ICM3 28472 19428 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ISOSPAGLUMIC ACID ISOSPAGLUMIC ACID 28473 19429 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SJ000044511 CHEMBL592124 28476 19430 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774822-Compound-Figure2Example1-1right 28477 19431 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME antisense oligonucleotide LY2181308 GATAPARSEN 28478 19432 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200809 AZELASTINE HYDROCHLORIDE 28479 19433 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545421 DERAZANTINIB 28481 19434 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME RANTES 10679062 28482 19435 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-78 CHEMBL579318 28485 19436 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE MESALAMINE MESALAMINE 28486 19437 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR radiotherapy 25026457,28796378 28488 19438 TUBB 203068 DRUGGABLE GENOME DAVLB-HYDRAZIDE 22814904 28489 19439 PDK4 5166 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME CPI-613 28490 19440 POLB 5423 DNA REPAIR, DRUGGABLE GENOME HAEMATOXYLIN HAEMATOXYLIN 28492 19441 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 354702298 28493 19442 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ATL1102 28494 19443 PDE10A 10846 ENZYME, DRUGGABLE GENOME DIPYRIDAMOLE DIPYRIDAMOLE 28495 19444 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME PMID28621580-Compound-WO2014079545C69 28497 19445 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL296419 ASTEMIZOLE 28498 19446 METAP2 10988 ENZYME, DRUGGABLE GENOME, KINASE, PROTEASE XMT-1107 28500 19447 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE MCI-186 EDARAVONE 28501 19448 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR MMV085203 CHEMBL586031 28503 19449 DNER 92737 NA Isoxazole-based bicyclic compound 12 28504 19450 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALCITRIOL CALCITRIOL 28506 19451 PDE4A 5141 DRUGGABLE GENOME, ENZYME IC-485 28508 19452 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL blocker 178100875 PICROTOXIN 28511 19453 ALB 213 TRANSPORTER, DRUGGABLE GENOME [19F]-HALOPERIDOL [19F]-HALOPERIDOL 28512 19454 ALOX15 246 ENZYME, DRUGGABLE GENOME 2',4'-DIHYDROXYCHALCONE 2',4'-DIHYDROXYCHALCONE 28514 19455 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME ERBITUX ERBITUX 12850474 28515 19456 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 252166507 28516 19457 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178100975 28518 19458 ALOX15 246 ENZYME, DRUGGABLE GENOME Triazole derivative 3 28519 19459 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME KX-01 ointment 28520 19460 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TRICETIN TRICETIN 28521 19461 RALBP1 10928 TRANSPORTER, ABC TRANSPORTER carbamazepine CARBAMAZEPINE 21738081 28522 19462 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR antagonist FULVESTRANT FULVESTRANT 28524 19463 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE EMD 1204831 25326232 28525 19464 SMN1 6606 DRUGGABLE GENOME CHRYSIN CHRYSIN 28526 19465 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING VINORELBIN DITARTRATE VINORELBINE TARTRATE 28528 19466 ATAD5 79915 NA NITROBENZYLMERCAPTOPURINE RIBONUCLEOSIDE NITROBENZYLMERCAPTOPURINE RIBONUCLEOSIDE 28529 19467 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-Table1Example30 28531 19468 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TAMATINIB R-406 28533 19469 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 4-PHENOXYPHENOL CHEMBL224318 28534 19470 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PMID28048944-Compound-3 28535 19471 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Pyrrolo-pyridinone derivative 6 28536 19472 CCNB1 891 DRUGGABLE GENOME PROTOAPIGENONE PROTOAPIGENONE 28538 19473 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR raloxifene RALOXIFENE 28539 19474 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE MIDOSTAURIN MIDOSTAURIN 27355533 28540 19475 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL1908391 MASITINIB 28542 19476 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-872 CHEMBL600342 28544 19477 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME RTX 9374538 28545 19478 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME ONO-1301 28547 19479 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER epirubicin EPIRUBICIN 28549 19480 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME ARGATROBAN ARGATROBAN 28550 19481 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ZINC 03369470 CHEMBL599013 28551 19482 TNFRSF9 3604 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE CD137 CAR-T Cell 28552 19483 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL1201748 CABAZITAXEL 28555 19484 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000128325 CHEMBL602718 28557 19485 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PMID25726713-Compound-47 28558 19486 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME ETOPOSIDE ETOPOSIDE 11391599 28559 19487 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Sonidegib SONIDEGIB 26124204 28561 19488 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545324 RG-7666 28562 19489 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL2338329 ROXADUSTAT 28564 19490 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor 178103126 28565 19491 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE REL-3,4-DICAFFEOYLQUINIC ACID CHEMBL249448 22921742 28566 19492 GLS 2744 ENZYME GALLIC ACID GALLIC ACID 28567 19493 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CS1229 28568 19494 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE LIF 7782459 28569 19495 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CLOTIAZEPAM CLOTIAZEPAM 28570 19496 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-47 28571 19497 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Doxorubicin DOXORUBICIN 28572 19498 GAK 2580 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor HTS-466284 CHEMBL261454 19035792 28575 19499 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE SB-220025 SB-220025 28577 19500 NPHS1 4868 NA losartan LOSARTAN 28578 19501 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 315661216 PLX8394 28581 19502 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ELLIPTECINE ELLIPTECINE 28582 19503 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME AMENTOFLAVONE AMENTOFLAVONE 28584 19504 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AG-537 CHEMBL67535 28585 19505 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AMITRIPTYLINE AMITRIPTYLINE 22931300 28586 19506 ATAD5 79915 NA GNF-PF-3756 CHEMBL597035 28587 19507 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor BOSUTINIB BOSUTINIB 28588 19508 MUC16 94025 DRUGGABLE GENOME DIFFERENTIATING AGENTS 1720110 28589 19509 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL44657 ETOPOSIDE 28590 19510 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME US9346821, B-13 28591 19511 DHFR 1719 DRUGGABLE GENOME, ENZYME PRALATREXATE PRALATREXATE 28592 19512 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CRIZOTINIB CRIZOTINIB 26729443,21716144,31584608,25971938,25922291,22162573,31416808,31809977,25971939,21623265,27325282,31932802,25232318,26892698,23729478,26547802,30339198,31391294 28593 19513 KDM4A 9682 DRUGGABLE GENOME, ENZYME DIPROTIN A DIPROTIN A 28594 19514 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NALBUPHINE NALBUPHINE 28597 19515 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE antibody MAPATUMUMAB MAPATUMUMAB 28600 19516 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL12 DIAZEPAM 28603 19517 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MYCOPHENOLIC ACID MYCOPHENOLIC ACID 28604 19518 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649809 28606 19519 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR EPINEPHRINE EPINEPHRINE 28607 19520 XDH 7498 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1467 ALLOPURINOL 28608 19521 TUBB3 10381 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 28609 19522 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ACRIDIN-1-YLAMINE CHEMBL146525 28610 19523 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ESTRIOL E3 28611 19524 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE NSC-95397 CHEMBL429095 28613 19525 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE 178101752 28614 19526 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-123868 CHEMBL548615 28617 19527 TXNRD1 7296 DRUGGABLE GENOME 4-aryl quinol derivative 5 28618 19528 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AG-1879 CHEMBL406845 28619 19529 CSNK2A2 1459 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME, TRANSCRIPTION FACTOR US8940736, 6 28620 19530 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650038 28622 19531 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME ethanol ALCOHOL 28624 19532 IMPA1 3612 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200826 LITHIUM CARBONATE 28625 19533 EPHX1 2052 ENZYME, DRUGGABLE GENOME cisplatin CISPLATIN 24533712 28626 19534 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Thalidomide THALIDOMIDE 28627 19535 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CURCUMIN CURCUMIN 25753330 28628 19536 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CHEMBL407 FLUMAZENIL 28629 19537 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME TROGLITAZONE TROGLITAZONE 14977862 28630 19538 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE FALNIDAMOL FALNIDAMOL 28631 19539 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2364626 RALIMETINIB 28632 19540 ESRRG 2104 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650324 CHEMBL193836 28633 19541 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-145 28634 19542 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AG-490 CHEMBL56543 28635 19543 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME DIPHENYLUREA DIPHENYLUREA 28636 19544 FOXO1 2308 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR cyclophosphamide CYCLOPHOSPHAMIDE 28638 19545 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME PMID27539678-Compound-7 28639 19546 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 315661235 NALDEMEDINE 28640 19547 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL564829 MILCICLIB 28641 19548 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Ponatinib PONATINIB 26270481 28642 19549 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ERLOTINIB ERLOTINIB 28644 19550 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HONOKIOL HONOKIOL 20695472 28645 19551 TOP2B 7155 DRUGGABLE GENOME, ENZYME Teniposide TENIPOSIDE 28646 19552 PTGS2 5743 DRUGGABLE GENOME, ENZYME Eicosapentaenoic acid/docosa-hexaenoic acid 28647 19553 TNFRSF12A 51330 DRUGGABLE GENOME Enavatuzumab ENAVATUZUMAB 28648 19554 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1201470 HYDROCODONE POLISTIREX 28649 19555 ALPL 249 ENZYME, DRUGGABLE GENOME 2-AMINOPHENOXAZINONE CHEMBL146710 28650 19556 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650161 28651 19557 TXNRD1 7296 DRUGGABLE GENOME Palmarumycin derivative 1 28652 19558 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AMG 337 26432108 28654 19559 IL1A 3552 CELL SURFACE, DRUGGABLE GENOME HYDROXYCHLOROQUINE HYDROXYCHLOROQUINE 8336306 28655 19560 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE E6201 E-6201 23039341 28656 19561 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-125296 CHEMBL311489 28658 19562 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AZD6482 AZD-6482 26563132 28660 19563 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor DACTOLISIB DACTOLISIB 28661 19564 GMNN 51053 DRUGGABLE GENOME PENTETIC ACID PENTETIC ACID 28662 19565 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ACY-957 25605023 28663 19566 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TYRPHOSTIN 47 TYRPHOSTIN 47 28664 19567 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER carvedilol CARVEDILOL 28665 19568 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 223366077 RGB-286638 28666 19569 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL3301604 RALINEPAG 28667 19570 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-119889 CHEMBL516616 28668 19571 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CARBOSULFAN CARBOSULFAN 28669 19572 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME CGS-15943 CGS-15943 28670 19573 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GDC-0077 GDC-0077 28671 19574 GMNN 51053 DRUGGABLE GENOME MICONAZOLE NITRATE MICONAZOLE NITRATE 28674 19575 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL2103852 CROLIBULIN 28675 19576 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME bevacizumab BEVACIZUMAB 29871907 28677 19577 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-659162 CHEMBL471005 28679 19578 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLOROPHENOTHANE CHLOROPHENOTHANE 28681 19579 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor REGORAFENIB REGORAFENIB 28682 19580 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR modulator CHEMBL260538 ULIPRISTAL ACETATE 28683 19581 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME lisinopril LISINOPRIL 28684 19582 NOS1 4842 DRUGGABLE GENOME, ENZYME GSPE 16555001 28685 19583 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER RESERPINE RESERPINE 28686 19584 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Sulfonamide derivative 18 28687 19585 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE XL418 XL-418 28688 19586 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME OXALIPLATIN OXALIPLATIN 15545975,14985457 28691 19587 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Procaterol PROCATEROL 28692 19588 CA2 760 DRUGGABLE GENOME, ENZYME ACETAZOLAMIDE ACETAZOLAMIDE 28694 19589 MAOB 4129 DRUGGABLE GENOME, ENZYME Benzylcinnamate 28695 19590 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME V3381 INDANTADOL 28697 19591 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-50 28699 19592 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME CLX-0921 CLX-0921 28700 19593 SMN2 6607 DRUGGABLE GENOME 7-METHOXY-BAPTIGENIN CHEMBL583578 28703 19594 IFNG 3458 DRUGGABLE GENOME Fumaric acid 28704 19595 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-1477 CHEMBL582675 28706 19596 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1051 LATANOPROST 28707 19597 IMPDH1 3614 ENZYME, DRUGGABLE GENOME VX-148 28709 19598 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Doxil DOXIL 21216929 28710 19599 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE GO-6976 GO-6976 28712 19600 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME IL-1 8698619 28713 19601 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 328083459 28715 19602 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE SORAFENIB SORAFENIB 21482694 28719 19603 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Pazopanib + Tyverb/Tykerb 28720 19604 REV1 51455 NA cisplatin CISPLATIN 28721 19605 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NANDROLONE NANDROLONE 28722 19606 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102290 AT-7519 28723 19607 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SPLITOMICIN SPLITOMICIN 28724 19608 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2103831 NAPROXCINOD 28725 19609 PPP3CA 5530 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME VOCLOSPORIN VOCLOSPORIN 28726 19610 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME TAMATINIB R-406 28727 19611 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure3-Lycojaponicumin B 28728 19612 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 22931300 28729 19613 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3350 CHEMBL600747 28731 19614 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamide derivative 26 28732 19615 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR EGCG EPIGALOCATECHIN GALLATE 16950787 28733 19616 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 315661265 28737 19617 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 354702288 LEVOSALBUTAMOL 28738 19618 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CAPSAZEPINE CAPSAZEPINE 28740 19619 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor MASITINIB MASITINIB 28741 19620 POLK 51426 DNA REPAIR, ENZYME ZINC 03369470 CHEMBL599013 28742 19621 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124518 CHEMBL527584 28743 19622 IFNGR2 3460 CLINICALLY ACTIONABLE, DRUGGABLE GENOME INTERFERON GAMMA-1B 28744 19623 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GW0742 CHEMBL38508 28745 19624 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417011 CHEMBL1386434 28746 19625 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Sulfatinib SURUFATINIB 28747 19626 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL494089 GSK-690693 28750 19627 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NSC-125296 CHEMBL311489 28752 19628 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ORTHOTOLIDINE ORTHOTOLIDINE 28753 19629 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE MAPK INHIBITORS 16170570 28754 19630 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIBENZOYLMETHANE DIBENZOYLMETHANE 28756 19631 GCLC 2729 DRUGGABLE GENOME, ENZYME CISPLATIN CISPLATIN 9660546 28757 19632 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZO[B]FLUORANTHENE BENZO[B]FLUORANTHENE 28758 19633 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N/A 28762 19634 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE IMATINIB MESYLATE 16205964,12910520 28763 19635 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-2A, RECOMBINANT 28766 19636 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 354702237 LANRAPLENIB 28772 19637 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27551786-Compound-IV 28773 19638 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor TIVANTINIB TIVANTINIB 28775 19639 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist,antagonist 135650312 28776 19640 FGB 2244 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, FIBRINOGEN, DRUGGABLE GENOME ALFIMEPRASE ALFIMEPRASE 28777 19641 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PROTON PUMP INHIBITOR 16815316 28778 19642 ASXL1 171023 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR Azacitidine AZACITIDINE 25224413 28779 19643 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2109623 STX-100 28780 19644 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME EFLORNITHINE EFLORNITHINE 28783 19645 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME SOTRASTAURIN SOTRASTAURIN 28784 19646 ENPP2 5168 ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING (S)-CARBA CYCLIC-PHOSPHATIDIC ACID CHEMBL1630084 21051230 28786 19647 MAPT 4137 DRUGGABLE GENOME GUTHION GUTHION 28787 19648 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MANZAMINE A MANZAMINE A 16872140 28789 19649 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 187051822 28791 19650 SMN2 6607 DRUGGABLE GENOME GNF-PF-1872 CHEMBL600103 28792 19651 TDO2 6999 ENZYME, DRUGGABLE GENOME HYDROGEN PEROXIDE 17212352 28793 19652 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor AZD8055 AZD-8055 28794 19653 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME BI-11634 28795 19654 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GOSSYPOL GOSSYPOL 3158419 28798 19655 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HOMIDIUM BROMIDE HOMIDIUM BROMIDE 28799 19656 DHFR 1719 DRUGGABLE GENOME, ENZYME inhibitor 178103737 DIFLUNISAL 28800 19657 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ILOPROST ILOPROST 28801 19658 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE BECAPLERMIN BECAPLERMIN 28802 19659 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME CART-meso cells 28804 19660 SLC29A4 222962 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER metformin METFORMIN 22722338 28805 19661 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1416955 CHEMBL1327172 28806 19662 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE RANTES 9174593 28807 19663 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 mephenytoin MEPHENYTOIN 9187528 28808 19664 HSPA4 3308 NA PHOTOSENSITIZERS 8625311 28810 19665 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Pindolol PINDOLOL 28811 19666 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor SELUMETINIB SELUMETINIB 28812 19667 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 28813 19668 PGAP6 58986 NA remifentanil REMIFENTANIL 29207912 28815 19669 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE DEXAMETHASONE DEXAMETHASONE 7670964 28819 19670 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PRACINOSTAT PRACINOSTAT 28821 19671 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE N/A 19584151,25681512,22504380,19478385,25749173,26947875,26861460,25760429 28822 19672 PSMD5 5711 NA inhibitor CARFILZOMIB CARFILZOMIB 28824 19673 TUBA1A 7846 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 28826 19674 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Vilanterol VILANTEROL 28828 19675 SMN1 6606 DRUGGABLE GENOME SU-4312 CHEMBL328710 28829 19676 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178103954 ABEMACICLIB 28830 19677 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Entrectinib ENTRECTINIB 28832 19678 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE NERATINIB NERATINIB 28833 19679 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor LGX818 ENCORAFENIB 28834 19680 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 28835 19681 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE NAVITOCLAX NAVITOCLAX 28837 19682 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor 178103777 INAMRINONE 28838 19683 MAP2K5 5607 KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor TRAMETINIB TRAMETINIB 28839 19684 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE BAY1179470 28840 19685 ITPR1 3708 ION CHANNEL, KINASE, DRUGGABLE GENOME, TRANSPORTER antagonist 178101161 28841 19686 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650627 28845 19687 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 4 28846 19688 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BAY-613606 CHEMBL541400 28848 19689 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Savolitinib SAVOLITINIB 28644771,27694386,25779944,28396313 28850 19690 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME QUAZEPAM QUAZEPAM 28851 19691 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL calcium channel blockers 16610939 28853 19692 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME IRIGINOL HEXAACEATATE IRIGINOL HEXAACEATATE 28854 19693 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR 6-HYDROXYDOPAMINE 16770736 28856 19694 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PONATINIB PONATINIB 20513156 28859 19695 LPAR5 57121 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 329968439 28860 19696 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME doxorubicin DOXORUBICIN 27234217 28861 19697 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 223365984 LUCITANIB 28863 19698 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist 135650586 28864 19699 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX CUDRAFLAVONE B CUDRAFLAVONE B 24901948 28865 19700 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GNF-PF-763 CHEMBL1576338 28867 19701 PDF 64146 DRUGGABLE GENOME Meprobamate MEPROBAMATE 28868 19702 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FAMPROFAZONE FAMPROFAZONE 28869 19703 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MAL formulation 28874 19704 BAZ2B 29994 NA 2-PYRIDYLKETONE THIOPHENECARBOXYL HYDRAZONE CHEMBL255068 28875 19705 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TYRPHOSTIN AG-835 CHEMBL261557 28876 19706 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-37 28877 19707 POLK 51426 DNA REPAIR, ENZYME NORSTICTIC ACID NORSTICTIC ACID 28878 19708 HPGDS 27306 ENZYME, DRUGGABLE GENOME inhibitor 178103274 CHEMBL574003 28881 19709 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME EDROPHONIUM EDROPHONIUM 28882 19710 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE PROSTAGLANDIN E1 7822278 28884 19711 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME DIBROMOACETIC ACID DIBROMOACETIC ACID 28887 19712 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 328083448 28888 19713 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 381118861 28891 19714 TSPYL1 7259 NA prednisolone PREDNISOLONE 28892 19715 MAPT 4137 DRUGGABLE GENOME 4-METHOXYDALBERGIONE 4-METHOXYDALBERGIONE 28894 19716 EPHA3 2042 ENZYME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565850 28895 19717 ATAD5 79915 NA SJ000072340 CHEMBL592813 28896 19718 POLI 11201 DNA REPAIR SULOCHRIN SULOCHRIN 28897 19719 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE DOVITINIB DOVITINIB 28898 19720 HLA-DQB1 3119 CLINICALLY ACTIONABLE amoxicillin AMOXICILLIN 10535882,30664875 28902 19721 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BETULINIC ACID BETULINIC ACID 18842418 28903 19722 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PHENYLBUTYRYLHYDROXAMIC ACID PHENYLBUTYRYLHYDROXAMIC ACID 21874153 28904 19723 GMNN 51053 DRUGGABLE GENOME DNDI1417827 CHEMBL1363249 28906 19724 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PARAMETHASONE ACETATE PARAMETHASONE ACETATE 28907 19725 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID25656651-Compound-46 28908 19726 NOS2 4843 DRUGGABLE GENOME, ENZYME ANTIDEPRESSANTS 16401669 28909 19727 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME ERLOTINIB ERLOTINIB 28910 19728 CBX1 10951 NA APTIGANEL APTIGANEL 28911 19729 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR nortriptyline NORTRIPTYLINE 19641488 28912 19730 UGT2B7 7364 DRUGGABLE GENOME aprepitant APREPITANT 26053558 28913 19731 ATAD5 79915 NA CALYCOSIN CALYCOSIN 28914 19732 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME RG-1530 RG-1530 28915 19733 IMPDH2 3615 DRUGGABLE GENOME, ENZYME Mycophenolate mofetil 28918 19734 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR US9359293, TM 28919 19735 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651029 28921 19736 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135651325 28922 19737 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME DIAZOXIDE DIAZOXIDE 16271703 28923 19738 CCNA2 890 DRUGGABLE GENOME, KINASE tamoxifen TAMOXIFEN 24622579 28924 19739 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PSEUDOEPHEDRINE PSEUDOEPHEDRINE 28926 19740 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor HESPERADIN HESPERADIN 19035792 28927 19741 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 VANIPREVIR VANIPREVIR 19841155 28928 19742 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR STI-571 IMATINIB 11368438,11234890 28929 19743 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LEUCOVORIN LEUCOVORIN 11977552,12576451 28931 19744 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME PMID26161698-Compound-34 28932 19745 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CHLOPHEDIANOL CHLOPHEDIANOL 28933 19746 DROSHA 29102 NA mercaptopurine MERCAPTOPURINE 24614921 28934 19747 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PRO22 topical gel 28935 19748 TUBA1C 84790 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 28936 19749 GBA 2629 DRUGGABLE GENOME, ENZYME DNQX DNQX 28937 19750 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-638080 CHEMBL136344 28938 19751 GMNN 51053 DRUGGABLE GENOME METHYLDOPA METHYLDOPA 28939 19752 TUBB 203068 DRUGGABLE GENOME BAL-101553 LISAVANBULIN 28942 19753 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1200363 PENBUTOLOL SULFATE 28943 19754 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200654 BENOXINATE HYDROCHLORIDE 28944 19755 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR ERLOTINIB ERLOTINIB 28945 19756 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR SB-220025 SB-220025 28947 19757 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-2950 CHEMBL602807 28950 19758 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GW1929 CHEMBL434063 28952 19759 PTGS2 5743 DRUGGABLE GENOME, ENZYME lumiracoxib LUMIRACOXIB 19602986 28954 19760 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME prednisone PREDNISONE 16044099 28955 19761 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-123927 CHEMBL531268 28956 19762 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR vincristine VINCRISTINE 24141364 28957 19763 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL113461 TEDISAMIL 28961 19764 ACVR2B 93 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME antibody 249565766 BIMAGRUMAB 28963 19765 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker CHEMBL2107762 NERISPIRDINE 28964 19766 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-PHENYLPHENOL 2-PHENYLPHENOL 28967 19767 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Sodium Nitrite 28969 19768 USP1 7398 DNA REPAIR, PROTEASE, ENZYME BRILLIANT GREEN OXALATE BRILLIANT GREEN OXALATE 28971 19769 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 1-BENZYLMALEIMIDE CHEMBL388979 28972 19770 CD38 952 CELL SURFACE, DRUGGABLE GENOME CAR-T cells targeting CD38 28973 19771 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Temozolomide TEMOZOLOMIDE 28974 19772 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Doxercalciferol DOXERCALCIFEROL 28975 19773 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GAMBOGIC AMIDE GAMBOGIC AMIDE 17911251 28976 19774 GUCY1A2 2977 ENZYME, DRUGGABLE GENOME NITRIC OXIDE 28977 19775 XDH 7498 DRUGGABLE GENOME, ENZYME Azole benzene derivative 4 28978 19776 RORB 6096 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, KINASE US9598431, 2 28979 19777 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 5,7-DIHYDROXYISOFLAVONE 5,7-DIHYDROXYISOFLAVONE 28980 19778 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PURPURIN PURPURIN 28981 19779 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME ZM-447439 CHEMBL202721 28982 19780 LAMP1 3916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE DIMETHYL SULFOXIDE 2243101 28985 19781 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CANRENONE CANRENONE 28987 19782 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME PHLORETIN PHLORETIN 28988 19783 PTGS2 5743 DRUGGABLE GENOME, ENZYME FLURBIPROFEN FLURBIPROFEN 28989 19784 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 178100454 28990 19785 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor CHEMBL608533 MIDOSTAURIN 28993 19786 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 178102681 WORTMANNIN 28994 19787 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 178102428 28995 19788 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Alogliptin ALOGLIPTIN 28997 19789 LAG3 3902 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE FS118 28999 19790 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28117607-Compound-5 29000 19791 TH 7054 ENZYME, DRUGGABLE GENOME METHADONE METHADONE 6125371 29001 19792 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AMCINAFIDE AMCINAFIDE 29002 19793 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL1922094 APITOLISIB 29003 19794 SMN2 6607 DRUGGABLE GENOME GNF-PF-2812 CHEMBL125044 29004 19795 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Piperazine derivative 7 29005 19796 NR1D2 9975 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 310264682 SR9009 29006 19797 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME PACLITAXEL PACLITAXEL 11800022 29007 19798 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME LY411575 26855149 29009 19799 NELFCD 51497 KINASE Thiazides, plain 29010 19800 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE IBUPROFEN IBUPROFEN 30683736 29014 19801 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PMID29671355-Compound-31 29015 19802 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CLIOQUINOL CLIOQUINOL 29016 19803 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE LY-255283 LY-255283 29018 19804 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 7 29019 19805 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 135652718 STRYCHNINE 29020 19806 MAPKAPK5 8550 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE GW843682X GW843682X 29023 19807 USP1 7398 DNA REPAIR, PROTEASE, ENZYME NANAOMYCIN NANAOMYCIN 29024 19808 KDM4A 9682 DRUGGABLE GENOME, ENZYME CRYPTOTANSHINONE CRYPTOTANSHINONE 29025 19809 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GDC0879 19276360 29026 19810 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565685 AR-12 29027 19811 MPHOSPH8 54737 NA RITANSERIN RITANSERIN 29028 19812 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FUMAGILLIN FUMAGILLIN 29029 19813 BAZ2B 29994 NA MMV006389 CHEMBL586000 29031 19814 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL969 PRAZEPAM 29032 19815 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-55 29033 19816 RORB 6096 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, KINASE US9598431, 1 29035 19817 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CYCLOBENZAPRINE HYDROCHLORIDE CYCLOBENZAPRINE HYDROCHLORIDE 29036 19818 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE PH-794428 29037 19819 HEBP1 50865 DRUGGABLE GENOME Benzo[d]oxazole derivative 1 29038 19820 FURIN 5045 ENZYME, PROTEASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178103178 29039 19821 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME IFOSFAMIDE IFOSFAMIDE 8621235 29040 19822 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE CI-1040 CI-1040 29041 19823 KDM4A 9682 DRUGGABLE GENOME, ENZYME NITRILOTRIACETIC ACID NITRILOTRIACETIC ACID 29044 19824 ALOX15 246 ENZYME, DRUGGABLE GENOME PURPURIN PURPURIN 29045 19825 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor 348353640 29046 19826 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL545315 CANERTINIB DIHYDROCHLORIDE 29047 19827 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 318164856 29048 19828 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 252166689 29050 19829 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE brivanib BRIVANIB 20124951 29052 19830 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL544665 FINGOLIMOD HYDROCHLORIDE 29053 19831 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME PINAFIDE PINAFIDE 29054 19832 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650033 BUPRANOLOL 29055 19833 HSPA4 3308 NA THIABENDAZOLE THIABENDAZOLE 11226373 29057 19834 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL1201740 NILOTINIB HYDROCHLORIDE MONOHYDRATE 29060 19835 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ethambutol ETHAMBUTOL 20941486 29062 19836 CAMK1D 57118 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME ENTRECTINIB ENTRECTINIB 29063 19837 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1201022 PHENAZOPYRIDINE HYDROCHLORIDE 29064 19838 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX OUABAIN OUABAIN 29065 19839 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650577 MEDROXYPROGESTERONE ACETATE 29066 19840 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DIPHENIDOL DIPHENIDOL 29067 19841 CD200 4345 CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1743067 SAMALIZUMAB 29072 19842 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE RDEA119 27821489 29073 19843 COL18A1 80781 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 29075 19844 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor ARRY-380 TUCATINIB 29077 19845 CYP27B1 1594 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 deferasirox DEFERASIROX 30651574 29078 19846 ALOX15B 247 DRUGGABLE GENOME, ENZYME PICEATANNOL PICEATANNOL 29079 19847 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BI-87E7 CHEMBL523200 29081 19848 ATXN2 6311 NA CYCLOSPORINE CYCLOSPORINE 29082 19849 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CLOFIBRATE CLOFIBRATE 16680159 29083 19850 SMN1 6606 DRUGGABLE GENOME CID 670282 CHEMBL260213 29084 19851 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Beta Blocking Agents 15864115,20643254,15861037,16815314,16153393,20352314,12709726,12921807,15735607,18075464,12844134,22543981,11052857,16189366,22617224,11787477,17496726,14534524,21311897,14502278,28351962,20235788,16402084 29085 19852 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME CLOMIPRAMINE CLOMIPRAMINE 29086 19853 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME GENERIC 18691996 29089 19854 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135651491 29090 19855 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR HYDROGEN PEROXIDE 11409888 29091 19856 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 29098 19857 GMNN 51053 DRUGGABLE GENOME CID 100335 CHEMBL1520346 29099 19858 LPAR2 9170 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 178100856 29100 19859 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE SEMUSTINE SEMUSTINE 29101 19860 EPHX2 2053 DRUGGABLE GENOME, ENZYME FULVESTRANT FULVESTRANT 23684894 29102 19861 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE norfloxacin NORFLOXACIN 29105 19862 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SU5402 23175443,23597562,21119661 29107 19863 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE NORETHISTERONE ACETATE 7450248 29108 19864 POLK 51426 DNA REPAIR, ENZYME NSC-228155 CHEMBL505670 29110 19865 RAD50 10111 CLINICALLY ACTIONABLE, KINASE, DNA REPAIR IRINOTECAN IRINOTECAN 24934408 29112 19866 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 2-ACETYLAMINOFLUORENE 2-ACETYLAMINOFLUORENE 29113 19867 KDM4A 9682 DRUGGABLE GENOME, ENZYME OLEOYL DOPAMINE OLEOYL DOPAMINE 29114 19868 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CARBENDAZIM CARBENDAZIM 29115 19869 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR TRAMETINIB TRAMETINIB 25673644,25899310,24982505 29116 19870 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4464 CHEMBL600692 29117 19871 TSPO 706 DRUGGABLE GENOME PMID27599163-Compound-79 29119 19872 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL activator 135650743 29120 19873 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651154 29121 19874 HNF1A 6927 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Norleucine NORLEUCINE 29122 19875 BCHE 590 DRUGGABLE GENOME, ENZYME Di-substituted piperidine derivative 2 29123 19876 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 3,4-METHYLENEDIOXYB-NITROSTYRENE CHEMBL596380 29125 19877 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 249565873 29127 19878 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME ESTRAMUSTINE ESTRAMUSTINE 15869997 29128 19879 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE FP-1039 FP-1039 29130 19880 FN1 2335 DRUGGABLE GENOME Ocriplasmin OCRIPLASMIN 29131 19881 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER furosemide FUROSEMIDE 26927285 29132 19882 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME pembrolizumab PEMBROLIZUMAB 29133 19883 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME ELLIPTECINE ELLIPTECINE 29134 19884 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER loperamide LOPERAMIDE 29135 19885 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE NERIDRONIC ACID 29136 19886 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Trametinib TRAMETINIB 29138 19887 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178100911 29139 19888 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-10 29140 19889 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TCMDC-123653 CHEMBL548540 29142 19890 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650904 RITANSERIN 29144 19891 GCLC 2729 DRUGGABLE GENOME, ENZYME ETHANOL ALCOHOL 10385658 29146 19892 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE EGFR/IGFR tandem adnectin 29147 19893 PNP 4860 ENZYME, DRUGGABLE GENOME FORODESINE HYDROCHLORIDE FORODESINE HYDROCHLORIDE 19386496,19386498 29148 19894 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GW501516 GW501516 29149 19895 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL289351 FOSBRETABULIN DISODIUM 29150 19896 DIO1 1733 DRUGGABLE GENOME, ENZYME Propylthiouracil PROPYLTHIOURACIL 29151 19897 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING URSOLIC ACID URSOLIC ACID 19534471 29153 19898 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME INTERLEUKIN-1-ALPHA 8321378 29154 19899 TUBB2B 347733 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 29155 19900 PDE5A 8654 ENZYME, DRUGGABLE GENOME SILDENAFIL SILDENAFIL 29156 19901 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SSR-103800 29157 19902 XDH 7498 DRUGGABLE GENOME, ENZYME MISONIDAZOLE MISONIDAZOLE 2799816 29158 19903 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL477 ADENOSINE 29159 19904 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL PMID30185082-Compound-64 29163 19905 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GEFITINIB GEFITINIB 29164 19906 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SLAZINIC ACID SLAZINIC ACID 29165 19907 CFD 1675 ENZYME, DRUGGABLE GENOME, PROTEASE antibody 252166506 LAMPALIZUMAB 29166 19908 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME TETRAIDOFLUORESCEIN TETRAIDOFLUORESCEIN 29168 19909 TNFRSF11A 8792 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE diclofenac DICLOFENAC 26398624 29169 19910 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE BMS-299897 CHEMBL247471 29170 19911 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PYROGALLOL RED PYROGALLOL RED 29172 19912 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR E-GUGGULSTERONE E-GUGGULSTERONE 29175 19913 SMN2 6607 DRUGGABLE GENOME FORMONONETIN FORMONONETIN 29176 19914 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PF-4989216 24240111 29177 19915 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 178101958 29179 19916 SAMHD1 25939 ENZYME, KINASE stavudine STAVUDINE 30273369 29180 19917 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE 9-AMINOCAMPTOTHECIN 9-AMINOCAMPTOTHECIN 29182 19918 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME sorafenib SORAFENIB 28362716 29183 19919 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE everolimus EVEROLIMUS 29184 19920 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TALIPEXOLE TALIPEXOLE 29187 19921 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THIOTHIXENE HYDROCHLORIDE THIOTHIXENE HYDROCHLORIDE 29188 19922 CD44 960 DRUGGABLE GENOME, CELL SURFACE RG7356 25762343 29189 19923 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE GOSSYPOL GOSSYPOL 11510695 29190 19924 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME zuclopenthixol ZUCLOPENTHIXOL 12107620,1927573 29191 19925 GMNN 51053 DRUGGABLE GENOME GNF-PF-2094 CHEMBL578928 29192 19926 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR WEDELOLACTONE WEDELOLACTONE 29193 19927 TBL1XR1 79718 TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE allopurinol ALLOPURINOL 30924126 29194 19928 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor 178103171 29197 19929 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TAS-108 SR16234 29199 19930 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CELECOXIB CELECOXIB 29201 19931 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR DEOXYVASICINONE DEOXYVASICINONE 29202 19932 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-405662 CHEMBL118378 29203 19933 GAA 2548 DRUGGABLE GENOME, ENZYME inhibitor 178101544 MIGLITOL 29206 19934 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME CENISERTIB CENISERTIB 29207 19935 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 posaconazole POSACONAZOLE 29208 19936 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor EVEROLIMUS EVEROLIMUS 29210 19937 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME QUINACRINE QUINACRINE 29211 19938 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME fentanyl FENTANYL 25825958 29212 19939 REG1A 5967 DRUGGABLE GENOME, GROWTH FACTOR INSULIN INSULIN 9930932 29215 19940 ASS1 445 ENZYME, DRUG RESISTANCE PLATINUM COMPOUND 19533750 29216 19941 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME CEDIRANIB CEDIRANIB 29218 19942 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200703 CHLORDIAZEPOXIDE HYDROCHLORIDE 29219 19943 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHENYLETHYL ALCOHOL PHENYLETHYL ALCOHOL 29221 19944 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CICLOPIROX OLAMINE CICLOPIROX OLAMINE 29226 19945 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME inhibitor 178103615 29227 19946 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Nestorone transdermal spray 29228 19947 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Bevacizumab BEVACIZUMAB 27466356,23670029,17145525 29229 19948 GNMT 27232 ENZYME VITAMIN B12 2738712 29230 19949 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RETINAL RETINAL 29231 19950 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ACACETIN DIACETATE ACACETIN DIACETATE 29232 19951 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE MPA PROGESTERONE 10597237 29235 19952 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 387065580 29236 19953 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ORTHO-PHTHALALDEHYDE ORTHO-PHTHALALDEHYDE 29237 19954 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE cyclophosphamide CYCLOPHOSPHAMIDE 16822847 29239 19955 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ALITRETIONINE 29241 19956 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist CHEMBL1201621 SOMATROPIN 29243 19957 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL499 TIMOLOL 29244 19958 ALDH1A1 216 DRUGGABLE GENOME, ENZYME MONASTROL MONASTROL 29245 19959 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 29246 19960 COL18A1 80781 DRUGGABLE GENOME VITAMIN E 12792883 29247 19961 HMGCR 3156 ENZYME, DRUGGABLE GENOME Sterol derivative 3 29248 19962 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BMS-564929 CHEMBL229264 29249 19963 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME CI-1040 CI-1040 26267534 29250 19964 F3 2152 DRUGGABLE GENOME, CELL SURFACE MORAb-066 29251 19965 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652006 29252 19966 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Voruciclib VORUCICLIB 29253 19967 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 387065589 29254 19968 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHELIDAMIC ACID CHELIDAMIC ACID 29255 19969 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1-NAPHTHYLISOTHIOCYANATE 1-NAPHTHYLISOTHIOCYANATE 29256 19970 CBX1 10951 NA NSC-353720 CHEMBL1408276 29261 19971 CD44 960 DRUGGABLE GENOME, CELL SURFACE TUMOR NECROSIS FACTOR 12867430 29265 19972 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME NICLOSAMIDE NICLOSAMIDE 29266 19973 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE sumatriptan SUMATRIPTAN 25096645 29268 19974 POLI 11201 DNA REPAIR ISOORIENTIN ISOORIENTIN 29269 19975 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE LAROTRECTINIB LAROTRECTINIB 30204247,29606586,29466156,24162815,29610391,31605106 29270 19976 IRF2 3660 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR INTERFERON GAMMA 10859338 29271 19977 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-119889 CHEMBL516616 29272 19978 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE AG-490 CHEMBL56543 29273 19979 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE INS-117548 29274 19980 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200440 MEPIVACAINE HYDROCHLORIDE 29275 19981 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Bis-aminopyrimidine derivative 3 29276 19982 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE LICOAGRONE LICOAGRONE 24047800 29277 19983 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 4-hydroxycyclophosphamide 4-HYDROXYCYCLOPHOSPHAMIDE 12684728,18496131 29278 19984 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PMID28906174-Compound-figure1g 29279 19985 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102657 SELICICLIB 29280 19986 ALDH1A1 216 DRUGGABLE GENOME, ENZYME E927A E927A 29282 19987 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE CENISERTIB CENISERTIB 29283 19988 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Doxorubicin DOXORUBICIN 18708578 29284 19989 GMNN 51053 DRUGGABLE GENOME SJ000032151 CHEMBL592600 29285 19990 ALDH5A1 7915 DRUGGABLE GENOME, ENZYME methadone METHADONE 24230997 29286 19991 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Necitumumab NECITUMUMAB 26766738 29287 19992 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-38b 29289 19993 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Thiazole derivative 5 29290 19994 GABBR2 9568 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL2107312 ARBACLOFEN PLACARBIL 29291 19995 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE ZAPRINAST ZAPRINAST 29292 19996 HPSE 10855 ENZYME, DRUGGABLE GENOME REL-CISAPRIDE REL-CISAPRIDE 23415087 29293 19997 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor BMS-754807 BMS-754807 29295 19998 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NIFUROXAZIDE NIFUROXAZIDE 29296 19999 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650705 29297 20000 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME L-PAM MELPHALAN 11507071 29298 20001 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE LY-2090314 LY-2090314 29299 20002 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME S-(P-AZIDOPHENACYL)GLUTATHIONE CHEMBL1256813 29302 20003 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME RO-3201195 RO-3201195 18539026,16509574 29303 20004 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR ICRF-187 DEXRAZOXANE 10487526 29305 20005 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME PMID27998201-Compound-12 29306 20006 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PLICAMYCIN PLICAMYCIN 22931300 29307 20007 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEPHARANTHINE CEPHARANTHINE 29309 20008 GZMB 3002 PROTEASE, DRUGGABLE GENOME, ENZYME HEXACHLOROPHENE HEXACHLOROPHENE 19633659 29310 20009 KDM4A 9682 DRUGGABLE GENOME, ENZYME RANOLAZINE HYDROCHLORIDE RANOLAZINE HYDROCHLORIDE 29311 20010 ICAM3 3385 DRUGGABLE GENOME GRANULOCYTE MACROPHAGE COLONY-STIMULATING FACTOR 12600815 29312 20011 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME RUXOLITINIB RUXOLITINIB 18805579,16293597,20339092,22829971,15781101,16081687,22955920,20631743,19287384,20585391,21120162,22041374,16709929,19470474,18394554,21689158,23115274,22368270,25157968,22818858,24986690,24404189,22422826,22571758 29314 20012 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Ibrutinib IBRUTINIB 26563132 29316 20013 CD58 965 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE Alefacept ALEFACEPT 29317 20014 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME TCMDC-125544 CHEMBL533602 29318 20015 TARDBP 23435 TUMOR SUPPRESSOR FLUCONAZOLE FLUCONAZOLE 29319 20016 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor 178101332 CHEMBL77287 29320 20017 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TZTX-001 29324 20018 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 3-(PHENYLAMINO)PHENOL CHEMBL1523215 29325 20019 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CHLOROPHENYLPIPERAZINE CHLOROPHENYLPIPERAZINE 29326 20020 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME TRAIL 15569667 29327 20021 MAP3K1 4214 CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME docetaxel DOCETAXEL 21636554 29329 20022 TOP2B 7155 DRUGGABLE GENOME, ENZYME Tafluposide TAFLUPOSIDE 29332 20023 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor 178103249 CLORGILINE 29333 20024 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HYPERICIN HYPERICIN 29335 20025 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme27LeucettineL41derivatives 29336 20026 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Phenformin PHENFORMIN 26574479 29337 20027 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-49 29338 20028 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR RG-1530 RG-1530 29339 20029 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE AZ628 CHEMBL2144069 29340 20030 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1091644 LINSITINIB 29341 20031 SMN2 6607 DRUGGABLE GENOME 7-METHOXYISOFLAVONE CHEMBL563919 29345 20032 ALDH5A1 7915 DRUGGABLE GENOME, ENZYME valproic acid 23407051 29350 20033 GAA 2548 DRUGGABLE GENOME, ENZYME DNDI1417470 CHEMBL1422873 29351 20034 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651214 29353 20035 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-44 29354 20036 PTHLH 5744 HORMONE ACTIVITY, DRUGGABLE GENOME PROTEOLYTIC ENZYMES 7556886 29357 20037 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Isoindole 1,3-dione analog 1 29359 20038 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor MEK162 BINIMETINIB 29360 20039 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 29361 20040 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE DOCETAXEL DOCETAXEL 22425996 29362 20041 PSIP1 11168 CLINICALLY ACTIONABLE US9132129, Cpd047 29363 20042 CBX1 10951 NA PYRROLIDINE DITHIOCARBAMATE PYRROLIDINE DITHIOCARBAMATE 29365 20043 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TRYPAN BLUE TRYPAN BLUE 29366 20044 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME LY2090314 LY-2090314 29367 20045 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER NSC-348401 CHEMBL515505 29368 20046 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Jte 013 29369 20047 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 404859048 29370 20048 CHD1 1105 NA EPIRUBICIN EPIRUBICIN 29371 20049 MAPT 4137 DRUGGABLE GENOME ERBSTATIN ERBSTATIN 29372 20050 RRM2 6241 DRUGGABLE GENOME, ENZYME inhibitor 178103428 HYDROXYUREA 29373 20051 TPP1 1200 PROTEASE, ENZYME, DRUGGABLE GENOME Cerliponase Alfa 29374 20052 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650497 L-796449 29375 20053 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9187437, 8 29376 20054 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651574 LEVOTHYROXINE SODIUM 29381 20055 KCNG1 3755 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 29382 20056 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RAUWOLFIA SERPENTINA RAUWOLFIA SERPENTINA 29384 20057 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-124640 CHEMBL547161 29385 20058 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME trimipramine TRIMIPRAMINE 9918137,20531370,1346258,15252821,14716707,18359183,14520122,8867869,8181196,17721180,1527229,17667959,15115913,12360109,14646691,15205367,11682257,16024198,10774635,16361630,17008819,23486447,10460069,9585799,16871470 29387 20059 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-1919 CHEMBL576409 29388 20060 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SERTRALINE SERTRALINE 16680159 29389 20061 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME Phenylalanine derivative 1 29390 20062 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GED-0507-34-Levo 29392 20063 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200694 SEVOFLURANE 29393 20064 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 2,6-DIMETHOXYQUINONE 2,6-DIMETHOXYQUINONE 29395 20065 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME GW441756X GW441756X 29397 20066 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CYCLOSPORINE CYCLOSPORINE 29398 20067 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 N-AMINOHEXYL-5-CHLORO-1-NAPTHALENESULFONAMIDE HYDROCHLORIDE N-AMINOHEXYL-5-CHLORO-1-NAPTHALENESULFONAMIDE HYDROCHLORIDE 29400 20068 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL1078178 MOMELOTINIB 29401 20069 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR INTERLEUKIN-1 RECEPTOR ANTAGONIST 14580934 29402 20070 LIPA 3988 ENZYME, DRUGGABLE GENOME TRIFLUOPERAZINE TRIFLUOPERAZINE 9270979 29403 20071 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PALIFERMIN PALIFERMIN 29404 20072 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL IBUTILIDE IBUTILIDE 29405 20073 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-A3 29406 20074 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor PWT33597 29407 20075 ATXN2 6311 NA NSC-228155 CHEMBL505670 29409 20076 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-7387 CHEMBL119878 29410 20077 BAZ2B 29994 NA GNF-PF-2954 CHEMBL582722 29413 20078 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-13 29414 20079 TXNRD1 7296 DRUGGABLE GENOME Terpyridineplatinum(II) complexe 5 29416 20080 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MORPHINE MORPHINE 29417 20081 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 252166864 CHEMBL407848 29420 20082 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PF-05280014 25001079 29421 20083 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-15 29422 20084 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PD0325901 29423 20085 POLI 11201 DNA REPAIR (-)-EPICATECHIN (-)-EPICATECHIN 29424 20086 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL2108401 ENLIMOMAB PEGOL 29425 20087 BMP2K 55589 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 29427 20088 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 385612237 BEMCENTINIB 29428 20089 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR DERRUBONE DERRUBONE 29430 20090 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME pimozide PIMOZIDE 9951426,23059146 29431 20091 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Anistreplase ANISTREPLASE 29432 20092 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR inhibitor 340590276 29433 20093 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-21 29434 20094 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME SGN-70 29435 20095 UCP2 7351 TRANSPORTER, DRUGGABLE GENOME ANTIOXIDANT 15642337 29437 20096 GUCY2C 2984 DRUGGABLE GENOME, KINASE agonist CHEMBL3301675 LINACLOTIDE 29438 20097 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER FLAVOPIRIDOL ALVOCIDIB 10496352 29440 20098 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE ESCULETIN ESCULETIN 29441 20099 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CAPTAN CAPTAN 29442 20100 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Methylscopolamine METHSCOPOLAMINE 29444 20101 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DAIDZEIN DAIDZEIN 29445 20102 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GO-6976 GO-6976 29446 20103 TUBB6 84617 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 29448 20104 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Alkyl sulfone derivative 1 29449 20105 POLK 51426 DNA REPAIR, ENZYME ELLAGIC ACID ELLAGIC ACID 29450 20106 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME HUMAN CHORIONIC GONADOTROPIN 11095483 29451 20107 EIF2AK4 440275 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME risperidone RISPERIDONE 24751813 29452 20108 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BMS-927711 RIMEGEPANT 29453 20109 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE CENISERTIB CENISERTIB 29455 20110 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX STROPHANTHIDIN STROPHANTHIDIN 29457 20111 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX VORICONAZOLE VORICONAZOLE 18625774 29459 20112 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR FULVESTRANT FULVESTRANT 29461 20113 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Crizotinib CRIZOTINIB 27595477,26432108 29462 20114 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SPIRAMIDE SPIRAMIDE 29463 20115 TSPO 706 DRUGGABLE GENOME Quinoline carboxamide derivative 6 29464 20116 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR RG-7304 RG-7304 25766633 29465 20117 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME ZINC SULFATE 14568236 29466 20118 APC 324 CLINICALLY ACTIONABLE Trastuzumab TRASTUZUMAB 27626067 29467 20119 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME BIX-01294 CHEMBL569864 29468 20120 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DOXEPIN DOXEPIN 29470 20121 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PLATINUM PLATINUM 12181446 29472 20122 PC 5091 ENZYME, CLINICALLY ACTIONABLE AMPHOTERICIN B 2015823 29473 20123 KMO 8564 DRUGGABLE GENOME, ENZYME Isoxazoles and isoxazoline derivative 5 29474 20124 GNMT 27232 ENZYME mercaptopurine MERCAPTOPURINE 27452984 29476 20125 TAT 6898 ENZYME ANDROGENS 2882620 29477 20126 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL750 ZONISAMIDE 29478 20127 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE tamatinib 29479 20128 GMNN 51053 DRUGGABLE GENOME TCMDC-124468 CHEMBL1376851 29480 20129 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Doxorubicin DOXORUBICIN 27893038 29484 20130 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102730 29487 20131 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LAMELLARIN D LAMELLARIN D 21783369 29489 20132 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 29490 20133 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE DAUNORUBICIN DAUNORUBICIN 21094049 29492 20134 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545420 AG-24322 29493 20135 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE 17 BETA-ESTRADIOL 2492346 29494 20136 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DEQUALINIUM DEQUALINIUM 29495 20137 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 29496 20138 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DICHLOROPHEN DICHLOROPHEN 29497 20139 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME SCH772984 27222538 29500 20140 ATXN2 6311 NA A-443654 A-443654 29501 20141 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 249565661 29502 20142 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125310 CHEMBL582030 29504 20143 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME IL-13 12620497 29505 20144 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PYRROLIDINE DITHIOCARBAMATE PYRROLIDINE DITHIOCARBAMATE 29507 20145 RPS6KB2 6199 DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME, KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3544935 XL-418 29508 20146 CRTC2 200186 KINASE PKI-587 GEDATOLISIB 29510 20147 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE GW843682X GW843682X 29511 20148 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME RG-1530 RG-1530 29512 20149 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME SAND-5 22990692 29514 20150 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135650171 DESIPRAMINE 29517 20151 MT3 4504 PROTEASE INHIBITOR, HISTONE MODIFICATION IL-6 9675420 29519 20152 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL931 HALOTHANE 29520 20153 S100A10 6281 KINASE DEXAMETHASONE DEXAMETHASONE 10358078 29521 20154 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102620 29523 20155 ATAD5 79915 NA 4'-METHOXYFLAVONE 4'-METHOXYFLAVONE 29524 20156 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ASPIRIN ASPIRIN 30683736,23094721 29525 20157 PSMC5 5705 TRANSCRIPTION FACTOR BINDING, PROTEASE CARFILZOMIB CARFILZOMIB 24524217 29526 20158 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME ABT-263 NAVITOCLAX 29527 20159 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE KU-55933 KU-55933 16767085 29528 20160 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MELATONIN MELATONIN 15813899 29529 20161 TUBB 203068 DRUGGABLE GENOME NSC-639829 29530 20162 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MORIN MORIN 29531 20163 TOP2B 7155 DRUGGABLE GENOME, ENZYME Enoxacin ENOXACIN 29533 20164 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER CEPHALEXIN CEPHALEXIN 22166395 29534 20165 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME NKP-1339 IT-139 29535 20166 TUBB2A 7280 DRUGGABLE GENOME CHEMBL2105643 FOSBRETABULIN TROMETHAMINE 29536 20167 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE CCT018159 CHEMBL399530 29537 20168 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3407 CHEMBL602990 29539 20169 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Biphenyl derivative 3 29540 20170 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-36 29541 20171 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR EVEROLIMUS EVEROLIMUS 26951309 29543 20172 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL592445 GEDATOLISIB 29544 20173 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ATEZOLIZUMAB ATEZOLIZUMAB 25428504 29545 20174 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 29546 20175 TNKS 8658 DRUGGABLE GENOME, ENZYME 2X-121 2X-121 29547 20176 ABCC5 10057 DRUGGABLE GENOME, ABC TRANSPORTER, TRANSPORTER oxaliplatin OXALIPLATIN 24924344 29548 20177 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE LAUROGUADINE LAUROGUADINE 29549 20178 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 404859027 29551 20179 PSMD4 5710 NA inhibitor CHEMBL2103884 OPROZOMIB 29553 20180 UBA3 9039 TUMOR SUPPRESSOR, ENZYME MLN-4924 PEVONEDISTAT 29555 20181 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR RO-5068760 CHEMBL1956073 20053779 29556 20182 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650599 METOPROLOL 29557 20183 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650856 PROPAFENONE 29558 20184 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL Debio-0824 22637724 29559 20185 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME allosteric modulator 249565625 REFAMETINIB 29565 20186 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME BEVACIZUMAB BEVACIZUMAB 29566 20187 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE JSM 6427 29567 20188 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CLOZAPINE CLOZAPINE 17052361 29568 20189 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor GSK2636771 GSK-2636771 29570 20190 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Triazolo-pyridine derivative 1 29571 20191 MAPT 4137 DRUGGABLE GENOME CYSTAMINE HYDROCHLORIDE CYSTAMINE HYDROCHLORIDE 29572 20192 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TCMDC-125543 CHEMBL546170 29574 20193 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565645 MK-2461 29578 20194 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Oxaliplatin OXALIPLATIN 26540314,26341920,23209813,21468686 29579 20195 TSPO 706 DRUGGABLE GENOME Dextofisopam DEXTOFISOPAM 29581 20196 ASNS 440 CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE L-ASPARAGINASE ASPARAGINASE 11556848 29583 20197 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CETRIMONIUM BROMIDE CETRIMONIUM BROMIDE 29584 20198 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Desoxycorticosterone Acetate 29588 20199 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME GAMBOGIC ACID GAMBOGIC ACID 17911251 29589 20200 RGS4 5999 DRUGGABLE GENOME GBR-12909 VANOXERINE 29590 20201 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME SCRIPTAID SCRIPTAID 19966789 29592 20202 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BAY80-6946 COPANLISIB 29593 20203 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 135650355 DEXANABINOL 29594 20204 TSPO 706 DRUGGABLE GENOME Imidazo[1,2-b]pyridazine acetamide derivative 3 29595 20205 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME PYROGALLOL RED PYROGALLOL RED 29596 20206 CXCL8 3576 DRUGGABLE GENOME ALUMINUM HYDROXIDE 10466876 29597 20207 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651785 29598 20208 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NSC-123414 CHEMBL16751 29599 20209 AQP3 360 ION CHANNEL, TRANSPORTER inhibitor 381118898 AUPHEN 29600 20210 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650525 LISURIDE 29602 20211 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL AZIETOMIDATE AZIETOMIDATE 16884293 29604 20212 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme8NCGC-00189310 29610 20213 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 1,2,3,4,5,6-HEXABROMO-CYCLOHEXANE CHEMBL444236 29612 20214 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR KB-003 LENZILUMAB 29613 20215 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL2106798 NERAMEXANE MESYLATE 29614 20216 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE NERATINIB MALEATE 29617 20217 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME leucovorin LEUCOVORIN 29618 20218 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PF-4217903 PF-04217903 29619 20219 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TESTOSTERONE PROPIONATE TESTOSTERONE PROPIONATE 29620 20220 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME BDBM50011553 29623 20221 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE folic acid 29662106,16672082,22926161,20634689,29317847,19307503 29627 20222 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 178103309 29630 20223 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-6 29631 20224 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL572881 MOTESANIB 29632 20225 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE CYC-116 CYC-116 29633 20226 JUNB 3726 TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR CYTOKINES 9591138 29634 20227 NDUFB10 4716 ENZYME inhibitor CHEMBL3545135 NV-128 29636 20228 PGF 5228 GROWTH FACTOR, DRUGGABLE GENOME TB-403 TB-403 29637 20229 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR 5,4'-DIHYDROXYFLAVONE CHEMBL484662 29638 20230 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME atorvastatin ATORVASTATIN 27839692 29639 20231 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME MARIZOMIB MARIZOMIB 24269479 29640 20232 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 5-METHOXYFLAVANONE CHEMBL317869 29641 20233 CLCN7 1186 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER blocker 178101087 29642 20234 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME GNF-PF-4242 CHEMBL584514 29643 20235 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650756 OLANZAPINE 29644 20236 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE XL147 PILARALISIB 25637314 29645 20237 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-4418 CHEMBL604321 29647 20238 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR inhibitor 348353652 29648 20239 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 252166862 29649 20240 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 354702247 ELISMETREP 29650 20241 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 29651 20242 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR BDBM50158755 29652 20243 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Fluorometholone FLUOROMETHOLONE 29653 20244 PGD 5226 ENZYME, DRUGGABLE GENOME PHENOBARBITAL PHENOBARBITAL 7827108 29654 20245 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US10100051, Compound 11 29656 20246 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME GENISTEIN GENISTEIN 15290869 29658 20247 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FURAZABOL FURAZABOL 29659 20248 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL41306 CNS-5161 29661 20249 POLK 51426 DNA REPAIR, ENZYME DOXORUBICIN DOXORUBICIN 29662 20250 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PSAMMAPLIN A PSAMMAPLIN A 25884112 29663 20251 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME EUPAFOLIN EUPAFOLIN 29664 20252 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GNF-PF-3955 CHEMBL605747 29665 20253 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HARMALINE HARMALINE 29666 20254 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PREDNISONE PREDNISONE 22931300 29668 20255 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR PLX4720 PLX-4720 21383288,19915144 29669 20256 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE 2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE CHEMBL412603 29670 20257 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE STANOLONE STANOLONE 22014751 29671 20258 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME FTI-277 8620483 29674 20259 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565794 29675 20260 GMNN 51053 DRUGGABLE GENOME SILIBININ SILIBININ 29677 20261 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TG02, SB1317 29678 20262 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME SIROLIMUS SIROLIMUS 27482884,27279227 29679 20263 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR irinotecan IRINOTECAN 27160286 29680 20264 PSMA1 5682 PROTEASE, DRUGGABLE GENOME inhibitor CARFILZOMIB CARFILZOMIB 29681 20265 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166694 29682 20266 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Veltuzumab VELTUZUMAB 29686 20267 COL18A1 80781 DRUGGABLE GENOME H2O2 12832291 29687 20268 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE MSC2363318A MSC-2363318A 27186432 29688 20269 ATXN2 6311 NA SERTRALINE HYDROCHLORIDE SERTRALINE HYDROCHLORIDE 29689 20270 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME IL-4 10891465 29690 20271 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE inhibitor 178103263 PROPYLTHIOURACIL 29691 20272 MAPT 4137 DRUGGABLE GENOME IRIGINOL HEXAACEATATE IRIGINOL HEXAACEATATE 29693 20273 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AZATHIOPRINE AZATHIOPRINE 29694 20274 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-2954 CHEMBL582722 29695 20275 HCP5 10866 NA carboplatin CARBOPLATIN 31616045 29696 20276 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ARA-C 15632314 29697 20277 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME XL228 XL-228 29698 20278 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE LY294002 18262558 29700 20279 POLK 51426 DNA REPAIR, ENZYME SCLEROTIORIN SCLEROTIORIN 29702 20280 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE Pyrrolo-pyrazine derivative 3 29703 20281 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR L-165041 CHEMBL153057 29707 20282 IRF6 3664 TRANSCRIPTION FACTOR interferon beta-1b 30013178 29708 20283 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103753 ESMOLOL 29709 20284 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MISOPROSTOL MISOPROSTOL 29710 20285 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL3545103 AZD3199 29712 20286 KDM4A 9682 DRUGGABLE GENOME, ENZYME N-OXALYLGLYCINE N-OXALYLGLYCINE 19359167 29713 20287 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SNS-314 SNS-314 29714 20288 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR NCG-C00094421-01 CHEMBL553503 29715 20289 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR SUBEROHYDROXAMIC ACID SUBEROHYDROXAMIC ACID 16921367 29716 20290 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 381118867 29717 20291 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL517712 ATROPINE 29719 20292 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME DORAMAPIMOD DORAMAPIMOD 29720 20293 GAA 2548 DRUGGABLE GENOME, ENZYME HYPEROSIDE HYPEROSIDE 29721 20294 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 7,3'-DIHYDROXYFLAVONE CHEMBL253786 29722 20295 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor EVEROLIMUS EVEROLIMUS 29723 20296 ALDH1A1 216 DRUGGABLE GENOME, ENZYME FUROXAN FUROXAN 29724 20297 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GLYCINE GLYCINE 22931300 29725 20298 MAOB 4129 DRUGGABLE GENOME, ENZYME Selegiline Hydrochloride 29727 20299 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME Quinazolines and azaquinazoline derivative 1 29729 20300 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-2272 CHEMBL601757 29731 20301 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651413 SEROTONIN 29733 20302 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALVOCIDIB HYDROCHLORIDE ALVOCIDIB HYDROCHLORIDE 29734 20303 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000040829 CHEMBL589711 29736 20304 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MODAFINIL MODAFINIL 22931300 29739 20305 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 178103925 VILANTEROL 29740 20306 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL1201733 PAZOPANIB HYDROCHLORIDE 29741 20307 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TCMDC-123951 CHEMBL587849 29742 20308 TSPO 706 DRUGGABLE GENOME 18F-FEDAA-1106 29743 20309 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417719 CHEMBL1420370 29744 20310 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GAMBOGIC ACID GAMBOGIC ACID 17911251 29745 20311 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 252827481 29746 20312 TNIK 23043 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE SB-202190 SB-202190 22951114 29747 20313 STING1 340061 CLINICALLY ACTIONABLE, KINASE antagonist 381118832 29748 20314 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 252827489 29749 20315 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR VEGF 11704858 29750 20316 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE HALOFANTRINE HYDROCHLORIDE HALOFANTRINE HYDROCHLORIDE 29753 20317 AKR1C3 8644 ENZYME, DRUGGABLE GENOME N-(benzimidazole/indole) benzoic acid derivative 2 29756 20318 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ARBUTAMINE ARBUTAMINE 29757 20319 BAZ2B 29994 NA N'-(2-HYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE SALINAZID 29759 20320 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME DNDI1318925 CHEMBL1390716 29761 20321 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR GNF-PF-3832 CHEMBL261693 29763 20322 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE DIPYRIDAMOLE DIPYRIDAMOLE 29764 20323 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING LARGAZOLE LARGAZOLE 21420302,25203782,20491440 29765 20324 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 336446966 29766 20325 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME Linopirdine LINOPIRDINE 29768 20326 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME PMSG 15798021 29769 20327 POLB 5423 DNA REPAIR, DRUGGABLE GENOME DNDI1417346 CHEMBL1490332 29771 20328 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CLOBAZAM CLOBAZAM 29773 20329 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 135652720 29774 20330 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1201023 ORPHENADRINE HYDROCHLORIDE 29775 20331 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1201728 DESVENLAFAXINE SUCCINATE 29777 20332 CD38 952 CELL SURFACE, DRUGGABLE GENOME Anti-CD38 CAR-T cells 29778 20333 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TPM-1/Morphine 22020140 29781 20334 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Decyle nelycorine dibromo salt derivative 1 29782 20335 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651541 EPOPROSTENOL 29784 20336 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE MEGESTROL ACETATE 15345738 29785 20337 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SURAMIN HEXASODIUM SURAMIN HEXASODIUM 29786 20338 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TRIFLUOPERAZINE TRIFLUOPERAZINE 12415616 29788 20339 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE ELLAGIC ACID ELLAGIC ACID 29789 20340 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor CHEMBL1946170 REGORAFENIB 29790 20341 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Etoposide ETOPOSIDE 27216155 29791 20342 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HERACLENOL HERACLENOL 29792 20343 TUBA1A 7846 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 29793 20344 POLK 51426 DNA REPAIR, ENZYME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 29794 20345 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME MICHLER'S KETONE MICHLER'S KETONE 29795 20346 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR Tazemetostat TAZEMETOSTAT 28135235,28231254,26360609,26676756,24563539 29796 20347 PRIM1 5557 DRUGGABLE GENOME 3'-DEOXYADENOSINE 8827435 29797 20348 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL3545341 SAR-407899 29798 20349 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR abemaciclib ABEMACICLIB 29800 20350 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE AT-7867 24978597,20423992 29801 20351 PRSS3 5646 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 315661094 29802 20352 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Palifosfamide PALIFOSFAMIDE 29803 20353 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE acetaminophen ACETAMINOPHEN 23279026,26049587,16696573,11714888 29805 20354 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL NITRAZEPAM NITRAZEPAM 29806 20355 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID27724045-Compound-14 29807 20356 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME Vemurafenib VEMURAFENIB 25939769 29808 20357 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL OCINAPLON OCINAPLON 29809 20358 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Tetrabenazine TETRABENAZINE 29810 20359 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR tamoxifen TAMOXIFEN 29812 20360 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AMITRIPTYLINE AMITRIPTYLINE 22931300 29813 20361 SLC28A2 9153 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME URIDINE URIDINE 23388705 29815 20362 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HALAZONE HALAZONE 29818 20363 CCL21 6366 DRUGGABLE GENOME ANTIANGIOGENIC 10925282 29819 20364 HPSE 10855 ENZYME, DRUGGABLE GENOME NARINGIN NARINGIN 23415087 29820 20365 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME rifampin RIFAMPIN 27053325,17638512,28389387 29822 20366 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102915 29824 20367 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE N/A 26276366,25729899 29826 20368 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AFIMOXIFENE AFIMOXIFENE 29827 20369 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME SULFOBROMOPHTHALEIN SULFOBROMOPHTHALEIN 21422191 29829 20370 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME NICOTINE NICOTINE 15225679 29830 20371 MGAT4A 11320 DRUGGABLE GENOME bevacizumab BEVACIZUMAB 26222057 29831 20372 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME PF-562271 PF-00562271 29833 20373 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135652664 ALCURONIUM 29835 20374 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE ENTRECTINIB ENTRECTINIB 29836 20375 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME DALANTERCEPT DALANTERCEPT 29837 20376 CTAG2 30848 NA AUTOLOGOUS ANTI-NY-ESO-1/LAGE-1 TCR-TRANSDUCED C259 T LYMPHOCYTES GSK3377794 26193344 29838 20377 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-31 29839 20378 ATXN2 6311 NA TYRPHOSTIN A9 TYRPHOSTIN A9 29840 20379 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL2107842 ALBINTERFERON ALFA-2B 29841 20380 MAPT 4137 DRUGGABLE GENOME 3',4'-DIHYDROXYFLAVONE CHEMBL222556 29842 20381 DLG5 9231 KINASE capecitabine CAPECITABINE 29843 20382 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NCI-13239 CHEMBL187216 29844 20383 ALOX15 246 ENZYME, DRUGGABLE GENOME CUMENE HYDROPEROXIDE CUMENE HYDROPEROXIDE 29845 20384 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE BPTES 24333121 29846 20385 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-36398 CHEMBL483206 29847 20386 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651151 29848 20387 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000027778 CHEMBL592588 29849 20388 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE risperidone RISPERIDONE 29852 20389 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER FENOFIBRATE FENOFIBRATE 16316932 29853 20390 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Alcaftadine ALCAFTADINE 29854 20391 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME MITOXANTRONE MITOXANTRONE 29856 20392 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417264 CHEMBL1467200 29857 20393 LIPA 3988 ENZYME, DRUGGABLE GENOME TRIIODOTHYRONINE LIOTHYRONINE SODIUM 6713293 29858 20394 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME DASATINIB DASATINIB 29859 20395 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRICYCLAZOLE TRICYCLAZOLE 29860 20396 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR STICTIC ACID STICTIC ACID 29861 20397 APC 324 CLINICALLY ACTIONABLE PKF115-584 14749129 29862 20398 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-129 29863 20399 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME PARA-SIRTINOL CHEMBL372375 23189967 29865 20400 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Aromatic bicyclic compound 3 29868 20401 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME blocker 135650114 CLOTRIMAZOLE 29869 20402 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PAZOPANIB PAZOPANIB 23786770,24550739 29870 20403 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 22931300 29871 20404 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AMB 16127053 29872 20405 ALOX15 246 ENZYME, DRUGGABLE GENOME CHOLECALCIFEROL CHOLECALCIFEROL 29873 20406 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR INDACATEROL INDACATEROL 29874 20407 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417181 CHEMBL1537417 29875 20408 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME PF-4554878 29876 20409 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE ADRIAMYCIN ADRIAMYCIN 10831167 29877 20410 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650911 29879 20411 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 374883884 29880 20412 TUBB2B 347733 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 29881 20413 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SIMVASTATIN SIMVASTATIN 17928392 29884 20414 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR PICEATANNOL PICEATANNOL 29888 20415 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MICAFUNGIN MICAFUNGIN 16205037 29889 20416 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR platinum PLATINUM 19786980,22188361,18347182,21902499,25069034,21057378,29662106,19362955,27498158,21262916,22026922,22329723 29890 20417 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Tonabersat TONABERSAT 29891 20418 CBX1 10951 NA NSC-628113 CHEMBL176599 29895 20419 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME RANIBIZUMAB RANIBIZUMAB 29896 20420 ALDH1A1 216 DRUGGABLE GENOME, ENZYME aldophosphamide ALDOPHOSPHAMIDE 29899 20421 FGG 2266 DRUGGABLE GENOME, FIBRINOGEN, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor CHEMBL1201505 FIBRINOLYSIN, HUMAN 29900 20422 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME tramadol TRAMADOL 24849324 29902 20423 RAB9A 9367 ENZYME, DRUGGABLE GENOME PIFEXOLE PIFEXOLE 29904 20424 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor CHEMBL3544933 VS-4718 29905 20425 MPI 4351 ENZYME, DRUGGABLE GENOME APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 29906 20426 TPM3 7170 KINASE, CLINICALLY ACTIONABLE ACTH CORTICOTROPIN 17877367 29907 20427 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME AST-487 AST-487 29908 20428 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE SOMATROPIN RECOMBINANT 29909 20429 ATXN2 6311 NA SORAFENIB TOSYLATE SORAFENIB TOSYLATE 29911 20430 USP1 7398 DNA REPAIR, PROTEASE, ENZYME LAURYL ISOQUINOLINIUM LAURYL ISOQUINOLINIUM 29912 20431 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME ANDROGENS 2229290 29913 20432 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NIA-114 29918 20433 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-2243 CHEMBL600908 29919 20434 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PSAMMAPLIN A PSAMMAPLIN A 25884112 29922 20435 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ERIBULIN ERIBULIN 26006067 29923 20436 GBA 2629 DRUGGABLE GENOME, ENZYME GNF-PF-1295 CHEMBL579837 29924 20437 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME WORTMANNIN WORTMANNIN 17135248 29925 20438 NOS2 4843 DRUGGABLE GENOME, ENZYME BXT-51072 ALT-2074 29926 20439 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 1-METHYLEVODIAMINE CHEMBL2171778 22867019 29929 20440 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME AZD-1080 AZD-1080 29930 20441 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE TRIAMCINOLONE TRIAMCINOLONE 1197440 29933 20442 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CAPSAZEPINE CAPSAZEPINE 29934 20443 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SIMETRIDE SIMETRIDE 29935 20444 HMGCR 3156 ENZYME, DRUGGABLE GENOME LOVASTATIN LOVASTATIN 24726306 29938 20445 ATXN2 6311 NA GNF-PF-78 CHEMBL579318 29939 20446 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE GNF-PF-5151 CHEMBL576208 29941 20447 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103492 29943 20448 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE CISPLATIN CISPLATIN 9219734 29945 20449 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE TAPENTADOL TAPENTADOL 29948 20450 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PROCHLORPERAZINE PROCHLORPERAZINE 22931300 29950 20451 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL598797 CUDC-101 29951 20452 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE antibody PERTUZUMAB PERTUZUMAB 29952 20453 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BACLOFEN BACLOFEN 29953 20454 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 363894208 ILORASERTIB 29954 20455 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101291 29955 20456 MARCHF8 220972 ENZYME Focetria A(H1N1) 29956 20457 IL7R 3575 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CYT-107 29958 20458 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME TAK-715 TAK-715 29960 20459 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PKI-587 GEDATOLISIB 29961 20460 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RILUZOLE RILUZOLE 29963 20461 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME docetaxel DOCETAXEL 21151855 29964 20462 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW832467X GW832467X 29965 20463 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ranitidine RANITIDINE 29967 20464 TMEM97 27346 NA CT1812 29968 20465 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CEFMETAZOLE CEFMETAZOLE 22166395 29970 20466 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE DOVITINIB DOVITINIB 29973 20467 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE cetuximab CETUXIMAB 29974 20468 FAAH 2166 ENZYME, DRUGGABLE GENOME Boronic acid derivative 5 29975 20469 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 diltiazem DILTIAZEM 9187528 29976 20470 MAOA 4128 DRUGGABLE GENOME, ENZYME Moclobemide MOCLOBEMIDE 29977 20471 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIBUTYLCHLOROSTANNANE TRIBUTYLCHLOROSTANNANE 29979 20472 POLI 11201 DNA REPAIR GNF-PF-159 CHEMBL599924 29980 20473 GMNN 51053 DRUGGABLE GENOME DIBUCAINE DIBUCAINE 29981 20474 ITPA 3704 ENZYME methotrexate METHOTREXATE 26237184,19858780,27217051,29520081,16947783 29982 20475 COL18A1 80781 DRUGGABLE GENOME RED CELLS 15181823 29984 20476 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL2108589 CLAZAKIZUMAB 29986 20477 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR DES DIETHYLSTILBESTROL 17292805 29989 20478 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2103840 DINACICLIB 29990 20479 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE DORAMAPIMOD DORAMAPIMOD 29992 20480 CDC37 11140 KINASE GELDANAMYCIN GELDANAMYCIN 21486005 29995 20481 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2107731 AXOMADOL 29997 20482 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR SURGICAL ADJUVANT 10764421 29998 20483 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Selumetinib SELUMETINIB 26438159 29999 20484 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker 178100912 30000 20485 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-72b 30001 20486 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-2B, RECOMBINANT 30004 20487 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Methylprednisolone Acetate 30005 20488 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE Metformin METFORMIN 17062558,18006825 30006 20489 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CHEMBL407 FLUMAZENIL 30008 20490 EDN3 1908 DRUGGABLE GENOME, HORMONE ACTIVITY HUMAN CHORIONIC GONADOTROPIN 9870082 30009 20491 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GLABROL GLABROL 20022509 30010 20492 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME inhibitor 381744899 30011 20493 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MEQUITAZINE MEQUITAZINE 30012 20494 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649675 30013 20495 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-4803 CHEMBL585240 30015 20496 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CHIR-265 RAF-265 30016 20497 NDUFV3 4731 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 30018 20498 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR RALOXIFEN RALOXIFEN 30019 20499 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 1,5-ISOQUINOLINEDIOL CHEMBL338314 30020 20500 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE BMS-299897 CHEMBL247471 30021 20501 NDUFAF3 25915 NA inhibitor CHEMBL3545135 NV-128 30022 20502 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME DNDI1417076 CHEMBL1526167 30024 20503 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Ruxolitinib cream 30025 20504 SETBP1 26040 CLINICALLY ACTIONABLE N/A 23832012 30026 20505 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE AMUVATINIB AMUVATINIB 30027 20506 TSPO 706 DRUGGABLE GENOME Temazepam TEMAZEPAM 30029 20507 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME CTP-543 30030 20508 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650345 HALOPERIDOL 30032 20509 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DDD 7587937 30034 20510 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 7-Vanillic acid 30035 20511 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PLX4720 PLX-4720 20538618,26351322,24265153,21383288,23242808,27924459,19915144,24983357,18287029,27523909,26461489,22281684,27217440,26573800 30036 20512 F7 2155 ENZYME, DRUGGABLE GENOME, PROTEASE F-7TG 30037 20513 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TANNIC ACID TANNIC ACID 30038 20514 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE PMID29130358-Compound-Figure17(12) 30041 20515 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE CB-10-01 30042 20516 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545027 XL-281 30044 20517 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR Autologous melanoma cell vaccine 30045 20518 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TRIFLOXYSTROBIN TRIFLOXYSTROBIN 30046 20519 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GNF-PF-4218 CHEMBL585269 30047 20520 BAZ2B 29994 NA SJ000292689 CHEMBL602954 30048 20521 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE TRABECTEDIN TRABECTEDIN 28454547 30050 20522 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE JUGLONE JUGLONE 30051 20523 DNER 92737 NA PMID26924192-Compound-54 30053 20524 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME KD019 TESEVATINIB 30054 20525 POLB 5423 DNA REPAIR, DRUGGABLE GENOME PROSTAGLANDIN A2 PROSTAGLANDIN A2 30055 20526 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 315661184 LUMATEPERONE 30056 20527 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHOXYCHLOR METHOXYCHLOR 30057 20528 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID2350207 CHEMBL259615 30058 20529 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME MLN0128 SAPANISERTIB 26272063 30059 20530 MAPT 4137 DRUGGABLE GENOME CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE 30064 20531 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 363894214 SITRAVATINIB 30065 20532 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SULPIRIDE SULPIRIDE 22931300 30066 20533 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE IBUPROFEN IBUPROFEN 16997128 30069 20534 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1201190 LEVOCETIRIZINE DIHYDROCHLORIDE 30074 20535 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor 178103971 IBUDILAST 30075 20536 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-3 30076 20537 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649707 2-METHYLHISTAMINE 30077 20538 TSPO 706 DRUGGABLE GENOME Oxazepam OXAZEPAM 30078 20539 TNFRSF12A 51330 DRUGGABLE GENOME agonist CHEMBL1743011 ENAVATUZUMAB 30079 20540 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR 2-O, 3-O DESULFATED HEPARIN 30080 20541 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE PF-562271 PF-00562271 30085 20542 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9522888, 618 30086 20543 GMNN 51053 DRUGGABLE GENOME GNF-PF-1702 CHEMBL600313 30087 20544 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUFENAMIC ACID FLUFENAMIC ACID 17911242 30088 20545 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE ABACAVIR ABACAVIR 17172311 30089 20546 RAMP1 10267 DRUGGABLE GENOME, CELL SURFACE SALMON CALCITONIN 30090 20547 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR LINIFANIB LINIFANIB 30091 20548 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER ETOCARLIDE ETOCARLIDE 30092 20549 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DISULFIRAM DISULFIRAM 30094 20550 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor NINTEDANIB NINTEDANIB 30095 20551 ALDH1A1 216 DRUGGABLE GENOME, ENZYME IODOACETAMIDE IODOACETAMIDE 30096 20552 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 252166567 30097 20553 TLK2 11011 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME GO6983 27694828 30100 20554 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GLUFOSFAMIDE GLUFOSFAMIDE 30101 20555 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CIPROFLOXACIN CIPROFLOXACIN 30102 20556 GPR183 1880 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178101167 30103 20557 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-N1 30108 20558 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Quinoline carboxamide derivative 2 30109 20559 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME TAE-684 TAE-684 30110 20560 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PAPAVERINE HYDROCHLORIDE PAPAVERINE HYDROCHLORIDE 30111 20561 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650861 PRUCALOPRIDE 30112 20562 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE DACARBAZINE DACARBAZINE 9378540 30114 20563 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 7 30116 20564 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 4,4'-METHYLENEDIANILINE 4,4'-METHYLENEDIANILINE 30120 20565 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor ENZASTAURIN ENZASTAURIN 30122 20566 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIHYDROXIDINE DIHYDROXIDINE 30123 20567 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE DOVITINIB DOVITINIB 30124 20568 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor 315661236 CRISABOROLE 30125 20569 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL519504 ALEGLITAZAR 30128 20570 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE partial agonist CHEMBL500 PINDOLOL 30129 20571 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME antagonist,activator 135652731 30130 20572 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Nilotinib NILOTINIB 30133 20573 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135649866 30135 20574 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 328083477 30137 20575 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-123764 CHEMBL533226 30138 20576 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME 6-HYDROXYDOPAMINE 15504737 30140 20577 ACSS2 55902 ENZYME, TRANSCRIPTION FACTOR inhibitor 405560508 30141 20578 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHYSTICIN METHYSTICIN 30143 20579 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TILIQUINOL TILIQUINOL 30144 20580 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHLOROGENIC ACID CHLOROGENIC ACID 30146 20581 VCAM1 7412 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME 6-MERCAPTOPURINE MERCAPTOPURINE 7694584 30147 20582 ABL2 27 KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME DASATINIB DASATINIB 30148 20583 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3996 CHEMBL584458 30149 20584 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME TG003 30150 20585 GJB3 2707 TRANSPORTER, ION CHANNEL inhibitor 178100972 CARBENOXOLONE 30152 20586 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200606 MEXILETINE HYDROCHLORIDE 30153 20587 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR IBUPROFEN IBUPROFEN 8870119,9118476 30154 20588 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103080 CIPEMASTAT 30155 20589 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME blocker 178100912 30157 20590 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME cytarabine CYTARABINE 26663398,22584460 30158 20591 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE MN-221 BEDORADRINE SULFATE 30159 20592 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AC-100,DENTONIN 30160 20593 GCLM 2730 ENZYME CISPLATIN CISPLATIN 10399958 30161 20594 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE folic acid 18322994 30163 20595 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody SYM004 30164 20596 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 5 30166 20597 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME DIETHYLDITHIOCARBAMATE DITIOCARB 6135240 30168 20598 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE TOLFENAMIC ACID TOLFENAMIC ACID 30170 20599 ULK3 25989 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565900 30171 20600 CBX1 10951 NA LEVODOPA LEVODOPA 30172 20601 ATXN2 6311 NA THONZONIUM BROMIDE THONZONIUM BROMIDE 30173 20602 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME INAMRINONE INAMRINONE 30174 20603 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-13 30175 20604 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200638 DEXBROMPHENIRAMINE MALEATE 30176 20605 KDM4A 9682 DRUGGABLE GENOME, ENZYME ACITRETIN ACITRETIN 30177 20606 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Cisplatin CISPLATIN 26517239 30178 20607 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PAZOPANIB PAZOPANIB 30179 20608 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX doxorubicin DOXORUBICIN 30181 20609 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE LENALIDOMIDE LENALIDOMIDE 30182 20610 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 4'-EPICHAETOVIRIDIN A CHEMBL1306556 30183 20611 MAP3K5 4217 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, ENZYME GS-4977 30184 20612 MTRR 4552 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VITAMIN B12 12807760 30185 20613 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE PALBOCICLIB PALBOCICLIB 30186 20614 HEBP1 50865 DRUGGABLE GENOME 1,2,3,4-tetrahydroisoquinoline derivative 1 30187 20615 NME1 4830 KINASE zidovudine ZIDOVUDINE 22960662 30188 20616 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102897 ACETALDEHYDE 30189 20617 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THIOTEPA THIOTEPA 30190 20618 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR SCRIPTAID SCRIPTAID 19966789 30193 20619 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME Venetoclax VENETOCLAX 27520294 30194 20620 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL41355 EZOGABINE 30195 20621 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME vaccine PRINOMASTAT PRINOMASTAT 30196 20622 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE vaccine EP-2101 30198 20623 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 252166577 PRACINOSTAT 30199 20624 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-11 30200 20625 ALOX5 240 DRUGGABLE GENOME, ENZYME VIA-2291 ATRELEUTON 30201 20626 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ANDROGENS 6770999 30202 20627 HTT 3064 DRUGGABLE GENOME TCMDC-125614 CHEMBL580609 30203 20628 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1201463 CODEINE POLISTIREX 30204 20629 ATXN2 6311 NA BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 30208 20630 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SULFASALAZINE SULFASALAZINE 22931300 30209 20631 CLDN18 51208 KINASE, DRUGGABLE GENOME CHEMBL2109427 ZOLBETUXIMAB 30211 20632 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME PLATINUM COMPOUND 27209210 30213 20633 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE CENISERTIB CENISERTIB 30214 20634 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DISULFIRAM DISULFIRAM 30216 20635 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME celecoxib CELECOXIB 22336956 30217 20636 SMN1 6606 DRUGGABLE GENOME RUTAECARPINE RUTAECARPINE 30219 20637 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX Tretinoin TRETINOIN 30220 20638 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME DHT ANDROSTANOLONE 16773205 30221 20639 SOD1 6647 ENZYME, DRUGGABLE GENOME OXYTETRACYCLINE OXYTETRACYCLINE 30222 20640 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DOVITINIB DOVITINIB 30226 20641 DDC 1644 ENZYME, DRUGGABLE GENOME Patrome 30229 20642 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CYMOXANIL CYMOXANIL 30230 20643 CDK11B 984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL445813 AT-7519 30231 20644 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CID 1245272 CHEMBL408850 30232 20645 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE BMS-936557 ELDELUMAB 30233 20646 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Vistusertib VISTUSERTIB 26725216 30234 20647 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME REGN910 NESVACUMAB 30235 20648 FZD1 8321 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, KINASE NICLOSAMIDE NICLOSAMIDE 23453073 30236 20649 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR DS-6051 30237 20650 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9422240, 1-286 30238 20651 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ERBB3 antibody 27196767 30239 20652 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor PI-103 PI-103 30240 20653 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE SERIBANTUMAB SERIBANTUMAB 20227043 30241 20654 MYO9B 4650 NA WORTMANNIN WORTMANNIN 15823093 30242 20655 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME Platinum compounds 29662106 30245 20656 POLK 51426 DNA REPAIR, ENZYME TAXIFOLIN TAXIFOLIN 30246 20657 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650310 30247 20658 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178103073 DESIRUDIN 30249 20659 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHOSMET PHOSMET 30252 20660 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME HYDROXYZINE PAMOATE HYDROXYZINE PAMOATE 30253 20661 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TRITIOZINE TRITIOZINE 30254 20662 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heteroaryl-carboxamide derivative 9 30256 20663 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Imidazo bicyclic iminium derivative 8 30257 20664 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ETOCRYLENE ETOCRYLENE 30259 20665 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-312948A GSK-312948A 30260 20666 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135651962 30261 20667 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SGN-14 10866315 30262 20668 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32x 30264 20669 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME ALPHA-DIFLUOROMETHYLORNITHINE 6144574 30265 20670 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GLYCYRRHIZIN GLYCYRRHIZIN 30268 20671 ENG 2022 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL2109321 CAROTUXIMAB 30269 20672 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 1 30270 20673 RRM2 6241 DRUGGABLE GENOME, ENZYME inhibitor 178101495 GEMCITABINE 30271 20674 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TIOTROPIUM TIOTROPIUM 30272 20675 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR 4SC-202 DOMATINOSTAT 30274 20676 HMGCR 3156 ENZYME, DRUGGABLE GENOME Poly-substituted azoles statin lactone derivative 2 30276 20677 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Herbimycin A 30277 20678 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE 9-AMINOCAMPTOTHECIN 9-AMINOCAMPTOTHECIN 10803925 30278 20679 NR1D1 9572 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME lithium LITHIUM 20348464 30279 20680 AKR1C3 8644 ENZYME, DRUGGABLE GENOME Nitrogen/sulfur-substituted estrene derivative 1 30280 20681 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR QUINALIZARIN QUINALIZARIN 30282 20682 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Pirbuterol PIRBUTEROL 30283 20683 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200332 PROTRIPTYLINE HYDROCHLORIDE 30286 20684 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR ALSTERPAULLONE ALSTERPAULLONE 30287 20685 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200382 BEPRIDIL HYDROCHLORIDE 30288 20686 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TCMDC-124479 CHEMBL587259 30289 20687 PSMD8 5714 NA inhibitor CHEMBL451887 CARFILZOMIB 30290 20688 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SELECTIVE ESTROGEN RECEPTOR MODULATORS 16198475 30292 20689 POLK 51426 DNA REPAIR, ENZYME NSC-61836 CHEMBL521171 30293 20690 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME GNF-PF-2301 CHEMBL578061 30294 20691 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TERTATOLOL TERTATOLOL 2903243 30295 20692 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 178102613 ISOGRANULATIMIDE 30298 20693 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-21 30299 20694 PSMC6 5706 NA inhibitor CHEMBL451887 CARFILZOMIB 30300 20695 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 178102301 RAF-265 30302 20696 IL1B 3553 KINASE, DRUGGABLE GENOME CYT013-IL1BQB 30303 20697 MAPT 4137 DRUGGABLE GENOME CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 30305 20698 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 30306 20699 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PIPOXOLAN HYDROCHLORIDE PIPOXOLAN HYDROCHLORIDE 30308 20700 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR toremifene TOREMIFENE 30309 20701 CD55 1604 DRUGGABLE GENOME, CELL SURFACE ETHANOL ALCOHOL 17383432 30310 20702 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PACHYRRIZINE PACHYRRIZINE 30312 20703 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME TRAMETINIB TRAMETINIB 30314 20704 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR TAE684 25688157 30315 20705 EPHB2 2048 KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 249565821 30317 20706 RORA 6095 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE citalopram CITALOPRAM 19846067 30318 20707 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 135650566 MAPROTILINE 30319 20708 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135651337 ISRAPAFANT 30321 20709 ATAD5 79915 NA GNF-PF-1307 CHEMBL585030 30322 20710 TOP2B 7155 DRUGGABLE GENOME, ENZYME Lomefloxacin LOMEFLOXACIN 30323 20711 PRKACB 5567 ENZYME, KINASE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE FASUDIL FASUDIL 22257127 30324 20712 FAAH 2166 ENZYME, DRUGGABLE GENOME Benzyl pyrrolyloxoacetamide derivative 2 30325 20713 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME LY294002 22871572 30327 20714 MPHOSPH8 54737 NA GOSSYPOL GOSSYPOL 30330 20715 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BISPHENOL A BISPHENOL A 30331 20716 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE RETIGABINE EZOGABINE 30332 20717 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 WIN-55212-2 WIN-552122 30333 20718 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CALCIPOTRIENE CALCIPOTRIENE 30334 20719 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME SB1518 PACRITINIB 30335 20720 TLR7 51284 DRUGGABLE GENOME Hydroxychloroquine HYDROXYCHLOROQUINE 30336 20721 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE amoxicillin AMOXICILLIN 30664875 30337 20722 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE AKT INHIBITOR MK2206 27297869 30339 20723 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ALITRETINOIN ALITRETINOIN 30341 20724 GMNN 51053 DRUGGABLE GENOME TCMDC-124681 CHEMBL536008 30342 20725 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER etoposide ETOPOSIDE 12969965 30344 20726 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR THIOTEPA THIOTEPA 30345 20727 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HEXACONAZOLE HEXACONAZOLE 30346 20728 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ASPIRIN ASPIRIN 22931300 30347 20729 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650056 CARBACYCLIN 30350 20730 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PEMIROLAST PEMIROLAST 30351 20731 HEBP1 50865 DRUGGABLE GENOME 1-phenyl-1,3,4-triazole derivative 2 30352 20732 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor TAK901 30353 20733 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Metipranolol METIPRANOLOL 30354 20734 CPA1 1357 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 252166827 30355 20735 BCHE 590 DRUGGABLE GENOME, ENZYME mivacurium MIVACURIUM 27031121 30356 20736 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 223365982 AC-480 30358 20737 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEBRISOQUIN SULFATE DEBRISOQUIN SULFATE 30359 20738 MSH6 2956 CLINICALLY ACTIONABLE, DNA REPAIR N/A 21242281,19125127,26582061 30360 20739 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER DOXYCYCLINE DOXYCYCLINE 11850258 30362 20740 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BMS-182874 BMS-182874 30363 20741 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US10149841, Compound 1 30364 20742 ALOX15B 247 DRUGGABLE GENOME, ENZYME GNF-PF-5114 CHEMBL601952 30366 20743 POLK 51426 DNA REPAIR, ENZYME CATECHIN CATECHIN 30369 20744 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE SULINDAC SULINDAC 12654560 30370 20745 GMNN 51053 DRUGGABLE GENOME NSC-102742 CHEMBL1519374 30372 20746 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE CNS-5161 CNS-5161 30373 20747 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR KINASE INHIBITOR 16951152 30374 20748 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME SB-216763 SB-216763 30375 20749 TUBA1C 84790 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 30376 20750 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE SORAFENIB TOSYLATE SORAFENIB TOSYLATE 30377 20751 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE CEFACLOR CEFACLOR 22166395 30379 20752 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SR-2640 SR-2640 30380 20753 POLK 51426 DNA REPAIR, ENZYME METHYLDOPA METHYLDOPA 30381 20754 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Levobetaxolol LEVOBETAXOLOL 30382 20755 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 30385 20756 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL917 FLOXURIDINE 30387 20757 NDUFV3 4731 ENZYME inhibitor CHEMBL3545135 NV-128 30390 20758 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 315661146 PF-03882845 30391 20759 KDM4A 9682 DRUGGABLE GENOME, ENZYME GBR-12909 VANOXERINE 30392 20760 TUBB 203068 DRUGGABLE GENOME Taxol PACLITAXEL 30394 20761 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PF-04691502 PF-04691502 30396 20762 DNER 92737 NA OTX-015 BIRABRESIB 30397 20763 GGPS1 9453 DRUGGABLE GENOME, ENZYME DIGERANYL BISPHOSPHONATE DIGERANYL BISPHOSPHONATE 24726306 30398 20764 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE ALPHA-TOCOPHEROL VITAMIN E 16679868 30399 20765 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE LY-2090314 LY-2090314 30400 20766 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME DNDI1416917 CHEMBL1335833 30402 20767 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-638080 CHEMBL136344 30404 20768 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PGF2alpha 30406 20769 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE NAPROXEN NAPROXEN 1908176 30407 20770 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL2104992 VESTIPITANT MESYLATE 30408 20771 PSMC2 5701 PROTEASE, TRANSCRIPTION FACTOR inhibitor CARFILZOMIB CARFILZOMIB 30409 20772 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CID2350207 CHEMBL259615 30410 20773 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMOXICILLIN AMOXICILLIN 12152002 30411 20774 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE (4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE (4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE 30413 20775 TXNRD1 7296 DRUGGABLE GENOME Triazole gold complexe 2 30414 20776 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME EFEGATRAN SULFATE HYDRATE 30415 20777 F11 2160 DRUGGABLE GENOME, PROTEASE, ENZYME EP-7041 30416 20778 MAPT 4137 DRUGGABLE GENOME LMT-X 30418 20779 STING1 340061 CLINICALLY ACTIONABLE, KINASE agonist 381118837 30419 20780 HEBP1 50865 DRUGGABLE GENOME Benzamide derivative 5 30421 20781 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR Platinum compounds 18538445,18483375,22134350,21642870,24361227 30423 20782 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1023 BEXAROTENE 30424 20783 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME oxaliplatin OXALIPLATIN 24338217,20530282 30425 20784 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME amphetamine AMPHETAMINE 30426 20785 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 L-741742 CHEMBL444309 30427 20786 MAPT 4137 DRUGGABLE GENOME Z-PRO-PROLINAL Z-PRO-PROLINAL 30428 20787 PSMD10 5716 TRANSCRIPTION FACTOR BINDING inhibitor BORTEZOMIB BORTEZOMIB 30429 20788 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody 310264711 ISTIRATUMAB 30431 20789 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR RG-1530 RG-1530 30433 20790 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME CPT-11 IRINOTECAN HYDROCHLORIDE 15956246 30434 20791 BAZ2B 29994 NA 3-MORPHOLINOSYDNONIMINE HCL CHEMBL538104 30437 20792 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Dacomitinib DACOMITINIB 24857124,28363995,21764376,26561558,27913578,25456362,25939761,26206867,18089823 30438 20793 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE DASATINIB DASATINIB 30440 20794 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME TRIAZOLAM TRIAZOLAM 30441 20795 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL488436 AZD-5438 30443 20796 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE DOXORUBICIN DOXORUBICIN 12576455 30444 20797 ACAT2 39 ENZYME inhibitor 381118860 30445 20798 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PENTABROMOPHENOL PENTABROMOPHENOL 30446 20799 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ROSIGLITAZONE ROSIGLITAZONE 22819190,22934537,24890090,26384286,22070604,19719236,25442322,23273519,15745794,21030263,16680159,25497132 30448 20800 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RECOMBINANT HUMAN INTERLEUKIN-2 12174877 30450 20801 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102236 30451 20802 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME IL-6 8096510 30452 20803 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme15-3 30453 20804 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE TOZASERTIB TOZASERTIB 30454 20805 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME agonist 135651492 GLYCINE 30455 20806 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME nicotine NICOTINE 17015050,17638512,11470993,18004205,25652250 30456 20807 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SOTALOL SOTALOL 22931300 30459 20808 FAAH 2166 ENZYME, DRUGGABLE GENOME Tetra-substituted urea derivative 1 30460 20809 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DESVENLAFAXINE DESVENLAFAXINE 30461 20810 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME HL-018 30462 20811 KDM4A 9682 DRUGGABLE GENOME, ENZYME NOREPINEPHRINE NOREPINEPHRINE 30463 20812 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR OXYQUINOLINE OXYQUINOLINE 30464 20813 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200382 BEPRIDIL HYDROCHLORIDE 30465 20814 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2006015124 30466 20815 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Pazopanib PAZOPANIB 30467 20816 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Cyclic sulfonamide derivative 2 30469 20817 FAAH 2166 ENZYME, DRUGGABLE GENOME risperidone RISPERIDONE 20631561 30470 20818 DPP9 91039 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 363894187 30471 20819 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME BRYOSTATIN BRYOSTATIN 30472 20820 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 385612170 KZR-616 30473 20821 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor PELITINIB PELITINIB 30474 20822 ATXN2 6311 NA GNF-PF-3641 CHEMBL599098 30475 20823 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR GM-CSF REGRAMOSTIM 8260700 30476 20824 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME NSC-677438 CHEMBL118678 30478 20825 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE TETRODOTOXIN TETRODOTOXIN 30479 20826 FKBP4 2288 DRUGGABLE GENOME IMMUNOSUPPRESSIVE 1716886 30480 20827 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 3,6-DIMETHOXYFLAVONE 3,6-DIMETHOXYFLAVONE 30481 20828 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AMOXICILLIN AMOXICILLIN 22931300 30482 20829 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME agonist 178101033 30483 20830 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Kevetrin 4-ISOTHIOUREIDOBUTYRONITRILE 30484 20831 ABCC5 10057 DRUGGABLE GENOME, ABC TRANSPORTER, TRANSPORTER FLOXURIDINE FLOXURIDINE 20930123 30487 20832 F5 2153 DRUGGABLE GENOME inhibitor 178103394 30488 20833 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GNF-PF-5510 CHEMBL578741 30492 20834 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING 2-ENE-VALPROATE CHEMBL117487 17566732 30493 20835 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PMID25416646-Compound-Figure2-N 30495 20836 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 384403651 30497 20837 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-9 30499 20838 POLK 51426 DNA REPAIR, ENZYME GNF-PF-5510 CHEMBL578741 30500 20839 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GW-409544 30501 20840 CD27 939 PROTEASE INHIBITOR, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PROTEASE INHIBITORS 17309824 30502 20841 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR PHENYLSTIBONIC ACID PHENYLSTIBONIC ACID 30504 20842 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor PALBOCICLIB PALBOCICLIB 30505 20843 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Recombinant RGD-hirudin 30507 20844 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 VASOPRESSIN VASOPRESSIN 18431272 30509 20845 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE IRINOTECAN IRINOTECAN 25003995,23360284,24507920 30510 20846 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor MK-1775 ADAVOSERTIB 30513 20847 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AMPHOTERICIN B AMPHOTERICIN B 22931300 30514 20848 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME paliperidone PALIPERIDONE 30516 20849 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE IMMUNOSUPPRESSIVE 17015702 30517 20850 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME SGI-1776 SGI-1776 26472029 30518 20851 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY DEXAMETHASONE DEXAMETHASONE 1174132 30521 20852 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE MORPHINE MORPHINE 12829326 30522 20853 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL428647 PACLITAXEL 30523 20854 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE corticosteroids 26774659,19932356,24279851 30524 20855 CD38 952 CELL SURFACE, DRUGGABLE GENOME CD38 CAR T cells 30525 20856 AKR1B1 231 DRUGGABLE GENOME, ENZYME ANTISERUM 2158468 30526 20857 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ENDO-ATROPINE ENDO-ATROPINE 22931300 30527 20858 ENO2 2026 CELL SURFACE SODIUM BUTYRATE 7276941 30529 20859 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2103838 DILMAPIMOD 30530 20860 RIPK2 8767 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 384403681 30531 20861 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200833 DIPIVEFRIN HYDROCHLORIDE 30532 20862 KCND3 3752 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 30533 20863 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL1980391 RG-1530 30534 20864 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 30535 20865 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME 2-HYDROXYPHENAZINE 5,10-DIOXIDE CHEMBL179611 30536 20866 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR EXEMESTANE EXEMESTANE 30537 20867 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHLORANIL CHLORANIL 30542 20868 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-37 30544 20869 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-16 30545 20870 GUCY2C 2984 DRUGGABLE GENOME, KINASE antibody 252827376 30548 20871 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR citalopram CITALOPRAM 18195729 30551 20872 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Pemetrexed PEMETREXED 27213589 30553 20873 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GRAVEOLINE GRAVEOLINE 30555 20874 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 310264722 30556 20875 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER VCR 9864280 30559 20876 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1201747 ALCAFTADINE 30560 20877 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER SU-6656 CHEMBL605003 30561 20878 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR CX-4945 SILMITASERTIB 30562 20879 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125232 CHEMBL531079 30563 20880 NOS1 4842 DRUGGABLE GENOME, ENZYME ADJUVANT 8991992 30565 20881 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ritonavir RITONAVIR 30567 20882 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IDARUBICIN IDARUBICIN 30568 20883 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 20 30570 20884 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1417181 CHEMBL1537417 30572 20885 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-BROMOETHANOL 2-BROMOETHANOL 30575 20886 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 30578 20887 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-516 CHEMBL602970 30579 20888 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Geminally-substituted cyanoethylpypazolo pyridone derivative 2 30580 20889 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PWT-33597 30581 20890 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 STAVUDINE STAVUDINE 22931300 30582 20891 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEXPROPRANOLOL DEXPROPRANOLOL 30583 20892 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ACRIDIN-1-YLAMINE CHEMBL146525 30584 20893 UGT1A10 54575 DRUGGABLE GENOME, ENZYME febuxostat FEBUXOSTAT 27798726 30587 20894 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1421 DASATINIB 30588 20895 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CIS-(Z)-FLUPENTHIXOL DIHYDROCHLORIDE CHEMBL1256995 30589 20896 XDH 7498 DRUGGABLE GENOME, ENZYME Oxypurinol OXYPURINOL 30591 20897 ATAD5 79915 NA MMV009085 CHEMBL581225 30593 20898 CAMK1 8536 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME LINIFANIB LINIFANIB 30594 20899 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ISOVELLERAL ISOVELLERAL 30595 20900 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME NBQX NBQX 30597 20901 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SPIRAMIDE SPIRAMIDE 30598 20902 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CSL 360 30599 20903 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GENISTEIN GENISTEIN 10400830 30600 20904 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Mocetinostat MOCETINOSTAT 27443263 30601 20905 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SENNOSIDE B SENNOSIDE B 30603 20906 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 135650607 MIBOLERONE 30604 20907 ITGB6 3694 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor CHEMBL2109623 STX-100 30605 20908 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4809 CHEMBL585439 30606 20909 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-1919 CHEMBL576409 30607 20910 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE PROPOFOL PROPOFOL 17223697 30608 20911 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LE-SN38 30609 20912 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE ZM-447439 CHEMBL202721 30612 20913 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER TRICHOSTATIN A 17332941 30614 20914 GALC 2581 ENZYME, DRUGGABLE GENOME BUSULFAN BUSULFAN 2034480,8101401 30615 20915 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE 30616 20916 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 348353615 30617 20917 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Trastuzumab TRASTUZUMAB 30618 20918 CBX1 10951 NA NSC-130813 CHEMBL463783 30619 20919 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE R115777 16101130 30621 20920 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE amphetamine AMPHETAMINE 30623 20921 CYBB 1536 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME, ENZYME inhibitor 363894227 30625 20922 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR INDOLE-3-CARBINOL INDOLE-3-CARBINOL 30626 20923 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 328083525 NEMIRALISIB 30628 20924 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SR-2640 SR-2640 30631 20925 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ENOXOLONE ENOXOLONE 22931300 30632 20926 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SAR-113945 SAR-113945 21896960 30633 20927 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR NKP-1339 IT-139 30634 20928 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651280 TRIPITRAMINE 30635 20929 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL457 GEMFIBROZIL 30638 20930 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 arteether 18064444,18979093,19926036,19851082,18350255,12920490,12844133 30639 20931 KMO 8564 DRUGGABLE GENOME, ENZYME Aryl pyrimidine derivative 6 30640 20932 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME N,N'-DIPHENYL-P-PHENYLENEDIAMINE N,N'-DIPHENYL-P-PHENYLENEDIAMINE 30641 20933 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL1201748 CABAZITAXEL 30642 20934 ASPH 444 ENZYME, TRANSPORTER warfarin WARFARIN 27488176 30644 20935 ATP2C1 27032 ENZYME, TRANSPORTER, DRUGGABLE GENOME ISOFLURANE ISOFLURANE 30645 20936 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME 1,5-NAPHTHALENEDIAMINE CHEMBL538965 30648 20937 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME U-0126 U-0126 30649 20938 ATAD5 79915 NA HELENALIN HELENALIN 30652 20939 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor PWT33597 30655 20940 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME IONOMYCIN IONOMYCIN 12193581,15845548 30658 20941 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE GW441756X GW441756X 30659 20942 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL450 METHARBITAL 30660 20943 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR fluoxetine FLUOXETINE 18794724 30663 20944 ATP1A2 477 ENZYME, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME inhibitor CHEMBL254219 DIGITOXIN 30664 20945 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NITRALIN NITRALIN 30665 20946 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL274654 ORANTINIB 30667 20947 PSMC3 5702 NA inhibitor CHEMBL2103884 OPROZOMIB 30668 20948 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME CANDESARTAN CILEXETIL CANDESARTAN CILEXETIL 30669 20949 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ribavirin RIBAVIRIN 25713999,27139837 30671 20950 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651070 30676 20951 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE CADMIUM ACETATE CADMIUM ACETATE 30677 20952 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PROCHLORPERAZINE PROCHLORPERAZINE 30678 20953 TPP1 1200 PROTEASE, ENZYME, DRUGGABLE GENOME cerliponase alfa 30680 20954 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist CHEMBL1082407 ENZALUTAMIDE 30681 20955 XDH 7498 DRUGGABLE GENOME, ENZYME VCR 9461035 30682 20956 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 6ALPHA-METHYLPREDNISOLONE ACETATE METHYLPREDNISOLONE ACETATE 30684 20957 PSMC6 5706 NA CARFILZOMIB CARFILZOMIB 24524217 30685 20958 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME 6-METHOXY-HARMALAN CHEMBL338115 30686 20959 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PSC-833 15456083 30687 20960 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TAMOXIFEN TAMOXIFEN 3793272 30688 20961 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Azacitidine AZACITIDINE 30691 20962 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NICARDIPINE HYDROCHLORIDE NICARDIPINE HYDROCHLORIDE 30692 20963 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PSORALEN PSORALEN 30693 20964 BMP7 655 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR methotrexate METHOTREXATE 26590194 30694 20965 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1671 PROPRANOLOL HYDROCHLORIDE 30696 20966 CBL 867 KINASE, ENZYME, CLINICALLY ACTIONABLE SU11274 28835699 30698 20967 SLC5A6 8884 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSPORTER Gabapentin enacarbil 30699 20968 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-13 30701 20969 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Peptidomimetic analog 1 30702 20970 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR SNS-314 SNS-314 30703 20971 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-367089 CHEMBL1543865 30704 20972 HSPA4 3308 NA Minnelide MINNELIDE 30707 20973 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Rogaratinib ROGARATINIB 30711 20974 GMNN 51053 DRUGGABLE GENOME BENZIODARONE BENZIODARONE 30713 20975 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TPA ALTEPLASE 1394224 30716 20976 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE FELBAMATE FELBAMATE 30717 20977 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 354702207 30718 20978 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 pyrazinamide PYRAZINAMIDE 20941486 30719 20979 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TCMDC-124327 CHEMBL581929 30720 20980 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 223366096 30724 20981 UTRN 7402 NA SMT-C1100 EZUTROMID 30725 20982 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051814 30726 20983 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME A-substituted phenylpropionic acid derivative 2 30727 20984 ALOX15 246 ENZYME, DRUGGABLE GENOME 3,3',4'-TRIHYDROXYFLAVONE CHEMBL122701 30730 20985 SETD4 54093 METHYL TRANSFERASE daunorubicin DAUNORUBICIN 19204081 30734 20986 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE AMCINONIDE AMCINONIDE 30735 20987 CPS1 1373 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME positive modulator CHEMBL1201780 CARGLUMIC ACID 30736 20988 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Tesofensine TESOFENSINE 30737 20989 PSMC1 5700 PROTEASE inhibitor CHEMBL2103884 OPROZOMIB 30738 20990 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 318164817 30739 20991 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1416955 CHEMBL1327172 30740 20992 IRF3 3661 KINASE, TRANSCRIPTION FACTOR IFN 10692430 30743 20993 HTT 3064 DRUGGABLE GENOME NITROVIN NITROVIN 30745 20994 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Chloroprocaine CHLOROPROCAINE 30746 20995 BAZ2B 29994 NA NSC-367089 CHEMBL1543865 30747 20996 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650690 30748 20997 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DE-098 30749 20998 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE STM 434 30750 20999 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE Tricyclic compound 5 30757 21000 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROCHLORAZ PROCHLORAZ 30758 21001 CD36 948 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME, CLINICALLY ACTIONABLE antagonist 404859035 30759 21002 TRPC4 7223 ION CHANNEL, KINASE, DRUGGABLE GENOME, CELL SURFACE activator 252166584 30760 21003 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME R-RUGULACTONE R-RUGULACTONE 19093800 30762 21004 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MK-2461 MK-2461 30763 21005 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME VASOPRESSIN VASOPRESSIN 15845548 30764 21006 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor DINACICLIB DINACICLIB 30765 21007 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Aryl methoxyacrylate derivative 2 30767 21008 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE BMS-690514 BMS-690514 23490650 30772 21009 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Imidazo bicyclic iminium derivative 6 30773 21010 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102757 30774 21011 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE GLUCOCORTICOID 10739632 30775 21012 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GENISTEIN GENISTEIN 30777 21013 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL463981 BEGACESTAT 30778 21014 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL LORAZEPAM LORAZEPAM 30779 21015 PDE4A 5141 DRUGGABLE GENOME, ENZYME Oglemilast OGLEMILAST 18660832 30780 21016 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PHENYLBUTYRYLHYDROXAMIC ACID PHENYLBUTYRYLHYDROXAMIC ACID 21874153 30781 21017 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107771 RALFINAMIDE 30782 21018 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PARDOPRUNOX PARDOPRUNOX 30783 21019 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PH-011685 CHEMBL126804 30784 21020 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PF-05212384 GEDATOLISIB 12068308,21325073 30785 21021 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE FUSARIC ACID FUSARIC ACID 30787 21022 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ZM-449829 CHEMBL154580 30790 21023 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME LAVENDUSTIN C LAVENDUSTIN C 30791 21024 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME Marimastat MARIMASTAT 30793 21025 GMNN 51053 DRUGGABLE GENOME DNDI1417614 CHEMBL1567571 30794 21026 TAT 6898 ENZYME MITOMYCIN-C 610 30795 21027 ECE1 1889 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE inhibitor 178103121 30796 21028 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ROSIGLITAZONE ROSIGLITAZONE 30798 21029 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Nerenone 30800 21030 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME FILGRASTIM FILGRASTIM 30801 21031 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DEXAMETHASONE DEXAMETHASONE 23276449,20308375 30803 21032 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE GANTENERUMAB GANTENERUMAB 30804 21033 ATAD5 79915 NA DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 30805 21034 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545423 AZD-1208 30806 21035 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650612 MK-0767 30807 21036 ATAD5 79915 NA CV-1808 CHEMBL1256672 30808 21037 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FTI-277 CHEMBL135561 30809 21038 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AMSACRINE AMSACRINE 19155103,22537681,17911018,19725581,25626146 30810 21039 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME IDDBCP161883 30812 21040 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-32 30813 21041 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor NIRAPARIB NIRAPARIB 30814 21042 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE CSA CYCLOSPORINE 11571455,11817607,11683823 30815 21043 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE TRETINOIN TRETINOIN 19965647,21719597 30816 21044 HBB 3043 DRUGGABLE GENOME, ENZYME HYDROXYCAMPTOTHECIN HYDROXYCAMPTOTHECIN 30818 21045 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL494 ILOPROST 30820 21046 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LAMOTRIGINE LAMOTRIGINE 22931300 30821 21047 MAPT 4137 DRUGGABLE GENOME AG-808 CHEMBL68534 30822 21048 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE THEOPHYLLINE THEOPHYLLINE 10666409 30824 21049 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Iboctadekin + rituximab 30825 21050 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-97 30826 21051 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417195 CHEMBL1303948 30827 21052 PEMT 10400 ENZYME CHEMBL2109637 HUHMFG1 30828 21053 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Pyrimidine derivative 31 30829 21054 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PINACIDIL PINACIDIL 30830 21055 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LINEZOLID LINEZOLID 24044938 30832 21056 TLR7 51284 DRUGGABLE GENOME GS-9620 VESATOLIMOD 30833 21057 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PD-98059 CHEMBL35482 30834 21058 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME Masitinib MASITINIB 30835 21059 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 387065602 30836 21060 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 2-BENZOYL-5-METHOXYBENZOQUINONE 2-BENZOYL-5-METHOXYBENZOQUINONE 30838 21061 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker 178100970 30839 21062 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE SCH-527123 NAVARIXIN 30841 21063 FAAH 2166 ENZYME, DRUGGABLE GENOME Azole derivative 1 30842 21064 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME 3,4,5-TRIHYDROXY-BENZOIC ACID PHENETHYL ESTER CHEMBL151146 30843 21065 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LAVENDUSTIN A LAVENDUSTIN A 30844 21066 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AZD4547 26936917 30845 21067 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME ILORASERTIB ILORASERTIB 30846 21068 PDE4B 5142 DRUGGABLE GENOME, ENZYME OX-914 HT-0712 30847 21069 STAT5A 6776 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AZD-1480 AZD-1480 21138246 30848 21070 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TETRADIFON TETRADIFON 30850 21071 PRKG1 5592 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 178101884 GSK-690693 30855 21072 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE LAPATINIB LAPATINIB 18408761 30857 21073 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Phenylpyrrolidinone derivative 5 30860 21074 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIMETHISTERONE DIMETHISTERONE 30861 21075 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MANEB MANEB 30862 21076 ATXN2 6311 NA NSC-724440 CHEMBL515617 30863 21077 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Oxazolyl methylthiothiazole derivative 1 30864 21078 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ZAFIRLUKAST ZAFIRLUKAST 22931300 30865 21079 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME AVOBENZONE AVOBENZONE 30866 21080 NME2 4831 KINASE lamivudine LAMIVUDINE 30867 21081 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING CLOTRIMAZOLE CLOTRIMAZOLE 16680159 30868 21082 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR GSK2981278 30870 21083 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME US8609715, A-1 30871 21084 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100475 30872 21085 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR fluoxetine FLUOXETINE 18195729 30873 21086 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME inhibitor 53801012 30874 21087 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Tanespimycin TANESPIMYCIN 26009011 30875 21088 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE Peptide analog 59 30876 21089 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CRIZOTINIB CRIZOTINIB 30877 21090 GMNN 51053 DRUGGABLE GENOME ANGUSTIBALIN ANGUSTIBALIN 30878 21091 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR methadone METHADONE 31940240 30879 21092 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE STICTIC ACID STICTIC ACID 30880 21093 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME MELAGATRAN MELAGATRAN 30882 21094 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL1201752 IXABEPILONE 30883 21095 CCR6 1235 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR agonist 135652054 30886 21096 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME DIMETHYLADENINE DIMETHYLADENINE 30888 21097 THOP1 7064 DRUGGABLE GENOME, PROTEASE Karenitecin KARENITECIN 30890 21098 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200833 DIPIVEFRIN HYDROCHLORIDE 30891 21099 GLS 2744 ENZYME N'-(2,4-DIHYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE CHEMBL199592 30892 21100 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE hmg coa reductase inhibitors 30893 21101 PDE5A 8654 ENZYME, DRUGGABLE GENOME Papaverine PAPAVERINE 30895 21102 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-159 CHEMBL599924 30896 21103 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PMID25416646-Compound-Figure5-A 30898 21104 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Ponatinib PONATINIB 25122427 30899 21105 ALDH1A1 216 DRUGGABLE GENOME, ENZYME vitamin a 30901 21106 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR CISPLATIN CISPLATIN 14977831,24595080 30902 21107 GMNN 51053 DRUGGABLE GENOME NITROXOLINE NITROXOLINE 30904 21108 ACP1 52 ENZYME, DRUGGABLE GENOME, PROTEIN PHOSPHATASE NCI-372939 CHEMBL84440 30907 21109 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE MMF MYCOPHENOLATE MOFETIL 14550820 30908 21110 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102695 30909 21111 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 252827426 30910 21112 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME AMD-070 MAVORIXAFOR 30911 21113 TXNRD1 7296 DRUGGABLE GENOME Palmarumycin derivative 4 30913 21114 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Oxaliplatin OXALIPLATIN 26432108 30914 21115 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR activator ILOPROST ILOPROST 30916 21116 MAP2K3 5606 KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE ROSIGLITAZONE ROSIGLITAZONE 11591391 30918 21117 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652040 30919 21118 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME isoniazid ISONIAZID 28389387 30922 21119 ATAD5 79915 NA 1,2-BIS(3-FLUOROBENZYLIDENE)HYDRAZINE CHEMBL371811 30926 21120 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME 7RH 26855149 30927 21121 FAAH 2166 ENZYME, DRUGGABLE GENOME JNJ-42165279 JNJ-42165279 30928 21122 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE JNJ-38877605 JNJ-38877605 30929 21123 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR R-1487 R-1487 30931 21124 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OUABAIN OUABAIN 30932 21125 RPL13 6137 NA docetaxel DOCETAXEL 20038957 30933 21126 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR GSK3196165 OTILIMAB 30934 21127 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 2-ENE-VALPROATE CHEMBL117487 17566732 30936 21128 IL1B 3553 KINASE, DRUGGABLE GENOME Ibudilast IBUDILAST 30937 21129 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME SEMAXANIB SEMAXANIB 30938 21130 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME TAK-379 30939 21131 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ACACETIN ACACETIN 30940 21132 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CHEMBL1341 METHOXYFLURANE 30941 21133 ATXN2 6311 NA OSAJIN OSAJIN 30943 21134 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR RETASPIMYCIN RETASPIMYCIN 30945 21135 PLEKHH2 130271 NA atenolol ATENOLOL 27670767 30946 21136 GMNN 51053 DRUGGABLE GENOME ALPHA,BETA-DEHYDROCURVULARIN CHEMBL482050 30949 21137 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702258 DERAZANTINIB 30951 21138 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LITHOCHOLIC ACID LITHOCHOLIC ACID 30953 21139 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR AZITHROMYCIN AZITHROMYCIN 16113783 30954 21140 GLA 2717 ENZYME, DRUGGABLE GENOME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 30955 21141 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME RG7155 30958 21142 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650799 PD-156707 30959 21143 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A1 30960 21144 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME PF-562271 PF-00562271 30962 21145 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor DACTOLISIB DACTOLISIB 30964 21146 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TROLEANDOMYCIN TROLEANDOMYCIN 22931300 30965 21147 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE LOVASTATIN LOVASTATIN 17472962 30966 21148 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 178102337 SORAFENIB 30967 21149 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Lusutrombopag LUSUTROMBOPAG 30969 21150 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GBR-12909 VANOXERINE 30970 21151 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME SB-415286 CHEMBL322970 30972 21152 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME AZD-1775 ADAVOSERTIB 30973 21153 EPHA4 2043 DRUGGABLE GENOME, KINASE, CELL SURFACE, TYROSINE KINASE inhibitor 249565821 30974 21154 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME atorvastatin ATORVASTATIN 30975 21155 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE HKI-272 NERATINIB 30976 21156 HTT 3064 DRUGGABLE GENOME GSK311739 30977 21157 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR LEVOFLOXACIN LEVOFLOXACIN 12714806 30978 21158 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 310264723 EDICOTINIB 30979 21159 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ESTROGEN ESTROGEN 30984 21160 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NITROFEN NITROFEN 30986 21161 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GO-6976 GO-6976 30989 21162 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000201681 CHEMBL602135 30990 21163 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-26 30991 21164 SLC15A4 121260 DRUGGABLE GENOME, TRANSPORTER 178101385 30995 21165 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL107 COLCHICINE 30996 21166 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 328083502 30997 21167 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GSK269962A 30998 21168 KDM5C 8242 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 178103605 31000 21169 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR 4-(4-AMINOPHENYL)BUTANOIC ACID CHEMBL1650245 24044874 31001 21170 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR TRAMADOL TRAMADOL 15464068 31004 21171 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME Pyrazolo-triazine derivative 1 31005 21172 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TAZAROTENE TAZAROTENE 31006 21173 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR OXYMETHOLONE OXYMETHOLONE 31008 21174 MDM4 4194 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, DRUGGABLE GENOME docetaxel DOCETAXEL 24958282 31009 21175 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 354702226 31012 21176 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Tetrahydrofolic acid 31013 21177 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE AZD-1775 ADAVOSERTIB 31014 21178 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SNS-314 SNS-314 31015 21179 DDC 1644 ENZYME, DRUGGABLE GENOME inhibitor 178101902 31017 21180 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL378544 VINBLASTINE SULFATE 31018 21181 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CISPLATIN CISPLATIN 16079468 31019 21182 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HYDROQUINONE HYDROQUINONE 17118622 31020 21183 POLI 11201 DNA REPAIR FENOLDOPAM BROMIDE FENOLDOPAM BROMIDE 31021 21184 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING ZINC 03369470 CHEMBL599013 31023 21185 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER JQ1 24231268 31024 21186 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DACTINOMYCIN DACTINOMYCIN 31026 21187 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HYDROCORTISONE HYDROCORTISONE 31028 21188 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE Peptide analog 56 31029 21189 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor AS703569 CENISERTIB 31030 21190 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZARIBINE AZARIBINE 31031 21191 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist,antagonist 178102776 CP-195543 31033 21192 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR antagonist CHEMBL1358 FULVESTRANT 31040 21193 COL1A2 1278 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 31041 21194 GMNN 51053 DRUGGABLE GENOME GNF-PF-98 CHEMBL244023 31042 21195 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER METHYL 4-(3-METHOXYBENZAMIDO)BENZOATE CHEMBL1214407 31043 21196 CA1 759 DRUGGABLE GENOME, ENZYME CHLOROTHIAZIDE CHLOROTHIAZIDE 31045 21197 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FINASTERIDE FINASTERIDE 22931300 31046 21198 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 178102681 WORTMANNIN 31047 21199 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor VALPROIC ACID DEPAKOTE 31048 21200 KDM4A 9682 DRUGGABLE GENOME, ENZYME THIOGUANOSINE THIOGUANOSINE 31049 21201 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL285674 ESTAZOLAM 31050 21202 POLI 11201 DNA REPAIR MYRICETIN MYRICETIN 31051 21203 CBL 867 KINASE, ENZYME, CLINICALLY ACTIONABLE N/A 26230957,23690417,19901108 31052 21204 ALOX5AP 241 DRUGGABLE GENOME inhibitor CHEMBL1922660 FIBOFLAPON 31053 21205 ATXN2 6311 NA CP-55940 CP-55940 31056 21206 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE R1507 31058 21207 PAPPA 5069 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE ANTISERUM 2475160 31059 21208 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Phthalazine ketone derivative 2 31061 21209 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CLIOQUINOL CLIOQUINOL 23799643 31063 21210 CSF3 1440 GROWTH FACTOR, DRUGGABLE GENOME F-627 BENEGRASTIM 31064 21211 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CARVEDILOL CARVEDILOL 31066 21212 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Diaminopyridine analog 5 31067 21213 SFTPA1 653509 DRUGGABLE GENOME HEPARIN HEPARIN 7980398 31069 21214 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE Clofibrate CLOFIBRATE 31070 21215 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1721885 SU-014813 31073 21216 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 405067337 31074 21217 P2RX4 5025 ION CHANNEL, DRUGGABLE GENOME antagonist 336446927 31076 21218 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CLINAFLOXACIN CLINAFLOXACIN 31077 21219 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PYROGALLOL PYROGALLOL 31079 21220 HDC 3067 DRUGGABLE GENOME, ENZYME Lixivaptan LIXIVAPTAN 31080 21221 ALDH1A1 216 DRUGGABLE GENOME, ENZYME LINOLEIC ACID LINOLEIC ACID 31081 21222 GMNN 51053 DRUGGABLE GENOME OTILONIUM OTILONIUM 31082 21223 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ALPHA-TOCOPHEROL VITAMIN E 7649489 31083 21224 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXYFLUORFEN OXYFLUORFEN 31084 21225 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE OLAPARIB OLAPARIB 28148839 31088 21226 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE cocaine COCAINE 11840318,16387451,31246565 31089 21227 BAZ2B 29994 NA PROMETHAZINE HYDROCHLORIDE PROMETHAZINE HYDROCHLORIDE 31090 21228 ADRM1 11047 ENZYME CARFILZOMIB CARFILZOMIB 24524217 31091 21229 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME inhibitor BAY869766 31092 21230 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor 178101975 31093 21231 PML 5371 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE tretinoin TRETINOIN 31094 21232 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178103494 IBRUTINIB 31096 21233 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE GONADOTROPINS 18321442 31098 21234 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL87992 ESLICARBAZEPINE ACETATE 31099 21235 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR EUPAFOLIN EUPAFOLIN 31100 21236 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL861 MEPHENYTOIN 31101 21237 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL ethanol ALCOHOL 31634677 31102 21238 CALR 811 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME OLTIPRAZ OLTIPRAZ 15961673 31105 21239 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PONATINIB PONATINIB 22238366,26619011,18552176,23908597,23002168 31106 21240 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1946170 REGORAFENIB 31107 21241 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 328083456 31108 21242 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GOSSYPOL GOSSYPOL 31109 21243 ATAD5 79915 NA PD-98059 CHEMBL35482 31110 21244 CA2 760 DRUGGABLE GENOME, ENZYME IL-3 11112384 31111 21245 NOS2 4843 DRUGGABLE GENOME, ENZYME RHIL-11 10587516 31112 21246 STX4 6810 CELL SURFACE phenprocoumon PHENPROCOUMON 21063236 31113 21247 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102272 31114 21248 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ETHYNODIOL DIACETATE 31117 21249 IPO9 55705 NA MKC-1 ENMD-981693 31118 21250 RACGAP1 29127 NA TCMDC-125528 CHEMBL375673 31120 21251 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125606 CHEMBL536166 31122 21252 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CEPHARANTHINE CEPHARANTHINE 31123 21253 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL931 HALOTHANE 31128 21254 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE KAEMPFEROL KAEMPFEROL 31130 21255 ALOX15 246 ENZYME, DRUGGABLE GENOME DNDI1417523 CHEMBL598663 31131 21256 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PERUVOSIDE PERUVOSIDE 31132 21257 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME STAVUDINE STAVUDINE 22931300 31134 21258 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CHELERYTHRINE CHELERYTHRINE 31136 21259 GNE 10020 ENZYME, KINASE GNE Lipoplex 31137 21260 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME inhibitor 249565871 31138 21261 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Dihydrodiazepinocarbazolone derivative 1 31140 21262 DEPTOR 64798 KINASE inhibitor OSI-027 OSI-027 31141 21263 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 310264777 31143 21264 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1723 ALFUZOSIN HYDROCHLORIDE 31145 21265 POLK 51426 DNA REPAIR, ENZYME N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 31150 21266 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL3545395 BI-811283 31151 21267 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME activator 404859097 31152 21268 POLK 51426 DNA REPAIR, ENZYME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 31153 21269 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL BENZYL ISOTHIOCYANATE BENZYL ISOTHIOCYANATE 26263397 31156 21270 GAA 2548 DRUGGABLE GENOME, ENZYME HYDROXYTYROSOL HYDROXYTYROSOL 31157 21271 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 31158 21272 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DEXBROMPHENIRAMINE DEXBROMPHENIRAMINE 31159 21273 NOS2 4843 DRUGGABLE GENOME, ENZYME FLUOXETINE FLUOXETINE 16413968 31160 21274 BBOX1 8424 DRUGGABLE GENOME EBSELEN EBSELEN 25266780 31164 21275 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DEBRISOQUIN SULFATE DEBRISOQUIN SULFATE 31166 21276 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1,8-DINITRO-NAPHTHALENE CHEMBL167529 31167 21277 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 31169 21278 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BEZ235 DACTOLISIB 31171 21279 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR Tabalumab TABALUMAB 31173 21280 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL522892 DOVITINIB 31177 21281 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BUTOCONAZOLE NITRATE BUTOCONAZOLE NITRATE 31178 21282 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-3464 CHEMBL602213 31180 21283 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCDD 14510636 31181 21284 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE JNJ-26483327 JNJ-26483327 31182 21285 BRDT 676 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE PMID26924192-Compound-104 31183 21286 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Timolol TIMOLOL 31184 21287 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR RETINOIC ACID 8940178 31185 21288 DGAT1 8694 ENZYME, DRUGGABLE GENOME Carbamide derivative 3 31187 21289 FOXO1 2308 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FAS LIGAND 12172378 31189 21290 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 249565590 CHEMBL1236539 31190 21291 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME acetaldehyde ACETALDEHYDE 31002879 31192 21292 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHENANTHROLINE PHENANTHROLINE 31194 21293 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE INSULIN INSULIN 11527158 31196 21294 NDUFA13 51079 ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545320 ME-344 31198 21295 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102916 31199 21296 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-2357 CHEMBL578257 31200 21297 SIK1 150094 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565818 31201 21298 SCNN1G 6340 ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE P-552 31202 21299 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LOSARTAN LOSARTAN 31204 21300 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE EVEROLIMUS EVEROLIMUS 24836070 31206 21301 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME US8609715, A-26 31208 21302 GMNN 51053 DRUGGABLE GENOME CALCITRIOL CALCITRIOL 31209 21303 DUSP6 1848 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE DIMETHYL SULFOXIDE 10702230 31210 21304 CFD 1675 ENZYME, DRUGGABLE GENOME, PROTEASE Anti-Factor D 31211 21305 POLK 51426 DNA REPAIR, ENZYME NSC-69187 CHEMBL19954 31215 21306 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1201649 ESTROGENS, CONJUGATED 31216 21307 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM BROMIDE 31217 21308 NDUFC1 4717 ENZYME inhibitor CHEMBL3545320 ME-344 31218 21309 PSMD4 5710 NA TALAZOPARIB TALAZOPARIB 28316110 31219 21310 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor GDC-0941 PICTILISIB 31220 21311 POLK 51426 DNA REPAIR, ENZYME MESALAMINE MESALAMINE 31221 21312 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 7,3'-DIMETHOXYFLAVONE 7,3'-DIMETHOXYFLAVONE 31222 21313 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME JNJ-7706621 JNJ-7706621 31223 21314 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 31229 21315 HMGCR 3156 ENZYME, DRUGGABLE GENOME Lovastatin LOVASTATIN 31230 21316 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALFAXALONE ALFAXALONE 31232 21317 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 178102589 31235 21318 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CAPSAZEPINE CAPSAZEPINE 31236 21319 ATAD5 79915 NA 2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE CHEMBL201325 31237 21320 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE US9695118, 4 31241 21321 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE ONC201 ONC-201 23390247 31242 21322 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PMI-005 31243 21323 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL650 METHYLPREDNISOLONE 31247 21324 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Pyrrolo[1,2-f]triazine derivative 2 31248 21325 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GNF-PF-2301 CHEMBL578061 31250 21326 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE REVERSE TRANSCRIPTASE INHIBITOR 15522931,16152760 31252 21327 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor PANOBINOSTAT PANOBINOSTAT 31253 21328 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE Mecasermin MECASERMIN 31254 21329 MPHOSPH8 54737 NA SALIRASIB SALIRASIB 31255 21330 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 9523002 31257 21331 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 28-THIOBETULINIC ACID CHEMBL1080077 19691293 31258 21332 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FENOFIBRATE FENOFIBRATE 22931300 31261 21333 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ARN-810 BRILANESTRANT 31262 21334 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME FISETIN FISETIN 31263 21335 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ANTIDEPRESSANT 16740621 31264 21336 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AGN-214868 SENREBOTASE 31265 21337 KLC3 147700 NA Platinum compounds 19434073,22188361,29662106,22026922,21449681 31266 21338 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR APIGENIN APIGENIN 25190466 31268 21339 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE DASATINIB DASATINIB 31270 21340 KDM4A 9682 DRUGGABLE GENOME, ENZYME ESCITALOPRAM OXALATE ESCITALOPRAM OXALATE 31272 21341 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AT13387 31274 21342 PCSK6 5046 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE inhibitor 252166848 31276 21343 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE LORECLEZOLE LORECLEZOLE 31277 21344 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200804 DICLOFENAC POTASSIUM 31278 21345 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1708 PAROXETINE HYDROCHLORIDE 31279 21346 NPR3 4883 DRUGGABLE GENOME antagonist 178101717 31281 21347 HTT 3064 DRUGGABLE GENOME VANOXERINE VANOXERINE 31282 21348 SMARCA2 6595 NA TCMDC-125813 CHEMBL580076 31284 21349 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Fosphenytoin FOSPHENYTOIN 31285 21350 MAOB 4129 DRUGGABLE GENOME, ENZYME SAFINAMIDE SAFINAMIDE 31287 21351 BCHE 590 DRUGGABLE GENOME, ENZYME ECHOTHIOPHATE IODIDE 31288 21352 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CETUXIMAB CETUXIMAB 31290 21353 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE MP470 31291 21354 SGPL1 8879 ENZYME, DRUGGABLE GENOME LX3305 LX-2931 31293 21355 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME Pyrrolo-pyrrolone derivative 6 31295 21356 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178102312 31296 21357 TNKS 8658 DRUGGABLE GENOME, ENZYME inhibitor 404859121 31298 21358 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME HALOPERIDOL HALOPERIDOL 17052361 31299 21359 NOS1 4842 DRUGGABLE GENOME, ENZYME HSP70 17150954 31300 21360 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE RG7440 31302 21361 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-4300 CHEMBL585656 31305 21362 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME radiotherapy 25054431 31306 21363 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BROMPERIDOL BROMPERIDOL 31307 21364 CEP68 23177 NA aspirin ASPIRIN 31310 21365 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METHAMPHETAMINE METHAMPHETAMINE 31311 21366 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9422240, 1-297 31312 21367 ATAD5 79915 NA NSC-92207 CHEMBL139935 31315 21368 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME NATALIZUMAB NATALIZUMAB 31316 21369 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Nebivolol NEBIVOLOL 31317 21370 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200806 NAPROXEN SODIUM 31321 21371 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PIPERTRAMINE AMIDE PIPERTRAMINE AMIDE 31323 21372 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178103584 31324 21373 SMN1 6606 DRUGGABLE GENOME N-HISTIDYL-2-AMINONAPHTHALENE (BETANA) N-HISTIDYL-2-AMINONAPHTHALENE (BETANA) 31325 21374 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL2110725 VINFLUNINE 31326 21375 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker 135652732 31327 21376 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135651430 31328 21377 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ETHANOL ALCOHOL 16478533 31330 21378 GMNN 51053 DRUGGABLE GENOME OLVANIL OLVANIL 31331 21379 CD47 961 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE ALX148 ALX-148 31332 21380 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL1200675 TOREMIFENE CITRATE 31333 21381 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME sertindole SERTINDOLE 31334 21382 UGT2B7 7364 DRUGGABLE GENOME fentanyl FENTANYL 32401749 31335 21383 SLC1A3 6507 TRANSPORTER, DRUGGABLE GENOME, CELL SURFACE ANTISERUM 9068840 31337 21384 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR RIBAVIRIN RIBAVIRIN 31338 21385 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME GO-6976 GO-6976 31339 21386 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE 178101646 31340 21387 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Octreotide OCTREOTIDE 31341 21388 CD9 928 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PROPIONIBACTERIUM ACNES 15902693 31342 21389 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PREDNISONE PREDNISONE 31343 21390 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Mometasone MOMETASONE 31344 21391 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CAMPTOTHECIN CAMPTOTHECIN 12464623 31345 21392 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHOPRENE METHOPRENE 31346 21393 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PROPACHLOR PROPACHLOR 31347 21394 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME STAVUDINE STAVUDINE 31348 21395 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor IRINOTECAN IRINOTECAN 31349 21396 VAMP2 6844 DRUGGABLE GENOME INSULIN INSULIN 7796801,9267469,9430681,8973549 31350 21397 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TCMDC-125603 CHEMBL528734 31351 21398 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 328083454 HARMINE 31352 21399 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE antagonist 252166532 ABT 737 31353 21400 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE GARLIC GARLIC 7604070 31354 21401 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE SJ000089102 CHEMBL606460 31355 21402 NAMPT 10135 DRUGGABLE GENOME CHS-828 CHS-828 31356 21403 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Dasatinib DASATINIB 31357 21404 APH1B 83464 PROTEASE, DRUGGABLE GENOME BMS-299897 CHEMBL247471 31359 21405 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ANTI-CD3 ANTIBODY 10712669 31360 21406 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DESIPRAMINE DESIPRAMINE 31361 21407 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME ICasp9M28z T cell 31363 21408 TUBB6 84617 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 31364 21409 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-9 31366 21410 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME DONEPEZIL DONEPEZIL 31368 21411 ACVR2A 92 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CELL SURFACE ACE-011 SOTATERCEPT 31369 21412 PSMA7 5688 PROTEASE, DRUGGABLE GENOME CARFILZOMIB CARFILZOMIB 24524217 31370 21413 MAOA 4128 DRUGGABLE GENOME, ENZYME PHENELZINE PHENELZINE 31372 21414 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER R547 17121911 31373 21415 APOE 348 DRUGGABLE GENOME ACE INHIBITOR 12105166,15585195 31374 21416 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR CELECOXIB CELECOXIB 17167033,17166886,15131590,16597647 31375 21417 FXYD2 486 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL1614 DESLANOSIDE 31376 21418 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE STI571 IMATINIB MESYLATE 31377 21419 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TCMDC-124224 CHEMBL580421 31378 21420 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME inhibitor ENDOSTATIN (84-114)-NH2 (JKC367) 31379 21421 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE PALBOCICLIB PALBOCICLIB 31380 21422 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Selumetinib SELUMETINIB 26343583,26272063 31381 21423 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 315661335 31382 21424 POLK 51426 DNA REPAIR, ENZYME GOSSYPETIN GOSSYPETIN 31383 21425 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR 4'-EPICHAETOVIRIDIN A CHEMBL1306556 31385 21426 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR GLAUCARUBINONE GLAUCARUBINONE 19199792 31386 21427 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR GW7604 CHEMBL195515 20334372 31389 21428 LTC4S 4056 ENZYME, DRUGGABLE GENOME montelukast MONTELUKAST 31390 21429 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR THIOCYCLAM HYDROGEN OXALATE THIOCYCLAM HYDROGEN OXALATE 31391 21430 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 178103597 31393 21431 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor ALVOCIDIB ALVOCIDIB 31396 21432 MAP3K7 6885 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565876 31398 21433 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 53801072 31400 21434 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL3545049 BAY-1125976 31402 21435 CSNK1G3 1456 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 249565894 31404 21436 SDF4 51150 NA ETHANOL ALCOHOL 18355758 31405 21437 PDE8A 5151 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL932 DIPYRIDAMOLE 31407 21438 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME GSK-269962A GSK-269962A 31409 21439 HSPB1 3315 DRUGGABLE GENOME PROTEIN KINASE C INHIBITOR 8875961 31410 21440 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650647 31411 21441 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE inhibitor 381118849 31415 21442 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 404859065 31420 21443 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL2103796 BERUBICIN HYDROCHLORIDE 31422 21444 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor XL147 PILARALISIB 31423 21445 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME inhibitor 252827503 CGS-27023A 31424 21446 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AMGMDS3 25730903 31425 21447 SERPINF1 5176 DRUGGABLE GENOME, PROTEASE INHIBITOR AdPEDR 31426 21448 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SCRIPTAID SCRIPTAID 19966789 31427 21449 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ZILEUTON ZILEUTON 22931300 31428 21450 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME MIDAZOLAM MIDAZOLAM 31429 21451 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE NAVITOCLAX, ABT-263 31430 21452 SULT1A3 6818 DRUGGABLE GENOME, ENZYME o-desmethyl-tramadol 31431 21453 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 178102336 BOSUTINIB 31432 21454 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Bicyclic heteroaryl benzamide derivative 1 31434 21455 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-66209 CHEMBL175266 31437 21456 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MOLINATE MOLINATE 31438 21457 TSPO 706 DRUGGABLE GENOME ALPIDEM ALPIDEM 31439 21458 MPI 4351 ENZYME, DRUGGABLE GENOME HAEMATOXYLIN HAEMATOXYLIN 31441 21459 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor NINTEDANIB NINTEDANIB 31442 21460 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PAZOPANIB PAZOPANIB 31443 21461 DPP8 54878 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166752 31445 21462 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TOLUENE DIISOCYANATE TOLUENE DIISOCYANATE 31446 21463 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor GSK1363089 FORETINIB 31448 21464 TESK1 7016 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565797 31449 21465 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-14 31451 21466 USP14 9097 ENZYME, CELL SURFACE, PROTEASE inhibitor 252827537 31454 21467 MPHOSPH8 54737 NA DEPHOSTATIN DEPHOSTATIN 31456 21468 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TCMDC-124327 CHEMBL581929 31458 21469 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE WEHI-539 27974663 31459 21470 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200950 CLIDINIUM BROMIDE 31461 21471 MAPKAPK5 8550 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL3545338 GLPG-0259 31462 21472 MAGEA1 4100 NA 5-AZA-2'-DEOXYCYTIDINE 8757382,15256472,7511051,8698626 31463 21473 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GDC-0032 TASELISIB 25172762,28331003,26333383,26589432,23662903 31466 21474 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Trametinib + 2141795 31467 21475 TUBB2A 7280 DRUGGABLE GENOME CHEMBL2103826 DAVUNETIDE 31468 21476 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME KPT-9274 KPT-9274 31469 21477 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-3237 CHEMBL602206 31471 21478 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4576 CHEMBL527336 31472 21479 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051792 PANOBINOSTAT 31475 21480 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1237132 CLEVIDIPINE 31476 21481 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417413 CHEMBL1343568 31477 21482 CD276 80381 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME MGA271 ENOBLITUZUMAB 23114578 31480 21483 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR EUPAROTIN ACETATE EUPAROTIN ACETATE 31481 21484 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650108 CLIDINIUM 31482 21485 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NEOSTIGMINE METHYLSULFATE NEOSTIGMINE METHYLSULFATE 31484 21486 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME HYDRALAZINE HYDRALAZINE 31485 21487 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SPIPERONE SPIPERONE 31486 21488 MAPT 4137 DRUGGABLE GENOME LY3303560 ZAGOTENEMAB 31488 21489 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR SM-122 CHEMBL481422 21462933 31489 21490 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-74 31490 21491 RGS4 5999 DRUGGABLE GENOME BAY-11-7082 CHEMBL403183 31491 21492 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME APIGENIN APIGENIN 25190466 31492 21493 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE EMODIN EMODIN 22212721 31493 21494 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME IMMUNOSUPPRESSANT 11567647 31494 21495 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545096 BGT-226 31495 21496 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME VANDETANIB VANDETANIB 31496 21497 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME Larotrectinib LAROTRECTINIB 31499 21498 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR PEPEROMIN E PEPEROMIN E 19559609 31500 21499 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME Benzoimidazole derivative 1 31502 21500 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM BROMIDE 31505 21501 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Fluorouracil FLUOROURACIL 25714871,28424201 31506 21502 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-377852 CHEMBL1466186 31507 21503 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL antagonist 178103291 CHEMBL190883 31508 21504 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PIMOZIDE PIMOZIDE 31509 21505 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650765 31510 21506 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER fluphenazine FLUPHENAZINE 31511 21507 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor E-3810 RABEPRAZOLE SODIUM 31512 21508 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Netoglitazone NETOGLITAZONE 31513 21509 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DEZOCINE DEZOCINE 31514 21510 E2F1 1869 TRANSCRIPTION FACTOR ANTISENSE OLIGONUCLEOTIDES 10207094 31515 21511 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE P-552 31517 21512 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor ARQ 197 TIVANTINIB 31518 21513 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR TAS-108 SR16234 31519 21514 MAOA 4128 DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 22071524 31520 21515 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 187051805 QUISINOSTAT 31521 21516 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Norepinephrine NOREPINEPHRINE 31522 21517 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 178104006 BUDESONIDE 31523 21518 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME PROTEIN KINASE A INHIBITOR 9093533 31525 21519 NME2 4831 KINASE tenofovir TENOFOVIR 31529 21520 BAZ2B 29994 NA NSC-175743 CHEMBL1609016 31530 21521 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MOLINDONE MOLINDONE 31532 21522 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Olaparib OLAPARIB 31533 21523 KLK5 25818 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166696 31537 21524 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE AG-1879 CHEMBL406845 31539 21525 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME EVEROLIMUS EVEROLIMUS 31540 21526 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME APO-010 31542 21527 POLB 5423 DNA REPAIR, DRUGGABLE GENOME EMODIC ACID EMODIC ACID 31543 21528 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE SULFONATES 12161163 31545 21529 CA2 760 DRUGGABLE GENOME, ENZYME Curcumin CURCUMIN 31546 21530 POLK 51426 DNA REPAIR, ENZYME AMPICILLIN AMPICILLIN 31547 21531 GLS 2744 ENZYME ICOSAPENT ICOSAPENT 31548 21532 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Megestrol MEGESTROL 31549 21533 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 310264758 31551 21534 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME MIBEFRADIL MIBEFRADIL 31552 21535 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TOZASERTIB TOZASERTIB 31553 21536 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2016054807Example80 31555 21537 GMNN 51053 DRUGGABLE GENOME GERONTOXANTHONE I GERONTOXANTHONE I 31556 21538 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME N-OXALYLGLYCINE N-OXALYLGLYCINE 26022078 31557 21539 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135651446 ADENOSINE TRIPHOSPHATE 31559 21540 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649665 31560 21541 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 381744995 SELITRECTINIB 31561 21542 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SKF-82526 CHEMBL1161520 31562 21543 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE allosteric modulator 178102420 31564 21544 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 135651223 T091317 31568 21545 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme8NCGC-00010037 31569 21546 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PROADIFEN PROADIFEN 31570 21547 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR abemaciclib ABEMACICLIB 31571 21548 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 381118895 31572 21549 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ALSTERPAULLONE ALSTERPAULLONE 31576 21550 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PT-101 CHEMBL316796 31577 21551 TUBA3C 7278 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 31578 21552 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE CRENOLANIB CRENOLANIB 24132921,22745105 31580 21553 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201124 KETOROLAC TROMETHAMINE 31582 21554 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE peginterferon alfa-2b 28703131 31583 21555 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ChronSeal 31584 21556 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CLORAZEPATE CLORAZEPIC ACID 31585 21557 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-5 31586 21558 UGT1A7 54577 DRUGGABLE GENOME, ENZYME febuxostat FEBUXOSTAT 27798726 31587 21559 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX JQ1 28151717 31588 21560 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PD98509 22662154 31590 21561 PRMT1 3276 ENZYME, METHYL TRANSFERASE inhibitor 178103616 31592 21562 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME DEPHOSTATIN DEPHOSTATIN 31593 21563 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR ARSENIC TRIOXIDE 14619570 31594 21564 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR FENTANYL FENTANYL 9527747 31595 21565 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102780 31597 21566 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE ONONIN ONONIN 31598 21567 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DOX 12810556 31599 21568 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651513 31603 21569 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650599 METOPROLOL 31605 21570 KEAP1 9817 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING 385612246 31606 21571 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIETHYLSTILBESTROL DIETHYLSTILBESTROL 22931300 31607 21572 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 OFLOXACIN OFLOXACIN 22931300 31608 21573 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NADOLOL NADOLOL 2903243 31609 21574 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 249565633 DACTOLISIB 31610 21575 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 223365969 31611 21576 TNFRSF9 3604 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE antibody 318164830 URELUMAB 31613 21577 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME INC280 CAPMATINIB 28783719 31614 21578 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZEARALANONE ZEARALANONE 31615 21579 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR L-655708 CHEMBL52030 22137933 31617 21580 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Cisplatin CISPLATIN 31618 21581 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270010-Compound-Figure17-1 31619 21582 FTO 79068 ENZYME interferon alfa-2a, recombinant 25367448 31621 21583 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL3184679 AZD-4547 31622 21584 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE METHYLCURCUMIN METHYLCURCUMIN 25753330 31623 21585 POLI 11201 DNA REPAIR 5,7,3',5'-TETRAHYDROXYFLAVANONE CHEMBL307893 31625 21586 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME LINOLENIC ACID LINOLENIC ACID 31627 21587 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Cinnarizine CINNARIZINE 31629 21588 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BENZOTHIAZYL DISULFIDE BENZOTHIAZYL DISULFIDE 31630 21589 PDF 64146 DRUGGABLE GENOME MCB-3837 31631 21590 BAZ2B 29994 NA MYRICETIN MYRICETIN 31632 21591 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE ICO-007 31633 21592 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE RIBOCICLIB RIBOCICLIB 29306020 31634 21593 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL Lercanidipine LERCANIDIPINE 31639 21594 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CARBOPLATIN CARBOPLATIN 29584549 31640 21595 TARDBP 23435 TUMOR SUPPRESSOR IBUPROFEN IBUPROFEN 31641 21596 MMP10 4319 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 249565939 31642 21597 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME DOCETAXEL DOCETAXEL 16210916 31643 21598 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000024553 CHEMBL589238 31646 21599 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-28081 CHEMBL512832 31647 21600 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650336 GW501516 31648 21601 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GR-127935 GR-127935 31649 21602 BCL2L11 10018 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR imatinib IMATINIB 24223824 31650 21603 CACNB4 785 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL940 GABAPENTIN 31651 21604 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650390 INDOMETHACIN 31652 21605 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AG-555 CHEMBL53898 31653 21606 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody AMG 479 31655 21607 APOE 348 DRUGGABLE GENOME CORTICOSTEROIDS 1903065 31656 21608 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL520733 SEMAGACESTAT 31658 21609 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 31659 21610 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor VORINOSTAT VORINOSTAT 31661 21611 METAP2 10988 ENZYME, DRUGGABLE GENOME, KINASE, PROTEASE D-Methionine 31662 21612 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR TOPOTECAN TOPOTECAN 15569250 31663 21613 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ELIPRODIL ELIPRODIL 31664 21614 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME E-4031 CHEMBL327980 31665 21615 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650824 PILOCARPINE 31666 21616 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650160 DARIFENACIN 31667 21617 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ALSTERPAULLONE ALSTERPAULLONE 31672 21618 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME URSOLIC ACID URSOLIC ACID 19534471 31673 21619 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PIPLARTINE PIPLARTINE 31674 21620 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME BAY 10-00394 31676 21621 ARNT 405 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR HYDROCORTISONE HYDROCORTISONE 10048155 31677 21622 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TOLONIUM CHLORIDE TOLONIUM CHLORIDE 31678 21623 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Aripiprazole ARIPIPRAZOLE 31682 21624 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL NICARDIPINE NICARDIPINE 31683 21625 GMNN 51053 DRUGGABLE GENOME CARPHENAZINE CARPHENAZINE 31684 21626 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Pyrido[1,2-a]indole-1.-carboxylic acid analog 5 31685 21627 BRCA2 675 CLINICALLY ACTIONABLE Cisplatin CISPLATIN 25193512,26801247 31686 21628 TOP2B 7155 DRUGGABLE GENOME, ENZYME BMY-43748 31687 21629 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR NSC-39249 CHEMBL482792 31689 21630 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor LINIFANIB LINIFANIB 31690 21631 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME GSK-269962A GSK-269962A 31691 21632 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR HESPERETIN HESPERETIN 22429094 31692 21633 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GW843682X GW843682X 31693 21634 CD38 952 CELL SURFACE, DRUGGABLE GENOME SAR650984 31694 21635 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL antagonist 178103292 31695 21636 SENP3 26168 PROTEASE methylphenidate METHYLPHENIDATE 29382897 31696 21637 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TGF 11687963 31698 21638 MICB 4277 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE ribavirin RIBAVIRIN 31699 21639 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor XL647 TESEVATINIB 31700 21640 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PEMETREXED PEMETREXED 31605797,24636847 31701 21641 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE inhibitor PX-478 PX-478 31703 21642 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE VATALANIB VATALANIB 31704 21643 HSPD1 3329 DRUGGABLE GENOME, ENZYME, CELL SURFACE CETRORELIX CETRORELIX 9805247 31705 21644 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 252166794 31706 21645 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BUDESONIDE BUDESONIDE 22931300 31708 21646 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor GEFITINIB GEFITINIB 31709 21647 PRSS8 5652 DRUGGABLE GENOME, PROTEASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 223366189 31710 21648 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE BRIGATINIB BRIGATINIB 28287083 31713 21649 DUSP1 1843 PROTEIN PHOSPHATASE, KINASE, DRUGGABLE GENOME HYDROXYUREA HYDROXYUREA 15856297 31714 21650 PTGS2 5743 DRUGGABLE GENOME, ENZYME SALICYLIC ACID 31716 21651 PTBP1 5725 DRUGGABLE GENOME ELLIPTECINE ELLIPTECINE 31717 21652 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GW3965 CHEMBL59030 31718 21653 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE platinum PLATINUM 25677447 31720 21654 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL25 ASPIRIN 31721 21655 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR TACI-IG ATACICEPT 31723 21656 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE XL147 PILARALISIB 31724 21657 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-992 CHEMBL602561 31725 21658 CBX1 10951 NA SARCOLYSIN SARCOLYSIN 31726 21659 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHOXYVONE METHOXYVONE 31727 21660 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PX-866 SONOLISIB 31728 21661 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101291 31729 21662 HNF1B 6928 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX platinum PLATINUM 27561454 31730 21663 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 329968448 31731 21664 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 381118904 31732 21665 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME HUMAX-CD20 OFATUMUMAB 31733 21666 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYSTEINE CYSTEINE 31735 21667 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Dobutamine DOBUTAMINE 31736 21668 ABCA1 19 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178103851 PROBUCOL 31737 21669 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE THYMIDINE THYMIDINE 1868466 31741 21670 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-23 31742 21671 ACVR2A 92 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CELL SURFACE antibody 249565766 BIMAGRUMAB 31743 21672 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER bepridil BEPRIDIL 31744 21673 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR COR-1 31745 21674 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 363894208 ILORASERTIB 31746 21675 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME VORINOSTAT VORINOSTAT 31747 21676 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrazolopyridine derivative 3 31748 21677 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ECONAZOLE NITRATE ECONAZOLE NITRATE 31749 21678 TMEM97 27346 NA agonist 178103297 31750 21679 ENPP2 5168 ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING NSC-1741 CHEMBL483302 20349977 31751 21680 GSTA1 2938 ENZYME, DRUGGABLE GENOME PHYTOCHEMICALS 15672752 31752 21681 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OLOPATADINE OLOPATADINE 31753 21682 ALB 213 TRANSPORTER, DRUGGABLE GENOME DIAZEPAM DIAZEPAM 20869876 31754 21683 FAAH 2166 ENZYME, DRUGGABLE GENOME Thiopental THIOPENTAL 31756 21684 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BEPRIDIL BEPRIDIL 31757 21685 IL1R2 7850 DRUGGABLE GENOME IL-1 31760 21686 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIRLOTAPIDE DIRLOTAPIDE 22094027 31761 21687 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME STICTIC ACID STICTIC ACID 31762 21688 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antagonist CHEMBL2109357 AVE-1642 31763 21689 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TCMDC-123884 CHEMBL580955 31764 21690 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AG-527 CHEMBL258767 31765 21691 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor 340590240 31766 21692 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178100901 31767 21693 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR 4SC-202 DOMATINOSTAT 31769 21694 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR ROMIDEPSIN ROMIDEPSIN 31770 21695 SRI 6717 NA ADRIAMYCIN ADRIAMYCIN 1975203 31771 21696 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME NEUROPROTECTANTS 10460254 31772 21697 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DOVITINIB DOVITINIB 31773 21698 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Isoquinoline sulfonyl derivative 2 31774 21699 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE RISEDRONATE RISEDRONIC ACID 31775 21700 LPAR5 57121 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651488 31777 21701 DHFR 1719 DRUGGABLE GENOME, ENZYME MDAM (y-methylene-10-deazaaminopterin) 31778 21702 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE FENOTEROL FENOTEROL 31781 21703 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000113257 CHEMBL528694 31782 21704 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL496102 AMG-208 31784 21705 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Sphingosomal topotecan 31785 21706 USP1 7398 DNA REPAIR, PROTEASE, ENZYME HEXACHLOROPHENE HEXACHLOROPHENE 31787 21707 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GR-127935 GR-127935 31789 21708 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Fulvestrant FULVESTRANT 31791 21709 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BEXAROTENE BEXAROTENE 19791803,23391145 31792 21710 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NIACIN NIACIN 31795 21711 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Cediranib CEDIRANIB 22238366 31796 21712 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME HYPERFORIN HYPERFORIN 31797 21713 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PF-05212384 GEDATOLISIB 24042735,17314276,21325073 31798 21714 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200909 PREDNISOLONE TEBUTATE 31799 21715 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME EP42675 31800 21716 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-59 31801 21717 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545053 EMD-1204831 31803 21718 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME GM-CSF REGRAMOSTIM 16403261 31804 21719 ANKFN1 162282 NA hydrochlorothiazide HYDROCHLOROTHIAZIDE 31805 21720 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 318164817 31806 21721 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL428647 PACLITAXEL 31807 21722 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE BROMOCRIPTINE BROMOCRIPTINE 11680511 31809 21723 CBX1 10951 NA SIB-1757 CHEMBL88553 31811 21724 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650624 MORPHINE 31812 21725 SLPI 6590 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR HEPARIN HEPARIN 8615699,9593692 31813 21726 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1201179 LAPATINIB DITOSYLATE 31814 21727 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE CENISERTIB CENISERTIB 31815 21728 ATXN2 6311 NA ECONAZOLE NITRATE ECONAZOLE NITRATE 31817 21729 MPHOSPH8 54737 NA AG-537 CHEMBL67535 31820 21730 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor 178101520 TIAGABINE 31823 21731 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Crizotinib CRIZOTINIB 31824 21732 RAB9A 9367 ENZYME, DRUGGABLE GENOME TRANILAST TRANILAST 31826 21733 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor CHEMBL189963 PALBOCICLIB 31827 21734 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Ladostigil LADOSTIGIL 31828 21735 PDE5A 8654 ENZYME, DRUGGABLE GENOME ROLIPRAM ROLIPRAM 31830 21736 MAPT 4137 DRUGGABLE GENOME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 31833 21737 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME METIXENE METHIXENE 31834 21738 CD38 952 CELL SURFACE, DRUGGABLE GENOME 4SCAR19 and 4SCAR38 31835 21739 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CCT196969 25500121,23431193 31836 21740 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE KP201 BENZHYDROCODONE HYDROCHLORIDE 31837 21741 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Cabozantinib CABOZANTINIB 31838 21742 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 4-NONYLPHENOL 4-NONYLPHENOL 31840 21743 SEM1 7979 NA CARFILZOMIB CARFILZOMIB 24524217 31841 21744 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Emepepimut-S EMEPEPIMUT-S 31843 21745 ETV4 2118 CLINICALLY ACTIONABLE, DRUG RESISTANCE TRAMETINIB TRAMETINIB 28178529 31844 21746 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GW282974X GW282974X 31847 21747 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-119889 CHEMBL516616 31848 21748 NOD1 10392 CLINICALLY ACTIONABLE, DRUGGABLE GENOME GNF-PF-3971 CHEMBL599890 31849 21749 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME BAY-613606 CHEMBL541400 31850 21750 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL482967 CYC-116 31852 21751 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE UROKINASE UROKINASE 31853 21752 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 178103870 SOTALOL 31856 21753 TMEM97 27346 NA Piperazinyl norbenzomorphane compound 2 31858 21754 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200745 OXPRENOLOL HYDROCHLORIDE 31859 21755 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE VINBLASTINE SULFATE VINBLASTINE SULFATE 31861 21756 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-300014A GSK-300014A 31862 21757 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135652672 BRUCINE 31863 21758 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 31864 21759 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2311030 ERGOLOID MESYLATES 31865 21760 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PHANQUONE PHANQUONE 31866 21761 GMNN 51053 DRUGGABLE GENOME SALIRASIB SALIRASIB 31867 21762 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-747259 CHEMBL561679 31872 21763 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL1230609 FORETINIB 31873 21764 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE agonist 178100891 31874 21765 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL511142 BUPRENORPHINE 31875 21766 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE trastuzumab TRASTUZUMAB 31876 21767 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 31877 21768 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CARFENTRAZONE-ETHYL CARFENTRAZONE-ETHYL 31879 21769 HMGCR 3156 ENZYME, DRUGGABLE GENOME SIMVASTATIN SIMVASTATIN 31881 21770 GAA 2548 DRUGGABLE GENOME, ENZYME inhibitor 178101359 31882 21771 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE ataluren ATALUREN 18722008,21233271,26840186,20622033 31884 21772 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CVT-6883 GS 6201 31885 21773 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor 178103944 APREMILAST 31886 21774 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-123851 CHEMBL548458 31888 21775 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TOREMIFENE TOREMIFENE 9871429 31889 21776 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PCM-075 ONVANSERTIB 31890 21777 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL101253 VATALANIB 31891 21778 HSPA8 3312 TUMOR SUPPRESSOR ANTIBIOTIC ANTIBIOTIC 14966137 31892 21779 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME AST-487 AST-487 31893 21780 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Lapatinib LAPATINIB 26270481 31894 21781 MAPT 4137 DRUGGABLE GENOME DNDI1417063 CHEMBL2094422 31895 21782 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178103494 IBRUTINIB 31896 21783 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GAMMA-PROPARGYLAMINO-ATP CHEMBL557670 19410453 31897 21784 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GSK9772 CHEMBL493241 18800767,22873709 31898 21785 PSMD2 5708 NA inhibitor BORTEZOMIB BORTEZOMIB 31900 21786 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME Larotrectinib LAROTRECTINIB 31901 21787 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DZNep 26676756 31902 21788 EYA2 2139 DNA REPAIR AMARANTH AMARANTH 31903 21789 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Tositumomab TOSITUMOMAB 31904 21790 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (R)-MELPHALAN (R)-MELPHALAN 31908 21791 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102572 31910 21792 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Rivaroxaban RIVAROXABAN 31911 21793 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100385 31913 21794 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME NSC-228155 CHEMBL505670 31916 21795 TSPO 706 DRUGGABLE GENOME Flumazenil FLUMAZENIL 31917 21796 CACNB3 784 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ION CHANNEL modulator CHEMBL1059 PREGABALIN 31918 21797 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BI 113823 31919 21798 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME antagonist 178103270 31921 21799 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TRIAMTERENE TRIAMTERENE 31922 21800 ALOX15B 247 DRUGGABLE GENOME, ENZYME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 31926 21801 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 375973268 31928 21802 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME (+)-TAXIFOLIN (+)-TAXIFOLIN 31929 21803 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor SUNITINIB SUNITINIB 31931 21804 ALPI 248 DRUGGABLE GENOME, ENZYME CURCUMIN CURCUMIN 31932 21805 COMT 1312 DRUGGABLE GENOME, ENZYME norepinephrine NOREPINEPHRINE 31933 21806 TAF1 6872 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE DOXORUBICIN DOXORUBICIN 10070062 31934 21807 POLA1 5422 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, DNA REPAIR CLOFARABINE CLOFARABINE 31936 21808 KDM1A 23028 DRUGGABLE GENOME, ENZYME, CELL SURFACE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING activator 252166601 31937 21809 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR NSAIDS 16452198 31940 21810 BAZ2B 29994 NA DNDI1417420 CHEMBL1546223 31941 21811 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AM-404 CHEMBL39878 31942 21812 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Cycloalkyl nitrile pyrazole carboxamide derivative 1 31944 21813 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME succinylcholine SUXAMETHONIUM 25989378,12411786,26951757,8828983,19919814,17710899,7829078,9334205,21965348,11063719,20837722,20301325,9037193,12467748,10823104,20681998,25611019,19648156,25256590,12220451,11668625,23736090,23223104,14500992,9066328,14641996,18945287,25960145,7889656,26031886,11575529,18212565,16284304,8602662,18306019,28326467,25424378,11928716,18502356,12761368,10352931,11725865,12151923,11525881,17122579,16917943,8220422,24291096,10700782,16163667,17226826,9389851,16732128,16835904,11448278,29101530,9450902,7547049,23628358,19807743,9543323,18313359,24361844,26994242,12208234,15448513,16621918,21455645,11553045,10625004,12124989,3177917,19020143,19191329,15537710,27918309,8220423,12059893,10612851,16732084,10793526,23069638,27382027,15108991,12709367,12123492,19018722,26381711,10360872,25268394,28063098,11493496,12434264,17182726,12411788,19685112,25735680,8902717,29608462,27663056,7751854,8012359,9520251,15731587,26068069,15210166,1510267,10888602,22030266,25466363,17483490,28403410,12237752,9873004,1774074,17081152,18564801,10484775,21282829,20888934,16244001,7586638,19191333,25086907,7633940,17667581,15299003,12883402,19346234,1354642,22415532 31945 21814 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Pyrazole derivative 62 31946 21815 PSMD2 5708 NA BORTEZOMIB BORTEZOMIB 31947 21816 CXCL8 3576 DRUGGABLE GENOME ATRA TRETINOIN 8900181 31949 21817 ALOX5 240 DRUGGABLE GENOME, ENZYME 5-OXO-ETE 5-OXO-ETE 24924423 31951 21818 EPHX2 2053 DRUGGABLE GENOME, ENZYME inhibitor 381118834 31952 21819 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2012830453910 31955 21820 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 252166674 31956 21821 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Brivanib BRIVANIB 22238366 31957 21822 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME dexamethasone DEXAMETHASONE 25055799 31958 21823 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Lorlatinib LORLATINIB 31959 21824 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME peginterferon alfa-2a 20812847 31960 21825 PSMD5 5711 NA inhibitor BORTEZOMIB BORTEZOMIB 31961 21826 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FOLPET FOLPET 31963 21827 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE CGM097 CGM-097 27507190 31964 21828 ATAD5 79915 NA DNDI1417263 CHEMBL1431115 31965 21829 CD38 952 CELL SURFACE, DRUGGABLE GENOME THROMBIN THROMBIN 9654134 31967 21830 CD3D 915 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE MT-103 BLINATUMOMAB 31968 21831 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 252166674 31969 21832 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GNF-PF-3582 CHEMBL606167 31974 21833 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE panitumumab PANITUMUMAB 18681783,14990633,16467544,23959273,16377102,14990632,18784101,16257339,18003960,23022519,11255078,19339720,18316547,12648464,22594511 31978 21834 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR RO-31-8220 15327748 31979 21835 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CHLOROQUINE CHLOROQUINE 22931300 31981 21836 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER CPT-11 IRINOTECAN HYDROCHLORIDE 9918583 31983 21837 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178101124 31984 21838 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE AG-538 CHEMBL56393 31985 21839 POLI 11201 DNA REPAIR KAEMPFEROL KAEMPFEROL 31988 21840 CAST 831 PROTEASE INHIBITOR STAUROSPORINE STAUROSPORINE 12576481 31989 21841 RRM2 6241 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1637 GEMCITABINE HYDROCHLORIDE 31991 21842 FAM177A1 283635 NA lithium LITHIUM 29121268 31993 21843 LCAT 3931 ENZYME, TRANSPORTER, DRUGGABLE GENOME MEDI6012 RECOMBINANT HUMAN LECITHIN:CHOLESTEROL ACYLTRANSFERASE 25657982 31995 21844 FAAH 2166 ENZYME, DRUGGABLE GENOME N-alkyl-4-oxazolecar boxamide derivative 2 31997 21845 ANO1 55107 ION CHANNEL activator 135652731 31998 21846 MAP3K9 4293 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565579 APITOLISIB 31999 21847 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Doxylamine DOXYLAMINE 32000 21848 ATAD5 79915 NA NIMODIPINE NIMODIPINE 32001 21849 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME SIROLIMUS SIROLIMUS 17031644 32003 21850 GBA 2629 DRUGGABLE GENOME, ENZYME CASTANOSPERMINE CASTANOSPERMINE 32005 21851 ATXN2 6311 NA SERTRALINE SERTRALINE 32006 21852 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DACTINOMYCIN DACTINOMYCIN 32007 21853 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR PYRITHIONE PYRITHIONE 32008 21854 DIABLO 56616 NA STAUROSPORINE STAUROSPORINE 14985459,15466201 32009 21855 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652320 32010 21856 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME CAR-T Cells targeting Mesothelin 32014 21857 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4078 CHEMBL584883 32015 21858 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PHA-767491 CHEMBL225519 32016 21859 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CADMIUM DICHLORIDE CADMIUM DICHLORIDE 32018 21860 NOX1 27035 ION CHANNEL, ENZYME, TRANSPORTER, DRUGGABLE GENOME PHENOTHIAZINE PHENOTHIAZINE 32020 21861 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MECLIZINE MECLIZINE 22931300 32021 21862 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME 178101604 CILMOSTIM 32023 21863 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE SUFENTANIL SUFENTANIL 32025 21864 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME HALAZEPAM HALAZEPAM 32026 21865 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR PD-0166285 PD-0166285 32029 21866 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565693 32031 21867 ATXN2 6311 NA BIX-01294 CHEMBL569864 32034 21868 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Imidazo[4,5-c]pyridine derivative 2 32035 21869 ESRRG 2104 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist CHEMBL10041 AFIMOXIFENE 32036 21870 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 381118877 TOMIVOSERTIB 32037 21871 GNL3 26354 NA fluorouracil FLUOROURACIL 32039 21872 ACVR1B 91 SERINE THREONINE KINASE, CELL SURFACE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 404859109 32041 21873 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR SORAFENIB SORAFENIB 32042 21874 RRM2 6241 DRUGGABLE GENOME, ENZYME TRIAPINE TRIAPINE 32044 21875 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZO(K)FLUORANTHENE BENZO(K)FLUORANTHENE 32045 21876 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ZOLMITRIPTAN ZOLMITRIPTAN 32046 21877 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE LABETALOL LABETALOL 4050551 32047 21878 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Nortriptyline NORTRIPTYLINE 32049 21879 COMT 1312 DRUGGABLE GENOME, ENZYME sufentanil SUFENTANIL 28006928,23686330,21398039,23302985,26902643,29474345,23773341,25155931,25185591,19514130,28745577,27027462 32050 21880 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE MASITINIB MASITINIB 32053 21881 SREBF1 6720 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR INSULIN INSULIN 10627507,12576518,14594997 32054 21882 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor PKI-587 GEDATOLISIB 32055 21883 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BGJ398 INFIGRATINIB 32056 21884 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PTHRP 3395323 32058 21885 HKDC1 80201 DRUGGABLE GENOME, KINASE 2,6-DIMETHOXYQUINONE 2,6-DIMETHOXYQUINONE 32059 21886 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TROGLITAZONE TROGLITAZONE 22579484,22342624,22424300,16680159 32061 21887 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE inhibitor 178103157 32064 21888 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CHLORHEXIDINE CHLORHEXIDINE 32066 21889 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-Figure4b 32068 21890 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652032 32069 21891 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200562 HYDROCORTISONE VALERATE 32070 21892 GLS 2744 ENZYME CEFAMANDOLE NAFATE CEFAMANDOLE NAFATE 32071 21893 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ORPHENADRINE ORPHENADRINE 32074 21894 POLK 51426 DNA REPAIR, ENZYME CARBOPLATIN CARBOPLATIN 32075 21895 CLU 1191 CELL SURFACE, DRUGGABLE GENOME antisense oligonucleotide CUSTIRSEN CUSTIRSEN 32077 21896 MARCHF8 220972 ENZYME Arepanrix 32078 21897 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE APRATOXIN F APRATOXIN F 32079 21898 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE JNJ-42756493 ERDAFITINIB 26324363,28341788 32081 21899 MPHOSPH8 54737 NA KETOCONAZOLE KETOCONAZOLE 32082 21900 TARDBP 23435 TUMOR SUPPRESSOR BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 32083 21901 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE OSI-632 OSI-632 32085 21902 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NALMEFENE NALMEFENE 32087 21903 RABEP1 9135 CLINICALLY ACTIONABLE, GROWTH FACTOR risperidone RISPERIDONE 28694205 32088 21904 SRD5A1 6715 DRUGGABLE GENOME BEXLOSTERIDE BEXLOSTERIDE 32091 21905 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR DOVITINIB DOVITINIB 32092 21906 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Doxepin DOXEPIN 32093 21907 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-39 32094 21908 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CLIOXANIDE CLIOXANIDE 32095 21909 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ET-1 32096 21910 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1564 DIPHENYLPYRALINE HYDROCHLORIDE 32098 21911 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL491473 CEDIRANIB 32099 21912 AKR1B1 231 DRUGGABLE GENOME, ENZYME ADMVA 32101 21913 EML4 27436 CLINICALLY ACTIONABLE, KINASE PF-06463922 LORLATINIB 27432227,26698910,26144315,26554404 32102 21914 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651697 CORTISTATIN-14 32103 21915 TARDBP 23435 TUMOR SUPPRESSOR SESAMIN SESAMIN 32104 21916 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE ONO-4578 32105 21917 AKR1C3 8644 ENZYME, DRUGGABLE GENOME Flufenamic Acid 32107 21918 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR TAK-441 TAK-441 32108 21919 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHENYLBUTANOIC ACID PHENYLBUTANOIC ACID 24044874 32110 21920 EML4 27436 CLINICALLY ACTIONABLE, KINASE Afatinib AFATINIB 26682573 32111 21921 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ALAPROCLATE ALAPROCLATE 32112 21922 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE ABT-957 32113 21923 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MILBEMYCIN A4 MILBEMYCIN A4 32114 21924 ATXN2 6311 NA KEPONE KEPONE 32115 21925 GMNN 51053 DRUGGABLE GENOME RESCINNAMINE RESCINNAMINE 32117 21926 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE PROPYLTHIOURACIL PROPYLTHIOURACIL 32118 21927 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE DEOXYCYTIDINE DEOXYCYTIDINE 10471381,11952160 32119 21928 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME TNP-470 O-CHLOROACETYLCARBAMOYLFUMAGILLOL 10481942 32120 21929 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME BDBM50173323 32121 21930 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102776 CP-195543 32122 21931 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 A-315456 CHEMBL362863 32124 21932 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PYROGALLOL RED PYROGALLOL RED 32125 21933 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AMINACRINE AMINACRINE 32126 21934 ALOX5 240 DRUGGABLE GENOME, ENZYME LICOFELONE LICOFELONE 32127 21935 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GLAUCINE METHIODIDE GLAUCINE METHIODIDE 32129 21936 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL58323 ERLOSAMIDE 32130 21937 BBOX1 8424 DRUGGABLE GENOME THIRAM THIRAM 25266780 32132 21938 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 21 32133 21939 SPP1 6696 DRUGGABLE GENOME TPA ALTEPLASE 12009309 32134 21940 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650727 32137 21941 CACNB3 784 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ION CHANNEL modulator CHEMBL2103836 IMAGABALIN 32138 21942 CASP8 841 DRUGGABLE GENOME, PROTEASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL197672 EMRICASAN 32139 21943 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE CENISERTIB CENISERTIB 32140 21944 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME PMID28460551-Compound-6 32141 21945 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-15 32145 21946 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE LY-2090314 LY-2090314 32146 21947 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE NITIDINE CHLORIDE NITIDINE CHLORIDE 21435753 32147 21948 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CNS-7056 REMIMAZOLAM 32148 21949 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SORBINIL SORBINIL 24819954 32149 21950 TNFRSF11A 8792 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE risperidone RISPERIDONE 32150 21951 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Trametinib TRAMETINIB 26343583,28783719,26882569,27222538 32151 21952 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHEMBL1200789 TRICLOFOS SODIUM 32152 21953 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TOCILIZUMAB TOCILIZUMAB 32153 21954 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ASP-4058 ASP-4058 32156 21955 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme21Right 32157 21956 CYB5R3 1727 DRUGGABLE GENOME, ENZYME chloroprocaine CHLOROPROCAINE 32158 21957 AQP1 358 ION CHANNEL, DRUGGABLE GENOME blocker 405560380 32159 21958 ALOX5 240 DRUGGABLE GENOME, ENZYME ZILEUTON ZILEUTON 11454666 32160 21959 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE PD-0166285 PD-0166285 32162 21960 GUCY1A2 2977 ENZYME, DRUGGABLE GENOME NCX 4016 32163 21961 RPS6KA4 8986 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, ENZYME LINIFANIB LINIFANIB 32166 21962 USP1 7398 DNA REPAIR, PROTEASE, ENZYME QUINALDINE BLUE QUINALDINE BLUE 32167 21963 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 381118865 32168 21964 MARCKS 4082 KINASE BIO-11006 BIO-11006 32170 21965 NCAM1 4684 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE LORVOTUZUMAB 32171 21966 TNFRSF1A 7132 CELL SURFACE, DRUGGABLE GENOME 178101757 32172 21967 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METOPROLOL METOPROLOL 2903243 32173 21968 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PI-103 PI-103 32175 21969 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME BMS-309403 CHEMBL247920 17554340 32177 21970 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE nppb 32178 21971 SMN1 6606 DRUGGABLE GENOME NITAZOXANIDE NITAZOXANIDE 32179 21972 CAST 831 PROTEASE INHIBITOR ACE INHIBITOR 11159730 32182 21973 MAPT 4137 DRUGGABLE GENOME ELLAGIC ACID ELLAGIC ACID 32183 21974 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor 178102629 32186 21975 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE heroin DIACETYLMORPHINE 12657887,19891732,11424981,31853823,28692418,11933204,11338173,23651028 32188 21976 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE rituximab RITUXIMAB 27173875 32189 21977 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor GDC-0980 APITOLISIB 32190 21978 MARCHF8 220972 ENZYME GMZ-2 22166048 32191 21979 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Obinutuzumab OBINUTUZUMAB 32192 21980 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Olaparib OLAPARIB 22172724 32193 21981 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Trastuzumab TRASTUZUMAB 27108243,26243863 32195 21982 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1237085 32196 21983 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME FREUND'S ADJUVANT 15146439 32197 21984 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME VALPROPYLHYDROXAMIC ACID VALPROPYLHYDROXAMIC ACID 21874153 32198 21985 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 16 32199 21986 GMNN 51053 DRUGGABLE GENOME 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 32201 21987 CYP27B1 1594 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 INTERFERON GAMMA 12055341 32202 21988 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE XANTHOANGELOL B XANTHOANGELOL B 32203 21989 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2011788838110 32205 21990 KDM4A 9682 DRUGGABLE GENOME, ENZYME BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 32210 21991 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ENDOSULFAN ENDOSULFAN 32214 21992 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME ISOSILYBIN B ISOSILYBIN B 23401473 32215 21993 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR HYDROXYUREA HYDROXYUREA 32217 21994 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor DASATINIB DASATINIB 32218 21995 PTGS2 5743 DRUGGABLE GENOME, ENZYME BROMFENAC BROMFENAC 32219 21996 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME LOVASTATIN LOVASTATIN 11884371 32221 21997 CERS6 253782 ENZYME Tumor necrosis factor alpha (TNF-alpha) inhibitors 32222 21998 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 223365984 LUCITANIB 32223 21999 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 384403651 32226 22000 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrimidopyridazinone derivative 1 32227 22001 COL22A1 169044 DRUGGABLE GENOME salbutamol ALBUTEROL 32228 22002 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE Midostaurin MIDOSTAURIN 32231 22003 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3544945 SAR-113945 32232 22004 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME TETRABROMOBENZOTRIAZOLE TETRABROMOBENZOTRIAZOLE 32233 22005 SMN2 6607 DRUGGABLE GENOME 4'-METHOXYFLAVONE 4'-METHOXYFLAVONE 32234 22006 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR cisplatin CISPLATIN 21642870 32236 22007 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrrole derivative 7 32237 22008 LIMK2 3985 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565833 32239 22009 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 187051786 SOLIFENACIN 32240 22010 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GEFITINIB GEFITINIB 32241 22011 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR RHAMNETIN RHAMNETIN 24397781 32244 22012 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL3545085 XL-228 32245 22013 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28270010-Compound-Figure24-b 32246 22014 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME PECTOLINARIGENIN PECTOLINARIGENIN 32247 22015 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE TAE-684 TAE-684 32249 22016 TSPO 706 DRUGGABLE GENOME DIAZEPAM DIAZEPAM 32250 22017 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650703 32251 22018 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HMAF IROFULVEN 9195958 32252 22019 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXYCARBOXIN OXYCARBOXIN 32253 22020 GCLC 2729 DRUGGABLE GENOME, ENZYME sulfamethoxazole SULFAMETHOXAZOLE 22824134 32254 22021 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER QUINIDINE QUINIDINE 1671173 32255 22022 MAPT 4137 DRUGGABLE GENOME FELODIPINE FELODIPINE 32256 22023 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CEPHALOCHROMIN CEPHALOCHROMIN 32257 22024 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROMETHAZINE PROMETHAZINE 32258 22025 NOS1 4842 DRUGGABLE GENOME, ENZYME ICI 182,780 15790731 32264 22026 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker CHEMBL1398126 AMILORIDE HYDROCHLORIDE 32267 22027 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME CYC-116 CYC-116 32272 22028 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 fluconazole FLUCONAZOLE 26886310 32273 22029 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist CHEMBL1095097 EPLERENONE 32274 22030 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER cisplatin CISPLATIN 23478653 32276 22031 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE PD-0166285 PD-0166285 32277 22032 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL FLUDIAZEPAM FLUDIAZEPAM 32278 22033 ATAD5 79915 NA TCMDC-124381 CHEMBL579919 32279 22034 SIRT6 51548 TRANSCRIPTION FACTOR, ENZYME inhibitor 252827474 32280 22035 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ASTEMIZOLE ASTEMIZOLE 32281 22036 PDE4D 5144 DRUGGABLE GENOME, ENZYME Piclamilast PICLAMILAST 32283 22037 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TRYPAN BLUE TRYPAN BLUE 32285 22038 ALOX15 246 ENZYME, DRUGGABLE GENOME U-73122 CHEMBL1256678 32287 22039 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME XIMELAGATRAN XIMELAGATRAN 32288 22040 E2F1 1869 TRANSCRIPTION FACTOR ADRIAMYCIN ADRIAMYCIN 9863003 32289 22041 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 1 32290 22042 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1201575 EFALIZUMAB 32295 22043 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649746 32296 22044 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR (TRICYCLO[5.2.1.0~2,6~]DEC-8-YLOXY)CARBONOTHIOYLSULFIDE CHEMBL404954 32299 22045 KLK6 5653 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 404859023 32301 22046 CFLAR 8837 DRUG RESISTANCE, DRUGGABLE GENOME, PROTEASE FINASTERIDE FINASTERIDE 11399535 32303 22047 PDE4D 5144 DRUGGABLE GENOME, ENZYME DYPHYLLINE DYPHYLLINE 32304 22048 SMN2 6607 DRUGGABLE GENOME LAPACHOL LAPACHOL 32305 22049 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamate derivative 9 32306 22050 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE DIFFERENTIATING AGENTS 2842422 32307 22051 CST3 1471 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR DIGOXIN DIGOXIN 17698593 32313 22052 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME AG-1879 CHEMBL406845 32314 22053 USP1 7398 DNA REPAIR, PROTEASE, ENZYME QUINACRINE DIHYDROCHLORIDE QUINACRINE DIHYDROCHLORIDE 32317 22054 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME GW441756X GW441756X 32318 22055 TXNRD1 7296 DRUGGABLE GENOME MOTEXAFIN GADOLINIUM 32319 22056 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135650659 32320 22057 GTF2B 2959 TRANSCRIPTION FACTOR VITAMIN D 9013769,7876247 32322 22058 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 53801088 32323 22059 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE BAFETINIB BAFETINIB 26703895 32324 22060 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CURCUMIN CURCUMIN 23742639 32326 22061 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-J2 32327 22062 F5 2153 DRUGGABLE GENOME Avatrombopag AVATROMBOPAG 32328 22063 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME Diaryl amine derivative 4 32329 22064 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565838 32330 22065 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE INGENOL MEBUTATE 32331 22066 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE FERULIC ACID 32332 22067 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ALITRETIONINE 32333 22068 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DIENESTROL DIENESTROL 32334 22069 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GSK2636771 GSK-2636771 32335 22070 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE WORTMANNIN WORTMANNIN 12133829,9484773 32336 22071 RIPK3 11035 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 381118865 32337 22072 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME GW-813893 32339 22073 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565890 32340 22074 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TAE-684 TAE-684 32342 22075 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 2,3,4,6-TETRACHLORO-PHENOL CHEMBL320361 32343 22076 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565621 MILCICLIB 32344 22077 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME GSK2245840 32346 22078 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TYRPHOSTIN 23 TYRPHOSTIN 23 32347 22079 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GLUCOCORTICOID 10524567 32349 22080 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GW7647 GW7647 23102891,18665581,23171045,18162399 32350 22081 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 315661180 ZOTIRACICLIB 32351 22082 BAZ2B 29994 NA ERBSTATIN ERBSTATIN 32352 22083 TARDBP 23435 TUMOR SUPPRESSOR FLAVANONE FLAVANONE 32353 22084 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Golvatinib GOLVATINIB 22789825 32354 22085 CA1 759 DRUGGABLE GENOME, ENZYME DICHLORPHENAMIDE DICHLORPHENAMIDE 32356 22086 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME TETRACYCLINE TETRACYCLINE 9470171 32357 22087 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ABT-700 TELISOTUZUMAB 32358 22088 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CAMPHOR CAMPHOR 32359 22089 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALPHA-ENDOSULFAN ALPHA-ENDOSULFAN 32360 22090 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 223366064 SARACATINIB 32361 22091 ATXN2 6311 NA GNF-PF-4459 CHEMBL585502 32362 22092 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545332 CEP-2563 32363 22093 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Vandetanib VANDETANIB 32364 22094 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 178102082 ADAPALENE 32365 22095 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL278703 ERTEBEREL 32366 22096 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3544983 TESEVATINIB 32367 22097 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE OXATOMIDE OXATOMIDE 32368 22098 MUC16 94025 DRUGGABLE GENOME DOCETAXEL DOCETAXEL 9288793,14756546 32369 22099 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZD9291 OSIMERTINIB 25870145,27252416 32370 22100 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME SIMVASTATIN SIMVASTATIN 16797728 32371 22101 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL484785 CRISABOROLE 32374 22102 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-699479 CHEMBL1701915 32375 22103 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME AZD4573 32378 22104 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-948 CHEMBL602158 32379 22105 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 32380 22106 MAPT 4137 DRUGGABLE GENOME GOSSYPETIN GOSSYPETIN 32381 22107 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 178102304 TOFACITINIB 32383 22108 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 374883851 32385 22109 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHYL YELLOW METHYL YELLOW 32387 22110 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER levetiracetam LEVETIRACETAM 32388 22111 NOS2 4843 DRUGGABLE GENOME, ENZYME OESTRADIOL ESTRADIOL 17068060 32389 22112 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME THAPSIGARGIN THAPSIGARGIN 32390 22113 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 381744924 32391 22114 SIRT3 23410 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME SURAMIN SURAMIN 22835719 32392 22115 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor CHEMBL3545051 CEP-37440 32394 22116 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-22 32395 22117 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SB-623 32398 22118 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE M-COPA 27197184 32399 22119 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor MLN0128 SAPANISERTIB 32400 22120 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MOCETINOSTAT MOCETINOSTAT 23829483,26287310 32401 22121 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor TOZASERTIB TOZASERTIB 19035792 32402 22122 SPP1 6696 DRUGGABLE GENOME TACROLIMUS TACROLIMUS 16103732 32403 22123 PSMA4 5685 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL451887 CARFILZOMIB 32405 22124 AMPD1 270 DRUGGABLE GENOME, ENZYME regadenoson REGADENOSON 26554440 32406 22125 POLK 51426 DNA REPAIR, ENZYME ISOORIENTIN ISOORIENTIN 32407 22126 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PESUDOGINSENOSIDE RP1 METHYL ESTER PESUDOGINSENOSIDE RP1 METHYL ESTER 20951582 32408 22127 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CLIOQUINOL CLIOQUINOL 32411 22128 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME RO-410960 CHEMBL1256291 32412 22129 MAPT 4137 DRUGGABLE GENOME SANGUINARINE SULFATE SANGUINARINE SULFATE 32414 22130 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 187051822 32416 22131 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE LAPATINIB LAPATINIB 32418 22132 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Everolimus EVEROLIMUS 28151717 32419 22133 ALOX5 240 DRUGGABLE GENOME, ENZYME montelukast MONTELUKAST 32422 22134 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CEAROIN CEAROIN 32423 22135 APOE 348 DRUGGABLE GENOME ANTI-INFLAMMATORY DRUGS 15084783 32425 22136 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AG-808 CHEMBL68534 32426 22137 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL2106468 TRICETAMIDE 32428 22138 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DECITABINE DECITABINE 32429 22139 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200532 METHDILAZINE HYDROCHLORIDE 32430 22140 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Doramapimod DORAMAPIMOD 32431 22141 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 32433 22142 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 249565925 32434 22143 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER dexrazoxane DEXRAZOXANE 25558979,20938465,25567217,16331627 32435 22144 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ABT-510 ABT-510 32436 22145 ALPL 249 ENZYME, DRUGGABLE GENOME Asfotase alfa 32438 22146 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651536 PARICALCITOL 32439 22147 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE IBUPROFEN IBUPROFEN 9118476 32440 22148 SULT1A1 6817 DRUGGABLE GENOME, ENZYME minoxidil MINOXIDIL 2390100 32441 22149 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ISOKAEMPFERIDE ISOKAEMPFERIDE 32443 22150 TNC 3371 DRUGGABLE GENOME, FIBRINOGEN 8H9 8H9 131I 32444 22151 SLC29A4 222962 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 178101327 RHODAMINE123 32445 22152 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PMID28048944-Compound-21 32446 22153 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PROGESTERONE PROGESTERONE 32447 22154 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX LOPINAVIR LOPINAVIR 32448 22155 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Aminopyridine derivative 3 32450 22156 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE FENTICLOR FENTICLOR 32451 22157 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TRIS(2,3-DIBROMOPROPYL)PHOSPHATE TRIS(2,3-DIBROMOPROPYL)PHOSPHATE 32454 22158 ATP2C1 27032 ENZYME, TRANSPORTER, DRUGGABLE GENOME SEVOFLURANE SEVOFLURANE 32455 22159 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417319 CHEMBL1392244 32456 22160 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 404859145 32457 22161 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3,4-DICHLOROISOCOUMARIN CHEMBL24983 32458 22162 SLC11A2 4891 TRANSPORTER, DRUGGABLE GENOME, CELL SURFACE inhibitor 252827472 32459 22163 GMNN 51053 DRUGGABLE GENOME TCMDC-125142 CHEMBL528791 32460 22164 NTS 4922 DRUGGABLE GENOME MAGNESIUM SULFATE 1758237 32461 22165 CSNK1G3 1456 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME SP-600125 SP-600125 32463 22166 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TRETINOIN TRETINOIN 32464 22167 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 385612185 32466 22168 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TAK-715 TAK-715 32467 22169 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME GANITUMAB GANITUMAB 23741071,24727326 32468 22170 ENOSF1 55556 ENZYME 3TC LAMIVUDINE 10864683 32471 22171 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PD-153035 CHEMBL29197 20095624 32472 22172 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PANOBINOSTAT PANOBINOSTAT 32473 22173 MAP3K14 9020 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE inhibitor 374883852 32474 22174 TMEM97 27346 NA MIN-101 ROLUPERIDONE HYDROCHLORIDE 32475 22175 FCGR2A 2212 CLINICALLY ACTIONABLE, DRUGGABLE GENOME cetuximab CETUXIMAB 23296156,27897268,28719596,30318772 32476 22176 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME agonist CHEMBL979 MEPROBAMATE 32478 22177 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650810 PERPHENAZINE 32479 22178 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 374883887 32480 22179 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178102559 NINTEDANIB 32481 22180 PBRM1 55193 CLINICALLY ACTIONABLE CTLA-4 INHIBITOR 29301960 32482 22181 PIKFYVE 200576 SERINE THREONINE KINASE, ENZYME, KINASE Apilimod dimesylate 32483 22182 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL antidepressants 23394390 32485 22183 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE dacomitinib DACOMITINIB 32488 22184 PTGS2 5743 DRUGGABLE GENOME, ENZYME MEFENAMIC ACID 32491 22185 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE articaine / epinephrine 32492 22186 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-3037 CHEMBL600336 32493 22187 RPS6KA2 6196 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565819 32494 22188 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ELLIPTECINE ELLIPTECINE 32496 22189 BRCA2 675 CLINICALLY ACTIONABLE Evofosfamide EVOFOSFAMIDE 25193512 32497 22190 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL1569 AMANTADINE HYDROCHLORIDE 32498 22191 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IODOMELATONIN IODOMELATONIN 32499 22192 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649788 32501 22193 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GSK2126458 OMIPALISIB 32502 22194 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor MK4827 NIRAPARIB 32503 22195 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652110 32504 22196 ATAD5 79915 NA TCMDC-123748 CHEMBL530609 32505 22197 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 32506 22198 NDUFA1 4694 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 32508 22199 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME (S)APOMORPHINE (S)APOMORPHINE 32509 22200 TSPO 706 DRUGGABLE GENOME CLORAZEPATE CLORAZEPIC ACID 32510 22201 TSPO 706 DRUGGABLE GENOME Aryl oxyanilide derivative 1 32511 22202 PDE4A 5141 DRUGGABLE GENOME, ENZYME IBUDILAST IBUDILAST 32512 22203 PTK6 5753 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, ENZYME CEDIRANIB CEDIRANIB 32513 22204 PSMD11 5717 KINASE inhibitor CHEMBL451887 CARFILZOMIB 32514 22205 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Isoflavone derivative 7 32515 22206 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Bevacizumab BEVACIZUMAB 25363205 32517 22207 FAAH 2166 ENZYME, DRUGGABLE GENOME PF-750 CHEMBL560590 23287055 32518 22208 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE hydrocodone HYDROCODONE 23703421 32519 22209 BAZ2B 29994 NA TCMDC-123600 CHEMBL531296 32521 22210 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR Conjugated Estrogens 32524 22211 COL4A2 1284 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 32525 22212 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650104 CISAPRIDE 32529 22213 AKR1C3 8644 ENZYME, DRUGGABLE GENOME Indomethacin analog 2 32530 22214 PTGS2 5743 DRUGGABLE GENOME, ENZYME ETORICOXIB ETORICOXIB 32532 22215 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE 2-piperidine thiazole derivative 2 32533 22216 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME oxaliplatin OXALIPLATIN 32534 22217 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100866 32536 22218 CBL 867 KINASE, ENZYME, CLINICALLY ACTIONABLE Quizartinib QUIZARTINIB 22990016 32537 22219 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME RO-5068760 CHEMBL1956073 20053779 32538 22220 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE RUCAPARIB RUCAPARIB 32541 22221 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE activator 385612180 32542 22222 LNPEP 4012 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, TRANSPORTER, PROTEASE US10023583, Example 8 32545 22223 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-60339 CHEMBL1448793 32546 22224 HSPB1 3315 DRUGGABLE GENOME NSC-67746 CHEMBL333177 32547 22225 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor 363894172 32548 22226 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL3544971 DEXTROAMPHETAMINE SULFATE 32549 22227 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Lepirudin LEPIRUDIN 32551 22228 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650948 32552 22229 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PF-562271 PF-00562271 32553 22230 ATXN2 6311 NA INDIRUBIN SULFATE SU-9516 32554 22231 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 94777 CHEMBL407501 32555 22232 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 7,12-DIMETHYL-BENZO[A]ANTHRACENE CHEMBL329673 32556 22233 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 178102341 32557 22234 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE TYROSINE KINASE INHIBITOR 11978788 32558 22235 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 6-13 32559 22236 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 LIOTHYRONINE LIOTHYRONINE 22931300 32562 22237 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE medroxyprogesterone MEDROXYPROGESTERONE ACETATE 18695978 32563 22238 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR RADICICOL RADICICOL 24984936,17603540,16499313 32564 22239 SLC25A5 292 DRUGGABLE GENOME, TRANSPORTER TRICHOSTATIN A 10657244 32566 22240 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER felodipine FELODIPINE 32567 22241 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 310264693 ACALABRUTINIB 32568 22242 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHOLINE CHLORIDE CHOLINE CHLORIDE 32569 22243 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IONOMYCIN IONOMYCIN 15294043 32570 22244 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor ENZASTAURIN ENZASTAURIN 32572 22245 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 381118866 32573 22246 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PF-562271 PF-00562271 32575 22247 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME MOCETINOSTAT MOCETINOSTAT 23829483,26287310 32576 22248 SDHB 6390 ENZYME, CLINICALLY ACTIONABLE DOXORUBICIN DOXORUBICIN 6672210,16278810 32577 22249 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OXYBUTYNIN OXYBUTYNIN 32578 22250 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME NU172 32579 22251 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR GW7647 GW7647 32580 22252 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER FLAVANONE FLAVANONE 32581 22253 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-574 CHEMBL582737 32584 22254 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Anti-HER2 CAR-T 32585 22255 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GERONTOXANTHONE H GERONTOXANTHONE H 25838141 32587 22256 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER RO 31-8220 8624264 32588 22257 GPD2 2820 DRUGGABLE GENOME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 32589 22258 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650373 32591 22259 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652471 OCTREOTIDE 32592 22260 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME SAND-26 BEGELOMAB 32593 22261 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CEFSULODIN SODIUM CEFSULODIN SODIUM 32594 22262 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER LAMIVUDINE LAMIVUDINE 17172311 32595 22263 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178101539 BUMETANIDE 32597 22264 PLCG1 5335 ENZYME, KINASE, PHOSPHOLIPASE, DRUGGABLE GENOME 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 32599 22265 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FIPRONIL FIPRONIL 32600 22266 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR AZD-1080 AZD-1080 32602 22267 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NAPHAZOLINE NAPHAZOLINE 32603 22268 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME DASATINIB DASATINIB 32604 22269 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME BICALUTAMIDE BICALUTAMIDE 9622849 32605 22270 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME SAR-114137 32607 22271 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME MELPHALAN MELPHALAN 8621235 32609 22272 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 252166576 ITACITINIB 32610 22273 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL PMID30185082-Compound-57 32611 22274 ATAD5 79915 NA AMSACRINE AMSACRINE 32617 22275 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR COLCHICINE COLCHICINE 1946455 32619 22276 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME irinotecan IRINOTECAN 32620 22277 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DSC-103 32621 22278 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651970 32625 22279 ETFDH 2110 ENZYME methylphenidate METHYLPHENIDATE 29382897 32626 22280 ABHD6 57406 PHOSPHOLIPASE, ENZYME inhibitor 329968420 32627 22281 EED 8726 ENZYME, CLINICALLY ACTIONABLE allosteric modulator 387065597 32628 22282 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GSK461364 GSK-461364 32629 22283 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME LY3127804 32631 22284 CXCL8 3576 DRUGGABLE GENOME ACE INHIBITOR 9846973 32632 22285 HMGCR 3156 ENZYME, DRUGGABLE GENOME PRAVASTATIN PRAVASTATIN 32633 22286 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR RETINOID 8940178 32634 22287 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TACRINE TACRINE 22931300 32636 22288 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 252827469 32639 22289 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME MEDI-3617 MEDI-3617 32640 22290 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 32641 22291 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME Methylbenzenesulfonamide derivative 1 32642 22292 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE NECITUMUMAB NECITUMUMAB 32643 22293 KDM4A 9682 DRUGGABLE GENOME, ENZYME THIOGUANINE THIOGUANINE 32645 22294 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 381744955 32647 22295 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME YANGONIN YANGONIN 32648 22296 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ILOPERIDONE ILOPERIDONE 32649 22297 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FAS LIGAND 12660450,10974031 32651 22298 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE WORTMANNIN WORTMANNIN 10187855 32652 22299 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565837 32654 22300 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME FENOLDOPAM FENOLDOPAM 32655 22301 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME VERAPAMIL VERAPAMIL 9354939 32657 22302 KDM4A 9682 DRUGGABLE GENOME, ENZYME LAVENDUSTIN B LAVENDUSTIN B 32658 22303 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE IL-2 ALDESLEUKIN 2528593,1827816 32659 22304 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE LASALOCID A SODIUM LASALOCID A SODIUM 32660 22305 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR tiratricol TIRATRICOL 32661 22306 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL2001019 PF-04217903 32662 22307 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE ANTIBIOTIC ANTIBIOTIC 2654492 32663 22308 UGT2B7 7364 DRUGGABLE GENOME (S)-methadone 17178267 32664 22309 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 atorvastatin ATORVASTATIN 18528690,19802823 32665 22310 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE LINIFANIB LINIFANIB 32667 22311 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 354702222 32668 22312 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TAMOXIFEN CITRATE TAMOXIFEN CITRATE 32669 22313 CDC5L 988 DNA REPAIR gemcitabine GEMCITABINE 22838950 32670 22314 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor LAPATINIB DITOSYLATE 32671 22315 GMNN 51053 DRUGGABLE GENOME TCMDC-123579 CHEMBL533954 32672 22316 CD44 960 DRUGGABLE GENOME, CELL SURFACE GP-120 7539755 32673 22317 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRADIOL ESTRADIOL 32675 22318 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-2A, RECOMBINANT 32676 22319 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PHENYLBUTAZONE PHENYLBUTAZONE 32677 22320 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody AV203 32678 22321 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE M-CSF CILMOSTIM 11061591 32680 22322 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CATECHOL CATECHOL 32681 22323 IL1B 3553 KINASE, DRUGGABLE GENOME LY-2189102 32682 22324 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Epoxysuccinate derivative 4 32685 22325 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR inhibitor 187051779 LORLATINIB 32687 22326 PNMT 5409 DRUGGABLE GENOME, ENZYME NERVE GROWTH FACTOR 16926281 32688 22327 RRM2B 50484 ENZYME, DRUGGABLE GENOME, DNA REPAIR MOTEXAFIN GADOLINIUM 32690 22328 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME PD-0166285 PD-0166285 32691 22329 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178102616 32692 22330 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR H2O2 9406937 32693 22331 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME activator 135652731 32695 22332 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE FLOXURIDINE FLOXURIDINE 32696 22333 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ILOPROST ILOPROST 32699 22334 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-33 32700 22335 PDE4B 5142 DRUGGABLE GENOME, ENZYME OGLEMILAST OGLEMILAST 32701 22336 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL521 IBUPROFEN 32703 22337 GSTM1 2944 DRUGGABLE GENOME, ENZYME METHOTREXATE METHOTREXATE 17180579 32704 22338 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME LINIFANIB LINIFANIB 32706 22339 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GARCINOLIC ACID GARCINOLIC ACID 32707 22340 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR Vorinostat VORINOSTAT 25605023 32708 22341 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE DIGOXIN DIGOXIN 32709 22342 TNFRSF18 8784 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME TRX518 32712 22343 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME GAMOLENIC ACID GAMOLENIC ACID 32715 22344 TUBA4A 7277 DRUGGABLE GENOME CABAZITAXEL CABAZITAXEL 32718 22345 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TRIPROLIDINE TRIPROLIDINE 32720 22346 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE AST-005 32722 22347 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE SPIRONOLACTONE SPIRONOLACTONE 7079590 32723 22348 PERP 64065 NA cyclophosphamide CYCLOPHOSPHAMIDE 32724 22349 MAP3K5 4217 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565813 32725 22350 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL2103741 LEVOTHYROXINE SODIUM 32726 22351 ALOX15 246 ENZYME, DRUGGABLE GENOME GUTHION GUTHION 32727 22352 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33i 32728 22353 USP1 7398 DNA REPAIR, PROTEASE, ENZYME MK-571 MK-571 32730 22354 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CHELERYTHRINE CHELERYTHRINE 32731 22355 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL cerivastatin CERIVASTATIN 21386754 32732 22356 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE LASALOCID A SODIUM LASALOCID A SODIUM 32734 22357 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME QUINALIZARIN QUINALIZARIN 32735 22358 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SL-327 CHEMBL261237 32737 22359 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME SORAFENIB SORAFENIB 32739 22360 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME heroin DIACETYLMORPHINE 21723677 32741 22361 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TREMELIMUMAB TREMELIMUMAB 32744 22362 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL593430 ATAGABALIN 32746 22363 KDM4A 9682 DRUGGABLE GENOME, ENZYME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 32747 22364 PSMA3 5684 PROTEASE, DRUGGABLE GENOME inhibitor BORTEZOMIB BORTEZOMIB 32750 22365 MAPT 4137 DRUGGABLE GENOME SJ000059275 CHEMBL603952 32751 22366 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor 363894172 32753 22367 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NILUTAMIDE NILUTAMIDE 22931300 32754 22368 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METHYSERGIDE METHYSERGIDE 32755 22369 TARDBP 23435 TUMOR SUPPRESSOR SJ000032154 CHEMBL591876 32756 22370 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LINIFANIB LINIFANIB 32757 22371 POLK 51426 DNA REPAIR, ENZYME S(+)-ISOPROTERENOL-BITARTRATE CHEMBL1257092 32761 22372 CRBN 51185 ENZYME, DRUG RESISTANCE CC-122 AVADOMIDE 32762 22373 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AFATINIB AFATINIB 23982599,24035188,32193290,25589191,26051236,24439929,32226941,27083334,24353160,22452895,23816960,25948633,27304188 32763 22374 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Ceftriaxone CEFTRIAXONE 32764 22375 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL1234354 PF-04691502 32766 22376 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TALIPEXOLE HYDROCHLORIDE TALIPEXOLE HYDROCHLORIDE 32767 22377 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 32768 22378 GDF15 9518 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR RESVERATROL RESVERATROL 11895857 32771 22379 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SLAZINIC ACID SLAZINIC ACID 32773 22380 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE Trametinib TRAMETINIB 32775 22381 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Erythromycin ERYTHROMYCIN 32779 22382 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME ETOPOSIDE ETOPOSIDE 15019164 32780 22383 MPHOSPH8 54737 NA IODOACETAMIDE IODOACETAMIDE 32781 22384 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103918 MK-0249 32782 22385 NOX1 27035 ION CHANNEL, ENZYME, TRANSPORTER, DRUGGABLE GENOME TCMDC-125505 CHEMBL587104 32783 22386 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor FK-228 ROMIDEPSIN 32784 22387 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE Clobetasol CLOBETASOL 32785 22388 CEL 1056 CELL SURFACE, DRUGGABLE GENOME, ENZYME RESVERATROL RESVERATROL 16099206 32786 22389 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Trametinib TRAMETINIB 28783719 32791 22390 CD55 1604 DRUGGABLE GENOME, CELL SURFACE COXSACKIEVIRUS TYPE A21 32792 22391 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SELENIUM 12669817 32793 22392 PTGS2 5743 DRUGGABLE GENOME, ENZYME Naproxen NAPROXEN 32795 22393 TRPC4 7223 ION CHANNEL, KINASE, DRUGGABLE GENOME, CELL SURFACE blocker 381744972 32796 22394 F2RL3 9002 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME RUSALATIDE RUSALATIDE 32799 22395 PDE3A 5139 ENZYME, DRUGGABLE GENOME Aminophylline AMINOPHYLLINE 32800 22396 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BYL719 ALPELISIB 32802 22397 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE AVI-5126 32803 22398 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR U-0126 U-0126 32805 22399 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NSC-11437 CHEMBL1814509 32806 22400 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 223366150 32807 22401 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker 135651249 32808 22402 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE GW441756X GW441756X 32809 22403 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALCIMYCIN CALCIMYCIN 32811 22404 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER aldosterone ALDOSTERONE 32813 22405 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE (R)-FLECAINIDE (R)-FLECAINIDE 32814 22406 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MYCOPHENOLATE MOFETIL MYCOPHENOLATE MOFETIL 32815 22407 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME 3-acylidene-2-oxoindole derivative 2 32816 22408 CCNB1 891 DRUGGABLE GENOME SELICICLIB SELICICLIB 21080703 32817 22409 GALNT14 79623 ENZYME fluorouracil FLUOROURACIL 31611591,21635146 32818 22410 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CHEMBL2068724 ACAMPROSATE CALCIUM 32820 22411 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE MORIN MORIN 32824 22412 CA9 768 DRUGGABLE GENOME, ENZYME PHENOL PHENOL 32825 22413 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 32827 22414 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-45382 CHEMBL1214274 32828 22415 IRS2 8660 KINASE, CLINICALLY ACTIONABLE ASPIRIN ASPIRIN 18059035 32829 22416 MPHOSPH8 54737 NA PD-169316 PD-169316 32830 22417 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL203567 RO-3201195 32831 22418 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GEMCITABINE GEMCITABINE 29941343 32834 22419 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME CAP1-6D 32835 22420 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE HYDROGEN PEROXIDE 8959153 32836 22421 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor CHEMBL3545052 FIMEPINOSTAT 32837 22422 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER tetrabenazine TETRABENAZINE 32838 22423 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-46 32839 22424 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR DIFFERENTIATING AGENTS 11720243 32840 22425 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE ENTRECTINIB ENTRECTINIB 32841 22426 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER INGN-225 32842 22427 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Ceritinib CERITINIB 25394791 32843 22428 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE VANDETANIB VANDETANIB 32844 22429 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Pyrrolo[2,3-d]pyrimidine derivative 2 32846 22430 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor ARQ736 32847 22431 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652643 32849 22432 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE PMID25726713-Compound-49 32850 22433 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 178103584 32851 22434 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER METHADONE METHADONE 15876424 32852 22435 KAT2B 8850 ENZYME, DRUGGABLE GENOME 6-DECYLSALICYLIC ACID CHEMBL416038 20655754 32853 22436 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL586701 ZSTK-474 32854 22437 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PROTEASOME INHIBITOR 15613543 32856 22438 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 387065606 32857 22439 SMN1 6606 DRUGGABLE GENOME CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 32858 22440 TNFRSF1B 7133 DRUGGABLE GENOME infliximab INFLIXIMAB 25850964,18565259,25537528,22129793 32859 22441 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROBENECID PROBENECID 32861 22442 PSMA6 5687 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL2103884 OPROZOMIB 32862 22443 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HYDROXYCAMPTOTHECIN HYDROXYCAMPTOTHECIN 32863 22444 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ETHINYL ESTRADIOL 32867 22445 CLK3 1198 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, TYROSINE KINASE LEUCETTAMINE B LEUCETTAMINE B 22998443 32868 22446 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 381118852 32869 22447 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NIMESULIDE NIMESULIDE 22931300 32870 22448 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor TIVANTINIB TIVANTINIB 32872 22449 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROCHLORPERAZINE PROCHLORPERAZINE 32873 22450 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SULISOBENZONE SULISOBENZONE 32874 22451 GLS 2744 ENZYME OXYTETRACYCLINE HYDROCHLORIDE OXYTETRACYCLINE HYDROCHLORIDE 32875 22452 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SNC-80 SNC-80 32876 22453 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Imidazo pyridine derivative 3 32878 22454 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE SJ000044511 CHEMBL592124 32879 22455 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROPARGITE PROPARGITE 32880 22456 IL13RA2 3598 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ICT-107 32881 22457 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-5051 CHEMBL600773 32882 22458 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 310264781 ADL-5747 32883 22459 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652086 32884 22460 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MITOXANTRONE MITOXANTRONE 23442188 32885 22461 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CENISERTIB CENISERTIB 32886 22462 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BYL719 ALPELISIB 32888 22463 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME PMID25468267-Compound-56 32889 22464 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CCT018159 CHEMBL399530 32890 22465 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TIMOLOL TIMOLOL 32891 22466 TUBB4B 10383 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 32892 22467 MGLL 11343 DRUGGABLE GENOME, ENZYME Piperazine carbamic compound 2 32893 22468 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-992 CHEMBL602561 32894 22469 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE GSK1070916 GSK-1070916 32895 22470 HR 55806 NUCLEAR HORMONE RECEPTOR LCB-2183 32898 22471 LTC4S 4056 ENZYME, DRUGGABLE GENOME inhibitor 252827532 32899 22472 KDM4A 9682 DRUGGABLE GENOME, ENZYME RESCINNAMINE RESCINNAMINE 32901 22473 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME TAE-684 TAE-684 32902 22474 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE CARBOPLATIN CARBOPLATIN 10081494 32904 22475 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TRAZODONE TRAZODONE 32905 22476 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME VIOXX ROFECOXIB 14627349 32907 22477 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme25-3 32908 22478 PDE4A 5141 DRUGGABLE GENOME, ENZYME PENTOXIFYLLINE PENTOXIFYLLINE 32909 22479 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL1201752 IXABEPILONE 32910 22480 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GO-6976 GO-6976 32911 22481 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 WAY-629 CHEMBL258465 32912 22482 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE GEFITINIB GEFITINIB 24685132 32914 22483 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antagonist CHEMBL1743019 FIGITUMUMAB 32915 22484 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DACTINOMYCIN DACTINOMYCIN 32916 22485 RPSA 3921 NA MITOXANTRONE MITOXANTRONE 8630412 32918 22486 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROTHYMOSIN ALPHA 15657435 32919 22487 PSMD1 5707 NA inhibitor CHEMBL325041 BORTEZOMIB 32920 22488 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL DIAZEPAM DIAZEPAM 32921 22489 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker 223366051 32922 22490 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PENCYCURON PENCYCURON 32925 22491 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545322 PANULISIB 32927 22492 JUNB 3726 TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR DEXAMETHASONE DEXAMETHASONE 9024781 32928 22493 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GANCICLOVIR GANCICLOVIR 8986436 32930 22494 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CINALUKAST CINALUKAST 32931 22495 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 1245272 CHEMBL408850 32932 22496 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CINOLAZEPAM CINOLAZEPAM 32933 22497 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PW2101 32934 22498 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZOMEPIRAC SODIUM ZOMEPIRAC SODIUM 32937 22499 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GLIOTOXIN GLIOTOXIN 32939 22500 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TAMOXIFEN CITRATE TAMOXIFEN CITRATE 32941 22501 NDUFS7 374291 ENZYME inhibitor CHEMBL3545135 NV-128 32942 22502 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CYSTEINE CYSTEINE 32943 22503 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor PONATINIB PONATINIB 32944 22504 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL568 OXAZEPAM 32945 22505 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 328083476 32947 22506 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME ALVOCIDIB ALVOCIDIB 32949 22507 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX RETINOIDS 1323296 32950 22508 TARDBP 23435 TUMOR SUPPRESSOR PIPLARTINE PIPLARTINE 32951 22509 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME EOTAXIN 12576300 32952 22510 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SULCONAZOLE NITRATE SULCONAZOLE NITRATE 32953 22511 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME L-689560 CHEMBL287327 32955 22512 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME OMEPRAZOLE OMEPRAZOLE 8529327 32956 22513 UGT2B4 7363 DRUGGABLE GENOME ibuprofen IBUPROFEN 25502615 32958 22514 HMGCR 3156 ENZYME, DRUGGABLE GENOME Pitavastatin derivative 1 32959 22515 GMNN 51053 DRUGGABLE GENOME GNF-PF-5058 CHEMBL601180 32961 22516 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE LY-2875358 EMIBETUZUMAB 32962 22517 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Aflibercept AFLIBERCEPT 32963 22518 IGF2R 3482 ENZYME, DRUGGABLE GENOME, CELL SURFACE EP-128504 32964 22519 CBX1 10951 NA TETRYDAMINE TETRYDAMINE 32965 22520 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DEQUALINIUM DEQUALINIUM 32966 22521 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME RETINOL RETINOL 17202653 32967 22522 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 135649822 32968 22523 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TIRAPAZAMINE TIRAPAZAMINE 9647614 32969 22524 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201063 PROPAFENONE HYDROCHLORIDE 32972 22525 UGT1A7 54577 DRUGGABLE GENOME, ENZYME ritonavir RITONAVIR 17058217 32973 22526 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE JNJ-61186372 JNJ-61186372 27216193 32974 22527 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE OSI-027 OSI-027 21673091 32975 22528 TGFBR2 7048 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME TG-C 32977 22529 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE 32978 22530 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME CARMINOMYCIN CARUBICIN 32979 22531 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 348353656 SOLCITINIB 32981 22532 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 249565620 DANUSERTIB 32984 22533 SLC29A4 222962 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER HISTAMINE HISTAMINE 22396231 32985 22534 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME RO-4882224 CHEMBL1077391 19762240 32986 22535 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 381118873 32987 22536 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102412 32989 22537 SLC47A1 55244 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER metformin METFORMIN 23267855,23873119,28834135,24624919,26004431,22882994,22722338 32992 22538 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 zidovudine ZIDOVUDINE 22960662 32993 22539 GPA33 10223 DRUGGABLE GENOME KRN-330 KRN-330 32994 22540 HTT 3064 DRUGGABLE GENOME TCMDC-125567 CHEMBL530049 32995 22541 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME levetiracetam LEVETIRACETAM 30020991 32998 22542 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROPIOMAZINE PROPIOMAZINE 32999 22543 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650688 NALTRIBEN 33001 22544 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME DEHYDROEPIANDROSTERONE PRASTERONE 15448171 33002 22545 GMNN 51053 DRUGGABLE GENOME DNDI1417719 CHEMBL1420370 33003 22546 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME DI-TERT-BUTYLHYDROQUINONE CHEMBL480626 33005 22547 LIPA 3988 ENZYME, DRUGGABLE GENOME HORMONES 6543190,7272337,7056842 33006 22548 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE LENVATINIB LENVATINIB 33009 22549 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-668394 CHEMBL336095 33011 22550 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650043 33013 22551 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200606 MEXILETINE HYDROCHLORIDE 33015 22552 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE METHYLNALTREXONE BROMIDE 33017 22553 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AG-537 CHEMBL67535 33019 22554 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE Other general anesthetics 30136624 33020 22555 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor BKM120 BUPARLISIB 33021 22556 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE BERKELEYAMIDE C BERKELEYAMIDE C 18330993 33023 22557 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RITANSERIN RITANSERIN 33024 22558 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 1,3-DIACETYLVILASININ CHEMBL463701 33025 22559 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000032159 CHEMBL591361 33026 22560 RRM2 6241 DRUGGABLE GENOME, ENZYME MOTEXAFIN GADOLINIUM 33027 22561 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417447 CHEMBL1307453 33030 22562 CPS1 1373 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME sodium benzoate / sodium phenylacetate 33031 22563 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME Tricyclic compound 10 33032 22564 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE HEN EGG LYSOZYME 9492007 33033 22565 GTF2B 2959 TRANSCRIPTION FACTOR PC4 8617240 33034 22566 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417447 CHEMBL1307453 33035 22567 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor FK-228 ROMIDEPSIN 33036 22568 PDE10A 10846 ENZYME, DRUGGABLE GENOME Pyrido[1,2,4]triazolo[4,3-a]pyrazine derivative 3 33037 22569 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BENOXINATE BENOXINATE 33039 22570 NT5C2 22978 ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE mercaptopurine MERCAPTOPURINE 15990089 33040 22571 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Nilotinib NILOTINIB 28843487,20442311,25594040,25209843,28327988,17699867,23582185 33043 22572 GC 2638 DRUGGABLE GENOME CHEMBL2105671 AFEGOSTAT TARTRATE 33046 22573 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 178101428 DILAZEP 33047 22574 ARSA 410 DRUGGABLE GENOME, ENZYME MELEVODOPA MELEVODOPA 33048 22575 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE IL-12 16751417 33049 22576 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BECLOMETHASONE BECLOMETHASONE 33052 22577 SLC9A3 6550 DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE, EXCHANGER inhibitor CHEMBL2107782 33053 22578 EGLN3 112399 DRUGGABLE GENOME, ENZYME inhibitor 252827454 33054 22579 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE EVEROLIMUS EVEROLIMUS 33056 22580 PDE10A 10846 ENZYME, DRUGGABLE GENOME PF-02545920 MARDEPODECT 33058 22581 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE JNJ-7706621 JNJ-7706621 33059 22582 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650725 33060 22583 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SCH772984 26267534,27222538,27312529 33061 22584 SLC2A3 6515 DRUGGABLE GENOME, TRANSPORTER 178101360 33063 22585 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME TOPOTECAN HYDROCHLORIDE TOPOTECAN HYDROCHLORIDE 33066 22586 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE 681640 CHEMBL379975 33069 22587 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Cytolin 33070 22588 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR RAC-ARISTOYUNNOLIN D CHEMBL2333543 33071 22589 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TETRAZOLIUM RED TETRAZOLIUM RED 33073 22590 BAZ2B 29994 NA ISOCONAZOLE ISOCONAZOLE 33077 22591 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DERRUBONE DERRUBONE 18020309 33078 22592 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE benazepril BENAZEPRIL 16081343,15226090 33080 22593 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CGP41251 15914319 33081 22594 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Linagliptin LINAGLIPTIN 33082 22595 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL661 ALPRAZOLAM 33083 22596 GMNN 51053 DRUGGABLE GENOME LIDAMIDINE HYDROCHLORIDE LIDAMIDINE HYDROCHLORIDE 33084 22597 GPR183 1880 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178101171 33085 22598 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 1-HEXYLPYRIDINIUM IODIDE CHEMBL555242 33086 22599 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9216972, 132 33088 22600 ABCA1 19 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE fenofibrate FENOFIBRATE 33090 22601 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 temazepam TEMAZEPAM 33091 22602 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100392 33093 22603 SLC38A4 55089 TRANSPORTER 178101263 33094 22604 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLURANDRENOLIDE FLURANDRENOLIDE 33096 22605 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135652067 33097 22606 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME RESMINOSTAT RESMINOSTAT 33098 22607 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE RAPAMYCIN SIROLIMUS 17010674 33100 22608 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545200 S-222611 33103 22609 GRAMD1B 57476 TRANSPORTER lithium LITHIUM 29121268 33104 22610 PDE6D 5147 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL628 PENTOXIFYLLINE 33108 22611 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE RESACTIN A RESACTIN A 33109 22612 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME Bosutinib BOSUTINIB 33110 22613 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Ethinyl Estradiol 33111 22614 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-Table1Example5 33112 22615 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE A-443654 A-443654 33113 22616 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX GDC-0941 PICTILISIB 27020857 33114 22617 CBX1 10951 NA INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 33115 22618 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PERVILLEINE B PERVILLEINE B 11754602 33116 22619 XRCC1 7515 CLINICALLY ACTIONABLE GEMCITABINE GEMCITABINE 19157633 33117 22620 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL1628502 GABAPENTIN ENACARBIL 33118 22621 ALOX15 246 ENZYME, DRUGGABLE GENOME HAEMATOXYLIN HAEMATOXYLIN 33119 22622 QPCT 25797 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252166568 33121 22623 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CID 2056784 CHEMBL261123 33122 22624 NOS1 4842 DRUGGABLE GENOME, ENZYME METHYLTESTOSTERONE METHYLTESTOSTERONE 15934456 33123 22625 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE PMID25656651-Compound-21b 33124 22626 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE 2-piperidine thiazole derivative 1 33126 22627 DYRK2 8445 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID28766366-Compound-Scheme16DMAT 33128 22628 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GENISTEIN GENISTEIN 33129 22629 CEACAM7 1087 DRUGGABLE GENOME IFN 14636419 33130 22630 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-19 33133 22631 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 135651723 33134 22632 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GW9662 CHEMBL375270 33135 22633 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DOBUTAMINE DOBUTAMINE 33136 22634 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE TENECTEPLASE TENECTEPLASE 33137 22635 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PD-0325901 PD-0325901 27488531 33138 22636 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Neratinib NERATINIB 26725216,26243863 33139 22637 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DESIPRAMINE DESIPRAMINE 33141 22638 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE LENVATINIB LENVATINIB 33142 22639 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME VALPROIC ACID VALPROIC ACID 18294844,16921367,25304896 33143 22640 PPAT 5471 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200751 MERCAPTOPURINE 33144 22641 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-117079 CHEMBL471225 33145 22642 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GW7647 GW7647 18162399 33146 22643 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE MK2206 MK-2206 27370604 33148 22644 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME Ruxolitinib derivative 1 33149 22645 PSMD1 5707 NA inhibitor CARFILZOMIB CARFILZOMIB 33150 22646 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-5 33151 22647 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE (-)-U-50488 (-)-U-50488 33152 22648 FIP1L1 81608 CLINICALLY ACTIONABLE, KINASE Imatinib IMATINIB 33156 22649 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator CHEMBL1200644 FONDAPARINUX SODIUM 33157 22650 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NALOXONE METHIODIDE NALOXONE METHIODIDE 33158 22651 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME ACNU 9537648 33161 22652 ARHGAP12 94134 ENZYME methylphenidate METHYLPHENIDATE 29382897 33162 22653 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PANITUMUMAB PANITUMUMAB 23020132,22608338,26619011,21483012,22351686,19001320,21156289,20368568,19255327,22048237,19561230,19010912,23549875,25024077,23489023,18541894,24586605,24508103,22773810,23833300,23812671,24576830,19238210,20818844,23612012,23251002,22356324,20857202,22536370,22997239,21163703,15035987,23470635,21663470,24594804,22586120,20413299,22805292,19537845,14679157,22663011,21975775,22038996,22448344,12068308,24163374,19773371,24354346,23325582,24583796,23031422,22735384,21683865,25370471,21639808,22281684,22649091,22241789,24570209,23918947,25989278,22389471,23934108,22180495,23524406,26678033,19018267,24388723,23845441,23614898,25157968,20619739,12460919,24107445,12460918,21594703,20350999,20630094,21426297,19404918,22743296,24396464,22972589,21129611,23406027 33165 22654 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME Prinomastat PRINOMASTAT 33167 22655 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IPI-504 RETASPIMYCIN HYDROCHLORIDE 33169 22656 GLS 2744 ENZYME 2-HYDROXYESTRADIOL CHEMBL467987 33174 22657 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-60 33176 22658 ATXN2 6311 NA NORTRIPTYLINE NORTRIPTYLINE 33177 22659 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME INCB18424 33181 22660 POLK 51426 DNA REPAIR, ENZYME BUTEIN BUTEIN 33184 22661 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GSK2256098 GSK-2256098 25833835 33185 22662 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 385612194 33186 22663 E2F1 1869 TRANSCRIPTION FACTOR 17 BETA-ESTRADIOL 12697671 33187 22664 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX TRETINOIN TRETINOIN 33189 22665 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 telaprevir TELAPREVIR 33190 22666 IFNG 3458 DRUGGABLE GENOME ALL-TRANS RETINOIC ACID 9792441 33193 22667 TOP2B 7155 DRUGGABLE GENOME, ENZYME GRC-6211 GRC-6211 33195 22668 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME 8-(3-CHLOROSTYRYL)CAFFEINE CHEMBL26138 33196 22669 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor PLX108-01 33197 22670 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE LEUCOVORIN LEUCOVORIN 33198 22671 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME IODOPHTHALEIN IODOPHTHALEIN 33200 22672 ATAD5 79915 NA TCMDC-125821 CHEMBL547977 33201 22673 COL5A3 50509 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 33203 22674 TUBB3 10381 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 33205 22675 UGT1A7 54577 DRUGGABLE GENOME, ENZYME mycophenolic acid 24220207 33206 22676 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor MEK162 BINIMETINIB 33208 22677 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR quinapril QUINAPRIL 11849656 33211 22678 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR lorlatinib LORLATINIB 33214 22679 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME SJ000047240 CHEMBL590706 33217 22680 CBX1 10951 NA RABEPRAZOLE SODIUM RABEPRAZOLE SODIUM 33218 22681 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME ASP8232 33219 22682 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE AT-101 ISOSORBIDE 33220 22683 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102626 33221 22684 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR TRASTUZUMAB TRASTUZUMAB 22842582 33222 22685 EGFL7 51162 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE MEGF0444A PARSATUZUMAB 33225 22686 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL448 PENTOBARBITAL 33226 22687 RCE1 9986 ENZYME, PROTEASE, DRUGGABLE GENOME FLUNARIZINE DIHYDROCHLORIDE FLUNARIZINE DIHYDROCHLORIDE 33227 22688 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE DASATINIB DASATINIB 33228 22689 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SB-228357 CHEMBL14276 33231 22690 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MELPHALAN MELPHALAN 15779864,1988111 33232 22691 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME ALISERTIB ALISERTIB 33233 22692 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME XL281 33235 22693 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME 2-ENE-VALPROATE CHEMBL117487 17566732 33236 22694 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL558752 RAF-265 33237 22695 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR Cholic acid - Asklepion 33238 22696 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME 4SCAR19 and 4SCAR70 33239 22697 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DACTINOMYCIN DACTINOMYCIN 33240 22698 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CGP-60474 CHEMBL300389 33241 22699 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Amocarzine AMOCARZINE 33243 22700 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GBR-12909 VANOXERINE 33245 22701 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME 3-HYDROXYANTHRANILIC ACID CHEMBL445304 18003900 33246 22702 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME TAMOXIFEN TAMOXIFEN 9067554 33247 22703 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Coenzyme Q10 analog 25343117 33248 22704 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DACOMITINIB DACOMITINIB 33249 22705 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GNF-PF-4997 CHEMBL306147 33251 22706 ENO2 2026 CELL SURFACE STREPTOZOTOCIN STREPTOZOCIN 2146046 33252 22707 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PMID29671355-Compound-56 33253 22708 KLKB1 3818 DRUGGABLE GENOME, PROTEASE, ENZYME ANTITHROMBIN 33255 22709 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CARVEDILOL CARVEDILOL 33256 22710 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102914 33258 22711 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL1795071 RUXOLITINIB PHOSPHATE 33261 22712 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR T091317 T091317 33262 22713 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RGB-286638 RGB-286638 33264 22714 TUBA1C 84790 DRUGGABLE GENOME CHEMBL2304041 SAGOPILONE 33266 22715 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR THIOLUTIN THIOLUTIN 33267 22716 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 esomeprazole ESOMEPRAZOLE 33270 22717 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME flucytosine FLUCYTOSINE 33271 22718 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HARMAN HARMAN 33275 22719 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE Eslicarbazepine ESLICARBAZEPINE 33276 22720 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor 178103398 ACETAZOLAMIDE 33277 22721 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RO-137410 CHEMBL275311 33278 22722 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BEZ235 DACTOLISIB 33279 22723 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL538943 VINORELBINE TARTRATE 33281 22724 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DACARBAZINE DACARBAZINE 22931300 33282 22725 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE CEDIRANIB CEDIRANIB 33283 22726 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME L-751250 33285 22727 ITIH3 3699 DRUGGABLE GENOME, PROTEASE INHIBITOR clozapine CLOZAPINE 27396837 33289 22728 ADCY1 107 DRUGGABLE GENOME, ENZYME Adenosine monophosphate 33290 22729 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SOTRASTAURIN SOTRASTAURIN 33291 22730 OGFR 11054 NA INNO-105 33294 22731 FES 2242 ENZYME, DRUGGABLE GENOME, KINASE, TYROSINE KINASE inhibitor 249565819 33297 22732 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR HGS-1029 33298 22733 PTGS1 5742 ENZYME, DRUGGABLE GENOME MESALAZINE MESALAMINE 33301 22734 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DAPSONE DAPSONE 22931300 33303 22735 ATAD5 79915 NA DNDI1417264 CHEMBL1467200 33304 22736 APCS 325 TRANSPORTER, DRUGGABLE GENOME inhibitor 249565936 MIRIDESAP 33305 22737 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Pioglitazone PIOGLITAZONE 33307 22738 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME WEDELOLACTONE WEDELOLACTONE 22926226 33309 22739 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-STYRYL-QUINOLINE CHEMBL127579 33311 22740 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER methotrexate METHOTREXATE 26086825,29743634,18256692,21317831 33313 22741 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 252166488 PALOVAROTENE 33314 22742 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SURAMIN HEXASODIUM SURAMIN HEXASODIUM 33315 22743 PSMA6 5687 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL325041 BORTEZOMIB 33316 22744 KDM4A 9682 DRUGGABLE GENOME, ENZYME 2,3,4-TRIHYDROXYBENZOPHENONE CHEMBL1527 33318 22745 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 252166749 33319 22746 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DAZOMET DAZOMET 33320 22747 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME ALISERTIB ALISERTIB 33324 22748 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Ridaforolimus RIDAFOROLIMUS 26725216 33325 22749 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME ACETYLSALICYLIC ACID 6108875 33326 22750 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MENADIONE MENADIONE 33327 22751 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CEFOXITIN SODIUM CEFOXITIN SODIUM 33328 22752 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-14 33329 22753 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GLUTAMIC ACID HYDROCHLORIDE GLUTAMIC ACID HYDROCHLORIDE 33330 22754 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor 249565784 LY-2874455 33331 22755 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME MESALAMINE MESALAMINE 33337 22756 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 33338 22757 SMN1 6606 DRUGGABLE GENOME SODIUM 4-PHENYLBUTYRATE 15523494 33340 22758 RAB9A 9367 ENZYME, DRUGGABLE GENOME DAIDZEIN DAIDZEIN 33341 22759 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 178103172 GISADENAFIL 33342 22760 MARCHF8 220972 ENZYME Grippol TC 33343 22761 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ADAPALENE ADAPALENE 33344 22762 PPCDC 60490 ENZYME docetaxel DOCETAXEL 33345 22763 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ESTRADIOL BENZOATE 11923430 33346 22764 MAPT 4137 DRUGGABLE GENOME NSC-663284 CHEMBL337173 33347 22765 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 7-HYDROXY ISOFLAVONE 7-HYDROXY ISOFLAVONE 33348 22766 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME TAK-715 TAK-715 33352 22767 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE Tricyclic compound 6 33353 22768 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME TRIBUTYRIN TRIBUTYRIN 16188956 33354 22769 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 223366154 33355 22770 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Glatiramer Acetate 33356 22771 MAOA 4128 DRUGGABLE GENOME, ENZYME PhyllanthoidA 33357 22772 PTK7 5754 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE PF-06647020 COFETUZUMAB PELIDOTIN 33358 22773 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE HTU-PA 33359 22774 MPHOSPH8 54737 NA CIS(Z)-FLUPENTIXOL DIHYDROCHLORIDE CHEMBL1496351 33360 22775 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE PD-98059 CHEMBL35482 11196459 33361 22776 EPHB4 2050 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL24828 VANDETANIB 33363 22777 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BIMATOPROST BIMATOPROST 33364 22778 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRIMETREXATE TRIMETREXATE 33365 22779 SMN2 6607 DRUGGABLE GENOME 4-BENZYLOXYANILINE 4-BENZYLOXYANILINE 33366 22780 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CRYPTOTANSHINONE CRYPTOTANSHINONE 33368 22781 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL1201752 IXABEPILONE 33370 22782 MAP2 4133 NA COLCHICINE COLCHICINE 7511033 33371 22783 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE AMINOCAPROIC ACID 33372 22784 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CEFTRIAXONE CEFTRIAXONE 22931300 33373 22785 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE boceprevir BOCEPREVIR 33376 22786 POLB 5423 DNA REPAIR, DRUGGABLE GENOME PROTOPORPHYRIN PROTOPORPHYRIN 33377 22787 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MMV666022 CHEMBL599100 33379 22788 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1201735 BUPROPION HYDROBROMIDE 33383 22789 BCHE 590 DRUGGABLE GENOME, ENZYME irinotecan IRINOTECAN 33384 22790 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 381118853 33385 22791 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID29757691-Compound-10 33386 22792 TUBB3 10381 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 33387 22793 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Isoindoline derivative 4 33389 22794 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-43 33390 22795 MGLL 11343 DRUGGABLE GENOME, ENZYME inhibitor 329968421 33392 22796 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Carbinoxamine CARBINOXAMINE 33393 22797 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME FEDRATINIB FEDRATINIB 18394554 33394 22798 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE REGN1400 33395 22799 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545244 ALLITINIB 33396 22800 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DARIFENACIN DARIFENACIN 33397 22801 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102815 33399 22802 SOST 50964 DRUGGABLE GENOME inhibitor CHEMBL2107874 ROMOSOZUMAB 33400 22803 GMNN 51053 DRUGGABLE GENOME MMV667491 CHEMBL1437888 33403 22804 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL2068724 ACAMPROSATE CALCIUM 33404 22805 DPP7 29952 PROTEASE, ENZYME, DRUGGABLE GENOME BDBM50382283 33406 22806 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3716 CHEMBL609606 33408 22807 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE XL999 33409 22808 MMP14 4323 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178103981 ILOMASTAT 33410 22809 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BAY 10-00394 33413 22810 CDKN3 1033 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, TUMOR SUPPRESSOR, ENZYME, KINASE inhibitor CHEMBL3544942 RONICICLIB 33414 22811 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEFIXIME CEFIXIME 33415 22812 SH2B1 25970 KINASE clozapine CLOZAPINE 28694205 33416 22813 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125495 CHEMBL532412 33417 22814 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 135651987 33418 22815 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200434 OXTRIPHYLLINE 33419 22816 NDUFB1 4707 ENZYME inhibitor CHEMBL3545135 NV-128 33421 22817 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 187051805 QUISINOSTAT 33422 22818 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200434 OXTRIPHYLLINE 33424 22819 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 363894211 PEXMETINIB 33425 22820 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR palbociclib PALBOCICLIB 33426 22821 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME PD-360324 PD-360324 33429 22822 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME XCT790 CHEMBL189753 33430 22823 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Proline amide derivative 1 33432 22824 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200578 THEOPHYLLINE SODIUM GLYCINATE 33433 22825 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 249565754 33436 22826 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME ANTHRACYCLINE 10641488 33440 22827 IL1B 3553 KINASE, DRUGGABLE GENOME TPN 8724378 33442 22828 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX STREPTONIGRIN STREPTONIGRIN 33444 22829 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PYROGALLOL PYROGALLOL 33446 22830 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DROMOSTANOLONE DROMOSTANOLONE 33449 22831 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PROGESTERONE PROGESTERONE 33450 22832 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE Cixutumumab CIXUTUMUMAB 33451 22833 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 7 33452 22834 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME FOLFOX 27002107 33455 22835 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CEDIRANIB CEDIRANIB 33457 22836 TUBB 203068 DRUGGABLE GENOME Oral paclitaxel 33458 22837 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PWT33597 33459 22838 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051824 33460 22839 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 4-(4-AMINOPHENYL)BUTANOIC ACID CHEMBL1650245 24044874 33463 22840 ERAP1 51752 PROTEASE, ENZYME, DRUGGABLE GENOME TCMDC-124673 CHEMBL587247 33464 22841 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME APAZONE APAZONE 33467 22842 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE EAI045 27251290 33468 22843 TUBB2B 347733 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 33469 22844 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME AZD-1775 ADAVOSERTIB 33470 22845 LAMB2 3913 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 33472 22846 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METIXENE METHIXENE 33474 22847 HIF1AN 55662 NA L-4-THIOPROLINE CHEMBL1800368 21665470 33475 22848 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE risperidone RISPERIDONE 33476 22849 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE vaccine PRINOMASTAT PRINOMASTAT 33477 22850 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING CEFDINIR CEFDINIR 33479 22851 GMNN 51053 DRUGGABLE GENOME TCMDC-123868 CHEMBL548615 33480 22852 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR HEPARIN HEPARIN 11150580 33482 22853 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MMV006937 CHEMBL580381 33483 22854 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME CINNAMTANNIN B1 CINNAMTANNIN B1 17602466 33484 22855 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME AZD-1080 AZD-1080 33485 22856 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-1919 CHEMBL576409 33486 22857 BAZ2B 29994 NA DNDI1417156 CHEMBL1504679 33488 22858 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME RG-1530 RG-1530 33490 22859 GDF15 9518 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR CALCITRIOL CALCITRIOL 15386353 33492 22860 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME A-443654 A-443654 24978597,24569089 33493 22861 ACSS2 55902 ENZYME, TRANSCRIPTION FACTOR paclitaxel PACLITAXEL 21636554 33494 22862 BAZ2B 29994 NA BITHIONOL BITHIONOL 33495 22863 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LAPATINIB LAPATINIB 33496 22864 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 310264698 AMG-319 33497 22865 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RS-17053 CHEMBL88272 33498 22866 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 867101 CHEMBL406557 33499 22867 KDM4A 9682 DRUGGABLE GENOME, ENZYME PROCHLORPERAZINE PROCHLORPERAZINE 33500 22868 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor NILOTINIB NILOTINIB 33501 22869 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2107725 ANATIBANT 33503 22870 MAGEA4 4103 NA CAR-T cells targeting MAGE-A4 33504 22871 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME MORPHINE MORPHINE 11937560 33505 22872 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE LJM716 ELGEMTUMAB 33506 22873 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING CINNARIZINE CINNARIZINE 16680159 33507 22874 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2105683 NAPROXEN ETEMESIL 33509 22875 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor CHEMBL598797 CUDC-101 33510 22876 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SJ000014858 CHEMBL591628 33511 22877 NDUFA9 4704 ENZYME inhibitor CHEMBL3545320 ME-344 33512 22878 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201174 SITAGLIPTIN PHOSPHATE 33513 22879 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CURCUMIN CURCUMIN 23145932 33514 22880 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor MOTESANIB MOTESANIB 33515 22881 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PI3KBETA INHIBITOR AZD8186 26725216 33518 22882 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 318164808 SIPONIMOD 33519 22883 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker 381118869 BENIDIPINE 33520 22884 RICTOR 253260 CLINICALLY ACTIONABLE inhibitor MLN0128 SAPANISERTIB 33521 22885 PGLYRP4 57115 DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 27670765 33522 22886 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Erlotinib ERLOTINIB 27659046,27924459,22448344 33523 22887 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 315661279 ACUMAPIMOD 33524 22888 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROPERICIAZINE PERICIAZINE 33525 22889 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BUSPIRONE BUSPIRONE 33526 22890 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLUORANTHENE FLUORANTHENE 33527 22891 ALOX15 246 ENZYME, DRUGGABLE GENOME MK-886 CHEMBL29097 33528 22892 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565815 33529 22893 ILK 3611 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME US8754233, (4-Benzothiazol-2-yl-1H-pyrazol-3-yl)-[2-(1H-imidazol-4-yl)-ethyl]-amine 33530 22894 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL3544932 TAK-901 33531 22895 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 178102606 CHEMBL104264 33532 22896 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1685 DEZOCINE 33533 22897 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CYC-116 CYC-116 33534 22898 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROPACHLOR PROPACHLOR 33535 22899 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE everolimus EVEROLIMUS 33538 22900 ALOX15 246 ENZYME, DRUGGABLE GENOME HEXACHLOROPHENE HEXACHLOROPHENE 33539 22901 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE SORAFENIB SORAFENIB 33541 22902 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor GSK2126458 OMIPALISIB 33542 22903 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649868 A-123189 33544 22904 PLCD3 113026 KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHOLIPASE diltiazem DILTIAZEM 22525200 33545 22905 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 4-METHOXYDALBERGIONE 4-METHOXYDALBERGIONE 33548 22906 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-N1 33549 22907 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CISAPRIDE CISAPRIDE 1555639,7952869,12519861,7557734,8321323 33553 22908 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MEXILETINE MEXILETINE 9806111 33554 22909 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 252166682 33555 22910 HSPA4 3308 NA ISOPROTERENOL ISOPROTERENOL 8047983 33557 22911 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651471 DEXAMETHASONE 33558 22912 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-17 33560 22913 ABCC9 10060 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER CHEMBL1200338 PINACIDIL 33563 22914 CD52 1043 DRUGGABLE GENOME ALEMTUZUMAB ALEMTUZUMAB 33564 22915 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor SORAFENIB SORAFENIB 33565 22916 HTT 3064 DRUGGABLE GENOME DNDI1417548 CHEMBL2094789 33566 22917 POLK 51426 DNA REPAIR, ENZYME GW7647 GW7647 33567 22918 TMEM97 27346 NA PMID30185082-Compound-64 33569 22919 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE LOXO-101 LAROTRECTINIB 28578312,26216294,27093299 33570 22920 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1201020 DISOPYRAMIDE PHOSPHATE 33571 22921 GLS 2744 ENZYME NSC-228155 CHEMBL505670 33572 22922 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX 1,7-O-DIACETYLGEOPYXIN A CHEMBL1873045 33576 22923 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIENESTROL DIENESTROL 33577 22924 CAPN1 823 PROTEASE, DRUGGABLE GENOME, ENZYME BORTEZOMIB BORTEZOMIB 20875739 33579 22925 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 187051772 CICLESONIDE 33582 22926 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHYLPREDNISOLONE METHYLPREDNISOLONE 33583 22927 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CLOFLUCARBAN CLOFLUCARBAN 33585 22928 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SB-415286 CHEMBL322970 33586 22929 GMNN 51053 DRUGGABLE GENOME SORAFENIB TOSYLATE SORAFENIB TOSYLATE 33587 22930 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 Drugs used in nicotine dependence 26132489 33589 22931 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-16 33591 22932 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LEMILDIPINE LEMILDIPINE 33593 22933 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME AG-1879 CHEMBL406845 33594 22934 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2011137219 35(1-11) 33595 22935 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PAROXETINE PAROXETINE 33596 22936 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL586701 ZSTK-474 33599 22937 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1922094 APITOLISIB 33601 22938 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR EPINEPHRINE BITARTRATE EPINEPHRINE BITARTRATE 33603 22939 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE SELUMETINIB SELUMETINIB 27922010 33605 22940 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1201580 ADALIMUMAB 33606 22941 ITPR2 3709 ION CHANNEL, DRUGGABLE GENOME activator 178101040 33607 22942 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PF-562271 PF-00562271 33608 22943 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178100242 ROFECOXIB 33609 22944 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE REBASTINIB REBASTINIB 26703895 33610 22945 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR NICOTINE NICOTINE 14555188 33611 22946 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ALEXIDINE DIHYDROCHLORIDE ALEXIDINE DIHYDROCHLORIDE 33612 22947 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME NSC-228155 CHEMBL505670 33613 22948 SLC29A2 3177 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE gemcitabine GEMCITABINE 25162786 33614 22949 BCHE 590 DRUGGABLE GENOME, ENZYME succinylcholine SUXAMETHONIUM 21637541,18075469,25054547,21029050,22053728,2915989,26398623,1415224,12724618,21228368,12881446,15731589 33616 22950 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE RAPAMYCIN SIROLIMUS 11245436 33617 22951 NDUFA12 55967 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 33618 22952 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR Cediranib CEDIRANIB 26802156 33619 22953 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR thalidomide THALIDOMIDE 21435719 33622 22954 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Depatuxizumab DEPATUXIZUMAB 33623 22955 POLK 51426 DNA REPAIR, ENZYME SULFURETIN SULFURETIN 33624 22956 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody OFATUMUMAB OFATUMUMAB 33625 22957 ALOX15B 247 DRUGGABLE GENOME, ENZYME MERCURIC CHLORIDE MERCURIC CHLORIDE 33626 22958 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BEXAROTENE BEXAROTENE 33628 22959 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR FISPEMIFENE FISPEMIFENE 33629 22960 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CHLORANIL CHLORANIL 33632 22961 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL1201748 CABAZITAXEL 33633 22962 POLI 11201 DNA REPAIR CRYPTOTANSHINONE CRYPTOTANSHINONE 33634 22963 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL FOSPROPOFOL FOSPROPOFOL 33635 22964 GMNN 51053 DRUGGABLE GENOME PIROCTONE PIROCTONE 33636 22965 MAPT 4137 DRUGGABLE GENOME EXEBRYL-1 33638 22966 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR 192C86 19624532 33639 22967 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL2096631 CLORAZEPATE DIPOTASSIUM 33640 22968 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 223365977 33641 22969 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE dextropropoxyphene PROPOXYPHENE 20133509 33642 22970 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HYPEROSIDE HYPEROSIDE 33645 22971 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ROBUSTIC ACID ROBUSTIC ACID 33646 22972 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000044417 CHEMBL609438 33647 22973 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TETRACYCLINE TETRACYCLINE 33648 22974 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME arsenic trioxide 33649 22975 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1228 OXYPHENBUTAZONE 33651 22976 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME inhibitor CHEMBL1200826 LITHIUM CARBONATE 33652 22977 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME GNF-PF-4227 CHEMBL585654 33653 22978 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE MK2206 MK-2206 24265152,25551293 33655 22979 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Prednisolone PREDNISOLONE 28151717 33656 22980 XDH 7498 DRUGGABLE GENOME, ENZYME INSULIN INSULIN 17370312 33659 22981 FCGRT 2217 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antibody 354702250 33662 22982 SERPINA6 866 DRUGGABLE GENOME, PROTEASE INHIBITOR TRIAMCINOLONE TRIAMCINOLONE 33664 22983 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENYL 2-PHENYLETHENESULFONATE CHEMBL443343 33666 22984 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545332 CEP-2563 33667 22985 KDM4A 9682 DRUGGABLE GENOME, ENZYME 0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE 0-HEXYL-1,3-DIAMINE-PLATINUM 2,2-DICHLORIDE 33668 22986 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE ACETYLDIGITOXIN ACETYLDIGITOXIN 33670 22987 TSPO 706 DRUGGABLE GENOME Lorazepam LORAZEPAM 33671 22988 FGA 2243 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, FIBRINOGEN inhibitor CHEMBL1201505 FIBRINOLYSIN, HUMAN 33672 22989 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AG-34 CHEMBL80155 33674 22990 TLR6 10333 DRUGGABLE GENOME MALP-2S 33675 22991 PRKAG1 5571 ENZYME, KINASE METFORMIN METFORMIN 26471090 33677 22992 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 33678 22993 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GDC-0084 RG-7666 27638506 33679 22994 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C17 33683 22995 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL971 PENTOBARBITAL SODIUM 33685 22996 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME EZOGABINE EZOGABINE 21296466 33686 22997 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE HYDROXYCHLOROQUINE HYDROXYCHLOROQUINE 11117548 33687 22998 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME modulator CHEMBL1628502 GABAPENTIN ENACARBIL 33688 22999 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 381118815 33694 23000 POLB 5423 DNA REPAIR, DRUGGABLE GENOME RUTIN RUTIN 33695 23001 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIFLOXACIN HYDROCHLORIDE DIFLOXACIN HYDROCHLORIDE 33696 23002 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 310264739 LIFIRAFENIB 33697 23003 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TRICHOSTATIN A 17267518 33698 23004 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ELLIPTECINE ELLIPTECINE 33700 23005 LPAR2 9170 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 135651487 33701 23006 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL2104967 FIRATEGRAST 33702 23007 NEK3 4752 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565802 33703 23008 ATXN2 6311 NA GNF-PF-4029 CHEMBL596633 33704 23009 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE OK-432 1375873 33705 23010 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 3-AMINOEVODIAMINE CHEMBL2171795 22867019 33706 23011 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PSEUDOEPHEDRINE PSEUDOEPHEDRINE 33708 23012 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CASEARINONE A CASEARINONE A 9322361 33709 23013 BAZ2B 29994 NA TRIFLUPROMAZINE HYDROCHLORIDE TRIFLUPROMAZINE HYDROCHLORIDE 33712 23014 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-5478 CHEMBL586982 33713 23015 PROM1 8842 CELL SURFACE, DRUGGABLE GENOME CAR-T cells targeting CD133 33714 23016 KDM4A 9682 DRUGGABLE GENOME, ENZYME GERONTOXANTHONE I GERONTOXANTHONE I 33715 23017 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE JQ-1 21889194 33716 23018 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BIPHENYL BIPHENYL 33719 23019 SLC47A1 55244 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER rucaparib RUCAPARIB 33720 23020 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178102078 SULINDAC 33721 23021 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE PIXY 7874002 33724 23022 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TROLEANDOMYCIN TROLEANDOMYCIN 22931300 33725 23023 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHLOROXINE CHLOROXINE 33726 23024 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PYROGALLOL PYROGALLOL 33727 23025 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME PENT-1-ENE CHEMBL295337 33729 23026 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE ABT-737 ABT 737 27974663 33730 23027 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33l 33732 23028 FAAH 2166 ENZYME, DRUGGABLE GENOME Benzoxazole derivative 1 33733 23029 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE agonist 178103125 33734 23030 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE ME-401 ME-401 33735 23031 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CAR-T cells targeting CD123 33736 23032 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MORIN MORIN 33737 23033 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL282686 TESAGLITAZAR 33738 23034 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist,antagonist 178100399 33739 23035 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE 111In-hEGF 33741 23036 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME SBC-014 19175929 33742 23037 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME VVP-808 METHAZOLAMIDE 33743 23038 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-16 33747 23039 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME DOVITINIB DOVITINIB 33749 23040 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE ARX201 33750 23041 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1201468 ESTROGENS, ESTERIFIED 33751 23042 NAAA 27163 ENZYME, DRUGGABLE GENOME CYCLOPENTYL PALMITATE CYCLOPENTYL PALMITATE 20022504 33752 23043 EML4 27436 CLINICALLY ACTIONABLE, KINASE X-396 ENSARTINIB 21613408 33753 23044 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565784 LY-2874455 33755 23045 KIF11 3832 DRUGGABLE GENOME 4SC-205 33756 23046 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IMATINIB IMATINIB 18094422 33758 23047 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME LESTAURTINIB LESTAURTINIB 33760 23048 BAZ2B 29994 NA CEFOTETAN CEFOTETAN 33761 23049 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Entrectinib ENTRECTINIB 28183697 33762 23050 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR SM-101 VALZIFLOCEPT 33763 23051 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ISRAPAFANT ISRAPAFANT 33768 23052 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME TD-0714 33770 23053 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 381118892 33772 23054 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL NAV 1.7 BLOCKER 33773 23055 KDM5C 8242 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE EVEROLIMUS EVEROLIMUS 27751729 33774 23056 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE YM-024 24718026 33777 23057 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1256958 EPINEPHRINE BITARTRATE 33779 23058 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PHA-767491 CHEMBL225519 33780 23059 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650897 33781 23060 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 14 33782 23061 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR boceprevir BOCEPREVIR 25836019 33784 23062 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GESTRINONE GESTRINONE 33785 23063 MBP 4155 CELL SURFACE NBI-5788 TIPLIMOTIDE 33786 23064 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR THIRAM THIRAM 33787 23065 CREB1 1385 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR NICOTINE NICOTINE 11331423 33789 23066 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CORTICOTROPIN CORTICOTROPIN 11360665 33790 23067 ATXN2 6311 NA THIOTHIXENE THIOTHIXENE 33793 23068 MT1H 4496 NA CISPLATIN CISPLATIN 10422815 33794 23069 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER METHOTREXATE METHOTREXATE 17363498 33800 23070 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME GO-6976 GO-6976 33801 23071 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-139257 CHEMBL1256364 33802 23072 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME CORTISOL HYDROCORTISONE 7592884 33804 23073 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE 4-PHENOXYPHENOL CHEMBL224318 18952425 33805 23074 TMEM97 27346 NA Piperazinyl norbenzomorphane compound 3 33807 23075 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE CHIR-265 RAF-265 33808 23076 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PKI-402 CHEMBL589258 20371716 33809 23077 CBR1 873 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME anthracyclines and related substances 22124095 33810 23078 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIHYDROTACHYSTEROL DIHYDROTACHYSTEROL 33811 23079 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LY411575 27556950 33812 23080 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565806 SILMITASERTIB 33813 23081 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 178102434 33815 23082 TH 7054 ENZYME, DRUGGABLE GENOME inhibitor 178101810 33822 23083 CXCL13 10563 DRUGGABLE GENOME rituximab RITUXIMAB 26384320 33826 23084 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor GSAO 33828 23085 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE DOVITINIB DOVITINIB 33829 23086 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL2023349 R428 33830 23087 CCL4 6351 DRUGGABLE GENOME CLODRONATE CLODRONIC ACID 12388372 33831 23088 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor COMETRIQ COMETRIQ 33833 23089 ALOX15B 247 DRUGGABLE GENOME, ENZYME PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 33834 23090 TPT1 7178 DRUGGABLE GENOME 5-FLUOROURACIL FLUOROURACIL 15262975 33836 23091 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE ANISOMYCIN ANISOMYCIN 33838 23092 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE BIBW 2992 33839 23093 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SURAMIN SURAMIN 33841 23094 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 329968437 BMS-986020 33842 23095 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE LOMIFYLLINE LOMIFYLLINE 33843 23096 ATXN2 6311 NA GW405833 CHEMBL73711 33844 23097 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PEG-CAMPTOTHECIN 33846 23098 CHST11 50515 ENZYME, DRUGGABLE GENOME CHONDROITIN SULFATE 16079159 33847 23099 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY PD 098059 10781369 33849 23100 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28117607-Compound-20 33850 23101 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME ISOSILYBIN A ISOSILYBIN A 23401473 33851 23102 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649899 33852 23103 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20100022547C87 33853 23104 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 223366040 33856 23105 TSPO 706 DRUGGABLE GENOME TRIAZOLAM TRIAZOLAM 33857 23106 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1200848 HYDROXYPROGESTERONE CAPROATE 33860 23107 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHENETHYLISOTHIOCYANATE PHENETHYLISOTHIOCYANATE 23371965 33861 23108 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 252166513 33862 23109 SH2B1 25970 KINASE mirtazapine MIRTAZAPINE 28694205 33864 23110 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE BI-831266 33865 23111 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR GUTHION GUTHION 33866 23112 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME MLN-8054 MLN-8054 33868 23113 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL223360 LINIFANIB 33869 23114 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME Salirasib SALIRASIB 33870 23115 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE glimepiride GLIMEPIRIDE 33873 23116 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor AS703569 CENISERTIB 33875 23117 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL1200810 DOXERCALCIFEROL 33876 23118 DPP7 29952 PROTEASE, ENZYME, DRUGGABLE GENOME US8470836, 8 33877 23119 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1980297 ILORASERTIB 33878 23120 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME SIROLIMUS SIROLIMUS 19848404,17563385,24893224,24836070 33879 23121 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BUPROFEZIN BUPROFEZIN 33881 23122 POLK 51426 DNA REPAIR, ENZYME AG-1288 CHEMBL166486 33882 23123 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME GCC-4401 33885 23124 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME DASATINIB DASATINIB 26619011,21483012,19010912,23833300,19238210,22310681,19537845,18186519,12068308,22649091,25157968,12460919,12460918,20350999,21129611 33886 23125 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME Baricitinib BARICITINIB 33888 23126 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PMID29671355-Compound-21 33890 23127 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-1644 CHEMBL600734 33891 23128 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure3-Aspeverin 33892 23129 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE SF1126 33893 23130 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE DHM25 26237138 33896 23131 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DIPYRIDAMOLE DIPYRIDAMOLE 33897 23132 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE nifedipine NIFEDIPINE 22875663 33898 23133 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME 7-azaindole derivative 5 33901 23134 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CGM097 CGM-097 33902 23135 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 4-BENZYLOXYANILINE 4-BENZYLOXYANILINE 33906 23136 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 135650039 33907 23137 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650207 DONITRIPTAN 33910 23138 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PAPAVERINE PAPAVERINE 33911 23139 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME perphenazine PERPHENAZINE 2743709 33913 23140 GMNN 51053 DRUGGABLE GENOME TCMDC-125738 CHEMBL527585 33914 23141 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GDC-0032 TASELISIB 33916 23142 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL1201752 IXABEPILONE 33917 23143 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545096 BGT-226 33918 23144 MAOA 4128 DRUGGABLE GENOME, ENZYME 5-PHENOXYPHTHALIMIDE CHEMBL1813518 21778064 33919 23145 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE ARA-C 15936818 33920 23146 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-5 33922 23147 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROSTAGLANDIN D2 PROSTAGLANDIN D2 23566516 33923 23148 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DICYCLOMINE DICYCLOMINE 33924 23149 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CILNIDIPINE CILNIDIPINE 33927 23150 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR AMINOQUINURIDE AMINOQUINURIDE 33928 23151 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3148 CHEMBL81782 33930 23152 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NECA NECA 33931 23153 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME METHOXYARACHIDONOYL FLUOROPHOSPHONATE METHOXYARACHIDONOYL FLUOROPHOSPHONATE 33932 23154 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME SNS-314 SNS-314 33933 23155 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME DACTOLISIB DACTOLISIB 23549875 33934 23156 MAPT 4137 DRUGGABLE GENOME NSC-402083 CHEMBL1546228 33935 23157 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DAUNORUBICIN DAUNORUBICIN 33936 23158 IL1B 3553 KINASE, DRUGGABLE GENOME ANTICONVULSANT 16358339 33937 23159 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 404859045 33939 23160 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102298 BMS-387032 33941 23161 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CENISERTIB CENISERTIB 33942 23162 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Indoline derivative 10 33943 23163 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING NSC-60340 CHEMBL1534034 33945 23164 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME IPRIFLAVONE IPRIFLAVONE 33948 23165 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE Idelalisib IDELALISIB 33949 23166 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE DOXIFLURIDINE DOXIFLURIDINE 2972339 33950 23167 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 33951 23168 TUBA1C 84790 DRUGGABLE GENOME ABT-751 ABT-751 25468039 33952 23169 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-228155 CHEMBL505670 33953 23170 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 310264696 AZD-8835 33954 23171 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AV-412 MP-412 33955 23172 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 318164847 TAK-715 33958 23173 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SP-600125 SP-600125 33959 23174 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor PANOBINOSTAT PANOBINOSTAT 33960 23175 HBB 3043 DRUGGABLE GENOME, ENZYME Crizanlizumab-tmca 33961 23176 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ATRASENTAN ATRASENTAN 33962 23177 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SAPONIN 9342944 33963 23178 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE erythromycin ethylsuccinate / sulfisoxazole acetyl 33964 23179 HTT 3064 DRUGGABLE GENOME KETOROLAC TROMETHAMINE KETOROLAC TROMETHAMINE 33965 23180 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR DIFENOCONAZOLE DIFENOCONAZOLE 33969 23181 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor DOVITINIB DOVITINIB 33970 23182 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DIHYDREXIDINE DIHYDREXIDINE 33971 23183 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ANTIMYCIN A ANTIMYCIN A 33972 23184 UGT2B7 7364 DRUGGABLE GENOME lovastatin LOVASTATIN 33975 23185 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME 5-FLUOROURACIL FLUOROURACIL 15641988 33979 23186 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME oxymorphone OXYMORPHONE 33980 23187 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE AZD-1080 AZD-1080 33983 23188 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1944698 ZOTIRACICLIB 33984 23189 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 15746054,15228172,8242617,15919850 33986 23190 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor 135651454 33987 23191 NGFR 4804 CELL SURFACE, DRUGGABLE GENOME 178101723 33988 23192 RORB 6096 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, KINASE antagonist 135649927 33989 23193 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565751 33991 23194 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR RHEIN RHEIN 33992 23195 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SALINE SODIUM CHLORIDE 17187818 33994 23196 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-28 33995 23197 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYPROTERONE ACETATE CYPROTERONE ACETATE 33996 23198 POLK 51426 DNA REPAIR, ENZYME ESCULETIN ESCULETIN 33997 23199 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 310264675 CUDC-101 33998 23200 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MOSAPRAMINE MOSAPRAMINE 33999 23201 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DIETHYLSTILBESTROL DIETHYLSTILBESTROL 16598927 34000 23202 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TAE-684 TAE-684 34001 23203 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME LITHOCHOLIC ACID LITHOCHOLIC ACID 34002 23204 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZINC 03877300 CHEMBL1738937 22047606 34003 23205 PDE5A 8654 ENZYME, DRUGGABLE GENOME UDENAFIL UDENAFIL 34004 23206 ALOX15 246 ENZYME, DRUGGABLE GENOME MMV007363 CHEMBL601528 34005 23207 DHFR 1719 DRUGGABLE GENOME, ENZYME CH-1504 34006 23208 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TAMOXIFEN TAMOXIFEN 34009 23209 NPC1L1 29881 DRUGGABLE GENOME, TRANSPORTER EMZETIBE 34011 23210 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER PROTEASE INHIBITORS 16078135 34013 23211 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME 3-HYDROXY-3',4'-DIMETHOXYFLAVONE 3-HYDROXY-3',4'-DIMETHOXYFLAVONE 34015 23212 PTGS2 5743 DRUGGABLE GENOME, ENZYME etodolac ETODOLAC 19602986 34018 23213 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200613 TOLMETIN SODIUM 34019 23214 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL592445 GEDATOLISIB 34020 23215 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody U3-1287 AMG-888 34021 23216 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor CHEMBL445813 AT-7519 34023 23217 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL526 PROPOFOL 34024 23218 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME RO5045337 RO-5045337 34025 23219 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-48300 CHEMBL1091971 34026 23220 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR TEMOZOLOMIDE TEMOZOLOMIDE 12610499,16100942 34029 23221 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR 7-azaindole derivative 1 34030 23222 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ANTHRANILIC ACID ANTHRANILIC ACID 34031 23223 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL2219422 AFURESERTIB 34035 23224 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IMETIT IMETIT 34037 23225 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FENRETINIDE FENRETINIDE 10328240 34038 23226 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME INM-176 34040 23227 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2,4-DINITROPHENOL 2,4-DINITROPHENOL 34041 23228 CCL11 6356 DRUGGABLE GENOME inhibitor CHEMBL2109103 BERTILIMUMAB 34042 23229 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME inhibitor BORTEZOMIB BORTEZOMIB 34043 23230 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR eribulin ERIBULIN 34044 23231 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Imidazo cyclohexylamine derivative 1 34046 23232 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ASPIRIN ASPIRIN 12941295 34047 23233 FBXL17 64839 TUMOR SUPPRESSOR hydrochlorothiazide HYDROCHLOROTHIAZIDE 34051 23234 SLC47A1 55244 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER 178101296 34052 23235 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000114741 CHEMBL591370 34053 23236 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor SORAFENIB SORAFENIB 34055 23237 UCP2 7351 TRANSPORTER, DRUGGABLE GENOME TRIIODOTHYRONINE LIOTHYRONINE SODIUM 9428737,10444435 34058 23238 MAPT 4137 DRUGGABLE GENOME AG-494 CHEMBL56731 34059 23239 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME activator 135650729 34061 23240 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME R-1663 34062 23241 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Dihydropyrido phthalazinone derivative 2 34063 23242 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW852849X GW852849X 34065 23243 CRBN 51185 ENZYME, DRUG RESISTANCE 387065615 34067 23244 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME ZONISAMIDE ZONISAMIDE 34068 23245 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR US10022354, Example 5 34069 23246 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE niraparib NIRAPARIB 34070 23247 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE atorvastatin ATORVASTATIN 22186618,29178257 34071 23248 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME BRYOSTATIN BRYOSTATIN 34073 23249 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE 17 BETA-ESTRADIOL 11133691 34074 23250 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME SANGUINARIUM SANGUINARIUM 34075 23251 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PODOFILOX PODOFILOX 34076 23252 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ORBIFLOXACIN ORBIFLOXACIN 34077 23253 PDE7B 27115 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL932 DIPYRIDAMOLE 34079 23254 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL30219 METHOHEXITAL SODIUM 34080 23255 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SP-600125 SP-600125 34081 23256 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE RG-1530 RG-1530 34083 23257 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DNL151 34085 23258 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 187051798 BELINOSTAT 34087 23259 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL blocker 178101108 PROCAINE 34088 23260 MVD 4597 DRUGGABLE GENOME, ENZYME inhibitor 135650812 34090 23261 P4HB 5034 THIOREDOXIN, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE SYROSINGOPINE SYROSINGOPINE 34091 23262 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 34092 23263 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Quinoline and quinazoline derivative 8 34093 23264 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE OXYMORPHONE OXYMORPHONE 34094 23265 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME JNK-401 34095 23266 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Letrozole LETROZOLE 34096 23267 CA12 771 DRUGGABLE GENOME PARABEN PARABEN 34098 23268 POLI 11201 DNA REPAIR LEVODOPA LEVODOPA 34099 23269 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Vistusertib VISTUSERTIB 27974663 34101 23270 ACVR1B 91 SERINE THREONINE KINASE, CELL SURFACE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE US10030004, Compound 19 34103 23271 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-6 34104 23272 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-228155 CHEMBL505670 34105 23273 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR N'-(2-HYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE SALINAZID 34106 23274 TUBB4B 10383 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 34109 23275 GNA11 2767 CLINICALLY ACTIONABLE CABOZANTINIB CABOZANTINIB 28103611 34111 23276 SLAMF7 57823 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME antibody ELOTUZUMAB ELOTUZUMAB 34112 23277 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Nitrofurantoin NITROFURANTOIN 34113 23278 PRLR 5618 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, KINASE LFA-102 34114 23279 CBL 867 KINASE, ENZYME, CLINICALLY ACTIONABLE IL-2 ALDESLEUKIN 9461587 34115 23280 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL1213490 ROMIDEPSIN 34116 23281 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME rucaparib RUCAPARIB 34117 23282 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SP-600125 SP-600125 34118 23283 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME NORTRIPTYLINE NORTRIPTYLINE 34119 23284 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE MOTESANIB MOTESANIB 34121 23285 IL23R 149233 KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE Anti-IL-23 34122 23286 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME LUTEOLIN LUTEOLIN 25190466 34123 23287 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE JNJ-17305600 34124 23288 ATXN2 6311 NA QUINESTROL QUINESTROL 34127 23289 VKORC1 79001 DRUGGABLE GENOME, ENZYME Dicumarol DICUMAROL 34128 23290 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-402538 CHEMBL121556 34129 23291 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AG-120 IVOSIDENIB 34130 23292 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Desipramine DESIPRAMINE 34131 23293 VKORC1 79001 DRUGGABLE GENOME, ENZYME Acenocoumarol ACENOCOUMAROL 34132 23294 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME CONGO RED CONGO RED 34133 23295 TGFBR2 7048 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME inhibitor 249565755 34134 23296 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ERLOTINIB ERLOTINIB 34135 23297 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME EZN-3042 34137 23298 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME GAMBOGIC AMIDE GAMBOGIC AMIDE 17911251 34141 23299 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR FLUTICASONE PROPIONATE 10433509 34143 23300 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR ILORASERTIB ILORASERTIB 34144 23301 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135651956 34145 23302 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE LYS-6KAKT1 34146 23303 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650691 NARATRIPTAN 34148 23304 PTGS2 5743 DRUGGABLE GENOME, ENZYME MECLOFENAMIC ACID 34151 23305 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME UC-773587 25825487 34152 23306 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AMA-76 34153 23307 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE IL-6 8858917 34155 23308 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME ALVOCIDIB ALVOCIDIB 34159 23309 RAB9A 9367 ENZYME, DRUGGABLE GENOME TCMDC-125785 CHEMBL588525 34161 23310 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEPHARANTHINE CEPHARANTHINE 34164 23311 KAT2B 8850 ENZYME, DRUGGABLE GENOME inhibitor 178103614 34165 23312 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SORAFENIB SORAFENIB 34166 23313 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME sorafenib SORAFENIB 28362716 34169 23314 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135651026 34171 23315 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME INDOLE-3-CARBINOL INDOLE-3-CARBINOL 34172 23316 KDM4A 9682 DRUGGABLE GENOME, ENZYME 1-BENZYLMALEIMIDE CHEMBL388979 34173 23317 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Romidepsin ROMIDEPSIN 27443263 34174 23318 PTGS2 5743 DRUGGABLE GENOME, ENZYME rofecoxib ROFECOXIB 16678543,19602986 34176 23319 EGLN3 112399 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3544988 DAPRODUSTAT 34177 23320 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR 5,7,3',5'-TETRAHYDROXYFLAVANONE CHEMBL307893 34178 23321 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEFOTIAM HYDROCHLORIDE CEFOTIAM HYDROCHLORIDE 34181 23322 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL1944698 ZOTIRACICLIB 34182 23323 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650071 34184 23324 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL538943 VINORELBINE TARTRATE 34185 23325 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE AZD-1775 ADAVOSERTIB 34188 23326 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Everolimus EVEROLIMUS 34190 23327 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IOPANOIC ACID IOPANOIC ACID 34191 23328 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME AZD-3839 AZD-3839 34192 23329 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TCMDC-125784 CHEMBL581574 34193 23330 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 374883861 MK-8353 34194 23331 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 34195 23332 MPHOSPH8 54737 NA NICARDIPINE HYDROCHLORIDE NICARDIPINE HYDROCHLORIDE 34196 23333 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL1079175 MK-2206 34197 23334 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE HYDROMORPHONE HYDROMORPHONE 34199 23335 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Bipyridine derivative 1 34200 23336 COMT 1312 DRUGGABLE GENOME, ENZYME inhibitor 178103259 TOLCAPONE 34203 23337 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE PLX9486 34204 23338 MAPT 4137 DRUGGABLE GENOME NSC-9037 CHEMBL1451216 34208 23339 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE imatinib IMATINIB 34209 23340 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR SP-600125 SP-600125 34211 23341 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SUNITINIB SUNITINIB 34213 23342 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 2-(4-METHOXYPHENYL)BENZO[D]THIAZOLE CHEMBL460508 34214 23343 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE PROTON PUMP INHIBITOR 16925334 34216 23344 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHYLDOPA METHYLDOPA 22931300 34217 23345 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ALBUTEROL ALBUTEROL 2903243,16680159 34218 23346 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DOV 21947 34219 23347 ALOX15 246 ENZYME, DRUGGABLE GENOME TYRPHOSTIN 25 TYRPHOSTIN 25 34220 23348 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-31 34222 23349 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME activator 135650001 FLINDOKALNER 34223 23350 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CARFILZOMIB CARFILZOMIB 34224 23351 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SAR-125844 SAR-125844 34225 23352 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE PONATINIB PONATINIB 34227 23353 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE OSI-906 LINSITINIB 34229 23354 PDE7A 5150 ENZYME, DRUGGABLE GENOME inhibitor 178101846 34230 23355 CCR6 1235 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR agonist 135651668 34233 23356 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME CYPRODINIL CYPRODINIL 34235 23357 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR NSAID 12654560 34236 23358 NDUFV2 4729 ENZYME inhibitor CHEMBL3545135 NV-128 34237 23359 IDO2 169355 ENZYME inhibitor 381118836 34238 23360 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALPHA,BETA-DEHYDROCURVULARIN CHEMBL482050 34239 23361 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME sevoflurane SEVOFLURANE 25989378,12411786,26951757,8828983,19919814,17710899,7829078,9334205,21965348,11063719,10823104,20681998,25611019,19648156,25256590,12220451,11668625,23736090,14500992,9066328,14641996,18945287,25960145,7889656,11575529,18212565,16284304,8602662,18306019,28326467,11928716,18502356,10352931,12151923,11525881,17122579,16917943,8220422,10700782,16163667,17226826,9389851,16732128,16835904,11448278,29101530,9450902,7547049,23628358,9543323,24361844,26994242,12208234,15448513,16621918,21455645,11553045,12124989,19020143,19191329,27918309,8220423,12059893,10612851,16732084,10793526,27382027,15108991,12709367,12123492,26381711,25268394,28063098,11493496,12434264,12411788,19685112,25735680,8902717,29608462,27663056,7751854,8012359,9520251,15731587,15210166,1510267,10888602,22030266,25466363,17483490,28403410,12237752,1774074,17081152,18564801,10484775,21282829,16244001,7586638,19191333,25086907,7633940,17667581,12883402,19346234,1354642,22415532 34242 23362 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TEMEFOS TEMEFOS 34244 23363 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PROCHLORPERAZINE PROCHLORPERAZINE 22931300 34245 23364 IL1RN 3557 DRUGGABLE GENOME haloperidol HALOPERIDOL 27023437 34246 23365 PRMT5 10419 ENZYME, METHYL TRANSFERASE inhibitor 252166499 34247 23366 TNIK 23043 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 34249 23367 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9216972, 94 34250 23368 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE RESERPINE RESERPINE 2866100 34251 23369 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE latonduine a 27193581 34254 23370 TUBA3D 113457 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 34255 23371 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME blocker 135652738 34260 23372 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR THIOSEMICARBAZIDE THIOSEMICARBAZIDE 34262 23373 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102292 CEDIRANIB 34263 23374 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652473 PASIREOTIDE 34265 23375 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 329968438 34266 23376 KMO 8564 DRUGGABLE GENOME, ENZYME Benzene sulfonamide derivative 5 34268 23377 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL491473 CEDIRANIB 34270 23378 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME GW-2580 24186003 34271 23379 IFNGR2 3460 CLINICALLY ACTIONABLE, DRUGGABLE GENOME IFN-GAMMA INTERFERON GAMMA-1B 34276 23380 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-4337 CHEMBL277148 34277 23381 ALDH1A1 216 DRUGGABLE GENOME, ENZYME E-DOXEPIN E-DOXEPIN 34278 23382 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TCMDC-124059 CHEMBL530733 34279 23383 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DNDI1417467 CHEMBL1997335 34281 23384 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SORAFENIB SORAFENIB 19001320,18794803,28002790 34282 23385 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NOREPINEPHRINE NOREPINEPHRINE 2903243 34283 23386 GSTM1 2944 DRUGGABLE GENOME, ENZYME DOCETAXEL DOCETAXEL 16765145 34286 23387 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME EP-217609 34287 23388 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Formoterol FORMOTEROL 34288 23389 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE BMS-986202 34289 23390 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME GNF-PF-2893 CHEMBL312032 34291 23391 AREG 374 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE irinotecan IRINOTECAN 23959273 34292 23392 TMEM97 27346 NA Piperidine derivative 5 34293 23393 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652602 34296 23394 HUS1 3364 DNA REPAIR, KINASE CAMPTOTHECIN CAMPTOTHECIN 14762204 34297 23395 SLC47A2 146802 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME metformin METFORMIN 23417334,23267855,28834135,21956618,23652408,25939711,24624919,22722338 34298 23396 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2108566 NERELIMOMAB 34299 23397 CSK 1445 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE hydrochlorothiazide HYDROCHLOROTHIAZIDE 31327267 34300 23398 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Paclitaxel PACLITAXEL 26469692,24170767,26245675,21216929 34301 23399 NTS 4922 DRUGGABLE GENOME LITHIUM LITHIUM 7992199 34302 23400 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER TETRABENAZINE TETRABENAZINE 34303 23401 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE 681640 CHEMBL379975 34304 23402 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME inhibitor 178100439 GEMFIBROZIL 34305 23403 PPIA 5478 DRUGGABLE GENOME, ENZYME L-Proline PROLINE 34306 23404 HMMR 3161 KINASE, CELL SURFACE, DRUGGABLE GENOME HYALURONAN HYALURONAN 34307 23405 ATXN2 6311 NA CHLORHEXIDINE CHLORHEXIDINE 34308 23406 BRCA2 675 CLINICALLY ACTIONABLE Olaparib OLAPARIB 34310 23407 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TCMDC-124536 CHEMBL580851 34311 23408 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 34312 23409 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE RESVERATROL RESVERATROL 23799643 34317 23410 APC 324 CLINICALLY ACTIONABLE JW74 21199802 34318 23411 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME PROTOPORPHYRIN PROTOPORPHYRIN 34320 23412 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME RG7221 34321 23413 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING HTS-05057 CHEMBL372629 34322 23414 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE meloxicam MELOXICAM 18695978 34323 23415 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME GNF-2 CHEMBL483847 16415863 34324 23416 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PHENOLPHTHALEIN PHENOLPHTHALEIN 34326 23417 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PUROMYCIN HYDROCHLORIDE PUROMYCIN HYDROCHLORIDE 34327 23418 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Paclitaxel PACLITAXEL 24886365,26469692,27078022,24868024,27556950,26432108 34328 23419 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-718429A GSK-718429A 34329 23420 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL2180604 TAK-593 34330 23421 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1200946 NANDROLONE DECANOATE 34333 23422 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR thioguanine THIOGUANINE 24141364 34334 23423 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 EMODIN EMODIN 34335 23424 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Danazol DANAZOL 34336 23425 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 34337 23426 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME IDARUBICIN IDARUBICIN 34343 23427 GMNN 51053 DRUGGABLE GENOME (E)-DIBENZYLIDENEACETONE CHEMBL17201 34344 23428 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 223365885 DOTHIEPIN 34345 23429 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 310264699 SAMOTOLISIB 34346 23430 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER clomipramine CLOMIPRAMINE 21449676 34348 23431 ATAD5 79915 NA NSC-102042 CHEMBL273103 34349 23432 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL1090479 GSK-1070916 34350 23433 FFAR4 338557 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102222 34351 23434 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649972 ATORVASTATIN 34352 23435 ATAD5 79915 NA DNDI1417368 CHEMBL2094652 34353 23436 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MIM-D3 TAVILERMIDE 34354 23437 BAZ2B 29994 NA GNF-PF-4945 CHEMBL585628 34356 23438 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TRASTUZUMAB TRASTUZUMAB 15655555 34357 23439 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL 4-HYDROXYNON-2-ENAL 4-HYDROXYNON-2-ENAL 17684094 34358 23440 BCL6 604 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE inhibitor 348353631 34359 23441 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL445813 AT-7519 34360 23442 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-5134 CHEMBL602969 34361 23443 CBX1 10951 NA 2-HYDROXYPHENAZINE 5,10-DIOXIDE CHEMBL179611 34363 23444 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR THIRAM THIRAM 34364 23445 ATP5F1D 513 TRANSPORTER METHOXYFLURANE METHOXYFLURANE 34366 23446 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PD-0166285 PD-0166285 34368 23447 PEMT 10400 ENZYME CHEMBL1742998 CANTUZUMAB RAVTANSINE 34370 23448 KCNS3 3790 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107762 NERISPIRDINE 34371 23449 GJB4 127534 ION CHANNEL inhibitor 178101095 OCTANOL 34375 23450 TUBA3D 113457 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 34376 23451 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 223365899 METHYLNALTREXONE 34377 23452 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 135651751 GALANIN 34378 23453 CP 1356 DRUGGABLE GENOME, ENZYME PROGESTERONE PROGESTERONE 8619904 34380 23454 TUBB4B 10383 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 34381 23455 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE GSK-269962A GSK-269962A 34382 23456 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR NORGESTIMATE NORGESTIMATE 34383 23457 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 34384 23458 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE D3263 34385 23459 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX RETINOIC ACID 11602619 34387 23460 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BUCLIZINE BUCLIZINE 34388 23461 FFAR4 338557 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102224 34389 23462 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200732 AMCINONIDE 34391 23463 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor BAY80-6946 COPANLISIB 34392 23464 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AG-538 CHEMBL56393 34393 23465 MAP3K10 4294 SERINE THREONINE KINASE, ENZYME, KINASE, DRUGGABLE GENOME inhibitor 249565786 34396 23466 MSH2 4436 CLINICALLY ACTIONABLE, DNA REPAIR ANTI-PD-1 MONOCLONAL ANTIBODY MEDI0680 26674132 34397 23467 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 336446949 34398 23468 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 381744891 TROLEANDOMYCIN 34399 23469 FAAH 2166 ENZYME, DRUGGABLE GENOME Tetrazolyl urea derivative 1 34402 23470 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1201103 METHOXAMINE HYDROCHLORIDE 34403 23471 CD14 929 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor CHEMBL2109330 IC14 34404 23472 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Chlamydocin CHLAMYDOCIN 34405 23473 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HER2-specific T cells 34406 23474 CYP7A1 1581 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME cholic acid 34407 23475 TF 7018 CELL SURFACE, DRUGGABLE GENOME Ademetionine ADEMETIONINE 34408 23476 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 178102336 BOSUTINIB 34412 23477 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW695874X GW695874X 34414 23478 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-12 34415 23479 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Ivosidenib IVOSIDENIB 34417 23480 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100683 34418 23481 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TAMOXIFEN CITRATE TAMOXIFEN CITRATE 34419 23482 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Gemcitabine GEMCITABINE 26540314,27167172,26156229,26091808,27975152,26228206 34423 23483 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME OSI-632 OSI-632 34424 23484 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DNDI1417155 CHEMBL1548739 34426 23485 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator CHEMBL1201460 DALTEPARIN SODIUM 34427 23486 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYPRODINIL CYPRODINIL 34428 23487 NECTIN4 81607 DRUGGABLE GENOME ENFORTUMAB VEDOTIN 27013195 34429 23488 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DISULFIRAM DISULFIRAM 34431 23489 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Thiazides, plain 19247266 34432 23490 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32m 34433 23491 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GIVINOSTAT GIVINOSTAT 34434 23492 CLOCK 9575 ENZYME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX salbutamol ALBUTEROL 23508266 34435 23493 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE INS117548 34436 23494 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SU-6656 CHEMBL605003 34437 23495 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME activator 178104015 34438 23496 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650199 DOBUTAMINE 34439 23497 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME MENADIONE MENADIONE 34441 23498 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ANDROGENS 10468769 34442 23499 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME NSAIDS 2571317 34444 23500 HEBP1 50865 DRUGGABLE GENOME 1-phenyl-1,3,4-triazole derivative 3 34446 23501 SLC28A1 9154 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE THYMIDINE THYMIDINE 10353719 34447 23502 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME ETOMIDATE ETOMIDATE 16884293 34448 23503 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR CHF 4227 34449 23504 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME HELENALIN HELENALIN 34450 23505 DGAT2 84649 ENZYME PMID25470667-Compound-Figure4-1A 34451 23506 BAZ2B 29994 NA 5-CHLORO-[1,10]PHENANTHROLINE CHEMBL317115 34452 23507 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX RETINOID 10319995 34453 23508 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HYCANTHONE HYCANTHONE 22931300 34455 23509 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TAK-715 TAK-715 34456 23510 CPT2 1376 DRUGGABLE GENOME PROPIONYL-L-CARNITINE 34460 23511 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Pyrrolo-pyrrolone derivative 5 34461 23512 SLC15A2 6565 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101226 34462 23513 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor BAY80-6946 COPANLISIB 34463 23514 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 310264695 CC-223 34465 23515 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY CALCITRIOL CALCITRIOL 15319350 34466 23516 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CHRYSENE-1,4-DIONE CHEMBL421215 34467 23517 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL6 INDOMETHACIN 34469 23518 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE TAMOXIFEN TAMOXIFEN 15750629 34470 23519 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SAR125844 SAR-125844 25504634 34471 23520 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME Selective serotonin reuptake inhibitors 22776887 34473 23521 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 348353661 34474 23522 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE TOPOTECAN HYDROCHLORIDE TOPOTECAN HYDROCHLORIDE 34478 23523 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 178102481 34479 23524 DSE 29940 ENZYME abiraterone ABIRATERONE 34481 23525 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 178102556 AZD-1480 34484 23526 GALT 2592 ENZYME HyperAcute vaccine 34485 23527 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR ERISMODEGIB SONIDEGIB 34486 23528 ATP2A2 488 ENZYME, DRUGGABLE GENOME, TRANSPORTER celecoxib CELECOXIB 22336956 34487 23529 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 caffeine CAFFEINE 11394901,16402128,15940289,16952495,19238117,18698229,16891249,10544257,15660270,20860463,11241319,15475735,18212800,15592323,20089352,11725533,19921195,15980104,11237731,19845430,10999944,20155256,16272956,17130279,12042667,15900015,21494765,10448083,20596643,12223434,12844137,19604090,15265511,11197315,15308589,21521021,16452582,19225447,11779172,17267622,12749606,18380793,14981342,17220563,17112802 34488 23530 ELK1 2002 TRANSCRIPTION FACTOR DHPG 12220559 34489 23531 UNC13D 201294 NA emapalumab EMAPALUMAB 34491 23532 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-11c 34492 23533 BST1 683 DRUGGABLE GENOME Beta blocking agents, selective 34493 23534 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE LY2801653 34494 23535 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor PX-866 SONOLISIB 34495 23536 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLUOXASTROBIN FLUOXASTROBIN 34497 23537 ITGA2 3673 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE aspirin ASPIRIN 17157856,16493486,15205592,22940005,16214444 34498 23538 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE CHLORDANE CHLORDANE 34500 23539 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE mirtazapine MIRTAZAPINE 18695978 34501 23540 ITGB6 3694 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist CHEMBL1743032 INTETUMUMAB 34508 23541 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SNS-314 SNS-314 34511 23542 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL574737 UCN-01 34512 23543 SMN1 6606 DRUGGABLE GENOME 2-(PHENOXYMETHYL)BENZOTHIAZOLE 2-(PHENOXYMETHYL)BENZOTHIAZOLE 34513 23544 NOS2 4843 DRUGGABLE GENOME, ENZYME KD-7040 34514 23545 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ASTERRIC ACID ASTERRIC ACID 34515 23546 TARDBP 23435 TUMOR SUPPRESSOR SJ000117447 CHEMBL592611 34516 23547 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER nevirapine NEVIRAPINE 20017669,16912957,16912956 34517 23548 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL ZONISAMIDE ZONISAMIDE 34518 23549 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE antibody 318164853 TIGATUZUMAB 34521 23550 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Prasugrel PRASUGREL 34522 23551 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor AXITINIB AXITINIB 34524 23552 HMGCR 3156 ENZYME, DRUGGABLE GENOME PITAVASTATIN PITAVASTATIN 34525 23553 PRSS2 5645 DRUGGABLE GENOME, PROTEASE, ENZYME CYANOPEPTOLIN SS CYANOPEPTOLIN SS 34526 23554 PSCA 8000 DRUGGABLE GENOME CAR-T Cells targeting PSCA 34528 23555 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrazolopyridine derivative 6 34530 23556 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING ROMIDEPSIN ROMIDEPSIN 34531 23557 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE AZD5363 CAPIVASERTIB 34532 23558 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DAUNORUBICIN DAUNORUBICIN 34533 23559 TNKS2 80351 DRUGGABLE GENOME, ENZYME inhibitor 404859123 34534 23560 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME LATREPIRDINE LATREPIRDINE 34535 23561 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NALBUPHINE NALBUPHINE 34537 23562 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178101837 BATIMASTAT 34538 23563 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135650296 GALLAMINE 34539 23564 IL18 3606 DRUGGABLE GENOME THYROXINE THYROXINE 16061828 34540 23565 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ACRIDIN-1-YLAMINE CHEMBL146525 34541 23566 ATXN2 6311 NA TETRABROMOBENZOTRIAZOLE TETRABROMOBENZOTRIAZOLE 34542 23567 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIS(4-ISOPROPYLPHENYL) PHOSPHATE CHEMBL458602 34545 23568 SLC7A5 8140 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME melphalan MELPHALAN 34547 23569 QRFPR 84109 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651878 34550 23570 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 34551 23571 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR TOREMIFENE TOREMIFENE 34552 23572 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR antagonist 135650353 34553 23573 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HALOPERIDOL HALOPERIDOL 34554 23574 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Navitoclax NAVITOCLAX 25665005,26725216 34556 23575 ATXN2 6311 NA DOCEBENONE DOCEBENONE 34558 23576 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE AVB-S6-500 34559 23577 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE R-salbutamol sulphate 34560 23578 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR VUF-10497 CHEMBL452847 19053770 34561 23579 POLK 51426 DNA REPAIR, ENZYME DIOSMIN DIOSMIN 34562 23580 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650757 OLMESARTAN 34563 23581 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE amiodarone AMIODARONE 18695978 34564 23582 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DE-110 34565 23583 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 310264778 34566 23584 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650476 CHEMBL306645 34568 23585 MGLL 11343 DRUGGABLE GENOME, ENZYME inhibitor 329968422 34569 23586 PSMD8 5714 NA BORTEZOMIB BORTEZOMIB 24524217 34570 23587 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650405 IODOPHENPROPIT 34571 23588 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PEMBROLIZUMAB PEMBROLIZUMAB 26918451,26086854,27718847,28472902,25891174 34572 23589 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Temsirolimus TEMSIROLIMUS 24323026 34574 23590 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE FS118 34575 23591 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME PH-797804 PH-797804 34576 23592 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE 178101574 34577 23593 SMN1 6606 DRUGGABLE GENOME RG7800 25147906 34578 23594 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-640583 CHEMBL1287895 21074425 34582 23595 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIPHENYLSTANNANOL TRIPHENYLSTANNANOL 34584 23596 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CLENBUTEROL CLENBUTEROL 34585 23597 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL17 DICHLORPHENAMIDE 34586 23598 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heteroaryl-carboxamide derivative 8 34588 23599 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PIMOZIDE PIMOZIDE 34589 23600 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE 178101725 34590 23601 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor AZD4547 34591 23602 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Trifluridine TRIFLURIDINE 25700705 34592 23603 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor AZD 2281 34593 23604 HTT 3064 DRUGGABLE GENOME Oxazolyl methylthiothiazole derivative 1 34594 23605 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 34595 23606 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CINTREDEKIN BESUDOTOX 34596 23607 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GLUCOCORTICOID 17072757 34597 23608 UGT2B10 7365 DRUGGABLE GENOME cotinine COTININE 34601 23609 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TCMDC-125758 CHEMBL546797 34603 23610 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME AZD-1775 ADAVOSERTIB 34604 23611 ATAD5 79915 NA GW405833 CHEMBL73711 34606 23612 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ACTH CORTICOTROPIN 16330021 34607 23613 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME OLTIPRAZ OLTIPRAZ 12818361 34608 23614 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR 12-EPI-SALVINORIN B ETHOXYMETHYL ETHER CHEMBL1941031 22204910 34609 23615 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIMETHYLPINOCEMBRIN DIMETHYLPINOCEMBRIN 34610 23616 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL2107771 RALFINAMIDE 34611 23617 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METACETAMOL METACETAMOL 22613176 34612 23618 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE PIOGLITAZONE PIOGLITAZONE 34615 23619 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201542 INSULIN ZINC SUSP EXTENDED PURIFIED BEEF 34617 23620 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor NINTEDANIB NINTEDANIB 34620 23621 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AZATHIOPRINE AZATHIOPRINE 34621 23622 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Tricyclic pyrrolopyridine compound 1 34622 23623 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME AMPHOTERICIN B 2871108 34623 23624 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR IRIGENOL IRIGENOL 34624 23625 KDM4A 9682 DRUGGABLE GENOME, ENZYME 4-TERT-BUTYLCATECHOL CHEMBL220845 34626 23626 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR Emapalumab-lzsg EMAPALUMAB 34629 23627 SLC47A1 55244 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 178101502 PYRIMETHAMINE 34630 23628 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DIBENZ[A,H]ANTHRACENE DIBENZ[A,H]ANTHRACENE 34631 23629 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SYROSINGOPINE SYROSINGOPINE 34632 23630 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL538943 VINORELBINE TARTRATE 34633 23631 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PENT-1-ENE CHEMBL295337 34635 23632 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR inhibitor 363894175 34636 23633 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 135651718 34637 23634 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE THALIDOMIDE THALIDOMIDE 14995997 34638 23635 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PALBINONE PALBINONE 19716700 34639 23636 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Lobeglitazone LOBEGLITAZONE 34640 23637 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DAIDZEIN DAIDZEIN 34641 23638 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102049 34642 23639 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE GLUCOCORTICOID 9032457 34643 23640 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR ELLAGIC ACID ELLAGIC ACID 34644 23641 SLC28A1 9154 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE anthracyclines and related substances 23441093,21900104 34645 23642 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE PMID26882240-Compound-7 34646 23643 AQP9 366 ION CHANNEL inhibitor 178101032 34647 23644 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME blocker 178101077 34648 23645 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NOCODAZOLE NOCODAZOLE 34649 23646 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545396 BMS-690514 34650 23647 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BETA-LAPACHONE LAPACHONE 34652 23648 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TG02 ZOTIRACICLIB 34653 23649 SAE1 10055 ENZYME, DRUGGABLE GENOME 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 34654 23650 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME GW632580X GW632580X 34656 23651 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 pyridoxal phosphate 16770646 34657 23652 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CRYSTAL VIOLET HEXAMETHYL PARAROSANILINE 34659 23653 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-358518 CHEMBL352222 34661 23654 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DEPHOSTATIN DEPHOSTATIN 34663 23655 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SELENOMETHIONINE SELENOMETHIONINE 1759407 34665 23656 ALDH1A1 216 DRUGGABLE GENOME, ENZYME THIOMERSAL THIMEROSAL 34666 23657 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CB7969312 CHEMBL599255 34667 23658 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME NSC-107022 CHEMBL1601846 34669 23659 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE PYRANTEL PAMOATE PYRANTEL PAMOATE 34671 23660 EPHX2 2053 DRUGGABLE GENOME, ENZYME AR9281 AR9281 34672 23661 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME asparaginase ASPARAGINASE 24970932,25987655 34673 23662 GMNN 51053 DRUGGABLE GENOME IDAZOXAN HYDROCHLORIDE IDAZOXAN HYDROCHLORIDE 34675 23663 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW284372X GW284372X 34677 23664 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE METHIXENE HYDROCHLORIDE METHIXENE HYDROCHLORIDE 34678 23665 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 178100460 ZINTEROL 34679 23666 POLA1 5422 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, DNA REPAIR CLOFARABINE CLOFARABINE 34683 23667 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CHLOROQUINE CHLOROQUINE 22931300 34684 23668 MCOLN1 57192 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER activator 178103003 34685 23669 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CAMPTOTHECIN CAMPTOTHECIN 11205246 34687 23670 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME inhibitor SELUMETINIB SELUMETINIB 34688 23671 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 252166579 TACEDINALINE 34689 23672 PLCG1 5335 ENZYME, KINASE, PHOSPHOLIPASE, DRUGGABLE GENOME diclofenac DICLOFENAC 26398624 34690 23673 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor XL647 TESEVATINIB 34691 23674 PTGS1 5742 ENZYME, DRUGGABLE GENOME SALICYLIC ACID 34692 23675 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 34693 23676 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME 178101388 34694 23677 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-640353 CHEMBL1288253 21074425 34696 23678 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650759 34697 23679 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL2103810 EZATIOSTAT HYDROCHLORIDE 34698 23680 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL3545326 TAS-119 34699 23681 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR CEDIRANIB CEDIRANIB 34700 23682 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651740 34702 23683 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Ragaglitazar RAGAGLITAZAR 34703 23684 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME CYC-116 CYC-116 34704 23685 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE SP-600125 SP-600125 34705 23686 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-11 34706 23687 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102680 VX-702 34707 23688 KDM4A 9682 DRUGGABLE GENOME, ENZYME OMEPRAZOLE OMEPRAZOLE 34708 23689 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME PLX3397 PEXIDARTINIB 25939769,26222558 34711 23690 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME ML-10302 CHEMBL286136 34714 23691 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL564829 MILCICLIB 34716 23692 QRFPR 84109 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 329968383 34717 23693 KMO 8564 DRUGGABLE GENOME, ENZYME Cyclopropane 1-carboxylic acid derivative 10 34719 23694 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545083 RGB-286638 34720 23695 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME TDZD-8 34721 23696 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 310264761 CONESSINE 34722 23697 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL235191 TACEDINALINE 34723 23698 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Budesonide BUDESONIDE 34724 23699 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR dexamethasone DEXAMETHASONE 18285546 34725 23700 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME carboplatin CARBOPLATIN 26194361 34726 23701 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DNDI1417434 CHEMBL394883 34727 23702 MAPT 4137 DRUGGABLE GENOME 2',3'-DIHYDROXYFLAVONE CHEMBL242171 34728 23703 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrrolo-pyridine derivative 3 34730 23704 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RESORCINOL RESORCINOL 34731 23705 LGR6 59352 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178101191 34732 23706 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE FOLIC ACID 6732760 34734 23707 POLI 11201 DNA REPAIR SURAMIN HEXASODIUM SURAMIN HEXASODIUM 34735 23708 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME LY2228820 RALIMETINIB 34736 23709 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR APIGENIN APIGENIN 34737 23710 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE LAUROGUADINE LAUROGUADINE 34738 23711 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Trastuzumab TRASTUZUMAB 17936563,21676217,24470511 34740 23712 USP1 7398 DNA REPAIR, PROTEASE, ENZYME MIRIPIRIUM MIRIPIRIUM 34741 23713 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 34743 23714 SLC47A1 55244 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER Metformin METFORMIN 34744 23715 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1201777 TAPENTADOL HYDROCHLORIDE 34745 23716 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178101057 34747 23717 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE METIPRANOLOL METIPRANOLOL 34748 23718 DHFR 1719 DRUGGABLE GENOME, ENZYME inhibitor 405560261 ICLAPRIM 34749 23719 ERCC5 2073 DRUGGABLE GENOME, CLINICALLY ACTIONABLE platinum PLATINUM 22158331 34750 23720 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-52 34751 23721 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER VORINOSTAT VORINOSTAT 25669829 34754 23722 EZR 7430 CLINICALLY ACTIONABLE, KINASE TNF-ALPHA 15965500 34755 23723 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650115 CLOZAPINE 34759 23724 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL230011 TG100-115 34764 23725 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME GM6001 34766 23726 MPHOSPH8 54737 NA CGS-15943 CGS-15943 34767 23727 CBX1 10951 NA PYROGALLOL RED PYROGALLOL RED 34771 23728 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3544929 ABROCITINIB 34772 23729 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE CYC-116 CYC-116 34774 23730 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL2103839 RIDAFOROLIMUS 34775 23731 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR TCMDC-139459 CHEMBL86464 34776 23732 CRBN 51185 ENZYME, DRUG RESISTANCE 387065622 34777 23733 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME CLX-0921 CLX-0921 34778 23734 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE Entrectinib ENTRECTINIB 26884591,26939704 34779 23735 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PROPAFENONE PROPAFENONE 34781 23736 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY ANTISERUM 1827257 34782 23737 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BGJ398 INFIGRATINIB 34785 23738 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Oxindole derivative 4 34789 23739 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME antagonist 178103613 34790 23740 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR PT2399 27595393 34791 23741 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE nitrofurantoin NITROFURANTOIN 5897424,20701405,12659,1669155 34793 23742 UGT2B15 7366 DRUGGABLE GENOME phenytoin PHENYTOIN 26049587 34795 23743 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TANSHINONE IIA SULFONATE TANSHINONE IIA SULFONATE 34796 23744 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME OFLOXACIN OFLOXACIN 15008519 34798 23745 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE TAE-684 TAE-684 34801 23746 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME RHuEPO 34805 23747 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER TROXACITABINE TROXACITABINE 12451476 34806 23748 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CEDIRANIB CEDIRANIB 34807 23749 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-19063 CHEMBL1310138 34809 23750 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103493 34810 23751 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CARBOQUONE CARBOQUONE 34812 23752 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor XL281 XL-281 34813 23753 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RESVERATROL RESVERATROL 11279601 34814 23754 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE KRC-00715 26801760 34815 23755 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OSTHOLE OSTHOLE 34816 23756 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME CADMIUM DICHLORIDE CADMIUM DICHLORIDE 34817 23757 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE PF-228 CHEMBL514554 34818 23758 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRENBOLONE ACETATE TRENBOLONE ACETATE 34819 23759 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DIETHYLDITHIOCARBAMATE DITIOCARB 2992773 34820 23760 RBL2 5934 TRANSCRIPTION FACTOR COMPLEX, ENZYME RAPAMYCIN SIROLIMUS 8895523 34821 23761 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME LINIFANIB LINIFANIB 34822 23762 SLC25A20 788 DRUGGABLE GENOME, TRANSPORTER PROPIONYL-L-CARNITINE 34823 23763 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GW843682X GW843682X 34825 23764 ATXN2 6311 NA SAQUINAVIR MESYLATE SAQUINAVIR MESYLATE 34827 23765 CRP 1401 DRUGGABLE GENOME ISIS-CRPRX 34828 23766 MALAT1 378938 NA ZD-7288 CHEMBL2052019 34829 23767 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SC-514 CHEMBL193093 34833 23768 GGCX 2677 DRUGGABLE GENOME, ENZYME PHYTONADIONE PHYTONADIONE 34834 23769 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME CIPEMASTAT CIPEMASTAT 34835 23770 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING TROPISETRON TROPISETRON 34836 23771 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Insulin-glulisine 34837 23772 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DT-061 28504649 34838 23773 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CANDIDIN CANDIDIN 34839 23774 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR HOMATROPINE METHYLBROMIDE 34840 23775 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IDAZOXAN HYDROCHLORIDE IDAZOXAN HYDROCHLORIDE 34844 23776 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ketoconazole KETOCONAZOLE 34845 23777 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR KEPONE KEPONE 34846 23778 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417085 CHEMBL1522984 34847 23779 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-2491 CHEMBL577851 34849 23780 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR Topotecan TOPOTECAN 26936505 34850 23781 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR SB-220025 SB-220025 34851 23782 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135651526 NOREPINEPHRINE BITARTRATE 34852 23783 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DOVITINIB DOVITINIB 34856 23784 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20100022547C88 34857 23785 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ALDICARB ALDICARB 34858 23786 TSPO 706 DRUGGABLE GENOME Imidazopyridine acetamide analog 6 34859 23787 KMO 8564 DRUGGABLE GENOME, ENZYME Cyclopropane 1-carboxylic acid derivative 6 34862 23788 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 310264678 34863 23789 USP1 7398 DNA REPAIR, PROTEASE, ENZYME QUINOCIDE QUINOCIDE 34864 23790 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135650232 ENPROSTIL 34869 23791 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565831 34870 23792 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-4746 CHEMBL584868 34871 23793 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME SF1126 34872 23794 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME N-BENZOYLANTHRANILIC ACID CHEMBL198666 34873 23795 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MC-3002 34874 23796 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417777 CHEMBL1412002 34875 23797 RAPGEF3 10411 ENZYME BITHIONOLOXIDE BITHIONOLOXIDE 34876 23798 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME LINIFANIB LINIFANIB 34878 23799 POLK 51426 DNA REPAIR, ENZYME 5,7-DIHYDROXYISOFLAVONE 5,7-DIHYDROXYISOFLAVONE 34879 23800 NCOA3 8202 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, ENZYME METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 34880 23801 AKT1S1 84335 KINASE, DRUGGABLE GENOME inhibitor OSI-027 OSI-027 34881 23802 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME Ravulizumab RAVULIZUMAB 34882 23803 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Ximelegatran 34884 23804 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME BELACTOSIN A BELACTOSIN A 23547757 34885 23805 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CITRIC ACID CITRIC ACID 34886 23806 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE MENTHOL MENTHOL 17293875 34887 23807 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DAMNACANTHAL DAMNACANTHAL 34889 23808 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE TIVOZANIB TIVOZANIB 34890 23809 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME DAUNORUBICIN DAUNORUBICIN 34891 23810 GAA 2548 DRUGGABLE GENOME, ENZYME ACARBOSE ACARBOSE 34893 23811 CEL 1056 CELL SURFACE, DRUGGABLE GENOME, ENZYME SIMVASTATIN SIMVASTATIN 16955753 34894 23812 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE RALTITREXED RALTITREXED 34895 23813 DMD 1756 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME PRO044 34897 23814 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-5061 CHEMBL601385 34899 23815 CAMKK2 10645 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE CQ7 34901 23816 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL Imagabalin IMAGABALIN 34903 23817 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201628 INSULIN SUSP PROTAMINE ZINC BEEF/PORK 34905 23818 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 135651285 34909 23819 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR Mavrilimumab MAVRILIMUMAB 34910 23820 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GSK343 26676756 34913 23821 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PD-0166285 PD-0166285 34914 23822 CYP51A1 1595 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 252827457 AZALANSTAT 34915 23823 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CEPHALOCHROMIN CEPHALOCHROMIN 34916 23824 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Palbociclib/ribociclib analog 1 34919 23825 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GUANFACINE GUANFACINE 34921 23826 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME SB-509 34922 23827 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE paroxetine PAROXETINE 34923 23828 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR E319 E319 34924 23829 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GDC-0032 TASELISIB 28331003 34926 23830 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Tetra-cyclic pyridophthalazinone derivative 1 34927 23831 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME TRAMETINIB TRAMETINIB 23020132,22608338,26619011,21483012,2493360,22351686,19001320,21156289,20368568,19255327,22048237,19561230,19010912,23549875,25024077,22798288,23489023,18541894,24586605,24508103,22773810,23833300,23812671,24576830,19238210,20818844,23612012,23251002,22356324,20857202,22536370,22997239,21163703,15035987,23470635,21663470,24594804,22586120,20413299,23715574,22805292,19537845,14679157,22663011,21975775,22038996,22448344,12068308,24163374,19773371,24354346,23325582,24583796,23031422,22735384,21683865,25370471,21639808,22281684,22649091,22241789,24570209,23918947,25989278,22389471,23934108,22180495,23524406,26678033,19018267,24388723,23845441,23614898,25157968,20619739,12460919,24107445,12460918,21594703,20350999,20630094,21426297,19404918,22743296,24396464,22972589,21129611,23406027,25656898 34928 23832 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 381118861 34929 23833 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor 310264733 FIMEPINOSTAT 34930 23834 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 249565643 RABUSERTIB 34932 23835 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL971 PENTOBARBITAL SODIUM 34934 23836 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor LEE011 RIBOCICLIB 34935 23837 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PF-431396 CHEMBL472212 27793840 34937 23838 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Hydroxyzine HYDROXYZINE 34939 23839 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 12-HYDROXY-OCTADECANOIC ACID CHEMBL292352 34940 23840 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL BROMAZEPAM BROMAZEPAM 34943 23841 ERAP2 64167 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE ESCULETIN ESCULETIN 34944 23842 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Quinoline and quinazoline derivative 10 34945 23843 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649667 34946 23844 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 340590276 34947 23845 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE POLYPHENOL 16707458 34948 23846 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME FLUTICASONE PROPIONATE 34949 23847 MAPK7 5598 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 328083508 34950 23848 CASP8 841 DRUGGABLE GENOME, PROTEASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL2105721 NIVOCASAN 34951 23849 PRMT1 3276 ENZYME, METHYL TRANSFERASE inhibitor 178103608 34952 23850 XDH 7498 DRUGGABLE GENOME, ENZYME FOLIC ACID 6547955 34953 23851 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-13 34954 23852 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CUDC-101 CUDC-101 34955 23853 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000120449 CHEMBL609027 34959 23854 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102578 34961 23855 SMN2 6607 DRUGGABLE GENOME NSC-102045 CHEMBL483633 34962 23856 CPB1 1360 DRUGGABLE GENOME, PROTEASE, ENZYME US8710232, 8 34964 23857 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TANSHINONE I TANSHINONE I 34965 23858 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545003 MSC-2363318A 34966 23859 MAPT 4137 DRUGGABLE GENOME OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 34967 23860 PCSK7 9159 ENZYME, PROTEASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 252166858 34968 23861 PCSK5 5125 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166868 34969 23862 P2RX4 5025 ION CHANNEL, DRUGGABLE GENOME antagonist 336446928 34970 23863 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR PMID25980951-Compound-1 34972 23864 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051798 BELINOSTAT 34974 23865 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUNITROLOL BUNITROLOL 2903243 34975 23866 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING GEMFIBROZIL GEMFIBROZIL 16680159 34977 23867 KMT2D 8085 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE HDAC INHIBITOR AR-42 25273096 34978 23868 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 381744939 34982 23869 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-4300 CHEMBL585656 34983 23870 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PILOCARPINE PILOCARPINE 34986 23871 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL1980391 RG-1530 34988 23872 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE THROMBIN THROMBIN 15559761,15280447,11504518,10027305,15383630,12707033,11841573,15386385,14699102 34989 23873 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 34995 23874 ABCA1 19 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE 315661263 34996 23875 RHOA 387 KINASE, CLINICALLY ACTIONABLE ROTTLERIN ROTTLERIN 22093759 34998 23876 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME lifitegrast LIFITEGRAST 34999 23877 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE U0126 19078957 35000 23878 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PACLITAXEL PACLITAXEL 35001 23879 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BENZO[B]FLUORANTHENE BENZO[B]FLUORANTHENE 35003 23880 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CERITINIB CERITINIB 26870817 35004 23881 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CB-03-01 CLASCOTERONE 35005 23882 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GLYCYRRHIZIN GLYCYRRHIZIN 35006 23883 BRDT 676 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE (+)-JQ1 35007 23884 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DCMU DCMU 35008 23885 MAPT 4137 DRUGGABLE GENOME AG-1288 CHEMBL166486 35010 23886 LPAR5 57121 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 381744912 35012 23887 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-39 35014 23888 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 348353622 35015 23889 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SERTACONAZOLE NITRATE SERTACONAZOLE NITRATE 35016 23890 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28117607-Compound-4 35017 23891 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME SNS-314 SNS-314 35018 23892 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Acitretin ACITRETIN 35019 23893 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 35020 23894 CAMK1D 57118 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME inhibitor 178102336 BOSUTINIB 35021 23895 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Bicalutamide BICALUTAMIDE 35022 23896 DBI 1622 NA HORMONES 9712181 35023 23897 SMN1 6606 DRUGGABLE GENOME CID 893238 CHEMBL473735 35024 23898 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CENISERTIB CENISERTIB 35025 23899 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME TAK-733 TAK-733 35026 23900 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1201006 PYRILAMINE MALEATE 35028 23901 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE antibody DULANERMIN DULANERMIN 35029 23902 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 384403666 35030 23903 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME CAR-T Cells targeting CEA 35031 23904 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Tbo-Filgrastim FILGRASTIM 35032 23905 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME RFIX 35033 23906 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR NERVE GROWTH FACTOR 10894779 35034 23907 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ANDROSTENEDIONE ANDROSTENEDIONE 9384522 35035 23908 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE S-49076 23804704 35038 23909 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER NEVIRAPINE NEVIRAPINE 21189339 35044 23910 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR (1R)-TRANS-TETRAMETHRIN (1R)-TRANS-TETRAMETHRIN 35045 23911 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME larotrectinib sulfate 35047 23912 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PRACINOSTAT PRACINOSTAT 35049 23913 POLK 51426 DNA REPAIR, ENZYME CONGO RED CONGO RED 35050 23914 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Antegren 35051 23915 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ZYH-7 35052 23916 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE benazepril BENAZEPRIL 15554460 35053 23917 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BOLDINE BOLDINE 35054 23918 PHKG1 5260 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565884 A-443654 35058 23919 POLR2A 5430 NA gemcitabine GEMCITABINE 35062 23920 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200990 FLURBIPROFEN SODIUM 35064 23921 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DERRUSNIN DERRUSNIN 35065 23922 SMN1 6606 DRUGGABLE GENOME BIOCHANIN BIOCHANIN 35067 23923 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUCINDOLOL BUCINDOLOL 35071 23924 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-28 35072 23925 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME JL-18 CHEMBL63329 35073 23926 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Midostaurin MIDOSTAURIN 25209843 35074 23927 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4102 CHEMBL596836 35075 23928 MAOA 4128 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 4 35076 23929 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE Becaplermin BECAPLERMIN 35078 23930 BCOR 54880 CLINICALLY ACTIONABLE Tretinoin TRETINOIN 25790901 35079 23931 ALOX15 246 ENZYME, DRUGGABLE GENOME 5,7,3',5'-TETRAHYDROXYFLAVANONE CHEMBL307893 35081 23932 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Binimetinib BINIMETINIB 26206338,28152546,25167228,27556948,27422710 35083 23933 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CABOZANTINIB CABOZANTINIB 35084 23934 APEH 327 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166764 35085 23935 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME PACLITAXEL PACLITAXEL 12574211 35087 23936 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PLUMBAGIN PLUMBAGIN 35088 23937 PSMD13 5719 NA inhibitor CHEMBL451887 CARFILZOMIB 35089 23938 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME KOBOPHENOL A KOBOPHENOL A 17300930 35090 23939 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Methacholine Chloride 35091 23940 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE PHENOL PHENOL 35093 23941 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DIPHENIDOL DIPHENIDOL 35094 23942 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME agonist 135651597 35095 23943 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-4459 CHEMBL585502 35096 23944 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor REGORAFENIB REGORAFENIB 35097 23945 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MIANSERIN MIANSERIN 35098 23946 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MEDRYSONE MEDRYSONE 35100 23947 TPM3 7170 KINASE, CLINICALLY ACTIONABLE PROGESTERONE PROGESTERONE 17549730 35101 23948 IRS1 3667 KINASE, CLINICALLY ACTIONABLE INOSITOL INOSITOL 9693122 35104 23949 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME THC DRONABINOL 7945419 35105 23950 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE HOMIDIUM BROMIDE HOMIDIUM BROMIDE 35106 23951 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FURAZOLIDONE FURAZOLIDONE 35107 23952 MLST8 64223 KINASE inhibitor MLN0128 SAPANISERTIB 35109 23953 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE DASATINIB DASATINIB 35110 23954 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650056 CARBACYCLIN 35112 23955 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Copanlisib COPANLISIB 24170767 35113 23956 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TCMDC-125578 CHEMBL195350 35114 23957 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BETA-SITOSTEROL BETA-SITOSTEROL 19716700 35115 23958 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor CHEMBL1946170 REGORAFENIB 35121 23959 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor XL-765 VOXTALISIB 35122 23960 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE RG7116 35123 23961 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME ENZASTAURIN ENZASTAURIN 22333600 35124 23962 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor CHEMBL506871 VELIPARIB 35125 23963 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PALIPERIDONE PALIPERIDONE 35126 23964 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL377300 BRIVANIB 35128 23965 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178102577 35129 23966 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL429736 RETOSIBAN 35130 23967 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME GLEEVEC IMATINIB 15805252,15155841 35131 23968 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ETOMIDATE ETOMIDATE 16884293,20704351 35132 23969 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR VX-745 NEFLAMAPIMOD 35133 23970 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565803 35134 23971 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ALFATRADIOL ALFATRADIOL 35135 23972 RIT1 6016 CLINICALLY ACTIONABLE PICTILISIB PICTILISIB 24469055 35136 23973 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CR665 35137 23974 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102736 35139 23975 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 URAPIDIL URAPIDIL 35141 23976 CBX1 10951 NA FLUPENTIXOL FLUPENTIXOL 35143 23977 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33a 35146 23978 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TAXIFOLIN TAXIFOLIN 35147 23979 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE Paclitaxel PACLITAXEL 28514312 35148 23980 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME AMG-102 RILOTUMUMAB 35149 23981 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Pyrimidine derivative 20 35150 23982 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME TAE-684 TAE-684 35151 23983 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4853 CHEMBL599957 35154 23984 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE phenytoin PHENYTOIN 12083967 35157 23985 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROMAZINE PROMAZINE 35160 23986 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MAPROTILINE MAPROTILINE 22931300 35162 23987 IL33 90865 DRUGGABLE GENOME AMG 282 35163 23988 PDE4A 5141 DRUGGABLE GENOME, ENZYME Apremilast APREMILAST 35164 23989 CTSF 8722 DRUGGABLE GENOME, PROTEASE, ENZYME PMID27998201-Compound-5 35165 23990 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BUMETANIDE BUMETANIDE 35168 23991 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL49642 INDIBULIN 35169 23992 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE CORTISOL HYDROCORTISONE 1597147 35170 23993 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE DASATINIB DASATINIB 35172 23994 ERAP2 64167 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE inhibitor 348353641 35173 23995 SMN1 6606 DRUGGABLE GENOME LUTEOLIN LUTEOLIN 35174 23996 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR SNS-314 SNS-314 35179 23997 F2RL3 9002 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME VORAPAXAR VORAPAXAR 35180 23998 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE TAS-120 FUTIBATINIB 35181 23999 ATXN2 6311 NA GNF-PF-4300 CHEMBL585656 35183 24000 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR RALOXIFENE RALOXIFENE 35185 24001 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 7 35188 24002 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR MART1 16968820 35190 24003 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE AZD-1152-HQPA AZD-1152-HQPA 35191 24004 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME LUTEOLIN LUTEOLIN 35192 24005 HMGCR 3156 ENZYME, DRUGGABLE GENOME LAROPIPRANT LAROPIPRANT 35193 24006 ALOX15B 247 DRUGGABLE GENOME, ENZYME 4-METHOXYDALBERGIONE 4-METHOXYDALBERGIONE 35194 24007 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TELMISARTAN TELMISARTAN 35195 24008 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME 3,4-DIHYDROXYPHENYLACETIC ACID 3,4-DIHYDROXYPHENYLACETIC ACID 35197 24009 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME AZD8055 AZD-8055 26544513 35198 24010 RFC1 5981 DNA REPAIR PRALATREXATE PRALATREXATE 35199 24011 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME ZEARALENONE ZEARALENONE 35200 24012 SMARCB1 6598 CLINICALLY ACTIONABLE DZNeP 23190500 35201 24013 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Everolimus EVEROLIMUS 26951309,20664174,20664172,22473592,21358673,22662154,28330462 35202 24014 MPHOSPH8 54737 NA SU-6656 CHEMBL605003 35203 24015 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL2141712 PALOMID-529 35205 24016 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE SF1126 35209 24017 PTPA 5524 PROTEIN PHOSPHATASE LB-100 LB-100 35210 24018 SGMS1 259230 ENZYME, KINASE inhibitor 252827492 35212 24019 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE JNJ-7706621 JNJ-7706621 35214 24020 DHODH 1723 DRUGGABLE GENOME, ENZYME IMMUNOSUPPRESSIVE 7575649 35215 24021 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL898 DIFLUNISAL 35216 24022 VEGFC 7424 GROWTH FACTOR, TRANSPORTER, DRUGGABLE GENOME VGX-100 VGX-100 35219 24023 ATXN2 6311 NA GNF-PF-5151 CHEMBL576208 35221 24024 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME modulator CHEMBL593430 ATAGABALIN 35222 24025 MPHOSPH8 54737 NA NCG-C00093820-01 CHEMBL544115 35223 24026 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 223366046 AZD-7762 35224 24027 GMNN 51053 DRUGGABLE GENOME ALBENDAZOLE ALBENDAZOLE 35226 24028 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CIS-2,4,3',5'-TETRAMETHOXYSTILBENE CHEMBL221300 35227 24029 MAOA 4128 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 2 35228 24030 FST 10468 DRUGGABLE GENOME ALPHA-ADRENERGIC AGONIST 9427529 35229 24031 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE LAPATINIB LAPATINIB 23680147 35230 24032 APOE 348 DRUGGABLE GENOME GANCICLOVIR GANCICLOVIR 16322528 35232 24033 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE GELDANAMYCIN GELDANAMYCIN 7662976 35233 24034 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Chlorotrianisene CHLOROTRIANISENE 35235 24035 PSMD4 5710 NA CARFILZOMIB CARFILZOMIB 27033953 35237 24036 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME NICOTINE NICOTINE 16011614 35239 24037 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SB-415286 CHEMBL322970 35240 24038 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PF-04995274 PF-04995274 35241 24039 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 178102286 QUIZARTINIB 35242 24040 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VANOXERINE VANOXERINE 35245 24041 MAPT 4137 DRUGGABLE GENOME DIAMIDE DIAMIDE 35246 24042 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Insulin Lyspro recombinant 35248 24043 POLB 5423 DNA REPAIR, DRUGGABLE GENOME 2'-HYDROXYGENISTEIN CHEMBL6665 35249 24044 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor 315661304 RAVOXERTINIB 35250 24045 MAPT 4137 DRUGGABLE GENOME INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 35253 24046 BAZ2B 29994 NA GNF-PF-1319 CHEMBL235891 35254 24047 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-5151 CHEMBL576208 35255 24048 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME EMBELIN EMBELIN 35256 24049 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR GEMFIBROZIL GEMFIBROZIL 8941582 35257 24050 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME KRAS mutant-specific TIL 27959684 35258 24051 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE N-(3-PHENYLPROPYL)BENZAMIDE CHEMBL1404865 35262 24052 ARSA 410 DRUGGABLE GENOME, ENZYME SPIROXATRINE SPIROXATRINE 35263 24053 RPS6KA6 27330 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME CEP-1347 CEP-1347 24044867 35264 24054 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CETRIMONIUM BROMIDE CETRIMONIUM BROMIDE 35266 24055 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE SOTRASTAURIN SOTRASTAURIN 35267 24056 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GW7647 GW7647 35269 24057 BAZ2B 29994 NA DNDI1417777 CHEMBL1412002 35270 24058 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE OK-432 1963635 35271 24059 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX HALOPERIDOL HALOPERIDOL 16893530 35272 24060 CD36 948 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ABT-510 ABT-510 35273 24061 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ELINAFIDE ELINAFIDE 21880496 35274 24062 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LAUROGUADINE LAUROGUADINE 35275 24063 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650330 CHEMBL434063 35277 24064 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PALINURIN PALINURIN 23354070 35279 24065 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME VANOXERINE VANOXERINE 35281 24066 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LY2090314 LY-2090314 35283 24067 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-123579 CHEMBL533954 35284 24068 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PROPYLPYRAZOLETRIOL PROPYLPYRAZOLETRIOL 35285 24069 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GLUCOCORTICOID 15544592 35286 24070 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL activator 178100888 35287 24071 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME SENNOSIDE B SENNOSIDE B 35291 24072 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ACETAMINOPHEN ACETAMINOPHEN 8699917 35293 24073 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE TRICETIN TRICETIN 35294 24074 ALOX15 246 ENZYME, DRUGGABLE GENOME NEROLIDOL NEROLIDOL 35295 24075 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8536181, A41 35296 24076 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE sulfinpyrazone SULFINPYRAZONE 22981363 35297 24077 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME MDCO-216 35298 24078 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor LY2940680 35301 24079 HTT 3064 DRUGGABLE GENOME MGCD-0103 MOCETINOSTAT 35302 24080 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 223366209 CEP-32496 35303 24081 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649770 35304 24082 HLA-E 3133 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE infliximab INFLIXIMAB 35305 24083 BAZ2B 29994 NA N'-(2,4-DIHYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE CHEMBL199592 35306 24084 CBX1 10951 NA PIMOZIDE PIMOZIDE 35307 24085 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Necitumumab NECITUMUMAB 35308 24086 PBRM1 55193 CLINICALLY ACTIONABLE ANTI-PD-L1 MONOCLONAL ANTIBODY 29301960 35312 24087 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR IUDR 1313063 35313 24088 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Protriptyline PROTRIPTYLINE 35315 24089 CACNB4 785 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL593430 ATAGABALIN 35316 24090 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CHEMBL1200789 TRICLOFOS SODIUM 35317 24091 TPSAB1 7177 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 223366193 GABEXATE 35318 24092 EYA2 2139 DNA REPAIR 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 35319 24093 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor CHEMBL2108742 SIPLIZUMAB 35320 24094 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651792 35322 24095 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR NN-7415 35323 24096 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 135651519 35324 24097 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE METHYL 2-(2-METHOXYBENZAMIDO)BENZOATE CHEMBL249190 35325 24098 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3707400 INDANTADOL 35326 24099 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE NIC5-15 METHYLINOSITOL 35327 24100 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE RISEDRONATE RISEDRONIC ACID 35328 24101 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Asimadoline ASIMADOLINE 35329 24102 NQO2 4835 DRUGGABLE GENOME, ENZYME NSC-640583 CHEMBL1287895 21074425 35331 24103 UGT1A6 54578 ENZYME, DRUGGABLE GENOME allopurinol ALLOPURINOL 27798726 35333 24104 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME Venetoclax VENETOCLAX 35335 24105 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE FLUORESCEIN SODIUM FLUORESCEIN SODIUM 22889313 35337 24106 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 348353615 35338 24107 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME quetiapine QUETIAPINE 23859574,20031235 35339 24108 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 135652071 35341 24109 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE EPO EPOETIN ALFA 1300984 35342 24110 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DZNep 26676756 35343 24111 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID28048944-Compound-2 35346 24112 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY SUMATRIPTAN SUMATRIPTAN 9486164 35347 24113 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3,3',4'-TRIHYDROXYFLAVONE CHEMBL122701 35348 24114 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CARNOSIC ACID CARNOSIC ACID 35350 24115 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME carbimazole CARBIMAZOLE 35351 24116 BAZ2B 29994 NA S-NITROSOGLUTATHIONE S-NITROSOGLUTATHIONE 35352 24117 SLC16A7 9194 DRUGGABLE GENOME, TRANSPORTER inhibitor 404859052 35353 24118 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178103999 VILAZODONE 35355 24119 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Avapritinib AVAPRITINIB 35358 24120 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL1201770 METHYLNALTREXONE BROMIDE 35360 24121 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GENTIAN VIOLET GENTIAN VIOLET 35361 24122 SMAD2 4087 KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ATRA TRETINOIN 15799023 35362 24123 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE HARMALOL HARMALOL 35363 24124 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR morphine MORPHINE 29259946 35364 24125 TMEM97 27346 NA Benzamide derivative 3 35365 24126 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 35367 24127 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR PALBOCICLIB PALBOCICLIB 35368 24128 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BERBERINE CHLORIDE BERBERINE CHLORIDE 35369 24129 KDM4A 9682 DRUGGABLE GENOME, ENZYME 4,4'-DITHIODIPYRIDINE CHEMBL1232076 35372 24130 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DANAZOL DANAZOL 22931300 35373 24131 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Bicyclic heteroaryl benzamide derivative 2 35375 24132 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE MP-412 MP-412 35376 24133 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1200695 PHENYLPROPANOLAMINE HYDROCHLORIDE 35377 24134 PTGS2 5743 DRUGGABLE GENOME, ENZYME KETOPROFEN KETOPROFEN 35378 24135 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 670282 CHEMBL260213 35379 24136 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1215923 BIMOSIAMOSE 35381 24137 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENAZEPRIL HYDROCHLORIDE BENAZEPRIL HYDROCHLORIDE 35383 24138 S100A12 6283 DRUGGABLE GENOME, KINASE METHOTREXATE METHOTREXATE 15077313 35384 24139 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE AN0128 35385 24140 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Umeclidinium UMECLIDINIUM 35387 24141 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE VEGF 16138928 35388 24142 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Epirubicin EPIRUBICIN 17388661 35389 24143 COMT 1312 DRUGGABLE GENOME, ENZYME entacapone ENTACAPONE 21280081 35391 24144 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MI-503 25817203 35398 24145 SLC15A2 6565 TRANSPORTER, DRUGGABLE GENOME 178101217 35399 24146 ENTPD1 953 DRUGGABLE GENOME, CELL SURFACE, ENZYME inhibitor 315661108 CHEMBL608559 35400 24147 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME RIBOFLAVIN RIBOFLAVIN 35401 24148 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RIFAMPICIN RIFAMPIN 35402 24149 CYB5R3 1727 DRUGGABLE GENOME, ENZYME metoclopramide METOCLOPRAMIDE 11418378 35404 24150 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 4-AMINOBENZAMIDINE DIHYDROCHLORIDE CHEMBL545184 35405 24151 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME ERYTHROMYCIN ERYTHROMYCIN 17007374 35407 24152 CFH 3075 DRUGGABLE GENOME photodynamic therapy 26780119,18292785,18050121 35408 24153 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE OSI-632 OSI-632 35410 24154 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 223366035 ADAVOSERTIB 35411 24155 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Radiotherapy 21992793,26358474,18026198,28062704,21799033,26162687 35412 24156 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE XL418 XL-418 35413 24157 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8481586, 5 35414 24158 DUSP6 1848 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE TRAMETINIB TRAMETINIB 22169769 35415 24159 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME BENZIODARONE BENZIODARONE 35416 24160 XDH 7498 DRUGGABLE GENOME, ENZYME Curcumin CURCUMIN 35417 24161 KDM4A 9682 DRUGGABLE GENOME, ENZYME FENRETINIDE FENRETINIDE 35421 24162 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME CYCLOTHIAZIDE CYCLOTHIAZIDE 35424 24163 SMN2 6607 DRUGGABLE GENOME 2-AMINO-ANTHRAQUINONE CHEMBL84685 35425 24164 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652337 35426 24165 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME VESNARINONE VESNARINONE 15356428 35428 24166 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565781 SPLITOMICIN 35429 24167 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE NSC-628113 CHEMBL176599 35430 24168 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545088 PUQUITINIB 35432 24169 SOAT1 6646 DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 7485476 35433 24170 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME TTA-A8 35436 24171 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE GNF-PF-108 CHEMBL578929 35437 24172 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME DAUNORUBICIN DAUNORUBICIN 22260166 35438 24173 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8598210, Table XV, 1 35441 24174 AKR1C3 8644 ENZYME, DRUGGABLE GENOME exemestane EXEMESTANE 27111237 35442 24175 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE INCB28060 CAPMATINIB 35443 24176 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1201649 ESTROGENS, CONJUGATED 35444 24177 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ESTRIOL ESTRIOL 35445 24178 SMN2 6607 DRUGGABLE GENOME ANISINDIONE ANISINDIONE 35446 24179 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME (+)-EPITAXIFOLIN (+)-EPITAXIFOLIN 35447 24180 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW829115X GW829115X 35451 24181 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BAY-11-7082 CHEMBL403183 35454 24182 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER TIOPRONIN TIOPRONIN 21657271 35455 24183 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-41 35456 24184 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME SHIKONIN SHIKONIN 35457 24185 TUBB 203068 DRUGGABLE GENOME CHEMBL2103826 DAVUNETIDE 35459 24186 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME amodiaquine AMODIAQUINE 17361129,21998472,23204183,18855526 35460 24187 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX IMATINIB IMATINIB 35461 24188 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE fluorouracil FLUOROURACIL 23816762 35462 24189 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME peginterferon alfa-2b 23360626 35464 24190 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE BUSULFAN BUSULFAN 2635153 35465 24191 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32r 35467 24192 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME AG-490 CHEMBL56543 35468 24193 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649963 35470 24194 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102249 GS 6201 35471 24195 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LINIFANIB LINIFANIB 35472 24196 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 35473 24197 ATAD5 79915 NA AG1295 AG1295 35475 24198 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545008 SAR-260301 35476 24199 LIPF 8513 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL175247 ORLISTAT 35478 24200 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE BGB-290 PAMIPARIB 35482 24201 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFACON-1 35485 24202 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Isoxazole derivative 2 35486 24203 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR ANTIOXIDANT 12520757 35487 24204 TUBA3D 113457 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 35489 24205 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651110 35490 24206 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MVA HER-2 AutoVac 35491 24207 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Netarsudil NETARSUDIL 35492 24208 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178102342 FEDRATINIB 35493 24209 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME REL-CARINATIN B CHEMBL2332126 35495 24210 PAK2 5062 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 310264719 35496 24211 KDM4A 9682 DRUGGABLE GENOME, ENZYME 5,7,3',5'-TETRAHYDROXYFLAVANONE CHEMBL307893 35499 24212 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Lasofoxifene LASOFOXIFENE 35500 24213 GPX1 2876 DRUGGABLE GENOME, PROTEASE INHIBITOR GP-120 16871233 35502 24214 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Atrasentan ATRASENTAN 35503 24215 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ULIPRISTAL ULIPRISTAL 35504 24216 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 178100958 APIGENIN 35506 24217 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor XL647 TESEVATINIB 35507 24218 CA2 760 DRUGGABLE GENOME, ENZYME Salicyclic acid 35508 24219 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PROROXAN HYDROCHLORIDE PROROXAN HYDROCHLORIDE 35510 24220 TXN2 25828 DRUGGABLE GENOME, THIOREDOXIN GAMBOGIC ACID GAMBOGIC ACID 22663155 35513 24221 PTGS1 5742 ENZYME, DRUGGABLE GENOME FENBUFEN FENBUFEN 35514 24222 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHENELZINE PHENELZINE 35515 24223 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PD-153035 CHEMBL29197 35516 24224 SMN1 6606 DRUGGABLE GENOME BROXURIDINE BROXURIDINE 35518 24225 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME troglitazone TROGLITAZONE 14977862 35520 24226 PTGS2 5743 DRUGGABLE GENOME, ENZYME Celecoxib CELECOXIB 35521 24227 PTGS2 5743 DRUGGABLE GENOME, ENZYME CG-100649 POLMACOXIB 35522 24228 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL3185958 CLOMIPHENE CITRATE 35523 24229 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR OPHIOBOLIN O OPHIOBOLIN O 22130129 35524 24230 ATAD5 79915 NA 6-HYDROXYFLAVONE 6-HYDROXYFLAVONE 35526 24231 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-10 35527 24232 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 252166787 35528 24233 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLORAZEPATE CLORAZEPIC ACID 35529 24234 MAGEA12 4111 NA vaccine MAGE-12 PEPTIDE VACCINE 35531 24235 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING BRUCEANTIN BRUCEANTIN 19199792 35532 24236 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL1200641 CISATRACURIUM BESYLATE 35533 24237 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Pyrrolo[2,3-d]pyrimidine derivative 9 35534 24238 POLK 51426 DNA REPAIR, ENZYME NSC-180246 CHEMBL484640 35535 24239 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200409 LIDOCAINE HYDROCHLORIDE 35536 24240 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LATANOPROST LATANOPROST 35537 24241 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME 3-HYDROXYBENZYLHYDRAZINE DIHYDROCHLORIDE 35538 24242 IMPDH2 3615 DRUGGABLE GENOME, ENZYME MYCOPHENOLATE MOFETIL 35539 24243 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102907 ISOVELLERAL 35540 24244 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE TOPOTECAN TOPOTECAN 10803925 35542 24245 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DRONEDARONE DRONEDARONE 35544 24246 ATAD5 79915 NA AZACITIDINE AZACITIDINE 35547 24247 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor CHEMBL1580 PENTOSTATIN 35548 24248 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER IL-6 7564516 35550 24249 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 METARAMINOL METARAMINOL 22931300 35551 24250 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 384403666 35552 24251 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BUTANOIC ACID BUTANOIC ACID 19053749 35555 24252 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-2776 CHEMBL578294 35557 24253 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BITHIONOL BITHIONOL 35559 24254 MPHOSPH8 54737 NA FLUSPIRILENE FLUSPIRILENE 35560 24255 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 178103659 35561 24256 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE FUROSPONGOLIDE FUROSPONGOLIDE 18989978 35562 24257 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PINDOLOL PINDOLOL 35563 24258 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651383 35564 24259 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE HIF-1ALPHA 35566 24260 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 363894195 35567 24261 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHENANTHROLINE PHENANTHROLINE 35570 24262 CHST3 9469 DRUGGABLE GENOME, ENZYME docetaxel DOCETAXEL 20038957 35571 24263 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 375973268 35572 24264 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR TPA ALTEPLASE 18815270,18563704 35573 24265 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RAUWOLFIA SERPENTINA RAUWOLFIA SERPENTINA 35574 24266 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE Rosiglitazone + metformin 35576 24267 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME CISPLATIN CISPLATIN 11800022,12519017 35577 24268 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ORPHENADRINE CITRATE ORPHENADRINE CITRATE 35579 24269 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PROPYLPYRAZOLETRIOL PROPYLPYRAZOLETRIOL 35580 24270 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME PURPUROGALLIN PURPUROGALLIN 35582 24271 PSMB7 5695 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL3545432 IXAZOMIB CITRATE 35585 24272 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 404859089 35586 24273 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 385612240 35588 24274 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651388 35589 24275 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200880 DIPHEMANIL METHYLSULFATE 35590 24276 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 328083526 CITARINOSTAT 35593 24277 GCLM 2730 ENZYME SULFORAPHANE SULFORAPHANE 11535546 35594 24278 ATXN2 6311 NA 3,4-METHYLENEDIOXYB-NITROSTYRENE CHEMBL596380 35598 24279 APH1B 83464 PROTEASE, DRUGGABLE GENOME IC261 IC261 20350806 35599 24280 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 375973257 APROCITENTAN 35602 24281 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE RG-1530 RG-1530 35603 24282 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ROBINETIN ROBINETIN 35604 24283 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME FLUNISOLIDE FLUNISOLIDE 35605 24284 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOLVAPTAN TOLVAPTAN 35606 24285 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALPHA 35608 24286 MARK4 57787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DOVITINIB DOVITINIB 35609 24287 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-7f 35610 24288 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CYSTAMINE DIHYDROCHLORIDE CYSTAMINE DIHYDROCHLORIDE 35614 24289 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 3R14S-OCHRATOXIN A 3R14S-OCHRATOXIN A 35615 24290 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-38 35616 24291 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178103973 NIMESULIDE 35617 24292 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME CUDC-101 CUDC-101 35618 24293 CYP27A1 1593 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RETINOID 15340076 35619 24294 NRXN1 9378 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER antipsychotics 35621 24295 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE BMS-754807 BMS-754807 35622 24296 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME ATORVASTATIN ATORVASTATIN 15313180 35625 24297 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BW-373U86 CHEMBL25230 35626 24298 ALOX15 246 ENZYME, DRUGGABLE GENOME LINOLENIC ACID LINOLENIC ACID 35631 24299 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Ado-Trastuzumab Emtansine 35633 24300 HTT 3064 DRUGGABLE GENOME GSK3117391 GSK-3117391 19065135 35634 24301 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545213 BENTAMAPIMOD 35635 24302 FST 10468 DRUGGABLE GENOME NERVE GROWTH FACTOR 9770356 35637 24303 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME eletriptan ELETRIPTAN 35639 24304 TNKS 8658 DRUGGABLE GENOME, ENZYME inhibitor 404859123 35640 24305 PTGS1 5742 ENZYME, DRUGGABLE GENOME MEFENAMIC ACID 35642 24306 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL1536 ERGOCALCIFEROL 35644 24307 HSPA4 3308 NA EPO EPOETIN ALFA 15943180 35646 24308 KCNC3 3748 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL284348 DALFAMPRIDINE 35647 24309 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 1058137-23-7 LUCITANIB 35648 24310 BAZ2B 29994 NA TOLONIUM CHLORIDE TOLONIUM CHLORIDE 35649 24311 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HYDRALAZINE HYDRALAZINE 22931300 35650 24312 MAPT 4137 DRUGGABLE GENOME EMODIN EMODIN 35652 24313 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565894 35653 24314 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME AVOBENZONE AVOBENZONE 35655 24315 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-66209 CHEMBL175266 35656 24316 NCK1 4690 KINASE AX-024 35657 24317 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 3-phenyl isoquinolin-1(2H) derivative 1 35658 24318 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 WAY-100,635 WAY-100,635 35660 24319 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PLATELET FACTOR 4 7790818 35661 24320 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME LEVOFLOXACIN LEVOFLOXACIN 15008519 35662 24321 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PMID29671355-Compound-56 35664 24322 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Pyrazolopyrimidine and thienopyrimidine amide derivative 2 35665 24323 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545267 UMBRALISIB TOSYLATE 35666 24324 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW678313X GW678313X 35667 24325 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME raltitrexed RALTITREXED 11705857 35668 24326 TESK1 7016 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565799 35671 24327 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME TAMATINIB R-406 35672 24328 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 404859101 LICOGLIFLOZIN 35674 24329 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE T-817MA T-817 MALEATE 35675 24330 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME EBSELEN EBSELEN 35676 24331 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor INIPARIB INIPARIB 35677 24332 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME PHENYLSTIBONIC ACID PHENYLSTIBONIC ACID 35678 24333 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE NILE RED NILE RED 35679 24334 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TOMELUKAST TOMELUKAST 35680 24335 ABCC6 368 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER thalidomide THALIDOMIDE 20038957 35681 24336 BLVRA 644 ENZYME Ursodeoxycholic acid 35686 24337 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SANGUINARIUM SANGUINARIUM 35687 24338 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VALRUBICIN VALRUBICIN 35688 24339 CACNB3 784 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ION CHANNEL modulator CHEMBL1628502 GABAPENTIN ENACARBIL 35689 24340 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178100732 35690 24341 TUBB 203068 DRUGGABLE GENOME Verubulin VERUBULIN 35692 24342 SLC1A2 6506 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE 178100898 35696 24343 CA7 766 DRUGGABLE GENOME, ENZYME activator 135651493 HISTAMINE 35697 24344 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Imidazo bicyclic iminium derivative 1 35701 24345 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor ENZASTAURIN ENZASTAURIN 35706 24346 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME rocuronium ROCURONIUM 28409297 35707 24347 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE ADENOSINE DEAMINASE INHIBITOR 11969266 35709 24348 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650837 35710 24349 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-69187 CHEMBL19954 35711 24350 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 178103635 35712 24351 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ART621 PLACULUMAB 35713 24352 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER BROMOCRIPTINE BROMOCRIPTINE 11856485,9514944 35715 24353 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Refametinib REFAMETINIB 26582713 35718 24354 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME nebivolol NEBIVOLOL 35719 24355 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AP32788 35720 24356 ULK3 25989 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE imatinib IMATINIB 15073101 35721 24357 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 178102616 35722 24358 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651565 35723 24359 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ALBUMIN ALBUMIN HUMAN 11246175 35724 24360 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE PEMETREXED PEMETREXED 35725 24361 SMN1 6606 DRUGGABLE GENOME FRENTIZOLE FRENTIZOLE 35726 24362 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER mitomycin MITOMYCIN 35727 24363 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME OXYPHENBUTAZONE OXYPHENBUTAZONE 35728 24364 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-124176 CHEMBL588038 35730 24365 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME Sampatrilat SAMPATRILAT 35731 24366 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE PHYTOESTROGEN 14583453 35732 24367 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 404859135 35735 24368 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 35736 24369 PEMT 10400 ENZYME CHEMBL1742997 CANTUZUMAB MERTANSINE 35737 24370 STN1 79991 ENZYME atenolol ATENOLOL 31327267 35738 24371 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Trametinib TRAMETINIB 26343583,27488531,22983396 35740 24372 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL672 FENOFIBRATE 35741 24373 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TT-100 35742 24374 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME OMEPRAZOLE OMEPRAZOLE 35744 24375 MAPT 4137 DRUGGABLE GENOME AMINOHIPPURIC ACID AMINOHIPPURIC ACID 35746 24376 PREX2 80243 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE VEMURAFENIB VEMURAFENIB 24265155 35748 24377 NAT1 9 ENZYME, DRUGGABLE GENOME thioguanine THIOGUANINE 35749 24378 ATAD5 79915 NA TCMDC-125204 CHEMBL588028 35750 24379 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Methylene Blue 35751 24380 MYB 4602 CLINICALLY ACTIONABLE 5-FLUOROURACIL FLUOROURACIL 15001837 35753 24381 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PLX4720 PLX-4720 25500121,23431193 35754 24382 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AG-808 CHEMBL68534 35755 24383 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL107 COLCHICINE 35757 24384 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE ZNCL2 15596258 35758 24385 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PENTABROMOPHENOL PENTABROMOPHENOL 35759 24386 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME TPKI-48 CHEMBL2333445 22819505 35760 24387 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME EP-42675 35762 24388 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201497 INSULIN GLARGINE 35765 24389 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Cerdulatinib CERDULATINIB 35767 24390 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 187051806 35768 24391 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER RESERPINE RESERPINE 23273047,22148475 35770 24392 POLB 5423 DNA REPAIR, DRUGGABLE GENOME BENZBROMARONE BENZBROMARONE 35772 24393 KCNG1 3755 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107762 NERISPIRDINE 35774 24394 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565692 35777 24395 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CYCLOVALONE CYCLOVALONE 35778 24396 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ECONAZOLE NITRATE ECONAZOLE NITRATE 35779 24397 SMN1 6606 DRUGGABLE GENOME NECROSTATIN NECROSTATIN 35780 24398 RARS1 5917 ENZYME, DRUGGABLE GENOME cisplatin CISPLATIN 27150640 35782 24399 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor VALPROIC ACID DEPAKOTE 35783 24400 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103698 AZELASTINE 35786 24401 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NSC59984 26294215 35789 24402 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME SURAMIN SURAMIN 35791 24403 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR GENISTEIN GENISTEIN 16038533 35792 24404 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE FLAVANONE FLAVANONE 35793 24405 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME GSK-269962A GSK-269962A 35795 24406 ALOX15 246 ENZYME, DRUGGABLE GENOME LEVONORDEFRIN LEVONORDEFRIN 35797 24407 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651283 TROGLITAZONE 35798 24408 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TACEDINALINE TACEDINALINE 18692397 35799 24409 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME activator 178100888 35800 24410 HMGCR 3156 ENZYME, DRUGGABLE GENOME atorvastatin ATORVASTATIN 17563401,18815589,18332269,16103896,20031582,18261733,15199031,26408409 35803 24411 MAP3K7 6885 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565757 CHEMBL1077979 35804 24412 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR CLOFIBRATE CLOFIBRATE 35805 24413 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE FOLFOX 27002107 35806 24414 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist CHEMBL3183409 APALUTAMIDE 35808 24415 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME FLUSPIRILENE FLUSPIRILENE 35812 24416 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME 178103300 35813 24417 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CUDC-907 FIMEPINOSTAT 22693356 35814 24418 TARDBP 23435 TUMOR SUPPRESSOR 3-(PHENYLAMINO)PHENOL CHEMBL1523215 35816 24419 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Dronabinol DRONABINOL 35817 24420 RBP4 5950 DRUGGABLE GENOME A1-10436 35818 24421 COL4A2 1284 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 35819 24422 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 375973260 35820 24423 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 178103872 TADALAFIL 35821 24424 AMH 268 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIETHYLSTILBESTROL DIETHYLSTILBESTROL 2286533 35822 24425 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist 178100606 35825 24426 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW711782X GW711782X 35826 24427 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 THIOPERAMIDE THIOPERAMIDE 35827 24428 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 35829 24429 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9340511, 5 35830 24430 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR ERGOSTEROL PEROXIDE ERGOSTEROL PEROXIDE 22014750 35831 24431 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER elbasvir / grazoprevir 35832 24432 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE TAK-901 TAK-901 35833 24433 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649832 35834 24434 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ETHACRYNIC ACID ETHACRYNIC ACID 35835 24435 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Mepyramine PYRILAMINE 35836 24436 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 348353622 35837 24437 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE INGENOL MEBUTATE 35838 24438 ACE2 59272 ENZYME, TRANSPORTER, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, CELL SURFACE, PROTEASE GSK2586881 GSK-2586881 25893478 35839 24439 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DIHYDROSPINGOSINE DIHYDROSPINGOSINE 35840 24440 RAC2 5880 NA idarubicin IDARUBICIN 28485375 35841 24441 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 astemizole ASTEMIZOLE 15861034 35844 24442 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ANISOTROPINE METHYLBROMIDE 35845 24443 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE PF-04691502 PF-04691502 35846 24444 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 30-NORHEDERAGENIN CHEMBL1081326 19716700 35848 24445 CGA 1081 DRUGGABLE GENOME, HORMONE ACTIVITY IL-18 11712764 35851 24446 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE PAI-1 35856 24447 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650452 35858 24448 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor GEFITINIB GEFITINIB 35859 24449 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RO-09-4889 35860 24450 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ZINC 03369470 CHEMBL599013 35861 24451 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 1096708-71-2 35864 24452 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652451 35865 24453 MAPT 4137 DRUGGABLE GENOME ISOLIQUIRITIGENIN ISOLIQUIRITIGENIN 35866 24454 KDM4A 9682 DRUGGABLE GENOME, ENZYME GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE CHEMBL1255944 35868 24455 TXNRD2 10587 DRUGGABLE GENOME MOTEXAFIN GADOLINIUM 35870 24456 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE NG7 35871 24457 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Crizotinib CRIZOTINIB 35872 24458 APC 324 CLINICALLY ACTIONABLE CGP049090 14749129 35874 24459 IL1B 3553 KINASE, DRUGGABLE GENOME Rilonacept RILONACEPT 35875 24460 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL GSK683699 35877 24461 ATXN2 6311 NA BI-87E7 CHEMBL523200 35878 24462 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CT-P6 28592386 35879 24463 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME VEMURAFENIB VEMURAFENIB 35880 24464 HTT 3064 DRUGGABLE GENOME GNF-PF-3268 CHEMBL582073 35881 24465 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 315661114 MOMETASONE 35883 24466 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ACACETIN DIACETATE ACACETIN DIACETATE 35887 24467 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME vincristine VINCRISTINE 35888 24468 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545216 FX-005 35889 24469 CSMD1 64478 NA oxaliplatin OXALIPLATIN 24444404 35890 24470 ATXN2 6311 NA TCMDC-123869 CHEMBL546597 35892 24471 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CY-208243 CHEMBL313737 35894 24472 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE antibody ADO-TRASTUZUMAB EMTANSINE 35895 24473 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL1200675 TOREMIFENE CITRATE 35897 24474 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE larotrectinib sulfate 35898 24475 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE RECOMBINANT INTERLEUKIN 14960573 35900 24476 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-25 35901 24477 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE infliximab INFLIXIMAB 16720636,16909270,23057546,26244882,12847678,18050183,18713756,19365401,22760475,24192118,17343250,22960943,22129793,25311255,12190096,18438841,17673491,15695296 35903 24478 POLK 51426 DNA REPAIR, ENZYME DIHYDROGAMBOGIC ACID DIHYDROGAMBOGIC ACID 35904 24479 ADAM10 102 ENZYME, CELL SURFACE, TRANSPORTER, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE inhibitor 178103981 ILOMASTAT 35905 24480 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME SPERMINE TRIS-1-NAPG CHEMBL2347632 23434419 35907 24481 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist 404859102 NIDUFEXOR 35908 24482 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SORAFENIB SORAFENIB 35910 24483 TARDBP 23435 TUMOR SUPPRESSOR DNDI1417025 CHEMBL1320453 35913 24484 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE RG7601 VENETOCLAX 35914 24485 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SYM015 35915 24486 SCGB1A1 7356 DRUGGABLE GENOME RHIGF-1 17697625 35916 24487 KDM4A 9682 DRUGGABLE GENOME, ENZYME MALTOL MALTOL 35918 24488 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME GATIFLOXACIN GATIFLOXACIN 35919 24489 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BISINDOLYLMALEIMIDE IX BISINDOLYLMALEIMIDE IX 35921 24490 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE rigosertib RIGOSERTIB 23873848,27104980 35927 24491 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102704 35928 24492 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-11d 35930 24493 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY CTX LORNOXICAM 10067836 35931 24494 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-1 35932 24495 RACGAP1 29127 NA TOLONIUM CHLORIDE TOLONIUM CHLORIDE 35934 24496 KMT2E 55904 ENZYME, METHYL TRANSFERASE duloxetine DULOXETINE 28696415 35935 24497 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME docetaxel DOCETAXEL 27234217 35937 24498 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL1200629 VECURONIUM BROMIDE 35938 24499 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor 252827365 DEUTETRABENAZINE 35939 24500 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PYRONIN Y PYRONIN Y 35940 24501 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NIFUROXAZIDE NIFUROXAZIDE 35941 24502 TUBB3 10381 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 35942 24503 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Nivolumab NIVOLUMAB 27225694,28407039 35943 24504 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor MK2206 MK-2206 35944 24505 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME RITANSERIN RITANSERIN 35946 24506 DHFR 1719 DRUGGABLE GENOME, ENZYME PRALATREXATE PRALATREXATE 35947 24507 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 252166796 35948 24508 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME rucaparib RUCAPARIB 35949 24509 BAZ2B 29994 NA GNF-PF-1644 CHEMBL600734 35951 24510 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE SB-656933 ELUBRIXIN 35952 24511 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME nilotinib NILOTINIB 17611564,24898899 35953 24512 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME pravastatin PRAVASTATIN 10190398 35954 24513 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IRIGINOL HEXAACEATATE IRIGINOL HEXAACEATATE 35955 24514 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR ILORASERTIB ILORASERTIB 35956 24515 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Bb2121 IDECABTAGENE VICLEUCEL 35957 24516 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR GEMCITABINE GEMCITABINE 35958 24517 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL AMLODIPINE AMLODIPINE 35959 24518 IL1A 3552 CELL SURFACE, DRUGGABLE GENOME olanzapine OLANZAPINE 21107309 35963 24519 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TRYPTANTHRIN TRYPTANTHRIN 20373766 35964 24520 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TCMDC-125617 CHEMBL545900 35965 24521 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MHHFJYABEVJNEG-UHFFFAOYSA-N 35966 24522 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW561436X GW561436X 35967 24523 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AT13148 AT-13148 22781553 35968 24524 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565717 35969 24525 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DAUNORUBICIN DAUNORUBICIN 9494516 35970 24526 PTGS2 5743 DRUGGABLE GENOME, ENZYME Darbufelone DARBUFELONE 35973 24527 COL3A1 1281 DRUGGABLE GENOME COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 35974 24528 CD44 960 DRUGGABLE GENOME, CELL SURFACE INTERFERON GAMMA 11369659 35975 24529 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR VORINOSTAT VORINOSTAT 35976 24530 FURIN 5045 ENZYME, PROTEASE, CELL SURFACE, DRUGGABLE GENOME US9266828, B 35977 24531 SMN1 6606 DRUGGABLE GENOME NSC-116702 CHEMBL1477383 35978 24532 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 olanzapine OLANZAPINE 23559402 35981 24533 TOP2B 7155 DRUGGABLE GENOME, ENZYME Aclarubicin ACLARUBICIN 35982 24534 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RHEIN RHEIN 35983 24535 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-123598 CHEMBL547269 35985 24536 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE LY2780301 35986 24537 TLE3 7090 TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR PACLITAXEL PACLITAXEL 35987 24538 PDK2 5164 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 328083464 35988 24539 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR N/A 35989 24540 TOP2B 7155 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL44657 ETOPOSIDE 35990 24541 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 187051805 QUISINOSTAT 35991 24542 MAPT 4137 DRUGGABLE GENOME NORSTICTIC ACID NORSTICTIC ACID 35992 24543 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 315661254 35993 24544 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AV-412 MP-412 35994 24545 ALOX15 246 ENZYME, DRUGGABLE GENOME LUFENURON LUFENURON 35995 24546 ADH1B 125 DRUGGABLE GENOME, ENZYME ethanol ALCOHOL 16571603,15902904,23240771,32451486 35996 24547 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME DIETHYL-2-UNDECYLIDENEMALONATE CHEMBL1797707 21292492 35997 24548 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-46 35998 24549 EWSR1 2130 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SUNITINIB SUNITINIB 24703573 36000 24550 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor TEMSIROLIMUS TEMSIROLIMUS 36001 24551 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BI-44370 TA 36002 24552 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor VORINOSTAT VORINOSTAT 36003 24553 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PHA-767491 CHEMBL225519 36005 24554 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE LINIFANIB LINIFANIB 36006 24555 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor ALVOCIDIB ALVOCIDIB 36007 24556 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 223365911 EDOXABAN 36008 24557 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Pyridino tricyclic compound 1 36010 24558 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE HYDROCODONE HYDROCODONE 36011 24559 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor CHEMBL3545001 MK-8353 36012 24560 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE GNF-PF-992 CHEMBL602561 36014 24561 POLI 11201 DNA REPAIR PHYSODIC ACID PHYSODIC ACID 36015 24562 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650996 36016 24563 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor 354702258 DERAZANTINIB 36017 24564 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650856 PROPAFENONE 36018 24565 ATAD5 79915 NA HARMINE HYDROCHLORIDE HARMINE HYDROCHLORIDE 36020 24566 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BRILLIANT GREEN OXALATE BRILLIANT GREEN OXALATE 36021 24567 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1671 PROPRANOLOL HYDROCHLORIDE 36023 24568 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 53801057 NIMODIPINE 36024 24569 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL EVT-201 36025 24570 SMN2 6607 DRUGGABLE GENOME CID2350207 CHEMBL259615 36028 24571 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HYDROCORTISONE SODIUM PHOSPHATE HYDROCORTISONE SODIUM PHOSPHATE 36029 24572 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Dexamethasone sodium phosphate 36031 24573 CDK12 51755 KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR, SERINE THREONINE KINASE Cemiplimab CEMIPLIMAB 36033 24574 ATXN2 6311 NA TCMDC-124032 CHEMBL536375 36034 24575 CA9 768 DRUGGABLE GENOME, ENZYME Sulfonamide-thiadiazole derivative 2 36035 24576 PSMB10 5699 PROTEASE, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 24524217 36036 24577 GMNN 51053 DRUGGABLE GENOME TDR77578 CHEMBL1364172 36037 24578 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-13 36038 24579 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DOPAMINE DOPAMINE 36039 24580 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651590 DENUFOSOL 36040 24581 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME CARBOPLATIN CARBOPLATIN 12168940 36041 24582 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 METYROSINE METYROSINE 22931300 36043 24583 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR HYPERBARIC OXYGEN 12515318 36045 24584 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL568 OXAZEPAM 36047 24585 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TCMDC-123730 CHEMBL530280 36050 24586 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4674 CHEMBL584452 36051 24587 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL744 RILUZOLE 36056 24588 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RAC-NUTLIN-3 CHEMBL211045 36058 24589 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CHR-3996 NANATINOSTAT 36061 24590 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME PTHRP 11136536 36063 24591 TSPO 706 DRUGGABLE GENOME Indole-based analog 10 36064 24592 TUBB2B 347733 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 36065 24593 BAZ2B 29994 NA EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 36067 24594 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Aryl carbamate analog 1 36069 24595 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SJ000118780 CHEMBL591836 36070 24596 HSPB1 3315 DRUGGABLE GENOME E-GUGGULSTERONE E-GUGGULSTERONE 36071 24597 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CLOBAZAM CLOBAZAM 36072 24598 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME POSIPHEN PHENSERINE, (+)- 36073 24599 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE TOZASERTIB TOZASERTIB 36074 24600 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135650016 36075 24601 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200990 FLURBIPROFEN SODIUM 36077 24602 ATAD5 79915 NA THIOINOSINE THIOINOSINE 36078 24603 PRKCH 5583 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE INGENOL MEBUTATE 36079 24604 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GESTODENE GESTODENE 36080 24605 CA12 771 DRUGGABLE GENOME ACETAZOLAMIDE ACETAZOLAMIDE 36081 24606 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME Antihypertensives 18425130,21127457 36082 24607 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE LINIFANIB LINIFANIB 36085 24608 DNER 92737 NA Isoxazole-based bicyclic compound 5 36086 24609 RGS4 5999 DRUGGABLE GENOME URIDINE-5'-MONOPHOSPHATE CHEMBL214393 36087 24610 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER montelukast MONTELUKAST 36088 24611 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLOROTRIPHENYLSTANNANE CHLOROTRIPHENYLSTANNANE 36089 24612 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ISOPRENALINE ISOPROTERENOL 36090 24613 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE TAI-GPC3-CART cells 36095 24614 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHEMBL1257 ENFLURANE 36096 24615 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AZAKENPAULLONE AZAKENPAULLONE 36097 24616 UGT2B7 7364 DRUGGABLE GENOME losartan LOSARTAN 36098 24617 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME V3381 INDANTADOL 36099 24618 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200328 DULOXETINE HYDROCHLORIDE 36100 24619 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650146 36102 24620 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME XmAb13676 PLAMOTAMAB 36103 24621 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650903 RISPERIDONE 36108 24622 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE Peptide analog 61 36109 24623 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PF-06463922 LORLATINIB 36110 24624 NOS1 4842 DRUGGABLE GENOME, ENZYME PENICILLIN PENICILLIN G POTASSIUM 11367745 36111 24625 CTSD 1509 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166874 36112 24626 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE BAF 10217271 36113 24627 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Dacomitinib DACOMITINIB 36114 24628 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE PD-98059 CHEMBL35482 11031257 36116 24629 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200323 LABETALOL HYDROCHLORIDE 36117 24630 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SP-600125 SP-600125 36118 24631 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-acylpyrrolidine ether derivative 1 36119 24632 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CARBETAPENTANE CARBETAPENTANE 36120 24633 PML 5371 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TAMIBAROTENE TAMIBAROTENE 30289902 36122 24634 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1166 ARGATROBAN 36123 24635 XDH 7498 DRUGGABLE GENOME, ENZYME RICIN 8624583 36125 24636 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL75133 IRX-4204 36126 24637 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME ANDROSTENEDIONE ANDROSTENEDIONE 8907816 36129 24638 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FLUPIRTINE MALEATE FLUPIRTINE MALEATE 36130 24639 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PURPUROGALLIN PURPUROGALLIN 36131 24640 BAZ2B 29994 NA OXYTETRACYCLINE OXYTETRACYCLINE 36134 24641 GMNN 51053 DRUGGABLE GENOME SJ000114741 CHEMBL591370 36135 24642 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROPICONAZOLE PROPICONAZOLE 36136 24643 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TCMDC-125785 CHEMBL588525 36139 24644 RGS4 5999 DRUGGABLE GENOME inhibitor 249565714 36143 24645 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-43 36144 24646 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME TINZAPARIN TINZAPARIN 36145 24647 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor X-82 X-82 36148 24648 RIPK3 11035 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 384403668 36149 24649 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME TCDD 15459018 36150 24650 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GNF-PF-2893 CHEMBL312032 36152 24651 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE URSOLIC ACID URSOLIC ACID 21453996 36153 24652 NFKBIA 4792 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME GAMBOGIC ACID GAMBOGIC ACID 22472167 36155 24653 GMNN 51053 DRUGGABLE GENOME DNDI1417529 CHEMBL1990783 36156 24654 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651563 36158 24655 ATAD5 79915 NA TYRPHOSTIN A9 TYRPHOSTIN A9 36159 24656 HYAL2 8692 DRUGGABLE GENOME, CELL SURFACE DEXAMETHASONE DEXAMETHASONE 212383 36161 24657 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Nilotinib NILOTINIB 36162 24658 PSCA 8000 DRUGGABLE GENOME CAR-T cells targeting PSCA 36163 24659 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE rituximab RITUXIMAB 19018870,26167726,23505228,30457672,12975461,16609067 36164 24660 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2013009582Example16 36167 24661 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER lithium LITHIUM 21449676 36169 24662 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 (S)-AMPA (S)-AMPA 36170 24663 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SULFINPYRAZONE SULFINPYRAZONE 36172 24664 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Meprednisone MEPREDNISONE 36174 24665 RRM2 6241 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2105467 TEZACITABINE 36177 24666 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL GABAPENTIN GABAPENTIN 36178 24667 E2F1 1869 TRANSCRIPTION FACTOR RAS INHIBITORS 16496386 36179 24668 CDC42 998 DRUGGABLE GENOME ZU-0073945 CHEMBL563777 19527032 36180 24669 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME hydroxyamitriptyline 36181 24670 TAGLN 6876 NA TGFBETA1 16876108 36182 24671 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 23622981 36184 24672 PSMD13 5719 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 36185 24673 FTO 79068 ENZYME ribavirin RIBAVIRIN 25367448 36188 24674 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME BUSULFAN BUSULFAN 7742532 36190 24675 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor PF-4217903 PF-04217903 36191 24676 ATAD5 79915 NA TRANILAST TRANILAST 36192 24677 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 405067335 36193 24678 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR APD-811 RALINEPAG 21687516 36196 24679 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ESTRADIOL ACETATE 36199 24680 FCGR2A 2212 CLINICALLY ACTIONABLE, DRUGGABLE GENOME rituximab RITUXIMAB 30457672 36201 24681 CSF3 1440 GROWTH FACTOR, DRUGGABLE GENOME MK-4214 36202 24682 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 404859096 36203 24683 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201613 INSULIN GLULISINE 36204 24684 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-108 CHEMBL578929 36205 24685 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL NITRAZEPAM NITRAZEPAM 36207 24686 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE CIS-RESVERATROL CIS-RESVERATROL 36208 24687 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 36211 24688 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME ANTIHEMOPHILIC FACTOR 36213 24689 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME NISOLDIPINE NISOLDIPINE 36214 24690 RGS4 5999 DRUGGABLE GENOME DAPH DAPH 36216 24691 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102548 ALSTERPAULLONE 36218 24692 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 135650177 DICLOFENAC 36219 24693 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE DNDI1417156 CHEMBL1504679 36220 24694 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME BENZOQUINONE BENZOQUINONE 36222 24695 GHRL 51738 DRUGGABLE GENOME PLANT STEROLS 18066136 36224 24696 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-60339 CHEMBL1448793 36227 24697 PLD1 5337 ENZYME, DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 19136975 36228 24698 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE DDTC 9726816 36230 24699 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR AMPICILLIN AMPICILLIN 9931456 36231 24700 HDAC11 79885 DRUGGABLE GENOME, ENZYME ENTINOSTAT ENTINOSTAT 19966789,20491440 36232 24701 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL2103852 CROLIBULIN 36233 24702 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-17 36235 24703 FST 10468 DRUGGABLE GENOME BICALUTAMIDE BICALUTAMIDE 14761877 36237 24704 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FINASTERIDE FINASTERIDE 36238 24705 BAP1 8314 PROTEASE, TUMOR SUPPRESSOR, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE SUNITINIB SUNITINIB 27751729 36240 24706 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TAFA-93 36243 24707 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GOSSYPOL GOSSYPOL 36245 24708 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-123713 CHEMBL586135 36246 24709 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME TAK-632 27523909 36247 24710 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VER-49009 CHEMBL365617 36249 24711 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme4Bottom 36250 24712 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME CHEMBL3707253 BEVACIZUMAB 111IN 36252 24713 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME leucovorin LEUCOVORIN 36253 24714 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME BAICALEIN BAICALEIN 36254 24715 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL856 PRIMIDONE 36256 24716 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GNF-PF-159 CHEMBL599924 36257 24717 SMARCB1 6598 CLINICALLY ACTIONABLE Vorinostat VORINOSTAT 23764045 36259 24718 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME FENTICLOR FENTICLOR 36261 24719 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME OSM-S-85 CHEMBL1494650 36263 24720 CA1 759 DRUGGABLE GENOME, ENZYME CG100649 POLMACOXIB 36265 24721 CXCL2 2920 DRUGGABLE GENOME BB-94 BATIMASTAT 18477053 36266 24722 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE NILOTINIB NILOTINIB 26703895 36272 24723 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHYTANIC ACID PHYTANIC ACID 20695472 36273 24724 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200463 OXAPROZIN POTASSIUM 36275 24725 DHODH 1723 DRUGGABLE GENOME, ENZYME LAS-186323 36276 24726 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR RESVERATROL RESVERATROL 36277 24727 NDUFB2 4708 ENZYME inhibitor CHEMBL3545320 ME-344 36278 24728 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 178103206 EFALIZUMAB 36279 24729 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565856 36281 24730 SMN1 6606 DRUGGABLE GENOME AMIKACIN AMIKACIN 15790598 36286 24731 CCNA2 890 DRUGGABLE GENOME, KINASE SURAMIN SURAMIN 10208280 36288 24732 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (-)-U-50488 (-)-U-50488 36289 24733 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 328083455 36290 24734 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME TROFOSFAMIDE TROFOSFAMIDE 10447581 36291 24735 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-3515 CHEMBL602365 36293 24736 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE EPTIFIBATIDE EPTIFIBATIDE 36295 24737 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LY3381916 36297 24738 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL inhibitor 223365904 36298 24739 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL289351 FOSBRETABULIN DISODIUM 36299 24740 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 idarubicin IDARUBICIN 22584460 36300 24741 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-asCEBP-1 36301 24742 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME METYROSINE METYROSINE 22931300 36304 24743 TARDBP 23435 TUMOR SUPPRESSOR N-(4-FLUOROBENZYLCARBAMOTHIOYL)BENZAMIDE CHEMBL1545737 36305 24744 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor 252827493 36306 24745 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PT-102 CHEMBL317356 36307 24746 ELN 2006 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PRT-201 VONAPANITASE 36310 24747 ALOX5 240 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL93 ZILEUTON 36311 24748 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE SORAFENIB SORAFENIB 36314 24749 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor PD 0332991 36316 24750 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102921 36318 24751 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CADMIUM DICHLORIDE CADMIUM DICHLORIDE 36321 24752 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER mycophenolate mofetil 18444945 36322 24753 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE LY2874455 LY-2874455 36326 24754 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME ZINC 03369470 CHEMBL599013 36328 24755 KDM4A 9682 DRUGGABLE GENOME, ENZYME FASUDIL HYDROCHLORIDE FASUDIL HYDROCHLORIDE 36329 24756 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TREPROSTINIL TREPROSTINIL 36330 24757 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE TENOFOVIR TENOFOVIR 17172311 36332 24758 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GW7074 CHEMBL72365 36334 24759 SMN1 6606 DRUGGABLE GENOME JNJ-16259685 CHEMBL174588 36335 24760 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL679 EPINEPHRINE 36336 24761 ALOX5 240 DRUGGABLE GENOME, ENZYME Silymarin SILYBIN A 36340 24762 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1200377 AMPHETAMINE ASPARTATE 36341 24763 KDM4A 9682 DRUGGABLE GENOME, ENZYME PYRAZINOIC ACID PYRAZINOIC ACID 36343 24764 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER HOMIDIUM BROMIDE HOMIDIUM BROMIDE 36344 24765 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ZAPRINAST ZAPRINAST 36345 24766 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL3833330 CINPANEMAB 36346 24767 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PATULIN PATULIN 16680159 36347 24768 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 178102324 NILOTINIB 36350 24769 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL1967878 CENISERTIB 36351 24770 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIHYDROGAMBOGIC ACID DIHYDROGAMBOGIC ACID 36352 24771 HSPA8 3312 TUMOR SUPPRESSOR inhibitor CHEMBL2105726 36353 24772 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE REMIFENTANIL REMIFENTANIL 36354 24773 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 36355 24774 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL552212 LEXIBULIN 36356 24775 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME SCUTELLARIN SCUTELLARIN 22822035 36358 24776 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545088 PUQUITINIB 36359 24777 RAPGEF3 10411 ENZYME DAPHNORETIN DAPHNORETIN 36361 24778 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL207197 OLCEGEPANT 36362 24779 LTF 4057 CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, PROTEASE RESERPINE RESERPINE 3608900 36365 24780 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME 3,4-DICHLOROISOCOUMARIN CHEMBL24983 36368 24781 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME Lusutrombopag LUSUTROMBOPAG 36370 24782 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE CHEMBL201325 36371 24783 MAOB 4129 DRUGGABLE GENOME, ENZYME Budipine BUDIPINE 36373 24784 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Contusugene ladenovec 36374 24785 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL2109224 ROVELIZUMAB 36375 24786 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GOSSYPETIN GOSSYPETIN 36377 24787 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PROSTAGLANDIN D2 PROSTAGLANDIN D2 23566516 36378 24788 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135651327 36379 24789 TUBB 203068 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 36382 24790 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-J5 36383 24791 NOS2 4843 DRUGGABLE GENOME, ENZYME ISOTHIOUREA 36384 24792 ALOX15B 247 DRUGGABLE GENOME, ENZYME BITHIONOL BITHIONOL 36385 24793 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME 3-amino-5-benzyl-substituted indazole derivative 1 36386 24794 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 36387 24795 ATAD5 79915 NA 7-METHOXY-BAPTIGENIN CHEMBL583578 36389 24796 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178103084 BIVALIRUDIN 36391 24797 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 385612227 36392 24798 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR EMODIC ACID EMODIC ACID 36394 24799 SMN2 6607 DRUGGABLE GENOME NSC-93401 CHEMBL452954 36395 24800 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE sertraline SERTRALINE 18695978 36396 24801 PTGS2 5743 DRUGGABLE GENOME, ENZYME Ibuprofen IBUPROFEN 36397 24802 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 2-(STYRYL)-BENZIMIDAZOLE CHEMBL473721 36400 24803 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Acrivastine ACRIVASTINE 36401 24804 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Panitumumab PANITUMUMAB 26843189,17664472,22270724,27312529 36402 24805 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME 5,7,3',5'-TETRAHYDROXYFLAVANONE CHEMBL307893 36403 24806 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PIRENOXINE PIRENOXINE 36404 24807 SMN1 6606 DRUGGABLE GENOME 7,2'-DIHYDROXYFLAVONE CHEMBL475908 36405 24808 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 252827463 36406 24809 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME DASATINIB DASATINIB 19462975,25835317 36407 24810 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 328083456 36408 24811 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor FORETINIB FORETINIB 36409 24812 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME EPINEPHRINE EPINEPHRINE 36410 24813 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ISOBOLDINE ISOBOLDINE 36411 24814 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME CYC-116 CYC-116 36412 24815 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME ESTAZOLAM ESTAZOLAM 36414 24816 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE blinatumomab BLINATUMOMAB 36415 24817 MAPT 4137 DRUGGABLE GENOME OBTUSAQUINONE OBTUSAQUINONE 36417 24818 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL DIAZEPAM DIAZEPAM 36418 24819 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME antagonist LCL161 LCL-161 36420 24820 TAT 6898 ENZYME PREDNISOLONE PREDNISOLONE 6127207 36421 24821 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME REL-CARINATIN D CHEMBL2332128 36422 24822 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VITAMIN E 17029404 36425 24823 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3544956 PYROTINIB 36426 24824 UGCG 7357 ENZYME, DRUGGABLE GENOME ELIGLUSTAT ELIGLUSTAT 36427 24825 CCR7 1236 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR agonist 135651663 36428 24826 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545236 BPI-9016 36429 24827 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Aurora Kinase Inhibitor II 26842935 36431 24828 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PYRANTEL PAMOATE PYRANTEL PAMOATE 36432 24829 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DERRUBONE DERRUBONE 36434 24830 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME PF-562271 PF-00562271 36435 24831 MAPT 4137 DRUGGABLE GENOME OLEOYL DOPAMINE OLEOYL DOPAMINE 36437 24832 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE EGCG EPIGALOCATECHIN GALLATE 11936850 36438 24833 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PYRROLIDINE DITHIOCARBAMATE PYRROLIDINE DITHIOCARBAMATE 36439 24834 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-236687 CHEMBL318892 36440 24835 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist 178101665 36442 24836 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125788 CHEMBL529986 36444 24837 GGPS1 9453 DRUGGABLE GENOME, ENZYME ZOLEDRONATE ZOLEDRONIC ACID 36445 24838 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TAE-684 TAE-684 36446 24839 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CHEMBL1102 GLUTETHIMIDE 36449 24840 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200982 BUTABARBITAL SODIUM 36450 24841 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PMID27376512-Compound-MTC-422 36451 24842 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME cyclophosphamide CYCLOPHOSPHAMIDE 27234217 36452 24843 PRKAG2 51422 ENZYME, KINASE hydrochlorothiazide HYDROCHLOROTHIAZIDE 31327267 36453 24844 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME SHIKONIN SHIKONIN 36454 24845 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DIETHYLDITHIOCARBAMATE DITIOCARB 17052849 36455 24846 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-78 CHEMBL579318 36456 24847 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME Dersalazine DERSALAZINE 21790535 36457 24848 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 5-(4-PHENYLBUTOXY)PSORALEN CHEMBL1256851 36458 24849 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NITROSCANATE NITROSCANATE 36459 24850 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME chlorpromazine CHLORPROMAZINE 8739822 36460 24851 IFNGR2 3460 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Interferon gamma-1b 36461 24852 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 10 36466 24853 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650178 DICYCLOMINE 36467 24854 DHFR 1719 DRUGGABLE GENOME, ENZYME methotrexate METHOTREXATE 25084201,19648163,25778468,19902562,21747412,19861437,26335211 36469 24855 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135649663 36470 24856 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-42 36471 24857 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR METHYLPREDNISOLONE METHYLPREDNISOLONE 14966352 36474 24858 NUDT15 55270 ENZYME, CLINICALLY ACTIONABLE AZATHIOPRINE AZATHIOPRINE 26878724 36475 24859 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 22 36476 24860 KDM4A 9682 DRUGGABLE GENOME, ENZYME Selenium compound 3 36477 24861 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166899 VERUBECESTAT 36478 24862 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE CNS-5161 CNS-5161 36479 24863 CHRNA5 1138 DRUGGABLE GENOME, ION CHANNEL partial agonist CHEMBL127071 POZANICLINE 36481 24864 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR BRYOSTATIN-1 36483 24865 ATAD5 79915 NA DNDI1417300 CHEMBL1401091 36484 24866 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 329968395 36485 24867 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inotuzumab ozogamicin 36486 24868 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Duvelisib DUVELISIB 36487 24869 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME NAPHMETHONIUM NAPHMETHONIUM 25051097 36488 24870 CD276 80381 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME 124I-8H9 36489 24871 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME HTS-05058 CHEMBL261692 36492 24872 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CD20-Specific CAR T Cells 36494 24873 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME IFN 16140920 36495 24874 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C4 36496 24875 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX LANATOSIDE C LANATOSIDE C 36497 24876 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CID 27456 CHEMBL1708510 21950657 36499 24877 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR peginterferon alfa-2a 25713999 36501 24878 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR HGS1029 36503 24879 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE FASUDIL FASUDIL 36504 24880 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417072 CHEMBL1310701 36506 24881 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor GDC-0980 APITOLISIB 36507 24882 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME CYC116 36509 24883 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE terazosin TERAZOSIN 18695978 36510 24884 NR2F2 7026 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CYCLOHEXIMIDE CYCLOHEXIMIDE 36511 24885 GMNN 51053 DRUGGABLE GENOME WOGONIN WOGONIN 36512 24886 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE LOVASTATIN LOVASTATIN 8663292 36514 24887 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME METOLAZONE METOLAZONE 36515 24888 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651538 36516 24889 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE LEE011 RIBOCICLIB 36517 24890 TOP2B 7155 DRUGGABLE GENOME, ENZYME AMONAFIDE AMONAFIDE 36518 24891 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME arteether 36519 24892 DDAH1 23576 ENZYME 2-ETHYL-BENZIMIDAZOLE CHEMBL351569 22921743 36520 24893 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CLIOQUINOL CLIOQUINOL 36521 24894 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE DIPYRIDAMOLE DIPYRIDAMOLE 36522 24895 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Fostamatinib FOSTAMATINIB 22237022 36523 24896 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NAVEGLITAZAR NAVEGLITAZAR 36524 24897 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME Diaryl amine derivative 2 36525 24898 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME modulator CHEMBL3545020 MBX-2044 36526 24899 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 178103303 36529 24900 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CLOCORTOLONE PIVALATE CLOCORTOLONE PIVALATE 36530 24901 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BYL719 ALPELISIB 36531 24902 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DL-CATECHIN TRIHYDRATE CHEMBL1172228 36532 24903 ALDH1A1 216 DRUGGABLE GENOME, ENZYME P-CYANOCHALCONE CHEMBL445153 36533 24904 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL antagonist 178100925 36538 24905 RACGAP1 29127 NA THUNBERGINOL A THUNBERGINOL A 36540 24906 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME PEMETREXED PEMETREXED 26317331,21879757 36541 24907 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE GAMBOGIC AMIDE GAMBOGIC AMIDE 17911251 36542 24908 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AFATINIB AFATINIB 23930994,24565969 36543 24909 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Aminopyrimidine derivative 9 36544 24910 POLB 5423 DNA REPAIR, DRUGGABLE GENOME EDGEWORIN EDGEWORIN 18343122 36545 24911 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BUNAMIDINE HYDROCHLORIDE BUNAMIDINE HYDROCHLORIDE 36546 24912 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1200760 BALSALAZIDE DISODIUM 36547 24913 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 249565841 36549 24914 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX INDOPROFEN INDOPROFEN 36550 24915 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL443684 NAVITOCLAX 36552 24916 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE TETRAHYDROURIDINE TETRAHYDROURIDINE 17296311 36555 24917 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE CYC-116 CYC-116 36556 24918 ALPL 249 ENZYME, DRUGGABLE GENOME NSC-234945 CHEMBL260311 36558 24919 RGS4 5999 DRUGGABLE GENOME PHLORETIN PHLORETIN 36559 24920 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SEMAXANIB SEMAXANIB 36560 24921 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME IFOSFAMIDE IFOSFAMIDE 16282887 36561 24922 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-18 36562 24923 PDE4A 5141 DRUGGABLE GENOME, ENZYME MILRINONE MILRINONE 36563 24924 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DICHLOROPHEN DICHLOROPHEN 36564 24925 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Imidazolidine derivative 1 36565 24926 B2M 567 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PEMBROLIZUMAB PEMBROLIZUMAB 27433843 36567 24927 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME OXYTETRACYCLINE OXYTETRACYCLINE 36570 24928 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2-MERCAPTOBENZOTHIAZOLE 2-MERCAPTOBENZOTHIAZOLE 36571 24929 ALOX15B 247 DRUGGABLE GENOME, ENZYME CHELERYTHRINE CHELERYTHRINE 36572 24930 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TAMATINIB R-406 36575 24931 NDUFA11 126328 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 36576 24932 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SJ000066481 CHEMBL588749 36578 24933 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TRIAMCINOLONE TRIAMCINOLONE 36580 24934 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE entrectinib ENTRECTINIB 36581 24935 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103140 36582 24936 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME MORAb-009 AMATUXIMAB 36583 24937 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL3545179 AZD-7451 36584 24938 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Carboplatin CARBOPLATIN 28514312 36585 24939 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR 681640 CHEMBL379975 36586 24940 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TAE-684 TAE-684 36589 24941 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Nivolumab NIVOLUMAB 26645196 36590 24942 ALPI 248 DRUGGABLE GENOME, ENZYME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 36591 24943 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROMETHAZINE HYDROCHLORIDE PROMETHAZINE HYDROCHLORIDE 36592 24944 LIPA 3988 ENZYME, DRUGGABLE GENOME LOVASTATIN LOVASTATIN 11380065 36593 24945 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME VARESPLADIB VARESPLADIB 36594 24946 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565818 36595 24947 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME WR-243246 CHEMBL117217 36596 24948 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CLEMASTINE CLEMASTINE 36597 24949 RGS4 5999 DRUGGABLE GENOME DIAMIDE DIAMIDE 36598 24950 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL272621 HYODEOXYCHOLIC_ACID 36600 24951 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR RALOXIFENE RALOXIFENE 36601 24952 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING MGCD-0103 MOCETINOSTAT 36602 24953 PTGS2 5743 DRUGGABLE GENOME, ENZYME INDOMETHACIN INDOMETHACIN 36603 24954 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DIHYDROTANSHINONE I DIHYDROTANSHINONE I 26339922 36604 24955 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER MARIJUANA 16439618 36605 24956 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LXR-623 LXR-623 20350005 36606 24957 BCHE 590 DRUGGABLE GENOME, ENZYME SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 36607 24958 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME (+)-EPITAXIFOLIN (+)-EPITAXIFOLIN 36609 24959 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HYDROCORTISONE PROBUTATE HYDROCORTISONE PROBUTATE 36610 24960 TNFAIP3 7128 PROTEASE, ENZYME, CLINICALLY ACTIONABLE, KINASE methotrexate METHOTREXATE 20921970 36611 24961 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME IPILIMUMAB IPILIMUMAB 26095797 36612 24962 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE NU7441 23761041 36615 24963 TSPO 706 DRUGGABLE GENOME Quinazoline derivative 3 36616 24964 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 187051803 36617 24965 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR CLOSANTEL CLOSANTEL 36618 24966 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 363894214 SITRAVATINIB 36619 24967 MGAT2 4247 ENZYME Bicyclic pyrimidine derivative 1 36622 24968 TH 7054 ENZYME, DRUGGABLE GENOME Tetrahydrobiopterin SAPROPTERIN 36623 24969 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW779439X GW779439X 36624 24970 RGS4 5999 DRUGGABLE GENOME PROPENTOFYLLINE PROPENTOFYLLINE 36625 24971 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178103994 DACOMITINIB 36627 24972 GJB6 10804 ION CHANNEL inhibitor 135650269 36629 24973 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL675 ALENDRONATE SODIUM 36630 24974 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AG-555 CHEMBL53898 36631 24975 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE MITONAFIDE MITONAFIDE 36635 24976 ATP2C1 27032 ENZYME, TRANSPORTER, DRUGGABLE GENOME ISOFLURANE ISOFLURANE 36636 24977 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VANIPREVIR VANIPREVIR 19841155 36637 24978 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651254 THEOPHYLLINE 36641 24979 MPHOSPH8 54737 NA DEQUALINIUM CHLORIDE DEQUALINIUM CHLORIDE 36642 24980 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE example 98 (WO2011020806) 36644 24981 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Cyclopropyl-spiro piperidine derivative 2 36645 24982 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME losartan LOSARTAN 36646 24983 APH1B 83464 PROTEASE, DRUGGABLE GENOME UNII-DRL23N424R 36648 24984 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AVI-4557 36649 24985 POLB 5423 DNA REPAIR, DRUGGABLE GENOME N-BENZOYLANTHRANILIC ACID CHEMBL198666 36650 24986 GMNN 51053 DRUGGABLE GENOME TCMDC-124518 CHEMBL527584 36651 24987 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor IMATINIB IMATINIB 36652 24988 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME CHEMBL3833393 EMICIZUMAB 36653 24989 USP5 8078 ENZYME, PROTEASE VIALININ A VIALININ A 23791076 36654 24990 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL592054 IMIGLITAZAR 36656 24991 NOS1 4842 DRUGGABLE GENOME, ENZYME inhibitor 252827417 36658 24992 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178100981 36659 24993 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GM-CSF REGRAMOSTIM 11591765 36660 24994 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR HEPARIN HEPARIN 36663 24995 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-PG-11047 36664 24996 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Lmw heparin 36666 24997 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE KAMEBANIN KAMEBANIN 36667 24998 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DOCUSATE DOCUSATE 36668 24999 RACGAP1 29127 NA DNDI1417884 CHEMBL1346025 36670 25000 TXK 7294 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 318164804 36673 25001 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR CHEMOSENSITIZER 8620409 36675 25002 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MIZORIBINE MIZORIBINE 36676 25003 TSPO 706 DRUGGABLE GENOME Imidazopyridine acetamide analog 2 36679 25004 ABCC9 10060 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER Repaglinide REPAGLINIDE 36680 25005 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200762 BETAMETHASONE SODIUM PHOSPHATE 36681 25006 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652513 36682 25007 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1726 NISOLDIPINE 36683 25008 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TYRPHOSTIN 25 TYRPHOSTIN 25 36684 25009 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME HEPARAN SULFATE 18499669 36685 25010 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR DOVITINIB DOVITINIB 36686 25011 RGS4 5999 DRUGGABLE GENOME 5-HYDROXYFLAVONE 5-HYDROXYFLAVONE 36688 25012 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme25-4 36689 25013 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-US20120277229 39(1.1) 36690 25014 C1S 716 ENZYME, PROTEASE, DRUGGABLE GENOME Cinryze CINRYZE 36691 25015 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 2-((4-(DIMETHYLAMINO)PHENYL)DIAZENYL)BENZOIC ACID CHEMBL375971 36692 25016 TH 7054 ENZYME, DRUGGABLE GENOME TETRAHYDROBIOPTERIN SAPROPTERIN 36693 25017 HTT 3064 DRUGGABLE GENOME GNF-PF-1919 CHEMBL576409 36694 25018 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650681 NALMEFENE 36696 25019 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE POLIDOCANOL POLIDOCANOL 36697 25020 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE TASELISIB TASELISIB 26589432 36699 25021 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200773 TOCAINIDE HYDROCHLORIDE 36700 25022 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR EPHEDRINE EPHEDRINE 36705 25023 HLA-DQA1 3117 CLINICALLY ACTIONABLE Lapatinib LAPATINIB 36711 25024 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Myo-inositol 36712 25025 RAB9A 9367 ENZYME, DRUGGABLE GENOME ROEMERINE ROEMERINE 36713 25026 FMO5 2330 ENZYME, DRUGGABLE GENOME metformin METFORMIN 26306225 36714 25027 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME THROMBIN THROMBIN 2119237 36716 25028 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME TPN 8443268 36722 25029 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MUSCARINE MUSCARINE 36723 25030 SMN2 6607 DRUGGABLE GENOME 6,4'-DIMETHOXYFLAVONE 6,4'-DIMETHOXYFLAVONE 36728 25031 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LANSOPRAZOLE LANSOPRAZOLE 36730 25032 SMN2 6607 DRUGGABLE GENOME DNDI1416988 CHEMBL1389794 36732 25033 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE ZILEUTON ZILEUTON 24074025 36733 25034 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE NSC348884 21719597 36734 25035 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 178102672 36735 25036 MARCHF8 220972 ENZYME H5N1 influenza vaccine 36736 25037 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL TEZAMPANEL TEZAMPANEL 36737 25038 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE WX-671 UPAMOSTAT 36738 25039 MUC16 94025 DRUGGABLE GENOME CYCLOSPORINE CYCLOSPORINE 12169874 36739 25040 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME LY-2090314 LY-2090314 36741 25041 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL2443262 OLICERIDINE 36742 25042 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE TAMATINIB R-406 36743 25043 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200613 TOLMETIN SODIUM 36745 25044 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE calcein 22027652 36747 25045 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AMOXICILLIN AMOXICILLIN 22931300 36748 25046 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor CHEMBL3137331 DEFACTINIB 36749 25047 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME ACNU 1518162 36750 25048 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME E7090 E-7090 27535969,7506125 36751 25049 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Belinostat BELINOSTAT 36752 25050 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Ixabepilone IXABEPILONE 26864210 36753 25051 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME COCAINE COCAINE 36754 25052 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor EVEROLIMUS EVEROLIMUS 36756 25053 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Docetaxel DOCETAXEL 36758 25054 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565697 36759 25055 PDF 64146 DRUGGABLE GENOME Trimetrexate TRIMETREXATE 36762 25056 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DOPAMINE DOPAMINE 36763 25057 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME OSI-632 OSI-632 36764 25058 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 6,7-ADTN HYDROBROMIDE CHEMBL1255656 36767 25059 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME RITUXIMAB RITUXIMAB 36768 25060 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME RG-1530 RG-1530 36769 25061 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX DIOSMETIN DIOSMETIN 25190466 36771 25062 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME MDX-1411 MDX-1411 36774 25063 LNPEP 4012 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, TRANSPORTER, PROTEASE US10059720, Example 80 36775 25064 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 223365978 AEE-788 36777 25065 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor BKM120 BUPARLISIB 36778 25066 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3,3'-DIMETHOXYBENZIDINE CHEMBL398363 36779 25067 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SALMETEROL XINAFOATE SALMETEROL XINAFOATE 36780 25068 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYSTEINE METHYL-ESTER HCL CHEMBL1426508 36781 25069 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545297 PEXMETINIB 36784 25070 SLC16A7 9194 DRUGGABLE GENOME, TRANSPORTER methotrexate METHOTREXATE 36785 25071 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Debio1347 DEBIO-1347 36786 25072 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME KENPAULLONE KENPAULLONE 36787 25073 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE moviprep 36788 25074 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-162 36789 25075 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER R101933 36791 25076 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor CHEMBL488436 AZD-5438 36792 25077 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BUTYLPARABEN BUTYLPARABEN 36793 25078 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NITAZOXANIDE NITAZOXANIDE 36794 25079 CBX1 10951 NA NSC-720622 CHEMBL1287980 36795 25080 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL2107771 RALFINAMIDE 36796 25081 FKBP5 2289 DRUGGABLE GENOME paroxetine PAROXETINE 18597649,21449676,20709156,19676097,15565110,23733030,17467808 36797 25082 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE STZ STREPTOZOCIN 16130182 36798 25083 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PHENOLPHTHALEIN PHENOLPHTHALEIN 36799 25084 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL515387 GOSOGLIPTIN 36800 25085 RGS4 5999 DRUGGABLE GENOME CHELERYTHRINE CHELERYTHRINE 36801 25086 CYP24A1 1591 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME Lunacalcipol LUNACALCIPOL 36804 25087 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 busulfan BUSULFAN 24165757 36805 25088 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 36806 25089 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545322 PANULISIB 36808 25090 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE IDARUBICIN IDARUBICIN 22081665 36809 25091 ALB 213 TRANSPORTER, DRUGGABLE GENOME Gadobenate Dimeglumine 36810 25092 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME CS-3030 36811 25093 TUBB2B 347733 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 36813 25094 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING SCRIPTAID SCRIPTAID 19966789 36815 25095 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 36818 25096 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SPIPERONE SPIPERONE 36820 25097 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565829 36821 25098 ALPL 249 ENZYME, DRUGGABLE GENOME (+)-CATECHIN HYDRATE CHEMBL1256783 36823 25099 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TCMDC-123591 CHEMBL588234 36824 25100 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-270822A GSK-270822A 36825 25101 BCHE 590 DRUGGABLE GENOME, ENZYME Volanesorsen VOLANESORSEN 36827 25102 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FGF-1 FIBROBLAST GROWTH FACTOR-1 36828 25103 TUBB 203068 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 36830 25104 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME MIFEPRISTONE MIFEPRISTONE 10717784 36831 25105 S100A12 6283 DRUGGABLE GENOME, KINASE Eptinezumab EPTINEZUMAB 36832 25106 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CID 667285 CHEMBL267160 36833 25107 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME FESOTERODINE FESOTERODINE 36836 25108 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE TAE-684 TAE-684 36837 25109 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE Sym013 36838 25110 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OLANZAPINE OLANZAPINE 36839 25111 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE TYROSINE KINASE INHIBITOR 11245436 36840 25112 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME QUINOXALINE-2-CARBOXYLIC ACID CHEMBL151797 36841 25113 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR (R)-ALPHA-METHYLHISTAMINE CHEMBL268229 36843 25114 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Bis-aminopyrimidine derivative 3 36844 25115 ADAM10 102 ENZYME, CELL SURFACE, TRANSPORTER, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE INCB7839 36845 25116 ORAI1 84876 TRANSCRIPTION FACTOR, ION CHANNEL, TRANSPORTER blocker 381118798 36847 25117 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Abituzumab ABITUZUMAB 36848 25118 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL2105755 NALDEMEDINE 36849 25119 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 178102336 BOSUTINIB 36850 25120 GMNN 51053 DRUGGABLE GENOME DNDI1417759 CHEMBL1446254 36852 25121 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CYC-116 CYC-116 36853 25122 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 6-12 36854 25123 PTPRD 5789 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE verapamil VERAPAMIL 26425837 36855 25124 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-60 36857 25125 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME inhibitor 178103236 36859 25126 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200790 METHYPRYLON 36860 25127 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE MEK162 BINIMETINIB 27507190 36862 25128 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR EPOPROSTENOL EPOPROSTENOL 36863 25129 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OLOPATADINE OLOPATADINE 36866 25130 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME ROMIDEPSIN ROMIDEPSIN 36867 25131 STAG2 10735 CLINICALLY ACTIONABLE, DRUG RESISTANCE Trametinib TRAMETINIB 27500726 36868 25132 LGALS3 3958 CELL SURFACE, DRUGGABLE GENOME GR-MD-02 BELAPECTIN 36872 25133 TRPM7 54822 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ION CHANNEL, ENZYME, TRANSPORTER blocker 178101079 NAFAMOSTAT 36873 25134 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Bidentate ligands of Markush derivative 2 36874 25135 KDM4A 9682 DRUGGABLE GENOME, ENZYME Heteroaryl-cyclopropylamine derivative 4 36875 25136 CFLAR 8837 DRUG RESISTANCE, DRUGGABLE GENOME, PROTEASE BICALUTAMIDE BICALUTAMIDE 22623731 36877 25137 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-5510 CHEMBL578741 36879 25138 KDM4A 9682 DRUGGABLE GENOME, ENZYME DOXYCYCLINE HYCLATE DOXYCYCLINE HYCLATE 36881 25139 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME OXYMETHOLONE OXYMETHOLONE 36883 25140 ATAD5 79915 NA AZATHIOPRINE AZATHIOPRINE 36885 25141 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX DEHYDROXYMETHYLEPOXYQUINOMICIN DEHYDROXYMETHYLEPOXYQUINOMICIN 18729348 36887 25142 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME NOREPINEPHRINE NOREPINEPHRINE 36890 25143 GAA 2548 DRUGGABLE GENOME, ENZYME ELLIPTECINE ELLIPTECINE 36891 25144 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE celecoxib CELECOXIB 22336956 36892 25145 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRILOSTANE TRILOSTANE 36893 25146 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME TAK-733 TAK-733 22798288,24398428,26439693 36894 25147 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ER2 27040853 36895 25148 PSMA7 5688 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 36896 25149 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE IMETELSTAT IMETELSTAT 36897 25150 PSMD11 5717 KINASE inhibitor CARFILZOMIB CARFILZOMIB 36899 25151 QPRT 23475 ENZYME NIACIN NIACIN 36900 25152 GMNN 51053 DRUGGABLE GENOME DNDI1417411 CHEMBL1445650 36901 25153 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 252166676 36903 25154 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TAMIBAROTENE TAMIBAROTENE 36904 25155 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor CHEMBL1969664 AZD-1080 36905 25156 BIRC7 79444 PROTEASE INHIBITOR, TUMOR SUPPRESSOR, DRUG RESISTANCE antagonist AT-406 AT-406 36907 25157 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY PROGESTERONE PROGESTERONE 8404664 36908 25158 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR antipsychotics 16633140,25560300 36910 25159 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHLORHEXIDINE HYDROCHLORIDE CHLORHEXIDINE HYDROCHLORIDE 36911 25160 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER GEFITINIB GEFITINIB 16651435 36912 25161 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Methotrexate METHOTREXATE 28151717 36914 25162 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME BI-2536 BI-2536 25685941 36917 25163 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650113 CLOPROSTENOL 36919 25164 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 desipramine DESIPRAMINE 36920 25165 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-acylpiperidine ether derivative 7 36924 25166 PDE4A 5141 DRUGGABLE GENOME, ENZYME MK-0873 MK-0873 36926 25167 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-124176 CHEMBL588038 36927 25168 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL572881 MOTESANIB 36929 25169 CSNK2A2 1459 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME, TRANSCRIPTION FACTOR US8791257, 4 36931 25170 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME TOZASERTIB TOZASERTIB 36932 25171 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 310264733 FIMEPINOSTAT 36935 25172 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-Figure16 36936 25173 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER LX4211 36938 25174 GPR12 2835 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR 24-EPI-CYCLOCITRINOL CHEMBL496266 18656987 36939 25175 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER CEFAMANDOLE CEFAMANDOLE 22166395 36941 25176 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Benzothiazepine analog 10 36944 25177 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DIETHYL-2-TETRADECYLIDENEMALONATE CHEMBL257748 21292492 36947 25178 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TCMDC-124518 CHEMBL527584 36948 25179 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE URACIL URACIL 10607743 36949 25180 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME RG-1530 RG-1530 36951 25181 KISS1 3814 DRUGGABLE GENOME TAK-448 TAK-448 36954 25182 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE ropivacaine ROPIVACAINE 36956 25183 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME dapsone DAPSONE 29233746 36958 25184 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Sapanisertib SAPANISERTIB 25261369 36960 25185 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL940 GABAPENTIN 36961 25186 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Tolterodine TOLTERODINE 36962 25187 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER SULFINPYRAZONE SULFINPYRAZONE 36963 25188 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Abemaciclib ABEMACICLIB 27217383 36964 25189 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLOBENPROPIT CLOBENPROPIT 36966 25190 CBX1 10951 NA GNF-PF-4992 CHEMBL275177 36968 25191 AQP8 343 ION CHANNEL inhibitor 178101032 36970 25192 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 336446949 36971 25193 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THIORIDAZINE HYDROCHLORIDE THIORIDAZINE HYDROCHLORIDE 36972 25194 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX 9-AMINOCAMPTOTHECIN 9-AMINOCAMPTOTHECIN 36973 25195 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Sapitinib SAPITINIB 24886365,20145185 36975 25196 HPN 3249 DRUGGABLE GENOME, PROTEASE, CELL SURFACE Meclizine MECLIZINE 36976 25197 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME PIRFENIDONE PIRFENIDONE 36977 25198 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME IMMUNOSUPPRESSIVE 10342319 36978 25199 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE TGX-221 23674493,26577700 36979 25200 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MPA PROGESTERONE 16684279 36980 25201 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FRENTIZOLE FRENTIZOLE 36981 25202 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649887 36982 25203 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DOXEPIN DOXEPIN 36983 25204 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME E6201 E-6201 23039341 36984 25205 ATXN2 6311 NA THAPSIGARGIN THAPSIGARGIN 36985 25206 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR TRAIL 14596484,14739605 36986 25207 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ETHANOL ALCOHOL 16272348 36987 25208 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALISERTIB ALISERTIB 36988 25209 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 36989 25210 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 3,5-DIPHENYLISOXAZOLE 3,5-DIPHENYLISOXAZOLE 36991 25211 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor CHEMBL574737 UCN-01 36992 25212 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL451887 CARFILZOMIB 36995 25213 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Abemaciclib ABEMACICLIB 27217383,26183925 36996 25214 NOS1 4842 DRUGGABLE GENOME, ENZYME NXN-188 36998 25215 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL1096885 VALRUBICIN 37003 25216 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 838877 CHEMBL405317 37004 25217 AKR1C3 8644 ENZYME, DRUGGABLE GENOME doxorubicin DOXORUBICIN 23116553,20837989,21048526 37006 25218 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-10 37007 25219 CBX1 10951 NA CLOZAPINE CLOZAPINE 37008 25220 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZD8835 AZD-8835 26839307 37013 25221 FBP1 2203 DRUGGABLE GENOME, ENZYME MB07803 MB-07803 37014 25222 VKORC1 79001 DRUGGABLE GENOME, ENZYME PHENINDIONE PHENINDIONE 37015 25223 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Crizotinib CRIZOTINIB 28476735 37016 25224 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE RUCAPARIB RUCAPARIB 37017 25225 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Pyrazolo-triazine derivative 2 37018 25226 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME O6-Benzylguanine alkylade 37020 25227 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME RESOKAEMPFEROL RESOKAEMPFEROL 37021 25228 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-321 CHEMBL581044 37022 25229 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR methamphetamine METHAMPHETAMINE 19386276 37023 25230 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PKI-587 GEDATOLISIB 37024 25231 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 37025 25232 FBXW7 55294 DNA REPAIR, CLINICALLY ACTIONABLE AR-42 AR-42 23274910 37026 25233 CDK10 8558 DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3544942 RONICICLIB 37027 25234 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL2107823 GANDOTINIB 37028 25235 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE NSC-341622 CHEMBL79513 20155916,21823606,22329436,24502276 37029 25236 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE blocker 135650306 GLYBURIDE 37033 25237 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MIRTAZAPINE MIRTAZAPINE 37034 25238 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE 2-(4-NITROPHENYL)BENZO[D]THIAZOLE CHEMBL477841 19147351 37036 25239 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR TETRADECANOYL PHORBOL ACETATE TETRADECANOYL PHORBOL ACETATE 20121237 37038 25240 HR 55806 NUCLEAR HORMONE RECEPTOR ETX-9101 37040 25241 CCL2 6347 DRUGGABLE GENOME NOX-E36 37043 25242 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000117447 CHEMBL592611 37044 25243 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Temsirolimus TEMSIROLIMUS 21216929 37045 25244 A2M 2 ENZYME, TRANSPORTER, DRUGGABLE GENOME, PROTEASE INHIBITOR COBALT 6663071 37047 25245 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GW0742 CHEMBL38508 23273519 37050 25246 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME INHIBINS 15590985 37051 25247 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME 681640 CHEMBL379975 37052 25248 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178100909 37053 25249 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-157 37054 25250 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102242 ISTRADEFYLLINE 37055 25251 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR AZD5363 CAPIVASERTIB 37056 25252 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR GEMCITABINE GEMCITABINE 37060 25253 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178101521 FEXOFENADINE 37061 25254 ABCC9 10060 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER montelukast MONTELUKAST 28940478 37062 25255 ATXN2 6311 NA GNF-PF-3350 CHEMBL600747 37063 25256 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE URAPIDIL URAPIDIL 37066 25257 TFF2 7032 DRUGGABLE GENOME Aprotinin APROTININ 37067 25258 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 363894144 GW-406381 37068 25259 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR VASOPRESSIN VASOPRESSIN 7482412 37070 25260 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RILMENIDINE RILMENIDINE 37071 25261 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME RG-1530 RG-1530 37072 25262 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE nevirapine NEVIRAPINE 20017669,19228205,21824325 37073 25263 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist CHEMBL1265 ADAPALENE 37075 25264 PADI2 11240 ENZYME O-CL-AMIDINE CHEMBL1910971 21882827 37076 25265 USP14 9097 ENZYME, CELL SURFACE, PROTEASE PMID26077642-Compound-Figure3A 37078 25266 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4837 CHEMBL600769 37079 25267 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GENISTEIN GENISTEIN 37080 25268 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-143 37081 25269 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 354702263 37082 25270 GMNN 51053 DRUGGABLE GENOME GNF-PF-2936 CHEMBL582503 37084 25271 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PAZOPANI 37085 25272 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME activator 135652675 CAFFEINE 37088 25273 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 22225636 37089 25274 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor SF1126 37092 25275 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Epoxysuccinate derivative 6 37093 25276 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 dorzolamide DORZOLAMIDE 9187528 37094 25277 LRMDA 83938 NA tamoxifen TAMOXIFEN 22180457 37095 25278 APBB1 322 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING Clofarabine CLOFARABINE 37097 25279 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ARCTIGENIN ARCTIGENIN 37098 25280 ILK 3611 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME US8754233, 4-(5-Fluoro-6-methoxy-benzothiazol-2-yl)-5-(2-fluoro-phenyl)-2H-pyrazol-3-ylamine 37099 25281 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NIRIDAZOLE NIRIDAZOLE 37100 25282 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZIPRASIDONE ZIPRASIDONE 37103 25283 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NEBULARINE NEBULARINE 37104 25284 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 223366025 ELUXADOLINE 37105 25285 ALPI 248 DRUGGABLE GENOME, ENZYME TERPYRIDINE TERPYRIDINE 37108 25286 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PUROMYCIN PUROMYCIN 8423352 37110 25287 TUBB4B 10383 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 37112 25288 TUBA1C 84790 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 37114 25289 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME Antithyroid Preparations 27157822 37115 25290 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650039 37116 25291 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Metaproterenol Sulfate 37117 25292 PSMB7 5695 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL371405 MARIZOMIB 37118 25293 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TAMOXIFEN TAMOXIFEN 11916237,15901136,17266042 37123 25294 TARDBP 23435 TUMOR SUPPRESSOR PROGESTERONE PROGESTERONE 37127 25295 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY IL-2 ALDESLEUKIN 2149997 37128 25296 ST14 6768 ENZYME, DRUGGABLE GENOME, PROTEASE US8569313, Inhibitor 18 37129 25297 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650504 37130 25298 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE HEXACHLOROPHENE HEXACHLOROPHENE 37131 25299 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR VALSARTAN VALSARTAN 37132 25300 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649874 37133 25301 ATP2A2 488 ENZYME, DRUGGABLE GENOME, TRANSPORTER ISTAROXIME ISTAROXIME 37134 25302 GAA 2548 DRUGGABLE GENOME, ENZYME SULFURETIN SULFURETIN 37138 25303 SMN1 6606 DRUGGABLE GENOME GNF-PF-1235 CHEMBL585769 37139 25304 IL1B 3553 KINASE, DRUGGABLE GENOME TPA ALTEPLASE 8615653 37141 25305 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor GEFITINIB GEFITINIB 37142 25306 RAB9A 9367 ENZYME, DRUGGABLE GENOME LEFLUNOMIDE LEFLUNOMIDE 37144 25307 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 223366077 RGB-286638 37145 25308 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL483321 CP-724714 37146 25309 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1131 ACITRETIN 37148 25310 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CIGLITAZONE CIGLITAZONE 37149 25311 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ILORASERTIB ILORASERTIB 37150 25312 HSPB1 3315 DRUGGABLE GENOME VASOPRESSIN VASOPRESSIN 9925748 37151 25313 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX SELICICLIB SELICICLIB 21417417 37152 25314 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE IMATINIB IMATINIB 23835704,26703895,24186319,16960151,32068648 37154 25315 NUCB1 4924 DRUGGABLE GENOME antagonist 252166902 37155 25316 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID30259754-Compound-INT-767 37156 25317 CCR6 1235 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR agonist 178100550 37157 25318 ALPL 249 ENZYME, DRUGGABLE GENOME HAEMATOXYLIN HAEMATOXYLIN 37158 25319 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE DE-766 37159 25320 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650682 NALORPHINE 37160 25321 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME TAMATINIB R-406 37161 25322 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUAZINAM FLUAZINAM 37162 25323 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Onartuzumab ONARTUZUMAB 27918764 37164 25324 ABL2 27 KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME inhibitor TOZASERTIB TOZASERTIB 19035792 37165 25325 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL223360 LINIFANIB 37166 25326 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR RAPAMYCIN SIROLIMUS 11145585 37167 25327 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE IBANDRONATE IBANDRONIC ACID 37168 25328 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-4467 CHEMBL598883 37170 25329 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 24 37171 25330 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER INDOPROFEN INDOPROFEN 37172 25331 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Alkaloid derivative 4 37174 25332 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200606 MEXILETINE HYDROCHLORIDE 37176 25333 GABBR2 9568 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL1200682 SODIUM OXYBATE 37177 25334 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-18 37178 25335 GJB1 2705 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER inhibitor 178101095 OCTANOL 37179 25336 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Matairesinol derivative 1 37180 25337 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135649947 APAFANT 37181 25338 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE IBRUTINIB IBRUTINIB 24915291 37189 25339 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR COUMERMYCIN A1 COUMERMYCIN A1 24360559 37190 25340 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME Pyrrolo[2,3-d]pyrimidine derivative 4 37192 25341 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYL PARATHIONE METHYL PARATHIONE 37194 25342 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 135651714 37195 25343 BAZ2B 29994 NA MERCAPTOPURINE HYDRATE MERCAPTOPURINE 37197 25344 ATAD5 79915 NA BROMOENOL LACTONE BROMOENOL LACTONE 37198 25345 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Methotrexate METHOTREXATE 28151717 37201 25346 NGFR 4804 CELL SURFACE, DRUGGABLE GENOME 178101729 37202 25347 PLA2G7 7941 DRUGGABLE GENOME, ENZYME Indolizine derivative 1 37203 25348 SIRT5 23408 ENZYME OLEOYL DOPAMINE OLEOYL DOPAMINE 37204 25349 POLK 51426 DNA REPAIR, ENZYME BISANHYDRORUTILANTINONE BISANHYDRORUTILANTINONE 37205 25350 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME Quisinostat QUISINOSTAT 37206 25351 MPHOSPH8 54737 NA GYKI-52895 CHEMBL1256984 37207 25352 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650407 37208 25353 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME PMID27998201-Compound-6 37212 25354 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 2 37213 25355 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 3R14S-OCHRATOXIN A 3R14S-OCHRATOXIN A 37214 25356 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Oxazolyl methylthiothiazole derivative 1 37215 25357 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE trastuzumab TRASTUZUMAB 25199759 37216 25358 CBX1 10951 NA R-N-PROPYLNORAPOMORPHINE R-N-PROPYLNORAPOMORPHINE 37217 25359 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200733 DESFLURANE 37218 25360 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR VX-745 NEFLAMAPIMOD 37219 25361 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651539 DINOPROSTONE 37220 25362 POLK 51426 DNA REPAIR, ENZYME PHYSODIC ACID PHYSODIC ACID 37224 25363 ITGB8 3696 DRUGGABLE GENOME, CELL SURFACE US10035778, Example 16 37225 25364 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TRANILAST TRANILAST 37226 25365 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N,N-bis(5-pyrazoyl)urea derivative 1 37227 25366 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME GSK2586184 SOLCITINIB 37228 25367 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE SJ000039423 CHEMBL589207 37229 25368 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 249565735 37232 25369 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 37233 25370 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE activator CHEMBL2108358 SERELAXIN 37236 25371 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AG-490 CHEMBL56543 37237 25372 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ALL-TRANS RETINOIC ACID 9447832 37240 25373 ALDH1A1 216 DRUGGABLE GENOME, ENZYME AG-1288 CHEMBL166486 37241 25374 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CID 739615 CHEMBL260560 37243 25375 SLC25A6 293 TRANSPORTER, DRUGGABLE GENOME CLODRONATE CLODRONIC ACID 37244 25376 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL DIAZEPAM DIAZEPAM 37245 25377 KDM4A 9682 DRUGGABLE GENOME, ENZYME BENZANTHRONE BENZANTHRONE 37247 25378 RIPK2 8767 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102513 PONATINIB 37248 25379 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME CENISERTIB CENISERTIB 37250 25380 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-73 37251 25381 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650986 37252 25382 NPC1L1 29881 DRUGGABLE GENOME, TRANSPORTER antagonist 178103422 EZETIMIBE 37253 25383 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR SNX-5422 CHEMBL553939 37254 25384 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody MEHD7945A DULIGOTUZUMAB 37255 25385 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE ACTB1003 37256 25386 THBS2 7058 DRUGGABLE GENOME BEVACIZUMAB BEVACIZUMAB 16365183 37257 25387 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE HERBIMYCIN A 11139143 37258 25388 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652300 37259 25389 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE DELAVIRDINE DELAVIRDINE 17172311 37261 25390 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-acylpyrrolidine ether derivative 2 37262 25391 MCOLN1 57192 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER activator 178103002 37263 25392 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CHEMBL591 ETHCHLORVYNOL 37264 25393 POLK 51426 DNA REPAIR, ENZYME PICEATANNOL PICEATANNOL 37265 25394 AKR1C2 1646 DRUGGABLE GENOME, ENZYME URSODEOXYCHOLIC ACID 37266 25395 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-4864 CHEMBL583558 37267 25396 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMODIAQUINE DIHYDROCHLORIDE AMODIAQUINE DIHYDROCHLORIDE 37268 25397 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE DOVITINIB DOVITINIB 37270 25398 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR BELINOSTAT BELINOSTAT 25937017 37272 25399 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME JCXGHZCWAHCYGY-UHFFFAOYSA-N 37273 25400 ALDH1A1 216 DRUGGABLE GENOME, ENZYME MYRICETIN MYRICETIN 37275 25401 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME ALOSETRON HYDROCHLORIDE ALOSETRON HYDROCHLORIDE 37276 25402 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL454 BUTALBITAL 37278 25403 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BIOALLETHRIN S-CYCLOPENTENYL ISOMER BIOALLETHRIN S-CYCLOPENTENYL ISOMER 37279 25404 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CLOTRIMAZOLE CLOTRIMAZOLE 22931300 37280 25405 CBX1 10951 NA GBR-12935 CHEMBL26320 37283 25406 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER 4-(4-CHLOROPHENOXY)ANILINE CHEMBL1521156 37284 25407 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 7 37286 25408 LHFPL3 375612 NA corticosteroids 30697902 37287 25409 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417941 CHEMBL2095095 37288 25410 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1648 ISRADIPINE 37290 25411 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-62406 CHEMBL1332182 37291 25412 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651353 ZACOPRIDE 37293 25413 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ERGOCORNINE ERGOCORNINE 37294 25414 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE HYDROXYUREA HYDROXYUREA 2422298 37295 25415 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-747260 CHEMBL595912 37296 25416 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME JNJ-42756493 ERDAFITINIB 37297 25417 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist 135650003 37298 25418 MAP2K3 5606 KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE inhibitor BAY869766 37299 25419 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID30259754-Compound-WAY-362450 37300 25420 HPRT1 3251 DRUGGABLE GENOME, ENZYME MERCAPTOPURINE MERCAPTOPURINE 37301 25421 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE CHLORHEXIDINE CHLORHEXIDINE 10225852 37303 25422 PDE4A 5141 DRUGGABLE GENOME, ENZYME CC-1088 CDC-801 37304 25423 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SJ000111093 CHEMBL585045 37305 25424 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9181182, 47 37306 25425 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AMBAZONE AMBAZONE 37307 25426 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL605525 DP001 37308 25427 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NEOPETROFORMYNE A NEOPETROFORMYNE A 22928967 37309 25428 PTGS2 5743 DRUGGABLE GENOME, ENZYME DEXIBUPROFEN DEXIBUPROFEN 20143779 37310 25429 PPP2R5D 5528 PROTEIN PHOSPHATASE, ENZYME epirubicin EPIRUBICIN 37311 25430 MAOB 4129 DRUGGABLE GENOME, ENZYME RASAGILINE RASAGILINE 37312 25431 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Alitretinoin ALITRETINOIN 37314 25432 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MK-2461 MK-2461 37315 25433 MS4A2 2206 EXTERNAL SIDE OF PLASMA MEMBRANE OMALIZUMAB OMALIZUMAB 37316 25434 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Spirolaxine derivative 1 37317 25435 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL2104984 SODELGLITAZAR 37318 25436 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME Autologous T cells transfected with chimeric anti-mesothelin immunoreceptor SS1 37321 25437 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GW7647 GW7647 37322 25438 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL3545209 NKTR-171 37323 25439 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR PH-797804 PH-797804 37324 25440 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR GNF-PF-4464 CHEMBL600692 37325 25441 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL799 CILOSTAZOL 37326 25442 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE naloxone NALOXONE 11751037,12627468,18004207,16123758 37327 25443 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIPERIDOLATE HYDROCHLORIDE PIPERIDOLATE HYDROCHLORIDE 37331 25444 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SOTRASTAURIN SOTRASTAURIN 37332 25445 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565821 37333 25446 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TICRYNAFEN TICRYNAFEN 22931300 37335 25447 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME ETHYL CAFFEATE ETHYL CAFFEATE 25314129 37336 25448 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR BI-87E7 CHEMBL523200 37337 25449 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PRN1109 37338 25450 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE vincristine VINCRISTINE 37339 25451 CDA 978 ENZYME, DRUGGABLE GENOME cytarabine CYTARABINE 21325291,21521023,22304580,22379997,25003625,19458626,23651026,23230131,18473752 37340 25452 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-3501 CHEMBL581910 37342 25453 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BKM120 BUPARLISIB 24470511,26098748,28119489 37345 25454 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR inhibitor CHEMBL2105467 TEZACITABINE 37347 25455 BAZ2B 29994 NA TCMDC-125543 CHEMBL546170 37348 25456 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-42258 CHEMBL1410004 37349 25457 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-123730 CHEMBL530280 37350 25458 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DEPHOSTATIN DEPHOSTATIN 37351 25459 APC 324 CLINICALLY ACTIONABLE CCT036477 20610623 37352 25460 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME PMID29130358-Compound-Figure10(2a) 37354 25461 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651148 37355 25462 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-D2 37357 25463 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE THIOGUANOSINE THIOGUANOSINE 37360 25464 BAZ2B 29994 NA GNF-PF-3416 CHEMBL579550 37361 25465 CBX1 10951 NA MORIN MORIN 37365 25466 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 404859105 37366 25467 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME ADRENOCORTICOTROPIN CORTICOTROPIN 2444616 37367 25468 MAOA 4128 DRUGGABLE GENOME, ENZYME Tranylcypromine TRANYLCYPROMINE 37368 25469 HMGCR 3156 ENZYME, DRUGGABLE GENOME PMID27537201-Compound-Figure13b 37369 25470 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649917 ALLOXAZINE 37372 25471 ALOX15 246 ENZYME, DRUGGABLE GENOME QUERCETIN QUERCETIN 17869117 37373 25472 TUBB3 10381 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 37374 25473 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Sapanisertib SAPANISERTIB 25261369,23085766 37375 25474 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RESORCINOL MONOACETATE RESORCINOL MONOACETATE 37376 25475 TPCN1 53373 ION CHANNEL, DRUGGABLE GENOME blocker 135651305 VERAPAMIL 37379 25476 MAP2K3 5606 KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE inhibitor GDC-0973 COBIMETINIB 37382 25477 HSPB1 3315 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 37383 25478 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE JNJ-26483327 JNJ-26483327 37384 25479 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE METHYLENE BLUE CHLORIDE HYDRATE METHYLENE BLUE 37385 25480 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652140 37389 25481 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417601 CHEMBL1503729 37390 25482 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565761 37392 25483 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100628 37394 25484 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TINORIDINE TINORIDINE 37396 25485 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SPLITOMICIN SPLITOMICIN 37398 25486 UGT1A6 54578 ENZYME, DRUGGABLE GENOME SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 37399 25487 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 2,7-BIS[3-(DIMETHYLAMINO)PROPIONAMIDO]ANTHRAQUINONE CHEMBL89977 18571928 37401 25488 MAPT 4137 DRUGGABLE GENOME TYRPHOSTIN 23 TYRPHOSTIN 23 37402 25489 CBX1 10951 NA TCMDC-123916 CHEMBL493863 37403 25490 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE 11C-AZD-2184 23324871 37404 25491 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Vorinostat VORINOSTAT 26009011,25669829 37405 25492 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR SERM 12901849 37406 25493 C3 718 PROTEASE INHIBITOR, DRUGGABLE GENOME, CELL SURFACE Imprime PGG immunotherapeutic 37407 25494 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GNF-PF-806 CHEMBL547101 37411 25495 IL7R 3575 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME RUXOLITINIB (IN SH2B3 DELETED) 22897847,22955920 37413 25496 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-25 37414 25497 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE NSC-139257 CHEMBL1256364 37416 25498 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SJ000244621 CHEMBL600175 37417 25499 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE BAY-613606 CHEMBL541400 37418 25500 MPHOSPH8 54737 NA 3,4-DICHLOROISOCOUMARIN CHEMBL24983 37419 25501 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 249565686 BX-795 37420 25502 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME INTERLEUKIN-2 EXPRESSING PLASMID 37421 25503 SMN1 6606 DRUGGABLE GENOME CID2350207 CHEMBL259615 37422 25504 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME PROCARBAZINE PROCARBAZINE 11839668 37424 25505 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178102337 SORAFENIB 37425 25506 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 252827366 GILTERITINIB 37426 25507 POLK 51426 DNA REPAIR, ENZYME TDR77578 CHEMBL1364172 37427 25508 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SQ-789 CHEMBL211042 37428 25509 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 178101947 RUBOXISTAURIN 37430 25510 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 17-BETA ESTRADIOL 37431 25511 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 37434 25512 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DYCLONINE HYDROCHLORIDE DYCLONINE HYDROCHLORIDE 37436 25513 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pembrolizumab PEMBROLIZUMAB 37437 25514 SGPL1 8879 ENZYME, DRUGGABLE GENOME inhibitor 363894145 LX-2931 37438 25515 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME LAUROGUADINE LAUROGUADINE 37439 25516 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3582 CHEMBL606167 37441 25517 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY ISOTRETINOIN ISOTRETINOIN 12656659 37443 25518 ALOX15 246 ENZYME, DRUGGABLE GENOME LINOLEIC ACID LINOLEIC ACID 37445 25519 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TRIIODOTHYRONINE (T3) 37446 25520 EGFL7 51162 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE ANTI-EGFL7 37447 25521 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Bimosiamose BIMOSIAMOSE 37449 25522 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR PACLITAXEL PACLITAXEL 23038758 37451 25523 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 223365939 37453 25524 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME VANDETANIB VANDETANIB 37454 25525 GAPDH 2597 DRUGGABLE GENOME, ENZYME TCMDC-124224 CHEMBL580421 37455 25526 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL HALAZEPAM HALAZEPAM 37459 25527 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200322 ESCITALOPRAM OXALATE 37460 25528 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Epoxysuccinate derivative 3 37461 25529 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20120264760C87 37462 25530 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ILORASERTIB ILORASERTIB 37463 25531 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TYRPHOSTIN A9 TYRPHOSTIN A9 37464 25532 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL24828 VANDETANIB 37466 25533 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor BGJ398 INFIGRATINIB 37467 25534 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PHENYLBUTANOIC ACID PHENYLBUTANOIC ACID 24044874 37468 25535 GLA 2717 ENZYME, DRUGGABLE GENOME Maltose MALTOSE 37469 25536 GLA 2717 ENZYME, DRUGGABLE GENOME Migalastat MIGALASTAT 37470 25537 DGAT2 84649 ENZYME ARI-3037MO 37471 25538 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PREDNISONE PREDNISONE 37473 25539 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor MK2461 37476 25540 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE EZN-2968 37477 25541 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR WHILE OLIVETOL WHILE OLIVETOL 37478 25542 SMN1 6606 DRUGGABLE GENOME DNDI1417195 CHEMBL1303948 37484 25543 LPAR2 9170 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 135649710 37485 25544 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE ENTRECTINIB ENTRECTINIB 37486 25545 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME FILGRASTIM FILGRASTIM 37487 25546 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 249565753 37489 25547 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE CHEMBL2364609 ESKETAMINE HYDROCHLORIDE 37490 25548 GPA33 10223 DRUGGABLE GENOME HuA33 HUA33 37491 25549 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1071 OXAPROZIN 37492 25550 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Resminostat RESMINOSTAT 37493 25551 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MIFEPRISTONE MIFEPRISTONE 37494 25552 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE AZD8186 AZD-8186 37495 25553 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2062264 PHENYLEPHRINE BITARTRATE 37496 25554 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 135651362 37498 25555 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PANITUMUMAB PANITUMUMAB 37502 25556 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME SODIUM HEPARIN 15205701 37503 25557 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE GDC-0944 37504 25558 IFNGR1 3459 DRUGGABLE GENOME, CLINICALLY ACTIONABLE agonist CHEMBL1201564 INTERFERON GAMMA-1B 37506 25559 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL CHEMBL256087 MENTHOL 37507 25560 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME PYRAFLUFEN-ETHYL PYRAFLUFEN-ETHYL 37508 25561 PTGS1 5742 ENZYME, DRUGGABLE GENOME URSOLIC ACID URSOLIC ACID 9784154 37509 25562 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE YU238259 26116172 37510 25563 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL586701 ZSTK-474 37511 25564 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CORTODOXONE CORTODOXONE 37513 25565 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Dihydrotachysterol DIHYDROTACHYSTEROL 37514 25566 STAG2 10735 CLINICALLY ACTIONABLE, DRUG RESISTANCE Camptothecin CAMPTOTHECIN 21852505,24356817 37515 25567 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DB-959 DB959 37516 25568 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL2103842 VARLITINIB 37518 25569 HBB 3043 DRUGGABLE GENOME, ENZYME THIOGUANINE THIOGUANINE 37521 25570 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor CHEMBL1200814 ACETAZOLAMIDE SODIUM 37522 25571 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME OPROZOMIB OPROZOMIB 37523 25572 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker 178101099 PHENCYCLIDINE 37524 25573 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL378544 VINBLASTINE SULFATE 37525 25574 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 37526 25575 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Azaindazole derivative 4 37527 25576 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ORCIPRENALINE METAPROTERENOL 37531 25577 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor GDC-0973 COBIMETINIB 37532 25578 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AC430 AC-430 37533 25579 KMO 8564 DRUGGABLE GENOME, ENZYME Cyclopropane 1-carboxylic acid derivative 3 37534 25580 HTT 3064 DRUGGABLE GENOME ALAZANINE ALAZANINE 37535 25581 POLL 27343 NA 1-DEOXYRUBRALACTONE CHEMBL260980 18178092 37536 25582 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-50 37537 25583 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 223366077 RGB-286638 37538 25584 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Pyrimidinone derivative 1 37540 25585 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-105827 CHEMBL171699 37541 25586 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DAPHNETIN DAPHNETIN 37542 25587 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR PF-562271 PF-00562271 37543 25588 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENOXACOR BENOXACOR 37544 25589 ME3 10873 ENZYME ASPIRIN ASPIRIN 8611656 37545 25590 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178103826 OXAPROZIN 37547 25591 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 14 37548 25592 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME CEFOTETAN CEFOTETAN 37550 25593 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR MEDROXYPROGESTERONE ACETATE MEDROXYPROGESTERONE ACETATE 37551 25594 IKBKG 8517 KINASE, DRUGGABLE GENOME primaquine PRIMAQUINE 37555 25595 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Metoprolol METOPROLOL 37556 25596 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NICLOSAMIDE NICLOSAMIDE 37557 25597 TAC1 6863 DRUGGABLE GENOME HALOPERIDOL HALOPERIDOL 6166743 37563 25598 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR Talimogene Laherparepvec 37564 25599 RALBP1 10928 TRANSPORTER, ABC TRANSPORTER DOX 12632060 37565 25600 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PALMITOYL-CARNITINE PALMITOYL-CARNITINE 37566 25601 TXNIP 10628 TRANSCRIPTION FACTOR FAS-LIGAND 12706526 37567 25602 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME blocker 135651249 37570 25603 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-19 37571 25604 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE LIPOSOMAL DOXORUBICIN 10914739 37572 25605 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME GS 6201 GS 6201 37575 25606 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200332 PROTRIPTYLINE HYDROCHLORIDE 37576 25607 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLONAZEPAM CLONAZEPAM 37579 25608 PSMA4 5685 DRUGGABLE GENOME, PROTEASE inhibitor BORTEZOMIB BORTEZOMIB 37580 25609 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER 6-DESOXYMORPHINE CHEMBL410907 18311899 37581 25610 APOE 348 DRUGGABLE GENOME simvastatin SIMVASTATIN 10736278 37582 25611 RBX1 9978 DNA REPAIR, ENZYME fluorouracil FLUOROURACIL 37583 25612 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565893 37584 25613 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME H2O2 9706151 37585 25614 KCND3 3752 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL284348 DALFAMPRIDINE 37586 25615 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NORELGESTROMIN NORELGESTROMIN 37587 25616 MAPT 4137 DRUGGABLE GENOME 12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE 12A-HYDROXY-5-DEOXYDEHYDROMUNDUSERONE 37588 25617 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TCMDC-124278 CHEMBL534423 37590 25618 TUBB 203068 DRUGGABLE GENOME Lexibulin iv infusion 37591 25619 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545264 LY-2874455 37593 25620 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL1614725 TAK-285 37595 25621 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE isotretinoin ISOTRETINOIN 18695978 37596 25622 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING CLOSANTEL CLOSANTEL 37598 25623 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1692 IMIPRAMINE HYDROCHLORIDE 37599 25624 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE A-443654 A-443654 24978597,19208828,24569089 37600 25625 TOP2B 7155 DRUGGABLE GENOME, ENZYME Nalidixic Acid 37601 25626 GMNN 51053 DRUGGABLE GENOME HALETHAZOLE HALETHAZOLE 37602 25627 RBP4 5950 DRUGGABLE GENOME US9434727, 63 37608 25628 BAZ2B 29994 NA SJ000236197 CHEMBL582496 37611 25629 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Ribociclib RIBOCICLIB 37612 25630 NOS2 4843 DRUGGABLE GENOME, ENZYME inhibitor DOXYCYCLINE DOXYCYCLINE 37613 25631 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR eribulin ERIBULIN 37614 25632 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CAS 902561-11-9 CHEMBL494081 37618 25633 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME TRAMADOL TRAMADOL 37620 25634 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL1614766 RO-4987655 37621 25635 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE ISIS-FGFR4Rx 37622 25636 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR GO-6976 GO-6976 37623 25637 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 385612233 37624 25638 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GINKGO GINKGO 15901353 37628 25639 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE AZD8055 AZD-8055 28446642,22271687 37630 25640 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR HEXADECYLPHOSPHOCHOLINE MILTEFOSINE 1555249 37632 25641 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4789 CHEMBL583351 37633 25642 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NISOLDIPINE NISOLDIPINE 37634 25643 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor 178102336 BOSUTINIB 37639 25644 ATP1B3 483 ENZYME, TRANSPORTER, DRUGGABLE GENOME inhibitor CHEMBL3545057 ACETYLDIGITOXIN 37640 25645 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Thiomorpholine derivative 1 37641 25646 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE fluorouracil FLUOROURACIL 23314736 37642 25647 MCOLN1 57192 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER activator 178100233 37644 25648 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LU302146 37647 25649 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME EC-145 VINTAFOLIDE 23242435 37648 25650 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME ENTRECTINIB ENTRECTINIB 37649 25651 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 381118843 37651 25652 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE LINIFANIB LINIFANIB 37652 25653 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PRAZEPAM PRAZEPAM 37653 25654 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102572 37654 25655 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ENDRIN ENDRIN 37655 25656 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-105827 CHEMBL171699 37656 25657 CEL 1056 CELL SURFACE, DRUGGABLE GENOME, ENZYME GELDANAMYCIN GELDANAMYCIN 11104697 37657 25658 MBNL1 4154 DRUGGABLE GENOME NOR-BINALTORPHIMINE DIHYDROCHLORIDE CHEMBL2374078 37660 25659 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE ENMD-2076 ENMD-2076 27406088 37661 25660 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR THONZONIUM BROMIDE THONZONIUM BROMIDE 37662 25661 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR PF-562271 PF-00562271 37663 25662 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GBR-12935 CHEMBL26320 37664 25663 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200339 PHENYLEPHRINE HYDROCHLORIDE 37665 25664 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor 178104000 MOCLOBEMIDE 37667 25665 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE LAK 7947458,8095153,10520177,8128185,7651927,2469657,3294581,8917631,1968054,1362916 37668 25666 PTGS1 5742 ENZYME, DRUGGABLE GENOME Aminosalicylic Acid 37669 25667 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUOROMETHOLONE FLUOROMETHOLONE 37670 25668 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME rifampin RIFAMPIN 25798582,29036176,27281183 37671 25669 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL1256818 DEXTROMETHORPHAN HYDROBROMIDE 37672 25670 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LY-320135 CHEMBL411481 37675 25671 MGLL 11343 DRUGGABLE GENOME, ENZYME inhibitor 404859108 37676 25672 LPAR5 57121 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651509 37678 25673 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GERONTOXANTHONE I GERONTOXANTHONE I 37679 25674 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor CHEMBL408513 BELINOSTAT 37680 25675 POLB 5423 DNA REPAIR, DRUGGABLE GENOME AG-537 CHEMBL67535 37682 25676 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 348353627 37685 25677 MT1E 4493 NA NAC ACETYLCYSTEINE 7592595 37686 25678 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c][1,2,4]benzotriazine derivative 4 37688 25679 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178102746 37690 25680 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 N-DESMETHYLCLOZAPINE N-DESMETHYLCLOZAPINE 37691 25681 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME DIFLORASONE DIFLORASONE 37694 25682 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 223365976 ICOTINIB 37696 25683 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650009 BMY-7378 37697 25684 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor CUDC-101 CUDC-101 37698 25685 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 1R,9S-HYDRASTINE 1R,9S-HYDRASTINE 37699 25686 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME HYDROXYZINE HYDROXYZINE 37700 25687 IRS2 8660 KINASE, CLINICALLY ACTIONABLE INSULIN INSULIN 11522686,9421369,16037106,12687350 37701 25688 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor VORINOSTAT VORINOSTAT 37702 25689 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135650240 37703 25690 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL3544959 ARRY-382 37704 25691 PDE11A 50940 DRUGGABLE GENOME, ENZYME inhibitor 178103173 37706 25692 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Drospirenone DROSPIRENONE 37707 25693 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor PIMASERTIB PIMASERTIB 37708 25694 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200682 SODIUM OXYBATE 37709 25695 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BENFLUOREX HYDROCHLORIDE BENFLUOREX HYDROCHLORIDE 37710 25696 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 135650118 COLCHICINE 37712 25697 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1096 AMLEXANOX 37713 25698 PI4KB 5298 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, ENZYME inhibitor 252827496 37715 25699 CBX1 10951 NA TETRADECYLTHIOACETIC ACID TETRADECYLTHIOACETIC ACID 37718 25700 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GW405833 CHEMBL73711 37719 25701 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR VORINOSTAT VORINOSTAT 19344175,19966789,26211462,23622981,25974739,22260166,20491440,21548582,19084294 37720 25702 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 19 37724 25703 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE AVI-4126 37725 25704 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CNS-7056 REMIMAZOLAM 37728 25705 MUC2 4583 DRUGGABLE GENOME CHONDROITIN 12770776 37730 25706 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE LAPATINIB LAPATINIB 22885469 37731 25707 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 efavirenz EFAVIRENZ 16267764,15622315 37733 25708 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CHEMBL220492 TOPIRAMATE 37734 25709 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORHEXIDINE HYDROCHLORIDE CHLORHEXIDINE HYDROCHLORIDE 37735 25710 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OXYTOCIN OXYTOCIN 37736 25711 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist,antagonist 187051763 37737 25712 GRK2 156 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, G PROTEIN COUPLED RECEPTOR, ENZYME US9493490, C 37738 25713 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CAMBENDAZOLE CAMBENDAZOLE 37739 25714 USP1 7398 DNA REPAIR, PROTEASE, ENZYME EVANS BLUE EVANS BLUE 37740 25715 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME INFIGRATINIB INFIGRATINIB 26015511,27535980,27870574 37741 25716 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CADMIUM DICHLORIDE CADMIUM DICHLORIDE 37742 25717 BCL2L2 599 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 15813915 37743 25718 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME peginterferon alfa-2a 23360626 37745 25719 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME TCMDC-124059 CHEMBL530733 37746 25720 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Imidazo[1,5-a]pyridine derivative 1 37747 25721 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3137308 PEFICITINIB 37748 25722 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor ERISMODEGIB SONIDEGIB 37749 25723 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL1684984 PA-799 37750 25724 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178101879 37753 25725 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE pantoprazole PANTOPRAZOLE 18695978 37754 25726 DNER 92737 NA Quinazolinone derivative 4 37755 25727 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR TOZASERTIB TOZASERTIB 37756 25728 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1399 CHEMBL578504 37757 25729 HMGCR 3156 ENZYME, DRUGGABLE GENOME LOVASTATIN LOVASTATIN 37758 25730 MALAT1 378938 NA SKL-NP 37760 25731 CA9 768 DRUGGABLE GENOME, ENZYME inhibitor 381118859 37761 25732 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME AZD-1080 AZD-1080 37762 25733 NCF2 4688 NA PMA 9794433 37763 25734 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TH-4000 37764 25735 MAPT 4137 DRUGGABLE GENOME BROMOENOL LACTONE BROMOENOL LACTONE 37766 25736 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 37767 25737 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 328083490 37768 25738 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CLIOXANIDE CLIOXANIDE 37769 25739 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL131 PREDNISOLONE 37770 25740 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 252166729 AZD-8186 37771 25741 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 249565698 37772 25742 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Sunitinib SUNITINIB 19366796,18955458 37773 25743 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C20 37776 25744 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651103 37779 25745 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 12-CHLOROEVODIAMINE CHEMBL2171803 22867019 37780 25746 FAAH 2166 ENZYME, DRUGGABLE GENOME Ethylaminopyrimidine derivative 1 37782 25747 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE ENMD 2076 37783 25748 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NAPHTHALEN-1-YLAMINE CHEMBL57394 37784 25749 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL285674 ESTAZOLAM 37785 25750 FST 10468 DRUGGABLE GENOME ANDROGENS 14512439 37787 25751 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL258940 FALNIDAMOL 37790 25752 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MT-110 37791 25753 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ERYTHROMYCIN ERYTHROMYCIN 37797 25754 SLC9A3 6550 DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE, EXCHANGER AVE-0657 37798 25755 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HERZYME 37799 25756 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NIACIN NIACIN 22931300 37801 25757 XPO1 7514 CLINICALLY ACTIONABLE, KINASE LEPTOMYCIN B LEPTOMYCIN B 18835718 37802 25758 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER CYCLOSPORIN A 11189941 37803 25759 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROSTAGLANDIN A2 PROSTAGLANDIN A2 37804 25760 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR STREPTONIGRIN STREPTONIGRIN 37806 25761 CBX1 10951 NA BAY-11-7082 CHEMBL403183 37807 25762 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME inhibitor 381744900 37809 25763 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR LEVONORGESTREL LEVONORGESTREL 37810 25764 AQP1 358 ION CHANNEL, DRUGGABLE GENOME GLYBURIDE GLYBURIDE 14759764 37812 25765 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 252166839 37815 25766 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ADENOSINE TRIPHOSPHATE ADENOSINE TRIPHOSPHATE 16415863 37816 25767 MAPT 4137 DRUGGABLE GENOME GNF-PF-67 CHEMBL578512 37817 25768 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR EPINEPHRINE EPINEPHRINE 37818 25769 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-4242 CHEMBL584514 37819 25770 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Binimetinib BINIMETINIB 28284557,27307593,23414587,28152546,11238126,24569456,28514312 37821 25771 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENOVERINE FENOVERINE 37822 25772 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652545 37823 25773 TCF19 6941 TRANSCRIPTION FACTOR nevirapine NEVIRAPINE 21810746 37824 25774 UGT1A10 54575 DRUGGABLE GENOME, ENZYME ETOPOSIDE ETOPOSIDE 12695347 37825 25775 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102927 37826 25776 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME IRL-2500 CHEMBL72410 37828 25777 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME ENMD-2076 ENMD-2076 37831 25778 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 363894216 TUCATINIB 37833 25779 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME EPINEPHRINE EPINEPHRINE 37834 25780 CD82 3732 DRUGGABLE GENOME, CELL SURFACE NERVE GROWTH FACTOR 10353759 37835 25781 MPHOSPH8 54737 NA R(-)-PROPYLNORAPOMORPHINE HCL CHEMBL538542 37836 25782 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR EDARAVONE EDARAVONE 37837 25783 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GNF-PF-3201 CHEMBL581872 37838 25784 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME EVOXINE EVOXINE 37840 25785 POLI 11201 DNA REPAIR TDR77578 CHEMBL1364172 37847 25786 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 135650713 37849 25787 ABAT 18 DRUGGABLE GENOME, ENZYME Pyruvic acid 37852 25788 MAPT 4137 DRUGGABLE GENOME GNF-PF-1852 CHEMBL533293 37853 25789 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Acyl piperidine derivative 3 37854 25790 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME GNF-PF-4459 CHEMBL585502 37855 25791 ARG1 383 ENZYME inhibitor 178101800 37856 25792 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650582 37857 25793 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Binimetinib BINIMETINIB 26206338,26577700 37858 25794 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE IVOSIDENIB IVOSIDENIB 31300360,29860938 37859 25795 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PF-04217903 PF-04217903 27659046 37861 25796 TUBA3C 7278 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 37862 25797 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PLATELET-DERIVED GROWTH FACTOR (PDGF) 37863 25798 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 37865 25799 GMNN 51053 DRUGGABLE GENOME TDR77582 CHEMBL1329349 37866 25800 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL636 RIVASTIGMINE 37867 25801 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 405560192 37868 25802 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Malathion MALATHION 37869 25803 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR MOR103 OTILIMAB 37870 25804 SERPING1 710 DRUGGABLE GENOME, PROTEASE INHIBITOR C1-INH 37871 25805 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Indole-based analog 13 37872 25806 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Cisplatin CISPLATIN 37873 25807 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR asparaginase ASPARAGINASE 24141364 37875 25808 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 249565846 37876 25809 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody 178103464 CETUXIMAB 37877 25810 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR MELANOMA VACCINE 10093041 37878 25811 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 8 37882 25812 IL1B 3553 KINASE, DRUGGABLE GENOME ACNU 2350191,1331350 37883 25813 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR DNDI1417941 CHEMBL2095095 37884 25814 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PREDNISOLONE PREDNISOLONE 37885 25815 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TAMATINIB R-406 37890 25816 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Bapineuzumab BAPINEUZUMAB 37891 25817 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME STICTIC ACID STICTIC ACID 37892 25818 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PYRROLIDINE DITHIOCARBAMATE PYRROLIDINE DITHIOCARBAMATE 37893 25819 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 405560192 37894 25820 PDE4A 5141 DRUGGABLE GENOME, ENZYME AN-2728 CRISABOROLE 37895 25821 ADM 133 DRUGGABLE GENOME, HORMONE ACTIVITY INDOMETHACIN INDOMETHACIN 10830296 37897 25822 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 135651484 ESTRONE 37898 25823 SMN2 6607 DRUGGABLE GENOME CID 893238 CHEMBL473735 37899 25824 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CLOTIAZEPAM CLOTIAZEPAM 37900 25825 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID29757691-Compound-4 37902 25826 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Momelotinib MOMELOTINIB 37904 25827 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL2104986 TEDATIOXETINE 37909 25828 EGFL7 51162 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL2109387 PARSATUZUMAB 37910 25829 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE DG051 37912 25830 ATXN2 6311 NA 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 37913 25831 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE Pro-urokinase 37914 25832 EGLN2 112398 ENZYME, DRUGGABLE GENOME FG-4592 ROXADUSTAT 37917 25833 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR VITAMIN C 11120850 37918 25834 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL1059 PREGABALIN 37920 25835 MAPT 4137 DRUGGABLE GENOME GARCINONE E GARCINONE E 37922 25836 RACGAP1 29127 NA MITOXANTRONE MITOXANTRONE 37923 25837 GMNN 51053 DRUGGABLE GENOME GNF-PF-4832 CHEMBL601137 37924 25838 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME ACETAMINOPHEN ACETAMINOPHEN 22136404 37926 25839 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 178101770 37927 25840 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 404859073 37928 25841 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME antagonist 340590216 37929 25842 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME ezetimibe / rosuvastatin 37930 25843 DUSP3 1845 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE 1,4-DIMETHOXYANTHRAQUINONE 1,4-DIMETHOXYANTHRAQUINONE 37932 25844 NDUFAB1 4706 NA inhibitor CHEMBL3545135 NV-128 37934 25845 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 310264778 37935 25846 PTCH1 5727 CLINICALLY ACTIONABLE, TRANSPORTER Vismodegib VISMODEGIB 37936 25847 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 363894182 37937 25848 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME leucovorin LEUCOVORIN 24018773,24338217,20530282 37938 25849 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650039 37940 25850 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GC1118 26586721 37941 25851 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ADAPALENE ADAPALENE 37943 25852 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649876 37944 25853 RTN4 57142 DRUGGABLE GENOME ATI-355 ATINUMAB 22544872 37945 25854 PPP2CA 5515 PROTEIN PHOSPHATASE, ENZYME, KINASE VP-102 37947 25855 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE carbasalate calcium 37948 25856 CHRNA5 1138 DRUGGABLE GENOME, ION CHANNEL antagonist 178100835 37949 25857 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE Radiotherapy 27615706,28652249 37950 25858 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE antibody 384403634 37952 25859 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-111847 CHEMBL1984884 37953 25860 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417523 CHEMBL598663 37954 25861 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE DAMGO DAMGO 24613457,18380425,20235611 37955 25862 CD55 1604 DRUGGABLE GENOME, CELL SURFACE Coxsackievirus A21 37956 25863 ESRRG 2104 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650213 37957 25864 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SALMETEROL XINAFOATE SALMETEROL XINAFOATE 37960 25865 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME (4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE (4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE 37961 25866 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-46 37962 25867 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135650142 CV-6209 37963 25868 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Sorafenib SORAFENIB 23629727,26743856,24166906 37964 25869 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor BGJ398 INFIGRATINIB 37965 25870 ZEB1 6935 TRANSCRIPTION FACTOR, DRUG RESISTANCE DOXORUBICIN DOXORUBICIN 24013721 37966 25871 HES1 3280 TRANSCRIPTION FACTOR ALL-TRANS-RETINOIC ACID 12080040 37967 25872 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER RUBOXISTAURIN HYDROCHLORIDE 37969 25873 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER (Z)-PIPLARTINE (Z)-PIPLARTINE 37970 25874 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR CUDC-101 CUDC-101 37972 25875 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-123532 CHEMBL547833 37973 25876 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE COLCHICINE COLCHICINE 37974 25877 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME Dilmapimod DILMAPIMOD 37978 25878 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME RAPAMYCIN SIROLIMUS 15782132 37979 25879 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HYDROXYPROGESTERONE HYDROXYPROGESTERONE 37980 25880 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GDC-0994 RAVOXERTINIB 25320010 37981 25881 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL NITRAZEPAM NITRAZEPAM 37982 25882 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CHEMOKINES 11747824 37983 25883 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor REGORAFENIB REGORAFENIB 37984 25884 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 37985 25885 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE MEROPENEM MEROPENEM 8354907 37986 25886 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-4029 CHEMBL596633 37987 25887 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor 178103188 37989 25888 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE TRODUSQUEMINE TRODUSQUEMINE 37990 25889 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME LINIFANIB LINIFANIB 37991 25890 HSPB1 3315 DRUGGABLE GENOME CYROMAZINE CYROMAZINE 37992 25891 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME ALCLOMETASONE ALCLOMETASONE 37993 25892 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AG-537 CHEMBL67535 37994 25893 CDC42BPB 9578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565884 A-443654 37996 25894 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Nafamostat NAFAMOSTAT 37998 25895 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-29 38002 25896 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 223366022 38005 25897 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL289351 FOSBRETABULIN DISODIUM 38006 25898 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ibuprofen IBUPROFEN 25502615 38007 25899 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SB-200646 CHEMBL85194 38009 25900 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TANSHINONE IIA TANSHINONE IIA 38011 25901 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL METHYLPHENOBARBITAL MEPHOBARBITAL 38012 25902 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ZIDOVUDINE ZIDOVUDINE 22931300 38013 25903 KDM4A 9682 DRUGGABLE GENOME, ENZYME PMID25468267-Compound-46 38017 25904 HSPA4 3308 NA HALOPERIDOL HALOPERIDOL 9864262 38018 25905 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PEMBROLIZUMAB PEMBROLIZUMAB 27433843 38019 25906 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME CHEMOTHERAPEUTIC AGENT 16170020 38020 25907 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL48582 SAFINAMIDE MESYLATE 38022 25908 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ifosfamide IFOSFAMIDE 12386121,19702528,19442086,11038165,14704462,8886611 38023 25909 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE LEE011 RIBOCICLIB 38024 25910 ABL2 27 KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME PONATINIB PONATINIB 20513156 38025 25911 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Isoflavone derivative 2 38026 25912 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135650401 38029 25913 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME VEGF-121 38030 25914 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FINASTERIDE FINASTERIDE 22931300 38031 25915 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DASATINIB DASATINIB 38033 25916 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXYQUINOLINE OXYQUINOLINE 38034 25917 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 toremifene TOREMIFENE 9187528 38035 25918 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417457 CHEMBL1530911 38038 25919 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417207 CHEMBL256062 38040 25920 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GW0742 CHEMBL38508 38042 25921 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SJ000189154 CHEMBL604664 38043 25922 TUBA3D 113457 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 38044 25923 POLK 51426 DNA REPAIR, ENZYME PINAFIDE PINAFIDE 38045 25924 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SR 4233 8461036 38046 25925 CD3D 915 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE MT110 SOLITOMAB 38047 25926 SOD2 6648 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ANTIOXIDANT 12007958 38048 25927 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR APOMINE 38051 25928 CCL21 6366 DRUGGABLE GENOME CXC CHEMOKINES 10737895 38054 25929 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ENROFLOXACIN ENROFLOXACIN 38055 25930 NRP1 8829 DRUGGABLE GENOME PEGAPTANIB PEGAPTANIB SODIUM 38057 25931 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE BIIB 022 38058 25932 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NSC-95397 CHEMBL429095 38059 25933 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Pertuzumab PERTUZUMAB 22586653,23801166,23940356,27052654,28539475 38060 25934 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE inhibitor RO4929097 RG-4733 38063 25935 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME perhexiline PERHEXILINE 38065 25936 HSPB1 3315 DRUGGABLE GENOME OESTROGENS 7926277 38066 25937 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CARBIDOPA CARBIDOPA 38067 25938 CD3D 915 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE ANTI-CD3 MONOCLONAL ANTIBODY 38069 25939 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650735 NORMORPHINE 38070 25940 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DASATINIB DASATINIB 38071 25941 SMN1 6606 DRUGGABLE GENOME PICEATANNOL PICEATANNOL 38073 25942 UBE2N 7334 ENZYME, DRUGGABLE GENOME GNF-PF-254 CHEMBL461579 38074 25943 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL403989 TG100-801 38076 25944 FGA 2243 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, FIBRINOGEN eptifibatide EPTIFIBATIDE 20938371 38077 25945 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Ralimetinib RALIMETINIB 26725216 38080 25946 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 1-(4-HYDROXYPHENYL)MALEIMIDE CHEMBL565893 38081 25947 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER flupenthixol E-FLUPENTIXOL 38082 25948 RIPK3 11035 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 384403667 38083 25949 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL GC021109 38084 25950 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR CDP6038 OLOKIZUMAB 38085 25951 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PMID29130358-Compound-Figure18(14a) 38086 25952 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 L-687384 CHEMBL303336 38087 25953 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR tiratricol TIRATRICOL 38089 25954 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DESIPRAMINE DESIPRAMINE 38091 25955 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-40 38092 25956 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Alvespimycin ALVESPIMYCIN 26009011 38095 25957 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE L-796568 CHEMBL111201 38096 25958 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE TAMOXIFEN TAMOXIFEN 15138475 38097 25959 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR TCDD 16080534 38098 25960 APH1B 83464 PROTEASE, DRUGGABLE GENOME BMS-708163 AVAGACESTAT 38101 25961 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 38102 25962 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE GLPG-1837 38104 25963 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200841 PROCAINE HYDROCHLORIDE 38105 25964 ALDH1A1 216 DRUGGABLE GENOME, ENZYME RETINYL ACETATE RETINYL ACETATE 38106 25965 TUBA3C 7278 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 38107 25966 ALPI 248 DRUGGABLE GENOME, ENZYME 2-AMINOPHENOXAZINONE CHEMBL146710 38111 25967 PABPC1 26986 NA GNF-PF-4618 CHEMBL585964 38112 25968 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR LGX818 ENCORAFENIB 27312529 38113 25969 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1201577 CETUXIMAB 38114 25970 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID25399719-Compound-17 38115 25971 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GEFITINIB GEFITINIB 16282176 38116 25972 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 3-FLUOROEVODIAMINE CHEMBL2171781 22867019 38117 25973 GMNN 51053 DRUGGABLE GENOME CAPTAN CAPTAN 38118 25974 XDH 7498 DRUGGABLE GENOME, ENZYME ALLOPURINOL ALLOPURINOL 38119 25975 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-1509 CHEMBL576412 38120 25976 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PMID30107136-Compound-Example1 38121 25977 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE inhibitor CHEMBL3833374 ANDECALIXIMAB 38123 25978 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME GW3965 CHEMBL59030 38124 25979 DTNBP1 84062 KINASE corticosteroids 30697902 38126 25980 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DNDI1417467 CHEMBL1997335 38128 25981 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PCB 12230110 38129 25982 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Levormeloxifene non-steroidal 38130 25983 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 363894199 38131 25984 CRYBG2 55057 NA opioids 38135 25985 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Hexahydro quinoline derivative 1 38136 25986 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL1213490 ROMIDEPSIN 38138 25987 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AZATHIOPRINE AZATHIOPRINE 22931300 38139 25988 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651453 N6-CYCLOPENTYLADENOSINE 38140 25989 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE NINTEDANIB NINTEDANIB 38142 25990 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 38143 25991 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist 310264729 38144 25992 CDC42 998 DRUGGABLE GENOME GNRH GONADORELIN ACETATE 9626657 38146 25993 GBA 2629 DRUGGABLE GENOME, ENZYME Isofagomine tartrate 38147 25994 KMT5A 387893 ENZYME inhibitor 178103601 38149 25995 ABCB11 8647 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE pravastatin PRAVASTATIN 38151 25996 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MGL-3196 RESMETIROM 38153 25997 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CISPLATIN CISPLATIN 38154 25998 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TPCK TPCK 38155 25999 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME lifitegrast LIFITEGRAST 38156 26000 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200450 TRIPROLIDINE HYDROCHLORIDE 38157 26001 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME 2-(1-CYCLODODECYLETHYLIDENE)HYDRAZINECARBOTHIOAMIDE CHEMBL2316602 23350811 38158 26002 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 imatinib IMATINIB 38159 26003 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE Ouabain OUABAIN 38161 26004 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 354702275 38162 26005 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Daunoxome DAUNORUBICIN 16243804 38163 26006 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CARMINOMYCIN CARUBICIN 38164 26007 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 385612218 38165 26008 DHRS9 10170 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE PROTECTED SIPHONODICTYAL C PROTECTED SIPHONODICTYAL C 19188072 38166 26009 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DEXFENFLURAMINE DEXFENFLURAMINE 38168 26010 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR lapatinib LAPATINIB 38169 26011 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103934 38170 26012 COQ2 27235 ENZYME hmg coa reductase inhibitors 20347093 38171 26013 TOP2B 7155 DRUGGABLE GENOME, ENZYME Dhaq diacetate 38173 26014 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER APR-246 APR-246 22965953,21239882,21415220,26086967,27179933 38174 26015 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME LY-2090314 LY-2090314 38175 26016 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3137308 PEFICITINIB 38177 26017 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME modulator CHEMBL3545278 ATX08-001 38178 26018 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 310264675 CUDC-101 38179 26019 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ELLAGIC ACID ELLAGIC ACID 38180 26020 FAAH 2166 ENZYME, DRUGGABLE GENOME Boronic acid derivative 4 38182 26021 SMN2 6607 DRUGGABLE GENOME 7-HYDROXY ISOFLAVONE 7-HYDROXY ISOFLAVONE 38183 26022 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor 178103413 DICHLORPHENAMIDE 38185 26023 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR tacrolimus TACROLIMUS 24658827,24113216,29399716 38186 26024 MAPT 4137 DRUGGABLE GENOME CONGO RED CONGO RED 38188 26025 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROGESTERONE PROGESTERONE 38189 26026 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor XL228 XL-228 38190 26027 RAC1 5879 CLINICALLY ACTIONABLE, KINASE, DRUG RESISTANCE TCMDC-124310 CHEMBL579882 38191 26028 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135649873 A-349,821 38192 26029 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE GS-9901 GS-9901 38194 26030 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TASOSARTAN TASOSARTAN 38195 26031 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TRIIODOTHYRONINE LIOTHYRONINE SODIUM 9770474 38197 26032 NOS1 4842 DRUGGABLE GENOME, ENZYME inhibitor 363894143 GW-274150 38198 26033 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody BIIB022 38199 26034 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LISDEXAMFETAMINE LISDEXAMFETAMINE 38200 26035 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE PSYLLIUM PSYLLIUM SEED HUSKS 10696527 38201 26036 SUMO2 6613 ENZYME HEXACHLOROPHENE HEXACHLOROPHENE 38202 26037 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TIMOLOL TIMOLOL 2903243 38203 26038 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-128437 CHEMBL1370698 38204 26039 PSMA6 5687 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL371405 MARIZOMIB 38205 26040 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651190 38207 26041 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE DOVITINIB DOVITINIB 38208 26042 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME EUPAFOLIN EUPAFOLIN 38211 26043 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Infliximab INFLIXIMAB 38213 26044 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME LEVODOPA LEVODOPA 38214 26045 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DILTIAZEM DILTIAZEM 22931300 38215 26046 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AR-A014418 CHEMBL259850 38217 26047 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHANQUONE PHANQUONE 38218 26048 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR KEPONE KEPONE 38219 26049 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME CUDC-101 CUDC-101 38222 26050 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME PF-562271 PF-00562271 38223 26051 IL23A 51561 DRUGGABLE GENOME USTEKINUMAB USTEKINUMAB 38224 26052 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DIGITOXIN DIGITOXIN 38225 26053 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE antipsychotics 38226 26054 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER nitrendipine NITRENDIPINE 38228 26055 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-50688 CHEMBL1456848 38230 26056 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ALPRAZOLAM ALPRAZOLAM 38235 26057 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist CHEMBL3545275 LY2623091 38237 26058 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE DEXAMETHASONE DEXAMETHASONE 2707640,3398844 38238 26059 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TANSHINONE IIA TANSHINONE IIA 22175694 38239 26060 SMOX 54498 ENZYME, DRUGGABLE GENOME AZASERINE AZASERINE 7899459 38241 26061 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME COLCHICINE COLCHICINE 12815172 38247 26062 STK16 8576 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 38249 26063 NDUFAF3 25915 NA inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 38250 26064 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-53 38251 26065 MAPT 4137 DRUGGABLE GENOME 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 38252 26066 CYBB 1536 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME, ENZYME inhibitor 363894229 38253 26067 CYP24A1 1591 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME VITAMIN D 15225763 38254 26068 MAP3K9 4293 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 328083457 38255 26069 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 5-AZADEOXYCYTIDINE DECITABINE 11948118,11960994 38256 26070 PTGS2 5743 DRUGGABLE GENOME, ENZYME Rofecoxib ROFECOXIB 38257 26071 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE S-(+)-FLUOXETINE HCL CHEMBL1257031 38258 26072 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME activator 53801079 38261 26073 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 178102344 TOZASERTIB 38263 26074 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL1213490 ROMIDEPSIN 38264 26075 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE DMSO DIMETHYL SULFOXIDE 9678720 38266 26076 IL1B 3553 KINASE, DRUGGABLE GENOME tiludronate TILUDRONIC ACID 16257277 38268 26077 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor TAK-733 TAK-733 38270 26078 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE TACROLIMUS TACROLIMUS 38271 26079 VKORC1 79001 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1466 DICUMAROL 38274 26080 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR QUERCETIN QUERCETIN 17045724 38276 26081 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor VELIPARIB VELIPARIB 38277 26082 TSPO 706 DRUGGABLE GENOME Quinoline carboxamide derivative 10 38278 26083 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 375973252 38280 26084 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME MARIMASTAT MARIMASTAT 38283 26085 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR TIPLASININ TIPLASININ 17276980 38285 26086 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Crizotinib CRIZOTINIB 38286 26087 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100541 PRANLUKAST 38289 26088 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME TAE-684 TAE-684 38290 26089 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER paclitaxel PACLITAXEL 21151855 38293 26090 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3218576 COPANLISIB 38295 26091 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL ADX N05 38296 26092 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GNF-PF-2347 CHEMBL579045 38297 26093 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME FURAFYLLINE FURAFYLLINE 38298 26094 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROTEIN PHOSPHATASE INHIBITOR 12446695 38299 26095 DHRS9 10170 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE (+/-)-SPONGIAQUINONE CHEMBL514876 19188072 38300 26096 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME GO-6976 GO-6976 38301 26097 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME CLOPIDOGREL CLOPIDOGREL 38302 26098 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME OCTADEC-17-YNOIC ACID CHEMBL182310 38303 26099 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200409 LIDOCAINE HYDROCHLORIDE 38305 26100 CA1 759 DRUGGABLE GENOME, ENZYME activator 135651493 HISTAMINE 38306 26101 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR BENZOQUINONE BENZOQUINONE 38308 26102 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE AG140699 38309 26103 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 astemizole ASTEMIZOLE 9187528 38310 26104 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 38311 26105 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX Tazarotene TAZAROTENE 38312 26106 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CENISERTIB CENISERTIB 38313 26107 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Bicyclic heteroaryl benzamide derivative 7 38314 26108 BBOX1 8424 DRUGGABLE GENOME BENZENE SELENOIC ACID BENZENE SELENOIC ACID 25266780 38315 26109 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SN-32793 38317 26110 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE GW632580X GW632580X 38318 26111 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE LEUKOCYTE INTERFERON CETUXIMAB 3085922 38319 26112 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME INHIBITOR 26859458 38322 26113 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME GNF-PF-5159 CHEMBL1493528 38323 26114 PDE4A 5141 DRUGGABLE GENOME, ENZYME LIRIMILAST LIRIMILAST 18660832 38324 26115 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL79 LIDOCAINE 38325 26116 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL1201752 IXABEPILONE 38327 26117 USP1 7398 DNA REPAIR, PROTEASE, ENZYME IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 38328 26118 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 38329 26119 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-40 38330 26120 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR OSI-632 OSI-632 38331 26121 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DAUNORUBICIN DAUNORUBICIN 38334 26122 KAT2B 8850 ENZYME, DRUGGABLE GENOME inhibitor 178103580 GARCINOL 38336 26123 GMNN 51053 DRUGGABLE GENOME SOFALCONE SOFALCONE 38339 26124 GAA 2548 DRUGGABLE GENOME, ENZYME NSC-19803 CHEMBL522983 38340 26125 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME BERKELEYACETAL B BERKELEYACETAL B 17970594 38342 26126 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE XL647 TESEVATINIB 22722787 38343 26127 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE T8361 38345 26128 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME SNS-314 SNS-314 38346 26129 FPGS 2356 ENZYME, DRUGGABLE GENOME 5-FU FLUOROURACIL 9291820 38347 26130 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME RG-1530 RG-1530 38348 26131 MPHOSPH8 54737 NA FLUPIRTINE MALEATE FLUPIRTINE MALEATE 38349 26132 RORB 6096 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, KINASE agonist 310264687 38351 26133 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Indoline derivative 12 38352 26134 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR activator BEXAROTENE BEXAROTENE 38353 26135 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650838 38354 26136 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417099 CHEMBL1565444 38356 26137 KLKB1 3818 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166701 38357 26138 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER N-(3-CARBOXYPHENYL)RHODANINE CHEMBL442906 38358 26139 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LABETALOL LABETALOL 38359 26140 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CHLORPROMAZINE HYDROCHLORIDE CHLORPROMAZINE HYDROCHLORIDE 38360 26141 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DEBIO 0932 38361 26142 MRM2 29960 NA Plazomicin PLAZOMICIN 38364 26143 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 dronedarone DRONEDARONE 38365 26144 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL SA-5845 38366 26145 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Cyclophosphamide CYCLOPHOSPHAMIDE 17388661,16243804,26438783 38368 26146 CYP4F11 57834 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 warfarin WARFARIN 28620303 38369 26147 FBP1 2203 DRUGGABLE GENOME, ENZYME Managlinat dialanetil 38370 26148 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TRIFLUOPERAZINE HYDROCHLORIDE TRIFLUOPERAZINE HYDROCHLORIDE 38372 26149 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 315661268 38373 26150 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PIOGLITAZONE PIOGLITAZONE 24890090,15745794,21030263,16680159 38377 26151 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL DIQUAFOSOL DIQUAFOSOL 38379 26152 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545247 CAL-263 38380 26153 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER docetaxel DOCETAXEL 21151855 38381 26154 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MELOXICAM MELOXICAM 38383 26155 SFRP5 6425 DRUGGABLE GENOME Bisphosphonates 38384 26156 ALPL 249 ENZYME, DRUGGABLE GENOME DIHYDRODAPHNODORIN B DIHYDRODAPHNODORIN B 38385 26157 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PROTEASOME INHIBITOR 17159161 38386 26158 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 11 38387 26159 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor DABRAFENIB DABRAFENIB 38388 26160 POLK 51426 DNA REPAIR, ENZYME RUTIN RUTIN 38389 26161 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TCMDC-125620 CHEMBL530291 38390 26162 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER (+)-THALIPORPHINE CHEMBL1397308 38391 26163 PEBP1 5037 KINASE, PROTEASE INHIBITOR FLUTAMIDE FLUTAMIDE 12377983 38392 26164 RGS4 5999 DRUGGABLE GENOME TRIFLUOPERAZINE TRIFLUOPERAZINE 38393 26165 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178103707 BROMFENAC 38394 26166 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR KEPONE KEPONE 38397 26167 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE DNDI1417467 CHEMBL1997335 38398 26168 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AM-404 CHEMBL39878 38400 26169 IDE 3416 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, ENZYME, PROTEASE inhibitor 252166800 38402 26170 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME PLATINUM COMPOUND 24961465 38403 26171 TGFBR3 7049 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME antidepressants 23092981 38405 26172 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL1801204 AZD-8055 38406 26173 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200323 LABETALOL HYDROCHLORIDE 38407 26174 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME EPIRUBICIN EPIRUBICIN 16608080 38408 26175 CD200 4345 CELL SURFACE, DRUGGABLE GENOME ALXN6000 SAMALIZUMAB 21559315 38409 26176 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CLENBUTEROL CLENBUTEROL 16680159 38410 26177 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565818 38411 26178 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR STZ STREPTOZOCIN 8482431 38413 26179 POLB 5423 DNA REPAIR, DRUGGABLE GENOME DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 38414 26180 GMNN 51053 DRUGGABLE GENOME N-ETHYLMALEIMIDE N-ETHYLMALEIMIDE 38416 26181 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME AZD-1152-HQPA AZD-1152-HQPA 38417 26182 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL3545389 LY2245461 38422 26183 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR IMIPRAMINE IMIPRAMINE 16522641 38423 26184 GAL 51083 DRUGGABLE GENOME DHEA PRASTERONE 12195234 38424 26185 ACP1 52 ENZYME, DRUGGABLE GENOME, PROTEIN PHOSPHATASE CEFDINIR CEFDINIR 38425 26186 SMN1 6606 DRUGGABLE GENOME DAIDZEIN DAIDZEIN 38426 26187 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE DCC-2618 RIPRETINIB 38427 26188 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178100909 38428 26189 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE EFAVIRENZ EFAVIRENZ 21189339,17172311 38430 26190 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME OXYTETRACYCLINE OXYTETRACYCLINE 38431 26191 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135652706 38432 26192 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL1258517 PKI-179 38433 26193 RAB9A 9367 ENZYME, DRUGGABLE GENOME NICLOSAMIDE NICLOSAMIDE 38434 26194 FAAH 2166 ENZYME, DRUGGABLE GENOME clozapine CLOZAPINE 20631561 38436 26195 EPHA3 2042 ENZYME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 38437 26196 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME PMID27998201-Compound-12 38438 26197 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-METHOXY-1,4-NAPHTHOQUINONE 2-METHOXY-1,4-NAPHTHOQUINONE 38441 26198 SOD2 6648 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE valproic acid 38442 26199 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-24 38444 26200 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME IDARUBICIN IDARUBICIN 38445 26201 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BAY80-6946 COPANLISIB 38446 26202 TLR7 51284 DRUGGABLE GENOME CHLOROQUINE CHLOROQUINE 19949061,22239408 38448 26203 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor CHEMBL3545137 PF-00477736 38450 26204 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 310264778 38451 26205 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE PEMETREXED PEMETREXED 38452 26206 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ENZALUTAMIDE ENZALUTAMIDE 25634130 38453 26207 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL2105741 TRAMETINIB DIMETHYL SULFOXIDE 38454 26208 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Carbamide derivative 19 38455 26209 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR JNJ-7706621 JNJ-7706621 38456 26210 TNFRSF18 8784 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME INCAGN1876 38458 26211 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Curcumin analog 1 38461 26212 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME CLASTO-LACTACYSTIN BETA-LACTONE CHEMBL490829 18801655 38462 26213 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE US8889672, 252-036-001 38463 26214 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DERRUBONE DERRUBONE 38464 26215 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME BAY-613606 CHEMBL541400 38467 26216 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor SCH727965 DINACICLIB 38468 26217 DCLK1 9201 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TAE-684 TAE-684 38469 26218 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX EPIRUBICIN HYDROCHLORIDE EPIRUBICIN HYDROCHLORIDE 38470 26219 SIK3 23387 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 340590212 38471 26220 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LAWSONE LAWSONE 38472 26221 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor RECENTIN CEDIRANIB 38475 26222 DDIT4 54541 NA PF-04523655 38476 26223 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CLORAZEPATE CLORAZEPIC ACID 38477 26224 FGF1 2246 CLINICALLY ACTIONABLE, GROWTH FACTOR, DRUGGABLE GENOME CVBT-141H 38478 26225 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-4 38479 26226 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651087 NELIVAPTAN 38481 26227 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE carboplatin CARBOPLATIN 22901187 38484 26228 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME GNF-PF-254 CHEMBL461579 38485 26229 MAPT 4137 DRUGGABLE GENOME CURCUMIN CURCUMIN 38487 26230 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME METHOTREXATE METHOTREXATE 10732770 38489 26231 SCAP 22937 TRANSCRIPTION FACTOR atorvastatin ATORVASTATIN 18435918 38491 26232 BAZ2B 29994 NA DIHYDROERGOCRISTINE MESYLATE DIHYDROERGOCRISTINE MESYLATE 38493 26233 MGLL 11343 DRUGGABLE GENOME, ENZYME inhibitor 375973216 38494 26234 MAPT 4137 DRUGGABLE GENOME DIHYDROERGOTAMINE MESYLATE DIHYDROERGOTAMINE MESYLATE 38495 26235 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL25 ASPIRIN 38496 26236 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 252827496 38497 26237 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MB-07811 MB07811 38498 26238 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DAIDZEIN DAIDZEIN 16038533 38499 26239 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SIBUTRAMINE HYDROCHLORIDE SIBUTRAMINE HYDROCHLORIDE 38500 26240 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME N-(3-OXODODECANOYL)HOMOSERINELACTONE CHEMBL8483 18566250 38502 26241 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 223366077 RGB-286638 38503 26242 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ABBV-399 TELISOTUZUMAB VEDOTIN 27573171 38504 26243 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL284348 DALFAMPRIDINE 38505 26244 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 328083524 LENIOLISIB 38506 26245 HTT 3064 DRUGGABLE GENOME FLUOROSALAN FLUOROSALAN 38508 26246 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME VBY- 891 38509 26247 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor REGORAFENIB REGORAFENIB 38510 26248 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor XL-765 VOXTALISIB 38511 26249 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER gramicidin d 38512 26250 ECE2 9718 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252166821 38513 26251 PSMA8 143471 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL2103884 OPROZOMIB 38514 26252 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GNF-PF-3023 CHEMBL535331 38515 26253 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000293754 CHEMBL486706 38517 26254 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545052 FIMEPINOSTAT 38523 26255 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE BLEOMYCIN BLEOMYCIN 15855637 38524 26256 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Debio 1347 38525 26257 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor BMN673 38526 26258 BRDT 676 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE PMID26924192-Compound-105 38527 26259 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ENTRECTINIB ENTRECTINIB 38529 26260 LTC4S 4056 ENZYME, DRUGGABLE GENOME inhibitor 336446942 38530 26261 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ixabepilone IXABEPILONE 38531 26262 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME Pyrazolones 26398624 38533 26263 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor 363894172 38534 26264 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR BPTES 28346230 38535 26265 TUBA4A 7277 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 38536 26266 DHODH 1723 DRUGGABLE GENOME, ENZYME LEFLUNOMIDE LEFLUNOMIDE 38538 26267 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor PF00562271 38540 26268 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROTOPORPHYRIN PROTOPORPHYRIN 38542 26269 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TAMIBAROTENE TAMIBAROTENE 38543 26270 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE Carboplatin CARBOPLATIN 28514312 38544 26271 HSPB1 3315 DRUGGABLE GENOME DNDI1417169 CHEMBL2094499 38545 26272 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME AZD-1152-HQPA AZD-1152-HQPA 38546 26273 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FPL-55712 FPL-55712 38547 26274 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 178103494 IBRUTINIB 38551 26275 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 135649959 AMMONIUM TRICHLOROTELLURATE 38552 26276 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Chalcone derivative 5 38553 26277 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Linsitinib LINSITINIB 26561558 38554 26278 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME AE-941 38555 26279 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME CYC-116 CYC-116 38557 26280 POLK 51426 DNA REPAIR, ENZYME 7,8,3'-TRIHYDROXYFLAVONE CHEMBL225513 38558 26281 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PREDNISOLONE ACETATE PREDNISOLONE ACETATE 38559 26282 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TPCK TPCK 38560 26283 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME brivanib BRIVANIB 20124951 38561 26284 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TG-02 ZOTIRACICLIB 22148278 38562 26285 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 3R14S-OCHRATOXIN A 3R14S-OCHRATOXIN A 38563 26286 PSME2 5721 NA inhibitor BORTEZOMIB BORTEZOMIB 38565 26287 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME BUTANOIC ACID BUTANOIC ACID 19053749 38566 26288 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565794 38567 26289 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AZACITIDINE AZACITIDINE 38569 26290 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME CENISERTIB CENISERTIB 38570 26291 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 38572 26292 PLD1 5337 ENZYME, DRUGGABLE GENOME US9453017, 2 38573 26293 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR GUGGULSTERONE GUGGULSTERONE 38574 26294 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Nitrogen mustard derivative 1 38575 26295 NDUFA10 4705 ENZYME inhibitor CHEMBL3545320 ME-344 38576 26296 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 38579 26297 COL1A2 1278 DRUGGABLE GENOME IFN 14512876 38581 26298 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE MK-2206 MK-2206 38582 26299 MUC16 94025 DRUGGABLE GENOME N/A 38583 26300 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE Sulfonamide derivative 17 38584 26301 TNKS 8658 DRUGGABLE GENOME, ENZYME inhibitor 404859120 38585 26302 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (S)-VERAPAMIL (S)-VERAPAMIL 38586 26303 ALOX15 246 ENZYME, DRUGGABLE GENOME LY-255283 LY-255283 38587 26304 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE FAS-LIGAND 12730690 38590 26305 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650809 PERGOLIDE 38591 26306 POLK 51426 DNA REPAIR, ENZYME HOE-33342 CHEMBL343002 38592 26307 PTGS2 5743 DRUGGABLE GENOME, ENZYME MELOXICAM MELOXICAM 38593 26308 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor SB939 38595 26309 KDM6B 23135 ENZYME inhibitor 178103606 38596 26310 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME inhibitor 178103578 38597 26311 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VORICONAZOLE VORICONAZOLE 16141569 38599 26312 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IODOPHTHALEIN IODOPHTHALEIN 38603 26313 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME P-toluenesulfonate derivative 1 38604 26314 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PSEUDOEPHEDRINE PSEUDOEPHEDRINE 38606 26315 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR DIOSMETIN DIOSMETIN 25190466 38607 26316 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 404859074 38608 26317 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651501 38612 26318 ACE2 59272 ENZYME, TRANSPORTER, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, CELL SURFACE, PROTEASE ORE-1001 ORE-1001 38613 26319 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALOE-EMODIN ALOE-EMODIN 38615 26320 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL agonist 178101000 38616 26321 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774822-Compound-Figure10Example19 38617 26322 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE TRASTUZUMAB TRASTUZUMAB 20813970,15324695,16404430 38620 26323 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE EVODIAMINE EVODIAMINE 22867019,24103429 38621 26324 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Quinoline and quinazoline derivative 2 38622 26325 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DITHIAZANINE IODIDE DITHIAZANINE IODIDE 38623 26326 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 178102524 38629 26327 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL2048028 LIFITEGRAST 38630 26328 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Abiraterone ABIRATERONE 38631 26329 SMN1 6606 DRUGGABLE GENOME CID 739615 CHEMBL260560 38632 26330 CXCL8 3576 DRUGGABLE GENOME RETINOL RETINOL 38633 26331 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE paclitaxel PACLITAXEL 26179145,20212519 38635 26332 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor MIDOSTAURIN MIDOSTAURIN 38639 26333 HSPG2 3339 KINASE, DRUGGABLE GENOME D-20133 21649580 38640 26334 MAPT 4137 DRUGGABLE GENOME MESNA MESNA 38641 26335 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PMID29671355-Compound-43 38642 26336 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME NNC-0151-0000-0000 38643 26337 LIMK2 3985 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 363894133 38644 26338 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SANGUINARIUM SANGUINARIUM 38645 26339 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME SULFURETIN SULFURETIN 38646 26340 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 8-FLUOROTRYPTANTHRIN CHEMBL1098875 38647 26341 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR DERRUBONE DERRUBONE 18020309 38648 26342 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL1614710 OSI-930 38649 26343 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NALOXONE NALOXONE 14741437 38650 26344 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME GENTIAN VIOLET GENTIAN VIOLET 38651 26345 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SELUMETINIB SELUMETINIB 23515407,22392911 38652 26346 PSMD2 5708 NA CARFILZOMIB CARFILZOMIB 24524217 38653 26347 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE DINOPROSTONE DINOPROSTONE 38655 26348 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 38656 26349 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE 9F7-F11 25216528 38658 26350 CLU 1191 CELL SURFACE, DRUGGABLE GENOME PMSG 1547735 38660 26351 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TRICLOSAN TRICLOSAN 38661 26352 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3,6-DIMETHOXYFLAVONE 3,6-DIMETHOXYFLAVONE 38663 26353 SMN2 6607 DRUGGABLE GENOME CID 670282 CHEMBL260213 38664 26354 CACNA2D3 55799 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL593430 ATAGABALIN 38666 26355 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME ILORASERTIB ILORASERTIB 38667 26356 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME Cobimetinib COBIMETINIB 38668 26357 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 10-METHOXYLRUTAECARPINE CHEMBL85826 38669 26358 GMNN 51053 DRUGGABLE GENOME 2,3,4,4'-TETRAMETHOXYBIPHENYL 2,3,4,4'-TETRAMETHOXYBIPHENYL 38670 26359 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DNDI1417221 CHEMBL1459280 38671 26360 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME INSULIN INSULIN 11600523 38672 26361 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME B-701 VOFATAMAB 38673 26362 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Alpelisib ALPELISIB 38674 26363 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 384403673 38675 26364 IL1B 3553 KINASE, DRUGGABLE GENOME ustekinumab USTEKINUMAB 28696418 38677 26365 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR AG-1879 CHEMBL406845 38678 26366 EGFL7 51162 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE Anti-EGFL7 38679 26367 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR SONIDEGIB SONIDEGIB 26124204 38680 26368 AKR1B1 231 DRUGGABLE GENOME, ENZYME UVB 10391122 38681 26369 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL celecoxib CELECOXIB 22336956 38683 26370 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor BAY80-6946 COPANLISIB 38684 26371 AOX1 316 DRUGGABLE GENOME febuxostat FEBUXOSTAT 27798726 38686 26372 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE DCC-2618 RIPRETINIB 38689 26373 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 38690 26374 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FLUTAMIDE FLUTAMIDE 38691 26375 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650145 38693 26376 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor INC280 CAPMATINIB 38694 26377 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2012810604610 38695 26378 ATAD5 79915 NA QUINACRINE QUINACRINE 38696 26379 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING APICIDIN APICIDIN 19705846 38697 26380 XDH 7498 DRUGGABLE GENOME, ENZYME QUERCETIN QUERCETIN 21474216 38698 26381 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME S-METHYL-D-THIOCITRULLINE S-METHYL-D-THIOCITRULLINE 38699 26382 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE AST-487 AST-487 38700 26383 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LOMEFLOXACIN LOMEFLOXACIN 38701 26384 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TOMUDEX RALTITREXED 10047461 38702 26385 MAPT 4137 DRUGGABLE GENOME PHENAZOPYRIDINE HYDROCHLORIDE PHENAZOPYRIDINE HYDROCHLORIDE 38703 26386 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BETA-CCM BETA-CCM 38704 26387 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-47d 38705 26388 P4HB 5034 THIOREDOXIN, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE LIQUIRITIN LIQUIRITIN 38706 26389 EML4 27436 CLINICALLY ACTIONABLE, KINASE AP26113 CHEMBL3397300 27009859,27432227,25228534,26698910,27780853 38708 26390 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OCTABENZONE OCTABENZONE 38709 26391 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METERGOLINE METERGOLINE 38710 26392 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RESVERATROL RESVERATROL 38711 26393 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE INDOMETHACIN INDOMETHACIN 8557642 38712 26394 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-25 38713 26395 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103951 DINACICLIB 38716 26396 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME ENMD-2076 ENMD-2076 38717 26397 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR Doxorubicin DOXORUBICIN 26936505 38718 26398 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE MESO-2,3-DIMERCAPTOSUCCINIC ACID CHEMBL28721 38719 26399 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Tricyclic heterocycle derivative 5 38720 26400 GMNN 51053 DRUGGABLE GENOME GNF-PF-4029 CHEMBL596633 38721 26401 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL1230165 SILMITASERTIB 38722 26402 NLRP1 22861 PROTEASE agonist 178101721 38724 26403 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR NF-KB DECOY 38725 26404 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CARBOPLATIN CARBOPLATIN 25010864 38726 26405 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PREDNISOLONE PREDNISOLONE 38727 26406 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR SF1126 38728 26407 GPR183 1880 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178101170 38729 26408 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME IONOMYCIN IONOMYCIN 9045668 38730 26409 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 135650713 38731 26410 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Oral azacitidine 38732 26411 S100A12 6283 DRUGGABLE GENOME, KINASE BMS-927711 RIMEGEPANT 38734 26412 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 178102566 38735 26413 CCL21 6366 DRUGGABLE GENOME IMMUNOMODULATORS 14610196 38736 26414 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-47924 CHEMBL1269845 38737 26415 TSPO 706 DRUGGABLE GENOME Eszopiclone ESZOPICLONE 38738 26416 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Erlotinib ERLOTINIB 27207775 38744 26417 TPM3 7170 KINASE, CLINICALLY ACTIONABLE EO9 APAZIQUONE 8509220 38748 26418 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR allosteric modulator 178102297 BMS-345541 38749 26419 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HYDROCORTISONE SODIUM SUCCINATE HYDROCORTISONE SODIUM SUCCINATE 38751 26420 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 38752 26421 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-30 38754 26422 MAPT 4137 DRUGGABLE GENOME ALLOXAN ALLOXAN 38756 26423 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 38761 26424 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME SJ000259188 CHEMBL592578 38763 26425 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-125910 CHEMBL1529609 38766 26426 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME RICININE RICININE 25124862 38768 26427 TYMSOS 494514 NA cytarabine CYTARABINE 38769 26428 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ASTERRIC ACID ASTERRIC ACID 38771 26429 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Pimasertib PIMASERTIB 23629727,26228206 38772 26430 RGMA 56963 CELL SURFACE, KINASE antibody 318164809 ELEZANUMAB 38774 26431 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GOSSYPOL GOSSYPOL 38775 26432 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME E6201 E-6201 23039341 38776 26433 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME VORICONAZOLE VORICONAZOLE 17518356 38778 26434 MAPT 4137 DRUGGABLE GENOME 4,4'-DIMETHOXYDALBERGIONE 4,4'-DIMETHOXYDALBERGIONE 38779 26435 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 252166578 ABEXINOSTAT 38780 26436 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME arformoterol ARFORMOTEROL 38781 26437 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALD-401 38782 26438 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY HORMONES 11445246 38783 26439 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER APG-115 28498808 38784 26440 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GOSSYPOL GOSSYPOL 38785 26441 NDUFB5 4711 ENZYME inhibitor CHEMBL3545135 NV-128 38787 26442 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178103794 MELOXICAM 38788 26443 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Niraparib Tosylate 38792 26444 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL agonist 178103295 38793 26445 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME Elagolix ELAGOLIX 38796 26446 RAB9A 9367 ENZYME, DRUGGABLE GENOME Benzoic Acid 38797 26447 TAC1 6863 DRUGGABLE GENOME ETIDRONATE ETIDRONIC ACID 16133581 38798 26448 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME 681640 CHEMBL379975 38799 26449 AKR1C3 8644 ENZYME, DRUGGABLE GENOME inhibitor 381744943 38801 26450 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102415 38804 26451 POLB 5423 DNA REPAIR, DRUGGABLE GENOME MORIN MORIN 38805 26452 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME 2-(STYRYL)-BENZIMIDAZOLE CHEMBL473721 38806 26453 MAOB 4129 DRUGGABLE GENOME, ENZYME RASAGILINE RASAGILINE 38807 26454 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR ATRA TRETINOIN 8982293 38808 26455 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 178103533 DEXTROTHYROXINE 38809 26456 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME DOVITINIB DOVITINIB 38812 26457 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135650015 CHEMBL54004 38813 26458 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ADALIMUMAB ADALIMUMAB 38814 26459 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MEBEVERINE HYDROCHLORIDE MEBEVERINE HYDROCHLORIDE 38817 26460 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE FASUDIL FASUDIL 17018693 38818 26461 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 385612180 38819 26462 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NOREPINEPHRINE NOREPINEPHRINE 38820 26463 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 354702286 38821 26464 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PENTACHLOROPHENOL PENTACHLOROPHENOL 38823 26465 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor 178101475 38825 26466 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL3545160 SU-014813 38828 26467 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER rucaparib RUCAPARIB 38830 26468 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ETOXAZOLE ETOXAZOLE 38831 26469 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 178102326 38832 26470 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE TYRPHOSTIN AG-835 CHEMBL261557 38836 26471 USP1 7398 DNA REPAIR, PROTEASE, ENZYME STICTIC ACID STICTIC ACID 38839 26472 RRM2 6241 DRUGGABLE GENOME, ENZYME cladribine CLADRIBINE 24024897 38840 26473 CA2 760 DRUGGABLE GENOME, ENZYME GUAIACOL GUAIACOL 38841 26474 DHODH 1723 DRUGGABLE GENOME, ENZYME BAY2402234 38842 26475 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 23622981 38843 26476 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL2096631 CLORAZEPATE DIPOTASSIUM 38844 26477 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR CENISERTIB CENISERTIB 38845 26478 CRY1 1407 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR 252166810 38847 26479 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CISPLATIN CISPLATIN 27489350 38849 26480 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PROPYLPARABEN PROPYLPARABEN 38851 26481 PTGES3 10728 ENZYME DIETHYLSTILBESTROL DIETHYLSTILBESTROL 15229138 38852 26482 GMNN 51053 DRUGGABLE GENOME PARBENDAZOLE PARBENDAZOLE 38856 26483 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR Turofexorate isopropyl 38857 26484 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MELPHALAN MELPHALAN 38860 26485 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME AZD-6765 LANICEMINE 38862 26486 ACE2 59272 ENZYME, TRANSPORTER, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, CELL SURFACE, PROTEASE inhibitor 178103169 38863 26487 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SJ000082806 CHEMBL494668 38864 26488 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME NORSTICTIC ACID NORSTICTIC ACID 38866 26489 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 187051805 QUISINOSTAT 38867 26490 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ibritumomab IBRITUMOMAB TIUXETAN 38869 26491 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Her2-targeted autologous T-cell therapy 38870 26492 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR GENISTEIN GENISTEIN 12580099 38871 26493 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME SB-206553 CHEMBL297784 38872 26494 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-3201 CHEMBL581872 38874 26495 IL1B 3553 KINASE, DRUGGABLE GENOME CHEMBL1743026 GEVOKIZUMAB 38875 26496 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME TEMAZEPAM TEMAZEPAM 38877 26497 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Piperidinyl triazole derivative 6 38878 26498 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR 2,4-DINITROPHENOL 2,4-DINITROPHENOL 38879 26499 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE GEFITINIB GEFITINIB 38880 26500 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME PMID27998201-Compound-1 38882 26501 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL452 CLONAZEPAM 38883 26502 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHELIDONINE (+) CHELIDONINE (+) 38885 26503 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME WORTMANNIN WORTMANNIN 17135248 38887 26504 KDM4A 9682 DRUGGABLE GENOME, ENZYME MINAPRINE HYDROCHLORIDE MINAPRINE HYDROCHLORIDE 38888 26505 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody ABT-806 DEPATUXIZUMAB 38890 26506 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME 178103301 38893 26507 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER docetaxel DOCETAXEL 21151855 38894 26508 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 178101884 GSK-690693 38895 26509 TGFB3 7043 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR antibody FRESOLIMUMAB FRESOLIMUMAB 38896 26510 ALOX5 240 DRUGGABLE GENOME, ENZYME Diethylcarbamazine DIETHYLCARBAMAZINE 38899 26511 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 135650433 38900 26512 CDC42BPA 8476 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GSK-269962A GSK-269962A 38901 26513 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ALDRIN ALDRIN 38902 26514 RORA 6095 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE agonist 135651458 38903 26515 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME platinum PLATINUM 27462924 38904 26516 MTR 4548 ENZYME, DRUGGABLE GENOME ENZYME INHIBITOR 15148588 38905 26517 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR ANTIBIOTIC ANTIBIOTIC 9161031 38906 26518 RAB9A 9367 ENZYME, DRUGGABLE GENOME NSC-116702 CHEMBL1477383 38907 26519 TH 7054 ENZYME, DRUGGABLE GENOME Metyrosine METYROSINE 38909 26520 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR eltrombopag ELTROMBOPAG 38910 26521 SMARCA4 6597 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING TAZEMETOSTAT TAZEMETOSTAT 29650362 38911 26522 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LITHOCHOLIC ACID LITHOCHOLIC ACID 24818857 38917 26523 XDH 7498 DRUGGABLE GENOME, ENZYME ROXITHROMYCIN ROXITHROMYCIN 14730107 38918 26524 GPR183 1880 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178101169 38919 26525 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-44 38920 26526 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3545324 RG-7666 38921 26527 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TRICLOCARBAN TRICLOCARBAN 38924 26528 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BETA-TOXICAROL BETA-TOXICAROL 38925 26529 TXK 7294 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 354702234 38926 26530 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-71033 CHEMBL116548 38927 26531 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 187051782 ARFORMOTEROL 38929 26532 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme14BINDY 38930 26533 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE GW441756X GW441756X 38931 26534 CDH17 1015 TRANSPORTER, CELL SURFACE SQUALAMINE SQUALAMINE 11297269 38933 26535 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME BETA-LAPACHONE LAPACHONE 15753997 38934 26536 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE INIPARIB INIPARIB 38936 26537 HTT 3064 DRUGGABLE GENOME Sodium phenylbutyrate 38938 26538 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE Cobimetinib COBIMETINIB 38939 26539 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME DNDI1417467 CHEMBL1997335 38940 26540 BAZ2B 29994 NA MECLIZINE DIHCL MECLIZINE DIHCL 38941 26541 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ANCITABINE ANCITABINE 38942 26542 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME HYPERBARIC OXYGEN 16001273 38943 26543 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME VINPOCETINE VINPOCETINE 38945 26544 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 249565637 BMS-911543 38947 26545 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PENBUTOLOL PENBUTOLOL 38948 26546 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL451 CHLORDIAZEPOXIDE 38949 26547 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Piperidinyl pyrazole derivative 2 38950 26548 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CALCIMYCIN CALCIMYCIN 38951 26549 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CYPROTERONE CYPROTERONE 22931300 38953 26550 E2F1 1869 TRANSCRIPTION FACTOR HOECHST 33258 11151061 38954 26551 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 38955 26552 TUBB4B 10383 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 38957 26553 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 178102314 IMATINIB 38958 26554 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE midostaurin MIDOSTAURIN 38960 26555 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TETRADIFON TETRADIFON 38961 26556 HSPA4 3308 NA NIFEDIPINE NIFEDIPINE 7770620 38965 26557 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-3906 CHEMBL599102 38966 26558 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Monofluorine derivative 1 38967 26559 CBX1 10951 NA FLUPIRTINE FLUPIRTINE 38968 26560 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 178103305 PF-04457845 38969 26561 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE cisplatin CISPLATIN 25141953,22016816,31666714,27457817 38970 26562 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Trastuzumab biosimilar 38972 26563 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE GNF-PF-3023 CHEMBL535331 38973 26564 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL2110725 VINFLUNINE 38976 26565 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-37 38977 26566 ITPA 3704 ENZYME purine analogues 19129747 38978 26567 XRCC1 7515 CLINICALLY ACTIONABLE MUSTARD 8765433 38979 26568 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL3545133 JNJ-26483327 38980 26569 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR NCGC00381656-01 38981 26570 ALOX15B 247 DRUGGABLE GENOME, ENZYME DIPYRONE SODIUM DIPYRONE SODIUM 38982 26571 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE 6-TG THIOGUANINE 1988936 38983 26572 PSMC2 5701 PROTEASE, TRANSCRIPTION FACTOR CARFILZOMIB CARFILZOMIB 24524217 38984 26573 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-43 38985 26574 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1769 PROPOXYCAINE HYDROCHLORIDE 38986 26575 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL464 ETRETINATE 38989 26576 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUOXETINE FLUOXETINE 38990 26577 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-19 38991 26578 ATXN2 6311 NA NSC-106547 CHEMBL223575 38993 26579 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AZACITIDINE AZACITIDINE 38996 26580 PMP22 5376 DRUGGABLE GENOME, TRANSPORTER KETOPROFEN KETOPROFEN 38997 26581 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME MIDAZOLAM MIDAZOLAM 39000 26582 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 7,8,3'-TRIHYDROXYFLAVONE CHEMBL225513 39001 26583 GLS 2744 ENZYME PMID30273516-Compound-14 39002 26584 MAPT 4137 DRUGGABLE GENOME APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 39007 26585 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE atazanavir ATAZANAVIR 26287941 39008 26586 SMN2 6607 DRUGGABLE GENOME RETUSIN 7-METHYL ETHER RETUSIN 7-METHYL ETHER 39009 26587 ALOX5 240 DRUGGABLE GENOME, ENZYME BIM23A760 39010 26588 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID25726713-Compound-47 39011 26589 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor SB939 39012 26590 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PARAROSANILINE PARAROSANILINE 39013 26591 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE IODOCARB IODOCARB 39014 26592 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ARTHONIOIC ACID ARTHONIOIC ACID 39018 26593 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PROCHLORPERAZINE PROCHLORPERAZINE 22931300 39019 26594 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TCMDC-123764 CHEMBL533226 39022 26595 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL PRAZEPAM PRAZEPAM 39023 26596 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker 135652741 39024 26597 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3544966 GSK-1059615 39029 26598 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BENZQUINAMIDE BENZQUINAMIDE 39030 26599 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE GDC-0068 IPATASERTIB 39034 26600 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LINOLENIC ACID LINOLENIC ACID 39035 26601 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 39036 26602 EREG 2069 KINASE, GROWTH FACTOR, DRUGGABLE GENOME PANITUMUMAB PANITUMUMAB 26867820 39037 26603 BMP7 655 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR cyclophosphamide CYCLOPHOSPHAMIDE 26590194 39040 26604 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-67 39043 26605 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MANGOSTIN MANGOSTIN 39044 26606 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102574 39045 26607 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME ABBV-744 ABBV-744 39046 26608 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 374883879 39049 26609 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BOL-303259-X LATANOPROSTENE BUNOD 39052 26610 SLC1A2 6506 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE inhibitor 178101252 CHEMBL1628669 39053 26611 SFTPA1 653509 DRUGGABLE GENOME RETINYL PALMITATE 8023960 39055 26612 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME activator 178101017 39057 26613 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME XANTHINE AMINE CONGENER XANTHINE AMINE CONGENER 39059 26614 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE Epithalon 39060 26615 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL931 HALOTHANE 39062 26616 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102336 BOSUTINIB 39065 26617 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL564829 MILCICLIB 39066 26618 FAAH 2166 ENZYME, DRUGGABLE GENOME PMID29053063-Compound-11d 39067 26619 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 354702272 SELETALISIB 39068 26620 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME BEVACIZUMAB BEVACIZUMAB 39069 26621 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME PREDNISONE PREDNISONE 39070 26622 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME BROMAZEPAM BROMAZEPAM 39072 26623 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE olaratumab OLARATUMAB 39074 26624 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME SRT-1720 CHEMBL257991 18046409,23876989 39075 26625 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL2106615 BAZEDOXIFENE ACETATE 39078 26626 SMN1 6606 DRUGGABLE GENOME ANISINDIONE ANISINDIONE 39080 26627 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR O-DEMETHYLATED ADAPALENE O-DEMETHYLATED ADAPALENE 39082 26628 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SEMAXANIB SEMAXANIB 39083 26629 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME PMID27998201-Compound-9 39084 26630 PSMC5 5705 TRANSCRIPTION FACTOR BINDING, PROTEASE inhibitor BORTEZOMIB BORTEZOMIB 39085 26631 HEBP1 50865 DRUGGABLE GENOME Thiazole derivative 3 39091 26632 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 Methoxsalen METHOXSALEN 39093 26633 AQP1 358 ION CHANNEL, DRUGGABLE GENOME DIMETHYL SULFOXIDE 9374641 39095 26634 TCF7L2 6934 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR cyclosporine CYCLOSPORINE 23041303,21857094 39096 26635 PRMT1 3276 ENZYME, METHYL TRANSFERASE inhibitor 178103607 39097 26636 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651418 ALITRETINOIN 39098 26637 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME ezetimibe / rosuvastatin 39099 26638 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure1-Eryngiolide A 39100 26639 TUBB2A 7280 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 39102 26640 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DOCEBENONE DOCEBENONE 39103 26641 RACGAP1 29127 NA IMINOSTILBENE IMINOSTILBENE 39104 26642 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Ublituximab UBLITUXIMAB 39105 26643 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PYRAZINAMIDE PYRAZINAMIDE 22931300 39107 26644 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE INTRALIPID SOYBEAN OIL 10997602 39108 26645 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME EPOETIN ALFA 39110 26646 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL487 DROLOXIFENE 39112 26647 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-1702 CHEMBL600313 39113 26648 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DESOGESTREL DESOGESTREL 39114 26649 DPP7 29952 PROTEASE, ENZYME, DRUGGABLE GENOME US8470836, 2 39115 26650 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR OBETICHOLIC ACID OBETICHOLIC ACID 25247751,24387325,21459580 39117 26651 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DEXTROMEPROMAZINE DEXTROMEPROMAZINE 39120 26652 PBRM1 55193 CLINICALLY ACTIONABLE NIVOLUMAB NIVOLUMAB 29301960,31486842 39121 26653 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PD-98059 CHEMBL35482 39122 26654 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE LORATADINE LORATADINE 39123 26655 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE Anti-DR5 cells 39125 26656 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NATEGLINIDE NATEGLINIDE 22931300 39127 26657 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME cobimetinib COBIMETINIB 39130 26658 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 178102929 VILDAGLIPTIN 39131 26659 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BETA-LAPACHONE LAPACHONE 12689523 39135 26660 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Pyrazolo[1,5-a]-1,3,5-triazine derivative 1 39136 26661 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor PKI-587 GEDATOLISIB 39137 26662 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME PICEATANNOL PICEATANNOL 39138 26663 USP1 7398 DNA REPAIR, PROTEASE, ENZYME LINTITRIPT LINTITRIPT 39139 26664 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565696 39141 26665 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE RAMIPRIL RAMIPRIL 16166267 39142 26666 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Monoaryl-1,2-diamine derivative 4 39143 26667 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE PEGVISOMANT PEGVISOMANT 39146 26668 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE 7,4'-DIMETHOXYISOFLAVONE CHEMBL12658 39148 26669 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR CONICASTEROL B CONICASTEROL B 21428459 39149 26670 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DACARBAZINE DACARBAZINE 22931300 39153 26671 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME BROMAZEPAM BROMAZEPAM 39154 26672 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SGX523 19934279,26483207 39155 26673 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SB-202190 SB-202190 39156 26674 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE OXYCODONE OXYCODONE 39157 26675 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE PMID18163548C4 39158 26676 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HKI-272 NERATINIB 39159 26677 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 6-3'-DIMETHYLFLAVONE CHEMBL137498 39162 26678 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME FOSPROPOFOL FOSPROPOFOL 39164 26679 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NAN-190 NAN-190 39165 26680 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PALBOCICLIB PALBOCICLIB 39166 26681 CUL4A 8451 ENZYME, DNA REPAIR, CLINICALLY ACTIONABLE inhibitor CHEMBL468 THALIDOMIDE 39167 26682 LGMN 5641 ENZYME, DRUGGABLE GENOME, PROTEASE Legumain-cleavable doxorubicin prodrugs 39168 26683 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GABACULINE HYDROCHLORIDE GABACULINE HYDROCHLORIDE 39169 26684 HSPA8 3312 TUMOR SUPPRESSOR ELLAGIC ACID ELLAGIC ACID 39170 26685 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SANGUINARIUM CHLORIDE SANGUINARIUM CHLORIDE 39171 26686 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor PONATINIB PONATINIB 39172 26687 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE activator CHEMBL2108791 TENECTEPLASE 39173 26688 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-49 39174 26689 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CPI-006 39175 26690 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR GEDUNIN GEDUNIN 25756299,21129982 39177 26691 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 404859011 39178 26692 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor PD0332991 PALBOCICLIB 39179 26693 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PHENYLEPHRINE PHENYLEPHRINE 39180 26694 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LY2835219 ABEMACICLIB 39182 26695 POLI 11201 DNA REPAIR HAEMATOXYLIN HAEMATOXYLIN 39183 26696 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DIGOXIN DIGOXIN 22931300 39187 26697 RAPGEF3 10411 ENZYME ACRIFLAVINE CHLORIDE ACRIFLAVINE 39188 26698 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 363894149 PETESICATIB 39189 26699 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1071 OXAPROZIN 39190 26700 ENO2 2026 CELL SURFACE INSULIN INSULIN 7276941 39191 26701 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR INOSITOL INOSITOL 15560785 39193 26702 CDK12 51755 KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR, SERINE THREONINE KINASE inhibitor CHEMBL445813 AT-7519 39194 26703 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545421 DERAZANTINIB 39195 26704 KIF11 3832 DRUGGABLE GENOME ARRY-520 FILANESIB 39197 26705 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LEE011 RIBOCICLIB 39199 26706 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Drugs For Treatment Of Tuberculosis 23153709 39200 26707 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME US8609715, B-61 39201 26708 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE INFLIXIMAB INFLIXIMAB 39203 26709 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SAQUINAVIR SAQUINAVIR 39204 26710 SLC1A3 6507 TRANSPORTER, DRUGGABLE GENOME, CELL SURFACE inhibitor 178101329 39205 26711 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 387065612 39207 26712 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1200531 ALFENTANIL HYDROCHLORIDE 39209 26713 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TOZASERTIB TOZASERTIB 39210 26714 CDK14 5218 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME inhibitor CHEMBL445813 AT-7519 39211 26715 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE APALUTAMIDE APALUTAMIDE 23779130 39212 26716 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 404859109 39214 26717 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE Upamostat UPAMOSTAT 39215 26718 MPHOSPH8 54737 NA MYRICETIN MYRICETIN 39217 26719 HLA-E 3133 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE adalimumab ADALIMUMAB 39218 26720 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BUTYRATE 10444408,10720760 39219 26721 PTGS1 5742 ENZYME, DRUGGABLE GENOME ETHYL EICOSAPENTAENOIC ACID 39222 26722 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR GNTI 39225 26723 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME ALG-1001 RISUTEGANIB 39226 26724 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME PHENETHYLISOTHIOCYANATE PHENETHYLISOTHIOCYANATE 22607231 39227 26725 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL1230607 PHA-793887 39228 26726 STAG2 10735 CLINICALLY ACTIONABLE, DRUG RESISTANCE Dabrafenib DABRAFENIB 27500726 39229 26727 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Anastrozole ANASTROZOLE 39231 26728 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME CAPSAICIN CAPSAICIN 17603282 39232 26729 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE Refametinib REFAMETINIB 23434733 39235 26730 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-4945 CHEMBL585628 39239 26731 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 135650365 IBUPROFEN 39240 26732 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE FAZ053 39244 26733 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE tipiracil / trifluridine 39246 26734 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR RAD1901 RAD1901 39247 26735 CA1 759 DRUGGABLE GENOME, ENZYME Dichlorphenamide DICHLORPHENAMIDE 39248 26736 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME (R)-2,3-BIS(OCTYLOXY)PROPYL DIHYDROGEN PHOSPHATE CHEMBL202243 16263282 39249 26737 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774822-Compound-Figure10Compound4 39250 26738 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Pyrido[1,2-a]indole-1.-carboxylic acid analog 3 39251 26739 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor FK-228 ROMIDEPSIN 39252 26740 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR CRYPTOLEPINE HYDROCHLORIDE CRYPTOLEPINE HYDROCHLORIDE 23507189 39254 26741 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER IOXYNIL IOXYNIL 39255 26742 ATAD5 79915 NA ISOVELLERAL ISOVELLERAL 39256 26743 MUC16 94025 DRUGGABLE GENOME TOPOTECAN TOPOTECAN 17227902 39257 26744 PLK2 10769 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8598172, 1 39258 26745 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL TEMAZEPAM TEMAZEPAM 39259 26746 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649688 39260 26747 HSPA8 3312 TUMOR SUPPRESSOR NSC-119913 CHEMBL471004 39261 26748 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ERGOCORNINE ERGOCORNINE 39263 26749 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME PAZOPANIB PAZOPANIB 39264 26750 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE PEGVISOMANT PEGVISOMANT 39265 26751 RACGAP1 29127 NA NANAOMYCIN NANAOMYCIN 39266 26752 POLK 51426 DNA REPAIR, ENZYME LEVODOPA LEVODOPA 39267 26753 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GRINIMIBINE GRINIMIBINE 39270 26754 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor PAZOPANIB PAZOPANIB 39271 26755 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-36 39272 26756 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL918 PHENACEMIDE 39274 26757 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME INOSITOL INOSITOL 2498808 39275 26758 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650102 CIPROXIFAN 39276 26759 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PILSICAINIDE PILSICAINIDE 39277 26760 MAP3K2 10746 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME CI-1040 CI-1040 39279 26761 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Chloroacetyl ester derivative 1 39280 26762 TNFRSF4 7293 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE 178101769 39281 26763 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AER001,AEROVANT 39286 26764 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heteroaryl-carboxamide derivative 6 39287 26765 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ENOXOLONE ENOXOLONE 21888390 39288 26766 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL3544962 CT-1578 39290 26767 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ROTENONE ROTENONE 39291 26768 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR K-877 K-877 39292 26769 MYO9B 4650 NA TESTOSTERONE TESTOSTERONE 8409979 39293 26770 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651287 39294 26771 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME IL-6 1846631 39295 26772 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PROCHLORPERAZINE EDISYLATE PROCHLORPERAZINE EDISYLATE 39297 26773 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 1-O-ACETYLGEOPYXIN A CHEMBL1902074 39301 26774 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME sertraline SERTRALINE 39302 26775 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AG490 22159814 39303 26776 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AZD2461 27550455 39304 26777 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IPRONIAZID PHOSPHATE IPRONIAZID PHOSPHATE 39308 26778 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME ENTRECTINIB ENTRECTINIB 39309 26779 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545057 ACETYLDIGITOXIN 39310 26780 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Pyrimidinyl compound 5 39311 26781 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Kombiglyze XR/Komboglyze FDC 39312 26782 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Bevacizumab BEVACIZUMAB 26762204 39313 26783 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 384403668 39314 26784 MAOB 4129 DRUGGABLE GENOME, ENZYME CHF-3381 INDANTADOL 39315 26785 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor SAR302503 FEDRATINIB 39317 26786 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CADMIUM ACETATE CADMIUM ACETATE 39318 26787 JAG1 182 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, GROWTH FACTOR CORTISOL HYDROCORTISONE 11948681 39319 26788 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME SENNOSIDE B SENNOSIDE B 39320 26789 NEK4 6787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TAE-684 TAE-684 39321 26790 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL NITRAZEPAM NITRAZEPAM 39323 26791 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GNF-PF-4945 CHEMBL585628 39324 26792 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 310264691 39325 26793 PSMA4 5685 DRUGGABLE GENOME, PROTEASE inhibitor CARFILZOMIB CARFILZOMIB 39327 26794 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000121029 CHEMBL591631 39328 26795 MGLL 11343 DRUGGABLE GENOME, ENZYME OCTHILINONE OCTHILINONE 22056744 39329 26796 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUCINDOLOL BUCINDOLOL 39331 26797 MAPT 4137 DRUGGABLE GENOME MMV085203 CHEMBL586031 39332 26798 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-WO2009018344C78 39334 26799 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE XL999 39335 26800 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor CHEMBL574737 UCN-01 39336 26801 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HEXACHLOROPHENE HEXACHLOROPHENE 39337 26802 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TCMDC-123920 CHEMBL1606 39338 26803 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE IC261 IC261 20350806 39339 26804 PSIP1 11168 CLINICALLY ACTIONABLE US9132129, Cpd023 39340 26805 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE HUMAN CHORIONIC GONADOTROPIN 15590984 39342 26806 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 178102668 39344 26807 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-9 39348 26808 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME HORMONES 12660809 39350 26809 HLA-DQB1 3119 CLINICALLY ACTIONABLE flucloxacillin FLOXACILLIN 30664875 39351 26810 GAA 2548 DRUGGABLE GENOME, ENZYME SALACINOL SALACINOL 39352 26811 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER HYDRALAZINE HYDROCHLORIDE HYDRALAZINE HYDROCHLORIDE 39353 26812 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE CROFELEMER CROFELEMER 39356 26813 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651367 ZOTEPINE 39357 26814 CAST 831 PROTEASE INHIBITOR DHT ANDROSTANOLONE 12646165 39359 26815 PCBD1 5092 ENZYME H2O2 14530988 39360 26816 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME R3MAB 19381019 39362 26817 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME PHA-767491 CHEMBL225519 18469809 39363 26818 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME SOTRASTAURIN SOTRASTAURIN 39364 26819 ALOX15 246 ENZYME, DRUGGABLE GENOME 4,4'-DIMETHOXYDALBERGIONE 4,4'-DIMETHOXYDALBERGIONE 39365 26820 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LYCOPENE LYCOPENE 14640578 39366 26821 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL TRIAZOLAM TRIAZOLAM 39367 26822 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME SP-600125 SP-600125 39368 26823 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE acetaminophen ACETAMINOPHEN 21837673 39370 26824 MAPT 4137 DRUGGABLE GENOME DERRUBONE DERRUBONE 39371 26825 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE XL765 39372 26826 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE oxcarbazepine OXCARBAZEPINE 21449672,22630058,22188362,25155934,22256867,23697249,24567120,21799461 39373 26827 TH 7054 ENZYME, DRUGGABLE GENOME SAPONIN 9868557 39375 26828 CXCL8 3576 DRUGGABLE GENOME PMA 7510691 39376 26829 TDO2 6999 ENZYME, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 2 39377 26830 RACGAP1 29127 NA AMINODIMETHOXYQUINAZOLINYLPIPERAZINE AMINODIMETHOXYQUINAZOLINYLPIPERAZINE 39378 26831 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL INS-37217 DENUFOSOL TETRASODIUM 39379 26832 GMNN 51053 DRUGGABLE GENOME 4-(7-METHYLOCTYL)PHENOL CHEMBL503990 39380 26833 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PGF2ALPHA-IE 39381 26834 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-10 39382 26835 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CICHORIC ACID CICHORIC ACID 39384 26836 PTGS2 5743 DRUGGABLE GENOME, ENZYME NAPROXEN NAPROXEN 39385 26837 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER SAQUINAVIR MESYLATE 12384350 39386 26838 MAP3K13 9175 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 328083457 39387 26839 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR HEXAMETHYLENEBISACETAMIDE HEXAMETHYLENEBISACETAMIDE 7741753 39388 26840 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME PROGESTOGENS 11470238 39389 26841 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME MP0250 MP-0250 39390 26842 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE CYC-116 CYC-116 39392 26843 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME TCMDC-124307 CHEMBL546865 39393 26844 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE daunorubicin DAUNORUBICIN 25119182 39394 26845 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE DIFLOMOTECAN DIFLOMOTECAN 39396 26846 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TIOXOLONE TIOXOLONE 39397 26847 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OLEANOLIC_ACID OLEANOLIC_ACID 19716700 39400 26848 GZMA 3001 PROTEASE, DRUGGABLE GENOME, ENZYME CC CHEMOKINES 8598480 39401 26849 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AZD1480 AZD-1480 39402 26850 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME SJ000044511 CHEMBL592124 39404 26851 HDAC11 79885 DRUGGABLE GENOME, ENZYME PMID29671355-Compound-36 39405 26852 PC 5091 ENZYME, CLINICALLY ACTIONABLE CORTISOL HYDROCORTISONE 942746 39406 26853 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200802 TALBUTAL 39407 26854 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Aminooxazole carboxamide derivative 1 39408 26855 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR NICOTINE NICOTINE 11592233 39409 26856 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor CHEMBL3544955 BAY-1217389 39411 26857 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME TRANSPLATIN TRANSPLATIN 39412 26858 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417722 CHEMBL1503190 39413 26859 TNFRSF1B 7133 DRUGGABLE GENOME 178101766 39414 26860 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL FELODIPINE FELODIPINE 39415 26861 CTSE 1510 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166834 39416 26862 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE TRETINOIN TRETINOIN 39417 26863 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 39419 26864 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CIPROFLOXACIN CIPROFLOXACIN 22931300 39420 26865 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME HALOPERIDOL HALOPERIDOL 11080184 39421 26866 LIPG 9388 DRUGGABLE GENOME, ENZYME, LIPASE, CELL SURFACE, PHOSPHOLIPASE inhibitor 404859111 39422 26867 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TETRACYCLINE TETRACYCLINE 22931300 39423 26868 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 REMOXIPRIDE REMOXIPRIDE 22931300 39424 26869 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL MIDAZOLAM MIDAZOLAM 39426 26870 CALR 811 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GENTAMICIN GENTAMICIN 15351734 39427 26871 BAZ2B 29994 NA HINOKITIOL HINOKITIOL 39428 26872 COL3A1 1281 DRUGGABLE GENOME COLLAGENASE COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 39429 26873 CBX1 10951 NA DEPHOSTATIN DEPHOSTATIN 39431 26874 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 4-CHLOROBENZALDEHYDE CHEMBL1474 39432 26875 CFI 3426 ENZYME, DRUGGABLE GENOME, PROTEASE TGFBETA1 17320177 39433 26876 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DEPHOSTATIN DEPHOSTATIN 39435 26877 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Olaparib OLAPARIB 39436 26878 KMO 8564 DRUGGABLE GENOME, ENZYME Cyclopropane 1-carboxylic acid derivative 4 39439 26879 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME SJ000189154 CHEMBL604664 39440 26880 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME HEMATOXYLIN HEMATOXYLIN 39441 26881 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Carboplatin CARBOPLATIN 25637314,16043828,26307133,21216929,27998224 39444 26882 TSPO 706 DRUGGABLE GENOME Quinoline carboxamide derivative 8 39445 26883 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200382 BEPRIDIL HYDROCHLORIDE 39446 26884 NFKBIA 4792 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME gefitinib GEFITINIB 31664190 39447 26885 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor CHEMBL1094636 NIRAPARIB 39448 26886 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME VITAMIN A 6517947 39449 26887 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-234945 CHEMBL260311 39452 26888 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DOCUSATE DOCUSATE 39455 26889 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-J3 39457 26890 KDM5C 8242 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 249565909 39459 26891 CBX1 10951 NA OXOLINIC ACID OXOLINIC ACID 39462 26892 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PROGESTERONE PROGESTERONE 10195429 39464 26893 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE ENTRECTINIB ENTRECTINIB 39465 26894 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ZINC 03369470 CHEMBL599013 39466 26895 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 178100448 39467 26896 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR OP-R003 19934301 39468 26897 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TERAZOSIN TERAZOSIN 39470 26898 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor E-3810 RABEPRAZOLE SODIUM 39472 26899 EIF4E 1977 DRUGGABLE GENOME inhibitor ISIS-EIF4ERX 39473 26900 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MEDETOMIDINE MEDETOMIDINE 39474 26901 GADD45A 1647 DNA REPAIR, TUMOR SUPPRESSOR, KINASE CISPLATIN CISPLATIN 9013707,10779360 39475 26902 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME THIOURACIL THIOURACIL 10967532 39476 26903 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-56 39477 26904 PDE4B 5142 DRUGGABLE GENOME, ENZYME AMRINONE INAMRINONE 39478 26905 ALB 213 TRANSPORTER, DRUGGABLE GENOME (-)-EPICATECHIN (-)-EPICATECHIN 20598557 39480 26906 MAPT 4137 DRUGGABLE GENOME N-(4-NITROPHENYL)ANTHRANILIC ACID CHEMBL1574420 39481 26907 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-acylpiperidine ether derivative 1 39482 26908 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR 12-O-TETRADECANOYLPHORBOL-13-ACETATE 7982951 39483 26909 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DNDI1417181 CHEMBL1537417 39485 26910 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ACRIFLAVINE CHLORIDE ACRIFLAVINE 39486 26911 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 39487 26912 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-38 39488 26913 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MACROCARPAL A MACROCARPAL A 22934600 39489 26914 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Brivanib BRIVANIB 22238366 39491 26915 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE SB-220025 SB-220025 39492 26916 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1644 CHEMBL600734 39493 26917 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME GNF-PF-67 CHEMBL578512 39495 26918 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 celecoxib CELECOXIB 22336956 39497 26919 KAT5 10524 TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, ENZYME 6-DECYLSALICYLIC ACID CHEMBL416038 22100137 39499 26920 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201543 INSULIN ZINC SUSP SEMISYNTHETIC PURIFIED HUMAN 39500 26921 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 23622981 39506 26922 GMNN 51053 DRUGGABLE GENOME CAMBENDAZOLE CAMBENDAZOLE 39507 26923 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE ALSTERPAULLONE ALSTERPAULLONE 39508 26924 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ZYT-1 39509 26925 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-20 39510 26926 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER GENTIAN VIOLET GENTIAN VIOLET 39511 26927 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103455 TOPIRAMATE 39512 26928 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER SOM3355 39513 26929 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER unspecified ERBB3 antibody 27196767 39516 26930 KDM4A 9682 DRUGGABLE GENOME, ENZYME N-DEACETYLCOLCHICEINE CHEMBL517186 39517 26931 KIF11 3832 DRUGGABLE GENOME inhibitor 223366041 AZD-4877 39519 26932 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME VS-5584 VS-5584 39520 26933 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IBUPROFEN IBUPROFEN 22931300 39522 26934 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Androgen restored contraceptive 39524 26935 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 39525 26936 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR CHIDAMIDE CHIDAMIDE 39526 26937 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CY-208243 CHEMBL313737 39527 26938 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651331 XANOMELINE 39528 26939 GAK 2580 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 223366123 BARICITINIB 39529 26940 ABCC5 10057 DRUGGABLE GENOME, ABC TRANSPORTER, TRANSPORTER zidovudine ZIDOVUDINE 22960662 39530 26941 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Taxol PACLITAXEL 39531 26942 POLK 51426 DNA REPAIR, ENZYME QUERCETIN QUERCETIN 39532 26943 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE AMINOGLYCOSIDES 10900094 39533 26944 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650706 NECA 39534 26945 COL1A2 1278 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 39536 26946 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 39539 26947 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ranolazine RANOLAZINE 9187528 39540 26948 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme9EHT3356 39542 26949 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Pertuzumab PERTUZUMAB 23940356 39543 26950 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE Sulfamylon SULFAMYLON 39544 26951 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME celecoxib CELECOXIB 22336956 39548 26952 GMNN 51053 DRUGGABLE GENOME TOZASERTIB TOZASERTIB 39550 26953 MAOA 4128 DRUGGABLE GENOME, ENZYME 8-[3-(TRIFLUOROMETHYL)PHENOXYMETHYL]CAFFEINE CHEMBL2088303 22705191 39552 26954 KLB 152831 ENZYME ethanol ALCOHOL 39553 26955 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME LTB 019 39558 26956 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME PMID27998201-Compound-11 39560 26957 NFKBIA 4792 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME (+)-TUBERIFERIN CHEMBL1940084 22153345 39561 26958 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GSK-269962A GSK-269962A 39562 26959 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR EPROTIROME EPROTIROME 39563 26960 CES1 1066 DRUGGABLE GENOME, ENZYME trandolapril TRANDOLAPRIL 19185566 39565 26961 ABCC5 10057 DRUGGABLE GENOME, ABC TRANSPORTER, TRANSPORTER inhibitor 252827486 39567 26962 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE CILENGITIDE CILENGITIDE 24095096 39568 26963 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102587 39569 26964 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100419 39570 26965 SDC1 6382 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME BT-062 INDATUXIMAB RAVTANSINE 39571 26966 IL17RA 23765 DRUGGABLE GENOME CNTO-6785 39572 26967 NTS 4922 DRUGGABLE GENOME NIFEDIPINE NIFEDIPINE 8770786 39573 26968 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PROPYLTHIOURACIL PROPYLTHIOURACIL 22931300 39575 26969 HSF1 3297 TRANSCRIPTION FACTOR, DNA REPAIR BIMOCLOMOL BIMOCLOMOL 39576 26970 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FLUVOXAMINE FLUVOXAMINE 22931300 39577 26971 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GW7647 GW7647 39578 26972 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME MAPK INHIBITORS 14511403 39579 26973 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME FASUDIL FASUDIL 39580 26974 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR SNX-5422 CHEMBL553939 39581 26975 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHRYSIN CHRYSIN 39583 26976 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Emedastine EMEDASTINE 39584 26977 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1256 ISOFLURANE 39585 26978 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL723 CARVEDILOL 39587 26979 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR ZEARALANONE ZEARALANONE 39588 26980 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 178103108 DABRAFENIB 39589 26981 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1237132 CLEVIDIPINE 39591 26982 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE EMD-1214063 TEPOTINIB 39592 26983 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TANGERETIN TANGERETIN 39594 26984 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-38b 39596 26985 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL2068724 ACAMPROSATE CALCIUM 39597 26986 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL378544 VINBLASTINE SULFATE 39598 26987 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL2110725 VINFLUNINE 39599 26988 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE BMS-777607 BMS-777607 22286523,20515943,28396313 39602 26989 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102260 39605 26990 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651412 39606 26991 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE haloperidol HALOPERIDOL 27023437 39608 26992 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649942 39609 26993 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME inhibitor DABRAFENIB MESYLATE 39616 26994 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NPC-01 39618 26995 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650564 39619 26996 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME DEOXYVASICINONE DEOXYVASICINONE 39622 26997 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CARBOPLATIN CARBOPLATIN 26006067 39623 26998 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1200405 BITOLTEROL MESYLATE 39624 26999 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-43 39626 27000 NQO2 4835 DRUGGABLE GENOME, ENZYME NSC-645809 C-1311 39628 27001 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME ILORASERTIB ILORASERTIB 39629 27002 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME CICLOSPORIN CYCLOSPORINE 16805961 39630 27003 TJP1 7082 KINASE, TRANSCRIPTION FACTOR ETHANOL ALCOHOL 9952110 39632 27004 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Tricyclic heterocycle derivative 6 39634 27005 RCE1 9986 ENZYME, PROTEASE, DRUGGABLE GENOME HTS-9915 CHEMBL512935 39637 27006 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166766 39638 27007 POLK 51426 DNA REPAIR, ENZYME IRIGENOL IRIGENOL 39639 27008 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR allosteric modulator 178102303 CI-1040 39640 27009 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417025 CHEMBL1320453 39641 27010 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MMV396678 CHEMBL1459149 39642 27011 SFTPA1 653509 DRUGGABLE GENOME 9-CIS-RETINOIC ACID 8944731 39643 27012 PSMA1 5682 PROTEASE, DRUGGABLE GENOME CARFILZOMIB CARFILZOMIB 24524217 39645 27013 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 252166504 39647 27014 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR amlodipine AMLODIPINE 39651 27015 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE MU DELTA 39652 27016 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CYC065 CYC-065 39653 27017 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME METERGOLINE METERGOLINE 39654 27018 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 KETANSERIN KETANSERIN 39656 27019 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Thioridazine THIORIDAZINE 39657 27020 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL371405 MARIZOMIB 39658 27021 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME CAR-T cells targeting Muc1 39659 27022 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AFIMOXIFENE AFIMOXIFENE 39660 27023 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 39662 27024 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 39663 27025 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR URSOLIC ACID URSOLIC ACID 21855333 39666 27026 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor BMS-599626 AC-480 39667 27027 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL3833329 ERENUMAB 39668 27028 RIPK2 8767 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 385612179 39669 27029 MAOB 4129 DRUGGABLE GENOME, ENZYME V3381 INDANTADOL 39670 27030 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ETOPOSIDE ETOPOSIDE 22931300 39672 27031 DNER 92737 NA Isoxazole-based bicyclic compound 8 39674 27032 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL217092 SARACATINIB 39679 27033 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HARMALINE HARMALINE 39680 27034 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE Pyrrolo[2,3-d]pyrimidine derivative 28 39681 27035 IDO2 169355 ENZYME 2,3-diamino-benzo[b]thiophene derivative 8 39682 27036 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME OSI-632 OSI-632 39683 27037 PFKFB3 5209 ENZYME, KINASE inhibitor 336446948 39684 27038 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650972 39685 27039 ATAD5 79915 NA RESVERATROL RESVERATROL 39686 27040 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME HYDRALAZINE HYDRALAZINE 39687 27041 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650559 LY-518674 39688 27042 ADAMTS4 9507 ENZYME, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE CHONDROITIN SULFATE 14701864 39690 27043 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR BINIMETINIB BINIMETINIB 31227518 39691 27044 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178101149 39692 27045 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME lumiracoxib LUMIRACOXIB 20639878 39693 27046 KDM4A 9682 DRUGGABLE GENOME, ENZYME TOREMIFENE CITRATE TOREMIFENE CITRATE 39694 27047 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ETOPOSIDE ETOPOSIDE 22931300 39696 27048 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Triazolo[4,3-b]pyridazine derivative 2 39698 27049 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 39699 27050 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR SUVANINE'S SODIUM SALT SUVANINE'S SODIUM SALT 23656455 39701 27051 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR GNF-PF-3148 CHEMBL81782 39702 27052 PAK3 5063 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor HESPERADIN HESPERADIN 19035792 39703 27053 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-92 39705 27054 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME irinotecan IRINOTECAN 20125120,25955730 39708 27055 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651539 DINOPROSTONE 39710 27056 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PHENOLPHTHALEIN PHENOLPHTHALEIN 39713 27057 FZD5 7855 G PROTEIN COUPLED RECEPTOR, KINASE, CELL SURFACE antibody 381118907 VANTICTUMAB 39715 27058 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AMSACRINE AMSACRINE 39716 27059 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AMINOCARB AMINOCARB 39717 27060 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 187051804 RESMINOSTAT 39718 27061 GLS 2744 ENZYME SULFURETIN SULFURETIN 39721 27062 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200371 FROVATRIPTAN SUCCINATE 39722 27063 TRPM7 54822 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ION CHANNEL, ENZYME, TRANSPORTER activator 135650688 NALTRIBEN 39723 27064 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2,4,5,10-TETRAHYDROPYRAZOLO[3,4-A]CARBAZOLE CHEMBL512649 39724 27065 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 336446938 39725 27066 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102231 REGADENOSON 39727 27067 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1133 OXYBUTYNIN CHLORIDE 39728 27068 BAZ2B 29994 NA 3,8'-BIAPIGENIN CHEMBL515252 39729 27069 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 39734 27070 TSPO 706 DRUGGABLE GENOME Benzimidazolone acetamide derivative 2 39735 27071 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 24524217,23547757 39736 27072 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor BELINOSTAT BELINOSTAT 39737 27073 DDHD1 80821 PHOSPHOLIPASE warfarin WARFARIN 27488176 39738 27074 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE LABETALOL LABETALOL 39739 27075 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL3137308 PEFICITINIB 39741 27076 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME VANITIOLIDE VANITIOLIDE 39742 27077 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME NSC-348401 CHEMBL515505 39743 27078 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Abemaciclib ABEMACICLIB 39744 27079 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR TEW-7197 VACTOSERTIB 39745 27080 ATAD5 79915 NA TCMDC-125465 CHEMBL536151 39748 27081 SLC47A1 55244 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER 178101231 39750 27082 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE Farglitazar FARGLITAZAR 18004211 39752 27083 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR VITAMIN K3H2 VITAMIN K3H2 39753 27084 ALDH1A1 216 DRUGGABLE GENOME, ENZYME N-(4-(CYANO(PHENYL)METHYL)PHENYL)ACETAMIDE CHEMBL1580175 39757 27085 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SJ000294102 CHEMBL607309 39758 27086 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR MITOXANTRONE MITOXANTRONE 39760 27087 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME inhibitor 348353616 VARESPLADIB 39761 27088 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME Oxotetrahydro-2-H-furo[3.2-b]pyrrol-4(5-H)-yl derivative 1 39762 27089 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHYL PARATHIONE METHYL PARATHIONE 39763 27090 PDE4A 5141 DRUGGABLE GENOME, ENZYME THEOPHYLLINE THEOPHYLLINE 39765 27091 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SPIRONOLACTONE SPIRONOLACTONE 39769 27092 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Pyrrolo-benzo-diazine derivative 1 39770 27093 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 178101871 FASUDIL 39771 27094 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178101750 SEMAXANIB 39772 27095 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE CENISERTIB CENISERTIB 39773 27096 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2016054807Example82 39774 27097 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125602 CHEMBL580183 39775 27098 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE AST-487 AST-487 39776 27099 RIPOR2 9750 NA rifampin RIFAMPIN 30720667 39777 27100 BRCA2 675 CLINICALLY ACTIONABLE PLATINUM COMPOUND 24240112,25072261 39778 27101 MGAT2 4247 ENZYME Pyrimidine-4(3H)-one derivative 1 39779 27102 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME (RS)-ROSCOVITINE (RS)-ROSCOVITINE 39780 27103 HSPA4 3308 NA ANTINEOPLASTIC 12530536 39781 27104 CDA 978 ENZYME, DRUGGABLE GENOME Tetrahydrouridine TETRAHYDROURIDINE 39782 27105 CD9 928 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE EOTAXIN 10704064 39784 27106 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1922094 APITOLISIB 39785 27107 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME EP-42675 39786 27108 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GLAFENINE GLAFENINE 22931300 39787 27109 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Abemaciclib ABEMACICLIB 39788 27110 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HARMALOL HYDROCHLORIDE HARMALOL HYDROCHLORIDE 39789 27111 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR ACLARUBICIN ACLARUBICIN 7689127 39790 27112 IL10RB 3588 DRUGGABLE GENOME agonist CHEMBL2108723 PEGINTERFERON LAMBDA-1A 39791 27113 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-2950 CHEMBL602807 39794 27114 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BROMOCRIPTINE MESYLATE BROMOCRIPTINE MESYLATE 39795 27115 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE CID 4101591 CHEMBL428789 39796 27116 GSTO1 9446 ENZYME, DRUGGABLE GENOME inhibitor 405067312 39798 27117 PSMC2 5701 PROTEASE, TRANSCRIPTION FACTOR inhibitor CHEMBL2103884 OPROZOMIB 39799 27118 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL TEMAZEPAM TEMAZEPAM 39800 27119 MAOB 4129 DRUGGABLE GENOME, ENZYME L-DOPA LEVODOPA 7867755,6420516 39801 27120 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME carbamazepine CARBAMAZEPINE 24399721,23830818 39803 27121 ATAD5 79915 NA DNDI1417457 CHEMBL1530911 39804 27122 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME FASUDIL FASUDIL 39805 27123 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALLISAN ALLISAN 39807 27124 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE CILENGITIDE CILENGITIDE 39808 27125 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE RIBOPRINE RIBOPRINE 25184810 39809 27126 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor AFATINIB AFATINIB 39810 27127 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXENDOLONE OXENDOLONE 39811 27128 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL52885 ENMD-981693 39812 27129 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1201063 PROPAFENONE HYDROCHLORIDE 39814 27130 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KETOCONAZOLE KETOCONAZOLE 2546501 39815 27131 SP3 6670 TRANSCRIPTION FACTOR DOXORUBICIN DOXORUBICIN 17511886 39816 27132 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 rifampin RIFAMPIN 20941486 39817 27133 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CHLORHEXIDINE HYDROCHLORIDE CHLORHEXIDINE HYDROCHLORIDE 39818 27134 BAZ2B 29994 NA GW7647 GW7647 39819 27135 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4-TERT-BUTYLCATECHOL CHEMBL220845 39821 27136 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE NAKIJIQUINONES G NAKIJIQUINONES G 18676149 39822 27137 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE MORPHINE MORPHINE 17616524,18193048,18380425 39823 27138 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DNDI1417388 CHEMBL1528359 39824 27139 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR trastuzumab TRASTUZUMAB 39826 27140 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL ETAZOLATE ETAZOLATE 39827 27141 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE agonist 135651597 39828 27142 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 39829 27143 BRCA2 675 CLINICALLY ACTIONABLE E7449 2X-121 26513298 39830 27144 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE BREFELDIN A BREFELDIN A 39831 27145 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE XL418 XL-418 19644473 39832 27146 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL591118 CARMEGLIPTIN 39833 27147 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650592 39835 27148 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CALCIMYCIN CALCIMYCIN 39837 27149 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Refametinib REFAMETINIB 23434733 39838 27150 MT1H 4496 NA H2O2 8385930 39839 27151 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX PINAFIDE PINAFIDE 39840 27152 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE PF-562271 PF-00562271 39841 27153 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME KD-025 CHEMBL2005186 39843 27154 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BETAXOLOL HYDROCHLORIDE BETAXOLOL HYDROCHLORIDE 39847 27155 ATXN2 6311 NA TRIFLUOPERAZINE HYDROCHLORIDE TRIFLUOPERAZINE HYDROCHLORIDE 39849 27156 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE TIPIFARNIB TIPIFARNIB 39850 27157 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 135650829 PIOGLITAZONE 39851 27158 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL781 MAZINDOL 39852 27159 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER SIROLIMUS SIROLIMUS 14569063 39855 27160 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME DNDI1416969 CHEMBL1453126 39856 27161 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650414 IRBESARTAN 39858 27162 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 328083468 39859 27163 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL254760 MGCD-265 39860 27164 YWHAG 7532 DRUGGABLE GENOME, KINASE DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 39862 27165 CERK 64781 KINASE, LIPID KINASE, ENZYME inhibitor 178103280 39863 27166 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME CHLORPROMAZINE CHLORPROMAZINE 39865 27167 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor GSK2126458 OMIPALISIB 39868 27168 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 39869 27169 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE N-ACETYLASPARTIC ACID N-ACETYLASPARTIC ACID 39872 27170 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PF-4691502 PF-04691502 39873 27171 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL70418 CLOBAZAM 39874 27172 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178103494 IBRUTINIB 39875 27173 GSTM1 2944 DRUGGABLE GENOME, ENZYME CURCUMIN CURCUMIN 15044619 39876 27174 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor CHEMBL3544936 XL-844 39879 27175 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650362 PICLIDENOSON 39881 27176 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PSI 25759020 39883 27177 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 39884 27178 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME U-0126 U-0126 39886 27179 ACKR3 57007 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135649932 PLERIXAFOR 39888 27180 RGS4 5999 DRUGGABLE GENOME DOCOSAPENTAENOIC ACID DOCOSAPENTAENOIC ACID 39890 27181 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Torkinib 27197158 39891 27182 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 135652717 STAUROSPORINE 39892 27183 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor AZD4547 39893 27184 HLA-DRA 3122 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE clavulanate CLAVULANIC ACID 30664875 39895 27185 TRPM6 140803 ION CHANNEL, DRUGGABLE GENOME, ENZYME, TRANSPORTER, KINASE, SERINE THREONINE KINASE blocker,activator 135652741 39898 27186 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BI-69A11 20531415,26603897 39899 27187 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor SF1126 39900 27188 NOS1 4842 DRUGGABLE GENOME, ENZYME DIURETIC 16496394,16712979 39901 27189 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM BROMIDE 39902 27190 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 363894237 39903 27191 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME KALOPANAX-SAPONIN F CHEMBL1833984 21889336 39904 27192 PRMT5 10419 ENZYME, METHYL TRANSFERASE inhibitor 252166606 39905 27193 ADD1 118 KINASE hydrochlorothiazide HYDROCHLOROTHIAZIDE 19057513,14553962,18591455,11882573,9149697,12623934,10523341 39906 27194 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 4101591 CHEMBL428789 39907 27195 ACVR2B 93 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ACE-031 RAMATERCEPT 39910 27196 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME stavudine STAVUDINE 39912 27197 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NIMESULIDE NIMESULIDE 39913 27198 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME dimethyl fumarate 26967570 39915 27199 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor BKM120 BUPARLISIB 39917 27200 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SPARFLOXACIN SPARFLOXACIN 39920 27201 NDUFB8 4714 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 39922 27202 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor AP26113 CHEMBL3397300 39923 27203 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Risedronate RISEDRONIC ACID 39924 27204 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor GSK2636771 GSK-2636771 39925 27205 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CAULIBUGULONE B CAULIBUGULONE B 39928 27206 PRRC2A 7916 NA carboplatin CARBOPLATIN 31616045 39929 27207 NEK4 6787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SNS-314 SNS-314 39931 27208 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649861 39932 27209 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID25656651-Compound-28a 39934 27210 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Golvatinib GOLVATINIB 19832844 39935 27211 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CI-1040 CI-1040 19018267,19372556 39936 27212 RAMP1 10267 DRUGGABLE GENOME, CELL SURFACE PRAMLINTIDE PRAMLINTIDE 39938 27213 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ONARTUZUMAB ONARTUZUMAB 22389872 39939 27214 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME BLEOMYCIN BLEOMYCIN 15149862 39940 27215 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Ulipristal ULIPRISTAL 39941 27216 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Piperidinyl triazole derivative 5 39944 27217 KDM4A 9682 DRUGGABLE GENOME, ENZYME 2-MERCAPTONICOTINIC ACID 2-MERCAPTONICOTINIC ACID 39945 27218 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-61 39946 27219 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650378 ILOPROST 39947 27220 HBB 3043 DRUGGABLE GENOME, ENZYME luspatercept-aamt 39950 27221 ATXN2 6311 NA NSC-402083 CHEMBL1546228 39951 27222 CA2 760 DRUGGABLE GENOME, ENZYME STX-140 39953 27223 IL11 3589 DRUGGABLE GENOME, KINASE, GROWTH FACTOR 5-FU FLUOROURACIL 7691257 39954 27224 MOB3B 79817 KINASE Tumor necrosis factor alpha (TNF-alpha) inhibitors 39960 27225 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME pravastatin PRAVASTATIN 39963 27226 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL378544 VINBLASTINE SULFATE 39964 27227 MAPT 4137 DRUGGABLE GENOME THIOLUTIN THIOLUTIN 39965 27228 MBP 4155 CELL SURFACE BHT-3009 39967 27229 KDM6B 23135 ENZYME inhibitor 249565910 39968 27230 ATAD5 79915 NA 5-METHOXYFLAVONE CHEMBL16685 39971 27231 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME inotuzumab ozogamicin 39972 27232 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MEDROXYPROGESTERONE ACETATE MEDROXYPROGESTERONE ACETATE 39973 27233 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE Cobimetinib COBIMETINIB 39976 27234 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HYDROCORTISONE BUTYRATE HYDROCORTISONE BUTYRATE 39977 27235 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (+)-TETRAHYDROBERBERINE CHEMBL476501 39978 27236 TRPC4 7223 ION CHANNEL, KINASE, DRUGGABLE GENOME, CELL SURFACE blocker 135649695 39979 27237 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR celecoxib CELECOXIB 22336956 39980 27238 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX VINCRISTINE VINCRISTINE 39981 27239 BAZ2B 29994 NA N-(2-PYRIDYLMETHYL)PHENYLAMINE CHEMBL402456 39982 27240 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Solifenacin SOLIFENACIN 39984 27241 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE IMATINIB IMATINIB 39986 27242 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ATRA TRETINOIN 14587026,16403261 39987 27243 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW833373X GW833373X 39990 27244 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME CIPROFLOXACIN CIPROFLOXACIN 10741713,12632069 39991 27245 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000089001 CHEMBL591618 39993 27246 NPR3 4883 DRUGGABLE GENOME CARDIODILATIN 39994 27247 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MORICIZINE HYDROCHLORIDE MORICIZINE HYDROCHLORIDE 39996 27248 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID29757691-Compound-4 39997 27249 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE sunitinib SUNITINIB 19248971,26935927,20124951 39998 27250 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR FESOTERODINE FESOTERODINE 40001 27251 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 249565840 40005 27252 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MALATHION MALATHION 40007 27253 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME GNF-PF-1919 CHEMBL576409 40008 27254 ATAD5 79915 NA TCMDC-124422 CHEMBL527620 40009 27255 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3545284 CERDULATINIB 40010 27256 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR GEFITINIB GEFITINIB 17205515 40012 27257 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ethambutol ETHAMBUTOL 22151084 40014 27258 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE IFN 15548813 40015 27259 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 223365957 THIOTEPA 40018 27260 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Fulvestrant FULVESTRANT 27174596 40019 27261 CBX1 10951 NA SENNOSIDE B SENNOSIDE B 40020 27262 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 8 40021 27263 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 354702293 40022 27264 BAZ2B 29994 NA NSC-402083 CHEMBL1546228 40024 27265 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE DHT ANDROSTANOLONE 7704433 40025 27266 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR SYNTHETIC CONJUGATED ESTROGENS 40026 27267 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Cutamesine 40029 27268 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135650208 DOXEPIN 40030 27269 BAZ2B 29994 NA TCMDC-125567 CHEMBL530049 40035 27270 PPP1R13L 10848 TRANSCRIPTION FACTOR BINDING gemcitabine GEMCITABINE 40036 27271 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Aryl carboxamide derivative 2 40039 27272 SPG7 6687 PROTEASE, ENZYME anthracyclines and related substances 23441093,21900104 40041 27273 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1201576 RITUXIMAB 40042 27274 ANO1 55107 ION CHANNEL blocker 135650716 40043 27275 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME TOZASERTIB TOZASERTIB 40044 27276 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME TETRADECYLTHIOACETIC ACID TETRADECYLTHIOACETIC ACID 40045 27277 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SILIBININ SILIBININ 40046 27278 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PF3644022 26140595 40047 27279 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL2180604 TAK-593 40049 27280 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor BEZ235 DACTOLISIB 40050 27281 TUBB4B 10383 DRUGGABLE GENOME CHEMBL2103826 DAVUNETIDE 40051 27282 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR RIGOSERTIB RIGOSERTIB 40053 27283 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL443684 NAVITOCLAX 40054 27284 GMNN 51053 DRUGGABLE GENOME GNF-PF-1241 CHEMBL528724 40055 27285 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Linsitinib LINSITINIB 26561558 40056 27286 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR CLOFARABINE CLOFARABINE 40057 27287 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE IMMUNOSUPPRESSIVE 8972557 40058 27288 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 404859006 VOXELOTOR 40060 27289 MBP 4155 CELL SURFACE CSA CYCLOSPORINE 9184637 40062 27290 PTGS1 5742 ENZYME, DRUGGABLE GENOME Suprofen SUPROFEN 40063 27291 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CLARITHROMYCIN CLARITHROMYCIN 16221754 40064 27292 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 252166660 IXAZOMIB 40067 27293 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-61 40068 27294 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL932 DIPYRIDAMOLE 40069 27295 E2F1 1869 TRANSCRIPTION FACTOR NAC ACETYLCYSTEINE 12754095 40070 27296 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor MK2206 MK-2206 40071 27297 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER mefloquine MEFLOQUINE 40072 27298 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 187051774 ALVIMOPAN 40074 27299 SMAD2 4087 KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX BLEOMYCIN BLEOMYCIN 17274978 40075 27300 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PYRITHIONE ZINC PYRITHIONE ZINC 40076 27301 ATXN2 6311 NA HELENALIN HELENALIN 40077 27302 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE ONO-4232 40078 27303 TMEM97 27346 NA Benzamide derivative 8 40079 27304 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 178101642 40080 27305 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR AMIKACIN AMIKACIN 7540696,8158029 40081 27306 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PX-866 SONOLISIB 40085 27307 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME CELECOXIB CELECOXIB 15539607 40087 27308 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME SOBUZOXANE SOBUZOXANE 40090 27309 MAP2K3 5606 KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE inhibitor 178102628 40091 27310 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3544966 GSK-1059615 40092 27311 HDAC11 79885 DRUGGABLE GENOME, ENZYME TRICHOSTATIN TRICHOSTATIN 21055848,16921367,19966789,19385600 40093 27312 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AMG102 40095 27313 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DICLOFENAC DICLOFENAC 22931300 40096 27314 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE 3-amino-5-benzyl-substituted indazole derivative 1 40097 27315 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LY-25582 CHEMBL300662 40099 27316 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 384403638 40100 27317 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IMETIT IMETIT 40101 27318 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW680975X GW680975X 40102 27319 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651280 TRIPITRAMINE 40103 27320 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 315661180 ZOTIRACICLIB 40106 27321 POLI 11201 DNA REPAIR N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 40107 27322 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor AUY922 40110 27323 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYL 3-(2,5-DIHYDROXYPHENYL)ACRYLATE CHEMBL17329 40111 27324 AKR1B1 231 DRUGGABLE GENOME, ENZYME Fidarestat FIDARESTAT 40113 27325 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650423 40115 27326 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR BECLOMETHASONE BECLOMETHASONE 40116 27327 C3 718 PROTEASE INHIBITOR, DRUGGABLE GENOME, CELL SURFACE POT-4 19025129 40117 27328 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME artemether ARTEMETHER 40118 27329 UGT2B7 7364 DRUGGABLE GENOME oxazepam OXAZEPAM 40120 27330 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL723 CARVEDILOL 40121 27331 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME DIPYRIDAMOLE DIPYRIDAMOLE 40122 27332 CHKA 1119 ENZYME, KINASE inhibitor CHEMBL3545084 TCD-717 40124 27333 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Monoaryl-1,2-diamine derivative 3 40125 27334 ARSA 410 DRUGGABLE GENOME, ENZYME methylphenidate METHYLPHENIDATE 29382897 40126 27335 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR lamotrigine LAMOTRIGINE 27610747,26213157 40127 27336 CDA 978 ENZYME, DRUGGABLE GENOME DEOXYCYTIDINE DEOXYCYTIDINE 12008078 40128 27337 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-125814 CHEMBL533082 40130 27338 MAPT 4137 DRUGGABLE GENOME P-PHENYLENEDIAMINE CHEMBL403741 40134 27339 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NIFEDIPINE NIFEDIPINE 40135 27340 PPP1CA 5499 KINASE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE CANTHARIDIN CANTHARIDIN 40137 27341 IMPDH1 3614 ENZYME, DRUGGABLE GENOME MYCOPHENOLATE MOFETIL 40138 27342 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME PMID27998201-Compound-5 40139 27343 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME OPROZOMIB OPROZOMIB 40140 27344 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR LINEZOLID LINEZOLID 14561977 40143 27345 CYP51A1 1595 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME VT-1129 40144 27346 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CYTARABINE CYTARABINE 22931300 40145 27347 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565752 CHEMBL1794051 40146 27348 POLI 11201 DNA REPAIR EPIRUBICIN HYDROCHLORIDE EPIRUBICIN HYDROCHLORIDE 40147 27349 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 40148 27350 CRTC1 23373 CLINICALLY ACTIONABLE N/A 40149 27351 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BI-135585 40150 27352 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Alendronate ALENDRONIC ACID 40151 27353 TDO2 6999 ENZYME, DRUGGABLE GENOME PMID27172114-Compound-30 40153 27354 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ETHAVERINE HYDROCHLORIDE ETHAVERINE HYDROCHLORIDE 40154 27355 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IID AESCULIOSIDE IID 20371180 40155 27356 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 252166695 VELDOREOTIDE 40156 27357 SMN2 6607 DRUGGABLE GENOME 2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE CHEMBL201325 40157 27358 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3128043 PF-03758309 40159 27359 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-119915 CHEMBL1481974 22524450 40160 27360 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-23 40161 27361 RRM2 6241 DRUGGABLE GENOME, ENZYME inhibitor 178101504 FLUDARABINE 40162 27362 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1697 DILTIAZEM HYDROCHLORIDE 40165 27363 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR SJ000044511 CHEMBL592124 40166 27364 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Quinoxaline derivative 2 40168 27365 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 178102625 40169 27366 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GO-6976 GO-6976 40170 27367 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY VASOPRESSIN VASOPRESSIN 9794722 40171 27368 SCNN1A 6337 DRUGGABLE GENOME, ION CHANNEL AMILORIDE AMILORIDE 40173 27369 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE TAMATINIB R-406 25222877 40174 27370 CPB2 1361 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166875 40175 27371 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME sunitinib SUNITINIB 25344452,26244574,24013576 40179 27372 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 381744994 LEROCICLIB 40180 27373 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME BAS03450373 CHEMBL1576310 40181 27374 MAP2K5 5607 KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 328083482 40183 27375 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME 8-GERANYLOXY PSORALEN CHEMBL1412710 22222157 40184 27376 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CILENGITIDE CILENGITIDE 24095096 40189 27377 CBX1 10951 NA S-(P-AZIDOPHENACYL)GLUTATHIONE CHEMBL1256813 40190 27378 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1200598 DIETHYLSTILBESTROL DIPHOSPHATE 40192 27379 ALDH1A1 216 DRUGGABLE GENOME, ENZYME LIOTHYRONINE SODIUM LIOTHYRONINE SODIUM 40194 27380 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME INCB54828 40196 27381 SMN1 6606 DRUGGABLE GENOME PHENAMIL METHANESULFONATE PHENAMIL METHANESULFONATE 40197 27382 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor CHEMBL91829 RUBOXISTAURIN 40198 27383 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100315 40202 27384 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SB-202190 SB-202190 40203 27385 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor CHEMBL488436 AZD-5438 40204 27386 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TOPOISOMERASE INHIBITORS 16981845 40205 27387 KDM4A 9682 DRUGGABLE GENOME, ENZYME FRAXETIN FRAXETIN 40206 27388 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL PF-05241328 PF-05241328 40207 27389 RACGAP1 29127 NA DNDI1417156 CHEMBL1504679 40208 27390 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28270010-Compound-Figure5-2 40209 27391 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE METFORMIN METFORMIN 26471090 40211 27392 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PHENYTOIN PHENYTOIN 15698863 40213 27393 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR SULODEXIDE SULODEXIDE 40214 27394 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL antagonist CHEMBL3545042 SELURAMPANEL 40216 27395 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 135650235 EPLERENONE 40217 27396 ATXN2 6311 NA VINBLASTINE SULFATE VINBLASTINE SULFATE 40218 27397 MAPT 4137 DRUGGABLE GENOME 4,6-BIS(4-MORPHOLINOSTYRYL)PYRIMIDINE CHEMBL2181046 22913544 40222 27398 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Imiglitazar IMIGLITAZAR 40223 27399 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME COBALT 6203298 40224 27400 PSMA6 5687 PROTEASE, DRUGGABLE GENOME CARFILZOMIB CARFILZOMIB 24524217 40225 27401 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE NVP-BEZ238 40226 27402 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 354702265 PF-114 40227 27403 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE IRIGENOL IRIGENOL 40228 27404 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE GW559768X GW559768X 17884497 40230 27405 PTPN6 5777 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE HEN EGG LYSOZYME 7600299 40231 27406 FAP 2191 PROTEASE, CELL SURFACE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Talabostat TALABOSTAT 40232 27407 MAPT 4137 DRUGGABLE GENOME Tau-binding PET tracer 40233 27408 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PACLITAXEL PACLITAXEL 25010864 40234 27409 CEP43 11116 CLINICALLY ACTIONABLE brivanib BRIVANIB 20124951 40235 27410 GMNN 51053 DRUGGABLE GENOME GNF-PF-4464 CHEMBL600692 40236 27411 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200733 DESFLURANE 40238 27412 DHFR 1719 DRUGGABLE GENOME, ENZYME TAMOXIFEN TAMOXIFEN 3978632 40240 27413 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CARTEOLOL CARTEOLOL 40241 27414 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CANAVANINE CANAVANINE 40242 27415 HTT 3064 DRUGGABLE GENOME RAFOXANIDE RAFOXANIDE 40243 27416 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ADAPALENE ADAPALENE 40244 27417 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PROGESTOGEN PROGESTOGEN 40245 27418 MAPT 4137 DRUGGABLE GENOME AG-537 CHEMBL67535 40246 27419 TOP2B 7155 DRUGGABLE GENOME, ENZYME Lucanthone LUCANTHONE 40248 27420 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FGFR INHIBITOR AZD4547 23082000,27535980 40250 27421 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1200594 40251 27422 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME THALIDOMIDE THALIDOMIDE 40253 27423 CSF3 1440 GROWTH FACTOR, DRUGGABLE GENOME DA-3031 40254 27424 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISOQUINE ISOQUINE 19222165,19284751 40255 27425 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CILOSTAZOL CILOSTAZOL 22931300 40256 27426 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102912 CHLOROPICRIN 40258 27427 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE BGB-283 LIFIRAFENIB 26208524 40259 27428 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PROMAZINE PROMAZINE 40263 27429 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR prednisone PREDNISONE 24141364 40264 27430 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE UCART123 40265 27431 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TCMDC-124571 CHEMBL533542 40266 27432 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CID 4101591 CHEMBL428789 40267 27433 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-19063 CHEMBL1310138 40269 27434 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL661 ALPRAZOLAM 40270 27435 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER fluoxetine glucuronide 40271 27436 MGAT2 4247 ENZYME N-containing heterocyclic derivative 1 40272 27437 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE PMID27841036-Compound-37 40273 27438 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME CEFOTAXIME CEFOTAXIME 15895687 40275 27439 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR cyclosporine CYCLOSPORINE 18444945 40276 27440 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE atorvastatin ATORVASTATIN 16103896,15900215,18727922,18695978,17289397,15284534 40280 27441 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DICOUMAROL DICUMAROL 14634213 40281 27442 IFNG 3458 DRUGGABLE GENOME VIR-201 40283 27443 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE IMMUNOSUPPRESSIVE 9862695 40284 27444 GJA1 2697 ION CHANNEL PROTEASOME INHIBITOR 16829709 40285 27445 UBE2N 7334 ENZYME, DRUGGABLE GENOME NSC-60339 CHEMBL1448793 40286 27446 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor GDC-0980 APITOLISIB 40287 27447 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Paclitaxel PACLITAXEL 16043828,26307133,21216929 40288 27448 RRM2B 50484 ENZYME, DRUGGABLE GENOME, DNA REPAIR GEMCITABINE GEMCITABINE 40289 27449 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor AZD7762 AZD-7762 40291 27450 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CYCLOASPEPTIDE A CYCLOASPEPTIDE A 40292 27451 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE OSI-027 OSI-027 21673091 40293 27452 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-8186 CHEMBL122355 40294 27453 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE Pyrimidine analogues 21325291,10652619,16249645,15918040,21273624,27864592,20819423,27995989,21167658,20714149,27001118,20638924,17203168,23263912,21362378,25677447,20385995,20165956,14522928,27557140,20665215,11913730,20932673,20647221,21919605,16182121,16818689,12782596 40296 27454 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Triazole derivative 7 40297 27455 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME PD-0166285 PD-0166285 40299 27456 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Fused thiophene derivative 1 40301 27457 TXK 7294 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 178103494 IBRUTINIB 40303 27458 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE CANERTINIB CANERTINIB 40304 27459 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE DNDI1417467 CHEMBL1997335 40305 27460 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER zidovudine ZIDOVUDINE 22960662,23996099 40306 27461 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL403989 TG100-801 40307 27462 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME CYC-116 CYC-116 40308 27463 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME BIVALIRUDIN BIVALIRUDIN 40310 27464 MAPT 4137 DRUGGABLE GENOME GNF-PF-1549 CHEMBL227959 40311 27465 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL1852688 INFIGRATINIB 40314 27466 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1091 HYDROCORTISONE ACETATE 40316 27467 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME agonist 135651492 GLYCINE 40317 27468 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor AFATINIB AFATINIB 40319 27469 TSPO 706 DRUGGABLE GENOME Clotiazepam CLOTIAZEPAM 40320 27470 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MITOMYCIN MITOMYCIN 40321 27471 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-242717 CHEMBL269450 40322 27472 MAPT 4137 DRUGGABLE GENOME MACLURAXANTHONE MACLURAXANTHONE 40323 27473 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR somatropin recombinant 23567489 40324 27474 BAZ2B 29994 NA TCMDC-124176 CHEMBL588038 40325 27475 FPGS 2356 ENZYME, DRUGGABLE GENOME methotrexate METHOTREXATE 19902562 40327 27476 BAZ2B 29994 NA CEPHALOCHROMIN CEPHALOCHROMIN 40328 27477 TET2 54790 CLINICALLY ACTIONABLE, ENZYME N/A 24507812,23099237,24994606,26769228,24524305,25224413,25412851,19666869 40329 27478 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME AMG900 AMG-900 40330 27479 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BUTACHLOR BUTACHLOR 40332 27480 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE FGF/VEGF RECEPTOR TYROSINE KINASE INHIBITOR, PD173074 24124571 40333 27481 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE BLM BLEOMYCIN 16224526 40334 27482 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 252166898 40335 27483 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE VANDETANIB VANDETANIB 40338 27484 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZO[E]PYRENE BENZO[E]PYRENE 40339 27485 MAPT 4137 DRUGGABLE GENOME CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE CHEMBL457504 40340 27486 ABHD6 57406 PHOSPHOLIPASE, ENZYME Piperazine carbamic compound 4 40341 27487 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PIPOBROMAN PIPOBROMAN 40344 27488 DNER 92737 NA PMID26924192-Compound-56 40349 27489 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE XL147 PILARALISIB 25637314 40350 27490 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 384403641 RG-1530 40351 27491 EIF2AK2 5610 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR BCG BCG VACCINE 16301626 40352 27492 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE LAROTRECTINIB LAROTRECTINIB 32315394,29606586,29920189 40353 27493 DHFR 1719 DRUGGABLE GENOME, ENZYME Iclaprim ICLAPRIM 40354 27494 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GNF-PF-3084 CHEMBL601135 40355 27495 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PD-98059 CHEMBL35482 40356 27496 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX ANTISENSE AGENT 9185577 40357 27497 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL979 MEPROBAMATE 40359 27498 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE SORBITOL SORBITOL 11879194 40360 27499 SLC28A2 9153 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME ribavirin RIBAVIRIN 26071337 40361 27500 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE ACTB1003 40362 27501 ENO2 2026 CELL SURFACE GABAPENTIN GABAPENTIN 15780189 40363 27502 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER elacridar ELACRIDAR 40365 27503 RAPGEF3 10411 ENZYME GNF-PF-2272 CHEMBL601757 40366 27504 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 252827523 CEBRANOPADOL 40367 27505 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 4 40368 27506 RGS4 5999 DRUGGABLE GENOME LEUKOTRIENE D4 LEUKOTRIENE D4 40370 27507 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 310264783 40372 27508 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Levobunolol LEVOBUNOLOL 40375 27509 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PODOFILOX PODOFILOX 40377 27510 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL235191 TACEDINALINE 40382 27511 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MI-63 21725357 40383 27512 PTGS2 5743 DRUGGABLE GENOME, ENZYME SALSALATE SALSALATE 40384 27513 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IBUFENAC IBUFENAC 40386 27514 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE TAE-684 TAE-684 40387 27515 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2015042088Example12 40389 27516 POLK 51426 DNA REPAIR, ENZYME ARACHIDONIC ACID ARACHIDONIC ACID 40390 27517 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BEZ235 DACTOLISIB 40391 27518 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NANDROLONE PHENPROPIONATE NANDROLONE PHENPROPIONATE 40392 27519 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR INSULIN INSULIN 17392554 40393 27520 MAPT 4137 DRUGGABLE GENOME ETHOPROPAZINE HYDROCHLORIDE ETHOPROPAZINE HYDROCHLORIDE 40394 27521 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ISOFLAVONES 17182792 40395 27522 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME darifenacin DARIFENACIN 40396 27523 GAA 2548 DRUGGABLE GENOME, ENZYME RUTIN RUTIN 40397 27524 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201560 PEGINTERFERON ALFA-2A 40398 27525 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME BAY-613606 CHEMBL541400 40400 27526 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME OXOGLAUCINE OXOGLAUCINE 40401 27527 ATXN2 6311 NA FLUPENTIXOL FLUPENTIXOL 40402 27528 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GNF-PF-1192 CHEMBL584854 40403 27529 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DEXAMETHASONE-SPERMINE CHEMBL1275761 20308375 40404 27530 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR VORINOSTAT VORINOSTAT 40405 27531 BRD1 23774 ENZYME inhibitor 336446910 40406 27532 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PMA 9528865 40412 27533 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME LINIFANIB LINIFANIB 40413 27534 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID27774824-Compound-Figure9Example2down 40414 27535 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ROSIGLITAZONE ROSIGLITAZONE 15998575 40416 27536 PAH 5053 DRUGGABLE GENOME, ENZYME SAPROPTERIN SAPROPTERIN 40417 27537 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Bevacizumab + Trastuzumab 40419 27538 PHEX 5251 ENZYME, PROTEASE, DRUGGABLE GENOME VITAMIN D 15951631,12579406 40421 27539 PDE4A 5141 DRUGGABLE GENOME, ENZYME TA-7906 40423 27540 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME CYC-116 CYC-116 40425 27541 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1,3-DIPHENYLTHIOUREA CHEMBL275260 40427 27542 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME STICTIC ACID STICTIC ACID 40429 27543 KLC1 3831 NA leucovorin LEUCOVORIN 17549067 40430 27544 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME Sotrastaurin acetate 40431 27545 NCOA3 8202 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, ENZYME CYTARABINE CYTARABINE 40432 27546 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DISULFIRAM DISULFIRAM 40433 27547 SLC15A1 6564 DRUGGABLE GENOME, TRANSPORTER 178101375 40434 27548 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650700 40437 27549 GMNN 51053 DRUGGABLE GENOME MEBENDAZOLE MEBENDAZOLE 40438 27550 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417701 CHEMBL1326164 40439 27551 IL1B 3553 KINASE, DRUGGABLE GENOME LITHIUM LITHIUM 9342951 40440 27552 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME N/A 23656643,24441292,24081659 40441 27553 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist,antagonist 135651403 40442 27554 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR BCG VACCINE 12126899 40444 27555 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 7-METHOXYISOFLAVONE CHEMBL563919 40445 27556 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ACEBUTOLOL ACEBUTOLOL 2903243 40446 27557 NDUFC2 4718 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 40447 27558 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antagonist CHEMBL1743001 CIXUTUMUMAB 40448 27559 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE PERIFOSINE PERIFOSINE 40450 27560 BAZ2B 29994 NA MORIN MORIN 40451 27561 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL628 PENTOXIFYLLINE 40453 27562 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE bevacizumab BEVACIZUMAB 29662106,20634689,19307503 40455 27563 POLK 51426 DNA REPAIR, ENZYME LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 40456 27564 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Azatadine AZATADINE 40458 27565 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE FAT EMULSION 8110872 40459 27566 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE ALPELISIB ALPELISIB 25544636,25409150 40462 27567 CD276 80381 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Omburtamab I-131 40463 27568 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMA 2564369,8104888,2547869,7693806 40464 27569 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR Pyrazolopyrimidine and thienopyrimidine amide derivative 2 40465 27570 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUTAPROST BUTAPROST 40466 27571 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR GNF-PF-4242 CHEMBL584514 40467 27572 FTO 79068 ENZYME atenolol ATENOLOL 40468 27573 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX GOSSYPETIN GOSSYPETIN 25190466 40469 27574 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 40471 27575 COL4A1 1282 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 40472 27576 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FP-1039 FP-1039 40474 27577 NOS1 4842 DRUGGABLE GENOME, ENZYME BCG BCG VACCINE 16142388 40476 27578 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLOTIAZEPAM CLOTIAZEPAM 40477 27579 GMNN 51053 DRUGGABLE GENOME BREFELDIN A BREFELDIN A 40478 27580 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE DOXORUBICIN DOXORUBICIN 21094049,19053767,17276690 40481 27581 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR DAUNORUBICIN DAUNORUBICIN 22260166 40482 27582 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE antibody DULANERMIN DULANERMIN 40483 27583 CPD 1362 ENZYME, DRUGGABLE GENOME, PROTEASE ANTISERUM 9490632 40486 27584 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE AMG 208 40487 27585 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US9682991, 7 40488 27586 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545080 RG-7256 40491 27587 SCD 6319 DRUGGABLE GENOME, ENZYME MK-8245 MK-8245 40492 27588 MAPT 4137 DRUGGABLE GENOME 2-AMINOPHENOXAZINONE CHEMBL146710 40493 27589 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METRONIDAZOLE METRONIDAZOLE 17374625 40494 27590 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2029988 CEP-32496 40495 27591 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZD8186 AZD-8186 26725216 40496 27592 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE prasugrel PRASUGREL 28820077,23859572 40497 27593 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE WR-243246 CHEMBL117217 40498 27594 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Sulfamoylamide derivative 1 40499 27595 IMPDH1 3614 ENZYME, DRUGGABLE GENOME MYCOPHENOLIC ACID 40500 27596 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID25991433-Compound-A1 40501 27597 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CHLORPROMAZINE CHLORPROMAZINE 40503 27598 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME regorafenib REGORAFENIB 40505 27599 TUBB2A 7280 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 40506 27600 AQP3 360 ION CHANNEL, TRANSPORTER inhibitor 178101032 40507 27601 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102230 BINODENOSON 40508 27602 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR FORETINIB FORETINIB 25688157,26372962 40514 27603 ALDH1A1 216 DRUGGABLE GENOME, ENZYME LINOLENIC ACID LINOLENIC ACID 40515 27604 TXNRD1 7296 DRUGGABLE GENOME Metal complex derivative 1 40516 27605 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR METHIOCARB METHIOCARB 40517 27606 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME clavulanate CLAVULANIC ACID 20800921,10535882,30664875 40518 27607 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102611 40519 27608 SLC22A11 55867 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER PROBENECID PROBENECID 40520 27609 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Cobimetinib COBIMETINIB 40521 27610 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CATECHOL CATECHOL 40523 27611 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR TALAROFLAVONE TALAROFLAVONE 18178092 40525 27612 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ANTIESTROGENS 9205071 40526 27613 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL284348 DALFAMPRIDINE 40528 27614 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR inhibitor CHEMBL1743022 FRESOLIMUMAB 40529 27615 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-8 40530 27616 PLA2G7 7941 DRUGGABLE GENOME, ENZYME inhibitor 354702269 40531 27617 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TAE226 26090892 40532 27618 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Binimetinib BINIMETINIB 40533 27619 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565816 40534 27620 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME PMID27998201-Compound-5 40536 27621 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL3707227 ATEZOLIZUMAB 40537 27622 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 223366212 CP-724714 40538 27623 ROR2 4920 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CELL SURFACE, ENZYME CCT301-59 (targeting ROR2) 40539 27624 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565590 CHEMBL1236539 40540 27625 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Succimer SUCCIMER 40541 27626 NDUFS3 4722 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545320 ME-344 40542 27627 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL457748 MB07811 40543 27628 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ALPRENOLOL ALPRENOLOL 40544 27629 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEFOTAXIME SODIUM CEFOTAXIME SODIUM 40545 27630 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1737 SILDENAFIL CITRATE 40548 27631 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 384403668 40549 27632 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE 7-azaindole derivative 1 40550 27633 DPP8 54878 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 363894200 TENELIGLIPTIN 40551 27634 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417055 CHEMBL1486366 40552 27635 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CISPLATIN CISPLATIN 8314134 40553 27636 TAT 6898 ENZYME ENZYME INHIBITOR 85301 40554 27637 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ZK-164015 CHEMBL184074 40555 27638 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ATAZANAVIR ATAZANAVIR 16355344 40556 27639 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME MVA-BN Breast 40557 27640 DHFR 1719 DRUGGABLE GENOME, ENZYME PYRIMETHAMINE PYRIMETHAMINE 25984755 40558 27641 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DPPE TESMILIFENE HYDROCHLORIDE 11556524 40561 27642 GMNN 51053 DRUGGABLE GENOME GNF-PF-2260 CHEMBL601351 40562 27643 KDM1A 23028 DRUGGABLE GENOME, ENZYME, CELL SURFACE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING inhibitor 178103602 40564 27644 KDM4A 9682 DRUGGABLE GENOME, ENZYME PARAROSANILINE PARAROSANILINE 40565 27645 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR LARGAZOLE LARGAZOLE 21420302,25203782,20491440 40566 27646 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor PD325901 40567 27647 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 385612230 40568 27648 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Ibandronate IBANDRONIC ACID 40569 27649 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME inhibitor 405067337 40570 27650 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135649968 ASTEMIZOLE 40571 27651 POLI 11201 DNA REPAIR S-(P-AZIDOPHENACYL)GLUTATHIONE CHEMBL1256813 40573 27652 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 quetiapine QUETIAPINE 40574 27653 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME BCG BCG VACCINE 9393826 40575 27654 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 178102551 KU-55933 40576 27655 SIK1 150094 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 178102336 BOSUTINIB 40577 27656 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CHEMBL2109271 MDX-210 40578 27657 PSMB6 5694 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL325041 BORTEZOMIB 40579 27658 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 363894211 PEXMETINIB 40580 27659 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL2108569 INSULIN PEGLISPRO 40583 27660 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 178100876 40584 27661 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE CURCUMIN CURCUMIN 40585 27662 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Benzimidazole derivative 7 40586 27663 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR ALD-518 CLAZAKIZUMAB 40587 27664 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor 178103944 APREMILAST 40588 27665 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE B-Lactams 40589 27666 RGS4 5999 DRUGGABLE GENOME inhibitor 252827386 40590 27667 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHANQUONE PHANQUONE 40591 27668 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PAROXETINE PAROXETINE 40593 27669 ATAD5 79915 NA QUERCETIN QUERCETIN 40598 27670 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE DASATINIB DASATINIB 22328973 40599 27671 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-4384 CHEMBL602763 40600 27672 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME ANTIANGIOGENIC 17138942 40602 27673 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1201728 DESVENLAFAXINE SUCCINATE 40605 27674 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 EGCG EPIGALOCATECHIN GALLATE 17108060 40606 27675 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-7387 CHEMBL119878 40612 27676 ADK 132 DRUGGABLE GENOME, ENZYME, KINASE LOMUSTINE LOMUSTINE 6317371 40613 27677 GMNN 51053 DRUGGABLE GENOME NORARMEPAVINE NORARMEPAVINE 40614 27678 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Saracatinib SARACATINIB 25394791,26802156 40615 27679 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TELMISARTAN TELMISARTAN 40616 27680 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Cerdulatinib CERDULATINIB 40617 27681 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PIPERINE PIPERINE 40618 27682 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor XL-765 VOXTALISIB 40619 27683 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AG-1288 CHEMBL166486 40621 27684 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NORGESTREL NORGESTREL 40622 27685 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 40623 27686 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE NIVOLUMAB NIVOLUMAB 29773717 40624 27687 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TIOTROPIUM TIOTROPIUM 40625 27688 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE LYNGBYABELLIN A LYNGBYABELLIN A 40626 27689 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL49642 INDIBULIN 40627 27690 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201743 SAXAGLIPTIN HYDROCHLORIDE 40628 27691 KDM4A 9682 DRUGGABLE GENOME, ENZYME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 40630 27692 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR OBTUSAQUINONE OBTUSAQUINONE 40631 27693 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 135651418 ALITRETINOIN 40635 27694 POLK 51426 DNA REPAIR, ENZYME NBQX NBQX 40636 27695 POLK 51426 DNA REPAIR, ENZYME METHACYCLINE HYDROCHLORIDE METHACYCLINE HYDROCHLORIDE 40637 27696 MAPT 4137 DRUGGABLE GENOME TCMDC-125580 CHEMBL528807 40639 27697 ABL2 27 KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME DASATINIB DASATINIB 40640 27698 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE fluorouracil FLUOROURACIL 40642 27699 BRCA2 675 CLINICALLY ACTIONABLE Everolimus EVEROLIMUS 26546619 40643 27700 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PROPRANOLOL PROPRANOLOL 22931300 40644 27701 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417149 CHEMBL1622802 40645 27702 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING AR-42 AR-42 40649 27703 ALDH3A1 218 DRUGGABLE GENOME, ENZYME ETHANOL ALCOHOL 15909415,12652939,14987799 40650 27704 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SALMETEROL XINAFOATE SALMETEROL XINAFOATE 40651 27705 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME PMID27774824-Compound-Figure6Example12 40652 27706 TXN2 25828 DRUGGABLE GENOME, THIOREDOXIN BIOTINYLATED GAMBOGIC ACID BIOTINYLATED GAMBOGIC ACID 22663155 40653 27707 MAPT 4137 DRUGGABLE GENOME GNF-PF-2968 CHEMBL582473 40654 27708 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor CHEMBL3545368 PANOBINOSTAT LACTATE 40657 27709 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR H3B-6545 40659 27710 TUBB3 10381 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 40661 27711 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME APG-115 40662 27712 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-47924 CHEMBL1269845 40667 27713 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 40668 27714 IGFBP3 3486 DRUGGABLE GENOME celecoxib CELECOXIB 22336956 40669 27715 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE TUMOR NECROSIS FACTOR 12584200 40670 27716 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Betamethasone Benzoate 40671 27717 TXNRD1 7296 DRUGGABLE GENOME Bis-sulfonamide derivative 1 40672 27718 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE AMG 337 27196749,25326232,27196782,26432108 40673 27719 BTC 685 DRUGGABLE GENOME, GROWTH FACTOR panitumumab PANITUMUMAB 40674 27720 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL592054 IMIGLITAZAR 40675 27721 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE DIENESTROL DIENESTROL 40676 27722 MAOB 4129 DRUGGABLE GENOME, ENZYME TRANYLCYPROMINE TRANYLCYPROMINE 40677 27723 PTGS2 5743 DRUGGABLE GENOME, ENZYME antiinflammatory and antirheumatic products, non-steroids 22336956 40679 27724 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 40681 27725 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Quinazolinone derivative 1 40682 27726 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ZOXAZOLAMINE ZOXAZOLAMINE 22931300 40683 27727 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE BUPRANOLOL BUPRANOLOL 2903243 40684 27728 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651637 BRADYKININ 40685 27729 GPER1 2852 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR agonist 135650883 RALOXIFENE 40686 27730 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE COLCHICINE COLCHICINE 40687 27731 APOE 348 DRUGGABLE GENOME Antivirals for treatment of HIV infections, combinations 17700364,15809899 40690 27732 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 4'-METHOXYCHALCONE 4'-METHOXYCHALCONE 40691 27733 MAPT 4137 DRUGGABLE GENOME 5-BENZYLOXYTRYPTAMINE 5-BENZYLOXYTRYPTAMINE 40692 27734 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE C-Met/PD-L1 CAR-T Cell 40693 27735 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Propranolol PROPRANOLOL 40695 27736 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME cisplatin CISPLATIN 21636554 40697 27737 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 40699 27738 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL408513 BELINOSTAT 40701 27739 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565847 40702 27740 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-1969 CHEMBL601364 40703 27741 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME MCS-110 MCS-110 40704 27742 PNMT 5409 DRUGGABLE GENOME, ENZYME inhibitor 178103244 40705 27743 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1201065 THIAMYLAL SODIUM 40706 27744 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor PERIFOSINE PERIFOSINE 40707 27745 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE CHEMBL457504 40708 27746 ADAMTS1 9510 ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE pravastatin PRAVASTATIN 18174457 40714 27747 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GW-409544 40715 27748 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545359 ARRY-300 40716 27749 CAMLG 819 NA CYCLOSPORINE CYCLOSPORINE 40717 27750 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamide derivative 24 40718 27751 PDE4A 5141 DRUGGABLE GENOME, ENZYME IPL455 40719 27752 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR allosteric modulator 404859053 40720 27753 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME methimazole METHIMAZOLE 26599303,26151496 40722 27754 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME CV-9201 40723 27755 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE TIAPROFENIC ACID TIAPROFENIC ACID 40724 27756 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE ARQ 087 40725 27757 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DANTROLENE DANTROLENE 22931300 40727 27758 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR SERM 11901050 40729 27759 BAZ2B 29994 NA RHEIN RHEIN 40731 27760 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL482767 SNS-314 40733 27761 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR N-PROPYL BROMIDE N-PROPYL BROMIDE 40734 27762 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-4325 CHEMBL598263 40735 27763 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE 9-AC 10803925 40738 27764 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3,7-DIMETHOXYFLAVONE 3,7-DIMETHOXYFLAVONE 40739 27765 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR BELINOSTAT BELINOSTAT 40742 27766 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PAEONOL PAEONOL 40743 27767 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME ECULIZUMAB ECULIZUMAB 40744 27768 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Salirasib SALIRASIB 21847063 40745 27769 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE AT-101 ISOSORBIDE 40748 27770 ALOX15 246 ENZYME, DRUGGABLE GENOME GERANIOL GERANIOL 40749 27771 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NIFEDIPINE NIFEDIPINE 40750 27772 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3545332 CEP-2563 40752 27773 ATXN2 6311 NA TANSHINONE I TANSHINONE I 40753 27774 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ERGOCRYPTINE ERGOCRYPTINE 40755 27775 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW876790X GW876790X 40756 27776 TAT 6898 ENZYME PHENOBARBITAL PHENOBARBITAL 1688552 40757 27777 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR R-N-PROPYLNORAPOMORPHINE R-N-PROPYLNORAPOMORPHINE 40758 27778 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BP-897 BP-897 40759 27779 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME AG-494 CHEMBL56731 40760 27780 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLEBOPRIDE MALEATE CLEBOPRIDE MALEATE 40761 27781 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ISOPRENALINE ISOPROTERENOL 40762 27782 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TETRADECYLTHIOACETIC ACID TETRADECYLTHIOACETIC ACID 20036122 40764 27783 SLC22A3 6581 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER lamivudine LAMIVUDINE 40765 27784 VEGFB 7423 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR inhibitor SORAFENIB TOSYLATE 40766 27785 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE GNF-PF-3023 CHEMBL535331 40768 27786 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME KA2507 40771 27787 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL1236107 SGX-523 40772 27788 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME WX-554 WX-554 40774 27789 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME antagonist HGS 1029 40775 27790 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545063 OSIMERTINIB MESYLATE 40777 27791 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 405560501 40778 27792 TNFRSF9 3604 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE CD28 and CD137 CAR-T Cells 40779 27793 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME TRAZODONE TRAZODONE 40780 27794 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 40781 27795 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565763 40782 27796 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR METHACYCLINE HYDROCHLORIDE METHACYCLINE HYDROCHLORIDE 40783 27797 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 3-(PHENYLAMINO)PHENOL CHEMBL1523215 40786 27798 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL2048028 LIFITEGRAST 40787 27799 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Carbamide derivative 7 40788 27800 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME inhibitor 252166600 40789 27801 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL19019 NALTREXONE 40791 27802 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR GLYCYRRHETINIC ACID 15070972 40794 27803 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CETIRIZINE CETIRIZINE 40795 27804 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR MERCURIC CHLORIDE MERCURIC CHLORIDE 40796 27805 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME inhibitor 252827445 40797 27806 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME APOMORPHINE APOMORPHINE 40800 27807 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 252827454 40801 27808 TNFRSF4 7293 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE MEDI0562 TAVOLIMAB 40802 27809 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME LEVOCABASTINE LEVOCABASTINE 40803 27810 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR sparsentan SPARSENTAN 40805 27811 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME activator 404859002 40806 27812 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROPYLENE GLYCOL MONOSTEARATE PROPYLENE GLYCOL MONOSTEARATE 40808 27813 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME inhibitor 178102663 40810 27814 MUC16 94025 DRUGGABLE GENOME B43.13 9671143 40812 27815 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2368861 BUPRENORPHINE HYDROCHLORIDE 40813 27816 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Cytarabine CYTARABINE 27443263 40814 27817 CA2 760 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL20 ACETAZOLAMIDE 40817 27818 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DIMETHYLCURCUMIN DIMETHYLCURCUMIN 25753330 40818 27819 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL396778 SAFINAMIDE 40819 27820 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 315661252 40821 27821 PSMC1 5700 PROTEASE inhibitor CHEMBL325041 BORTEZOMIB 40822 27822 RAB9A 9367 ENZYME, DRUGGABLE GENOME ILEPCIMIDE ILEPCIMIDE 40823 27823 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME STEEL FACTOR 11162574 40824 27824 KMT2C 58508 ENZYME, CLINICALLY ACTIONABLE, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, DRUG RESISTANCE ANASTROZOLE ANASTROZOLE 29755131 40825 27825 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200339 PHENYLEPHRINE HYDROCHLORIDE 40826 27826 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR D-DOPA CHEMBL211670 40827 27827 NOS1 4842 DRUGGABLE GENOME, ENZYME GINKGO BILOBA 11550802 40828 27828 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE IRINOTECAN IRINOTECAN 40829 27829 POLK 51426 DNA REPAIR, ENZYME EVANS BLUE EVANS BLUE 40830 27830 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR DEPHOSTATIN DEPHOSTATIN 40832 27831 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CHEMBL2068724 ACAMPROSATE CALCIUM 40833 27832 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270010-Compound-Figure5-3 40835 27833 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER RANITIDINE RANITIDINE 9862768 40837 27834 AMH 268 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TESTOSTERONE TESTOSTERONE 11248089,11545286,1292985,14584782,11315948,7962305,7818099 40838 27835 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME Platinum compounds 30672383 40839 27836 GP6 51206 CELL SURFACE, KINASE aspirin ASPIRIN 16493486 40841 27837 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR TCDD 9772220 40842 27838 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyrimidine derivative 5 40844 27839 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 buprenorphine BUPRENORPHINE 26407542,31676110 40845 27840 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Echothiophate Iodide 40846 27841 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL2103852 CROLIBULIN 40847 27842 P2RX4 5025 ION CHANNEL, DRUGGABLE GENOME antagonist 178101492 PAROXETINE 40848 27843 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 zolpidem ZOLPIDEM 9187528 40849 27844 CA9 768 DRUGGABLE GENOME, ENZYME PARABEN PARABEN 40851 27845 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME APX-3330 40852 27846 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CORTICOSTERONE CORTICOSTERONE 40854 27847 POLI 11201 DNA REPAIR GNF-PF-2272 CHEMBL601757 40855 27848 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CER-002 CER-002 40856 27849 SCD 6319 DRUGGABLE GENOME, ENZYME CLOFIBRATE CLOFIBRATE 11162472 40858 27850 KLK2 3817 PROTEASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 252166872 40859 27851 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SORAFENIB SORAFENIB 40860 27852 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PANITUMUMAB PANITUMUMAB 28275037 40863 27853 SMAD2 4087 KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX BISDEMETHOXYCURCUMIN BISDEMETHOXYCURCUMIN 23145932 40864 27854 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE PRED 11911117 40865 27855 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200964 AMITRIPTYLINE HYDROCHLORIDE 40866 27856 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antibody 223365910 DUPILUMAB 40868 27857 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE zolpidem ZOLPIDEM 40870 27858 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME 4-(thiazol-5-yl)-pyrimidine derivative 2 40871 27859 HMGCR 3156 ENZYME, DRUGGABLE GENOME Hexahydro naphthalene derivative 3 40872 27860 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Selumetinib SELUMETINIB 22197931,22327936,25394791,18632602,19915144,26582713,24448821,27312529 40873 27861 MPI 4351 ENZYME, DRUGGABLE GENOME 4-HYDROXYESTRADIOL CHEMBL1412489 40876 27862 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DICUMAROL DICUMAROL 12584558 40879 27863 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CINNARIZINE CINNARIZINE 40880 27864 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE TAXANES 12558997 40881 27865 EPHB3 2049 DRUGGABLE GENOME, TYROSINE KINASE, KINASE inhibitor 249565821 40882 27866 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Triptolidenol analog 1 40883 27867 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Indole-based analog 3 40884 27868 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME allosteric modulator 252166893 CHEMBL493241 40885 27869 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME GNF-PF-3148 CHEMBL81782 40887 27870 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3545423 AZD-1208 40888 27871 NAT1 9 ENZYME, DRUGGABLE GENOME ASPIRIN ASPIRIN 10547619 40889 27872 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TELENZEPINE TELENZEPINE 40892 27873 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 354702287 40893 27874 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Azathioprine AZATHIOPRINE 40894 27875 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE 178101779 40895 27876 KCNF1 3754 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 40896 27877 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DOCUSATE SODIUM DOCUSATE SODIUM 40897 27878 MAPT 4137 DRUGGABLE GENOME PBT-2 40898 27879 CAV1 857 TRANSPORTER, KINASE ETHANOL ALCOHOL 15845868 40899 27880 LGALS1 3956 KINASE, DRUGGABLE GENOME US8703720, Reference Compound 2 40900 27881 TNC 3371 DRUGGABLE GENOME, FIBRINOGEN CHEMBL1743077 TENATUMOMAB 40901 27882 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650057 CARVEDILOL 40902 27883 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME OLEIC ACID OLEIC ACID 40905 27884 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-3756 CHEMBL597035 40906 27885 POLK 51426 DNA REPAIR, ENZYME SB-415286 CHEMBL322970 40907 27886 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL MC-1 40908 27887 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107762 NERISPIRDINE 40910 27888 HTT 3064 DRUGGABLE GENOME PMID27376512-Compound-PG-11048 40911 27889 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CYPROHEPTADINE CYPROHEPTADINE 40912 27890 LIG3 3980 NA cyclophosphamide CYCLOPHOSPHAMIDE 24533712 40914 27891 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE GO-6976 GO-6976 40916 27892 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Thiadiazolidindione derivative 1 40917 27893 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SALT VOLANESORSEN SODIUM 10100098 40918 27894 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR 4-HC PERFOSFAMIDE 1283360 40919 27895 GALNS 2588 DRUGGABLE GENOME, ENZYME Elosulfase alfa 40920 27896 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-8 40921 27897 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Geminally-substituted cyanoethylpypazolo pyridone derivative 2 40922 27898 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CUDC-101 CUDC-101 40924 27899 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GATIFLOXACIN GATIFLOXACIN 40928 27900 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PYRANTEL PAMOATE PYRANTEL PAMOATE 40929 27901 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE KD-025 CHEMBL2005186 40930 27902 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102476 40934 27903 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE vaccine S-3304 S-3304 40935 27904 DKK3 27122 DRUGGABLE GENOME REIC gene therapy 40936 27905 HTT 3064 DRUGGABLE GENOME GNF-PF-4300 CHEMBL585656 40938 27906 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME MNU 10469609,10439048 40939 27907 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE BCP9000383 40941 27908 TNRC6A 27327 NA ethanol ALCOHOL 32451486 40942 27909 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE FENBENDAZOLE FENBENDAZOLE 40943 27910 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Azetidine derivative 5 40946 27911 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TAE-684 TAE-684 40947 27912 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor BORTEZOMIB BORTEZOMIB 40949 27913 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE INDOMETHACIN INDOMETHACIN 10403534 40950 27914 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CNQX DISODIUM CHEMBL1255647 40954 27915 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE CISPLATIN CISPLATIN 12894503 40956 27916 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Atezolizumab ATEZOLIZUMAB 40958 27917 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR fulvestrant FULVESTRANT 24185512,24185510 40959 27918 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DICHLON DICHLON 40960 27919 PRKAB1 5564 ENZYME, KINASE, DRUGGABLE GENOME metformin METFORMIN 22722338 40961 27920 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ROTENONE ROTENONE 40962 27921 PI4KA 5297 DRUGGABLE GENOME, ENZYME, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor 178102681 WORTMANNIN 40964 27922 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178102147 SULPIRIDE 40965 27923 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL2110814 DELUCEMINE 40966 27924 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 5 40967 27925 CXCL8 3576 DRUGGABLE GENOME CORONOPILIN CORONOPILIN 40968 27926 NAPEPLD 222236 ENZYME inhibitor 135649999 BITHIONOL 40969 27927 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TOPOTECAN TOPOTECAN 19501511,24502276 40971 27928 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Tihotungstate derivative 1 40972 27929 COL5A2 1290 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 40973 27930 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Prednisolone PREDNISOLONE 28151717 40975 27931 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR doxorubicin DOXORUBICIN 40977 27932 NCOR2 9612 NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 40979 27933 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME N-ETHYLMALEIMIDE N-ETHYLMALEIMIDE 40981 27934 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178103793 40983 27935 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX BUFOGENIN BUFOGENIN 40986 27936 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PITAVASTATIN CALCIUM PITAVASTATIN CALCIUM 40989 27937 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR AEG35156, GEM 640 40990 27938 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR INDOMETHACIN INDOMETHACIN 15131590 40991 27939 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102285 LINIFANIB 40992 27940 MAOB 4129 DRUGGABLE GENOME, ENZYME Sulphadoxine SULPHADOXINE 40993 27941 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 404859149 40994 27942 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-J5 40995 27943 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME MUC-1 dendritic cancer vaccine 40996 27944 FANCC 2176 CLINICALLY ACTIONABLE, DNA REPAIR MELPHALAN MELPHALAN 16243825 40997 27945 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME U-37883A CHEMBL333121 40998 27946 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BI-D1870 CHEMBL573107 40999 27947 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BENZO[B]FLUORANTHENE BENZO[B]FLUORANTHENE 41002 27948 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TOSUFLOXACIN TOSYLATE TOSUFLOXACIN TOSYLATE 41004 27949 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-67 CHEMBL578512 41005 27950 TSPO 706 DRUGGABLE GENOME OLESOXIME OLESOXIME 41006 27951 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LEUCINE LEUCINE 22931300 41009 27952 METAP1D 254042 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103847 TOSEDOSTAT 41011 27953 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1707 LOPERAMIDE HYDROCHLORIDE 41012 27954 POLI 11201 DNA REPAIR SELEGILINE HYDROCHLORIDE SELEGILINE HYDROCHLORIDE 41013 27955 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-17 41015 27956 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 30 41016 27957 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIFENOCONAZOLE DIFENOCONAZOLE 41017 27958 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYL ROBUSTONE METHYL ROBUSTONE 41018 27959 GMNN 51053 DRUGGABLE GENOME DICHLORVOS DICHLORVOS 41020 27960 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PIMOZIDE PIMOZIDE 41021 27961 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE OTSSP167 41023 27962 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME STICTIC ACID STICTIC ACID 41025 27963 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL2364605 CEBRANOPADOL 41027 27964 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Galantamine GALANTAMINE 41028 27965 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUOXASTROBIN FLUOXASTROBIN 41032 27966 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME propionic acid derivatives 26398624 41034 27967 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 354702293 41036 27968 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME EBSELEN EBSELEN 41037 27969 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE IMATINIB MESYLATE 26758680,15705718,22371878,19652056,16772610 41039 27970 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Erlotinib ERLOTINIB 41040 27971 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME SIROLIMUS SIROLIMUS 41042 27972 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SB-242235 SB-242235 41043 27973 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Indazole amide derivative 2 41045 27974 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE blocker CHEMBL2107647 LANICEMINE 41046 27975 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SP-600125 SP-600125 41047 27976 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME L-765314 L-765314 41048 27977 HSPA8 3312 TUMOR SUPPRESSOR DEXAMETHASONE DEXAMETHASONE 7542664 41049 27978 ATAD5 79915 NA GNF-PF-2776 CHEMBL578294 41050 27979 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE RETINOIC ACID 8396187 41051 27980 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX RESVERATROL RESVERATROL 41052 27981 SULT2A1 6822 DRUGGABLE GENOME METHOTREXATE METHOTREXATE 17163485 41053 27982 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL552212 LEXIBULIN 41054 27983 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE E7449 2X-121 26513298 41055 27984 CA2 760 DRUGGABLE GENOME, ENZYME FERULIC ACID 41056 27985 KMO 8564 DRUGGABLE GENOME, ENZYME Benzene sulfonamide derivative 4 41057 27986 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL603469 LESTAURTINIB 41059 27987 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER domperidone DOMPERIDONE 41060 27988 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME FENRETINIDE FENRETINIDE 41062 27989 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROPICONAZOLE PROPICONAZOLE 41063 27990 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE (5Z)-7-OXOZEAENOL CHEMBL1077979 41064 27991 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ERGOCRYPTINE ERGOCRYPTINE 41066 27992 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Adalimumab ADALIMUMAB 41067 27993 PTGS2 5743 DRUGGABLE GENOME, ENZYME SUPROFEN SUPROFEN 41069 27994 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METIPRANOLOL METIPRANOLOL 41071 27995 CTSD 1509 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166834 41073 27996 HSPB1 3315 DRUGGABLE GENOME OMEPRAZOLE OMEPRAZOLE 41074 27997 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 135650850 PREDNISOLONE 41075 27998 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AZD5363 CAPIVASERTIB 26910118 41076 27999 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR EPZ-6438 TAZEMETOSTAT 41082 28000 ATXN2 6311 NA NSC-102742 CHEMBL1519374 41083 28001 CES1 1066 DRUGGABLE GENOME, ENZYME irinotecan IRINOTECAN 41085 28002 IDO2 169355 ENZYME 2,3-diamino-benzo[b]thiophene derivative 2 41088 28003 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200437 QUINIDINE GLUCONATE 41089 28004 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1200543 ANILERIDINE PHOSPHATE 41090 28005 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 363894222 PUQUITINIB 41093 28006 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE MM-141 ISTIRATUMAB 41094 28007 PDE3A 5139 ENZYME, DRUGGABLE GENOME Anagrelide ANAGRELIDE 41097 28008 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650342 GSK-9578 41098 28009 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL288441 BOSUTINIB 41099 28010 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR LASOFOXIFENE LASOFOXIFENE 41100 28011 BCHE 590 DRUGGABLE GENOME, ENZYME RIVASTIGMINE RIVASTIGMINE 41106 28012 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200341 INDECAINIDE HYDROCHLORIDE 41107 28013 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TRANSTORINE TRANSTORINE 41108 28014 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GSK525762 MOLIBRESIB 41110 28015 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE COLCHICEINE COLCHICEINE 41111 28016 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME LY-2090314 LY-2090314 41112 28017 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 esomeprazole ESOMEPRAZOLE 41113 28018 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FENDILINE HYDROCHLORIDE FENDILINE HYDROCHLORIDE 41115 28019 NDUFS3 4722 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 41116 28020 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3545056 SAPANISERTIB 41117 28021 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ATEZOLIZUMAB ATEZOLIZUMAB 31086949 41118 28022 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DIMETHYLPINOCEMBRIN DIMETHYLPINOCEMBRIN 41120 28023 ALDH1A1 216 DRUGGABLE GENOME, ENZYME JUGLONE JUGLONE 41121 28024 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DIETHYL-2-DODECYLIDENEMALONATE CHEMBL1797708 21292492 41122 28025 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME RIVAROXABAN RIVAROXABAN 25559742 41123 28026 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FLUOROURACIL FLUOROURACIL 15330204 41125 28027 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME OMEPRAZOLE MAGNESIUM OMEPRAZOLE MAGNESIUM 41126 28028 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 4-(2-AMINOETHYL)BENZENESULFONYL FLUORIDE CHEMBL1096339 41129 28029 GDF15 9518 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR ETOPOSIDE ETOPOSIDE 10618379 41130 28030 RGS4 5999 DRUGGABLE GENOME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 41132 28031 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME GNF-PF-67 CHEMBL578512 41133 28032 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME TOSITUMOMAB TOSITUMOMAB 41134 28033 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PERIFOSINE PERIFOSINE 19706758 41136 28034 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SNX-5422 CHEMBL553939 41138 28035 LPIN1 23175 ENZYME rosiglitazone ROSIGLITAZONE 18693052 41139 28036 BAZ2B 29994 NA CARVEDILOL CARVEDILOL 41140 28037 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FENRETINIDE FENRETINIDE 41142 28038 MPI 4351 ENZYME, DRUGGABLE GENOME NSC-19803 CHEMBL522983 41143 28039 NDUFC1 4717 ENZYME inhibitor CHEMBL3545135 NV-128 41144 28040 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist 135650004 41145 28041 KDM4A 9682 DRUGGABLE GENOME, ENZYME TAMOXIFEN TAMOXIFEN 41146 28042 SRI 6717 NA COLCHICINE COLCHICINE 1975203 41150 28043 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR IONOMYCIN IONOMYCIN 12038986 41153 28044 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MIVACURIUM MIVACURIUM 41154 28045 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102918 41157 28046 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE CHEMBL201325 41158 28047 ABAT 18 DRUGGABLE GENOME, ENZYME DIVALPROEX SODIUM 41159 28048 AKAP13 11214 KINASE haloperidol HALOPERIDOL 27023437 41160 28049 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME METFORMIN METFORMIN 32444490 41161 28050 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Tricyclic benzimidazole derivative 1 41162 28051 NOTCH3 4854 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody REGN421 41163 28052 BAZ2B 29994 NA NSC-19063 CHEMBL1310138 41165 28053 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2,4,6-TRICHLOROPHENOL CHEMBL309917 41167 28054 CYP24A1 1591 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME CALCITRIOL CALCITRIOL 25148392 41168 28055 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER FENOFIBRATE FENOFIBRATE 16680159 41169 28056 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TCMDC-124059 CHEMBL530733 41173 28057 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE 404859024 41174 28058 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SJ000117911 CHEMBL589915 41175 28059 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Crizotinib CRIZOTINIB 41176 28060 GUCY2C 2984 DRUGGABLE GENOME, KINASE PLECANATIDE PLECANATIDE 41179 28061 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR RICCARDI C RICCARDI C 19103488 41180 28062 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651430 41181 28063 RGS4 5999 DRUGGABLE GENOME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 41182 28064 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 5-HYDROXYINDOLACETIC ACID CHEMBL395915 41186 28065 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE VEMURAFENIB VEMURAFENIB 24265155 41187 28066 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 374883864 41188 28067 SGSM3 27352 NA Demecolcine DEMECOLCINE 41193 28068 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL NICARDIPINE NICARDIPINE 41194 28069 HEBP1 50865 DRUGGABLE GENOME Naphthalene derivative 1 41196 28070 CAMKK2 10645 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE JNJ-7706621 JNJ-7706621 41197 28071 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GMI-1359 41199 28072 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102298 BMS-387032 41200 28073 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME activator 135650089 CHLORZOXAZONE 41201 28074 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178103717 CARPROFEN 41202 28075 PDE4B 5142 DRUGGABLE GENOME, ENZYME DG071 41205 28076 APC 324 CLINICALLY ACTIONABLE G007-LK 23539443 41206 28077 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE NINTEDANIB NINTEDANIB 18559524 41207 28078 PLD1 5337 ENZYME, DRUGGABLE GENOME AFIMOXIFENE AFIMOXIFENE 19136975 41208 28079 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 252827463 41209 28080 PSMB7 5695 DRUGGABLE GENOME, PROTEASE BORTEZOMIB BORTEZOMIB 24524217 41211 28081 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 363894212 SAVOLITINIB 41212 28082 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME METHYL ANTHRANILATE METHYL ANTHRANILATE 41213 28083 ATAD5 79915 NA MIBEFRADIL MIBEFRADIL 41215 28084 GC 2638 DRUGGABLE GENOME bevacizumab BEVACIZUMAB 29208668 41216 28085 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR AMCINONIDE AMCINONIDE 41219 28086 ENO2 2026 CELL SURFACE FLOXURIDINE FLOXURIDINE 2146046 41220 28087 MAPT 4137 DRUGGABLE GENOME GNF-PF-3582 CHEMBL606167 41221 28088 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CLORGYLINE HYDROCHLORIDE CLORGYLINE HYDROCHLORIDE 41222 28089 GLS 2744 ENZYME ELLAGIC ACID ELLAGIC ACID 41223 28090 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-22 41224 28091 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR SURAMIN HEXASODIUM SURAMIN HEXASODIUM 41226 28092 UBE2N 7334 ENZYME, DRUGGABLE GENOME IMIDOCARB DIPROPIONATE IMIDOCARB DIPROPIONATE 41227 28093 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MLN0128 SAPANISERTIB 26272063 41228 28094 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SULFACARBAMIDE SULFACARBAMIDE 41229 28095 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 doxepin DOXEPIN 41232 28096 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Abacavir ABACAVIR 41233 28097 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Selumetinib SELUMETINIB 26343583,22197931,22048237,23942066,26351322,27655129,24265152,19915144,27222538,26461489,27196754,27217440,24448821,27312529,26137449,23406027 41235 28098 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 178102291 41236 28099 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CALCIMYCIN CALCIMYCIN 41237 28100 KDM4A 9682 DRUGGABLE GENOME, ENZYME PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER 41238 28101 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME stavudine STAVUDINE 23089673 41239 28102 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR MEDRYSONE MEDRYSONE 41242 28103 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL180022 NERATINIB 41243 28104 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE OXYTETRACYCLINE OXYTETRACYCLINE 41244 28105 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 252166658 SPARSENTAN 41246 28106 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SANGUINARIUM SANGUINARIUM 41248 28107 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME VS-4718 VS-4718 41249 28108 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME VANITIOLIDE VANITIOLIDE 41250 28109 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER RESERPINE RESERPINE 41251 28110 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE DASATINIB DASATINIB 14745431,15256422,23676790,11853795,20697894,19466505,20367437,15381060,21895409,11964322,24456693,18615627,25157968,14559829,21562040,21505103,19652056,12399961 41254 28111 POLI 11201 DNA REPAIR CHALCONE CHALCONE 41255 28112 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE AG-1879 CHEMBL406845 41256 28113 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652247 41257 28114 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Binimetinib BINIMETINIB 41258 28115 NDUFS2 4720 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 41259 28116 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME RO-137410 CHEMBL275311 41260 28117 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE VITAMIN A 17988958 41261 28118 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SGI-1776 SGI-1776 41263 28119 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME inhibitor 328083484 41265 28120 PDE9A 5152 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL932 DIPYRIDAMOLE 41266 28121 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201022 PHENAZOPYRIDINE HYDROCHLORIDE 41267 28122 DNER 92737 NA PMID26924192-Compound-55 41269 28123 POLB 5423 DNA REPAIR, DRUGGABLE GENOME 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 41271 28124 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IXABEPILONE IXABEPILONE 18451235 41276 28125 PTGES 9536 DRUGGABLE GENOME, ENZYME PMID28627961-Compound-32 41277 28126 RASA1 5921 CLINICALLY ACTIONABLE TRAMETINIB TRAMETINIB 29127119 41278 28127 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 252166595 BIMIRALISIB 41280 28128 PCNA 5111 NA CAPSAICIN CAPSAICIN 9435579 41283 28129 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR MADOLIN A MADOLIN A 41284 28130 GMNN 51053 DRUGGABLE GENOME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 41286 28131 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GSK2141795 UPROSERTIB 24265152 41287 28132 HSPA4 3308 NA WORTMANNIN WORTMANNIN 16979664 41288 28133 NLRP1 22861 PROTEASE PERHEXILINE MALEATE PERHEXILINE MALEATE 41290 28134 CAST 831 PROTEASE INHIBITOR 12-O-TETRADECANOYLPHORBOL-13-ACETATE 1995645 41291 28135 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NORSTICTIC ACID NORSTICTIC ACID 41292 28136 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor 178103909 41293 28137 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RU-24969 RU-24969 41297 28138 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE Interferon alfacon-1 41298 28139 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Olmesartan medoxomil 41301 28140 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CDX-3379 26880266 41302 28141 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE NIMESULIDE NIMESULIDE 12839301 41304 28142 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AZD4547 41305 28143 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE 23814 25995436 41306 28144 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME PRAVASTATIN PRAVASTATIN 16540096 41309 28145 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIPHENOXYLATE HYDROCHLORIDE DIPHENOXYLATE HYDROCHLORIDE 41310 28146 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE CALCIUM CHANNEL BLOCKER 8381427 41311 28147 GMNN 51053 DRUGGABLE GENOME BAY-11-7085 BAY-11-7085 41312 28148 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545284 CERDULATINIB 41313 28149 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-139459 CHEMBL86464 41314 28150 SCTR 6344 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651911 VASOACTIVE INTESTINAL PEPTIDE 41315 28151 ALDH1A1 216 DRUGGABLE GENOME, ENZYME AMITRIPTYLINE HYDROCHLORIDE AMITRIPTYLINE HYDROCHLORIDE 41316 28152 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE INC280 CAPMATINIB 28783719,27694386,25971938,28765324,15494073,28396313 41318 28153 TNNT2 7139 DRUGGABLE GENOME PURPUROGALLIN PURPUROGALLIN 41320 28154 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist CHEMBL1657 TAZAROTENE 41321 28155 MGLL 11343 DRUGGABLE GENOME, ENZYME Pyrazole derivative 80 41323 28156 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE inhibitor 405560328 41324 28157 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR JUGLONE JUGLONE 41325 28158 RAB9A 9367 ENZYME, DRUGGABLE GENOME N-PHENETHYL-NICOTINAMIDE CHEMBL309848 41326 28159 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Diphenylpyraline DIPHENYLPYRALINE 41327 28160 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Nutlin-3a 21643018,25964101,21725357 41328 28161 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 328083489 CHEMBL2062804 41329 28162 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME (S)-WILLARDIINE (S)-WILLARDIINE 41330 28163 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BARDOXOLONE BARDOXOLONE 41331 28164 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MBX-2044 MBX-2044 41332 28165 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PRELADENANT PRELADENANT 41334 28166 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8759338, 12 41335 28167 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 135650338 41337 28168 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR TAMATINIB R-406 41339 28169 PSMC3 5702 NA inhibitor CHEMBL451887 CARFILZOMIB 41341 28170 AKR1B1 231 DRUGGABLE GENOME, ENZYME Terbutyline 41342 28171 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY IFN-ALPHA 2 2149997 41345 28172 PTGS2 5743 DRUGGABLE GENOME, ENZYME BROMFENAC BROMFENAC 41347 28173 DYRK4 8798 ENZYME, KINASE, DRUGGABLE GENOME, TYROSINE KINASE, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 41349 28174 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-203580 SB-203580 41350 28175 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 41352 28176 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ILORASERTIB ILORASERTIB 41355 28177 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SILIBININ SILIBININ 21273068 41357 28178 NUDT15 55270 ENZYME, CLINICALLY ACTIONABLE Thioguanine THIOGUANINE 41358 28179 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE RECOMBINANT INTERFERON ALFA-2B 41359 28180 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME CEDIRANIB CEDIRANIB 41360 28181 PDE4D 5144 DRUGGABLE GENOME, ENZYME MEM-1414 41362 28182 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TCMDC-125773 CHEMBL528451 41364 28183 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE sulfasalazine SULFASALAZINE 4386139 41365 28184 KDM1A 23028 DRUGGABLE GENOME, ENZYME, CELL SURFACE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING inhibitor 178101964 TRANYLCYPROMINE 41366 28185 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1224 ACRIVASTINE 41367 28186 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 5-FLUOROURACIL FLUOROURACIL 17179731,11501504 41368 28187 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IODOACETAMIDE IODOACETAMIDE 41369 28188 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C13 41371 28189 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME IP10.C8-1 41372 28190 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE risperidone RISPERIDONE 41374 28191 NOS1AP 9722 NA Dihydropyridine derivatives 41375 28192 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BAY-11-7082 CHEMBL403183 41376 28193 NOS2 4843 DRUGGABLE GENOME, ENZYME BANOXANTRONE BANOXANTRONE 18681417 41377 28194 HSPA4 3308 NA NDGA 8591993 41379 28195 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEXTROMEPROMAZINE DEXTROMEPROMAZINE 41382 28196 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor RETASPIMYCIN RETASPIMYCIN 41383 28197 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME L-NOREPINEPHRINE L-NOREPINEPHRINE 41384 28198 NQO2 4835 DRUGGABLE GENOME, ENZYME Melatonin MELATONIN 41385 28199 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PYRIDOSTIGMINE BROMIDE PYRIDOSTIGMINE BROMIDE 41387 28200 ALDH5A1 7915 DRUGGABLE GENOME, ENZYME T83193 41388 28201 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CEP-11981 CEP-11981 22148921 41390 28202 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-7c 41391 28203 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME modulator CHEMBL3707374 AMISELIMOD HYDROCHLORIDE 41393 28204 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PMID29671355-Compound-45a 41394 28205 ALDH1A1 216 DRUGGABLE GENOME, ENZYME O-NITROANISOLE CHEMBL166415 41397 28206 GAA 2548 DRUGGABLE GENOME, ENZYME ACARBOSE ACARBOSE 41398 28207 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GERONTOXANTHONE B GERONTOXANTHONE B 25838141 41400 28208 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME TAE-684 TAE-684 41401 28209 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-50 41403 28210 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TECNAZENE TECNAZENE 41404 28211 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME diclofenac DICLOFENAC 26398624 41405 28212 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GNF-PF-2335 CHEMBL601146 41406 28213 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME erdafitinib ERDAFITINIB 41407 28214 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALCITRIOL CALCITRIOL 41408 28215 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE BUNOLOL BUNOLOL 2903243 41409 28216 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 315661266 41410 28217 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CLOTRIMAZOLE CLOTRIMAZOLE 16680159 41413 28218 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1693 DIETHYLPROPION HYDROCHLORIDE 41415 28219 CCL11 6356 DRUGGABLE GENOME ROXITHROMYCIN ROXITHROMYCIN 11408771 41416 28220 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Imiglitazar IMIGLITAZAR 41418 28221 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 381118815 41419 28222 HTT 3064 DRUGGABLE GENOME CHLORHEXIDINE CHLORHEXIDINE 41424 28223 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER PARAROSANILINE PARAROSANILINE 41425 28224 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME CISPLATIN CISPLATIN 18667446 41426 28225 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ribavirin RIBAVIRIN 21159314 41430 28226 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME HEMATOXYLIN HEMATOXYLIN 41431 28227 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE TEMSIROLIMUS TEMSIROLIMUS 41433 28228 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROPANIL PROPANIL 41434 28229 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE RADIATION IONIZING RADIOTHERAPY 27489350 41435 28230 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000119988 CHEMBL589694 41437 28231 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 enalapril ENALAPRIL 9187528 41438 28232 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE tocilizumab TOCILIZUMAB 30457672 41439 28233 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651085 41440 28234 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-2260 CHEMBL601351 41442 28235 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 1540951 CHEMBL259421 41443 28236 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SALMETEROL SALMETEROL 41445 28237 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME PONATINIB PONATINIB 41446 28238 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FPL-64176 CHEMBL93655 41447 28239 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MENTHOFURAN MENTHOFURAN 22931300 41448 28240 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR BESTATIN METHYL ESTER BESTATIN METHYL ESTER 18448338 41449 28241 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Triazole piperazine derivative 1 41450 28242 ATXN2 6311 NA PYROGALLOL RED PYROGALLOL RED 41451 28243 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135649659 41452 28244 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Isoxazole derivative 1 41453 28245 PDE4A 5141 DRUGGABLE GENOME, ENZYME crisaborole CRISABOROLE 41454 28246 SMN1 6606 DRUGGABLE GENOME APIGENIN APIGENIN 41455 28247 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651013 41456 28248 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE LAMIVUDINE LAMIVUDINE 17172311 41457 28249 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME NSC-66209 CHEMBL175266 41458 28250 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ALISERTIB ALISERTIB 41459 28251 POR 5447 ENZYME, DRUGGABLE GENOME atorvastatin ATORVASTATIN 25521355 41460 28252 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE GW441756X GW441756X 41462 28253 UBE2N 7334 ENZYME, DRUGGABLE GENOME TCMDC-139459 CHEMBL86464 41463 28254 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135649821 41464 28255 KDM4A 9682 DRUGGABLE GENOME, ENZYME POMIFERIN POMIFERIN 41465 28256 MYLK 4638 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE activator 135652052 41466 28257 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR VP-16 ETOPOSIDE PHOSPHATE 14666661 41467 28258 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR 2,4-DIHYDROXY BENZOIC ACID HYDRAZIDE CHEMBL1339206 41468 28259 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHYSCION PHYSCION 41469 28260 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 WAY-100135 CHEMBL38288 41472 28261 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1200326 NICARDIPINE HYDROCHLORIDE 41473 28262 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METARAMINOL METARAMINOL 41476 28263 DPP8 54878 DRUGGABLE GENOME, PROTEASE, ENZYME Talabostat TALABOSTAT 41477 28264 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 187051805 QUISINOSTAT 41479 28265 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE CYC-116 CYC-116 41480 28266 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL1668 RESCINNAMINE 41482 28267 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PMID27774824-Compound-Figure6Example12 41486 28268 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-22357 CHEMBL327209 41487 28269 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SJ000029700 CHEMBL591864 41490 28270 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 9 41493 28271 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME MICHLER'S KETONE MICHLER'S KETONE 41495 28272 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL103667 DORAMAPIMOD 41496 28273 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DEXBUDESONIDE DEXBUDESONIDE 41497 28274 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103831 NAPROXCINOD 41499 28275 HTT 3064 DRUGGABLE GENOME GNF-PF-4078 CHEMBL584883 41503 28276 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TESTOSTERONE TESTOSTERONE 10809356 41504 28277 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor GSK2126458 OMIPALISIB 41506 28278 ATAD5 79915 NA (R,S)-INDATRALINE (R,S)-INDATRALINE 41508 28279 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650497 L-796449 41511 28280 MAPT 4137 DRUGGABLE GENOME NICLOSAMIDE NICLOSAMIDE 41512 28281 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Palbociclib PALBOCICLIB 27488531,22983396 41513 28282 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR EMODIN EMODIN 41515 28283 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME PF-562271 PF-00562271 41516 28284 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 15 41517 28285 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TCMDC-125606 CHEMBL536166 41518 28286 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE ANTIFOLATES 11501504 41519 28287 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ixabepilone IXABEPILONE 41520 28288 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Dihydrobenzoxazine and tetrahydroquinoxaline sulfonamide derivative 1 41521 28289 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LEE011 RIBOCICLIB 41522 28290 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE antibody MM111 41523 28291 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR KAI-9803 DELCASERTIB 41525 28292 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME L-741626 CHEMBL445102 41526 28293 TH 7054 ENZYME, DRUGGABLE GENOME FLUTAMIDE FLUTAMIDE 11223814 41527 28294 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE MANGOSTIN MANGOSTIN 41532 28295 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545369 EPACADOSTAT 41533 28296 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE NERATINIB MALEATE 41534 28297 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME SILYCHRISTIN SILICRISTIN 23401473 41537 28298 RNASEH2A 10535 ENZYME CAPSAICIN CAPSAICIN 10087087 41538 28299 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALCIPOTRIENE CALCIPOTRIENE 41539 28300 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 752709 CHEMBL429335 41540 28301 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PYM50028 41541 28302 ANGPT1 284 KINASE, DRUGGABLE GENOME, FIBRINOGEN inhibitor CHEMBL2108568 TREBANANIB 41544 28303 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME AMITRIPTYLINE AMITRIPTYLINE 41545 28304 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR ENTRECTINIB ENTRECTINIB 41546 28305 CDC42 998 DRUGGABLE GENOME ZU-4194738 CHEMBL554475 19527032 41547 28306 RGS4 5999 DRUGGABLE GENOME inhibitor 252827383 CHEMBL1604848 41548 28307 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 223365982 AC-480 41550 28308 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR CYTOKINES 12865631 41551 28309 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL2104955 BECOCALCIDIOL 41552 28310 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR E7449 2X-121 26513298 41554 28311 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LY-2090314 LY-2090314 41558 28312 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor ROMIDEPSIN ROMIDEPSIN 41560 28313 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Pyrazole derivative 61 41561 28314 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME THIRAM THIRAM 41562 28315 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-124685 CHEMBL587579 41563 28316 COL6A2 1292 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 41564 28317 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME E-DOXEPIN E-DOXEPIN 41565 28318 E2F1 1869 TRANSCRIPTION FACTOR 12-O-TETRADECANOYLPHORBOL-13-ACETATE 12947120 41566 28319 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME activator 135650028 41567 28320 MAP3K11 4296 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565853 CEP-1347 41568 28321 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200733 DESFLURANE 41569 28322 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE NAC ACETYLCYSTEINE 16713429 41570 28323 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201664 INSULIN ASPART PROTAMINE RECOMBINANT 41571 28324 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 1,2-NAPHTHOQUINONE 1,2-NAPHTHOQUINONE 41574 28325 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME T-82 41575 28326 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL150894 CEP-5214 41576 28327 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CANDESARTAN CANDESARTAN 41577 28328 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-1859 CHEMBL1520837 41578 28329 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE inhibitor 252827418 CHEMBL290376 41581 28330 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE ILORASERTIB ILORASERTIB 41582 28331 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL3545257 MIROGABALIN BESYLATE 41583 28332 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL TRICHLORMETHIAZIDE TRICHLORMETHIAZIDE 41584 28333 CP 1356 DRUGGABLE GENOME, ENZYME VINCRISTINE VINCRISTINE 9392881 41585 28334 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METARAMINOL METARAMINOL 22931300 41586 28335 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL1096380 PLINABULIN 41587 28336 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1416924 CHEMBL156959 41590 28337 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL ENFLURANE ENFLURANE 41591 28338 LSS 4047 ENZYME, DRUGGABLE GENOME inhibitor 178103325 41592 28339 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CAPECITABINE CAPECITABINE 16279094 41593 28340 HLA-DRA 3122 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE ATEZOLIZUMAB ATEZOLIZUMAB 26822383 41594 28341 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME Dihydrodiazepinocarbazolone derivative 1 41596 28342 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TCMDC-125578 CHEMBL195350 41597 28343 COMT 1312 DRUGGABLE GENOME, ENZYME clozapine CLOZAPINE 25560469 41598 28344 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL2103836 IMAGABALIN 41600 28345 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102250 41602 28346 PDE4B 5142 DRUGGABLE GENOME, ENZYME PENTOXIFYLLINE PENTOXIFYLLINE 41603 28347 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME MK-886 CHEMBL29097 41605 28348 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME ACID BLUE 129 ACID BLUE 129 41607 28349 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME KETANSERIN TARTRATE KETANSERIN TARTRATE 41609 28350 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE KAEMPFEROL KAEMPFEROL 41611 28351 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME (-)-EPICATECHIN (-)-EPICATECHIN 41612 28352 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID25656651-Compound-34b 41613 28353 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME Z-PRO-PROLINAL Z-PRO-PROLINAL 41614 28354 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ETHANOL ALCOHOL 11025487 41616 28355 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL24828 VANDETANIB 41617 28356 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME AMPICILLIN AMPICILLIN 41619 28357 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CLOSANTEL CLOSANTEL 41620 28358 RGS4 5999 DRUGGABLE GENOME antipsychotics 41621 28359 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER TCMDC-123653 CHEMBL548540 41622 28360 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Golnerminogene pradenovac 41623 28361 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE XL147 PILARALISIB 25637314 41624 28362 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545150 AZM-475271 41626 28363 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor AT9283 AT-9283 41627 28364 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE GSK-269962A GSK-269962A 41628 28365 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DAMNACANTHAL DAMNACANTHAL 41629 28366 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CC-90003 41631 28367 ACE2 59272 ENZYME, TRANSPORTER, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, CELL SURFACE, PROTEASE activator 223366197 41633 28368 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HARMOL HYDROCHLORIDE HARMOL HYDROCHLORIDE 41634 28369 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-57 41635 28370 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker 135651438 ANANDAMIDE 41636 28371 ITGB5 3693 CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL2109621 ABITUZUMAB 41637 28372 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME activator 135651446 ADENOSINE TRIPHOSPHATE 41638 28373 XDH 7498 DRUGGABLE GENOME, ENZYME LC-350189 41639 28374 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE OCV-101 41640 28375 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME BAY-11-7082 CHEMBL403183 41642 28376 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR QUINPIROLE QUINPIROLE 41643 28377 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565842 41644 28378 HMGCS2 3158 DRUGGABLE GENOME, ENZYME hydrochlorothiazide HYDROCHLOROTHIAZIDE 29523524 41646 28379 IRF1 3659 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR CYTOKINES 17947510 41647 28380 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Selumetinib SELUMETINIB 27222538 41648 28381 PICALM 8301 CLINICALLY ACTIONABLE, CELL SURFACE calcium channel blockers 24192120 41649 28382 ARID5B 84159 CLINICALLY ACTIONABLE haloperidol HALOPERIDOL 27023437 41650 28383 UGT1A6 54578 ENZYME, DRUGGABLE GENOME acetaminophen ACETAMINOPHEN 23279026,17164591,23462933,26049587,16696573,15761113,11714888 41651 28384 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Lapatinib LAPATINIB 41653 28385 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE MYCOPHENOLATE MOFETIL 12070425 41658 28386 CD163 9332 DRUGGABLE GENOME, KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE GLUCOCORTICOID 9712057 41659 28387 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME CENISERTIB CENISERTIB 41661 28388 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE KRESOXIM-METHYL KRESOXIM-METHYL 41662 28389 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 135649904 41663 28390 PDK2 5164 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME CPI-613 41664 28391 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL301742 ARBACLOFEN 41665 28392 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Imidazo[4,5-c]pyridine derivative 2 41666 28393 ABAT 18 DRUGGABLE GENOME, ENZYME TIAGABINE TIAGABINE 41667 28394 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ASP8273 NAQUOTINIB 41668 28395 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545156 KW-2450 41669 28396 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor CHEMBL3545007 RG-7602 41671 28397 PIKFYVE 200576 SERINE THREONINE KINASE, ENZYME, KINASE inhibitor 363894153 APILIMOD 41672 28398 IL1B 3553 KINASE, DRUGGABLE GENOME morphine MORPHINE 27649267 41673 28399 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Tricyclic benzimidazole derivative 1 41674 28400 CCND3 896 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BAY1000394 41676 28401 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR METHANANDAMIDE METHANANDAMIDE 41678 28402 CD9 928 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TYROSINE KINASE INHIBITOR 7592610 41679 28403 GNA11 2767 CLINICALLY ACTIONABLE SOTRASTAURIN ACETATE 24141786 41682 28404 BRCA2 675 CLINICALLY ACTIONABLE RUCAPARIB RUCAPARIB 27908594,30051098 41683 28405 CXCL8 3576 DRUGGABLE GENOME MIDAZOLAM MIDAZOLAM 9620522 41684 28406 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 41690 28407 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR NORMAL SALINE 18630696 41691 28408 COIL 8161 NA ANTI-P80 16246523 41692 28409 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CLOTIAZEPAM CLOTIAZEPAM 41693 28410 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CARBAMAZEPINE CARBAMAZEPINE 12673034 41694 28411 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Metoclopramide METOCLOPRAMIDE 41695 28412 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EMETINE EMETINE 41697 28413 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME Charybdotoxin 41698 28414 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SERTRALINE SERTRALINE 41699 28415 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE DOLASETRON DOLASETRON 11046096 41700 28416 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME EDOXABAN EDOXABAN 41701 28417 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME ADINAZOLAM ADINAZOLAM 41702 28418 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RAPAMYCIN SIROLIMUS 7982907,11698435 41703 28419 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Betaxolol BETAXOLOL 41704 28420 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER DIPYRIDAMOLE DIPYRIDAMOLE 9664131 41707 28421 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1922094 APITOLISIB 41708 28422 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Tricyclic benzimidazole derivative 1 41709 28423 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 252827413 41710 28424 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME JNJ-7706621 JNJ-7706621 41711 28425 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CEP-32496 CEP-32496 41713 28426 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651269 TOLTERODINE 41715 28427 IDO2 169355 ENZYME 2,3-diamino-benzo[b]thiophene derivative 6 41716 28428 KMO 8564 DRUGGABLE GENOME, ENZYME Pyrimidine benzenesulfonamide derivative 3 41718 28429 MAPT 4137 DRUGGABLE GENOME TRANSPLATIN TRANSPLATIN 41719 28430 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR T091317 T091317 41721 28431 MAP3K1 4214 CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME erlotinib ERLOTINIB 21636554 41722 28432 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ONAPRISTONE ONAPRISTONE 41723 28433 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME MLN-9708 IXAZOMIB CITRATE 41725 28434 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID27724045-Compound-19 41726 28435 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PRAZOSIN PRAZOSIN 41727 28436 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE interferons 17602083 41728 28437 CSNK2A2 1459 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME, TRANSCRIPTION FACTOR US8940736, 7 41729 28438 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SIROLIMUS SIROLIMUS 24934779 41731 28439 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING NEOCHAMAEJASMIN A NEOCHAMAEJASMIN A 18380477 41732 28440 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200418 DOBUTAMINE HYDROCHLORIDE 41733 28441 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME QUINELORANE QUINELORANE 41734 28442 ATXN2 6311 NA MENADIONE MENADIONE 41736 28443 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 41738 28444 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE epinephrine EPINEPHRINE 41740 28445 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135650568 41741 28446 GMNN 51053 DRUGGABLE GENOME N-(4-HYDROXYPHENYL)RHODANINE CHEMBL462430 41743 28447 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-23 41744 28448 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME DNDI1417467 CHEMBL1997335 41746 28449 HTT 3064 DRUGGABLE GENOME DNDI1417623 CHEMBL2002849 41747 28450 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE DASATINIB DASATINIB 41748 28451 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178103093 41749 28452 MSR1 4481 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME H2O2 15316030 41751 28453 PDE4B 5142 DRUGGABLE GENOME, ENZYME AVE-8112 24343458 41752 28454 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GT 389-255 41753 28455 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BI2536 26597303 41754 28456 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME ITOPRIDE ITOPRIDE 41755 28457 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL2103830 FOSTAMATINIB 41756 28458 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE inhibitor 178103356 ABIRATERONE 41757 28459 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX PYRITHIONE PYRITHIONE 41758 28460 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 178102512 EVEROLIMUS 41759 28461 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL2017974 BUPARLISIB 41760 28462 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Organon-3 41762 28463 LMNA 4000 CLINICALLY ACTIONABLE, DRUGGABLE GENOME SU-4312 CHEMBL328710 41763 28464 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Celecoxib CELECOXIB 41764 28465 CDS1 1040 KINASE, ENZYME inhibitor CHEMBL3544911 PREXASERTIB 41765 28466 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MACROLIDES 12814973 41766 28467 SMN2 6607 DRUGGABLE GENOME MYCOPHENOLIC ACID MYCOPHENOLIC ACID 41767 28468 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Temozolomide TEMOZOLOMIDE 25910950 41768 28469 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CLIOQUINOL CLIOQUINOL 41770 28470 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DASATINIB DASATINIB 27231123 41773 28471 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME NSC-228155 CHEMBL505670 41775 28472 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL452231 TENIPOSIDE 41776 28473 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME atorvastatin ATORVASTATIN 41778 28474 TMEM97 27346 NA Bicyclo-heptan-2-amine derivative 4 41780 28475 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE irinotecan IRINOTECAN 18981587,18221820 41782 28476 RACGAP1 29127 NA NSC-19063 CHEMBL1310138 41788 28477 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 310264726 41789 28478 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32h 41791 28479 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649802 4-METHYLHISTAMINE 41792 28480 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME TRIMETHOPRIM TRIMETHOPRIM 15606443 41793 28481 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BROMOCRIPTINE BROMOCRIPTINE 18455424 41795 28482 PSMA1 5682 PROTEASE, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 24524217 41796 28483 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME NERVE GROWTH FACTOR 2887561 41797 28484 MAPT 4137 DRUGGABLE GENOME 3-MORPHOLINOSYDNONIMINE HCL CHEMBL538104 41800 28485 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-123650 CHEMBL580727 41801 28486 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PMID28766366-Compound-Scheme21Left 41805 28487 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE VINBURNINE VINBURNINE 41806 28488 KLK4 9622 PROTEASE, DRUGGABLE GENOME, ENZYME Benzoxazinone derivative 2 41807 28489 IGHG1 3500 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE IGG1 ANTIBODY 41809 28490 CBX1 10951 NA R(-)-PROPYLNORAPOMORPHINE HCL CHEMBL538542 41812 28491 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME AG-1879 CHEMBL406845 41813 28492 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CHEMBL591 ETHCHLORVYNOL 41814 28493 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102559 NINTEDANIB 41815 28494 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TANSHINONE IIA TANSHINONE IIA 41816 28495 TOP2B 7155 DRUGGABLE GENOME, ENZYME MTC-DOX 41820 28496 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Formoterol FORMOTEROL 41821 28497 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME cyclosporine CYCLOSPORINE 18021981 41822 28498 PDE5A 8654 ENZYME, DRUGGABLE GENOME LORNEIC ACID A LORNEIC ACID A 19856955 41824 28499 GMNN 51053 DRUGGABLE GENOME PALMITOYL-DL-CARNITINE CHLORIDE CHEMBL1256761 41825 28500 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3261331 RESMETIROM 41826 28501 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Dasatinib DASATINIB 26855149 41827 28502 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor VORINOSTAT VORINOSTAT 41828 28503 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178103511 TIDEGLUSIB 41830 28504 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE SIFALIMUMAB SIFALIMUMAB 41831 28505 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER hydrocortisone HYDROCORTISONE 41832 28506 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 10 41833 28507 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME (-)-HERDMANINE K CHEMBL2208195 23189988 41835 28508 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR FONDAPARINUX FONDAPARINUX 41836 28509 PTPRD 5789 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CIXUTUMUMAB CIXUTUMUMAB 23800680 41837 28510 BMPR1B 658 DRUGGABLE GENOME, CELL SURFACE, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 249565824 41838 28511 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 187051821 OLAPARIB 41839 28512 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME antibody 249565932 41840 28513 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 53801030 DIARYLPROPIONITRILE 41842 28514 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME PAC1 41844 28515 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DAPIPRAZOLE DAPIPRAZOLE 41845 28516 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE MP0112 ABICIPAR PEGOL 41847 28517 TRIB2 28951 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME allopurinol ALLOPURINOL 30924126 41848 28518 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor DABRAFENIB DABRAFENIB 41849 28519 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL EVT-201 41850 28520 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME L-694247 L-694247 41851 28521 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 41852 28522 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LEVISOPRENALINE LEVISOPRENALINE 41854 28523 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ARTEMISIN ARTEMISIN 41855 28524 BUB1 699 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565790 41856 28525 POLK 51426 DNA REPAIR, ENZYME 3,5-DINITROCATECHOL (OR-486) 3,5-DINITROCATECHOL (OR-486) 41857 28526 TXNRD2 10587 DRUGGABLE GENOME methadone METHADONE 32407152 41858 28527 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1969 CHEMBL601364 41859 28528 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PU3 41861 28529 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE VANDETANIB VANDETANIB 41866 28530 ALOX15 246 ENZYME, DRUGGABLE GENOME U-0126 U-0126 41869 28531 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE CENISERTIB CENISERTIB 41870 28532 SMN2 6607 DRUGGABLE GENOME LUTEOLIN LUTEOLIN 41872 28533 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME FAS LIGAND 12749243 41876 28534 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIFLUNISAL DIFLUNISAL 41877 28535 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1416924 CHEMBL156959 41878 28536 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR STREPTONIGRIN STREPTONIGRIN 41879 28537 DDX43 55510 DRUG RESISTANCE TRAMETINIB TRAMETINIB 24899684 41880 28538 BRD9 65980 ENZYME inhibitor 336446908 41881 28539 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME CSL-112 41882 28540 ATAD5 79915 NA TCMDC-124585 CHEMBL587856 41883 28541 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 354702232 41887 28542 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650391 INDORAMIN 41889 28543 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 384403651 41892 28544 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178101025 41893 28545 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 252166784 41894 28546 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1254771 SAFOTIBANT 41895 28547 RAB9A 9367 ENZYME, DRUGGABLE GENOME TCMDC-123480 CHEMBL588683 41897 28548 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LEVOTHYROXINE LEVOTHYROXINE 41898 28549 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ALBUMIN ALBUMIN HUMAN 8788167 41899 28550 GJA1 2697 ION CHANNEL Act1 41901 28551 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1172 DESLORATADINE 41902 28552 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GP-120 15954144 41903 28553 MAPT 4137 DRUGGABLE GENOME NSC-107022 CHEMBL1601846 41904 28554 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 310264698 AMG-319 41905 28555 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NANDROLONE NANDROLONE 41908 28556 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME KLH 11768621 41909 28557 ABCB4 5244 TRANSPORTER, DRUGGABLE GENOME, ENZYME, ABC TRANSPORTER VINCRISTINE VINCRISTINE 1673638 41910 28558 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PHENYTOIN PHENYTOIN 12673034 41911 28559 BAZ2B 29994 NA GNF-PF-2893 CHEMBL312032 41912 28560 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-21 41913 28561 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20120264760C86 41914 28562 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SMT-D002 41915 28563 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 354702286 41916 28564 ATXN2 6311 NA GNF-PF-2853 CHEMBL576362 41918 28565 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33f 41919 28566 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1919 CHEMBL576409 41920 28567 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL2106615 BAZEDOXIFENE ACETATE 41922 28568 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW703087X GW703087X 41923 28569 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL2109177 ODULIMOMAB 41924 28570 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3544913 VIXOTRIGINE 41925 28571 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY FDG FLUDEOXYGLUCOSE-F18 8491223 41926 28572 HMGCR 3156 ENZYME, DRUGGABLE GENOME Simvastatin SIMVASTATIN 41927 28573 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Filgrastim FILGRASTIM 41928 28574 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor BKM120 BUPARLISIB 41929 28575 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER vitamin e 41930 28576 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ATENOLOL ATENOLOL 15453913 41931 28577 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 374883869 41932 28578 ABL2 27 KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME DASATINIB DASATINIB 25207766 41933 28579 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENZODODECINIUM CHLORIDE BENZODODECINIUM CHLORIDE 41934 28580 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Beta Blocking Agents 18855529 41935 28581 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE R1295 41936 28582 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER GLEEVEC IMATINIB 15155841 41938 28583 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDEIV-23C1 CHEMBL1094358 20371180 41939 28584 APC 324 CLINICALLY ACTIONABLE Celecoxib CELECOXIB 17909047 41942 28585 ALOX15 246 ENZYME, DRUGGABLE GENOME CADMIUM DICHLORIDE CADMIUM DICHLORIDE 41944 28586 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME TRAMETINIB TRAMETINIB 25452114 41945 28587 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652332 41946 28588 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME R115777 16818651 41948 28589 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME ROSIGLITAZONE ROSIGLITAZONE 18314419 41949 28590 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 178101509 DIPYRIDAMOLE 41952 28591 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GNF-PF-5233 CHEMBL528316 41954 28592 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor GDC-0941 PICTILISIB 41957 28593 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor VENETOCLAX VENETOCLAX 41959 28594 GJB6 10804 ION CHANNEL inhibitor 178100972 CARBENOXOLONE 41960 28595 HTT 3064 DRUGGABLE GENOME HELENALIN HELENALIN 41962 28596 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE MAFOSFAMIDE MAFOSFAMIDE 1515095 41964 28597 SLC2A3 6515 DRUGGABLE GENOME, TRANSPORTER CYTOKINES 15727913 41965 28598 TUBB3 10381 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 41966 28599 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000114961 CHEMBL590168 41967 28600 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CALYCOSIN CALYCOSIN 41968 28601 APOE 348 DRUGGABLE GENOME INTRALIPID SOYBEAN OIL 3021887 41970 28602 GMNN 51053 DRUGGABLE GENOME PERMETHRIN PERMETHRIN 41971 28603 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1416985 CHEMBL593211 41972 28604 STK10 6793 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178102336 BOSUTINIB 41973 28605 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BIFENAZATE BIFENAZATE 41974 28606 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ASPIRIN ASPIRIN 22931300 41975 28607 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651067 41979 28608 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1021 NEPAFENAC 41980 28609 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme15-2 41981 28610 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE avelumab AVELUMAB 41982 28611 APC 324 CLINICALLY ACTIONABLE Dasatinib DASATINIB 20473900 41984 28612 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 135649822 41987 28613 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Pemirolast PEMIROLAST 41988 28614 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME COBALT 11891799 41989 28615 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Ganetespib GANETESPIB 25077897 41991 28616 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 41992 28617 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PHOSMET PHOSMET 41993 28618 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE NIVOLUMAB NIVOLUMAB 30742119 41994 28619 TUBB3 10381 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 41995 28620 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME ASP-015K PEFICITINIB 41998 28621 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PAROXETINE HYDROCHLORIDE PAROXETINE HYDROCHLORIDE 42000 28622 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Ruxolitinib derivative 2 42001 28623 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME NSC-77833 CHEMBL1287981 42002 28624 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Carboplatin CARBOPLATIN 25567130,25658463,26494859,27998224 42004 28625 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 135652743 42005 28626 SLC2A5 6518 TRANSPORTER, DRUGGABLE GENOME STREPTOZOTOCIN STREPTOZOCIN 9756334 42007 28627 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME DTIC DACARBAZINE 12168066 42008 28628 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200406 DIMENHYDRINATE 42009 28629 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME PF-562271 PF-00562271 42010 28630 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEXAMETHASONE DEXAMETHASONE 42011 28631 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME IL-2 ALDESLEUKIN 7528775 42012 28632 SLC28A2 9153 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME peginterferon alfa-2b 26071337 42014 28633 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor AT101 42016 28634 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 328083526 CITARINOSTAT 42017 28635 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NSC-228155 CHEMBL505670 42020 28636 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SDZ-205557 CHEMBL287045 42021 28637 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Ivosidenib IVOSIDENIB 42022 28638 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-95909 CHEMBL1547715 42023 28639 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BENZBROMARONE BENZBROMARONE 42024 28640 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SAPPANONE A DIMETHYL ETHER SAPPANONE A DIMETHYL ETHER 42025 28641 MPI 4351 ENZYME, DRUGGABLE GENOME TCMDC-125319 CHEMBL527586 42026 28642 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME BM-ca 42027 28643 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Selumetinib SELUMETINIB 42028 28644 NUAK2 81788 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565727 42030 28645 VKORC1 79001 DRUGGABLE GENOME, ENZYME DICUMAROL DICUMAROL 42031 28646 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-4012 CHEMBL584269 42033 28647 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME RADIOSENSITIZERS 12033498 42036 28648 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor RUCAPARIB RUCAPARIB 42037 28649 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 385612233 42038 28650 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BUTANE-2,3-DIONE MONOOXIME CHEMBL335741 42039 28651 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HYDRASTININE HYDROCHLORIDE HYDRASTININE HYDROCHLORIDE 42041 28652 ATP1B1 481 DRUGGABLE GENOME, TRANSPORTER, ENZYME inhibitor CHEMBL1751 DIGOXIN 42042 28653 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 1 42043 28654 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Bicyclic heteroaryl benzamide derivative 6 42044 28655 SH2B1 25970 KINASE amisulpride AMISULPRIDE 28694205 42046 28656 ATXN2 6311 NA PROCHLORPERAZINE PROCHLORPERAZINE 42047 28657 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650709 NETOGLITAZONE 42050 28658 SULT1A1 6817 DRUGGABLE GENOME, ENZYME desmethylnaproxen 42051 28659 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 42052 28660 EIF2B1 1967 NA HORMONES 7893823 42054 28661 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 348353650 42056 28662 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME blocker 135652740 42057 28663 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DICHLOFLUANID DICHLOFLUANID 42058 28664 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL3544997 LS-104 42059 28665 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-34b 42060 28666 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649955 42061 28667 IDE 3416 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, ENZYME, PROTEASE Bacitracin BACITRACIN 42062 28668 ESRRG 2104 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135649858 DAIDZEIN 42063 28669 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEFOTIAM HYDROCHLORIDE CEFOTIAM HYDROCHLORIDE 42066 28670 E2F1 1869 TRANSCRIPTION FACTOR IRINOTECAN IRINOTECAN 9766655 42067 28671 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PARICALCITOL PARICALCITOL 42069 28672 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER 1614235 + 2330672 42070 28673 RUNX3 864 TRANSCRIPTION FACTOR IRINOTECAN IRINOTECAN 17372756 42072 28674 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 4 42073 28675 PRMT3 10196 DRUGGABLE GENOME, METHYL TRANSFERASE, ENZYME allosteric modulator 252166753 42075 28676 POLK 51426 DNA REPAIR, ENZYME ACID BLUE 129 ACID BLUE 129 42078 28677 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME CAPTOPRIL CAPTOPRIL 17531305 42079 28678 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 178103494 IBRUTINIB 42080 28679 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SB-224289 SB-224289 42082 28680 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565693 42083 28681 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL514800 APREMILAST 42084 28682 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BOSENTAN BOSENTAN 42086 28683 TARDBP 23435 TUMOR SUPPRESSOR SJ000112730 CHEMBL591178 42087 28684 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME antagonist 223366065 CHEMBL504559 42088 28685 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL107 COLCHICINE 42089 28686 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME GABOXADOL GABOXADOL 42090 28687 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE DASATINIB DASATINIB 42091 28688 POLK 51426 DNA REPAIR, ENZYME HOMIDIUM BROMIDE HOMIDIUM BROMIDE 42093 28689 MIF 4282 DRUGGABLE GENOME, CELL SURFACE TCMDC-124484 CHEMBL524449 21719283 42094 28690 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TRIMETREXATE TRIMETREXATE 42096 28691 ATXN2 6311 NA N-DESMETHYLCLOZAPINE N-DESMETHYLCLOZAPINE 42097 28692 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR THEONELLASTEROL G THEONELLASTEROL G 21428459 42100 28693 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3544968 GSK-610677 42101 28694 PTPN12 5782 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, KINASE CRIZOTINIB CRIZOTINIB 29578538 42102 28695 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 381118865 42105 28696 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Amidine oxime derivative 1 42106 28697 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR CYCLOOXYGENASE INHIBITOR 12814375 42107 28698 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME BFGF 15310753 42108 28699 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME SPERMINE BIS-2-NAPG CHEMBL2347631 23434419 42109 28700 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR GEMCITABINE GEMCITABINE 17245119 42112 28701 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE warfarin WARFARIN 27740732 42113 28702 MSH6 2956 CLINICALLY ACTIONABLE, DNA REPAIR DURVALUMAB DURVALUMAB 26674132 42116 28703 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL2103836 IMAGABALIN 42117 28704 EPAS1 2034 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX PUUPEHENONE PUUPEHENONE 22928967 42119 28705 TUBB3 10381 DRUGGABLE GENOME CHEMBL2105643 FOSBRETABULIN TROMETHAMINE 42120 28706 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545366 VOXTALISIB 42123 28707 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL1980297 ILORASERTIB 42124 28708 TARDBP 23435 TUMOR SUPPRESSOR WIN-55212-2 WIN-552122 42125 28709 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME MESTRANOL MESTRANOL 6744303 42127 28710 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor DASATINIB DASATINIB 42128 28711 CALM1 801 ION CHANNEL, KINASE, ENZYME, DRUGGABLE GENOME APRINDINE APRINDINE 42129 28712 TAT 6898 ENZYME VITAMIN A 8100575 42130 28713 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Oxcarbazepine OXCARBAZEPINE 42132 28714 PSMA4 5685 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL2103884 OPROZOMIB 42133 28715 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 135651418 ALITRETINOIN 42136 28716 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME RESMINOSTAT RESMINOSTAT 42137 28717 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE GGF-2 42138 28718 ALOX15 246 ENZYME, DRUGGABLE GENOME PTAEROXYLIN PTAEROXYLIN 42139 28719 GSTM3 2947 ENZYME, DRUGGABLE GENOME olanzapine OLANZAPINE 23559402 42140 28720 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Donitriptan DONITRIPTAN 42141 28721 EYA2 2139 DNA REPAIR CRYSTAL VIOLET HEXAMETHYL PARAROSANILINE 42142 28722 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GNF-PF-265 CHEMBL602418 42143 28723 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME ST 638 2144851 42144 28724 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Methdilazine METHDILAZINE 42145 28725 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 9-AMINOCAMPTOTHECIN 9-AMINOCAMPTOTHECIN 42147 28726 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME IDRAPARINUX IDRAPARINUX 42149 28727 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL408513 BELINOSTAT 42152 28728 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHLORPHRIFOS OXON CHLORPHRIFOS OXON 42153 28729 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE IRINOTECAN IRINOTECAN 16456808 42154 28730 ATAD2B 54454 ENZYME inhibitor 336446907 42155 28731 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antagonist CHEMBL2107861 ZALUTUMUMAB 42156 28732 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR nifedipine NIFEDIPINE 19444285 42157 28733 POLK 51426 DNA REPAIR, ENZYME SURAMIN SURAMIN 42160 28734 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 178103587 MOCETINOSTAT 42161 28735 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE OLTIPRAZ OLTIPRAZ 20655236 42162 28736 PTGES 9536 DRUGGABLE GENOME, ENZYME INDOMETHACIN INDOMETHACIN 19053751 42163 28737 NR2F2 7026 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GNF-PF-1678 CHEMBL580340 42165 28738 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE JNK-401 42166 28739 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TRIFLUOPERAZINE TRIFLUOPERAZINE 42169 28740 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1417941 CHEMBL2095095 42170 28741 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 178101454 SILDENAFIL 42171 28742 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL103 PROGESTERONE 42172 28743 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME inhibitor 178103947 42173 28744 BCHE 590 DRUGGABLE GENOME, ENZYME Egonol compound 1 42175 28745 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HALCINONIDE HALCINONIDE 42177 28746 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DOXYCYCLINE DOXYCYCLINE 16643899 42178 28747 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GW7074 CHEMBL72365 42180 28748 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CAPECITABINE CAPECITABINE 26920887 42181 28749 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PEN-866 PEN-866 42183 28750 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CISPLATIN CISPLATIN 9600935,11812076,8678559 42184 28751 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CYTOKINES 15728714 42185 28752 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE raltitrexed RALTITREXED 17203168,15353299,16456808 42186 28753 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL686 MEFENAMIC ACID 42189 28754 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUMETHASONE FLUMETHASONE 42191 28755 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MENADIONE MENADIONE 42193 28756 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PMID28766366-Compound-Scheme21Right 42194 28757 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-14 42195 28758 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Dasatinib DASATINIB 26483207 42197 28759 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME OXOPURPUREINE OXOPURPUREINE 42199 28760 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE nicotine NICOTINE 22260295,15007373,17224915,23223006,11840318,16387451,31246565,16960700 42202 28761 BAZ2B 29994 NA TCMDC-123828 CHEMBL588804 42203 28762 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE 178101617 42205 28763 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PF-06410293 42206 28764 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE AMG102 42207 28765 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL856 PRIMIDONE 42208 28766 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR CINNAMIC ACID HYDROXAMATE CINNAMIC ACID HYDROXAMATE 24074025 42211 28767 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR IRBESARTAN IRBESARTAN 42212 28768 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR CILOSTAZOL CILOSTAZOL 15744080 42214 28769 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SB-269970 CHEMBL282199 42215 28770 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NSC-98938 CHEMBL1939691 42216 28771 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR FORASARTAN FORASARTAN 42220 28772 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL2103852 CROLIBULIN 42221 28773 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Citatuzumab bogatox 42223 28774 LIG1 3978 DNA REPAIR, DRUGGABLE GENOME BLEOMYCIN BLEOMYCIN 42224 28775 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE 42226 28776 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Aromatic bicyclic compound 5 42227 28777 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR F-8-IL-10 fusion protein 42229 28778 P4HA1 5033 DRUGGABLE GENOME, ENZYME SAFIRONIL SAFIRONIL 42230 28779 KDM4A 9682 DRUGGABLE GENOME, ENZYME CARBETAPENTANE CITRATE CARBETAPENTANE CITRATE 42232 28780 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL1200645 ETOPOSIDE PHOSPHATE 42234 28781 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650172 DEXETIMIDE 42235 28782 RACGAP1 29127 NA 7-HYDROXYCHLORPROMAZINE 7-HYDROXYCHLORPROMAZINE 42236 28783 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor GDC-0973 COBIMETINIB 42237 28784 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE TEPLIZUMAB TEPLIZUMAB 42238 28785 FAAH 2166 ENZYME, DRUGGABLE GENOME OL-92 CHEMBL367966 23287055 42239 28786 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE SORAFENIB SORAFENIB 42240 28787 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MLN-8054 MLN-8054 42241 28788 ACTB 60 TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE ENVIRONMENTAL ESTROGEN 17288598 42242 28789 ATAD5 79915 NA RAC-GONIOTHALAMIN CHEMBL1170485 42243 28790 CXCL8 3576 DRUGGABLE GENOME IONOMYCIN IONOMYCIN 7510691 42244 28791 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE FLUPIRTINE FLUPIRTINE 42245 28792 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GRISEOFULVIN GRISEOFULVIN 42246 28793 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE MR1-1 42248 28794 RAPGEF3 10411 ENZYME PENTABROMOPHENOL PENTABROMOPHENOL 42249 28795 KDM4A 9682 DRUGGABLE GENOME, ENZYME PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE CHEMBL114544 42250 28796 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL3545285 XL-999 42251 28797 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR lisinopril LISINOPRIL 42252 28798 GMNN 51053 DRUGGABLE GENOME DNDI1416975 CHEMBL1415851 42253 28799 SMN1 6606 DRUGGABLE GENOME GNF-PF-2812 CHEMBL125044 42254 28800 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-20 42257 28801 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652338 42258 28802 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor VORINOSTAT VORINOSTAT 42259 28803 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL XEN-402 FUNAPIDE 42260 28804 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL2107842 ALBINTERFERON ALFA-2B 42261 28805 SMN1 6606 DRUGGABLE GENOME NICLOSAMIDE NICLOSAMIDE 42262 28806 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-51 42263 28807 UGT1A6 54578 ENZYME, DRUGGABLE GENOME aspirin ASPIRIN 42264 28808 HTT 3064 DRUGGABLE GENOME THIRAM THIRAM 42265 28809 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIMETHISOQUIN DIMETHISOQUIN 42266 28810 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ANDROSTENEDIONE ANDROSTENEDIONE 9260906 42268 28811 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEFAZOLIN CEFAZOLIN 42270 28812 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE PF-04950615 BOCOCIZUMAB 42271 28813 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GR-89696 CHEMBL603370 42272 28814 PARP3 10039 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR inhibitor CHEMBL3833368 RUCAPARIB CAMSYLATE 42275 28815 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Nicotinamide NIACINAMIDE 42276 28816 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR GONADOTROPINS 12969721 42277 28817 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME SurVaxM 42278 28818 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MMV665817 CHEMBL590919 42281 28819 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHLOROQUINE CHLOROQUINE 22931300 42283 28820 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER METHAMPHETAMINE METHAMPHETAMINE 42284 28821 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE IC261 IC261 20350806 42285 28822 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 252166527 PEFICITINIB 42286 28823 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 10-HYDROXYEVODIAMINE CHEMBL2171812 22867019 42288 28824 KMO 8564 DRUGGABLE GENOME, ENZYME Cyclopropane 1-carboxylic acid derivative 9 42289 28825 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME ETOMIDATE ETOMIDATE 16884293 42290 28826 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Sapanisertib SAPANISERTIB 25261369 42291 28827 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME irinotecan IRINOTECAN 24018773,18221820 42292 28828 POLI 11201 DNA REPAIR PYRONIN Y PYRONIN Y 42293 28829 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 223366084 TANESPIMYCIN 42294 28830 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME TAMATINIB R-406 42295 28831 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 178101517 METHOTREXATE 42296 28832 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2178577 AZD-5363 42298 28833 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-37642 CHEMBL1707907 42300 28834 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE SB-216763 SB-216763 42303 28835 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME Tetra-cyclic compound 1 42305 28836 BCL2L2 599 CLINICALLY ACTIONABLE, DRUGGABLE GENOME 2-CDA CLADRIBINE 15813915 42306 28837 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR NSC-632536 CHEMBL1367933 42308 28838 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME RECOMBINANT THROMBOMODULIN 42311 28839 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antagonist CHEMBL2109402 MM-121 42312 28840 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER GNF-PF-2671 CHEMBL578878 42313 28841 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROPIOMAZINE PROPIOMAZINE 42314 28842 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRETINOIN TRETINOIN 42316 28843 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Paclitaxel PACLITAXEL 42317 28844 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE EBSELEN EBSELEN 42318 28845 PDE4D 5144 DRUGGABLE GENOME, ENZYME AWD-12-281 42319 28846 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER lovastatin LOVASTATIN 42320 28847 PDE10A 10846 ENZYME, DRUGGABLE GENOME FRM-6308 42321 28848 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200864 42322 28849 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME TAMATINIB R-406 42324 28850 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Anti-CD123 CAR-T treatment 42326 28851 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE CHRYSIN CHRYSIN 42328 28852 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME HALOPERIDOL HALOPERIDOL 42329 28853 TUBB 203068 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 42330 28854 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Dabrafenib DABRAFENIB 27312529 42331 28855 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-3149 CHEMBL582507 42332 28856 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME THUNBERGINOL B THUNBERGINOL B 42333 28857 ITPKC 80271 ENZYME, KINASE inhibitor 336446934 42334 28858 MAPT 4137 DRUGGABLE GENOME (-)-ESEROLINE CHEMBL310934 42336 28859 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME TRANSFORMING GROWTH FACTOR 15138629 42337 28860 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 42339 28861 FST 10468 DRUGGABLE GENOME HEREGULIN 15609326 42341 28862 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME SB-206553 CHEMBL297784 42345 28863 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE SAR228810 42348 28864 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3-HYDROXYFLAVONOL CHEMBL242172 42351 28865 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-31 42353 28866 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BCMA CAR-T Cells 42354 28867 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor CHEMBL52885 ENMD-981693 42355 28868 KDM4A 9682 DRUGGABLE GENOME, ENZYME RABEPRAZOLE SODIUM RABEPRAZOLE SODIUM 42356 28869 ALDH1A2 8854 DRUGGABLE GENOME, ENZYME VITAMIN A 9666306,11133156 42357 28870 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PD-169316 PD-169316 42358 28871 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor PF-4691502 PF-04691502 42360 28872 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 252166613 RETOSIBAN 42361 28873 CXCL8 3576 DRUGGABLE GENOME ASPIRIN ASPIRIN 12576442 42362 28874 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME OESTRADIOL ESTRADIOL 10508216 42364 28875 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME APOMORPHINE APOMORPHINE 42365 28876 FBXW7 55294 DNA REPAIR, CLINICALLY ACTIONABLE Regorafenib REGORAFENIB 27399335 42366 28877 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ESTRADIOL ESTRADIOL 42368 28878 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TOLONIUM CHLORIDE TOLONIUM CHLORIDE 42369 28879 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Bevacizumab + Rituximab 42373 28880 CDH1 999 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Selumetinib SELUMETINIB 26251290 42377 28881 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DIENOGEST DIENOGEST 42378 28882 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Ribociclib RIBOCICLIB 42379 28883 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR URACIL MUSTARD URACIL MUSTARD 42382 28884 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1201023 ORPHENADRINE HYDROCHLORIDE 42383 28885 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 223366047 AZD-8055 42384 28886 XRCC5 7520 KINASE thalidomide THALIDOMIDE 21435719 42385 28887 SLC12A2 6558 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178101453 PIRETANIDE 42387 28888 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 178103405 CAPECITABINE 42388 28889 TOP1MT 116447 DRUGGABLE GENOME, ENZYME PEG-SN38 42389 28890 RGS4 5999 DRUGGABLE GENOME MRS-1220 CHEMBL88147 42391 28891 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME FAGARONINE FAGARONINE 42392 28892 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2,4-DIMETHYLPHENOL CHEMBL29878 42394 28893 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PLUMBAGIN PLUMBAGIN 24355130 42395 28894 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist 223366049 42396 28895 ALDH1L1 10840 DRUGGABLE GENOME methylphenidate METHYLPHENIDATE 42397 28896 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE CHZ868 29434033 42398 28897 MAPT 4137 DRUGGABLE GENOME OXOPURPUREINE OXOPURPUREINE 42399 28898 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 252827453 42400 28899 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PD-173074 PD-173074 42401 28900 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ELLAGIC ACID ELLAGIC ACID 42402 28901 ECE1 1889 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE inhibitor 252166818 42403 28902 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PALBOCICLIB PALBOCICLIB 25524798 42404 28903 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE DEPSIPEPTIDE ROMIDEPSIN 15059137 42406 28904 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BYL719 ALPELISIB 42408 28905 BAZ2B 29994 NA METHACYCLINE HYDROCHLORIDE METHACYCLINE HYDROCHLORIDE 42410 28906 CPB2 1361 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166857 42411 28907 ATXN2 6311 NA NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 42412 28908 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CURCUMIN CURCUMIN 19112019 42413 28909 CBX1 10951 NA FENRETINIDE FENRETINIDE 42414 28910 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME inhibitor 354702236 42415 28911 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PI-103 PI-103 22336586 42416 28912 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NOREPINEPHRINE NOREPINEPHRINE 42417 28913 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE OLEOYL DOPAMINE OLEOYL DOPAMINE 42418 28914 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR CENISERTIB CENISERTIB 42420 28915 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MAKALUVAMINE A MAKALUVAMINE A 8691207 42424 28916 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME ENU 1727384 42425 28917 MAPT 4137 DRUGGABLE GENOME DNDI1417722 CHEMBL1503190 42427 28918 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-130813 CHEMBL463783 42428 28919 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-3148 CHEMBL81782 42429 28920 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PAPAVERINE PAPAVERINE 42430 28921 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL VERAPAMIL VERAPAMIL 42433 28922 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE ISOBONDUCELLIN ISOBONDUCELLIN 20813535 42434 28923 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PANOBINOSTAT PANOBINOSTAT 42435 28924 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE GOLIMUMAB GOLIMUMAB 42436 28925 CBX1 10951 NA OXYTETRACYCLINE OXYTETRACYCLINE 42437 28926 ALOX15 246 ENZYME, DRUGGABLE GENOME GNF-PF-3464 CHEMBL602213 42438 28927 ALOX15 246 ENZYME, DRUGGABLE GENOME SJ000044511 CHEMBL592124 42439 28928 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CANCER VACCINES 16619291 42442 28929 VKORC1 79001 DRUGGABLE GENOME, ENZYME WARFARIN WARFARIN 42443 28930 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BEPOTASTINE BEPOTASTINE 42444 28931 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NICLOSAMIDE NICLOSAMIDE 42445 28932 HSPB1 3315 DRUGGABLE GENOME FEPRAZONE FEPRAZONE 42448 28933 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200492 NEFAZODONE HYDROCHLORIDE 42449 28934 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 363894223 42453 28935 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME ATENOLOL ATENOLOL 16995309 42454 28936 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PROPRANOLOL PROPRANOLOL 15023456 42455 28937 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MUNDULONE MUNDULONE 42456 28938 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ALLOPREGNANOLONE BREXANOLONE 42457 28939 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PF-06747143 PF-06747143 42458 28940 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201020 DISOPYRAMIDE PHOSPHATE 42459 28941 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE CEDIRANIB CEDIRANIB 42461 28942 PDE4B 5142 DRUGGABLE GENOME, ENZYME TA-7906 42462 28943 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 135650760 ONAPRISTONE 42464 28944 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE DACTOLISIB DACTOLISIB 42466 28945 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THYMOL IODIDE THYMOL IODIDE 42468 28946 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Tolbutamide TOLBUTAMIDE 42469 28947 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRIAZOPHOS TRIAZOPHOS 42470 28948 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CENISERTIB CENISERTIB 42471 28949 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Ponatinib PONATINIB 42473 28950 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor GDC-0973 COBIMETINIB 42474 28951 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 17-AAG TANESPIMYCIN 16203796 42475 28952 BAZ2B 29994 NA DNDI1417076 CHEMBL1526167 42477 28953 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1201584 ABCIXIMAB 42478 28954 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PMID27336223-Compound-10 42479 28955 MYD88 4615 CLINICALLY ACTIONABLE Vorinostat VORINOSTAT 27733371 42481 28956 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417697 CHEMBL1420457 42484 28957 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW589933X GW589933X 42486 28958 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DOXORUBICIN DOXORUBICIN 1830717 42487 28959 TH 7054 ENZYME, DRUGGABLE GENOME inhibitor 178103538 METYROSINE 42491 28960 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545419 TELISOTUZUMAB 42494 28961 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE inhibitor 381745000 OLUTASIDENIB 42495 28962 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103589 RICOLINOSTAT 42497 28963 NAMPT 10135 DRUGGABLE GENOME Daporinad DAPORINAD 42498 28964 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR fulvestrant FULVESTRANT 42500 28965 PDE4A 5141 DRUGGABLE GENOME, ENZYME AN-2898 42501 28966 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME atenolol ATENOLOL 42502 28967 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NIGULDIPINE NIGULDIPINE 42503 28968 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR neratinib NERATINIB 42504 28969 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE nivolumab NIVOLUMAB 26086854 42505 28970 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME PURPUROGALLIN PURPUROGALLIN 42506 28971 GMNN 51053 DRUGGABLE GENOME TDR77585 CHEMBL1333386 42508 28972 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-1000 CHEMBL600554 42509 28973 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME levomepromazine LEVOMEPROMAZINE 19308365,29472872 42510 28974 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 KAEMPFEROL KAEMPFEROL 42511 28975 SERPING1 710 DRUGGABLE GENOME, PROTEASE INHIBITOR RECOMBINANT HUMAN C1 ESTERASE INHIBITOR 42512 28976 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Cyclopentane carboxamide derivative 2 42513 28977 NUCB2 4925 DRUGGABLE GENOME hydrochlorothiazide HYDROCHLOROTHIAZIDE 31327267 42514 28978 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor VISMODEGIB VISMODEGIB 42515 28979 TUBB 203068 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 42517 28980 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 42518 28981 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE RG-1530 RG-1530 42520 28982 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DIFLUPREDNATE DIFLUPREDNATE 42521 28983 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE GDC-5573 42524 28984 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE CABOZANTINIB CABOZANTINIB 42528 28985 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TCMDC-123869 CHEMBL546597 42529 28986 MARCHF8 220972 ENZYME H1N1 influenza vaccine 42530 28987 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME FLUOCINOLONE ACETONIDE 42532 28988 GMNN 51053 DRUGGABLE GENOME FENBENDAZOLE FENBENDAZOLE 42533 28989 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR 385612241 42534 28990 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor PWT33597 42535 28991 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE clopidogrel CLOPIDOGREL 15166949,19106083,16458133,19530321,23834376,22028352 42536 28992 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE ANTHRACYCLINE 14654373 42537 28993 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1201066 VENLAFAXINE HYDROCHLORIDE 42538 28994 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DEL-22379 DEL-22379 26267534 42539 28995 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EPITIOSTANOL EPITIOSTANOL 42540 28996 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR MGCD-0103 MOCETINOSTAT 42541 28997 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Aromatic bicyclic compound 1 42542 28998 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor PF-4691502 PF-04691502 42543 28999 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER temozolomide TEMOZOLOMIDE 31624332 42544 29000 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME GOSSYPOL GOSSYPOL 42545 29001 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE LAK 9376592 42546 29002 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME EZATIOSTAT EZATIOSTAT 42551 29003 GJA1 2697 ION CHANNEL EGCG EPIGALOCATECHIN GALLATE 15736408 42552 29004 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ALKS 33 42554 29005 POLK 51426 DNA REPAIR, ENZYME METHYLENE BLUE METHYLENE BLUE 42555 29006 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CC-223 CC-223 24978597,25855786 42556 29007 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor PIVANEX AN-9 42558 29008 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178102322 TANDUTINIB 42559 29009 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-123723 CHEMBL525103 42562 29010 BCHE 590 DRUGGABLE GENOME, ENZYME HEXAFLURONIUM BROMIDE 42563 29011 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Biphenyl 1,2-diamine derivative 1 42566 29012 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE partial agonist CHEMBL299400 BUTORPHANOL TARTRATE 42567 29013 TLR7 51284 DRUGGABLE GENOME agonist 315661329 GSK-2245035 42568 29014 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor 249565633 DACTOLISIB 42570 29015 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor REGORAFENIB REGORAFENIB 42571 29016 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE CEFDINIR CEFDINIR 42572 29017 BTC 685 DRUGGABLE GENOME, GROWTH FACTOR cetuximab CETUXIMAB 42573 29018 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEMETHYLZEYLASTERONE DEMETHYLZEYLASTERONE 11678653 42575 29019 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor NECITUMUMAB NECITUMUMAB 42577 29020 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR Cabiralizumab CABIRALIZUMAB 42579 29021 GUCY2C 2984 DRUGGABLE GENOME, KINASE MLN0264 INDUSATUMAB VEDOTIN 42580 29022 CDC42BPA 8476 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CENISERTIB CENISERTIB 42581 29023 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AZOXYSTROBIN AZOXYSTROBIN 42582 29024 FPGS 2356 ENZYME, DRUGGABLE GENOME warfarin WARFARIN 42583 29025 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYSTICIN METHYSTICIN 42587 29026 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DESONIDE DESONIDE 42589 29027 PPP3CA 5530 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Pimecrolimus PIMECROLIMUS 42592 29028 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 2-(ALPHA-NAPHTHOYL)ETHYLTRIMETHYLAMMONIUM IODIDE CHEMBL1255936 42593 29029 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME RETINOIC ACID 1430209 42594 29030 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME RP6530 42597 29031 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME Cabiralizumab CABIRALIZUMAB 42598 29032 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SURAMIN SURAMIN 42599 29033 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME GO-6976 GO-6976 42600 29034 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE FLOXURIDINE FLOXURIDINE 42601 29035 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME HEPARIN HEPARIN 42603 29036 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME Anti-meso-CAR T cells 42604 29037 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ACITRETIN ACITRETIN 42605 29038 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME N-PHENETHYLCINNAMAMIDE CHEMBL1305393 42606 29039 VCP 7415 TRANSPORTER, ENZYME, DNA REPAIR, DRUGGABLE GENOME AMENTOFLAVONE AMENTOFLAVONE 42607 29040 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME XANTHOANGELOL B XANTHOANGELOL B 42608 29041 PLA2G7 7941 DRUGGABLE GENOME, ENZYME inhibitor 375973250 42609 29042 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME JNJ-68284528 42610 29043 ACTG1 71 NA THYMOSIN BETA-4 42611 29044 SLC2A5 6518 TRANSPORTER, DRUGGABLE GENOME GLUFOSFAMIDE GLUFOSFAMIDE 42613 29045 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1201119 LIOTHYRONINE SODIUM 42614 29046 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651193 42615 29047 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME BMS-582949 BMS-582949 42618 29048 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200382 BEPRIDIL HYDROCHLORIDE 42621 29049 SMN2 6607 DRUGGABLE GENOME KENPAULLONE KENPAULLONE 42623 29050 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PACLITAXEL PACLITAXEL 12761490 42624 29051 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE PATRITUMAB PATRITUMAB 26137564 42625 29052 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Taxol/Paraplatin/Herceptin 42627 29053 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BROMPHENIRAMINE BROMPHENIRAMINE 42628 29054 PDE10A 10846 ENZYME, DRUGGABLE GENOME inhibitor 384403679 42629 29055 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 celecoxib CELECOXIB 12893985,23996211,26360837,11337938,25585969,27864660,16401468,22336956,17681167,16153401 42632 29056 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Pyrazole and thiophene derivative 3 42633 29057 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR CYCLOPROPARADICICOL CYCLOPROPARADICICOL 17603540 42635 29058 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE JNJ-479655 42636 29059 NOS1 4842 DRUGGABLE GENOME, ENZYME STAUROSPORINE STAUROSPORINE 8901458 42638 29060 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist CHEMBL216981 NAVARIXIN 42639 29061 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROMAZINE PROMAZINE 42641 29062 INVS 27130 NA duloxetine DULOXETINE 29407288 42642 29063 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR PERIFOSINE PERIFOSINE 42643 29064 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER AUSTOCYSTIN D AUSTOCYSTIN D 21348461 42644 29065 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME OLAPARIB OLAPARIB 28148839 42645 29066 BAZ2B 29994 NA GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE CHEMBL1255944 42646 29067 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166828 42647 29068 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR DEXRAZOXANE DEXRAZOXANE 10487526 42649 29069 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME PURPUROGALLIN PURPUROGALLIN 42650 29070 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-PHENOXYETHANOL PHENOXYETHANOL 42651 29071 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYDROCORTISONE HEMISUCCINATE HYDROCORTISONE HEMISUCCINATE 42652 29072 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE GSK-269962A GSK-269962A 42653 29073 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TIZANIDINE TIZANIDINE 42654 29074 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL329123 ETALOCIB 42655 29075 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 1,5-NAPHTHALENEDIAMINE CHEMBL538965 42656 29076 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR LEQ-506 LEQ506 42657 29077 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME MEK165 42658 29078 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME PMID28621580-Compound-WO2013112959C68 42659 29079 TUBA3C 7278 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 42661 29080 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor SOPHORETIN QUERCETIN 42662 29081 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME RUTAECARPINE RUTAECARPINE 42663 29082 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LY-367265 CHEMBL1079460 42664 29083 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 384403681 42665 29084 PDE10A 10846 ENZYME, DRUGGABLE GENOME 1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 5 42666 29085 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Lesinurad LESINURAD 42667 29086 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GALLAMINE TRIETHIODIDE GALLAMINE TRIETHIODIDE 42668 29087 ATXN2 6311 NA DNDI1417413 CHEMBL1343568 42670 29088 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor MASITINIB MASITINIB 42671 29089 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR PD-0166285 PD-0166285 42672 29090 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist CHEMBL1201532 THYROTROPIN 42673 29091 COL1A1 1277 CLINICALLY ACTIONABLE, DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 42674 29092 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1497 BETAMETHASONE VALERATE 42676 29093 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1201063 PROPAFENONE HYDROCHLORIDE 42679 29094 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652005 42680 29095 NOS1 4842 DRUGGABLE GENOME, ENZYME BACLOFEN BACLOFEN 16137704,15476754 42681 29096 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE Indole-based analog 1 42682 29097 OCLN 100506658 DRUGGABLE GENOME, TRANSPORTER RETINOIC ACID 15500294 42683 29098 PPP1R18 170954 ENZYME carboplatin CARBOPLATIN 31616045 42685 29099 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE IPATASERTIB IPATASERTIB 30037818,23287563 42686 29100 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE DASATINIB DASATINIB 27582545 42688 29101 KCNIP4 80333 ION CHANNEL Ace Inhibitors, Plain 28084903,26169577 42691 29102 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME QUAZEPAM QUAZEPAM 42692 29103 CBX1 10951 NA NIFEDIPINE NIFEDIPINE 42693 29104 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ROCURONIUM ROCURONIUM 42695 29105 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 178102568 42696 29106 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650335 CHEMBL410478 42697 29107 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER THIOMERSAL THIMEROSAL 42698 29108 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME CANCER VACCINE 15746049 42699 29109 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SCH772984 27338794,27222538,26725216,27312529 42700 29110 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651310 42701 29111 HBB 3043 DRUGGABLE GENOME, ENZYME LentiGlobin 42702 29112 TPSAB1 7177 PROTEASE, DRUGGABLE GENOME, ENZYME Pentamidine PENTAMIDINE 42703 29113 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TRASTUZUMAB TRASTUZUMAB 15236790,16596213 42704 29114 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor 178101854 42707 29115 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2014078408Example26 42708 29116 XDH 7498 DRUGGABLE GENOME, ENZYME Fused heterocyclic compound 8 42709 29117 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL2103852 CROLIBULIN 42710 29118 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Durvalumab DURVALUMAB 42712 29119 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TETRACONAZOLE TETRACONAZOLE 42713 29120 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME MYRICETIN MYRICETIN 42714 29121 GLS 2744 ENZYME CEFIXIME CEFIXIME 42715 29122 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor 178103184 APROTININ 42716 29123 ADM 133 DRUGGABLE GENOME, HORMONE ACTIVITY NSC-106221 CHEMBL2063510 22884224 42717 29124 CAMKK2 10645 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE DOVITINIB DOVITINIB 42719 29125 DPP7 29952 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 178103152 42720 29126 PABPC1 26986 NA SJ000027778 CHEMBL592588 42721 29127 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ETHYLISOTHIOUREA ETHYLISOTHIOUREA 42722 29128 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE TRICIRIBINE TRICIRIBINE 42724 29129 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE N-ACETYLCOLCHINOL CHEMBL486504 42725 29130 MAPT 4137 DRUGGABLE GENOME GNF-PF-4659 CHEMBL584442 42726 29131 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100852 42727 29132 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL antagonist CHEMBL3545042 SELURAMPANEL 42728 29133 RAPGEF3 10411 ENZYME SENNOSIDE B SENNOSIDE B 42729 29134 ACP1 52 ENZYME, DRUGGABLE GENOME, PROTEIN PHOSPHATASE AKT INHIBITOR VIII CHEMBL258844 42730 29135 GBA 2629 DRUGGABLE GENOME, ENZYME METITEPINE METITEPINE 42731 29136 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME COUMESTROL COUMESTROL 42732 29137 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Trametinib TRAMETINIB 25370473,26644315,24265153,26566875,26582713,22389471,27312529,28179366,24265154 42733 29138 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Vemurafenib VEMURAFENIB 42734 29139 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME MK-8109 26357465 42735 29140 CLCC1 23155 ION CHANNEL opioids 42737 29141 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-269962A GSK-269962A 42738 29142 TLR7 51284 DRUGGABLE GENOME IM0-8400 42739 29143 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR RUTIN RUTIN 25496805 42740 29144 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE antibody 310264746 ONARTUZUMAB 42741 29145 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2-HYDROXYESTRADIOL CHEMBL467987 42743 29146 MTTP 4547 DRUGGABLE GENOME JNJ-16269110 USISTAPIDE 42744 29147 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME (4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE (4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE 42749 29148 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE FASUDIL FASUDIL 42752 29149 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1213490 ROMIDEPSIN 42753 29150 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651308 42754 29151 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE Peptide analog 8 42756 29152 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME GEMCITABINE GEMCITABINE 16818479 42758 29153 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME OFLOXACIN OFLOXACIN 42759 29154 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX ARTESUNATE ARTESUNATE 25074847 42762 29155 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ELND-002 42763 29156 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651246 TERGURIDE 42764 29157 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PACLITAXEL PACLITAXEL 15876424 42765 29158 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 348353666 LINRODOSTAT 42766 29159 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor SODIUM PHENYLBUTYRATE 42767 29160 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 42768 29161 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-91 42769 29162 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME olanzapine OLANZAPINE 23559402 42770 29163 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE EPINEPHRINE EPINEPHRINE 42771 29164 KDM4A 9682 DRUGGABLE GENOME, ENZYME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 42773 29165 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650378 ILOPROST 42774 29166 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR M118 42777 29167 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor XL147 PILARALISIB 42778 29168 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135652718 STRYCHNINE 42785 29169 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME EP-217609 42787 29170 ALOX15B 247 DRUGGABLE GENOME, ENZYME THIOMERSAL THIMEROSAL 42788 29171 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651660 42789 29172 TUBB2A 7280 DRUGGABLE GENOME IXABEPILONE IXABEPILONE 42790 29173 FES 2242 ENZYME, DRUGGABLE GENOME, KINASE, TYROSINE KINASE inhibitor 249565817 42791 29174 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE inhibitor 252827445 42792 29175 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 315661299 42793 29176 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME XL019 XL-019 42795 29177 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PHORBOL MYRISTATE ACETATE 9443649,9129206 42796 29178 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR GEMCITABINE GEMCITABINE 42798 29179 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME EW-A-401 42799 29180 ACSS2 55902 ENZYME, TRANSCRIPTION FACTOR gemcitabine GEMCITABINE 21636554 42800 29181 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY BACLOFEN BACLOFEN 7042732 42803 29182 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE Pyrrolo-pyrazine derivative 4 42804 29183 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545160 SU-014813 42805 29184 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIPHENHYDRAMINE DIPHENHYDRAMINE 22931300 42806 29185 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CHLORAMBUCIL CHLORAMBUCIL 11691913 42807 29186 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PROCHLORAZ PROCHLORAZ 42808 29187 POLK 51426 DNA REPAIR, ENZYME 5,8,11,14-EICOSATETRAYNOIC ACID CHEMBL458328 42809 29188 MGLL 11343 DRUGGABLE GENOME, ENZYME Piperazine carbamic compound 4 42810 29189 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PARAMETHASONE PARAMETHASONE 42811 29190 POLK 51426 DNA REPAIR, ENZYME ANAZOLENE ANAZOLENE 42812 29191 HMOX2 3163 ENZYME HORMONES 14985830 42813 29192 KCNC2 3747 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL2107762 NERISPIRDINE 42814 29193 RAB9A 9367 ENZYME, DRUGGABLE GENOME LASSBIO-294 CHEMBL233194 42816 29194 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PD-98059 CHEMBL35482 42817 29195 ATAD5 79915 NA CUCURBITACIN B CUCURBITACIN B 42818 29196 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651395 CHEMBL285819 42820 29197 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE U0126 21358673 42821 29198 CACNA2D3 55799 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL1059 PREGABALIN 42823 29199 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor 385612249 42824 29200 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME PRAZEPAM PRAZEPAM 42825 29201 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE CHEMBL1699 MEMANTINE HYDROCHLORIDE 42826 29202 TNFSF14 8740 DRUGGABLE GENOME inhibitor CHEMBL1742988 BAMINERCEPT 42827 29203 MAP2K5 5607 KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor MEK162 BINIMETINIB 42828 29204 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-3 42830 29205 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL612 DEXTROAMPHETAMINE 42831 29206 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Trodusquemine TRODUSQUEMINE 24845231 42832 29207 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 42835 29208 SP1 6667 TRANSCRIPTION FACTOR Terameprocol TERAMEPROCOL 42836 29209 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor CHEMBL520733 SEMAGACESTAT 42837 29210 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Ipatasertib IPATASERTIB 24141624,27872130 42838 29211 ACVR1B 91 SERINE THREONINE KINASE, CELL SURFACE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE BDBM108945 42839 29212 APBA1 320 NA TCMDC-125221 CHEMBL546649 42840 29213 MDH2 4191 NA GONADOTROPINS 10026128 42841 29214 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE MLN-8054 MLN-8054 42843 29215 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE methotrexate METHOTREXATE 28444425 42844 29216 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650612 MK-0767 42845 29217 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE VERAPAMIL VERAPAMIL 8622594 42846 29218 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME PD-0166285 PD-0166285 42847 29219 PSMD11 5717 KINASE CARFILZOMIB CARFILZOMIB 24524217 42848 29220 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME (S)-MEXILETINE (S)-MEXILETINE 42849 29221 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SJ000116228 CHEMBL577887 42850 29222 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER PIRARUBICIN PIRARUBICIN 12897808 42851 29223 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE GW1929 CHEMBL434063 42852 29224 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NSC319726 22624712 42853 29225 ALOX5 240 DRUGGABLE GENOME, ENZYME Zileuton ZILEUTON 42854 29226 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CAR-T Cells targeting EpCAM 42855 29227 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Ribociclib RIBOCICLIB 42856 29228 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR DHEA PRASTERONE 15675949 42858 29229 KDM4A 9682 DRUGGABLE GENOME, ENZYME SLAZINIC ACID SLAZINIC ACID 42859 29230 GMNN 51053 DRUGGABLE GENOME QUINESTROL QUINESTROL 42860 29231 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY CORDYCEPIN CORDYCEPIN 8354260 42861 29232 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME AZD-6765 LANICEMINE 42862 29233 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME QUERCETIN QUERCETIN 42863 29234 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-4068 CHEMBL584668 42865 29235 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR WITHAFERIN A WITHAFERIN A 20726569 42866 29236 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIPHENYLSTANNYL ACETATE TRIPHENYLSTANNYL ACETATE 42867 29237 HDAC11 79885 DRUGGABLE GENOME, ENZYME AR-42 AR-42 42868 29238 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME METFORMIN METFORMIN 25504439 42869 29239 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178100730 42871 29240 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR THIETHYLPERAZINE MALATE THIETHYLPERAZINE MALATE 42872 29241 IRS1 3667 KINASE, CLINICALLY ACTIONABLE ETHANOL ALCOHOL 7526037 42874 29242 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AVX901 42875 29243 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME EPO EPOETIN ALFA 9249773 42876 29244 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE blocker CHEMBL1200564 42878 29245 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3',4'-DIMETHOXYFLAVONE 3',4'-DIMETHOXYFLAVONE 42880 29246 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL572878 TOZASERTIB 42881 29247 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178100988 42882 29248 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TYRPHOSTIN A9 TYRPHOSTIN A9 42884 29249 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR ZM-447439 CHEMBL202721 42885 29250 CD276 80381 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Omburtamab I-124 42888 29251 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor BORTEZOMIB BORTEZOMIB 42889 29252 KIF11 3832 DRUGGABLE GENOME SB-743921 SB-743921 42891 29253 ALDH1A1 216 DRUGGABLE GENOME, ENZYME MERCURIC CHLORIDE MERCURIC CHLORIDE 42892 29254 COL6A3 1293 DRUGGABLE GENOME, PROTEASE INHIBITOR CHEMBL2095222 OCRIPLASMIN 42894 29255 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SB-203580 SB-203580 42896 29256 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PIRETANIDE PIRETANIDE 42897 29257 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL593430 ATAGABALIN 42900 29258 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MBX-8025 MBX-8025 42901 29259 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE lenalidomide LENALIDOMIDE 26521987 42902 29260 BAZ2B 29994 NA 4-METHYL-[1,10]PHENANTHROLINE CHEMBL316589 42905 29261 GABBR2 9568 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL BACLOFEN BACLOFEN 42906 29262 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-216385 CHEMBL274863 42907 29263 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TOLFENAMIC ACID TOLFENAMIC ACID 42909 29264 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE GLPG0187 GLPG-0187 42912 29265 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME SNS-314 SNS-314 42915 29266 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE N/A 42916 29267 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GALLIC ACID GALLIC ACID 42918 29268 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Anti-BCMA-CAR-transduced T cells 42919 29269 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL1200527 ATRACURIUM BESYLATE 42920 29270 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE GRN163 42921 29271 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME antibody 315661182 TIMOLUMAB 42922 29272 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME sorafenib SORAFENIB 20124951 42924 29273 TUBA3D 113457 DRUGGABLE GENOME CHEMBL2108628 PACLITAXEL POLIGLUMEX 42926 29274 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BIOCHANIN BIOCHANIN 42930 29275 POLB 5423 DNA REPAIR, DRUGGABLE GENOME MK-886 CHEMBL29097 42935 29276 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DROMOSTANOLONE DROMOSTANOLONE 42938 29277 BHMT2 23743 DRUGGABLE GENOME CHEMBL1201130 BETAINE HYDROCHLORIDE 42939 29278 KAT2B 8850 ENZYME, DRUGGABLE GENOME DIETHYL-2-TRIDECYLMALONATE CHEMBL1797711 21292492 42940 29279 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32d 42941 29280 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 4-METHOXYCINNAMIC ACID 4-METHOXYCINNAMIC ACID 42942 29281 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Encorafenib ENCORAFENIB 27307593,28363909,28351928,27312529 42943 29282 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME RO5126766 26438159,27669459 42944 29283 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US9434725, 315 42946 29284 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME etanercept ETANERCEPT 42947 29285 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor TELATINIB TELATINIB 42950 29286 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME RESVERATROL RESVERATROL 42951 29287 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Tremelimumab TREMELIMUMAB 42952 29288 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Quinoline and quinazoline derivative 9 42953 29289 SLC2A2 6514 TRANSPORTER, DRUGGABLE GENOME 178101360 42955 29290 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GF-109203 GF-109203 42957 29291 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SCLEROTIORIN SCLEROTIORIN 42958 29292 CEL 1056 CELL SURFACE, DRUGGABLE GENOME, ENZYME BILE SALT STIMULATED LIPASE 42959 29293 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor TRAMETINIB TRAMETINIB 42960 29294 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE gefitinib GEFITINIB 42962 29295 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody NECITUMUMAB NECITUMUMAB 42963 29296 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME BMS-387032 BMS-387032 42964 29297 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1200480 OCTREOTIDE ACETATE 42966 29298 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PARAROSANILINE PARAROSANILINE 42967 29299 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE P-HYDROXYPHENETHYL ANISATE CHEMBL1078244 42970 29300 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE ONO-AE1-437 42971 29301 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME TESOFENSINE TESOFENSINE 42972 29302 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651360 42973 29303 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE Carbimazole CARBIMAZOLE 42974 29304 ATXN2 6311 NA CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 42975 29305 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME GNF-PF-4464 CHEMBL600692 42976 29306 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SORAFENIB SORAFENIB 26619011,22310681,19537845,14679157,18186519,12068308,18794803,25157968,20619739,20350999,21129611 42978 29307 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor CHEMBL3833368 RUCAPARIB CAMSYLATE 42979 29308 XDH 7498 DRUGGABLE GENOME, ENZYME Topiroxostat TOPIROXOSTAT 42981 29309 PPP3CB 5532 TRANSCRIPTION FACTOR VOCLOSPORIN VOCLOSPORIN 42982 29310 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RITANSERIN RITANSERIN 42983 29311 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME amoxapine AMOXAPINE 42986 29312 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE KD-025 CHEMBL2005186 42987 29313 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RABEPRAZOLE SODIUM RABEPRAZOLE SODIUM 42988 29314 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Romiplostim ROMIPLOSTIM 42989 29315 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CRYPTOTANSHINONE CRYPTOTANSHINONE 42990 29316 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DAPSONE DAPSONE 22931300 42991 29317 POLI 11201 DNA REPAIR GNF-PF-1947 CHEMBL585591 42994 29318 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL587723 AEE-788 42995 29319 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME DESONIDE DESONIDE 42996 29320 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2-AMINOANTHRACENE 2-AMINOANTHRACENE 42999 29321 CYB5R1 51706 DRUGGABLE GENOME rasburicase RASBURICASE 43001 29322 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE KX2-391 KX2-391 24100628 43002 29323 EGLN2 112398 ENZYME, DRUGGABLE GENOME FG-4592 ROXADUSTAT 43003 29324 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651540 43004 29325 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PENTACHLOROPHENOL PENTACHLOROPHENOL 43005 29326 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-43 43006 29327 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PSAMMAPLIN A PSAMMAPLIN A 25884112 43007 29328 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENFURACARB BENFURACARB 43008 29329 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32a 43009 29330 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Tyverb/Tykerb 43011 29331 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME INTERFERON GAMMA 12861419 43012 29332 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000236197 CHEMBL582496 43014 29333 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 22(S)-HYDROXYCHOLESTEROL CHEMBL1243244 23830695 43015 29334 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR CARDAMOMIN CARDAMOMIN 25959811 43017 29335 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME inhibitor 135651437 43019 29336 ATXN2 6311 NA GNF-PF-2357 CHEMBL578257 43020 29337 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 43023 29338 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUNOLOL BUNOLOL 2903243 43024 29339 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-17 43025 29340 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE CEDIRANIB CEDIRANIB 43027 29341 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BERGAPTEN BERGAPTEN 43028 29342 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 252166682 43029 29343 KLC3 147700 NA platinum PLATINUM 19434073,22188361,29662106,22026922,21449681 43030 29344 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 43031 29345 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE NARINGENIN NARINGENIN 43032 29346 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CHLOROTHALONIL CHLOROTHALONIL 43033 29347 ADAM9 8754 DRUGGABLE GENOME, PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, CELL SURFACE, ENZYME inhibitor 178103981 ILOMASTAT 43034 29348 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3545153 DE-104 43036 29349 PDE10A 10846 ENZYME, DRUGGABLE GENOME 1,2,4-triazole [4,3-a]quinoxaline derivative 3 43037 29350 NME1 4830 KINASE LYCOPENE LYCOPENE 16140886 43038 29351 SMN2 6607 DRUGGABLE GENOME 2-ETHYLANTHRAQUINONE CHEMBL42355 43039 29352 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHENTHOATE PHENTHOATE 43042 29353 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565580 ENTOSPLETINIB 43043 29354 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME 3,4-METHYLENEDIOXYB-NITROSTYRENE CHEMBL596380 43044 29355 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ROSIGLITAZONE MALEATE ROSIGLITAZONE MALEATE 43045 29356 RAB9A 9367 ENZYME, DRUGGABLE GENOME 6,4'-DIHYDROXYFLAVONE CHEMBL484663 43046 29357 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR inhibitor 178101504 FLUDARABINE 43048 29358 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME TRYPAN BLUE TRYPAN BLUE 43051 29359 PSMD6 9861 NA BORTEZOMIB BORTEZOMIB 24524217 43053 29360 USP1 7398 DNA REPAIR, PROTEASE, ENZYME FLUPHENAZINE FLUPHENAZINE 43054 29361 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SB-206553 CHEMBL297784 43055 29362 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650535 43056 29363 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651140 43057 29364 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PEUCENIN PEUCENIN 43058 29365 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CRA-024781 ABEXINOSTAT 43060 29366 WNT5B 81029 DRUGGABLE GENOME Platinum compounds 24980784 43061 29367 MAPT 4137 DRUGGABLE GENOME ACID BLUE 129 ACID BLUE 129 43064 29368 GAPDH 2597 DRUGGABLE GENOME, ENZYME Omigapil OMIGAPIL 43065 29369 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PENBUTOLOL PENBUTOLOL 43066 29370 GPER1 2852 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR agonist 135650294 43067 29371 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DINOPROST TROMETHAMINE 43068 29372 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Ximelegatran 43069 29373 SULT2B1 6820 ENZYME, DRUGGABLE GENOME cytarabine CYTARABINE 22584460 43071 29374 KDM4A 9682 DRUGGABLE GENOME, ENZYME GALLIC ACID METHYL ESTER GALLIC ACID METHYL ESTER 43072 29375 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PHENFORMIN HYDROCHLORIDE PHENFORMIN HYDROCHLORIDE 43075 29376 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Savolitinib SAVOLITINIB 27694386 43076 29377 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME RIVASTIGMINE RIVASTIGMINE 43078 29378 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME RITONAVIR RITONAVIR 43079 29379 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Phenylpropylamine derivative 3 43080 29380 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXYPHENISATINE OXYPHENISATINE 43081 29381 MAPT 4137 DRUGGABLE GENOME GNF-PF-1529 CHEMBL586078 43082 29382 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TROPISETRON TROPISETRON 8013282 43083 29383 DOCK10 55619 NA INTERLEUKIN-4 18499258 43086 29384 NOS2 4843 DRUGGABLE GENOME, ENZYME inhibitor 178101804 43088 29385 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE gefitinib GEFITINIB 43090 29386 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE JNJ-7706621 JNJ-7706621 43091 29387 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-1 43093 29388 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PET-16 26984758 43095 29389 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 43096 29390 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR PYM-50028 43098 29391 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEFSULODIN SODIUM CEFSULODIN SODIUM 43099 29392 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL1201782 FOSAPREPITANT DIMEGLUMINE 43100 29393 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MICONAZOLE MICONAZOLE 43104 29394 TOP1MT 116447 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1607 TOPOTECAN HYDROCHLORIDE 43105 29395 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE cysteamine CYSTEAMINE 27035618 43106 29396 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE blocker CHEMBL41306 CNS-5161 43108 29397 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME BUTYRATE 16188956 43109 29398 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator 178101031 HEPARIN 43110 29399 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME agonist CHEMBL1201438 ALDESLEUKIN 43111 29400 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 10-METHOXYLRUTAECARPINE CHEMBL85826 43112 29401 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE DFP 13318 43113 29402 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME METAGLIDASEN METAGLIDASEN 43114 29403 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME MORIN MORIN 43117 29404 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 354702272 SELETALISIB 43120 29405 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME PMID25399719-Compound-17 43122 29406 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Indoline derivative 18 43123 29407 TUBA4A 7277 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 43124 29408 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MCLA-128 ZENOCUTUZUMAB 43127 29409 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ORG-34517 ORG-34517 43130 29410 HSPB2 3316 KINASE CSA CYCLOSPORINE 10076049 43131 29411 TUBA4A 7277 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 43133 29412 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE JNJ-55308942 43136 29413 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME A-23187 CALCIMYCIN 43138 29414 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL blocker 135651249 43141 29415 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYLDOPA (RACEMIC) METHYLDOPA (RACEMIC) 43142 29416 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AMLEXANOX AMLEXANOX 43143 29417 POLB 5423 DNA REPAIR, DRUGGABLE GENOME PENTAMIDINE DIISETHIONATE PENTAMIDINE ISETHIONATE 43144 29418 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650678 NADOLOL 43145 29419 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME Ospemifene OSPEMIFENE 43146 29420 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BIOCHANIN BIOCHANIN 43147 29421 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL NG2-73 ADIPIPLON 43148 29422 UGT2B7 7364 DRUGGABLE GENOME oxcarbazepine OXCARBAZEPINE 28837897,25823783 43149 29423 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER p28 23449360 43152 29424 STAG2 10735 CLINICALLY ACTIONABLE, DRUG RESISTANCE Temozolomide TEMOZOLOMIDE 21852505,24356817 43154 29425 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE GOSSYPOL GOSSYPOL 43156 29426 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME GARCINOL GARCINOL 19086895 43157 29427 ATAD5 79915 NA TCMDC-125784 CHEMBL581574 43158 29428 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR MUNDULONE MUNDULONE 43160 29429 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 5 43161 29430 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 328083497 TOFOGLIFLOZIN 43162 29431 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-677438 CHEMBL118678 43163 29432 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Oxeglitazar OXEGLITAZAR 43164 29433 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CILENGITIDE CILENGITIDE 43165 29434 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Pazopanib PAZOPANIB 26324075 43167 29435 RHOB 388 NA NSC-126188 CHEMBL1797159 24095759,21543141,23266181 43168 29436 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor GSK2126458 OMIPALISIB 43169 29437 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CART20 43170 29438 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE NPS-1034 24165158,23542356 43171 29439 PTGS2 5743 DRUGGABLE GENOME, ENZYME Niflumic Acid 43172 29440 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR Pyrazolopyrimidine and thienopyrimidine amide derivative 1 43173 29441 TPBG 7162 CELL SURFACE, DRUGGABLE GENOME Naptumomab estafenatox 43174 29442 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE MYRICETIN MYRICETIN 8759170 43175 29443 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE BESTATIN 9003465 43176 29444 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL12 DIAZEPAM 43177 29445 DYRK2 8445 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR HARMINE HARMINE 22998443 43179 29446 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME CUDC-101 CUDC-101 43181 29447 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME (-)-DICENTRINE CHEMBL478754 43183 29448 RAB9A 9367 ENZYME, DRUGGABLE GENOME FRENTIZOLE FRENTIZOLE 43184 29449 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Desmopressin DESMOPRESSIN 43190 29450 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SPERMIDINE SPERMIDINE 43191 29451 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SP-600125 SP-600125 43192 29452 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR BDBM50363773 43193 29453 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ANTIDEPRESSANT 1656988 43196 29454 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 249565719 43197 29455 TFF2 7032 DRUGGABLE GENOME Camostat CAMOSTAT 43198 29456 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR COMPLETE FREUND'S ADJUVANT 17974009 43199 29457 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE METFORMIN HYDROCHLORIDE 43200 29458 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 385612215 RACTOPAMINE 43202 29459 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME dronedarone DRONEDARONE 43203 29460 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor ROMIDEPSIN ROMIDEPSIN 43204 29461 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PERVILLEINE C PERVILLEINE C 11754602 43206 29462 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ROMIDEPSIN ROMIDEPSIN 43207 29463 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE trastuzumab TRASTUZUMAB 9788323,30071039,17693647 43208 29464 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME partial agonist CHEMBL18442 PLERIXAFOR 43209 29465 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIAMCINOLONE ACETONIDE TRIAMCINOLONE ACETONIDE 43210 29466 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-38 43211 29467 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 249565723 PF-00477736 43212 29468 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Bicyclic heteroaryl amide derivative 2 43213 29469 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ALMOTRIPTAN ALMOTRIPTAN 43214 29470 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-13 43217 29471 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME MONOCLONAL ANTIBODY 1F5 3500472 43218 29472 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor SF1126 43219 29473 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL861 MEPHENYTOIN 43220 29474 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 187051794 43221 29475 VKORC1L1 154807 DRUGGABLE GENOME, ENZYME warfarin WARFARIN 29054760 43222 29476 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME ZT-1 43224 29477 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652007 43225 29478 IMPDH2 3615 DRUGGABLE GENOME, ENZYME inhibitor 178103438 43226 29479 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME vortioxetine VORTIOXETINE 43228 29480 HSPB1 3315 DRUGGABLE GENOME OGX-427 APATORSEN 43229 29481 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 3,4-DIHYDROXYPHENYLACETIC ACID 3,4-DIHYDROXYPHENYLACETIC ACID 43230 29482 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE 3-amino-5-benzyl-substituted indazole derivative 1 43231 29483 SLC16A7 9194 DRUGGABLE GENOME, TRANSPORTER inhibitor 384403683 43232 29484 BAK1 578 TUMOR SUPPRESSOR, DRUGGABLE GENOME KERACYANIN KERACYANIN 17360708 43233 29485 NOX1 27035 ION CHANNEL, ENZYME, TRANSPORTER, DRUGGABLE GENOME inhibitor 363894225 43234 29486 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TOPOTECAN HYDROCHLORIDE TOPOTECAN HYDROCHLORIDE 43235 29487 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Dolutegravir DOLUTEGRAVIR 43236 29488 GMNN 51053 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 43238 29489 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX CID 867101 CHEMBL406557 43239 29490 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER KRESOXIM-METHYL KRESOXIM-METHYL 43240 29491 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NSC-95397 CHEMBL429095 43241 29492 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor 363894159 REVAMILAST 43242 29493 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135651034 43244 29494 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CO 1686 43245 29495 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649778 43247 29496 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 178100455 43248 29497 SCG5 6447 CLINICALLY ACTIONABLE, DRUGGABLE GENOME HISTONE DEACETYLASE INHIBITOR 14709802 43249 29498 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 249565753 43250 29499 HP 3240 DRUGGABLE GENOME, PROTEASE, ENZYME AT1001 22731712 43251 29500 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178100988 43252 29501 COMT 1312 DRUGGABLE GENOME, ENZYME opioids 27061230,24533707,28006928,31745220,23686330,21398039,23302985,26902643,29474345,25096645,23773341,25155931,25185591,19514130,28745577,27027462 43254 29502 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Imidazole derivative 9 43259 29503 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CSA CYCLOSPORINE 14550820 43260 29504 PTGES 9536 DRUGGABLE GENOME, ENZYME Boswellia acid derivative 1 43261 29505 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX antagonist 135650059 43262 29506 GMNN 51053 DRUGGABLE GENOME DIPHENADIONE DIPHENADIONE 43263 29507 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Dinaciclib DINACICLIB 26627013 43267 29508 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR GW7647 GW7647 43268 29509 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ILORASERTIB ILORASERTIB 43269 29510 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME AMG 820 43270 29511 AQP3 360 ION CHANNEL, TRANSPORTER inhibitor 381118899 43271 29512 STING1 340061 CLINICALLY ACTIONABLE, KINASE agonist 381118838 43272 29513 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor PF-00299804 DACOMITINIB 43273 29514 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE DS-1150b 43274 29515 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 7,8-DIHYDROXYFLAVONE 7,8-DIHYDROXYFLAVONE 43275 29516 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 dronabinol DRONABINOL 43276 29517 POLK 51426 DNA REPAIR, ENZYME 7-NITROINDAZOLE 7-NITROINDAZOLE 43278 29518 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201091 TERAZOSIN HYDROCHLORIDE HYDRATE 43280 29519 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME GW559768X GW559768X 17884497 43281 29520 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER DOXORUBICIN DOXORUBICIN 11408511 43282 29521 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL ZK-93423 CHEMBL1518572 43283 29522 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CLOTRIMAZOLE CLOTRIMAZOLE 43285 29523 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HOMIDIUM HOMIDIUM 43286 29524 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 simvastatin SIMVASTATIN 22594507,17289397 43287 29525 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NIFEDIPINE NIFEDIPINE 43288 29526 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR bucindolol BUCINDOLOL 15864115,20643254,15861037,16815314,20352314,12709726,12921807,15735607,18075464,12844134,22617224,17496726,14534524,21311897,14502278,20235788 43289 29527 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Cyproterone CYPROTERONE 43290 29528 SMN2 6607 DRUGGABLE GENOME GNF-PF-1235 CHEMBL585769 43291 29529 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR rituximab RITUXIMAB 22129793 43293 29530 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR GEMCITABINE GEMCITABINE 24588962 43296 29531 FGB 2244 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, FIBRINOGEN, DRUGGABLE GENOME abciximab ABCIXIMAB 20938371 43299 29532 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DIOTYROSINE DIOTYROSINE 43300 29533 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1201064 FLUOROMETHOLONE ACETATE 43301 29534 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME NEOSTIGMINE NEOSTIGMINE 43302 29535 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE CISPLATIN CISPLATIN 29338080,25847936,25072261 43303 29536 NT5C 30833 ENZYME gemcitabine GEMCITABINE 25162786 43304 29537 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 43306 29538 TUBA1B 10376 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 43308 29539 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYCLOSERINE CYCLOSERINE 43309 29540 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100785 43312 29541 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Fondaparinux sodium 43314 29542 USP1 7398 DNA REPAIR, PROTEASE, ENZYME 5,7-DIHYDROXYISOFLAVONE 5,7-DIHYDROXYISOFLAVONE 43315 29543 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE MOROLIC ACID MOROLIC ACID 21453996 43317 29544 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-95 43322 29545 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON BETA-1B 43325 29546 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHANDROSTENOLONE METHANDROSTENOLONE 43326 29547 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ANACARDIC ACID 19099397 43327 29548 BAZ2B 29994 NA TAMOXIFEN CITRATE TAMOXIFEN CITRATE 43328 29549 NOTCH3 4854 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor PF-03084014 NIROGACESTAT 43329 29550 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID29757691-Compound-4 43330 29551 KDM4A 9682 DRUGGABLE GENOME, ENZYME NANAOMYCIN NANAOMYCIN 43331 29552 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME DOVITINIB DOVITINIB 43332 29553 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PF-04691502 PF-04691502 26725216,21750219 43335 29554 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-48 43336 29555 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SELICICLIB SELICICLIB 21080703 43337 29556 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MYRICETIN MYRICETIN 8759170,7769390 43339 29557 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR CCT244747 CHEMBL2203843 23082860 43341 29558 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME LEVDOBUTAMINE LEVDOBUTAMINE 43342 29559 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 6 43344 29560 CYB5R1 51706 DRUGGABLE GENOME isosorbide dinitrate 43346 29561 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME LEVOCETIRIZINE LEVOCETIRIZINE 43347 29562 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR VINBLASTINE VINBLASTINE 10640980 43348 29563 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME oxaliplatin OXALIPLATIN 24090479,20125120,25955730 43349 29564 AICDA 57379 ENZYME JX-929 43353 29565 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-50 43354 29566 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651182 43355 29567 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE 5-METHOXYCANTHINONE 5-METHOXYCANTHINONE 43356 29568 DPP7 29952 PROTEASE, ENZYME, DRUGGABLE GENOME US8470836, 5 43357 29569 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 385612219 BREPOCITINIB 43359 29570 SAE1 10055 ENZYME, DRUGGABLE GENOME BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 43360 29571 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102271 43361 29572 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE EB-101 43362 29573 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Cobimetinib COBIMETINIB 23934108 43363 29574 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200895 PHENELZINE SULFATE 43364 29575 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME selegiline SELEGILINE 17638512,11470993 43366 29576 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR MONTELUKAST SODIUM MONTELUKAST SODIUM 43367 29577 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 1096708-71-2 43368 29578 GMNN 51053 DRUGGABLE GENOME DNDI1417623 CHEMBL2002849 43369 29579 PNPLA3 80339 ENZYME prednisolone PREDNISOLONE 28744905 43371 29580 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MK-0773 MK-0773 43372 29581 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE SORAFENIB SORAFENIB 43373 29582 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE IMATINIB IMATINIB 43374 29583 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-1319 CHEMBL235891 43377 29584 TGFB2 7042 GROWTH FACTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME antibody FRESOLIMUMAB FRESOLIMUMAB 43379 29585 FMO3 2328 ENZYME, DRUGGABLE GENOME rosuvastatin ROSUVASTATIN 20679960 43380 29586 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TCMDC-125473 CHEMBL535051 43383 29587 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PD-146176 CHEMBL180917 43384 29588 RGS4 5999 DRUGGABLE GENOME TYRPHOSTIN 23 TYRPHOSTIN 23 43385 29589 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 178102618 43386 29590 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CRENOLANIB CRENOLANIB 43387 29591 ADRM1 11047 ENZYME inhibitor CHEMBL451887 CARFILZOMIB 43388 29592 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Dabrafenib DABRAFENIB 27659046 43389 29593 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ZNCL2 8131214 43390 29594 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME SHP099 27362227 43392 29595 POLI 11201 DNA REPAIR NSC-36398 CHEMBL483206 43394 29596 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL1213490 ROMIDEPSIN 43395 29597 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME DORAMAPIMOD DORAMAPIMOD 43396 29598 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME THIOPERAMIDE THIOPERAMIDE 43397 29599 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TRIAMTERENE TRIAMTERENE 43399 29600 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 QUINOXALINE1 QUINOXALINE1 43400 29601 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-123605 CHEMBL547285 43401 29602 PARP3 10039 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR inhibitor CHEMBL521686 OLAPARIB 43404 29603 FAAH 2166 ENZYME, DRUGGABLE GENOME Tetra-hydro-naphthalene derivative 2 43405 29604 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE ETOPOSIDE ETOPOSIDE 9716508 43406 29605 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME CARMUSTINE CARMUSTINE 43407 29606 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DAUNORUBICIN DAUNORUBICIN 43408 29607 TUBA3C 7278 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 43409 29608 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ATD transdermal gel 43410 29609 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR enalapril ENALAPRIL 24059494 43411 29610 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Cisplatin CISPLATIN 27196758 43412 29611 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL70418 CLOBAZAM 43413 29612 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 381118855 43414 29613 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR SURAMIN SURAMIN 43415 29614 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1201099 CODEINE PHOSPHATE 43416 29615 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL1096380 PLINABULIN 43417 29616 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 2',3'-DIHYDROXYFLAVONE CHEMBL242171 43418 29617 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TANGERETIN TANGERETIN 43419 29618 TOP2B 7155 DRUGGABLE GENOME, ENZYME Gepotidacin GEPOTIDACIN 43420 29619 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 L-733060 CHEMBL27006 43421 29620 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BYL719 ALPELISIB 26504226,25544636,26577700,27604488,28119489 43422 29621 TUBB2A 7280 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 43425 29622 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CLOTRIMAZOLE CLOTRIMAZOLE 16680159 43426 29623 BAZ2B 29994 NA RESERPINE RESERPINE 43427 29624 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 178101152 CHEMBL177991 43429 29625 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Lucitanib LUCITANIB 27126994 43430 29626 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ANETHOLTRITHION ANETHOLTRITHION 43432 29627 PSMB4 5692 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL325041 BORTEZOMIB 43434 29628 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE IFOSFAMIDE IFOSFAMIDE 43435 29629 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 1,4,5,8-TETRAAMINO-ANTHRAQUINONE CHEMBL87568 43436 29630 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AZD9291 OSIMERTINIB 43437 29631 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME CARFILZOMIB CARFILZOMIB 43438 29632 HSPB1 3315 DRUGGABLE GENOME ALPHA-TERTHIENYL ALPHA-TERTHIENYL 43439 29633 CBX1 10951 NA AG-555 CHEMBL53898 43440 29634 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME ifosfamide IFOSFAMIDE 17638512,11470993 43441 29635 BUB1 699 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME SCHEMBL17766424 43442 29636 NR2F2 7026 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TCMDC-125620 CHEMBL530291 43444 29637 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody MEHD7945 A 43445 29638 MAOA 4128 DRUGGABLE GENOME, ENZYME HouttuynoidA 43446 29639 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1651 DEXAMETHASONE ACETATE 43447 29640 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROFLAVINE PROFLAVINE 43448 29641 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Peptide analog 45 43449 29642 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME blocker 178101099 PHENCYCLIDINE 43450 29643 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL101253 VATALANIB 43451 29644 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2-METHYL GRAMINE 2-METHYL GRAMINE 43453 29645 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 43455 29646 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME EP217609 43456 29647 MGAT2 4247 ENZYME Dihydropyrimidinone derivative 3 43458 29648 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 43459 29649 PAPLN 89932 PROTEASE INHIBITOR citalopram CITALOPRAM 43460 29650 MAPT 4137 DRUGGABLE GENOME SJ000024939 CHEMBL590691 43462 29651 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3',4'-DIHYDROXYFLAVONE CHEMBL222556 43463 29652 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651551 PROGESTERONE 43464 29653 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4012 CHEMBL584269 43466 29654 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Indazoletriazolephenyl derivative 1 43467 29655 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORAMPHENICOL PALMITATE CHLORAMPHENICOL PALMITATE 43469 29656 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME CEPHALOTHIN CEPHALOTHIN 43473 29657 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Pyrrolidine derivative 10 43474 29658 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME antagonist 178103613 43475 29659 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor RIBOCICLIB RIBOCICLIB 43477 29660 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 374883849 TRIFAROTENE 43478 29661 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4,4'-DIHYDROXYDIPHENYLMETHANE CHEMBL138061 43479 29662 TNNI3 7137 DRUGGABLE GENOME PURPUROGALLIN PURPUROGALLIN 43481 29663 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL1743032 INTETUMUMAB 43482 29664 HDAC11 79885 DRUGGABLE GENOME, ENZYME valproic acid 23407051 43485 29665 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME HINOKITIOL HINOKITIOL 43487 29666 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL984 MIVACURIUM CHLORIDE 43488 29667 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE WR-159412 WR-159412 43489 29668 HPSE 10855 ENZYME, DRUGGABLE GENOME inhibitor 363894164 43490 29669 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL blocker 178101137 43491 29670 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE NAKIJIQUINONE I NAKIJIQUINONE I 18676149 43492 29671 KDM4A 9682 DRUGGABLE GENOME, ENZYME N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 43493 29672 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-18 43494 29673 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE EPO EPOETIN ALFA 16337691 43495 29674 PSMC3 5702 NA BORTEZOMIB BORTEZOMIB 24524217 43497 29675 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3301623 PATIDEGIB 43498 29676 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-66209 CHEMBL175266 43500 29677 ACVR1B 91 SERINE THREONINE KINASE, CELL SURFACE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE US9682983, 1 43502 29678 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME 7,12-DIMETHYL-BENZO[A]ANTHRACENE CHEMBL329673 43504 29679 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE Rilapladib RILAPLADIB 43505 29680 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PENTABROMOPHENOL PENTABROMOPHENOL 43506 29681 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565698 43507 29682 FAAH 2166 ENZYME, DRUGGABLE GENOME Aryl urea derivative 2 43509 29683 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME L-THREO-BENZYLOXY ASPARTATE CHEMBL79140 43510 29684 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CID1067700 19477428,26247207 43511 29685 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME TAE-684 TAE-684 43512 29686 IFNG 3458 DRUGGABLE GENOME MELPHALAN MELPHALAN 9864423 43514 29687 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIFLUCORTOLONE 21-VALERATE DIFLUCORTOLONE 21-VALERATE 43516 29688 TUBB2B 347733 DRUGGABLE GENOME CHEMBL2108628 PACLITAXEL POLIGLUMEX 43519 29689 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RS-16566 CHEMBL145725 43521 29690 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME U-0126 U-0126 43522 29691 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor SNS-032 BMS-387032 43524 29692 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ANTINEOPLASTIC 12839976 43527 29693 CBX1 10951 NA EBSELEN EBSELEN 43528 29694 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 OXOTREMORINE OXOTREMORINE 43529 29695 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 315661146 PF-03882845 43532 29696 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE TRIIODOTHYRONINE LIOTHYRONINE SODIUM 9217278 43533 29697 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AG-555 CHEMBL53898 43535 29698 XDH 7498 DRUGGABLE GENOME, ENZYME IFN 8046245 43536 29699 F2RL3 9002 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 385612202 43538 29700 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178101884 GSK-690693 43541 29701 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR MAO INHIBITORS 14512210 43543 29702 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROGLUMETACIN PROGLUMETACIN 43544 29703 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SKI-758 CHEMBL219557 43546 29704 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650415 43548 29705 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME GSK812397 CHEMBL1242210 19949058 43549 29706 PTGS2 5743 DRUGGABLE GENOME, ENZYME IMRECOXIB IMRECOXIB 43550 29707 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR RNA POLYMERASE INHIBITOR 9406930 43551 29708 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME FENRETINIDE FENRETINIDE 43552 29709 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE poziotinib POZIOTINIB 21306821 43553 29710 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 paroxetine PAROXETINE 43554 29711 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLEMASTINE CLEMASTINE 43556 29712 CXCL8 3576 DRUGGABLE GENOME RO 31-8220 2163626 43557 29713 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL856 PRIMIDONE 43558 29714 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-81747 CHEMBL1371696 43560 29715 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ribavirin RIBAVIRIN 21572301 43561 29716 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 315661257 ALTIRATINIB 43563 29717 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SJ000291458 CHEMBL592598 43565 29718 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IIC AESCULIOSIDE IIC 20371180 43566 29719 EPHX2 2053 DRUGGABLE GENOME, ENZYME ALOE-EMODIN ALOE-EMODIN 26372074 43567 29720 CBX1 10951 NA FIDUXOSIN FIDUXOSIN 43569 29721 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SANGUINARIUM CHLORIDE SANGUINARIUM CHLORIDE 43570 29722 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 315661129 DIFELIKEFALIN 43572 29723 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TRIFLUOPERAZINE TRIFLUOPERAZINE 43573 29724 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL MIDAZOLAM MIDAZOLAM 43574 29725 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650553 43575 29726 PPAT 5471 DRUGGABLE GENOME, ENZYME Mercaptopurine MERCAPTOPURINE 43577 29727 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3545181 TIOTROPIUM BROMIDE 43578 29728 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MELPHALAN MELPHALAN 43579 29729 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR NIMODIPINE NIMODIPINE 11486117 43580 29730 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME CEA/MUC-1/VF/TRICOM 43583 29731 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-202190 SB-202190 43584 29732 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 135651305 VERAPAMIL 43586 29733 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME IPILIMUMAB IPILIMUMAB 43587 29734 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE OUABAIN OUABAIN 43589 29735 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-94 43590 29736 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE Alkynyl-substituted pyrimidinyl-pyrrole derivative 1 43591 29737 POLI 11201 DNA REPAIR DNDI1417086 CHEMBL1224755 43592 29738 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CYTOLIN 43593 29739 TRPM6 140803 ION CHANNEL, DRUGGABLE GENOME, ENZYME, TRANSPORTER, KINASE, SERINE THREONINE KINASE activator 135652738 43594 29740 TSPO 706 DRUGGABLE GENOME TLN-4601 DIAZEPINOMICIN 43595 29741 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 3,4-DIMETHOXYBENZALDEHYDE 3,4-DIMETHOXYBENZALDEHYDE 43596 29742 GGH 8836 PROTEASE, ENZYME, DRUGGABLE GENOME bevacizumab BEVACIZUMAB 43598 29743 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR ALSTERPAULLONE ALSTERPAULLONE 43599 29744 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 187051800 BUFEXAMAC 43600 29745 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL750 ZONISAMIDE 43601 29746 PSMB9 5698 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL325041 BORTEZOMIB 43604 29747 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL1743071 SIRUKUMAB 43605 29748 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-326757 CHEMBL1368535 43606 29749 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL1201023 ORPHENADRINE HYDROCHLORIDE 43610 29750 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CHOLESTYRAMINE CHOLESTYRAMINE 2110363 43611 29751 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774824-Compound-Figure9Example2down 43613 29752 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor XL281 XL-281 43614 29753 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TRIMETHOPRIM TRIMETHOPRIM 22931300 43615 29754 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Amidopyrazole derivative 5 43616 29755 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE inhibitor CHEMBL189963 PALBOCICLIB 43617 29756 RBX1 9978 DNA REPAIR, ENZYME epirubicin EPIRUBICIN 43618 29757 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651369 43619 29758 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135649663 43623 29759 IGFBP1 3484 DRUGGABLE GENOME BUSERELIN BUSERELIN 7544746 43624 29760 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE FENOTEROL HBR FENOTEROL HBR 43625 29761 NUCB1 4924 DRUGGABLE GENOME GS-5734 REMDESIVIR 43626 29762 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 178102555 JNJ-7706621 43628 29763 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102779 43629 29764 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE 178101615 43630 29765 ATXN2 6311 NA SJ000059275 CHEMBL603952 43632 29766 FAAH 2166 ENZYME, DRUGGABLE GENOME Ketoheterocycle derivative 3 43633 29767 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 178101956 43634 29768 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE PF-05212384 GEDATOLISIB 43635 29769 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL521686 OLAPARIB 43636 29770 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALLO-OCIMENE ALLO-OCIMENE 43637 29771 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 43638 29772 CD38 952 CELL SURFACE, DRUGGABLE GENOME Daratumumab DARATUMUMAB 43639 29773 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135649797 4-DAMP 43640 29774 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL52885 ENMD-981693 43645 29775 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102307 ALVOCIDIB 43651 29776 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME AG-537 CHEMBL67535 43652 29777 CDA 978 ENZYME, DRUGGABLE GENOME capecitabine CAPECITABINE 21325291,24167597,28347776,18473752,23736036 43655 29778 BRD7 29117 ENZYME inhibitor 310264731 43656 29779 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-95397 CHEMBL429095 43657 29780 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TROGLITAZONE TROGLITAZONE 22931300 43658 29781 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME apixaban APIXABAN 28678049,29457840 43659 29782 SMARCA2 6595 NA AMINACRINE HYDROCHLORIDE AMINACRINE HYDROCHLORIDE 43660 29783 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CINOBUFOTALIN CINOBUFOTALIN 43662 29784 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AZTREONAM AZTREONAM 22931300 43663 29785 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-2374 CHEMBL600298 43664 29786 APOE 348 DRUGGABLE GENOME IMMUNOSUPPRESSANT 12752312 43666 29787 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 4-DAMP 4-DAMP 43667 29788 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178100241 CELECOXIB 43669 29789 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME inhibitor 381745024 43670 29790 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200413 TETRAHYDROZOLINE HYDROCHLORIDE 43671 29791 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NAPROPAMIDE NAPROPAMIDE 43673 29792 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE Peptide analog 62 43674 29793 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Endocrine therapy 43675 29794 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL IBUTILIDE IBUTILIDE 43677 29795 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DINITRO CRESOL DINITRO CRESOL 43678 29796 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME gemcitabine GEMCITABINE 21636554 43679 29797 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PF-562271 PF-00562271 43680 29798 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE atorvastatin ATORVASTATIN 24311107,21151198 43683 29799 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Pyrotinib PYROTINIB 28498781 43685 29800 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE LEXATUMUMAB LEXATUMUMAB 43687 29801 TDO2 6999 ENZYME, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 5 43689 29802 GDA 9615 ENZYME NSC-7861 7-METHYLXANTHINE 20716488 43691 29803 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRICLOSAN TRICLOSAN 43692 29804 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BGJ398 INFIGRATINIB 43693 29805 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE U-0126 U-0126 43694 29806 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102569 43695 29807 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 178103589 RICOLINOSTAT 43696 29808 STK24 8428 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 178102336 BOSUTINIB 43697 29809 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL1200485 SORAFENIB TOSYLATE 43700 29810 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HEXACHLOROPHENE HEXACHLOROPHENE 43702 29811 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ENZYME INHIBITOR 17059765 43704 29812 CBX1 10951 NA ISOPROTERENOL ISOPROTERENOL 43705 29813 PRF1 5551 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 387065583 43709 29814 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 363894199 43710 29815 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MM-151 43711 29816 TRPM6 140803 ION CHANNEL, DRUGGABLE GENOME, ENZYME, TRANSPORTER, KINASE, SERINE THREONINE KINASE activator 135649695 43712 29817 KDM4A 9682 DRUGGABLE GENOME, ENZYME inhibitor 340590215 43713 29818 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL979 MEPROBAMATE 43715 29819 POLI 11201 DNA REPAIR BI-87E7 CHEMBL523200 43716 29820 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PURVALANOLA PURVALANOLA 43717 29821 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Isoquinoline derivative 5 43720 29822 ATP5F1D 513 TRANSPORTER METHOXYFLURANE METHOXYFLURANE 43721 29823 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 252827519 43722 29824 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MEGESTROL MEGESTROL 43723 29825 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE LINIFANIB LINIFANIB 43724 29826 TH 7054 ENZYME, DRUGGABLE GENOME ProSavin 43727 29827 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor CHEMBL494089 GSK-690693 43730 29828 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER 2-CHLORO-ADENOSINETRIPHOSPHATE CHEMBL1368696 43731 29829 PROX1 5629 TRANSCRIPTION FACTOR atenolol ATENOLOL 43733 29830 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102660 43734 29831 ALOX15 246 ENZYME, DRUGGABLE GENOME GINGKOLIC ACID GINGKOLIC ACID 43735 29832 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE inhibitor 178101437 DIGOXIN 43736 29833 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE CHEMBL1255944 43737 29834 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SELUMETINIB SELUMETINIB 25952648 43738 29835 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-60339 CHEMBL1448793 43741 29836 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NATEGLINIDE NATEGLINIDE 22931300 43742 29837 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CABOZANTANIB 43743 29838 ADK 132 DRUGGABLE GENOME, ENZYME, KINASE 2,3-DIDEOXYADENOSINE 3262616 43748 29839 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Capmatinib CAPMATINIB 43749 29840 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME THIETHYLPERAZINE THIETHYLPERAZINE 43750 29841 CCL2 6347 DRUGGABLE GENOME Carlumab CARLUMAB 43751 29842 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 43752 29843 LTC4S 4056 ENZYME, DRUGGABLE GENOME inhibitor 336446941 43753 29844 MAPKAPK5 8550 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE GLPG0259 GLPG-0259 43755 29845 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL TEMAZEPAM TEMAZEPAM 43756 29846 ATXN2 6311 NA THIORIDAZINE HYDROCHLORIDE THIORIDAZINE HYDROCHLORIDE 43757 29847 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200420 MIDAZOLAM HYDROCHLORIDE 43758 29848 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TBC-3711 43762 29849 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME UMBELLIFERONE UMBELLIFERONE 43766 29850 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3545332 CEP-2563 43767 29851 TSPO 706 DRUGGABLE GENOME Imidazo[1,2-b]pyridazine acetamide derivative 7 43768 29852 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1059 PREGABALIN 43769 29853 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME BMS-753493 EPOFOLATE 43770 29854 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR SANDOSTATIN SANDOSTATIN 12142738 43771 29855 COMT 1312 DRUGGABLE GENOME, ENZYME Tolcapone TOLCAPONE 43773 29856 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SANGUINARINE SULFATE SANGUINARINE SULFATE 43774 29857 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Nilotinib NILOTINIB 43775 29858 PSME4 23198 DNA REPAIR inhibitor BORTEZOMIB BORTEZOMIB 43776 29859 ALPI 248 DRUGGABLE GENOME, ENZYME BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 43777 29860 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 13 43779 29861 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL FELODIPINE FELODIPINE 43781 29862 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor 178103458 VORINOSTAT 43782 29863 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE PD-98059 CHEMBL35482 11978788 43783 29864 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL BUTABARBITAL BUTABARBITAL 43784 29865 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-154983 CHEMBL227298 43785 29866 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor 363894203 RG-7420 43788 29867 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GABAZINE GABAZINE 43790 29868 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Tyrosine kinase inhibitor - NS 43791 29869 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE ISOPROTERENOL ISOPROTERENOL 12509508 43792 29870 PDE4B 5142 DRUGGABLE GENOME, ENZYME AMRINONE INAMRINONE 43793 29871 KDM4A 9682 DRUGGABLE GENOME, ENZYME PENTACHLOROPHENOL PENTACHLOROPHENOL 43794 29872 PERP 64065 NA fluorouracil FLUOROURACIL 43795 29873 BAZ2B 29994 NA EBSELEN EBSELEN 43796 29874 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 249565825 43798 29875 EPB41 2035 TRANSPORTER bupropion BUPROPION 43799 29876 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME U-73122 CHEMBL1256678 43800 29877 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ESTRADIOL ESTRADIOL 20334368,20659801,25879485,16038533,16520733,19561619,24805199 43801 29878 GUCY1A2 2977 ENZYME, DRUGGABLE GENOME positive modulator CHEMBL2107834 RIOCIGUAT 43802 29879 HMGCR 3156 ENZYME, DRUGGABLE GENOME PITAVASTATIN PITAVASTATIN 43803 29880 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME APICIDIN APICIDIN 19705846 43804 29881 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROPIOMAZINE PROPIOMAZINE 43805 29882 ALOX15 246 ENZYME, DRUGGABLE GENOME LUTEOLIN LUTEOLIN 43806 29883 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NSC-119236 CHEMBL458765 43807 29884 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE SCH772984 25104330 43808 29885 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Decitabine DECITABINE 27418649 43809 29886 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL3545081 RG-7304 43811 29887 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE ATORVASTATIN ATORVASTATIN 16701707 43812 29888 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SULFADOXINE SULFADOXINE 22931300 43813 29889 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 328083463 CHEMBL561708 43814 29890 GMNN 51053 DRUGGABLE GENOME DNDI1417080 CHEMBL1498652 43816 29891 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLOROTRIANISENE CHLOROTRIANISENE 43817 29892 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL128 SUMATRIPTAN 43820 29893 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER N-(4-CARBOXYPHENYL)RHODANINE CHEMBL450802 43821 29894 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE CHOLESTYRAMINE CHOLESTYRAMINE 3906004 43822 29895 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME NALOXONE NALOXONE 2738884 43824 29896 NOS2 4843 DRUGGABLE GENOME, ENZYME NIMODIPINE NIMODIPINE 16044358 43826 29897 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TESTOSTERONE PROPIONATE TESTOSTERONE PROPIONATE 43827 29898 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE activator 53801036 43828 29899 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE KLUGINE KLUGINE 15974627 43829 29900 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 4SC-202 DOMATINOSTAT 43830 29901 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR QUINALIZARIN QUINALIZARIN 43832 29902 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135650663 43833 29903 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SALIRASIB SALIRASIB 22547163 43834 29904 HTT 3064 DRUGGABLE GENOME GNF-PF-1083 CHEMBL530361 43835 29905 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 43836 29906 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR ETHANOL ALCOHOL 15745088,14627336 43837 29907 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650347 43838 29908 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Valproic Acid 20739657 43839 29909 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 1 43841 29910 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 385612185 43842 29911 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 EBSELEN EBSELEN 43843 29912 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-228155 CHEMBL505670 43846 29913 GMNN 51053 DRUGGABLE GENOME GNF-PF-1319 CHEMBL235891 43848 29914 HTT 3064 DRUGGABLE GENOME BITHIONOL BITHIONOL 43849 29915 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 187051838 43850 29916 FGA 2243 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, FIBRINOGEN tirofiban TIROFIBAN 20938371 43852 29917 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY STAUROSPORINE STAUROSPORINE 8879350 43854 29918 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PD173074 21666749,21160078 43855 29919 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-677438 CHEMBL118678 43856 29920 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME GNF-PF-1852 CHEMBL533293 43857 29921 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME JNJ-42756493 ERDAFITINIB 26324363,28341788 43859 29922 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 178103527 METHYLTESTOSTERONE 43860 29923 ILF3 3609 KINASE, TRANSCRIPTION FACTOR CSA CYCLOSPORINE 9843854 43861 29924 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME N/A 21881046,22417203,22915647,24487413 43862 29925 TSPO 706 DRUGGABLE GENOME CHLORMEZANONE CHLORMEZANONE 43863 29926 APOE 348 DRUGGABLE GENOME fluvastatin FLUVASTATIN 17289397,30363031 43864 29927 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL SAFINAMIDE SAFINAMIDE 43865 29928 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tetra-hydro-isoquinoline derivative 1 43866 29929 DUSP3 1845 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE TDR77585 CHEMBL1333386 43871 29930 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME KENPAULLONE KENPAULLONE 43872 29931 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME AG-538 CHEMBL56393 43873 29932 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME IMETIT IMETIT 43875 29933 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TYROSINE KINASE INHIBITORS 11163336 43876 29934 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-MTC-423 43880 29935 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DOXORUBICIN DOXORUBICIN 22698404,17363498,9569050,24065105 43881 29936 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 43882 29937 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-695801 CHEMBL461193 43883 29938 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE H2O2 8732780 43885 29939 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ANGIOTENSIN II 43887 29940 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE HEXACHLOROPHENE HEXACHLOROPHENE 43891 29941 PTGS2 5743 DRUGGABLE GENOME, ENZYME DERSALAZINE DERSALAZINE 43892 29942 PTGS2 5743 DRUGGABLE GENOME, ENZYME INDOMETHACIN INDOMETHACIN 24697244,20684598,22818041 43896 29943 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor PD325901 43898 29944 SAE1 10055 ENZYME, DRUGGABLE GENOME GINGKOLIC ACID GINGKOLIC ACID 23920437 43899 29945 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL1096380 PLINABULIN 43901 29946 MAPT 4137 DRUGGABLE GENOME ETHACRIDINE LACTATE ETHACRIDINE LACTATE 43903 29947 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor PCI-24781 ABEXINOSTAT 43904 29948 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE Tricyclic compound 7 43905 29949 LPAR5 57121 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME (S)-CARBA CYCLIC-PHOSPHATIDIC ACID CHEMBL1630084 21051230 43906 29950 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE axitinib AXITINIB 20124951 43907 29951 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 43909 29952 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-98938 CHEMBL1939691 43910 29953 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Mepivacaine MEPIVACAINE 43912 29954 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE artemether ARTEMETHER 43915 29955 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME amiodarone AMIODARONE 43916 29956 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE D-Serine (D)-SERINE 43917 29957 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR TINZAPARIN TINZAPARIN 43919 29958 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR FLUAZINAM FLUAZINAM 43921 29959 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME LAUROGUADINE LAUROGUADINE 43923 29960 KDM4A 9682 DRUGGABLE GENOME, ENZYME HARMAN-3-CARBOXYLIC ACID HARMAN-3-CARBOXYLIC ACID 43925 29961 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CYCLOHEXIMIDE CYCLOHEXIMIDE 43926 29962 GAA 2548 DRUGGABLE GENOME, ENZYME AMLEXANOX AMLEXANOX 43927 29963 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME KAEMPFEROL KAEMPFEROL 43928 29964 PSMB3 5691 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL2103884 OPROZOMIB 43929 29965 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CYCLIZINE CYCLIZINE 43930 29966 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MIDODRINE MIDODRINE 22931300 43931 29967 FCER1G 2207 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE BENZYLPENICILLOYL POLYLYSINE 43932 29968 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 albendazole ALBENDAZOLE 19923256 43933 29969 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PHOSMET PHOSMET 43934 29970 RACGAP1 29127 NA 4-METHYLDAPHNETIN 4-METHYLDAPHNETIN 43935 29971 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545048 AMG-319 43937 29972 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DEPHOSTATIN DEPHOSTATIN 43939 29973 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME SJ000040829 CHEMBL589711 43940 29974 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME LITHOCHOLIC ACID LITHOCHOLIC ACID 43941 29975 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME SAR 1118 43944 29976 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME Sulfonamide derivative 16 43946 29977 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1201002 CARTEOLOL HYDROCHLORIDE 43947 29978 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor 318164849 CDP840 43948 29979 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER NSC-50688 CHEMBL1456848 43949 29980 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PIROXICAM PIROXICAM 22931300 43951 29981 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 KETOCONAZOLE KETOCONAZOLE 26360048,24996140,22931300,26052884 43952 29982 PBRM1 55193 CLINICALLY ACTIONABLE EVEROLIMUS EVEROLIMUS 27751729 43953 29983 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL3137307 PEFCALCITOL 43954 29984 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Descartes-08 43955 29985 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME Rapamycin SIROLIMUS 43957 29986 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 sulfamethoxazole SULFAMETHOXAZOLE 11186133 43959 29987 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE OLAPARIB OLAPARIB 43960 29988 SERPIND1 3053 DRUGGABLE GENOME, PROTEASE INHIBITOR ARDEPARIN 43961 29989 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 178102330 PLX-4720 43962 29990 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor BYL719 ALPELISIB 43963 29991 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PHENYLBUTANOIC ACID PHENYLBUTANOIC ACID 24044874 43965 29992 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ISOSILYBIN A ISOSILYBIN A 24597776 43966 29993 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE CLODRONATE CLODRONIC ACID 11984068 43969 29994 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE BYL719 ALPELISIB 43970 29995 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 328083528 FRUQUINTINIB 43971 29996 ATXN2 6311 NA 1,7-O-DIACETYLMETHYLGEOPYXIN A CHEMBL1889303 43972 29997 KDM4A 9682 DRUGGABLE GENOME, ENZYME GALUTEOLIN GALUTEOLIN 43973 29998 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE agonist 178103562 43974 29999 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL activator 135652724 VERATRIDINE 43977 30000 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CETYLPYRIDINIUM CHLORIDE CETYLPYRIDINIUM CHLORIDE 43978 30001 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR CISPLATIN CISPLATIN 11145600,15610860 43980 30002 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-3876 CHEMBL596631 43983 30003 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200948 TRIMIPRAMINE MALEATE 43984 30004 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME IMMUNOMODULATORS 1557611 43985 30005 USP1 7398 DNA REPAIR, PROTEASE, ENZYME INDOCYANINE GREEN INDOCYANINE GREEN 43986 30006 ATAD5 79915 NA ISOLIQUIRITIGENIN ISOLIQUIRITIGENIN 43987 30007 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME CHEMBL3039521 VINTAFOLIDE 43990 30008 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Cyclopropyl-spiro piperidine derivative 4 43991 30009 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME ANTIHEMOPHILIC FACTOR 43992 30010 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649986 43993 30011 KIF11 3832 DRUGGABLE GENOME S-TRITYL-L-CYSTEINE S-TRITYL-L-CYSTEINE 22749640 43994 30012 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-62 43995 30013 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-Figure17 43996 30014 DYRK2 8445 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR LEUCETTAMINE B LEUCETTAMINE B 22998443 43998 30015 HEBP1 50865 DRUGGABLE GENOME Thiazole derivative 2 44001 30016 DDC 1644 ENZYME, DRUGGABLE GENOME Carbidopa CARBIDOPA 44002 30017 GBA 2629 DRUGGABLE GENOME, ENZYME TRICHOSTATIN TRICHOSTATIN 44003 30018 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CAROTENOID 10051470 44005 30019 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor GDC-0980 APITOLISIB 44007 30020 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Pyrazole and thiophene derivative 4 44008 30021 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-2588 CHEMBL578636 44009 30022 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US10166249, Example 695 44011 30023 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR FENOFIBRIC ACID FENOFIBRIC ACID 22579484,21855333,23566516 44015 30024 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Benzimidazole carboxamide derivative 1 44017 30025 HSPB1 3315 DRUGGABLE GENOME HYMECROMONE HYMECROMONE 44019 30026 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL940 GABAPENTIN 44023 30027 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME AC-170 CETIRIZINE 44024 30028 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE agonist CHEMBL1201556 BECAPLERMIN 44025 30029 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL661 ALPRAZOLAM 44028 30030 HEXB 3074 ENZYME GENTAMICIN GENTAMICIN 2876489,8456116 44029 30031 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW513184X GW513184X 44030 30032 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 VERAPAMIL HYDROCHLORIDE VERAPAMIL HYDROCHLORIDE 44031 30033 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE efavirenz EFAVIRENZ 26774523 44033 30034 POLI 11201 DNA REPAIR AG-537 CHEMBL67535 44034 30035 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE SB-203580 SB-203580 17964780 44036 30036 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR PIRFENIDONE PIRFENIDONE 44037 30037 SLC40A1 30061 TRANSPORTER, DRUGGABLE GENOME Ferroportin mab 24552640 44038 30038 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME activator 135650163 44039 30039 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME ARC-1905 AVACINCAPTAD PEGOL SODIUM 44041 30040 KDM4A 9682 DRUGGABLE GENOME, ENZYME 3-MORPHOLINOSYDNONIMINE HCL CHEMBL538104 44042 30041 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME FLUOROURACIL FLUOROURACIL 23456958 44043 30042 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ARRY-614 PEXMETINIB 44044 30043 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-1935 CHEMBL588250 44045 30044 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME irinotecan IRINOTECAN 44046 30045 TUBA4A 7277 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 44050 30046 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE GW7647 GW7647 44051 30047 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL514800 APREMILAST 44053 30048 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE vincristine VINCRISTINE 22016816 44055 30049 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROMAZINE PROMAZINE 44056 30050 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME FLAVONE-8-ACETIC ACID 12930151 44057 30051 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-42 44058 30052 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody MM-151 44059 30053 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 5310655 CHEMBL408563 44062 30054 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR ARRY-300 ARRY-300 44063 30055 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417614 CHEMBL1567571 44064 30056 IDE 3416 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, ENZYME, PROTEASE OLEOYL DOPAMINE OLEOYL DOPAMINE 44068 30057 DGAT1 8694 ENZYME, DRUGGABLE GENOME P-7435 44069 30058 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME CHIR-99021 CHIR-99021 44070 30059 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE RP6530 44071 30060 MAPK7 5598 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR sorafenib SORAFENIB 20124951 44073 30061 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ALCLOMETASONE ALCLOMETASONE 44077 30062 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2008107444 44078 30063 HMMR 3161 KINASE, CELL SURFACE, DRUGGABLE GENOME fluorouracil FLUOROURACIL 44079 30064 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME PHA-767491 CHEMBL225519 44082 30065 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ZIRAM ZIRAM 44084 30066 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE phenylephrine PHENYLEPHRINE 26771271,25730298 44087 30067 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DS-7423 DS-7423 24504419 44088 30068 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER fluorouracil FLUOROURACIL 19696793 44089 30069 GMNN 51053 DRUGGABLE GENOME NSC-98938 CHEMBL1939691 44091 30070 KDM4A 9682 DRUGGABLE GENOME, ENZYME PIMOZIDE PIMOZIDE 44095 30071 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PACLITAXEL PACLITAXEL 19470925 44096 30072 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 363894222 PUQUITINIB 44097 30073 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor SF1126 44098 30074 XDH 7498 DRUGGABLE GENOME, ENZYME inhibitor 178103423 FEBUXOSTAT 44099 30075 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE TOZASERTIB TOZASERTIB 44100 30076 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE AZD-7762 AZD-7762 44102 30077 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-A6 44103 30078 MAPT 4137 DRUGGABLE GENOME GNF-PF-4300 CHEMBL585656 44104 30079 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TOLONIUM CHLORIDE TOLONIUM CHLORIDE 44106 30080 ATF2 1386 TRANSCRIPTION FACTOR TGFBETA1 16125722 44107 30081 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CYCLOSPORIN 11516824 44108 30082 GMNN 51053 DRUGGABLE GENOME THIOMERSAL THIMEROSAL 44109 30083 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME TCMDC-125758 CHEMBL546797 44110 30084 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME GW572016 LAPATINIB 16452223 44111 30085 KDM4A 9682 DRUGGABLE GENOME, ENZYME BI-87E7 CHEMBL523200 44112 30086 SMN1 6606 DRUGGABLE GENOME DNDI1417597 CHEMBL1330352 44114 30087 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker 135649825 5-BENZYLOXYTRYPTAMINE 44115 30088 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME rigosertib RIGOSERTIB 27104980 44116 30089 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE THYROXINE THYROXINE 10452218 44118 30090 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE ACTB1003 44120 30091 SQLE 6713 DRUGGABLE GENOME, ENZYME Tolnaftate TOLNAFTATE 44121 30092 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Lapatinib LAPATINIB 21464044,23365119 44123 30093 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1201124 KETOROLAC TROMETHAMINE 44124 30094 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist CHEMBL1358 FULVESTRANT 44125 30095 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ANGUSTIBALIN ANGUSTIBALIN 44126 30096 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ICI 118,551 44129 30097 ADH1A 124 DRUGGABLE GENOME abacavir ABACAVIR 24625462 44130 30098 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200473 CYCLOPENTOLATE HYDROCHLORIDE 44131 30099 PSMA7 5688 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL371405 MARIZOMIB 44133 30100 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist CHEMBL705 ALITRETINOIN 44134 30101 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME HMG-COA REDUCTASE INHIBITOR 12618273 44135 30102 MAPT 4137 DRUGGABLE GENOME PLUMBAGIN PLUMBAGIN 44136 30103 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 1,4-DIMETHOXYANTHRAQUINONE 1,4-DIMETHOXYANTHRAQUINONE 44144 30104 AKR1B1 231 DRUGGABLE GENOME, ENZYME TECTORIGENIN TECTORIGENIN 16870454 44146 30105 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Anisodamine ANISODAMINE 44147 30106 BCL2L11 10018 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR IMATINIB IMATINIB 22426421 44148 30107 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE inhibitor NITROGLYCERIN NITROGLYCERIN 44149 30108 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE FENTICLOR FENTICLOR 44150 30109 BAZ2B 29994 NA ELLAGIC ACID ELLAGIC ACID 44151 30110 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor ALVOCIDIB ALVOCIDIB 44152 30111 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051816 CHEMBL2153434 44153 30112 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NAFTOPIDIL NAFTOPIDIL 44154 30113 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME GO-6976 GO-6976 44155 30114 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650239 ERGOTAMINE 44157 30115 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OXYBUTYNIN OXYBUTYNIN 22931300 44158 30116 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CARMINIC ACID CARMINIC ACID 44159 30117 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GUTHION GUTHION 44160 30118 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1769 PROPOXYCAINE HYDROCHLORIDE 44161 30119 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR ROMIDEPSIN ROMIDEPSIN 44163 30120 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32v 44164 30121 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ANETHOLTRITHION ANETHOLTRITHION 44167 30122 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NITROFURANTOIN NITROFURANTOIN 22931300 44168 30123 PTK6 5753 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, ENZYME SB-202190 SB-202190 22951114 44169 30124 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8592455, 90 44170 30125 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ESTRONE ESTRONE 44171 30126 BCHE 590 DRUGGABLE GENOME, ENZYME Di-substituted piperidine derivative 3 44176 30127 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DIGOXIN DIGOXIN 44179 30128 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NITRILOTRIACETIC ACID NITRILOTRIACETIC ACID 44180 30129 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Torin 1 27974663 44182 30130 ABHD12 26090 ENZYME, DRUGGABLE GENOME, PHOSPHOLIPASE inhibitor 381744932 44183 30131 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ARGX-111 44184 30132 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SCOULERINE SCOULERINE 44185 30133 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PF-03715455 PF-03715455 21888439 44186 30134 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR GSK343 26676756 44187 30135 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-2895 CHEMBL524603 44190 30136 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33c 44192 30137 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor REGORAFENIB REGORAFENIB 44194 30138 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 187051798 BELINOSTAT 44196 30139 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZ628 27523909 44197 30140 HPSE 10855 ENZYME, DRUGGABLE GENOME HESPERIDIN HESPERIDIN 23415087 44198 30141 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE NEVIRAPINE NEVIRAPINE 12869587 44199 30142 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 44200 30143 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR URSODIOL URSODIOL 21158453 44201 30144 HSPA4 3308 NA DON 9142921 44203 30145 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor VATALANIB VATALANIB 44204 30146 BAZ2B 29994 NA NSC-601359 CHEMBL1306524 44206 30147 ADH1A 124 DRUGGABLE GENOME ethanol ALCOHOL 44207 30148 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME inhibitor BALICATIB BALICATIB 44208 30149 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-3403 CHEMBL602209 44210 30150 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ENPIROLINE ENPIROLINE 44213 30151 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR Trilostane TRILOSTANE 44214 30152 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DOPAMINE DOPAMINE 44215 30153 ITGB5 3693 CELL SURFACE, DRUGGABLE GENOME inhibitor 385612210 44216 30154 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME AZD-1152-HQPA AZD-1152-HQPA 44218 30155 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TYRPHOSTIN 51 TYRPHOSTIN 51 44219 30156 TUBA3C 7278 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 44220 30157 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200497 CYCLIZINE LACTATE 44222 30158 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL272621 HYODEOXYCHOLIC_ACID 44224 30159 OGA 10724 ENZYME, DRUGGABLE GENOME inhibitor 387065591 CHEMBL1213603 44225 30160 ATXN2 6311 NA TCMDC-123951 CHEMBL587849 44226 30161 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Cyclohexane carboxamide derivative 2 44227 30162 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR FLUDARABINE FLUDARABINE 44228 30163 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME AC-55649 CHEMBL425027 19239230 44229 30164 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL632 BETAMETHASONE 44230 30165 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ABBV-744 ABBV-744 44231 30166 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PS-178990 19079612 44232 30167 RAD21 5885 CLINICALLY ACTIONABLE N/A 15767545 44233 30168 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL119385 NEFLAMAPIMOD 44234 30169 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NSC-668394 CHEMBL336095 44236 30170 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME PMID27828716-Compound-18 44238 30171 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER DIHYDRO-12-HYDROXY-2,2-DIMETHYL-2H,6H-PYRANO[3,2-B]XANTHEN-6-ONE DIHYDRO-12-HYDROXY-2,2-DIMETHYL-2H,6H-PYRANO[3,2-B]XANTHEN-6-ONE 44244 30172 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR RAPAMYCIN SIROLIMUS 1284044 44246 30173 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME INK128 SAPANISERTIB 44250 30174 TRAF1 7185 NA infliximab INFLIXIMAB 23007924 44251 30175 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME VATALANIB VATALANIB 28759044 44253 30176 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist CHEMBL146032 LONAPRISAN 44254 30177 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METHIMAZOLE METHIMAZOLE 44255 30178 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE 2,2-dimethylbenzopyran derivative 3 44256 30179 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE CHEMBL1255944 44257 30180 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565590 CHEMBL1236539 44258 30181 GSTM1 2944 DRUGGABLE GENOME, ENZYME Platinum compounds 26803611 44260 30182 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545075 LAROTRECTINIB 44261 30183 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE MLN-8054 MLN-8054 44263 30184 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME aripiprazole lauroxil 44264 30185 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Cannabinoid quinone derivative 1 44265 30186 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200787 PHENOXYBENZAMINE HYDROCHLORIDE 44266 30187 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200952 METHAMPHETAMINE HYDROCHLORIDE 44267 30188 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ALENDRONATE ALENDRONIC ACID 12608943 44268 30189 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR LOVASTATIN LOVASTATIN 7600119 44269 30190 HSPA8 3312 TUMOR SUPPRESSOR HEXACHLOROPHENE HEXACHLOROPHENE 44270 30191 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Mercaptopurine MERCAPTOPURINE 28151717 44271 30192 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AZD9291 OSIMERTINIB 27252416 44272 30193 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 252827442 SGI-1776 44275 30194 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR FISETIN FISETIN 44276 30195 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER TRIMETREXATE TRIMETREXATE 10360822 44277 30196 ACO1 48 ENZYME ANTISERUM 8764614 44280 30197 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Apremilast APREMILAST 44282 30198 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LAPATINIB LAPATINIB 44283 30199 RGS17 26575 NA antidepressants 44284 30200 IL18 3606 DRUGGABLE GENOME Iboctadekin + Doxil 44285 30201 IL1B 3553 KINASE, DRUGGABLE GENOME Bisphosphonates 16257277 44286 30202 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME ALS 2-0426 44287 30203 TTC37 9652 NA duloxetine DULOXETINE 29407288 44288 30204 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ETHYLESTRENOL ETHYLESTRENOL 44289 30205 MASP2 10747 PROTEASE, DRUGGABLE GENOME, ENZYME OMS721 NARSOPLIMAB 44290 30206 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME RIDAFOROLIMUS RIDAFOROLIMUS 44291 30207 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE DIPHENOXYLATE DIPHENOXYLATE 44292 30208 SMN2 6607 DRUGGABLE GENOME CID 926663 CHEMBL265686 44294 30209 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR METHYSERGIDE METHYSERGIDE 44295 30210 SCNN1G 6340 ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TRIAMTERENE TRIAMTERENE 44296 30211 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME L-NOREPINEPHRINE L-NOREPINEPHRINE 44299 30212 PTGS1 5742 ENZYME, DRUGGABLE GENOME ETODOLAC ETODOLAC 44301 30213 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Indole-based analog 13 44302 30214 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE XL-147 PILARALISIB 44303 30215 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LOPERAMIDE LOPERAMIDE 44304 30216 XPA 7507 CLINICALLY ACTIONABLE, DNA REPAIR Platinum compounds 25069034 44307 30217 HSPA8 3312 TUMOR SUPPRESSOR ADENOSINE TRIPHOSPHATE ADENOSINE TRIPHOSPHATE 44308 30218 MAGEA3 4102 ENZYME, DRUGGABLE GENOME MAGE-A3 ASTUPROTIMUT-R 44309 30219 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE RIFAMPICIN RIFAMPIN 26291341 44310 30220 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME DIMETHYLSPINGOSINE DIMETHYLSPINGOSINE 19469544 44311 30221 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE AKT INHIBITOR MK2206 24504448 44313 30222 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Carboxyamidotriazole Orotate 44314 30223 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME TCMDC-125758 CHEMBL546797 44315 30224 THBS4 7060 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, GROWTH FACTOR VASOPRESSIN VASOPRESSIN 18541142 44317 30225 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CEP-11981 CEP-11981 22148921 44318 30226 VIM 7431 DRUGGABLE GENOME GELDANAMYCIN GELDANAMYCIN 16328963 44320 30227 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME caspofungin CASPOFUNGIN 15716364 44321 30228 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102778 CHEMBL422420 44323 30229 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR HYDROXYZINE PAMOATE HYDROXYZINE PAMOATE 44324 30230 IGFBP1 3484 DRUGGABLE GENOME SANDOSTATIN SANDOSTATIN 9420847 44328 30231 BAZ2B 29994 NA DOXYCYCLINE HYCLATE DOXYCYCLINE HYCLATE 44329 30232 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE Alisporivir ALISPORIVIR 44330 30233 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR L-161982 CHEMBL1179743 44332 30234 GJA1 2697 ION CHANNEL PROPYLTHIOURACIL PROPYLTHIOURACIL 12606457 44334 30235 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 135652593 BKT140 44335 30236 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PROTRIPTYLINE PROTRIPTYLINE 44337 30237 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE pyrazinamide PYRAZINAMIDE 22151084 44338 30238 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PAPAVERINE HYDROCHLORIDE PAPAVERINE HYDROCHLORIDE 44339 30239 KNG1 3827 DRUGGABLE GENOME, PROTEASE INHIBITOR Avoralstat AVORALSTAT 44341 30240 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200964 AMITRIPTYLINE HYDROCHLORIDE 44342 30241 ATAT1 79969 ENZYME carboplatin CARBOPLATIN 31616045 44343 30242 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME NIA-114 44344 30243 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHAPHIT METHAPHIT 44345 30244 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE 5-AZACYTIDINE AZACITIDINE 9006118 44346 30245 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZD5312 AZD-5312 44350 30246 TARDBP 23435 TUMOR SUPPRESSOR SIMVASTATIN SIMVASTATIN 44351 30247 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Vildagliptin VILDAGLIPTIN 44352 30248 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE Lumacaftor LUMACAFTOR 44353 30249 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME SUBEROHYDROXAMIC ACID SUBEROHYDROXAMIC ACID 16921367 44354 30250 USP1 7398 DNA REPAIR, PROTEASE, ENZYME VITAMIN B2 VITAMIN B2 44355 30251 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 252166602 NANATINOSTAT 44356 30252 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE inhibitor 249565818 44358 30253 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL TRICHLORMETHIAZIDE TRICHLORMETHIAZIDE 44359 30254 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR DIURETIC 8724667 44360 30255 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650354 44362 30256 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE BAFETINIB BAFETINIB 18191450 44364 30257 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE IODINE I-131 27493271 44365 30258 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CETUXIMAB CETUXIMAB 44366 30259 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor 328083506 44367 30260 XPO1 7514 CLINICALLY ACTIONABLE, KINASE inhibitor 375973225 ELTANEXOR 44368 30261 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ERGOCALCIFEROL ERGOCALCIFEROL 44370 30262 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CLORAZEPATE CLORAZEPIC ACID 44372 30263 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SALAGEN SALAGEN 44373 30264 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE C-Met/PD-L1 CAR-T Cell 44374 30265 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-108783 CHEMBL1489812 44375 30266 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME pazopanib PAZOPANIB 25504632 44376 30267 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE DES DIETHYLSTILBESTROL 15545218 44378 30268 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody MT110 SOLITOMAB 44379 30269 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor CHEMBL2386889 SCH-900776 44380 30270 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL482968 ENMD-2076 44382 30271 SLC25A1 6576 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101413 44383 30272 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PRAZOSIN PRAZOSIN 44384 30273 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178102339 SUNITINIB 44385 30274 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR MADOLIN T MADOLIN T 44386 30275 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE Lacosamide ERLOSAMIDE 44387 30276 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SB-216763 SB-216763 44389 30277 HBB 3043 DRUGGABLE GENOME, ENZYME TOPOTECAN HYDROCHLORIDE TOPOTECAN HYDROCHLORIDE 44390 30278 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR MITOTANE MITOTANE 44391 30279 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 310264738 CERDULATINIB 44394 30280 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 7 44395 30281 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL972 SELEGILINE 44396 30282 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHENELZINE PHENELZINE 22931300 44398 30283 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR LAUROGUADINE LAUROGUADINE 44399 30284 SGMS1 259230 ENZYME, KINASE inhibitor 375973242 44400 30285 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER nelfinavir NELFINAVIR 20662624,20860463,11809184,23734829,16267764,16912956 44401 30286 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR BRYOSTATIN BRYOSTATIN 22579485 44403 30287 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 178100604 44404 30288 IFNG 3458 DRUGGABLE GENOME 5'-DEOXY-5-FLUOROURIDINE 12553027 44405 30289 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 selegiline SELEGILINE 9187528 44406 30290 PDE1A 5136 ENZYME, DRUGGABLE GENOME inhibitor 178101953 44407 30291 IL15RA 3601 DRUGGABLE GENOME, CELL SURFACE BNZ-1 44408 30292 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DOFETILIDE DOFETILIDE 44409 30293 KLK4 9622 PROTEASE, DRUGGABLE GENOME, ENZYME Benzoxazinone derivative 2 44410 30294 MAPT 4137 DRUGGABLE GENOME GNF-PF-2298 CHEMBL578905 44413 30295 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR INDIGO INDIGO 44414 30296 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 135651578 THYMOL 44416 30297 DGAT1 8694 ENZYME, DRUGGABLE GENOME inhibitor 223366162 44417 30298 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Paclitaxel PACLITAXEL 24886365 44418 30299 HLA-DQB1 3119 CLINICALLY ACTIONABLE Drugs For Treatment Of Tuberculosis 25250564,12359646 44419 30300 BCL2L11 10018 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR KERACYANIN KERACYANIN 17360708 44420 30301 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME EVEROLIMUS EVEROLIMUS 26544513 44424 30302 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 178102308 CHEMBL525191 44425 30303 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL CLEVIDIPINE CLEVIDIPINE 44426 30304 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME RIMSULFURON RIMSULFURON 44427 30305 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PD-404182 CHEMBL595227 44428 30306 BCHE 590 DRUGGABLE GENOME, ENZYME HEXAFLURONIUM BROMIDE 44431 30307 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CALCIMYCIN CALCIMYCIN 44432 30308 CBX1 10951 NA TYRPHOSTIN 51 TYRPHOSTIN 51 44433 30309 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR HEXACHLOROPHENE HEXACHLOROPHENE 44435 30310 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000121257 CHEMBL592363 44437 30311 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME ARSENIC TRIOXIDE 15690072 44438 30312 AKR1C3 8644 ENZYME, DRUGGABLE GENOME daunorubicin DAUNORUBICIN 20837989 44439 30313 POLK 51426 DNA REPAIR, ENZYME IRETOL IRETOL 44441 30314 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME TETRACYCLINE TETRACYCLINE 19258275 44442 30315 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TRASTUZUMAB TRASTUZUMAB 44443 30316 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME DIPHENYLENEIODONIUM DIPHENYLENEIODONIUM 44444 30317 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME TEDATIOXETINE TEDATIOXETINE 44445 30318 NPEPPS 9520 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103847 TOSEDOSTAT 44446 30319 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR KAEMPFERIDE KAEMPFERIDE 25190466 44447 30320 DHFR 1719 DRUGGABLE GENOME, ENZYME PEMETREXED PEMETREXED 44448 30321 RAPGEF3 10411 ENZYME BAS03450373 CHEMBL1576310 44450 30322 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ZM-449829 CHEMBL154580 44453 30323 POLK 51426 DNA REPAIR, ENZYME QUERCITRIN QUERCITRIN 44454 30324 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME PHENTERMINE PHENTERMINE 44455 30325 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4300 CHEMBL585656 44456 30326 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME KETANSERIN KETANSERIN 44457 30327 MAPT 4137 DRUGGABLE GENOME CCT018159 CHEMBL399530 44458 30328 BAZ2B 29994 NA METERGOLINE METERGOLINE 44462 30329 POLL 27343 NA TALAROFLAVONE TALAROFLAVONE 18178092 44463 30330 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE HER1-VSSP vaccine 44464 30331 BRCA2 675 CLINICALLY ACTIONABLE CARBOPLATIN CARBOPLATIN 25847936 44465 30332 COL4A2 1284 DRUGGABLE GENOME AK107 44468 30333 POLK 51426 DNA REPAIR, ENZYME PYROGALLOL PYROGALLOL 44469 30334 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME TAMATINIB R-406 44470 30335 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME modulator CHEMBL3707374 AMISELIMOD HYDROCHLORIDE 44471 30336 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545096 BGT-226 44472 30337 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME ILORASERTIB ILORASERTIB 44475 30338 BAZ2B 29994 NA LUTEOLIN LUTEOLIN 44476 30339 APBA1 320 NA BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 44477 30340 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROROXAN HYDROCHLORIDE PROROXAN HYDROCHLORIDE 44478 30341 CUL4A 8451 ENZYME, DNA REPAIR, CLINICALLY ACTIONABLE inhibitor CHEMBL43452 POMALIDOMIDE 44480 30342 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SGI-1776 SGI-1776 44481 30343 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102284 MASITINIB 44483 30344 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 249565623 GEDATOLISIB 44484 30345 CARM1 10498 ENZYME, METHYL TRANSFERASE, DRUGGABLE GENOME inhibitor 178103610 44485 30346 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-48 44486 30347 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL RIMCAZOLE RIMCAZOLE 44489 30348 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 2 44490 30349 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME COAGULATION FACTOR VIIA 44492 30350 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TIBOLONE TIBOLONE 44493 30351 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor SORAFENIB TOSYLATE 44494 30352 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIELDRIN DIELDRIN 44498 30353 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE WARFARIN POTASSIUM WARFARIN POTASSIUM 44499 30354 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-30 44501 30355 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME RIBAVIRIN RIBAVIRIN 16104024 44502 30356 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR APICIDIN APICIDIN 19705846 44503 30357 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME PHENTERMINE PHENTERMINE 44504 30358 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME XP13512 GABAPENTIN ENACARBIL 44505 30359 CDC42BPA 8476 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LAUROGUADINE LAUROGUADINE 44507 30360 CEACAM1 634 KINASE, CELL SURFACE, DRUGGABLE GENOME ARCITUMOMAB ARCITUMOMAB 44508 30361 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650853 PRENALTEROL 44509 30362 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor PX-866 SONOLISIB 44510 30363 POLI 11201 DNA REPAIR LAVENDUSTIN C LAVENDUSTIN C 44511 30364 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME INAMRINONE INAMRINONE 44515 30365 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125606 CHEMBL536166 44517 30366 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL193 NIFEDIPINE 44518 30367 RACGAP1 29127 NA NSC-8186 CHEMBL122355 44520 30368 ALOX15 246 ENZYME, DRUGGABLE GENOME PSEUDOEPHEDRINE PSEUDOEPHEDRINE 44521 30369 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 3237815 CHEMBL410484 44522 30370 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE KW-2449 KW-2449 44523 30371 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME [3H]-PHORBOL 12,13-DIBUTYRATE CHEMBL27768 24794745 44524 30372 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CNS-7056 REMIMAZOLAM 44525 30373 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Promestriene PROMESTRIENE 44526 30374 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME S63845 27760111 44527 30375 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE GAP T cells 44528 30376 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME RUCAPARIB RUCAPARIB 44529 30377 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME AG-538 CHEMBL56393 44531 30378 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME 2-ENE-VALPROATE CHEMBL117487 17566732 44532 30379 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE CARBOPLATIN CARBOPLATIN 44534 30380 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PREDNISOLONE PREDNISOLONE 16324786 44535 30381 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR PROTON PUMP INHIBITOR 16815316 44536 30382 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE DERSALAZINE DERSALAZINE 44538 30383 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PICOTAMIDE PICOTAMIDE 44539 30384 TUBA1C 84790 DRUGGABLE GENOME CHEMBL2105643 FOSBRETABULIN TROMETHAMINE 44540 30385 PDE4A 5141 DRUGGABLE GENOME, ENZYME PENTOXIFYLLINE PENTOXIFYLLINE 44543 30386 KDM4A 9682 DRUGGABLE GENOME, ENZYME N-(2,4-DIMETHYLPHENYL)BENZENESULFONAMIDE CHEMBL492651 44544 30387 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 44549 30388 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALLANTOIN ALLANTOIN 44550 30389 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ESTROPIPATE ESTROPIPATE 44552 30390 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 252166793 44553 30391 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3545209 NKTR-171 44557 30392 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL723 CARVEDILOL 44558 30393 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROPIOMAZINE PROPIOMAZINE 44562 30394 ALDH1A1 216 DRUGGABLE GENOME, ENZYME HEMICHOLINIUM-3 HEMICHOLINIUM-3 44563 30395 UGT2B17 7367 ENZYME, DRUGGABLE GENOME ibuprofen IBUPROFEN 25502615 44564 30396 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME 2,4-DIHYDROXYBENZOPHENONE 2,4-DIHYDROXYBENZOPHENONE 44565 30397 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER IMIDAZOLE-CALIXARENE CHEMBL1801219 20605095 44566 30398 PDE4D 5144 DRUGGABLE GENOME, ENZYME TA-7906 44569 30399 EGR1 1958 NA GENIPIN GENIPIN 26283511 44570 30400 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Gefitinib GEFITINIB 44571 30401 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE antagonist 252166531 NAVITOCLAX 44573 30402 HCP5 10866 NA nevirapine NEVIRAPINE 24322967 44574 30403 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Anti-MUC1 CAR T Cells 44576 30404 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME KARANJIN KARANJIN 44578 30405 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102652 44582 30406 PSMD3 5709 NA BORTEZOMIB BORTEZOMIB 24524217 44583 30407 USP7 7874 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME, PROTEASE PMID26077642-Compound-Vif2 44584 30408 TUBA4A 7277 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 44586 30409 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME interferon alfa-2a, recombinant 12873589 44587 30410 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ARQ 751 26469692 44591 30411 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE Y-27632 Y-27632 17018693 44592 30412 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME VEL-0230 CHEMBL1085282 44593 30413 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Tetracaine TETRACAINE 44594 30414 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME Dasatinib DASATINIB 44595 30415 ATXN2 6311 NA NANAOMYCIN NANAOMYCIN 44596 30416 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist 249565881 GLASDEGIB 44598 30417 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A3 44600 30418 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE EGFRBi-armed autologous activated T cells 16397041 44601 30419 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Sorafenib SORAFENIB 26270481 44603 30420 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-25 44607 30421 GPR39 2863 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist 135652747 44609 30422 SLCO4C1 353189 TRANSPORTER, DRUGGABLE GENOME Digoxin DIGOXIN 44611 30423 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PMID28460551-Compound-2 44612 30424 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103980 ERIBAXABAN 44613 30425 ATAD5 79915 NA ZERANOL ZERANOL 44615 30426 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PERTUZUMAB PERTUZUMAB 31453370,22149875,30857956,29320312,25693012 44617 30427 ODC1 4953 DRUGGABLE GENOME, ENZYME inhibitor 178101866 EFLORNITHINE 44619 30428 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PF-562271 PF-00562271 44620 30429 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR T091317 T091317 44621 30430 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ONC201 ONC-201 26474387 44627 30431 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2107815 TREPROSTINIL DIOLAMINE 44628 30432 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-14 44629 30433 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NSC-19803 CHEMBL522983 44630 30434 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8759338, 1 44631 30435 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE entrectinib ENTRECTINIB 44632 30436 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME LY-2090314 LY-2090314 44634 30437 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NORETHINDRONE NORETHINDRONE 44637 30438 PDE1A 5136 ENZYME, DRUGGABLE GENOME inhibitor 178101968 VINPOCETINE 44639 30439 ALDH1A1 216 DRUGGABLE GENOME, ENZYME MICHLER'S KETONE MICHLER'S KETONE 44642 30440 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3545368 PANOBINOSTAT LACTATE 44645 30441 LEPR 3953 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Metreleptin METRELEPTIN 44646 30442 BPTF 2186 TRANSCRIPTION FACTOR inhibitor 252827533 44647 30443 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE BAY1000394 44648 30444 PER1 5187 TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE MELATONIN MELATONIN 15978008,12895514 44649 30445 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TOZASERTIB TOZASERTIB 44650 30446 CALR 811 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GLUCOCORTICOID 8910610,8107808 44652 30447 CFH 3075 DRUGGABLE GENOME TT-30 44653 30448 ATAD5 79915 NA GNF-PF-5251 CHEMBL576404 44654 30449 ANO1 55107 ION CHANNEL blocker 178100935 44655 30450 GMNN 51053 DRUGGABLE GENOME GNF-PF-5037 CHEMBL585828 44658 30451 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor 178101857 CILOSTAMIDE 44660 30452 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME ACID BLUE 129 ACID BLUE 129 44661 30453 TUBB 203068 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 44662 30454 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PMI-001 44664 30455 GMNN 51053 DRUGGABLE GENOME ENCLOMIPHENE CITRATE ENCLOMIPHENE CITRATE 44665 30456 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TAMSULOSIN TAMSULOSIN 44666 30457 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1700 SOTALOL HYDROCHLORIDE 44668 30458 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2105708 PONATINIB HYDROCHLORIDE 44669 30459 CBX1 10951 NA METHYLDOPA METHYLDOPA 44671 30460 TARDBP 23435 TUMOR SUPPRESSOR ESTRONE ESTRONE 44672 30461 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CETRIMONIUM BROMIDE CETRIMONIUM BROMIDE 44673 30462 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE prednisone PREDNISONE 44677 30463 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417809 CHEMBL1442783 44678 30464 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-516 CHEMBL602970 44680 30465 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME AZD-1775 ADAVOSERTIB 44684 30466 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR KINETIN RIBOSIDE KINETIN RIBOSIDE 44685 30467 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE ABACAVIR ABACAVIR 17172311 44687 30468 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CILENGITIDE CILENGITIDE 44689 30469 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME SMS 201-995 7628916 44690 30470 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor VORINOSTAT VORINOSTAT 44693 30471 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor DACOMITINIB DACOMITINIB 44694 30472 POLI 11201 DNA REPAIR PROSTAGLANDIN B1 PROSTAGLANDIN B1 44695 30473 ATXN2 6311 NA GNF-PF-159 CHEMBL599924 44698 30474 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 6-CHLOROMELATONIN CHEMBL34730 44699 30475 IL1A 3552 CELL SURFACE, DRUGGABLE GENOME AMG-108 AMG-108 44700 30476 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE Enzastaurin ENZASTAURIN 22253748 44701 30477 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Tetra-hydro-quinoline derivative 1 44703 30478 SMN2 6607 DRUGGABLE GENOME XANTHYLETIN XANTHYLETIN 44705 30479 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CLADRIN CLADRIN 44706 30480 PTPRD 5789 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE trandolapril TRANDOLAPRIL 26425837 44708 30481 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Dabrafenib DABRAFENIB 44711 30482 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME GNF-PF-3996 CHEMBL584458 44714 30483 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL649 NADOLOL 44716 30484 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE ONX 0801 44717 30485 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR inhibitor 249565779 44718 30486 GALNT18 374378 NA cisplatin CISPLATIN 27150640 44719 30487 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME SRT-1460 CHEMBL254156 18046409 44720 30488 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135650843 44722 30489 NF2 4771 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, DRUG RESISTANCE, KINASE SELUMETINIB SELUMETINIB 26359368 44723 30490 GPR87 53836 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650457 44724 30491 MAPT 4137 DRUGGABLE GENOME TOLONIUM CHLORIDE TOLONIUM CHLORIDE 44725 30492 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL PHENYTOIN PHENYTOIN 44726 30493 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LINOLEIC ACID LINOLEIC ACID 44727 30494 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SORAFENIB SORAFENIB 44728 30495 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417827 CHEMBL1363249 44730 30496 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE AZD8835 AZD-8835 26839307 44731 30497 HPSE 10855 ENZYME, DRUGGABLE GENOME AMODIAQUINE HYDROCHLORIDE AMODIAQUINE HYDROCHLORIDE 23415087 44735 30498 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE TAE-684 TAE-684 44736 30499 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565645 MK-2461 44737 30500 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RAPAMYCIN SIROLIMUS 15642745 44738 30501 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME inhibitor CHEMBL2108568 TREBANANIB 44739 30502 BAZ2B 29994 NA AG-494 CHEMBL56731 44740 30503 CTSE 1510 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166874 44741 30504 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL agonist 178103288 44742 30505 ATXN2 6311 NA EMETINE EMETINE 44743 30506 CDK16 5127 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 44745 30507 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME FASUDIL FASUDIL 44746 30508 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ACECLOFENAC ACECLOFENAC 44747 30509 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME HYDROGEN PEROXIDE 9624736 44750 30510 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Bosutinib BOSUTINIB 28416483 44752 30511 SOST 50964 DRUGGABLE GENOME AMG 167 23807838 44753 30512 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DIFLUPREDNATE DIFLUPREDNATE 44754 30513 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME PMID29130358-Compound-Figure16(9c) 44755 30514 KCNA7 3743 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL284348 DALFAMPRIDINE 44756 30515 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUFENACET FLUFENACET 44758 30516 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME VEMURAFENIB VEMURAFENIB 24265153 44759 30517 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TCMDC-123579 CHEMBL533954 44760 30518 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME ANTISENSE OLIGONUCLEOTIDES 10911621 44761 30519 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DYCLONINE DYCLONINE 44762 30520 SLC22A11 55867 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER methotrexate METHOTREXATE 26086825 44763 30521 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME Antivirals for treatment of HIV infections, combinations 22162992 44764 30522 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Camptosar CAMPTOSAR 18618574 44765 30523 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651361 44767 30524 HTT 3064 DRUGGABLE GENOME HARMALINE HARMALINE 44768 30525 MBNL1 4154 DRUGGABLE GENOME AZELAIC ACID AZELAIC ACID 44769 30526 ALDH1A1 216 DRUGGABLE GENOME, ENZYME AZEPANE AZEPANE 44770 30527 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DICLOFENAC DICLOFENAC 22931300 44771 30528 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE CENISERTIB CENISERTIB 44772 30529 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Ganetespib GANETESPIB 26009011 44774 30530 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME PHORBOL MYRISTATE ACETATE 8503863 44775 30531 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-93 44776 30532 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ALAZANINE ALAZANINE 44778 30533 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TYRPHOSTIN AG-1478 TYRPHOSTIN AG-1478 44779 30534 MPHOSPH8 54737 NA CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 44780 30535 PSMD2 5708 NA inhibitor CHEMBL2103884 OPROZOMIB 44784 30536 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor AT9283 AT-9283 44785 30537 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME inhibitor 405560408 44786 30538 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE 7-azaindole derivative 7 44787 30539 FAAH 2166 ENZYME, DRUGGABLE GENOME Isoxazoline derivative 4 44788 30540 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME NV-52 44789 30541 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-628 CHEMBL1448140 44790 30542 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME PHA-767491 CHEMBL225519 44792 30543 DPYS 1807 ENZYME fluorouracil FLUOROURACIL 26244261 44793 30544 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR BACILLUS CALMETTE-GUERIN 14742634 44795 30545 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (+)-9-DEMETHYLELEUTHERIN CHEMBL594695 19783445 44796 30546 CLU 1191 CELL SURFACE, DRUGGABLE GENOME inhibitor OGX-011 CUSTIRSEN SODIUM 44797 30547 POLI 11201 DNA REPAIR AMPICILLIN AMPICILLIN 44798 30548 ALDH1A1 216 DRUGGABLE GENOME, ENZYME RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 44799 30549 DMD 1756 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME eteplirsen ETEPLIRSEN 44802 30550 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PEG-DOCETAXEL 44803 30551 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8987457, 117 44804 30552 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GANAXOLONE GANAXOLONE 44805 30553 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200434 OXTRIPHYLLINE 44806 30554 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE MLN1117 SERABELISIB 44807 30555 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 44808 30556 MAOB 4129 DRUGGABLE GENOME, ENZYME PIPERINE PIPERINE 44809 30557 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650342 GSK-9578 44810 30558 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL538943 VINORELBINE TARTRATE 44812 30559 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor 374883879 44815 30560 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE 178101565 44818 30561 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-36 44819 30562 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME inhibitor 384403662 44822 30563 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME oxcarbazepine OXCARBAZEPINE 27666425 44824 30564 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565632 AT-9283 44825 30565 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CAPTAN CAPTAN 44826 30566 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX ANDROGRAPHOLIDE ANDROGRAPHOLIDE 22026410 44830 30567 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE inhibitor 315661293 IVOSIDENIB 44832 30568 PLIN3 10226 NA IDURSULFASE IDURSULFASE 44834 30569 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CEFDITORIN PIVOXIL CEFDITORIN PIVOXIL 44835 30570 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GW441756X GW441756X 44838 30571 BAZ2B 29994 NA TRIAZOLAM TRIAZOLAM 22137933 44839 30572 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE larotrectinib sulfate 44840 30573 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AMG 337 26432108 44841 30574 RACGAP1 29127 NA LASSBIO-1183 CHEMBL1173141 44842 30575 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 310264722 44843 30576 AKR1C3 8644 ENZYME, DRUGGABLE GENOME Indomethacin analog 1 44844 30577 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL3545213 BENTAMAPIMOD 44847 30578 MAPT 4137 DRUGGABLE GENOME TCMDC-125286 CHEMBL533965 44848 30579 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AMPICILLIN AMPICILLIN 44849 30580 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR REL-BENDIGOLE E CHEMBL1915270 21684166 44850 30581 CSF1 1435 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PLX73086 44851 30582 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL565612 SOTRASTAURIN 44852 30583 SMN2 6607 DRUGGABLE GENOME INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 44853 30584 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PROPANTHELINE BROMIDE PROPANTHELINE BROMIDE 44856 30585 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650596 METHYSERGIDE 44857 30586 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME ABT-494 UPADACITINIB 44858 30587 CCL4 6351 DRUGGABLE GENOME CYCLOSPORIN A 15153516 44859 30588 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor XL820 44860 30589 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PERPHENAZINE PERPHENAZINE 44861 30590 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 249565740 AMG-900 44863 30591 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-50 44864 30592 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CHEMBL220492 TOPIRAMATE 44865 30593 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ROTENONE ROTENONE 44866 30594 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 44867 30595 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME tranilast TRANILAST 19364970,19852077,18349289,12181437,17058217,12969965,1651156,18466101,14647407,20562211,19390945,17728214,12019197,10381366,11037804 44868 30596 EML4 27436 CLINICALLY ACTIONABLE, KINASE Ceritinib CERITINIB 26775591,27009859,25173427,27432227,25228534,26698910,27780853,24675041 44869 30597 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 252166558 44870 30598 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178102302 CANERTINIB 44871 30599 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME TCMDC-125764 CHEMBL586670 44872 30600 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor PANOBINOSTAT PANOBINOSTAT 44875 30601 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Anti-C-met CAR-T cells 44876 30602 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 315661256 REBASTINIB 44880 30603 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE CAL-101 IDELALISIB 44881 30604 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE NI-0401 FORALUMAB 44882 30605 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NU-1025 CHEMBL123904 44883 30606 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor PIVANEX AN-9 44885 30607 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CURCUMIN CURCUMIN 20666513,23601707 44886 30608 GMNN 51053 DRUGGABLE GENOME PODOFILOX PODOFILOX 44887 30609 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BTCP CHEMBL279556 44888 30610 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL3084748 TROSPIUM CHLORIDE 44889 30611 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor CHEMBL1230607 PHA-793887 44890 30612 PSMA2 5683 DRUGGABLE GENOME, PROTEASE inhibitor BORTEZOMIB BORTEZOMIB 44893 30613 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Gefitinib GEFITINIB 22323597 44895 30614 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME SENNOSIDE B SENNOSIDE B 44897 30615 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER sorafenib SORAFENIB 44898 30616 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 363894217 VORUCICLIB 44900 30617 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist 178100909 44901 30618 HNMT 3176 ENZYME, DRUGGABLE GENOME Metoprine METOPRINE 44902 30619 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID27172114-Compound-30 44905 30620 PSMB6 5694 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL451887 CARFILZOMIB 44906 30621 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Sulfonamide derivative 8 44907 30622 LGR6 59352 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100586 44909 30623 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 44912 30624 CA1 759 DRUGGABLE GENOME, ENZYME CG-100649 POLMACOXIB 44913 30625 AKR1B10 57016 DRUGGABLE GENOME, ENZYME OLEANOLIC_ACID OLEANOLIC_ACID 21561086 44914 30626 RGS4 5999 DRUGGABLE GENOME FLUPIRTINE FLUPIRTINE 44915 30627 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MK-2461 MK-2461 44917 30628 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 EMBELIN EMBELIN 44919 30629 TNKS 8658 DRUGGABLE GENOME, ENZYME inhibitor 404859118 44920 30630 HTT 3064 DRUGGABLE GENOME SNDX-275 ENTINOSTAT 44921 30631 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME AMOXAPINE AMOXAPINE 44922 30632 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR PMID25980951-Compound-44 44923 30633 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 44925 30634 REEP5 7905 NA citalopram CITALOPRAM 22795047 44926 30635 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LACTOFEN LACTOFEN 44927 30636 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER LASSBIO-294 CHEMBL233194 44930 30637 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CYCLIRAMINE MALEATE CYCLIRAMINE MALEATE 44932 30638 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL272980 MOCETINOSTAT 44933 30639 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CINNAMALDEHYDE CINNAMALDEHYDE 44934 30640 TSLP 85480 DRUGGABLE GENOME MEDI9929 44936 30641 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652448 44938 30642 GMNN 51053 DRUGGABLE GENOME GNF-PF-67 CHEMBL578512 44942 30643 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME LEFLUNOMIDE LEFLUNOMIDE 16762150 44943 30644 GAA 2548 DRUGGABLE GENOME, ENZYME GOSSYPOL GOSSYPOL 44944 30645 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1237104 PROPOXYPHENE HYDROCHLORIDE 44945 30646 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR REV131 44946 30647 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GUANIDINONALTRINDOLE GUANIDINONALTRINDOLE 44947 30648 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME TG100801 44948 30649 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR METITEPINE METITEPINE 44949 30650 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE DALOTUZUMAB DALOTUZUMAB 44950 30651 TOP2B 7155 DRUGGABLE GENOME, ENZYME Doxorubicin-eluting beads 44951 30652 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TAZAROTENE TAZAROTENE 44952 30653 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE IMATINIB IMATINIB 44953 30654 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 3,4-DIMETHOXYDALBERGIONE 3,4-DIMETHOXYDALBERGIONE 44954 30655 CDC25C 995 KINASE, PROTEIN PHOSPHATASE, DRUGGABLE GENOME 5-FU FLUOROURACIL 9743457 44955 30656 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PRAZOSIN PRAZOSIN 12095132 44956 30657 LINGO1 84894 DRUGGABLE GENOME antibody 310264704 OPICINUMAB 44957 30658 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME NALED NALED 44958 30659 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 5 44959 30660 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CUMENE HYDROPEROXIDE CUMENE HYDROPEROXIDE 44960 30661 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RS-67506 CHEMBL83899 44961 30662 ATAD5 79915 NA BIX-01294 CHEMBL569864 44962 30663 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 7 44964 30664 COMT 1312 DRUGGABLE GENOME, ENZYME olanzapine OLANZAPINE 44965 30665 COMT 1312 DRUGGABLE GENOME, ENZYME catecholamines 44966 30666 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME PMID27998201-Compound-17 44967 30667 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Peptidomimetic analog 7 44968 30668 APBB1 322 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING COH29 COH-29 44970 30669 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME taxanes 26194361 44971 30670 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 252827399 RESVERATROL 44973 30671 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 2-AMINOETHOXYDIPHENYL BORATE CHEMBL169233 44974 30672 KDM4A 9682 DRUGGABLE GENOME, ENZYME Disulfiram analog 2 44976 30673 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650652 44977 30674 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PHENYLEPHRINE HYDROCHLORIDE PHENYLEPHRINE HYDROCHLORIDE 44980 30675 ANXA5 308 KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER Diannexin 44981 30676 TSPO 706 DRUGGABLE GENOME Aryl oxyanilide derivative 2 44982 30677 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE inhibitor 252827534 44983 30678 CA1 759 DRUGGABLE GENOME, ENZYME METHAZOLAMIDE METHAZOLAMIDE 44984 30679 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR calcium CALCIUM 10692979,17274004,10707958,12608943,9933478,21418277,18443790,15861036,19020788,15739035,12162507 44985 30680 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178100901 44986 30681 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME IMIPRAMINE IMIPRAMINE 44988 30682 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE FLOXURIDINE FLOXURIDINE 44991 30683 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE inhibitor 354702209 TRODUSQUEMINE 44992 30684 PTGS2 5743 DRUGGABLE GENOME, ENZYME VACCINE 17159912 44994 30685 CSK 1445 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor 252827493 44995 30686 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DEXBROMPHENIRAMINE DEXBROMPHENIRAMINE 44996 30687 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CLINAFLOXACIN CLINAFLOXACIN 44997 30688 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 22 44998 30689 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME ASP015K PEFICITINIB 45000 30690 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME PF-06439535 45003 30691 TSPO 706 DRUGGABLE GENOME Imidazopyridine acetamide analog 1 45004 30692 LTBR 4055 DRUGGABLE GENOME Baminercept BAMINERCEPT 45006 30693 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 4-METHYL-[1,10]PHENANTHROLINE CHEMBL316589 45007 30694 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Naphthyridine and isoquinoline derivative 1 45008 30695 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE R763 45009 30696 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FASUDIL FASUDIL 45010 30697 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-45382 CHEMBL1214274 45011 30698 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CI-1033 CANERTINIB 45012 30699 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME CLOMIPRAMINE CLOMIPRAMINE 45013 30700 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME Patisiran PATISIRAN 45014 30701 ANO1 55107 ION CHANNEL blocker 53801058 MIBEFRADIL 45015 30702 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor SOPHORETIN QUERCETIN 45016 30703 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METOLACHOR METOLACHOR 45021 30704 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-101 45022 30705 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IMIDAZOLE ACETIC ACID IMIDAZOLE ACETIC ACID 45023 30706 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME romidepsin ROMIDEPSIN 27443263 45024 30707 POLI 11201 DNA REPAIR ALPHA,BETA-DEHYDROCURVULARIN CHEMBL482050 45027 30708 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL citalopram CITALOPRAM 19388002 45028 30709 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3,5-dimethyl-2-(3-pyridyl)thiazolidin-4-one 8627557,19075994,10087035 45029 30710 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX HEXACHLOROPHENE HEXACHLOROPHENE 45030 30711 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CYCLOHEXIMIDE CYCLOHEXIMIDE 45031 30712 PYGL 5836 DRUGGABLE GENOME, ENZYME asparaginase ASPARAGINASE 23007406 45033 30713 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-292213 CHEMBL222808 45034 30714 PRF1 5551 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Emapalumab-lzsg EMAPALUMAB 45035 30715 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE AROMATASE INHIBITOR 11577780 45036 30716 IL23A 51561 DRUGGABLE GENOME Ustekinumab USTEKINUMAB 45037 30717 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 249565576 ENMD-2076 45039 30718 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE IMATINIB IMATINIB 15517875 45040 30719 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE KENPAULLONE KENPAULLONE 45042 30720 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2364614 LIAFENSINE 45043 30721 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 178103584 45044 30722 GMNN 51053 DRUGGABLE GENOME 1-(4-HYDROXYPHENYL)MALEIMIDE CHEMBL565893 45045 30723 CYB5R4 51167 DRUGGABLE GENOME rasburicase RASBURICASE 45046 30724 MGLL 11343 DRUGGABLE GENOME, ENZYME inhibitor 375973250 45047 30725 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CEPHALOCHROMIN CEPHALOCHROMIN 45048 30726 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 249565824 45050 30727 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 2-AMINOANTHRACENE 2-AMINOANTHRACENE 45052 30728 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Organon ORGANON 45053 30729 POLK 51426 DNA REPAIR, ENZYME CATECHOL CATECHOL 45054 30730 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C11 45055 30731 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-H3 45056 30732 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200637 DEXAMETHASONE SODIUM PHOSPHATE 45057 30733 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 178102615 45058 30734 MSH6 2956 CLINICALLY ACTIONABLE, DNA REPAIR KU60648 28224663 45059 30735 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL608533 MIDOSTAURIN 45060 30736 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100327 45062 30737 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 315661323 NAQUOTINIB 45063 30738 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME NSC-69187 CHEMBL19954 45065 30739 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE N-PHENYLMALEIMIDE CHEMBL76012 45069 30740 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102614 45070 30741 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ALPRENOLOL ALPRENOLOL 45071 30742 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ABBV-221 45072 30743 MAPT 4137 DRUGGABLE GENOME GNF-PF-1399 CHEMBL578504 45073 30744 KDM4A 9682 DRUGGABLE GENOME, ENZYME MMV006389 CHEMBL586000 45074 30745 GUCA2A 2980 DRUGGABLE GENOME, ENZYME, HORMONE ACTIVITY SALT VOLANESORSEN SODIUM 10564101 45075 30746 SGK3 23678 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ION CHANNEL, TRANSPORTER, ENZYME inhibitor 328083523 45076 30747 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HYDROXYTOLUIC ACID HYDROXYTOLUIC ACID 45077 30748 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GITOXIN GITOXIN 45084 30749 BAZ2B 29994 NA SJ000117447 CHEMBL592611 45085 30750 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 223366050 SAPITINIB 45086 30751 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2108208 LENERCEPT 45087 30752 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 QUINACRINE DIHYDROCHLORIDE QUINACRINE DIHYDROCHLORIDE 45089 30753 PTGES 9536 DRUGGABLE GENOME, ENZYME PMID28627961-Compound-33 45090 30754 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROTEASE INHIBITORS 12441344 45091 30755 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Isoproterenol ISOPROTERENOL 45092 30756 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FLUPIRTINE FLUPIRTINE 45094 30757 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE GLYCAR T cells 45095 30758 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PHENSERINE TARTRATE 45097 30759 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GW282974X GW282974X 45098 30760 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650585 METHOCTRAMINE 45099 30761 MAP3K5 4217 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, ENZYME inhibitor 385612190 45100 30762 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE SUNITINIB SUNITINIB 45102 30763 ATAD5 79915 NA 5-NITRO-[1,10]PHENANTHROLINE CHEMBL101815 45104 30764 PTGS1 5742 ENZYME, DRUGGABLE GENOME DICLOFENAC DICLOFENAC 45105 30765 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor BGJ398 INFIGRATINIB 45106 30766 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CAPTAN CAPTAN 45107 30767 ALOX15 246 ENZYME, DRUGGABLE GENOME DIHYDROGAMBOGIC ACID DIHYDROGAMBOGIC ACID 45108 30768 PTGS2 5743 DRUGGABLE GENOME, ENZYME Carprofen CARPROFEN 45110 30769 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IMAZODAN IMAZODAN 45111 30770 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ribavirin RIBAVIRIN 45112 30771 MPHOSPH8 54737 NA CEPHALOSPORIN C ZINC SALT CEPHALOSPORIN C ZINC SALT 45113 30772 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Phthalazine ketone derivative 1 45114 30773 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Aminobenzoxazole analog 1 45115 30774 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SOTALOL SOTALOL 2903243 45117 30775 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME PMID27774824-Compound-Figure9Example2down 45119 30776 MDK 4192 GROWTH FACTOR, DRUGGABLE GENOME, KINASE RETINOIC ACID 1819274 45122 30777 KLK6 5653 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 252166855 45123 30778 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL49642 INDIBULIN 45124 30779 KMO 8564 DRUGGABLE GENOME, ENZYME Aryl pyrimidine derivative 8 45126 30780 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL698 TETRACAINE 45128 30781 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR BDBM50158703 45130 30782 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE inhibitor 1372540-25-4 GSK-2636771 45131 30783 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE GO-6976 GO-6976 45132 30784 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR SNS-314 SNS-314 45133 30785 TGFA 7039 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME LY3016859 45134 30786 DAPK1 1612 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 135652717 STAUROSPORINE 45135 30787 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ONO-5129 45139 30788 RHEB 6009 TUMOR SUPPRESSOR, DRUG RESISTANCE, KINASE, CLINICALLY ACTIONABLE 4,4'-HYDROXYBIPHENYL CHEMBL76398 24266771 45140 30789 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor SOPHORETIN QUERCETIN 45142 30790 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE AZAKENPAULLONE AZAKENPAULLONE 45143 30791 COL27A1 85301 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 45144 30792 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE BIFONAZOLE BIFONAZOLE 45145 30793 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME inhibitor 252166814 45146 30794 CYP27B1 1594 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SOY PROTEIN 12421875 45147 30795 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME GNF-PF-5159 CHEMBL1493528 45148 30796 MAPT 4137 DRUGGABLE GENOME GALLIC ACID GALLIC ACID 45149 30797 CASP8 841 DRUGGABLE GENOME, PROTEASE, ENZYME, CLINICALLY ACTIONABLE ISOQUINOLINE-1,3(2H,4H)-DIONE CHEMBL1210769 45150 30798 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SODIUM LAURYL SULFATE SODIUM LAURYL SULFATE 45151 30799 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 178103534 TAZAROTENE 45152 30800 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Docetaxel DOCETAXEL 45154 30801 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME XEN1101 45155 30802 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER (S)APOMORPHINE (S)APOMORPHINE 45156 30803 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 fluorouracil FLUOROURACIL 15940289,19238117,18698229,16378601,19921195,20155256,21494765,19604090,21521021,14981342 45157 30804 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-22 45158 30805 NCAM1 4684 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE duloxetine DULOXETINE 28696415 45159 30806 UGCG 7357 ENZYME, DRUGGABLE GENOME Miglustat MIGLUSTAT 45161 30807 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME CEDIRANIB CEDIRANIB 45162 30808 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY ANTIDEPRESSANT 8895943 45163 30809 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR aspirin ASPIRIN 19138248 45166 30810 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor AZD4547 45167 30811 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL VERAPAMIL VERAPAMIL 45168 30812 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ATROPINE ATROPINE 45169 30813 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL activator 135651446 ADENOSINE TRIPHOSPHATE 45172 30814 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE NAC ACETYLCYSTEINE 15629104 45173 30815 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE BMS-599626 AC-480 45174 30816 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PHLORETIN PHLORETIN 45175 30817 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME GNF-PF-5510 CHEMBL578741 45176 30818 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545283 RIVICICLIB 45178 30819 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CIS-RESVERATROL CIS-RESVERATROL 45179 30820 PTPRZ1 5803 PROTEIN PHOSPHATASE, DRUGGABLE GENOME RETINOIC ACID 10809755 45180 30821 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR ARA-C 10930419 45181 30822 DYRK2 8445 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR HARMINE HARMINE 45182 30823 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL RAUWOLFIA SERPENTINA ROOT 45183 30824 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PLUMBAGIN PLUMBAGIN 24355130 45184 30825 FHIT 2272 CLINICALLY ACTIONABLE, ENZYME, TRANSPORTER interferon beta-1b 27001119 45186 30826 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR INTERLEUKIN 1 8382509 45187 30827 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME CAR-T cells targeting CEA 45190 30828 PTGS1 5742 ENZYME, DRUGGABLE GENOME latanoprost LATANOPROST 25339146 45191 30829 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE AZD8186 AZD-8186 25544636,25514658 45192 30830 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME CAPSAICIN CAPSAICIN 9138695 45193 30831 GALNT14 79623 ENZYME sorafenib SORAFENIB 31611591 45195 30832 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545322 PANULISIB 45197 30833 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Meglitinides 45198 30834 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE CHEMBL201325 45200 30835 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure1-Chukrasone A 45202 30836 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME efavirenz EFAVIRENZ 23859571 45203 30837 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LOBARIC ACID LOBARIC ACID 45204 30838 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR BACLOFEN BACLOFEN 17074039 45205 30839 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME temozolomide TEMOZOLOMIDE 24444404 45206 30840 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 3,5-DICHLORO-BENZOIC ACID CHEMBL118280 45209 30841 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1201467 SYNTHETIC CONJUGATED ESTROGENS, B 45210 30842 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX IONOMYCIN IONOMYCIN 16051191,9705872 45211 30843 GJB4 127534 ION CHANNEL inhibitor 178100972 CARBENOXOLONE 45213 30844 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LINIFANIB LINIFANIB 45214 30845 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR NICOTINE NICOTINE 16790237 45216 30846 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ALSTERPAULLONE ALSTERPAULLONE 45217 30847 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor NINTEDANIB NINTEDANIB 45218 30848 RHOA 387 KINASE, CLINICALLY ACTIONABLE CLAUSINE E CLAUSINE E 22093759 45219 30849 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DESOXYCORTICOSTERONE DESOXYCORTICOSTERONE 45220 30850 TUBA3D 113457 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 45222 30851 SFTPA1 653509 DRUGGABLE GENOME ALBUMIN ALBUMIN HUMAN 1314502 45223 30852 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-WO2009018344C79 45225 30853 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CHLORPROTHIXENE CHLORPROTHIXENE 45226 30854 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME REOLYSIN PELAREOREP 45227 30855 APOE 348 DRUGGABLE GENOME BPDE 14753754 45228 30856 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE PARABEN PARABEN 45229 30857 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE SUNITINIB SUNITINIB 45230 30858 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 387065624 45232 30859 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME XL518 COBIMETINIB 45233 30860 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL451887 CARFILZOMIB 45234 30861 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178102605 CHEMBL406375 45235 30862 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1501 FLUOCINONIDE 45236 30863 IGFBP1 3484 DRUGGABLE GENOME RAPAMYCIN SIROLIMUS 11942857 45239 30864 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME methoxyflurane METHOXYFLURANE 25989378,12411786,26951757,8828983,19919814,17710899,7829078,9334205,21965348,11063719,10823104,20681998,25611019,19648156,25256590,12220451,11668625,23736090,14500992,9066328,14641996,18945287,25960145,7889656,11575529,18212565,16284304,8602662,18306019,28326467,11928716,18502356,10352931,12151923,11525881,17122579,16917943,8220422,10700782,16163667,17226826,9389851,16732128,16835904,11448278,29101530,9450902,7547049,23628358,9543323,24361844,26994242,12208234,15448513,16621918,21455645,11553045,12124989,19020143,19191329,27918309,8220423,12059893,10612851,16732084,10793526,27382027,15108991,12709367,12123492,26381711,25268394,28063098,11493496,12434264,12411788,19685112,25735680,8902717,29608462,27663056,7751854,8012359,9520251,15731587,15210166,1510267,10888602,22030266,25466363,17483490,28403410,12237752,1774074,17081152,18564801,10484775,21282829,16244001,7586638,19191333,25086907,7633940,17667581,12883402,19346234,1354642,22415532 45241 30865 GMNN 51053 DRUGGABLE GENOME DNDI1416985 CHEMBL593211 45243 30866 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL2110814 DELUCEMINE 45244 30867 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-31 45245 30868 POLI 11201 DNA REPAIR SJ000244629 CHEMBL592115 45247 30869 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL2109482 BI-505 45249 30870 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NORFLOXACIN NORFLOXACIN 45251 30871 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL Dalazatide DALAZATIDE 45253 30872 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Solanezumab SOLANEZUMAB 45255 30873 POLI 11201 DNA REPAIR GNF-PF-4384 CHEMBL602763 45256 30874 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Topotecan TOPOTECAN 25833835 45258 30875 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE IBRUTINIB IBRUTINIB 45259 30876 LOX 4015 ENZYME, DRUGGABLE GENOME inhibitor 385612244 45260 30877 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ROTTLERIN ROTTLERIN 45261 30878 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ACEQUINOCYL ACEQUINOCYL 45263 30879 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE VITAMIN C 9834927 45265 30880 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-390527 CHEMBL160937 45266 30881 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 HYDRALAZINE HYDRALAZINE 22931300 45267 30882 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL OXAZEPAM OXAZEPAM 45268 30883 CDK12 51755 KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR, SERINE THREONINE KINASE Nivolumab NIVOLUMAB 45269 30884 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE TAE-684 TAE-684 45271 30885 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RO6839921 45272 30886 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE abemaciclib ABEMACICLIB 45273 30887 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL197672 EMRICASAN 45274 30888 FAAH 2166 ENZYME, DRUGGABLE GENOME IPI-940 45275 30889 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE artesunate ARTESUNATE 45276 30890 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME FRAXINE FRAXINE 45277 30891 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL113461 TEDISAMIL 45278 30892 UGT1A6 54578 ENZYME, DRUGGABLE GENOME doxorubicin DOXORUBICIN 45279 30893 NNMT 4837 DRUGGABLE GENOME NIACIN NIACIN 45280 30894 IL23A 51561 DRUGGABLE GENOME USTEKINUMAB USTEKINUMAB 45281 30895 PLD1 5337 ENZYME, DRUGGABLE GENOME PHORBOL MYRISTATE ACETATE 9989263 45282 30896 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DAPH DAPH 45284 30897 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR NALOXONE NALOXONE 12359151 45285 30898 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 5-AMINOISOQUINOLINE CHEMBL216973 45286 30899 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE MESALAMINE MESALAMINE 45287 30900 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 3-METHOXY-MORPHANIN HCL CHEMBL1257022 45288 30901 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR GLUCAGON GLUCAGON 17924870 45289 30902 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE antibody 375973255 45290 30903 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650882 RAGAGLITAZAR 45291 30904 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE DS-7423 DS-7423 45292 30905 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL697 METHSUXIMIDE 45294 30906 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR CREMOPHOR 9352228 45295 30907 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor AMUVATINIB AMUVATINIB 45296 30908 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CIANIDANOL CIANIDANOL 45298 30909 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor CHEMBL3137320 TALAZOPARIB 45299 30910 POLI 11201 DNA REPAIR ERBSTATIN ERBSTATIN 45300 30911 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor AXITINIB AXITINIB 45301 30912 HKDC1 80201 DRUGGABLE GENOME, KINASE ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 45302 30913 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE Imatinib IMATINIB 26861905 45303 30914 CSF3 1440 GROWTH FACTOR, DRUGGABLE GENOME SPI-2012 EFLAPEGRASTIM 45304 30915 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME OXYMETHOLONE OXYMETHOLONE 1009362 45305 30916 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-1969 CHEMBL601364 45306 30917 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR TDR77225 CHEMBL1353528 45308 30918 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW559768X GW559768X 45310 30919 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MINOCYCLINE MINOCYCLINE 22931300 45311 30920 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MERCURIC IODIDE MERCURIC IODIDE 45315 30921 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ATHRAQUINONES A ATHRAQUINONES A 45316 30922 EGFL7 51162 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE antibody MEGF0444A PARSATUZUMAB 45318 30923 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TAE-684 TAE-684 45320 30924 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 384403667 45321 30925 CA7 766 DRUGGABLE GENOME, ENZYME activator 178101506 AMPHETAMINE 45322 30926 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR medroxyprogesterone MEDROXYPROGESTERONE ACETATE 9860300 45327 30927 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE granisetron GRANISETRON 27809336 45328 30928 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DICUMAROL DICUMAROL 45330 30929 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR exemestane EXEMESTANE 45331 30930 LAMB1 3912 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 45332 30931 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME ENTINOSTAT ENTINOSTAT 19966789,18381238,20491440 45333 30932 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME GLUCOCORTICOID 12887795,12639897 45335 30933 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER FLUOROURACIL FLUOROURACIL 45336 30934 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HYDROQUINONE HYDROQUINONE 45337 30935 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651331 XANOMELINE 45338 30936 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 336446957 45339 30937 GAA 2548 DRUGGABLE GENOME, ENZYME ISOQUERCETIN ISOQUERCETIN 45340 30938 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME CTP-543 45342 30939 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE 5-FU FLUOROURACIL 22336586 45343 30940 UGT2B7 7364 DRUGGABLE GENOME atorvastatin ATORVASTATIN 45344 30941 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR docetaxel DOCETAXEL 25495407 45346 30942 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102575 45347 30943 PTGS1 5742 ENZYME, DRUGGABLE GENOME HYDROCHLOROTHIAZIDE HYDROCHLOROTHIAZIDE 11703585 45349 30944 PSMB4 5692 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL3545432 IXAZOMIB CITRATE 45350 30945 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME NITAZOXANIDE NITAZOXANIDE 45351 30946 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER LY3009120 LY-3009120 26343583 45353 30947 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Benzanilide compound 2 45355 30948 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE LATREPIRDINE LATREPIRDINE 45358 30949 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-234945 CHEMBL260311 45360 30950 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-69187 CHEMBL19954 45361 30951 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR LOMUSTINE LOMUSTINE 23904111 45363 30952 HYKK 123688 KINASE varenicline VARENICLINE 45365 30953 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ketoconazole KETOCONAZOLE 9187528 45366 30954 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME R-roscovitine SELICICLIB 45367 30955 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SPICLOMAZINE SPICLOMAZINE 45368 30956 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Flavonoid derivative 8 45369 30957 FHIT 2272 CLINICALLY ACTIONABLE, ENZYME, TRANSPORTER antidepressants 45371 30958 POLK 51426 DNA REPAIR, ENZYME ENTACAPONE ENTACAPONE 45374 30959 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR metformin METFORMIN 24853734 45376 30960 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tacrine-indole hybrid derivative 1 45377 30961 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist 178103927 BAZEDOXIFENE 45378 30962 CBX1 10951 NA VANOXERINE VANOXERINE 45380 30963 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-123916 CHEMBL493863 45381 30964 POLI 11201 DNA REPAIR FAGARONINE FAGARONINE 45383 30965 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LEVOBUPIVACAINE LEVOBUPIVACAINE 45384 30966 IL18 3606 DRUGGABLE GENOME Iboctadekin + rituximab 45385 30967 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NICARDIPINE NICARDIPINE 45386 30968 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CETIRIZINE DIHYDROCHLORIDE CETIRIZINE HYDROCHLORIDE 45390 30969 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME simvastatin SIMVASTATIN 25504632 45391 30970 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LINEZOLID LINEZOLID 24044938 45392 30971 ANO1 55107 ION CHANNEL blocker 178101136 45393 30972 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650408 45396 30973 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME blocker 178100875 PICROTOXIN 45397 30974 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIGITOXIN DIGITOXIN 45398 30975 PERP 64065 NA epirubicin EPIRUBICIN 45399 30976 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135651077 FOROPAFANT 45400 30977 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PDGF-BB 45401 30978 HSPA4 3308 NA RANITIDINE RANITIDINE 11523209 45402 30979 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NELIVAPTAN NELIVAPTAN 45403 30980 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178101011 FLURBIPROFEN 45404 30981 IMPDH2 3615 DRUGGABLE GENOME, ENZYME inhibitor 405067333 MERIMEPODIB 45405 30982 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135649984 45406 30983 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE carboplatin CARBOPLATIN 23963862 45408 30984 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME KENPAULLONE KENPAULLONE 45409 30985 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE CEDIRANIB CEDIRANIB 45410 30986 SLC1A5 6510 TRANSPORTER GLUTAMINE GLUTAMINE 11997238 45411 30987 ALOX15 246 ENZYME, DRUGGABLE GENOME AG-538 CHEMBL56393 45412 30988 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-4798 CHEMBL584635 45413 30989 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HARMOL HARMOL 45414 30990 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL1090771 AVAGACESTAT 45415 30991 PDHA1 5160 ENZYME CPI-613 45416 30992 KDM6A 7403 ENZYME, CLINICALLY ACTIONABLE GSK343 28228601 45417 30993 ADAM17 6868 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, NEUTRAL ZINC METALLOPEPTIDASE, TRANSPORTER, ENZYME Apratastat APRATASTAT 45418 30994 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DOXORUBICIN DOXORUBICIN 18413364 45419 30995 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZK-91587 45422 30996 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545422 MIRANSERTIB 45423 30997 PLD1 5337 ENZYME, DRUGGABLE GENOME US9127005, P2C 45424 30998 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME MDX-1411 MDX-1411 45425 30999 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME ABI-011 45428 31000 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ISOTHYMONIN ISOTHYMONIN 45429 31001 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TAZAROTENE TAZAROTENE 45431 31002 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ECONAZOLE NITRATE ECONAZOLE NITRATE 45432 31003 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR VUF-10499 CHEMBL454890 19053770 45434 31004 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LOSARTAN LOSARTAN 16509571 45435 31005 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 385612212 45436 31006 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL3544984 TRADIPITANT 45437 31007 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME blocker 135650366 SENICAPOC 45438 31008 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651569 45439 31009 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 53801030 DIARYLPROPIONITRILE 45440 31010 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE 4-METHOXYPHENOXYBENZENE CHEMBL398021 18952425 45441 31011 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE fenoterol FENOTEROL 45442 31012 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER erythromycin ERYTHROMYCIN 45443 31013 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Donepezil DONEPEZIL 45445 31014 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE 4-HYDROPEROXYCYCLOPHOSPHAMIDE PERFOSFAMIDE 17046572 45446 31015 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME CLODRONIC ACID CLODRONIC ACID 45447 31016 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SELICICLIB SELICICLIB 21417417 45450 31017 CBX1 10951 NA GNF-PF-2893 CHEMBL312032 45452 31018 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME N-(pyridin-2-yl)pyrimidin-4-amine derivative 2 45453 31019 POLK 51426 DNA REPAIR, ENZYME ESTRAMUSTINE ESTRAMUSTINE 45454 31020 SCTR 6344 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1201616 SECRETIN SYNTHETIC PORCINE 45456 31021 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200434 OXTRIPHYLLINE 45457 31022 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor XL228 XL-228 45458 31023 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER boceprevir BOCEPREVIR 25836019 45461 31024 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker 381744981 PF-05105679 45465 31025 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR SALINE SODIUM CHLORIDE 12742641 45467 31026 ATAD5 79915 NA 3,4-METHYLENEDIOXYB-NITROSTYRENE CHEMBL596380 45469 31027 CRTC2 200186 KINASE tacrolimus TACROLIMUS 26644205 45470 31028 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME OCTREOTIDE OCTREOTIDE 7515212 45471 31029 MAOB 4129 DRUGGABLE GENOME, ENZYME 8-(3-BROMOPHENOXYMETHYL)CAFFEINE CHEMBL2088301 22705191 45472 31030 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178103113 45473 31031 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FLUCONAZOLE FLUCONAZOLE 45475 31032 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLOMETHIAZOLE CLOMETHIAZOLE 45476 31033 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE AST-487 AST-487 45477 31034 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL750 ZONISAMIDE 45478 31035 PRLR 5618 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, KINASE SOMATROPIN SOMATROPIN 45479 31036 PDK2 5164 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 328083452 45480 31037 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Erlotinib ERLOTINIB 26324372,25870087,27468240,28089594,27694386,27102076,27216155,23917401,24410791,26341921,19015641,27760111,26106072,27207775,27793840,24353160,25573954,18981003,17349580,23344264,20942962,25077897,27825638,26286086,27913578,22190593,26720423,19147750,24868098,28408243,26206867,25931286,28343545,17177598,24470557,19010870 45482 31038 COL18A1 80781 DRUGGABLE GENOME THROMBIN THROMBIN 15615851 45483 31039 AKR1B1 231 DRUGGABLE GENOME, ENZYME inhibitor 252166837 45484 31040 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-3037 CHEMBL600336 45485 31041 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER sufentanil SUFENTANIL 45486 31042 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL3545052 FIMEPINOSTAT 45487 31043 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR INGENOL MEBUTATE 45488 31044 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NORTRIPTYLINE NORTRIPTYLINE 45490 31045 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BENZTHIAZIDE BENZTHIAZIDE 45491 31046 PTGS1 5742 ENZYME, DRUGGABLE GENOME KETOPROFEN KETOPROFEN 45492 31047 NEK1 4750 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE inhibitor 249565860 45494 31048 UBE2N 7334 ENZYME, DRUGGABLE GENOME DIHYDROSPINGOSINE DIHYDROSPINGOSINE 45496 31049 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103774 HYDROXYZINE 45499 31050 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000040549 CHEMBL589421 45501 31051 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ethanol ALCOHOL 45506 31052 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE 45507 31053 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Vorinostat VORINOSTAT 27924459 45508 31054 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CARBARIL CARBARIL 45510 31055 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DOXACURIUM CHLORIDE 45511 31056 IL1B 3553 KINASE, DRUGGABLE GENOME GEVOKIZUMAB GEVOKIZUMAB 45513 31057 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME MM-141 ISTIRATUMAB 45515 31058 SMN2 6607 DRUGGABLE GENOME HOE-33342 CHEMBL343002 45516 31059 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist 135650334 45517 31060 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE XL-147 PILARALISIB 45520 31061 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-8 45521 31062 IFI27 3429 NUCLEAR HORMONE RECEPTOR TNF-ALPHA 15086558 45522 31063 TYMSOS 494514 NA daunorubicin DAUNORUBICIN 45525 31064 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME E319 E319 45528 31065 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HEXACHLOROPHENE HEXACHLOROPHENE 45529 31066 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1611 PHENYTOIN SODIUM 45530 31067 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE RAC-NUTLIN-3 CHEMBL211045 45532 31068 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor CHEMBL1201571 ALEFACEPT 45533 31069 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ABAMECTIN ABAMECTIN 45534 31070 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-2 45537 31071 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AP26113 CHEMBL3397300 27836716,27780853 45538 31072 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE CEPHALEXIN CEPHALEXIN 22166395 45539 31073 MPHOSPH8 54737 NA GNF-PF-1969 CHEMBL601364 45541 31074 MAPT 4137 DRUGGABLE GENOME GNF-PF-2776 CHEMBL578294 45542 31075 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE GENTAMICIN GENTAMICIN 14565862 45543 31076 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrazolopyridine derivative 7 45545 31077 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME methotrexate METHOTREXATE 21317831 45546 31078 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE 1,7-O-DIACETYLMETHYLGEOPYXIN A CHEMBL1889303 45547 31079 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 45548 31080 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565816 45549 31081 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR JNJ-38518168 TOREFORANT 25873897 45550 31082 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 404859048 45551 31083 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR M7824 M-7824 45552 31084 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Azachalcone derivative 1 45553 31085 ALPL 249 ENZYME, DRUGGABLE GENOME GNF-PF-1947 CHEMBL585591 45554 31086 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL2110725 VINFLUNINE 45558 31087 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME 20(S)-PROTOPANAXATRIOL CHEMBL255683 26420067 45559 31088 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PEMETREXED PEMETREXED 27876675 45561 31089 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL1201748 CABAZITAXEL 45562 31090 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist 135649822 45564 31091 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE RU 486 11742418 45565 31092 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR alendronate ALENDRONIC ACID 18470879,10692979,21651652,12608943,9933478,18443790,16210379,19020788,15739035,14685227,20500803,12162507,11450701 45566 31093 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE Briciclib BRICICLIB 45569 31094 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Sphinx 45570 31095 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Imidazo bicyclic iminium derivative 3 45571 31096 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL969 PRAZEPAM 45572 31097 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 5,8,11,14-EICOSATETRAYNOIC ACID CHEMBL458328 45573 31098 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Isoflavone derivative 9 45574 31099 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE agonist CHEMBL1743080 TIGATUZUMAB 45575 31100 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-12 45579 31101 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1628502 GABAPENTIN ENACARBIL 45580 31102 CP 1356 DRUGGABLE GENOME, ENZYME HYDROXYUREA HYDROXYUREA 9473738 45582 31103 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamide derivative 25 45585 31104 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2134724 IPRATROPIUM BROMIDE 45586 31105 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CAPECITABINE CAPECITABINE 20504363,17192538,19289619,25287822 45589 31106 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135650257 FENOTEROL 45590 31107 AKR7A2 8574 DRUGGABLE GENOME, ENZYME daunorubicin DAUNORUBICIN 20837989 45591 31108 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE ALVOCIDIB ALVOCIDIB 45592 31109 HBEGF 1839 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME ANTISERUM 7538797 45593 31110 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DIPYRIDAMOLE DIPYRIDAMOLE 45596 31111 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 363894176 45598 31112 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8987457, 15 45601 31113 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PMID29671355-Compound-43 45602 31114 MAPT 4137 DRUGGABLE GENOME HYPERICIN HYPERICIN 45603 31115 HTT 3064 DRUGGABLE GENOME PHENANTHROLINE PHENANTHROLINE 45604 31116 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PALBOCICLIB PALBOCICLIB 25002028 45607 31117 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL325041 BORTEZOMIB 45608 31118 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE methadone METHADONE 23651024 45609 31119 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Pyrrole derivative 7 45611 31120 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL108 CARBAMAZEPINE 45614 31121 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SODIUM NITRITE SODIUM NITRITE 45615 31122 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TROVAFLOXACIN MESYLATE TROVAFLOXACIN MESYLATE 45617 31123 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist CHEMBL3545390 BRILANESTRANT 45618 31124 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR norepinephrine NOREPINEPHRINE 12383575 45619 31125 XDH 7498 DRUGGABLE GENOME, ENZYME Fused heterocyclic compound 4 45620 31126 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PMID29671355-Compound-23 45624 31127 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1724 MEPENZOLATE BROMIDE 45625 31128 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 252827368 PEXIDARTINIB 45627 31129 HMBS 3145 ENZYME RAAV5-PBGD 45628 31130 RAB9A 9367 ENZYME, DRUGGABLE GENOME KENPAULLONE KENPAULLONE 45629 31131 COL15A1 1306 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 45630 31132 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE rifampin RIFAMPIN 18695978 45631 31133 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME ESTAZOLAM ESTAZOLAM 45633 31134 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LY-2090314 LY-2090314 45634 31135 POLG 5428 ENZYME KASANOSIN B KASANOSIN B 18308572 45635 31136 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE LYMPHOKINES 8007461 45636 31137 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor PONATINIB PONATINIB 45637 31138 ACP5 54 ENZYME, DRUGGABLE GENOME G-CSF FILGRASTIM 1724107 45640 31139 ATP5F1D 513 TRANSPORTER HALOTHANE HALOTHANE 45641 31140 GMNN 51053 DRUGGABLE GENOME DEFEROXAMINE MESYLATE DEFEROXAMINE MESYLATE 45642 31141 ADCY1 107 DRUGGABLE GENOME, ENZYME inhibitor 381118802 45643 31142 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR SAQUINAVIR MESYLATE SAQUINAVIR MESYLATE 45644 31143 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME SB-242235 SB-242235 45646 31144 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE AMG 319 45647 31145 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2-MERCAPTOBENZOTHIAZOLE 2-MERCAPTOBENZOTHIAZOLE 45648 31146 NOS1 4842 DRUGGABLE GENOME, ENZYME inhibitor 178101820 45649 31147 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Xanthine XANTHINE 45651 31148 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE RESVERATROL RESVERATROL 15925284 45653 31149 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL135 ESTRADIOL 45655 31150 PTGS2 5743 DRUGGABLE GENOME, ENZYME indomethacin INDOMETHACIN 19602986 45656 31151 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Ad.p53-DC vaccine 12082455,15297186,19621448,21927947,12082456 45659 31152 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME VELIPARIB VELIPARIB 45661 31153 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL3707400 INDANTADOL 45662 31154 CCR10 2826 DRUGGABLE GENOME, CELL SURFACE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 348353673 45663 31155 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER METHOTREXATE METHOTREXATE 45665 31156 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme7WO2012/098070upper 45666 31157 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR thalidomide THALIDOMIDE 20038957 45667 31158 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME PEMBROLIZUMAB PEMBROLIZUMAB 28351930 45669 31159 ATAD5 79915 NA PROTOAPIGENONE PROTOAPIGENONE 45671 31160 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-69187 CHEMBL19954 45672 31161 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 15022342 45673 31162 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135650219 VINBURNINE 45674 31163 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PYRIDOXINE PYRIDOXINE 12603263 45677 31164 USP1 7398 DNA REPAIR, PROTEASE, ENZYME L-162313 CHEMBL288174 45678 31165 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor CHEMBL27759 ENTINOSTAT 45679 31166 PTGS2 5743 DRUGGABLE GENOME, ENZYME CURCUMIN CURCUMIN 24920381 45681 31167 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME P276-00 RIVICICLIB 45683 31168 POLK 51426 DNA REPAIR, ENZYME GOSSYPOL GOSSYPOL 45684 31169 POLB 5423 DNA REPAIR, DRUGGABLE GENOME MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 45685 31170 ATXN2 6311 NA DNDI1417722 CHEMBL1503190 45687 31171 MVK 4598 KINASE, ENZYME inhibitor 135650252 45688 31172 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200347 ISOPROPAMIDE IODIDE 45690 31173 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1416955 CHEMBL1327172 45692 31174 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 4-(4-HYDROXYPHENYLSULFONYL)PHENOL CHEMBL384441 45694 31175 ALOX15 246 ENZYME, DRUGGABLE GENOME RHEIN RHEIN 45695 31176 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BRL-52537 CHEMBL71294 45697 31177 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 INDOMETHACIN INDOMETHACIN 22931300 45700 31178 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE DNDI1417467 CHEMBL1997335 45701 31179 CA1 759 DRUGGABLE GENOME, ENZYME Curcumin CURCUMIN 45702 31180 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrazolopyridine derivative 4 45703 31181 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200420 MIDAZOLAM HYDROCHLORIDE 45705 31182 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE STAUROSPORINE STAUROSPORINE 8895768 45708 31183 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PYRITHIONE ZINC PYRITHIONE ZINC 45709 31184 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME fluvastatin FLUVASTATIN 19842935 45711 31185 PHEX 5251 ENZYME, PROTEASE, DRUGGABLE GENOME CALCITRIOL CALCITRIOL 9835432 45712 31186 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SULINDAC SULFIDE SULINDAC SULFIDE 45713 31187 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR VENLAFAXINE VENLAFAXINE 14978196 45714 31188 CTNNBL1 56259 NA Alpha-acetyldigoxin CHEMBL112750 45715 31189 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ZINC959121 45716 31190 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 404859011 45718 31191 KDM4A 9682 DRUGGABLE GENOME, ENZYME CHLORTETRACYCLINE HYDROCHLORIDE CHLORTETRACYCLINE HYDROCHLORIDE 45721 31192 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 24166501 45722 31193 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Irinotecan IRINOTECAN 27638859 45724 31194 MPHOSPH8 54737 NA GUANIDINONALTRINDOLE GUANIDINONALTRINDOLE 45725 31195 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MECLIZINE MECLIZINE 45726 31196 TRAF1 7185 NA Tumor necrosis factor alpha (TNF-alpha) inhibitors 23007924 45727 31197 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor NERATINIB NERATINIB 45728 31198 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE Benzimidazole BENZIMIDAZOLE 45732 31199 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1128 EDROPHONIUM CHLORIDE 45733 31200 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE ISOCEPHAELINE ISOCEPHAELINE 15974627 45734 31201 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYDROCORTISONE BUTYRATE HYDROCORTISONE BUTYRATE 45735 31202 CD38 952 CELL SURFACE, DRUGGABLE GENOME CD38 CAR-T Cell 45736 31203 TSPO 706 DRUGGABLE GENOME Flurazepam FLURAZEPAM 45738 31204 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor RO4987655 RO-4987655 45739 31205 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200440 MEPIVACAINE HYDROCHLORIDE 45741 31206 WNT5B 81029 DRUGGABLE GENOME fluorouracil FLUOROURACIL 23817222 45742 31207 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE CHONDROITIN 12972284 45743 31208 ATXN2 6311 NA PHENANTHROLINE PHENANTHROLINE 45744 31209 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PMID29130358-Compound-Figure16(9c) 45746 31210 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-22 45747 31211 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Letrozole LETROZOLE 27126994 45748 31212 GLS 2744 ENZYME PSOROMIC ACID PSOROMIC ACID 45749 31213 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Tocilizumab TOCILIZUMAB 45750 31214 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL TRIAZOLAM TRIAZOLAM 45753 31215 CP 1356 DRUGGABLE GENOME, ENZYME NICOTINE NICOTINE 7740554 45754 31216 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE EMTRICITABINE EMTRICITABINE 17172311 45755 31217 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 223365883 CITALOPRAM 45756 31218 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ARZOXIFENE ARZOXIFENE 45757 31219 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME MK-1496 MK-1496 45762 31220 KDM4A 9682 DRUGGABLE GENOME, ENZYME CNQX DISODIUM CHEMBL1255647 45763 31221 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR STREPTONIGRIN STREPTONIGRIN 45766 31222 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID25726713-Compound-48 45767 31223 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE N-METHYL-D-ASPARTIC ACID (NMDA) N-METHYL-D-ASPARTIC ACID (NMDA) 45768 31224 CBX1 10951 NA ROTTLERIN ROTTLERIN 45769 31225 ENPP2 5168 ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 354702264 45770 31226 SI 6476 DRUGGABLE GENOME, ENZYME ACARBOSE ACARBOSE 45773 31227 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PAN-RAF INHIBITOR LY3009120 26732095 45774 31228 SCNN1G 6340 ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AMILORIDE AMILORIDE 45775 31229 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 223365882 BITOPERTIN 45777 31230 HKDC1 80201 DRUGGABLE GENOME, KINASE DEOXYVASICINONE DEOXYVASICINONE 45778 31231 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME FASUDIL FASUDIL 45779 31232 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 INDOMETHACIN MORPHOLINYLAMIDE INDOMETHACIN MORPHOLINYLAMIDE 45780 31233 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE PROTEASE INHIBITORS 12829635 45781 31234 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHENTOLAMINE MESYLATE PHENTOLAMINE MESYLATE 45782 31235 BAZ2B 29994 NA 2-AMINOFLURENE CHEMBL84472 45783 31236 MVD 4597 DRUGGABLE GENOME, ENZYME inhibitor 135650193 45784 31237 KAT2B 8850 ENZYME, DRUGGABLE GENOME inhibitor 178103581 45785 31238 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE FTI 12420225 45786 31239 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE COBALT 15147973,11358837 45787 31240 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE CSA CYCLOSPORINE 12639820 45790 31241 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME JNJ-7706621 JNJ-7706621 45791 31242 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR LUTEOLIN LUTEOLIN 25190466 45792 31243 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Steroid derivative 2 45793 31244 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Recoflavone eye drops 45795 31245 MAPT 4137 DRUGGABLE GENOME SJ000014858 CHEMBL591628 45797 31246 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 252827391 45798 31247 ACP5 54 ENZYME, DRUGGABLE GENOME ANALGESICS 12521129 45799 31248 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor TEMSIROLIMUS TEMSIROLIMUS 45800 31249 MARK4 57787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TAMATINIB R-406 45801 31250 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135650270 FLUOXETINE 45802 31251 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR BAS 01152706 CHEMBL2002487 45803 31252 ATAD5 79915 NA DNDI1417420 CHEMBL1546223 45807 31253 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Rogaratinib ROGARATINIB 45808 31254 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200420 MIDAZOLAM HYDROCHLORIDE 45809 31255 ATAD5 79915 NA 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 45810 31256 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR KENPAULLONE KENPAULLONE 45813 31257 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IODOQUINOL IODOQUINOL 45814 31258 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CGP-12177 CGP-12177 45815 31259 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING AMINEPTINE AMINEPTINE 45816 31260 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE GAMMA-INTERFERON 8572591 45819 31261 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 178100442 CHEMBL375270 45820 31262 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 1R,9S-HYDRASTINE 1R,9S-HYDRASTINE 45822 31263 MAPT 4137 DRUGGABLE GENOME SJ000262801 CHEMBL605077 45823 31264 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME MNU 2415236 45824 31265 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE inhibitor 178103981 ILOMASTAT 45826 31266 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ARSENIC TRIOXIDE 14719092 45830 31267 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Neu-P11 PIROMELATINE 45831 31268 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor DACTOLISIB DACTOLISIB 45832 31269 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME ISF-402 45833 31270 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Ace Inhibitors, Plain 22543981 45834 31271 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DNDI1416969 CHEMBL1453126 45836 31272 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Cyproheptadine CYPROHEPTADINE 45837 31273 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102603 45838 31274 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL1200648 ROCURONIUM BROMIDE 45840 31275 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200819 ARTICAINE HYDROCHLORIDE 45841 31276 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME PMID25435179-Compound-WO2012106509Salermide 45844 31277 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BAY 10-00394 45845 31278 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649758 45847 31279 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX MK-2206 MK-2206 45848 31280 GBA 2629 DRUGGABLE GENOME, ENZYME velaglucerase alfa 45849 31281 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TRETINOIN TRETINOIN 25838141,18511283 45850 31282 ATP1B3 483 ENZYME, TRANSPORTER, DRUGGABLE GENOME inhibitor CHEMBL254219 DIGITOXIN 45851 31283 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE inhibitor 249565657 ZOTAROLIMUS 45854 31284 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650040 45856 31285 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 4,4'-OXYDIANILINE CHEMBL354663 45857 31286 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE THROMBIN THROMBIN 7499260,11375274 45858 31287 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PF-573328 28416483 45859 31288 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4-TERT-BUTYLCATECHOL CHEMBL220845 45863 31289 GMNN 51053 DRUGGABLE GENOME GNF-PF-4516 CHEMBL586029 45864 31290 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PYRITHIONE ZINC PYRITHIONE ZINC 45865 31291 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 249565786 45867 31292 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BGJ398 INFIGRATINIB 45868 31293 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 45869 31294 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565730 CHEMBL2069623 45871 31295 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PIPERTRAMINE PIPERTRAMINE 45872 31296 CLCN7 1186 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER blocker 178101092 45873 31297 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ERYTHROSINE ERYTHROSINE 45875 31298 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME INTERFERON ALFA-2B 11915028 45877 31299 GLCCI1 113263 NA fluticasone propionate 21991891 45878 31300 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME TLN-232 TT-232 45879 31301 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 135651245 TERFENADINE 45880 31302 MPHOSPH8 54737 NA AG-808 CHEMBL68534 45881 31303 PDE4A 5141 DRUGGABLE GENOME, ENZYME CHF 6001 45884 31304 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME BAY-613606 CHEMBL541400 45886 31305 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME PMID27774822-Compound-Figure10CompoundA 45888 31306 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE MT110 SOLITOMAB 45889 31307 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME modulator CHEMBL146506 MOFAROTENE 45891 31308 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME TRISMETHOXYRESVERATROL TRISMETHOXYRESVERATROL 21880495 45892 31309 NGFR 4804 CELL SURFACE, DRUGGABLE GENOME 178101730 45893 31310 SMN1 6606 DRUGGABLE GENOME LAPACHOL LAPACHOL 45895 31311 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ISOETHARINE ISOETHARINE 45896 31312 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR OPHIOBOLIN O OPHIOBOLIN O 22130129 45897 31313 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651501 45898 31314 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER Alseroxylon ALSEROXYLON 45899 31315 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME HERBIMYCIN A 1515646 45901 31316 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649772 45902 31317 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 45903 31318 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME JNJ-7706621 JNJ-7706621 45905 31319 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102292 CEDIRANIB 45906 31320 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 docetaxel DOCETAXEL 19604090 45907 31321 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR RAMIPRIL RAMIPRIL 15716710 45908 31322 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL3545003 MSC-2363318A 45910 31323 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Selumetinib SELUMETINIB 26438159,19755509 45911 31324 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Dacomitinib DACOMITINIB 45913 31325 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ABT-806 DEPATUXIZUMAB 25895099 45914 31326 PTGS2 5743 DRUGGABLE GENOME, ENZYME FENOPROFEN FENOPROFEN 45915 31327 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CEFDITORIN PIVOXIL CEFDITORIN PIVOXIL 45916 31328 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR FROVATRIPTAN FROVATRIPTAN 45918 31329 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor GSK2126458 OMIPALISIB 45919 31330 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 340590250 LORECIVIVINT 45921 31331 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545296 ARQ-736 45922 31332 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-N1 45923 31333 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL598797 CUDC-101 45924 31334 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor SIROLIMUS SIROLIMUS 45925 31335 PDE4D 5144 DRUGGABLE GENOME, ENZYME OX-914 HT-0712 45926 31336 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NEVIRAPINE NEVIRAPINE 22931300 45927 31337 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL454 BUTALBITAL 45929 31338 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-125814 CHEMBL533082 45930 31339 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Arbutamine ARBUTAMINE 45931 31340 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DNDI1417485 CHEMBL1346468 45932 31341 BAZ2B 29994 NA PROCHLORPERAZINE PROCHLORPERAZINE 45933 31342 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE 178101322 45935 31343 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CARBOPROST TROMETHAMINE 45936 31344 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SNS-314 SNS-314 45937 31345 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CONGO RED CONGO RED 45938 31346 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650297 SOBETIROME 45939 31347 CCNB1 891 DRUGGABLE GENOME KENPAULLONE KENPAULLONE 45940 31348 AKR1C3 8644 ENZYME, DRUGGABLE GENOME Isoquinolone derivative 1 45941 31349 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL501867 VINCRISTINE SULFATE 45942 31350 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TRIFLUPROMAZINE TRIFLUPROMAZINE 45943 31351 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME HINOKITIOL HINOKITIOL 45944 31352 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1946170 REGORAFENIB 45945 31353 MSH6 2956 CLINICALLY ACTIONABLE, DNA REPAIR ANTI-PD-1 MONOCLONAL ANTIBODY MEDI0680 26674132 45946 31354 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL538943 VINORELBINE TARTRATE 45947 31355 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GNF-PF-3464 CHEMBL602213 45948 31356 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 381118865 45949 31357 ALPL 249 ENZYME, DRUGGABLE GENOME PYROGALLOL RED PYROGALLOL RED 45950 31358 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 328083475 45951 31359 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TRANILAST TRANILAST 45952 31360 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor 178101304 45953 31361 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 178103530 ETHYLESTRENOL 45954 31362 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL inhibitor 374883890 45955 31363 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHLOROTHALONIL CHLOROTHALONIL 45956 31364 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME NSC-95397 CHEMBL429095 45959 31365 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR STREPTOZOTOCIN STREPTOZOCIN 17968528 45960 31366 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME GALANTAMINE GALANTAMINE 23540646 45961 31367 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME ARA 290 45962 31368 CYB5R3 1727 DRUGGABLE GENOME, ENZYME ceftriaxone CEFTRIAXONE 45963 31369 USP1 7398 DNA REPAIR, PROTEASE, ENZYME NITROFURANTOIN NITROFURANTOIN 45964 31370 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME N/A 45966 31371 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-2357 CHEMBL578257 45967 31372 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1650595 AR-12 45969 31373 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME PF-562271 PF-00562271 45970 31374 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 404859074 45972 31375 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Osimertinib OSIMERTINIB 45973 31376 ELN 2006 DRUGGABLE GENOME, CLINICALLY ACTIONABLE CHEMBL3545070 VONAPANITASE 45975 31377 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE SAHA VORINOSTAT 15583844 45978 31378 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 45980 31379 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 252166567 45982 31380 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor AFATINIB AFATINIB 45983 31381 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL495727 AT-9283 45984 31382 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE RHGH 10195702 45985 31383 TGFBR2 7048 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME inhibitor 249565835 45986 31384 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZD8055 AZD-8055 22271687,26725216,24791855 45991 31385 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 178101771 45992 31386 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AT7519 AT-7519 45993 31387 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-12 45996 31388 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ALPROSTADIL ALPROSTADIL 22931300 45998 31389 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE KINETIN RIBOSIDE KINETIN RIBOSIDE 46000 31390 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LYCOPENE LYCOPENE 18566994 46001 31391 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ANISOTROPINE METHYLBROMIDE 46002 31392 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME FOLFOX-4 REGIMEN 25666295 46003 31393 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor CHEMBL235191 TACEDINALINE 46004 31394 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ETHACRYNIC ACID ETHACRYNIC ACID 46005 31395 ATXN2 6311 NA PARAROSANILINE PARAROSANILINE 46006 31396 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME OXALIPLATIN OXALIPLATIN 20921465 46007 31397 NOS1 4842 DRUGGABLE GENOME, ENZYME CORTICOSTEROIDS 12193391 46009 31398 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 135650177 DICLOFENAC 46010 31399 RABEP1 9135 CLINICALLY ACTIONABLE, GROWTH FACTOR olanzapine OLANZAPINE 28694205 46013 31400 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE IODOQUINOL IODOQUINOL 46015 31401 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 46016 31402 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-138263 CHEMBL535307 46017 31403 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CYCLIZINE CYCLIZINE 46018 31404 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR HELIPARVIFOLINE HELIPARVIFOLINE 46021 31405 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 252166521 DECERNOTINIB 46022 31406 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ONYX-015 LONTUCIREV (REPLICATING ADENOVIRUS) 46023 31407 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1417309 CHEMBL1341830 46024 31408 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178102665 46027 31409 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME tacrolimus TACROLIMUS 18769365,28316087,23426640 46028 31410 SLC1A3 6507 TRANSPORTER, DRUGGABLE GENOME, CELL SURFACE 178100898 46029 31411 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 178102599 46030 31412 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BUFOGENIN BUFOGENIN 46031 31413 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PMID29671355-Compound-67 46032 31414 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Panobinostat PANOBINOSTAT 27443263 46033 31415 COL11A2 1302 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 46034 31416 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE inhibitor 249565822 BALANOL 46035 31417 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Mestranol MESTRANOL 46036 31418 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR antagonist 178103306 46037 31419 BCHE 590 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL215645 RIVASTIGMINE TARTRATE 46040 31420 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME activator 178101006 46041 31421 POLI 11201 DNA REPAIR GNF-PF-3037 CHEMBL600336 46042 31422 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE VATALANIB VATALANIB 46043 31423 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PRAZEPAM PRAZEPAM 46044 31424 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE negative modulator CHEMBL2109095 ERLIZUMAB 46045 31425 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-123457 CHEMBL285157 46046 31426 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 cyclophosphamide CYCLOPHOSPHAMIDE 19376514 46047 31427 VEGFB 7423 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR bevacizumab BEVACIZUMAB 20124951 46048 31428 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1908394 GSK-461364 46049 31429 GATA2 2624 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX EPO EPOETIN ALFA 8677751,9028967 46050 31430 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CEFPIROME CEFPIROME 46051 31431 POLI 11201 DNA REPAIR CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 46052 31432 NR5A2 2494 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR GSK8470 CHEMBL385911 17154495 46053 31433 CDC42 998 DRUGGABLE GENOME ZU-3594419 CHEMBL562095 19527032 46055 31434 DNER 92737 NA Isoxazole-based bicyclic compound 10 46056 31435 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZD5153 AZD-5153 27573426 46059 31436 BAZ2B 29994 NA PYRIDINE-2,4-DICARBOXYLIC ACID CHEMBL316034 46061 31437 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1201151 MESTRANOL 46063 31438 TNFRSF1B 7133 DRUGGABLE GENOME LITHIUM LITHIUM 15565432 46064 31439 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE PS-938285 46065 31440 ALPI 248 DRUGGABLE GENOME, ENZYME THUNBERGINOL B THUNBERGINOL B 46066 31441 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME IFENPRODIL IFENPRODIL 46069 31442 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102275 46070 31443 ANKS1B 56899 NA ethanol ALCOHOL 31462767 46072 31444 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME SANGIVAMYCIN SANGIVAMYCIN 17371872 46073 31445 PDE4A 5141 DRUGGABLE GENOME, ENZYME HT-0712 HT-0712 46075 31446 GHRL 51738 DRUGGABLE GENOME INSULIN INSULIN 17449920 46077 31447 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ANTISENSE OLIGONUCLEOTIDES 15217956 46078 31448 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEFOTAXIME CEFOTAXIME 46081 31449 CD9 928 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ANDROGENS 16128989 46082 31450 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE NGI-1 27694802 46083 31451 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME carbimazole CARBIMAZOLE 26599303,26151496 46085 31452 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-METHOXYESTRADIOL 2-METHOXYESTRADIOL 46086 31453 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (+)-THALIPORPHINE CHEMBL1397308 46087 31454 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME HEXACHLOROPHENE HEXACHLOROPHENE 46088 31455 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Imidazo[1,2-b]pyridazine derivative 3 46089 31456 VKORC1 79001 DRUGGABLE GENOME, ENZYME WARFARIN WARFARIN 46090 31457 KLK5 25818 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166691 46091 31458 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ABBV-257 ABBV-257 46094 31459 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SULMAZOLE SULMAZOLE 46097 31460 ATP1B3 483 ENZYME, TRANSPORTER, DRUGGABLE GENOME inhibitor CHEMBL1614 DESLANOSIDE 46098 31461 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE DEOXY CHOLATE DEOXY CHOLATE 19102680 46099 31462 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALDOSTERONE ALDOSTERONE 46100 31463 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 363894223 46103 31464 SMN1 6606 DRUGGABLE GENOME 2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE CHEMBL201325 46104 31465 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178103733 DESVENLAFAXINE 46105 31466 GABPA 2551 TRANSCRIPTION FACTOR CISPLATIN CISPLATIN 18036733 46106 31467 CFH 3075 DRUGGABLE GENOME eculizumab ECULIZUMAB 26724167 46107 31468 CXCL2 2920 DRUGGABLE GENOME Laquinamod 46108 31469 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME inhibitor 252827429 46109 31470 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME inhibitor CHEMBL2103738 LITHIUM CITRATE 46111 31471 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CAFFEINE CAFFEINE 22931300 46112 31472 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor CHEMBL2103738 LITHIUM CITRATE 46113 31473 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE NVP-BEZ235 DACTOLISIB 46114 31474 DNER 92737 NA Isoxazole-based bicyclic compound 4 46115 31475 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 178102335 SGX-523 46116 31476 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME REL-CISAPRIDE REL-CISAPRIDE 22931300 46118 31477 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1201065 THIAMYLAL SODIUM 46119 31478 ALPL 249 ENZYME, DRUGGABLE GENOME AG-538 CHEMBL56393 46120 31479 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME fluorouracil FLUOROURACIL 27234217 46121 31480 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Letrozole LETROZOLE 46124 31481 PRLR 5618 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, KINASE DHT ANDROSTANOLONE 1544711 46126 31482 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist CHEMBL2178579 ELUBRIXIN 46127 31483 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417086 CHEMBL1224755 46128 31484 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-E5 46130 31485 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL1614713 CC-401 46131 31486 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 46132 31487 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME gefitinib GEFITINIB 31664190 46137 31488 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE TAE-684 TAE-684 46138 31489 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651372 46139 31490 KDM4A 9682 DRUGGABLE GENOME, ENZYME MERCAPTOPURINE MERCAPTOPURINE 46140 31491 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 135651483 ESTRIOL 46143 31492 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-3323 CHEMBL1270169 46144 31493 BCHE 590 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1677 TACRINE HYDROCHLORIDE 46145 31494 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Oxaliplatin OXALIPLATIN 26637369 46146 31495 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SSR149415 46148 31496 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist 178101709 INSULIN 46151 31497 HTT 3064 DRUGGABLE GENOME TRYPTANTHRIN TRYPTANTHRIN 46152 31498 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE SJ000047241 CHEMBL601933 46155 31499 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyrimidine derivative 11 46156 31500 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Five membered heterocyclic benzamide derivative 2 46157 31501 DHFR 1719 DRUGGABLE GENOME, ENZYME ZD1694 RALTITREXED 8698629 46158 31502 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME N-METHYLDOPAMINE HCL CHEMBL1256484 46159 31503 CBR3 874 ENZYME, DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, CLINICALLY ACTIONABLE cyclophosphamide CYCLOPHOSPHAMIDE 46161 31504 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100247 ETALOCIB 46163 31505 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 1,2-NAPHTHOQUINONE 1,2-NAPHTHOQUINONE 46164 31506 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE PAZOPANIB PAZOPANIB 46165 31507 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL566315 OBETICHOLIC ACID 46167 31508 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE TPN 7790321 46168 31509 SFTPA1 653509 DRUGGABLE GENOME CORTISOL HYDROCORTISONE 9575874 46171 31510 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Trametinib TRAMETINIB 28514312 46173 31511 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME BERKELEYAMIDE C BERKELEYAMIDE C 18330993 46174 31512 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE Platinum IV complexe 1 46175 31513 ALDH1A1 216 DRUGGABLE GENOME, ENZYME QUINOXALINE-2-CARBOXYLIC ACID CHEMBL151797 46176 31514 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME PROTEIN SYNTHESIS INHIBITOR 10029562 46177 31515 PSMB9 5698 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor BORTEZOMIB BORTEZOMIB 46178 31516 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103782 LABETALOL 46179 31517 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME PHOSPHOROTHIOATE OLIGONUCLEOTIDE 8832976 46181 31518 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MK-8342 46183 31519 MAPT 4137 DRUGGABLE GENOME PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT 46186 31520 RACGAP1 29127 NA GNF-PF-4029 CHEMBL596633 46187 31521 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178103859 PROTRIPTYLINE 46188 31522 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME Entrectinib ENTRECTINIB 46189 31523 MUC16 94025 DRUGGABLE GENOME ABAGOVOMAB ABAGOVOMAB 46190 31524 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Hydrazide derivative 5 46191 31525 XRCC1 7515 CLINICALLY ACTIONABLE Platinum compounds 19786980,22188361,27636246,21057378,29662106,24446315,22821704,19362955,16875718,24224851,22026922 46192 31526 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PF-562271 PF-00562271 46193 31527 NOS1 4842 DRUGGABLE GENOME, ENZYME THEOPHYLLINE THEOPHYLLINE 12223230 46194 31528 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 46195 31529 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor NILOTINIB NILOTINIB 46196 31530 NCAM1 4684 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE IMGN901 46197 31531 TYMSOS 494514 NA dexamethasone DEXAMETHASONE 46198 31532 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL BUTALBITAL BUTALBITAL 46200 31533 PDE5A 8654 ENZYME, DRUGGABLE GENOME Dipyridamole DIPYRIDAMOLE 46201 31534 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME Chlorzoxazone CHLORZOXAZONE 46202 31535 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 249565855 46205 31536 TOP2B 7155 DRUGGABLE GENOME, ENZYME Elsamitrucin ELSAMITRUCIN 46206 31537 TYMSOS 494514 NA folic acid 18322994 46208 31538 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME LESTAURTINIB LESTAURTINIB 46210 31539 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE APIGENIN APIGENIN 46212 31540 GMNN 51053 DRUGGABLE GENOME STROPHANTHIDIN STROPHANTHIDIN 46213 31541 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL2103836 IMAGABALIN 46214 31542 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER GANCICLOVIR GANCICLOVIR 12105214 46215 31543 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE AMILORIDE AMILORIDE 46216 31544 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178103701 BENZQUINAMIDE 46219 31545 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL3545241 AC-430 46220 31546 CASP2 835 PROTEASE, DRUGGABLE GENOME, ENZYME CETYLPYRIDINIUM CHLORIDE CETYLPYRIDINIUM CHLORIDE 18366176 46222 31547 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 mianserin MIANSERIN 9187528 46223 31548 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL198362 RIVAROXABAN 46225 31549 BAZ2B 29994 NA KETOCONAZOLE KETOCONAZOLE 46226 31550 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER IBUPROFEN IBUPROFEN 11583291 46228 31551 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR AC1LOJYQ 46230 31552 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-3201 CHEMBL581872 46232 31553 KDM4A 9682 DRUGGABLE GENOME, ENZYME ACETOSIDE ACETOSIDE 46233 31554 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME PTHRP 15611080 46234 31555 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CHEMBL2109447 LYM-1 46237 31556 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OCTREOTIDE OCTREOTIDE 46240 31557 VKORC1 79001 DRUGGABLE GENOME, ENZYME acenocoumarol ACENOCOUMAROL 22920394,26445138,25042728,19225451,19018719,23602689,18781852,24474498,16611310,27581200,27262824,17596133,25519826,19875892,19277427,27488176,24956252,18574025,29577257,30983536,29479633,27335128,25769357,25089947,21148049,26777610,25244877,28689179,23651023,25001883,18950464,19270263,24919870,24108193,22571356,18698879,18690342,23774101,25521356,21636598,22592842,22486182,29432897,23423913,23159639,28033245,16815313,23774941,20020283,23473641 46241 31558 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME inhibitor 249565823 46242 31559 ATXN2 6311 NA TCMDC-139459 CHEMBL86464 46243 31560 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 187051797 APICIDIN 46245 31561 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME EPIRUBICIN EPIRUBICIN 46246 31562 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SB-639 46249 31563 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL274654 ORANTINIB 46251 31564 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE BMN673 46252 31565 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PENTAMETHYLQUERCETIN PENTAMETHYLQUERCETIN 46253 31566 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ARCTIGENIN ARCTIGENIN 46255 31567 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FAS-LIGAND 11159548 46257 31568 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 glimepiride GLIMEPIRIDE 24442125,12235454,16325295 46258 31569 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 354702294 46259 31570 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ERLOTINIB ERLOTINIB 46263 31571 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME clavulanate CLAVULANIC ACID 30664875 46265 31572 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Y-39983 Y-39983 46267 31573 FAAH 2166 ENZYME, DRUGGABLE GENOME Pyrimidinyl ethylenediamine derivative 1 46268 31574 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135649987 BETAXOLOL 46269 31575 ABCA1 19 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE atorvastatin ATORVASTATIN 20031551 46270 31576 RRM2 6241 DRUGGABLE GENOME, ENZYME Triapine TRIAPINE 46271 31577 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR OLAPARIB OLAPARIB 28490518 46273 31578 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ACTH CORTICOTROPIN 12571407 46274 31579 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Etanercept ETANERCEPT 46277 31580 KDM4A 9682 DRUGGABLE GENOME, ENZYME HAEMATOXYLIN HAEMATOXYLIN 46279 31581 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure3-Fluevirosine A 46281 31582 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 252166566 HESPERADIN 46282 31583 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CYCLOHEXIMIDE CYCLOHEXIMIDE 46284 31584 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE US9241942, 32-12 46285 31585 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Steroid derivative 3 46286 31586 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (+)-9-DEMETHOXYELEUTHERIN CHEMBL594379 19783445 46287 31587 HMGCR 3156 ENZYME, DRUGGABLE GENOME Rosuvastatin ROSUVASTATIN 46288 31588 SMN2 6607 DRUGGABLE GENOME TDR77585 CHEMBL1333386 46290 31589 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102721 46291 31590 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrrolo-pyridone derivative 1 46292 31591 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ENZYME INHIBITOR 12377937 46293 31592 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME DNDI1318925 CHEMBL1390716 46295 31593 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 187051812 46296 31594 NGFR 4804 CELL SURFACE, DRUGGABLE GENOME PYM50028 46298 31595 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR dopamine DOPAMINE 46299 31596 AOPEP 84909 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL2103847 TOSEDOSTAT 46301 31597 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID25991433-Compound-O3 46304 31598 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ROSMARINIC ACID ROSMARINIC ACID 46305 31599 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-3407 CHEMBL602990 46306 31600 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR OXYTETRACYCLINE HYDROCHLORIDE OXYTETRACYCLINE HYDROCHLORIDE 46308 31601 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Rimacalib RIMACALIB 24600394 46309 31602 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649671 46310 31603 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME AMBENONIUM AMBENONIUM 46311 31604 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME KX2-391 KX2-391 22784709 46314 31605 CSK 1445 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor 249565754 46316 31606 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Pyrimidine derivative 22 46317 31607 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME NSC-180246 CHEMBL484640 46319 31608 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR CHLOROPHENYLPIPERAZINE CHLOROPHENYLPIPERAZINE 46320 31609 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ERBSTATIN ERBSTATIN 46321 31610 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GESTODENE GESTODENE 46323 31611 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Norgestimate NORGESTIMATE 46324 31612 GGCX 2677 DRUGGABLE GENOME, ENZYME Phytonadione PHYTONADIONE 46327 31613 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE ZOLEDRONATE ZOLEDRONIC ACID 46328 31614 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SJ000111093 CHEMBL585045 46329 31615 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIPERIDOLATE PIPERIDOLATE 46330 31616 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PLUMBAGIN PLUMBAGIN 46333 31617 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CMX-2043 CMX-2043 46334 31618 TSPO 706 DRUGGABLE GENOME Quazepam QUAZEPAM 46335 31619 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-3792 CHEMBL582983 46337 31620 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME CYC-116 CYC-116 46338 31621 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 178103612 MOLIBRESIB 46342 31622 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Pyrrolo[1,2-f]triazine derivative 1 46343 31623 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BETHANIDINE BETHANIDINE 46344 31624 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US10100051, Compound 10 46346 31625 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 384403638 46347 31626 UGT2B7 7364 DRUGGABLE GENOME efavirenz EFAVIRENZ 20860463,24080498,26774523,19487252,19779319,24729586,23172109 46348 31627 CBX1 10951 NA GOSSYPOL GOSSYPOL 46349 31628 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-D1 46352 31629 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 223366031 46354 31630 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-806 CHEMBL547101 46355 31631 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE INFIGRATINIB INFIGRATINIB 29182496,24122810 46356 31632 CCL11 6356 DRUGGABLE GENOME methadone METHADONE 29222992 46358 31633 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Curcumin analog 2 46359 31634 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MALATHION MALATHION 46360 31635 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER WARFARIN WARFARIN 46362 31636 TUBA1C 84790 DRUGGABLE GENOME CHEMBL492399 VERUBULIN 46363 31637 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-2374 CHEMBL600298 46365 31638 SRD5A1 6715 DRUGGABLE GENOME FR-146687 46366 31639 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR NOVOBIOCIN NOVOBIOCIN 23859777 46367 31640 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Estradiol Cypionate 46368 31641 AK2 204 ENZYME, KINASE adefovir dipivoxil 46369 31642 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor 135651454 46370 31643 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME OSAJIN OSAJIN 46371 31644 PTGS2 5743 DRUGGABLE GENOME, ENZYME NAPROXEN NAPROXEN 46372 31645 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ATRA TRETINOIN 9402847 46373 31646 ATAD5 79915 NA GNF-PF-4078 CHEMBL584883 46376 31647 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 46377 31648 GSTO1 9446 ENZYME, DRUGGABLE GENOME ARSENIC TRIOXIDE 15761769 46379 31649 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME ELACRIDAR ELACRIDAR 22266779 46380 31650 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE VASOPRESSIN VASOPRESSIN 11514571 46383 31651 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME AX-200 46384 31652 ALPL 249 ENZYME, DRUGGABLE GENOME SULFURETIN SULFURETIN 46385 31653 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102269 46387 31654 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE TILUDRONATE TILUDRONIC ACID 46390 31655 CROT 54677 DRUGGABLE GENOME PROPIONYL-L-CARNITINE 46392 31656 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE VINDESINE SULFATE VINDESINE SULFATE 46393 31657 DIABLO 56616 NA PMA 12920112 46395 31658 NDUFA1 4694 ENZYME inhibitor CHEMBL3545320 ME-344 46396 31659 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ISOPROTERENOL ISOPROTERENOL 46397 31660 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE ADRIAMYCIN ADRIAMYCIN 2007582 46398 31661 CALR 811 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ANTIANGIOGENIC 10498619 46399 31662 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102601 46400 31663 POLA1 5422 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, DNA REPAIR DIGALLIC ACID DIGALLIC ACID 1705574 46401 31664 UBE2N 7334 ENZYME, DRUGGABLE GENOME CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 46403 31665 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102775 46406 31666 GUCY2C 2984 DRUGGABLE GENOME, KINASE MD-1100 LINACLOTIDE 46407 31667 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME Apratastat APRATASTAT 46409 31668 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650696 46411 31669 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103586 ENTINOSTAT 46413 31670 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Quinoline and quinazoline derivative 3 46415 31671 PDE4B 5142 DRUGGABLE GENOME, ENZYME PENTOXIFYLLINE PENTOXIFYLLINE 46416 31672 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE AMG888/U3-1287 46417 31673 XRCC5 7520 KINASE PHENYLBUTYRATE PHENYLBUTANOIC ACID 16000590 46418 31674 GMNN 51053 DRUGGABLE GENOME LY-367265 CHEMBL1079460 46419 31675 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tacrine heterodimer derivative 1 46420 31676 POLI 11201 DNA REPAIR NSC-638080 CHEMBL136344 46422 31677 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 329968400 46423 31678 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545160 SU-014813 46424 31679 FST 10468 DRUGGABLE GENOME ADENOVIRUS VECTOR 16943576 46425 31680 TNNI3 7137 DRUGGABLE GENOME PYROGALLOL RED PYROGALLOL RED 46426 31681 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME DERMOLASTIN 46427 31682 KDM4A 9682 DRUGGABLE GENOME, ENZYME MYRICETIN MYRICETIN 46428 31683 PLD1 5337 ENZYME, DRUGGABLE GENOME HALOPEMIDE HALOPEMIDE 46429 31684 BAZ2B 29994 NA TCMDC-123605 CHEMBL547285 46430 31685 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE RG-7446 ATEZOLIZUMAB 24403232 46431 31686 SULT1A4 445329 ENZYME morphine MORPHINE 46433 31687 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-4012 CHEMBL584269 46434 31688 CYP24A1 1591 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME inhibitor 252827515 CHEMBL255088 46436 31689 KDM4A 9682 DRUGGABLE GENOME, ENZYME OXYPHENBUTAZONE OXYPHENBUTAZONE 46437 31690 POLK 51426 DNA REPAIR, ENZYME AMOXICILLIN AMOXICILLIN 46438 31691 IGFBP3 3486 DRUGGABLE GENOME fluorouracil FLUOROURACIL 20860465 46439 31692 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor AXITINIB AXITINIB 46442 31693 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL1200722 PIPECURONIUM BROMIDE 46443 31694 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL THIOCOLCHICOSIDE THIOCOLCHICOSIDE 46445 31695 SLC9A1 6548 TRANSPORTER, DRUGGABLE GENOME, EXCHANGER, CELL SURFACE HOE-694 CHEMBL62231 17493937 46446 31696 LSS 4047 ENZYME, DRUGGABLE GENOME inhibitor 178103321 46447 31697 EGLN2 112398 ENZYME, DRUGGABLE GENOME FG-2216 46448 31698 IL11 3589 DRUGGABLE GENOME, KINASE, GROWTH FACTOR ETIDRONATE ETIDRONIC ACID 12522661 46453 31699 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor 252827389 46454 31700 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 sufentanil SUFENTANIL 31773688,29926893 46456 31701 IL1B 3553 KINASE, DRUGGABLE GENOME AUTOANTIGEN 8781713 46461 31702 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MYCOPHENOLIC ACID MYCOPHENOLIC ACID 17618115 46462 31703 BCHE 590 DRUGGABLE GENOME, ENZYME Tacrine heterodimer derivative 1 46464 31704 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NORGESTREL NORGESTREL 46467 31705 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE oxcarbazepine OXCARBAZEPINE 27900402 46468 31706 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor BEZ235 DACTOLISIB 46470 31707 POLI 11201 DNA REPAIR MUCRONULATOL(+/-) MUCRONULATOL(+/-) 46471 31708 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor REGORAFENIB REGORAFENIB 46472 31709 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE ALENDRONIC ACID ALENDRONIC ACID 15012988 46473 31710 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Fluorouracil FLUOROURACIL 46475 31711 HSPA4 3308 NA PIOGLITAZONE PIOGLITAZONE 12871756 46476 31712 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MCP-201 46477 31713 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DIHYDROGAMBOGIC ACID DIHYDROGAMBOGIC ACID 46478 31714 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHLORPROMAZINE CHLORPROMAZINE 15135088 46479 31715 COQ2 27235 ENZYME rosuvastatin ROSUVASTATIN 20347093 46480 31716 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME RG-1530 RG-1530 46482 31717 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor PI-103 PI-103 46484 31718 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist 310264685 46485 31719 DTNBP1 84062 KINASE haloperidol HALOPERIDOL 27023437 46486 31720 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE AZD6482 AZD-6482 26563132 46487 31721 HNMT 3176 ENZYME, DRUGGABLE GENOME anthracyclines and related substances 23441093,21900104 46489 31722 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 1-(4-HYDROXYPHENYL)MALEIMIDE CHEMBL565893 46491 31723 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-74859 CHEMBL477936 46492 31724 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUTAPROST BUTAPROST 46493 31725 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE CGP-7930 CHEMBL1256697 46494 31726 TH 7054 ENZYME, DRUGGABLE GENOME inhibitor 178101788 46495 31727 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME OXITRIPTAN OXITRIPTAN 46496 31728 MYO9B 4650 NA PROPYLTHIOURACIL PROPYLTHIOURACIL 3989729 46497 31729 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102252 46498 31730 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 310264696 AZD-8835 46499 31731 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Imidazo[1,5-a]pyridine derivative 2 46500 31732 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TCMDC-124544 CHEMBL531322 46502 31733 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AST-1306 ALLITINIB 46503 31734 MAPT 4137 DRUGGABLE GENOME AM-404 CHEMBL39878 46504 31735 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER BRYOSTATIN 1 9607591 46506 31736 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME DALANTERCEPT DALANTERCEPT 46507 31737 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DIHYDREXIDINE HYDROCHLORIDE DIHYDREXIDINE HYDROCHLORIDE 46511 31738 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200987 EPROSARTAN MESYLATE 46512 31739 MMP7 4316 NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor CHEMBL1200699 DOXYCYCLINE 46513 31740 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EZN-4176 46515 31741 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-402538 CHEMBL121556 46517 31742 CSNK1E 1454 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, DNA REPAIR heroin DIACETYLMORPHINE 46520 31743 IGF1 3479 GROWTH FACTOR, HORMONE ACTIVITY, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE RECOMBINANT HUMAN INSULIN-LIKE GROWTH FACTOR BINDING PROTEIN-3 46522 31744 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ethinyl estradiol 18695978 46523 31745 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE E-GUGGULSTERONE E-GUGGULSTERONE 46524 31746 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-124266 CHEMBL124006 46525 31747 TOP2B 7155 DRUGGABLE GENOME, ENZYME Novobiocin NOVOBIOCIN 46527 31748 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-4786 CHEMBL602363 46531 31749 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME GDC-0879 CHEMBL525191 23549875 46533 31750 MAPT 4137 DRUGGABLE GENOME EPINEPHRINE EPINEPHRINE 46534 31751 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL105442 CI-1040 46535 31752 GLS 2744 ENZYME PMID30273516-Compound-1 46536 31753 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-3996 CHEMBL584458 46539 31754 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4,4'-DITHIODIPYRIDINE CHEMBL1232076 46540 31755 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE POL I INHIBITOR CX5461 28211448 46541 31756 AKR1C3 8644 ENZYME, DRUGGABLE GENOME N-(phenylamino)-benzoate derivative 1 46542 31757 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 verapamil VERAPAMIL 9187528 46543 31758 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DACTOLISIB DACTOLISIB 24356815 46544 31759 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZIRAM ZIRAM 46545 31760 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE inhibitor CHEMBL1201608 MUROMONAB-CD3 46546 31761 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME IOPHENOXIC ACID IOPHENOXIC ACID 46548 31762 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR MGCD-0103 MOCETINOSTAT 46549 31763 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE sorafenib SORAFENIB 25816720 46551 31764 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 INDIRUBIN SULFATE SU-9516 46553 31765 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME HOMIDIUM HOMIDIUM 46554 31766 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE URSOLIC ACID URSOLIC ACID 20100662 46556 31767 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 249565715 LEVOBETAXOLOL 46557 31768 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MUNDULONE ACETATE MUNDULONE ACETATE 46558 31769 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE VATALANIB VATALANIB 46559 31770 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR PROPRANOLOL PROPRANOLOL 15598146 46560 31771 COMT 1312 DRUGGABLE GENOME, ENZYME haloperidol HALOPERIDOL 27023437,23963056 46561 31772 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME HGF 9348194 46562 31773 SV2A 9900 DRUGGABLE GENOME, TRANSPORTER modulator CHEMBL607400 BRIVARACETAM 46564 31774 BAP1 8314 PROTEASE, TUMOR SUPPRESSOR, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE VORINOSTAT VORINOSTAT 22038994 46565 31775 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 135652455 46567 31776 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL605 PROCAINAMIDE HYDROCHLORIDE 46568 31777 GMNN 51053 DRUGGABLE GENOME GITOXIGENIN GITOXIGENIN 46570 31778 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ACIVICIN ACIVICIN 46572 31779 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME Inotersen INOTERSEN 46573 31780 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 404858998 46574 31781 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISOPRENALINE ISOPROTERENOL 46575 31782 PSORS1C1 170679 NA gemcitabine GEMCITABINE 31616045 46577 31783 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME AVA-101 46578 31784 HBB 3043 DRUGGABLE GENOME, ENZYME NEBULARINE NEBULARINE 46579 31785 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TESTOLACTONE TESTOLACTONE 46581 31786 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NORETHISTERONE NORETHINDRONE 46582 31787 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CYCLOSPORINE CYCLOSPORINE 22931300 46583 31788 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 4-METHYLESCULETIN 4-METHYLESCULETIN 46584 31789 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MONASTROL MONASTROL 46586 31790 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178100905 46589 31791 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CARBOPLATIN CARBOPLATIN 22139083 46590 31792 HKDC1 80201 DRUGGABLE GENOME, KINASE NSC-95397 CHEMBL429095 46591 31793 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME acamprosate ACAMPROSATE 25290263 46592 31794 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BAICALEIN BAICALEIN 46593 31795 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ALPHA,BETA-DEHYDROCURVULARIN CHEMBL482050 46594 31796 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650008 46595 31797 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GALLIC ACID GALLIC ACID 46597 31798 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL3545368 PANOBINOSTAT LACTATE 46599 31799 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROTOAPIGENONE PROTOAPIGENONE 46601 31800 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR EPINEPHRINE EPINEPHRINE 46602 31801 TUBB 203068 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 46603 31802 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE LY-294002 LY-294002 16767085 46605 31803 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IBUPROFEN IBUPROFEN 22931300 46608 31804 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE PF-05212384 GEDATOLISIB 21325073 46609 31805 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DISULFIRAM DISULFIRAM 46610 31806 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE XL999 46613 31807 GMNN 51053 DRUGGABLE GENOME 7,12-DIMETHYL-BENZO[A]ANTHRACENE CHEMBL329673 46615 31808 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Rilotumumab RILOTUMUMAB 24919569 46616 31809 ALOX15B 247 DRUGGABLE GENOME, ENZYME MESO-HEXESTROL MESO-HEXESTROL 46617 31810 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GUANIDINONALTRINDOLE GUANIDINONALTRINDOLE 46618 31811 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PHA-665752 PHA-665752 24165158,26124204,23542356 46620 31812 RGS4 5999 DRUGGABLE GENOME TCMDC-124022 CHEMBL548017 46621 31813 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1201063 PROPAFENONE HYDROCHLORIDE 46622 31814 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE DORAMAPIMOD DORAMAPIMOD 46623 31815 DHRS9 10170 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE (+/-)-HYATELLAQUINONE CHEMBL456414 19188072 46624 31816 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Azaindazole amide derivative 1 46626 31817 RAD51 5888 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR AMUVATINIB AMUVATINIB 46627 31818 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135649702 46628 31819 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE inhibitor 315661315 46631 31820 PSCA 8000 DRUGGABLE GENOME AGS-PSCA MK-4721 46632 31821 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ISOPROTERENOL HYDROCHLORIDE ISOPROTERENOL HYDROCHLORIDE 46633 31822 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL27759 ENTINOSTAT 46635 31823 POLB 5423 DNA REPAIR, DRUGGABLE GENOME COUMESTROL COUMESTROL 46636 31824 GREM2 64388 DRUGGABLE GENOME allopurinol ALLOPURINOL 30924126 46637 31825 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MERCURIC CHLORIDE MERCURIC CHLORIDE 46638 31826 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651525 46639 31827 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME BARASERTIB BARASERTIB 46640 31828 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR BUDESONIDE BUDESONIDE 46641 31829 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652306 46642 31830 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PHENOXYBENZAMINE PHENOXYBENZAMINE 46643 31831 NF2 4771 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, DRUG RESISTANCE, KINASE EVEROLIMUS EVEROLIMUS 25567352 46644 31832 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME RVT-505 46645 31833 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Bavencio avelumab 46647 31834 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 375973260 46648 31835 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PIFEXOLE PIFEXOLE 46649 31836 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650088 CHLORPROMAZINE 46650 31837 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL552212 LEXIBULIN 46653 31838 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor LAPATINIB DITOSYLATE 46657 31839 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565822 BALANOL 46658 31840 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME mercaptopurine MERCAPTOPURINE 29683944 46660 31841 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200609 PAROXETINE MESYLATE 46661 31842 RGS4 5999 DRUGGABLE GENOME GOSSYPOL GOSSYPOL 46662 31843 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME CEP-37440 CEP-37440 46663 31844 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME 3,8'-BIAPIGENIN CHEMBL515252 46665 31845 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GLABRANIN GLABRANIN 46666 31846 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR RDEA119 46667 31847 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Piperidinone derivative 1 46668 31848 PDE1A 5136 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL628 PENTOXIFYLLINE 46669 31849 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXYPHENISATIN ACETATE OXYPHENISATIN ACETATE 46670 31850 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 249565755 46678 31851 FN1 2335 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 46679 31852 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 9-CRA 9077483 46680 31853 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR 2-ENE-VALPROATE CHEMBL117487 17566732 46681 31854 CDKL2 8999 DRUGGABLE GENOME, KINASE, ENZYME, TUMOR SUPPRESSOR, SERINE THREONINE KINASE inhibitor 249565786 46683 31855 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME ZM-449829 CHEMBL154580 46684 31856 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 336446955 ASP-4058 46685 31857 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TCMDC-124440 CHEMBL547407 46687 31858 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR ACACETIN ACACETIN 46688 31859 HKDC1 80201 DRUGGABLE GENOME, KINASE SJ000032153 CHEMBL600862 46690 31860 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL454 BUTALBITAL 46691 31861 SMN2 6607 DRUGGABLE GENOME 7,3'-DIMETHOXYFLAVONE 7,3'-DIMETHOXYFLAVONE 46692 31862 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR ALVESPIMYCIN ALVESPIMYCIN 17603540 46693 31863 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CHELERYTHRINE CHLORIDE CHELERYTHRINE CHLORIDE 46696 31864 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME DI-Leu16-IL2 46697 31865 CBX1 10951 NA LY-367265 CHEMBL1079460 46698 31866 TUBB6 84617 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 46699 31867 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor PANOBINOSTAT PANOBINOSTAT 46700 31868 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR inhibitor CHEMBL1637 GEMCITABINE HYDROCHLORIDE 46702 31869 TARDBP 23435 TUMOR SUPPRESSOR NEOCUPROINE NEOCUPROINE 46704 31870 CA1 759 DRUGGABLE GENOME, ENZYME Acetazolamide ACETAZOLAMIDE 46705 31871 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1201113 CETIRIZINE HYDROCHLORIDE 46706 31872 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE DORAMAPIMOD DORAMAPIMOD 46707 31873 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650830 PIPAMPERONE 46708 31874 ABCB11 8647 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE rosuvastatin ROSUVASTATIN 46709 31875 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME R667 46711 31876 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE 187051784 LUMACAFTOR 46712 31877 PDE4B 5142 DRUGGABLE GENOME, ENZYME AWD-12-281 46713 31878 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR clodronate CLODRONIC ACID 10692979,12608943,18443790,19020788,15739035,12162507 46715 31879 STAG2 10735 CLINICALLY ACTIONABLE, DRUG RESISTANCE Olaparib OLAPARIB 21852505,24356817 46716 31880 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME GR-127935 GR-127935 46717 31881 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR TESTOSTERONE TESTOSTERONE 9288184 46718 31882 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DNDI1383301 CHEMBL1509103 46719 31883 MT1H 4496 NA STREPTOZOTOCIN STREPTOZOCIN 9176863 46720 31884 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 223366188 46722 31885 FGF1 2246 CLINICALLY ACTIONABLE, GROWTH FACTOR, DRUGGABLE GENOME inhibitor CHEMBL1615835 MUPARFOSTAT 46723 31886 TH 7054 ENZYME, DRUGGABLE GENOME META-IODOBENZYLGUANIDINE 7576974 46724 31887 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME QUERCETIN QUERCETIN 46725 31888 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Flourouracil 16243804 46726 31889 CACNB3 784 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ION CHANNEL blocker CHEMBL1200382 BEPRIDIL HYDROCHLORIDE 46727 31890 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor ARQ736 46728 31891 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE EMD 55900 46731 31892 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME CARMINIC ACID CARMINIC ACID 46732 31893 SLC12A5 57468 DRUGGABLE GENOME, TRANSPORTER inhibitor 178101310 46733 31894 BRD9 65980 ENZYME 387065623 46734 31895 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SJ000147993 CHEMBL601618 46735 31896 ATAD5 79915 NA ELLIPTECINE ELLIPTECINE 46736 31897 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PD-98059 CHEMBL35482 10753939,9467952 46737 31898 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GOSSYPOL GOSSYPOL 46738 31899 GRK3 157 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 252166647 46739 31900 PML 5371 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TAZAROTENE TAZAROTENE 16939905 46740 31901 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200384 BETAMETHASONE DIPROPIONATE 46741 31902 GAA 2548 DRUGGABLE GENOME, ENZYME BAS 01152706 CHEMBL2002487 46742 31903 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 5,7-DIHYDROXY-4-METHYLCOUMARIN 5,7-DIHYDROXY-4-METHYLCOUMARIN 46743 31904 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BETA-LAPACHONE LAPACHONE 46745 31905 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE gemcitabine GEMCITABINE 21636554 46746 31906 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Mercaptopurine MERCAPTOPURINE 46747 31907 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX anthracyclines and related substances 46748 31908 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BEPOTASTINE BEPOTASTINE 46749 31909 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PIMOZIDE PIMOZIDE 46750 31910 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY DXM 8842473 46751 31911 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-5114 CHEMBL601952 46752 31912 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME CAR-T cells targeting MUC1 46753 31913 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000007704 CHEMBL589469 46754 31914 PTGES 9536 DRUGGABLE GENOME, ENZYME inhibitor 252827419 46757 31915 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody IBRITUMOMAB TIUXETAN ZEVALIN 46759 31916 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Tanespimycin TANESPIMYCIN 46761 31917 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE METHIOTHEPIN MESYLATE METHIOTHEPIN MESYLATE 46762 31918 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor MOTESANIB MOTESANIB 46763 31919 DNER 92737 NA Isoxazole-based bicyclic compound 11 46764 31920 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-26 46765 31921 ADD1 118 KINASE furosemide FUROSEMIDE 20877298,21692745 46766 31922 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR inhibitor ASP3026 ASP-3026 46769 31923 COL2A1 1280 DRUGGABLE GENOME COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 46771 31924 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor SORAFENIB SORAFENIB 46772 31925 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL3545252 DOCETAXEL 46773 31926 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Retosiban RETOSIBAN 46776 31927 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RITUXIMAB RITUXIMAB 11895917 46778 31928 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR SIMVASTATIN SIMVASTATIN 18047562 46780 31929 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BICALUTAMIDE BICALUTAMIDE 46781 31930 MYH7B 57644 NA activator CHEMBL1800955 OMECAMTIV MECARBIL 46782 31931 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME Hematide PEGINESATIDE 46784 31932 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME Sulfatinib SURUFATINIB 46785 31933 PTGS1 5742 ENZYME, DRUGGABLE GENOME MECLOFENAMIC ACID 46787 31934 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME CS-3030 46788 31935 ATAD5 79915 NA PIPERINE PIPERINE 46789 31936 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME E7090 E-7090 23175443,27535969,19901323 46790 31937 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PF-4691502 PF-04691502 46791 31938 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DINOSEB DINOSEB 46793 31939 SRPRB 58477 NA ethanol ALCOHOL 31002879 46794 31940 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL612 DEXTROAMPHETAMINE 46795 31941 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GW843682X GW843682X 46796 31942 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ustekinumab USTEKINUMAB 23521149 46797 31943 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE paclitaxel PACLITAXEL 22370314,20573926,19692680,22581822,21783417,22285168,21900837,20022809 46798 31944 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR MERCURIC CHLORIDE MERCURIC CHLORIDE 46800 31945 ALB 213 TRANSPORTER, DRUGGABLE GENOME ANTISERUM 1378681 46801 31946 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME PMID27998201-Compound-17 46803 31947 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR TETANUS TOXOID 8704175 46804 31948 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-5183 CHEMBL577660 46805 31949 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 3-AMINOBENZAMIDE 3-AMINOBENZAMIDE 46806 31950 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY clozapine CLOZAPINE 24624910 46807 31951 HTT 3064 DRUGGABLE GENOME CARMINOMYCIN CARUBICIN 46808 31952 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE azacitidine AZACITIDINE 29205204 46809 31953 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ETHACRYNIC ACID ETHACRYNIC ACID 46810 31954 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL284121 ILX23-7553 46811 31955 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PIRENZEPINE PIRENZEPINE 46812 31956 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist 178100456 46813 31957 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE IFN 11391574 46814 31958 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME COUMARIN COUMARIN 8576174 46815 31959 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NIGULDIPINE NIGULDIPINE 46817 31960 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650452 46818 31961 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE SAR245409 VOXTALISIB 24583798,24634413 46819 31962 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME TYRPHOSTIN A9 TYRPHOSTIN A9 46820 31963 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102567 46822 31964 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME JUGLONE JUGLONE 46823 31965 LAT 27040 KINASE TRIDOLGOSIR TRIDOLGOSIR 17897956 46826 31966 ACSS2 55902 ENZYME, TRANSCRIPTION FACTOR ethanol ALCOHOL 28550509 46830 31967 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER (S)-FLUOXETINE CHEMBL1169388 46831 31968 ACYP2 98 NA cisplatin CISPLATIN 26928270,31666714 46833 31969 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BCMA nanobody CAR-T cells 46837 31970 LSS 4047 ENZYME, DRUGGABLE GENOME inhibitor 178103333 46838 31971 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME LUTEOLIN LUTEOLIN 46840 31972 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Peptide analog 54 46842 31973 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID26161698-Compound-25 46844 31974 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1237119 TREPROSTINIL 46846 31975 HSPA4 3308 NA SALINE SODIUM CHLORIDE 8724993 46848 31976 F5 2153 DRUGGABLE GENOME Lusutrombopag LUSUTROMBOPAG 46849 31977 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LAUROGUADINE LAUROGUADINE 46850 31978 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SBI-060756 26603897 46852 31979 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE AZ8010 22869148 46854 31980 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FLUNISOLIDE FLUNISOLIDE 22931300 46855 31981 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 249565652 AKN-028 46856 31982 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Interferon Alfa-2a, Recombinant 46857 31983 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CONJUGATED ESTROGENS 46859 31984 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FLUPHENAZINE FLUPHENAZINE 46861 31985 CASP8 841 DRUGGABLE GENOME, PROTEASE, ENZYME, CLINICALLY ACTIONABLE CONATUMUMAB CONATUMUMAB 26291055 46862 31986 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME ETHANOL ALCOHOL 14574224 46863 31987 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PD-81723 CHEMBL59532 46865 31988 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1766 DESOXIMETASONE 46866 31989 XDH 7498 DRUGGABLE GENOME, ENZYME Fused heterocyclic compound 10 46867 31990 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774822-Compound-Figure10Compound12 46868 31991 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1940832 MILVETEROL 46870 31992 ATXN2 6311 NA PROTOAPIGENONE PROTOAPIGENONE 46871 31993 PPA1 5464 ENZYME ETHANOL ALCOHOL 10349738 46872 31994 CBX1 10951 NA ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 46873 31995 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650868 QUADAZOCINE 46876 31996 CDS1 1040 KINASE, ENZYME inhibitor CHEMBL3544936 XL-844 46877 31997 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER DOMPERIDONE DOMPERIDONE 15285840 46878 31998 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE HARMINE HARMINE 46879 31999 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL377300 BRIVANIB 46880 32000 MARCHF8 220972 ENZYME HBV vaccine 46882 32001 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR (S)APOMORPHINE (S)APOMORPHINE 46883 32002 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1428 NIMODIPINE 46885 32003 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Opium derivatives and expectorants 46888 32004 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ALPRENOLOL ALPRENOLOL 46889 32005 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PF-562271 PF-00562271 46890 32006 ABCB4 5244 TRANSPORTER, DRUGGABLE GENOME, ENZYME, ABC TRANSPORTER CYCLOSPORINE CYCLOSPORINE 1972761 46892 32007 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME NORHARMANE NORHARMANE 46893 32008 POLI 11201 DNA REPAIR BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 46894 32009 IDO2 169355 ENZYME 2,3-diamino-benzo[b]thiophene derivative 7 46895 32010 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ABT-263 NAVITOCLAX 27659046 46896 32011 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SKF-75670 HYDROBROMIDE CHEMBL1256698 46897 32012 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1256958 EPINEPHRINE BITARTRATE 46898 32013 TUBB2B 347733 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 46900 32014 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AG-538 CHEMBL56393 46902 32015 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649924 46903 32016 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE LOPERAMIDE HYDROCHLORIDE LOPERAMIDE HYDROCHLORIDE 46904 32017 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Selumetinib SELUMETINIB 27196754,21358673,26232337 46905 32018 KDM4A 9682 DRUGGABLE GENOME, ENZYME inhibitor 381118851 46907 32019 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AUTOLOGOUS DENDRITIC CELLS 11034426 46908 32020 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROTOPORPHYRIN DISODIUM PROTOPORPHYRIN DISODIUM 46911 32021 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR E324 E324 46912 32022 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor CHEMBL463981 BEGACESTAT 46916 32023 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PBF-1129 46917 32024 SLC15A1 6564 DRUGGABLE GENOME, TRANSPORTER GLYCYLSARCOSINE GLYCYLSARCOSINE 22584254 46918 32025 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TRIAZOLAM TRIAZOLAM 22137933 46919 32026 MMUT 4594 ENZYME Hydroxocobalamin HYDROXOCOBALAMIN 46920 32027 HTT 3064 DRUGGABLE GENOME BRAIN-DERIVED NEUROTROPHIC FACTOR 12956709 46921 32028 KDM4A 9682 DRUGGABLE GENOME, ENZYME ISOKAEMPFERIDE ISOKAEMPFERIDE 46922 32029 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 46923 32030 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE chlorproguanil CHLORPROGUANIL 12387962,20599264,15183620 46924 32031 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1742428 DONITRIPTAN 46926 32032 CYB5R4 51167 DRUGGABLE GENOME primaquine PRIMAQUINE 46927 32033 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR SJ000128325 CHEMBL602718 46928 32034 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DICHLOROXYLENOL DICHLOROXYLENOL 46929 32035 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 U-50488 U-50488 METHANE SULFONATE 46930 32036 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Chlorpheniramine CHLORPHENIRAMINE 46931 32037 GMNN 51053 DRUGGABLE GENOME KENPAULLONE KENPAULLONE 46932 32038 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIPYRITHIONE DIPYRITHIONE 46933 32039 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417614 CHEMBL1567571 46934 32040 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE DINACICLIB DINACICLIB 46936 32041 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZM-39923 HCL CHEMBL538798 46937 32042 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PRECLINICAL 23020132,22608338,26619011,21483012,22351686,19001320,21156289,20368568,19255327,22048237,19561230,19010912,23549875,25024077,23489023,18541894,24586605,24508103,22773810,23833300,23812671,24576830,19238210,20818844,23612012,23251002,22356324,20857202,22536370,22997239,21163703,15035987,23470635,21663470,24594804,22586120,20413299,22805292,19537845,14679157,22663011,21975775,22038996,22448344,12068308,24163374,19773371,24354346,23325582,24583796,23031422,22735384,21683865,25370471,21639808,22281684,22649091,22241789,24570209,23918947,25989278,22389471,23934108,22180495,23524406,26678033,19018267,24388723,23845441,23614898,25157968,20619739,12460919,24107445,12460918,21594703,20350999,20630094,21426297,19404918,22743296,24396464,22972589,21129611,23406027 46938 32043 SMN2 6607 DRUGGABLE GENOME 10-METHOXYLRUTAECARPINE CHEMBL85826 46940 32044 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1677 TACRINE HYDROCHLORIDE 46942 32045 AQP4 361 ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME SUMATRIPTAN SUMATRIPTAN 18572411 46943 32046 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE Clocortolone CLOCORTOLONE 46944 32047 BAP1 8314 PROTEASE, TUMOR SUPPRESSOR, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE PANOBINOSTAT PANOBINOSTAT 22038994 46946 32048 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE SB3 46948 32049 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR FR139317 46949 32050 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL511142 BUPRENORPHINE 46950 32051 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIFLORASONE DIACETATE DIFLORASONE DIACETATE 46951 32052 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE GLABRIDIN GLABRIDIN 46952 32053 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-22 46953 32054 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME SOMATOTROPIN HUMAN GROWTH HORMONE 9834461 46954 32055 RGS4 5999 DRUGGABLE GENOME BAY-11-7085 BAY-11-7085 46956 32056 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PINDOLOL PINDOLOL 2903243 46957 32057 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME GF-109203 GF-109203 46958 32058 HNMT 3176 ENZYME, DRUGGABLE GENOME aspirin ASPIRIN 19178400 46959 32059 PRDX1 5052 ENZYME ANTIOXIDANT 9388242 46960 32060 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME REV-5901 REV-5901 46961 32061 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME DACTOLISIB DACTOLISIB 46962 32062 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ATG 7732566 46964 32063 RIT1 6016 CLINICALLY ACTIONABLE SELUMETINIB SELUMETINIB 24469055 46966 32064 PDE4D 5144 DRUGGABLE GENOME, ENZYME CC-1088 CDC-801 46967 32065 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE irinotecan IRINOTECAN 18347181 46969 32066 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9670220, 76 46970 32067 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 46971 32068 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHOSALONE PHOSALONE 46977 32069 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyrimidine derivative 6 46978 32070 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3545096 BGT-226 46981 32071 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME DETD-35 27048951 46982 32072 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1230609 FORETINIB 46985 32073 MUC16 94025 DRUGGABLE GENOME CHEMBL2107917 OREGOVOMAB 46988 32074 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor 252166686 46991 32075 PPP1R1A 5502 NA INSULIN INSULIN 10334321 46992 32076 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1,5-DINITRO-NAPHTHALENE CHEMBL167316 46994 32077 APC 324 CLINICALLY ACTIONABLE Fluorouracil FLUOROURACIL 27626067 46995 32078 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME BAY-11-7082 CHEMBL403183 16680159 46996 32079 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME METHOTRIMEPRAZINE LEVOMEPROMAZINE 46997 32080 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR inhibitor 178103591 46998 32081 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL3707183 QUINIDINE SULFATE 46999 32082 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Hexahydro azepinone derivative 1 47000 32083 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Sirolimus SIROLIMUS 21468343,23454836,1689463 47001 32084 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR PIMASERTIB PIMASERTIB 47003 32085 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE cyclophosphamide CYCLOPHOSPHAMIDE 47004 32086 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651360 47005 32087 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 385612186 47006 32088 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE STROPHANTHIDIN STROPHANTHIDIN 47007 32089 ALOX15 246 ENZYME, DRUGGABLE GENOME Imidazole derivative 10 47009 32090 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 COLCHICINE COLCHICINE 22931300 47010 32091 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME WAY-629 CHEMBL258465 47011 32092 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR SB-220025 SB-220025 47013 32093 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE EMBELIN EMBELIN 47016 32094 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR CISPLATIN CISPLATIN 9427537,8968078 47017 32095 ALDH1A1 216 DRUGGABLE GENOME, ENZYME EDARAVONE EDARAVONE 47018 32096 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ICI-199,441 ICI-199,441 47021 32097 DHRS9 10170 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE (+/-)-WIEDENDIOL B (+/-)-WIEDENDIOL B 19188072 47022 32098 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051815 47023 32099 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565855 47024 32100 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL1230607 PHA-793887 47027 32101 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX TAMARIXETIN TAMARIXETIN 25190466 47028 32102 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL2107797 NORGESTREL 47029 32103 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2-MERCAPTONICOTINIC ACID 2-MERCAPTONICOTINIC ACID 47032 32104 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 223366023 47034 32105 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ENDOSULFAN ENDOSULFAN 47035 32106 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PHENYLEPHRINE PHENYLEPHRINE 47037 32107 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 223366123 BARICITINIB 47039 32108 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 47040 32109 ALDH1A1 216 DRUGGABLE GENOME, ENZYME VANITIOLIDE VANITIOLIDE 47041 32110 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 363894131 47042 32111 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 4-METHYLBENZOIC ACID METHYL ESTER 4-METHYLBENZOIC ACID METHYL ESTER 47043 32112 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE COCAINE COCAINE 47045 32113 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME TAE-684 TAE-684 47047 32114 XDH 7498 DRUGGABLE GENOME, ENZYME theophylline THEOPHYLLINE 47049 32115 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650681 NALMEFENE 47050 32116 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ibuprofen IBUPROFEN 25502615 47051 32117 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178102325 PAZOPANIB 47052 32118 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-1010 CHEMBL1688556 47053 32119 OGFR 11054 NA IRT-102 47054 32120 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Monoaryl-1,2-diamine derivative 2 47055 32121 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 249565846 47056 32122 ALDH1A1 216 DRUGGABLE GENOME, ENZYME THIRAM THIRAM 47057 32123 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ABI-011 47058 32124 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER silibinin SILIBININ 26595166 47059 32125 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ISOPROPYL PALMITATE ISOPROPYL PALMITATE 47060 32126 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CURCUMIN CURCUMIN 15999103 47061 32127 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR BI-D1870 CHEMBL573107 47062 32128 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor REGORAFENIB REGORAFENIB 47063 32129 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TYRPHOSTIN AG-835 CHEMBL261557 47065 32130 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor 178101973 47066 32131 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Carbamide derivative 9 47068 32132 ALDH1A1 216 DRUGGABLE GENOME, ENZYME OXYMETHOLONE OXYMETHOLONE 47070 32133 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Talazoparib TALAZOPARIB 26546619,23881923,28242752 47072 32134 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLUTAMIDE FLUTAMIDE 16055512 47073 32135 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL547 ISOTRETINOIN 47074 32136 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545293 FGF401 47075 32137 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PENICILLIN PENICILLIN G POTASSIUM 17257217 47076 32138 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Cisplatin CISPLATIN 25519148 47077 32139 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 354702204 DEZAPELISIB 47079 32140 C8ORF34 116328 CLINICALLY ACTIONABLE, KINASE irinotecan IRINOTECAN 22664479 47080 32141 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE M7824 M-7824 47081 32142 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 223366140 47084 32143 CES1 1066 DRUGGABLE GENOME, ENZYME Dabigatran DABIGATRAN 23467860,27261537 47085 32144 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE Epigallocatechin gallate 47087 32145 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TPX-0005 47089 32146 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1064 SIMVASTATIN 47091 32147 REEP5 7905 NA fluoxetine FLUOXETINE 22795047 47092 32148 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE GSI-136 GSI-136 47093 32149 GPR183 1880 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178101168 47094 32150 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 47095 32151 KDM4A 9682 DRUGGABLE GENOME, ENZYME N-(2-phenylcyclopropyl) amino acid derivative 1 47096 32152 GJB3 2707 TRANSPORTER, ION CHANNEL inhibitor 135650269 47097 32153 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Raloxifene RALOXIFENE 47098 32154 GMNN 51053 DRUGGABLE GENOME OCTRIZOLE OCTRIZOLE 47099 32155 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 47100 32156 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TIOXOLONE TIOXOLONE 47101 32157 ALDH1A1 216 DRUGGABLE GENOME, ENZYME EMODIN EMODIN 47102 32158 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-2950 CHEMBL602807 47104 32159 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL2108591 ELSILIMOMAB 47106 32160 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652026 47107 32161 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME ENTRECTINIB ENTRECTINIB 47109 32162 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME IC261 IC261 24592867 47111 32163 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR US9611221, Example 9 47112 32164 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 178103584 47113 32165 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ALOE-EMODIN ALOE-EMODIN 16275083 47114 32166 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 252166678 47115 32167 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 47116 32168 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE AFATINIB AFATINIB 31068372,28950338,29802158,29169524,28502724 47117 32169 BRCA2 675 CLINICALLY ACTIONABLE CEDIRANIB CEDIRANIB 25218906 47118 32170 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE MORPHINE MORPHINE 47120 32171 RGS4 5999 DRUGGABLE GENOME 2-CHLORO-ADENOSINETRIPHOSPHATE CHEMBL1368696 47121 32172 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEHYDROEQUOL IDRONOXIL 47123 32173 SMN2 6607 DRUGGABLE GENOME AZARIBINE AZARIBINE 47126 32174 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME atorvastatin ATORVASTATIN 47129 32175 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GUANFACINE GUANFACINE 47130 32176 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME TCMDC-125758 CHEMBL546797 47132 32177 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ARANIDIPINE ARANIDIPINE 47133 32178 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 3-oxo-2,3-dihydro-1H-indazole-4-carboxamide derivative 1 47134 32179 F12 2161 DRUGGABLE GENOME, ENZYME, PROTEASE Enzymes 23280790 47135 32180 CFD 1675 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 252166508 47136 32181 IL1B 3553 KINASE, DRUGGABLE GENOME K-832 47137 32182 SERPINA6 866 DRUGGABLE GENOME, PROTEASE INHIBITOR Paramethasone PARAMETHASONE 47138 32183 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ACETOCHLOR ACETOCHLOR 47139 32184 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Bethanidine BETHANIDINE 47141 32185 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Irinotecan IRINOTECAN 47142 32186 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PD-153035 CHEMBL29197 47144 32187 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE NSC-74859 CHEMBL477936 47145 32188 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME EVEROLIMUS EVEROLIMUS 47146 32189 MMP16 4325 CELL SURFACE, DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103981 ILOMASTAT 47147 32190 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-21 47149 32191 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-52 47151 32192 MAPT 4137 DRUGGABLE GENOME DNDI1417519 CHEMBL1402376 47152 32193 IL13RA2 3598 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CINTREDEKIN BESUDOTOX 47154 32194 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE DCC-2618 RIPRETINIB 47155 32195 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 178102652 47156 32196 BAZ2B 29994 NA TCMDC-125764 CHEMBL586670 47157 32197 TARDBP 23435 TUMOR SUPPRESSOR MORUSINOL MORUSINOL 47158 32198 FAAH 2166 ENZYME, DRUGGABLE GENOME Boronic acid derivative 6 47159 32199 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Nicaraven NICARAVEN 47161 32200 TPSB2 64499 DRUGGABLE GENOME, PROTEASE SALT VOLANESORSEN SODIUM 3048411 47162 32201 ADAM17 6868 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, NEUTRAL ZINC METALLOPEPTIDASE, TRANSPORTER, ENZYME GW-3333 47165 32202 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051819 47166 32203 ATXN2 6311 NA TAMOXIFEN TAMOXIFEN 47167 32204 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178101093 47168 32205 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR oxaliplatin OXALIPLATIN 19786980,22188361,18347182,21902499,25069034,21057378,29662106,19362955,23314736,27498158,21262916,22026922,22329723 47169 32206 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-348401 CHEMBL515505 47170 32207 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KEPONE KEPONE 47171 32208 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ZAPA ZAPA 47173 32209 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SARACATINIB SARACATINIB 47175 32210 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME HYDROQUINONE HYDROQUINONE 47176 32211 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME NVP-BVB808 22271575 47178 32212 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CHLORPROPHAM CHLORPROPHAM 47180 32213 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Larotrectinib LAROTRECTINIB 47181 32214 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER vincristine VINCRISTINE 29938344,22016816,25637052,25582575,18408561 47182 32215 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor MK-2461 MK-2461 47184 32216 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CEFSULODIN SODIUM CEFSULODIN SODIUM 47185 32217 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TRICHOSTATIN A 12695546 47186 32218 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME NSC-164459 CHEMBL1567041 47187 32219 CXCL8 3576 DRUGGABLE GENOME GP-120 8995686 47188 32220 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE GNF-PF-5510 CHEMBL578741 47191 32221 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PHENDIMETRAZINE PHENDIMETRAZINE 47195 32222 KLF5 688 TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CID 926663 CHEMBL265686 47196 32223 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME RETINYL ACETATE 2897254 47197 32224 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 178100355 ZAFIRLUKAST 47198 32225 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HAEMATOXYLIN HAEMATOXYLIN 47202 32226 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 5,7-DIHYDROXYISOFLAVONE 5,7-DIHYDROXYISOFLAVONE 47203 32227 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME LOMOFUNGIN LOMOFUNGIN 47204 32228 PTGES 9536 DRUGGABLE GENOME, ENZYME celecoxib CELECOXIB 23778325 47205 32229 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME SULFASALAZINE SULFASALAZINE 9435300 47208 32230 FOLR2 2350 CELL SURFACE, DRUGGABLE GENOME LOMETREXOL LOMETREXOL 20085328 47209 32231 PTGS1 5742 ENZYME, DRUGGABLE GENOME TOLMETIN TOLMETIN 47210 32232 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR pertuzumab PERTUZUMAB 47211 32233 IL1B 3553 KINASE, DRUGGABLE GENOME LANSOPRAZOLE LANSOPRAZOLE 16815316 47212 32234 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 375973259 47213 32235 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Frovatriptan FROVATRIPTAN 47214 32236 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE AZD4721 47215 32237 ASS1 445 ENZYME, DRUG RESISTANCE Sodium Phenylbutyrate 47217 32238 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor 249565629 SOTRASTAURIN 47218 32239 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR VANDETANIB VANDETANIB 47219 32240 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME Blinatumomab BLINATUMOMAB 47221 32241 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GNF-PF-67 CHEMBL578512 47222 32242 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 381744995 SELITRECTINIB 47223 32243 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME PD-0166285 PD-0166285 47224 32244 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME DANTROLENE DANTROLENE 47225 32245 CTSC 1075 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 328083514 47227 32246 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor 178103915 EVOLOCUMAB 47228 32247 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME BLZ-945 47230 32248 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR N-(4-HYDROXYPHENYL)RETINAMIDE 12138118 47231 32249 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 2-CHLOROADENOSINE CHEMBL285819 47233 32250 POLB 5423 DNA REPAIR, DRUGGABLE GENOME HEXACHLOROPHENE HEXACHLOROPHENE 47234 32251 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL705 ALITRETINOIN 47235 32252 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Polyglutamate camptothecin 47236 32253 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3343 CHEMBL599943 47237 32254 POLK 51426 DNA REPAIR, ENZYME ERBSTATIN ERBSTATIN 47238 32255 MAOA 4128 DRUGGABLE GENOME, ENZYME CLORGILINE CLORGILINE 22078410 47239 32256 GMNN 51053 DRUGGABLE GENOME AURIN AURIN 47242 32257 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME Lanabecestat LANABECESTAT 47244 32258 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PRAZOSIN HYDROCHLORIDE PRAZOSIN HYDROCHLORIDE 47246 32259 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME allopurinol ALLOPURINOL 27798726 47249 32260 MAP2K6 5608 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE, TUMOR SUPPRESSOR inhibitor DABRAFENIB MESYLATE 47250 32261 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE GW441756X GW441756X 47252 32262 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-155693 CHEMBL68096 47253 32263 UGT1A7 54577 DRUGGABLE GENOME, ENZYME oxcarbazepine OXCARBAZEPINE 27900402 47254 32264 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MBX-8025 MBX-8025 47257 32265 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Huperzine A 47258 32266 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR modulator CHEMBL3707374 AMISELIMOD HYDROCHLORIDE 47260 32267 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-10 47262 32268 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ADJUVANT 7787697 47263 32269 CRLF2 64109 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME JAK INHIBITOR I 20018760 47265 32270 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-ACETYLAMINOFLUORENE 2-ACETYLAMINOFLUORENE 47266 32271 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Oncolym LYM-1 47269 32272 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DOCONEXENT DOCONEXENT 47270 32273 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651168 47271 32274 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 47272 32275 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Sym015 47273 32276 SRD5A1 6715 DRUGGABLE GENOME FINASTERIDE FINASTERIDE 47274 32277 POLI 11201 DNA REPAIR N-METHYLDOPAMINE HCL CHEMBL1256484 47275 32278 TUBA1A 7846 DRUGGABLE GENOME CHEMBL2103826 DAVUNETIDE 47276 32279 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL3544942 RONICICLIB 47278 32280 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-720622 CHEMBL1287980 47279 32281 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Peptide analog 52 47280 32282 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE COCAINE COCAINE 47281 32283 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Darifenacin DARIFENACIN 47282 32284 GMNN 51053 DRUGGABLE GENOME 4-HYDROXYDERRICIN CHEMBL458094 47283 32285 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 135650520 BEXAROTENE 47288 32286 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE LINIFANIB LINIFANIB 47290 32287 PSMB7 5695 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL2103884 OPROZOMIB 47292 32288 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE Sodium pyruvate 47293 32289 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PD-160170 CHEMBL422942 47294 32290 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE MITOXANTRONE MITOXANTRONE 47296 32291 SMN1 6606 DRUGGABLE GENOME 2-(STYRYL)-BENZIMIDAZOLE CHEMBL473721 47298 32292 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650246 ETORPHINE 47299 32293 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE VEMURAFENIB VEMURAFENIB 24265155 47300 32294 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL ADINAZOLAM ADINAZOLAM 47302 32295 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Midostaurin MIDOSTAURIN 26725216 47304 32296 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR TRAIL 16153452,16984382 47306 32297 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565868 47307 32298 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE SIROLIMUS SIROLIMUS 24893224,24836070 47308 32299 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Imatinib IMATINIB 47309 32300 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR 4-HYDROXYBENZOHYDRAZIDE CHEMBL124267 47311 32301 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME RG-1530 RG-1530 47312 32302 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ADEFOVIR DIPIVOXIL ADEFOVIR DIPIVOXIL 47313 32303 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME 2-CDA CLADRIBINE 12473386 47314 32304 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PROPANTHELINE PROPANTHELINE 47315 32305 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ritonavir RITONAVIR 24433361 47317 32306 GDA 9615 ENZYME 8-AZAGUANINE 8-AZAGUANINE 7384171 47318 32307 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME agonist 178100891 47319 32308 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ESTRONE ESTRONE 47321 32309 SMAD7 4092 KINASE GED-0301 MONGERSEN SODIUM 47322 32310 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CLOBETASOL CLOBETASOL 47323 32311 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME Tricyclic benzimidazole derivative 1 47324 32312 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENYLPYRUVATE PHENYLPYRUVATE 47326 32313 TARDBP 23435 TUMOR SUPPRESSOR JNJ-1661010 CHEMBL460273 47327 32314 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1684984 PA-799 47328 32315 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Bevacizumab + Trastuzumab 47329 32316 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR VALPROIC ACID VALPROIC ACID 18294844,16921367,25304896 47330 32317 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR Pyrrolidine carboxamide derivative 1 47331 32318 TUBA3D 113457 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 47334 32319 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PD-325901 47335 32320 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE Resimmune RESIMMUNE 47336 32321 KDM4A 9682 DRUGGABLE GENOME, ENZYME MECLIZINE DIHCL MECLIZINE DIHCL 47337 32322 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME RG-1530 RG-1530 47338 32323 AKR1C3 8644 ENZYME, DRUGGABLE GENOME 3-[(4-ACETYLPHENYL)AMINO]BENZOIC ACID CHEMBL1682201 22263837 47339 32324 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL197672 EMRICASAN 47340 32325 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME ARC1905 AVACINCAPTAD PEGOL SODIUM 47341 32326 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FENPYROXYMATE FENPYROXYMATE 47342 32327 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-34 47343 32328 DLK1 8788 DRUGGABLE GENOME GDC0134 47344 32329 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 252166577 PRACINOSTAT 47345 32330 MAPT 4137 DRUGGABLE GENOME 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 47346 32331 MVK 4598 KINASE, ENZYME inhibitor 135651490 47347 32332 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 178103636 47348 32333 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR RAD-1901 ELACESTRANT 47349 32334 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-292213 CHEMBL222808 47350 32335 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor CHEMBL2103879 GANETESPIB 47351 32336 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor BMS-754807 BMS-754807 47356 32337 KDM4A 9682 DRUGGABLE GENOME, ENZYME 6-METHOXY-HARMALAN CHEMBL338115 47357 32338 ALDH1A1 216 DRUGGABLE GENOME, ENZYME IODOFORM IODOFORM 47359 32339 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 387065624 47360 32340 APC 324 CLINICALLY ACTIONABLE HISTONE DEACETYLASE INHIBITOR 15087381 47362 32341 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Depudecin DEPUDECIN 47363 32342 BAZ2B 29994 NA N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 47364 32343 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DAPHNETIN DAPHNETIN 47365 32344 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-5102 CHEMBL603031 47368 32345 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME methotrexate METHOTREXATE 21317831 47371 32346 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ATENOLOL ATENOLOL 47372 32347 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Cetuximab CETUXIMAB 26715098,25714871,28446642,25724520,25838391,28424201,27002107 47373 32348 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL2107762 NERISPIRDINE 47374 32349 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE CHENODIOL CHENODIOL 19102680 47375 32350 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ROXINDOLE ROXINDOLE 47376 32351 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE RG-1530 RG-1530 47377 32352 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME PHA-767491 CHEMBL225519 47378 32353 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE 47379 32354 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Piperidine derivative 5 47380 32355 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PD-160170 CHEMBL422942 47382 32356 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545307 MERESTINIB 47383 32357 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER HDM201 47388 32358 ATAD5 79915 NA SU-4312 CHEMBL328710 47391 32359 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME 5'-FORMYLGLABRIDIN CHEMBL599165 20022509 47394 32360 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor REGORAFENIB REGORAFENIB 47396 32361 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL593430 ATAGABALIN 47397 32362 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR inhibitor 387065598 PF-06821497 47398 32363 GRB2 2885 NA ACTINOMYCIN D 15964235 47399 32364 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2010077680 103 47400 32365 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CLORINDIONE CLORINDIONE 47401 32366 GMNN 51053 DRUGGABLE GENOME PYRITHIONE PYRITHIONE 47402 32367 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme12-4 47403 32368 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TRIFLUOPERAZINE TRIFLUOPERAZINE 47404 32369 GMNN 51053 DRUGGABLE GENOME GNF-PF-4300 CHEMBL585656 47405 32370 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GDC-0941 PICTILISIB 22084396,22693356,19165201,26725216,22952903 47407 32371 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TESMILIFENE TESMILIFENE 47408 32372 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TUBASTATIN A TUBASTATIN A 25899338 47413 32373 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TCMDC-123764 CHEMBL533226 47414 32374 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SJ000029642 CHEMBL591126 47415 32375 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME A-23187 CALCIMYCIN 47416 32376 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 3,6-DIPHENYL-[1,2,4,5]TETRAZINE CHEMBL17784 47417 32377 IFNG 3458 DRUGGABLE GENOME IBUPROFEN IBUPROFEN 8931897 47419 32378 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE RV001 TEPROTUMUMAB 47420 32379 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PUERARIN PUERARIN 16038533 47422 32380 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR atorvastatin ATORVASTATIN 47423 32381 ENO2 2026 CELL SURFACE FENRETINIDE FENRETINIDE 17110918 47424 32382 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Insulin transdermal 47425 32383 HK1 3098 ENZYME, KINASE ADENOVIRUS VECTOR 8804424 47426 32384 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME LY3009120 LY-3009120 26343583,22798288,26732095 47429 32385 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CRA-024781 ABEXINOSTAT 47431 32386 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE agonist CHEMBL2108557 TELBERMIN 47433 32387 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor LINSITINIB LINSITINIB 47434 32388 ATXN2 6311 NA NSC-95397 CHEMBL429095 47435 32389 DEFA5 1670 DRUGGABLE GENOME SALT VOLANESORSEN SODIUM 9169780 47439 32390 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CABOZANTINIB CABOZANTINIB 47441 32391 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Sulfonamide derivative 7 47442 32392 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-155693 CHEMBL68096 47443 32393 DGAT1 8694 ENZYME, DRUGGABLE GENOME Lactam derivative 4 47445 32394 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BUTYLATED HYDROXYTOLUENE BUTYLATED HYDROXYTOLUENE 22931300 47446 32395 KCNA7 3743 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 47448 32396 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE Y-9680 47449 32397 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PD-0118057 CHEMBL521083 47450 32398 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHIMAZOLE METHIMAZOLE 10053173 47452 32399 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist CHEMBL1393 SPIRONOLACTONE 47453 32400 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CEPHALOCHROMIN CEPHALOCHROMIN 47456 32401 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE RETINOIC ACID 2465548 47457 32402 S100B 6285 DRUGGABLE GENOME, KINASE ONO-2506 47459 32403 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME entrectinib ENTRECTINIB 47460 32404 MAPK7 5598 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 249565744 47461 32405 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME LOBARIC ACID LOBARIC ACID 47462 32406 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3545248 DS-7423 47463 32407 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL2108313 CONBERCEPT 47465 32408 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE carboplatin CARBOPLATIN 47466 32409 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Imipramine IMIPRAMINE 47468 32410 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201152 NALMEFENE HYDROCHLORIDE 47469 32411 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL OPC-14523 47471 32412 SAE1 10055 ENZYME, DRUGGABLE GENOME PEVONEDISTAT PEVONEDISTAT 47473 32413 NOS1 4842 DRUGGABLE GENOME, ENZYME ANALGESICS 8880855 47474 32414 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR antagonist HGS 1029 47475 32415 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SAPONIN 16939894 47476 32416 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME DIOSMETIN DIOSMETIN 25190466 47478 32417 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ivermectin IVERMECTIN 47479 32418 GJC1 10052 ION CHANNEL inhibitor 178101095 OCTANOL 47482 32419 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Carbamide derivative 18 47483 32420 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TANSHINONE IIA TANSHINONE IIA 47484 32421 ATAD5 79915 NA LEFLUNOMIDE LEFLUNOMIDE 47485 32422 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103496 47486 32423 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME BMS-936564 ULOCUPLUMAB 47489 32424 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE TCMDC-125758 CHEMBL546797 47491 32425 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 385612180 47492 32426 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR DOVITINIB DOVITINIB 47493 32427 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178100447 47497 32428 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102751 47498 32429 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME ANTINEOPLASTIC 9515813 47500 32430 CDK12 51755 KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR, SERINE THREONINE KINASE OLAPARIB OLAPARIB 24240700 47501 32431 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1628688 ZIBOTENTAN 47502 32432 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME dasatinib DASATINIB 47503 32433 GMNN 51053 DRUGGABLE GENOME NSC-50690 CHEMBL1388703 47506 32434 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 178102328 PI-103 47507 32435 MAOA 4128 DRUGGABLE GENOME, ENZYME 8-(3-BROMOPHENOXYMETHYL)CAFFEINE CHEMBL2088301 22705191 47510 32436 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CYAZOFAMID CYAZOFAMID 47511 32437 BAZ2B 29994 NA DNDI1417147 CHEMBL2094484 47512 32438 FKBP5 2289 DRUGGABLE GENOME corticosteroids 21788965 47513 32439 DCPS 28960 ENZYME, DRUGGABLE GENOME RG3039 47514 32440 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Panobinostat PANOBINOSTAT 47517 32441 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME PMID28594589-Compound-TABLE3C1 47518 32442 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Anti-CD20-CAR-transduced T cells 47519 32443 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Imidazo quinoline derivative 1 47520 32444 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MEGESTROL ACETATE MEGESTROL ACETATE 47521 32445 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 252166785 47522 32446 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Bevacizumab BEVACIZUMAB 28408243 47525 32447 HMGCR 3156 ENZYME, DRUGGABLE GENOME Lactol derivative 2 47526 32448 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 340590256 TRILACICLIB 47527 32449 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor AT9283 AT-9283 47528 32450 SMN1 6606 DRUGGABLE GENOME 10-METHOXYLRUTAECARPINE CHEMBL85826 47530 32451 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LINOLENIC ACID LINOLENIC ACID 47531 32452 ATAD2 29028 NUCLEAR HORMONE RECEPTOR, ENZYME inhibitor 336446907 47532 32453 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SB-242235 SB-242235 47537 32454 GMNN 51053 DRUGGABLE GENOME AZACITIDINE AZACITIDINE 47538 32455 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME agonist CHEMBL1201565 EPOETIN ALFA 47539 32456 ATAD5 79915 NA GNF-PF-3501 CHEMBL581910 47540 32457 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE TESETAXEL TESETAXEL 47541 32458 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME STI571 IMATINIB MESYLATE 12509383 47542 32459 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-45a 47543 32460 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1416969 CHEMBL1453126 47544 32461 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TYROSINE KINASE INHIBITOR 15713908 47545 32462 APOC3 345 ENZYME, DRUGGABLE GENOME ritonavir RITONAVIR 15809899 47547 32463 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103006 APIXABAN 47549 32464 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME NSC-228155 CHEMBL505670 47550 32465 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR QUINIZARIN QUINIZARIN 47551 32466 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PK-11195 PK-11195 47552 32467 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE XMT-1001 47553 32468 SLC22A11 55867 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER PROBENECID PROBENECID 47554 32469 NDUFAF2 91942 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 47555 32470 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL2105705 LUNACALCIPOL 47556 32471 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ETIDRONIC ACID ETIDRONIC ACID 22931300 47558 32472 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME (-)-HERDMANINE I CHEMBL2208196 23189988 47559 32473 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LEVONORDEFRIN LEVONORDEFRIN 47561 32474 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE OSI-632 OSI-632 47563 32475 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR TAMATINIB R-406 47566 32476 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME CLOTRIMAZOLE CLOTRIMAZOLE 47568 32477 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE TZT-1027 SOBLIDOTIN 11855751 47569 32478 EPHB4 2050 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL403989 TG100-801 47572 32479 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE 2-CARBOPEROXYBENZOATE CHEMBL1162414 18595691 47573 32480 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565885 47574 32481 GAA 2548 DRUGGABLE GENOME, ENZYME TRIAMTERENE TRIAMTERENE 47575 32482 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TRASTUZUMAB TRASTUZUMAB 47576 32483 GMNN 51053 DRUGGABLE GENOME DNDI1417086 CHEMBL1224755 47577 32484 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME inhibitor 135650523 LINOPIRDINE 47578 32485 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1201065 THIAMYLAL SODIUM 47581 32486 CACNB4 785 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200382 BEPRIDIL HYDROCHLORIDE 47582 32487 KLK1 3816 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166697 47583 32488 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME DES DIETHYLSTILBESTROL 1980008 47586 32489 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DSM-106 CHEMBL444928 47587 32490 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist 178100437 47588 32491 SERPINA1 5265 DRUGGABLE GENOME, PROTEASE INHIBITOR Alpha1-proteinase inhibitor (human) modified process 47589 32492 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OSI-930 OSI-930 21068193 47590 32493 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ROMIDEPSIN ROMIDEPSIN 47592 32494 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BGJ398 INFIGRATINIB 47593 32495 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE SCHISANHENOL SCHISANHENOL 47595 32496 NOS1 4842 DRUGGABLE GENOME, ENZYME CARVEDILOL CARVEDILOL 16580580 47596 32497 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CetuGEX 47599 32498 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32b 47601 32499 GAPDH 2597 DRUGGABLE GENOME, ENZYME 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 47603 32500 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 5 47604 32501 CA2 760 DRUGGABLE GENOME, ENZYME SULFAMIDE SULFAMIDE 47605 32502 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE BMS-536924 CHEMBL401930 21804605 47608 32503 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MK-3207 MK3207 47609 32504 ATF4 468 TRANSPORTER, TRANSCRIPTION FACTOR VITAMIN E 11043924 47610 32505 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR 2-PHENYLACETYLAMINOBENZOTHIAZOLE CHEMBL1405979 47611 32506 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR ALPHA-TOCOPHEROL VITAMIN E 16909121 47612 32507 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 47614 32508 HTT 3064 DRUGGABLE GENOME PMID29671355-Compound-53 47615 32509 NTS 4922 DRUGGABLE GENOME haloperidol HALOPERIDOL 27023437 47617 32510 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 4-(HEXYLOXY)PHENOL CHEMBL225563 47621 32511 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NSC-255523 CHEMBL519155 18467108 47623 32512 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME modulator CHEMBL146506 MOFAROTENE 47624 32513 ATXN2 6311 NA DNDI1417400 CHEMBL1362503 47626 32514 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE ALSTERPAULLONE ALSTERPAULLONE 47628 32515 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DUTASTERIDE DUTASTERIDE 47630 32516 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ALTHIAZIDE ALTHIAZIDE 47631 32517 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antibody RAMUCIRUMAB RAMUCIRUMAB 47632 32518 MAPT 4137 DRUGGABLE GENOME LY-367265 CHEMBL1079460 47633 32519 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME AG-537 CHEMBL67535 47635 32520 CD9 928 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE INTERLEUKIN-16 16144798 47636 32521 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL HALOPERIDOL HALOPERIDOL 22055714 47638 32522 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME atorvastatin ATORVASTATIN 17700359 47640 32523 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE NORETHINDRONE NORETHINDRONE 1442974 47641 32524 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PYRIPROXYFEN PYRIPROXYFEN 47642 32525 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Pimozide PIMOZIDE 47643 32526 RABEP1 9135 CLINICALLY ACTIONABLE, GROWTH FACTOR mirtazapine MIRTAZAPINE 28694205 47644 32527 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR IDOXIFENE IDOXIFENE 11588112 47645 32528 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE ENMD-2076 ENMD-2076 47649 32529 MGLL 11343 DRUGGABLE GENOME, ENZYME Azetidinyl-piperidine derivative 2 47650 32530 ATIC 471 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PEMETREXED PEMETREXED 24256410 47652 32531 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR STREPTOZOCIN STREPTOZOCIN 16342200 47653 32532 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE OSI-632 OSI-632 47654 32533 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR TROGLITAZONE TROGLITAZONE 11553036 47657 32534 UBA1 7317 ENZYME HIMEIC ACID A HIMEIC ACID A 22695182 47659 32535 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MAKALUVAMINE F MAKALUVAMINE F 8691207 47660 32536 DGAT1 8694 ENZYME, DRUGGABLE GENOME Lactam derivative 5 47661 32537 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE GSK-269962A GSK-269962A 47662 32538 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MEPERIDINE MEPERIDINE 47663 32539 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135650610 47664 32540 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PT-103 CHEMBL398765 47665 32541 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DAPOXETINE DAPOXETINE 47666 32542 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649666 47667 32543 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR ALSTERPAULLONE ALSTERPAULLONE 47668 32544 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 47670 32545 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SB-242084 SB-242084 47672 32546 PLA2G7 7941 DRUGGABLE GENOME, ENZYME ERYTHROPOIETIN EPOETIN BETA 16421163 47674 32547 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE fluorouracil FLUOROURACIL 47676 32548 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2012520 LY377604 47677 32549 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HOMATROPINE HYDROBROMIDE HOMATROPINE HYDROBROMIDE 47681 32550 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor 249565819 47682 32551 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2,4-HEXADIENAL 2,4-HEXADIENAL 47684 32552 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR HALOBETASOL PROPIONATE 47685 32553 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE inhibitor 404859161 ALOXISTATIN 47686 32554 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HEPTACHLOR HEPTACHLOR 47688 32555 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE KETANSERIN KETANSERIN 47690 32556 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FIPEXIDE FIPEXIDE 47691 32557 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE antibody 340590228 ROVELIZUMAB 47692 32558 ARSA 410 DRUGGABLE GENOME, ENZYME 6-HYDROXYMELATONIN CHEMBL127421 47693 32559 VKORC1 79001 DRUGGABLE GENOME, ENZYME PHENINDIONE PHENINDIONE 47694 32560 HTT 3064 DRUGGABLE GENOME ACY-1215 RICOLINOSTAT 26031917 47697 32561 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR ACE-011 SOTATERCEPT 47698 32562 PTPN6 5777 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SORAFENIB SORAFENIB 22871485 47699 32563 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200443 MERETHOXYLLINE PROCAINE 47701 32564 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Rimexolone RIMEXOLONE 47703 32565 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Flutamide FLUTAMIDE 47704 32566 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR SANGUINARIUM SANGUINARIUM 47705 32567 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102716 47706 32568 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE SP-600125 SP-600125 23634759 47707 32569 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR RG-1530 RG-1530 47708 32570 PHF8 23133 ENZYME, DRUGGABLE GENOME inhibitor 178103604 47711 32571 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME inhibitor 249565704 LONAFARNIB 47712 32572 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL ALLYL ISOTHIOCYANATE ALLYL ISOTHIOCYANATE 26263397 47713 32573 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 404859119 47714 32574 HSPA4 3308 NA CHELATORS 11579132 47715 32575 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER CLIOXANIDE CLIOXANIDE 47717 32576 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-27 47718 32577 LPAR2 9170 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE MORPHINE MORPHINE 17090705 47719 32578 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CAR-T cells targeting HER2 47720 32579 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 178102314 IMATINIB 47721 32580 TUBA1C 84790 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 47724 32581 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DESOGESTREL DESOGESTREL 47725 32582 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HALOPROGIN HALOPROGIN 47726 32583 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AC480 AC-480 47730 32584 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY GENISTEIN GENISTEIN 16475902 47734 32585 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Anti-CD19 anti-CD20 Bispecific CAR-T 47735 32586 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NICARDIPINE HYDROCHLORIDE NICARDIPINE HYDROCHLORIDE 47737 32587 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR bevacizumab BEVACIZUMAB 29871907 47739 32588 SQLE 6713 DRUGGABLE GENOME, ENZYME AMIODARONE AMIODARONE 16451055 47740 32589 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME hydrocodone HYDROCODONE 9352573,12920424,25621429,24269714,20837591,7693389,16631290 47741 32590 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Perifosine PERIFOSINE 25519148 47742 32591 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650290 47743 32592 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME THROMBIN THROMBIN 8598231 47744 32593 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE ERLOTINIB ERLOTINIB 47745 32594 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 47746 32595 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE GOSSYPOL GOSSYPOL 47747 32596 CLK1 1195 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE HARMINE HARMINE 22998443 47748 32597 GMNN 51053 DRUGGABLE GENOME DNDI1417607 CHEMBL1588679 47749 32598 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000147993 CHEMBL601618 47750 32599 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Imidazo pyridine derivative 1 47751 32600 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SB-220025 SB-220025 47752 32601 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Cipatinib 47753 32602 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL416146 ETORICOXIB 47755 32603 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor CHEMBL2364655 EVOLOCUMAB 47756 32604 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-180736A GSK-180736A 47757 32605 IFNG 3458 DRUGGABLE GENOME AUTOLOGOUS LYMPHOCYTES 7750192 47758 32606 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 252166595 BIMIRALISIB 47759 32607 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-23 47761 32608 PSMA8 143471 DRUGGABLE GENOME, PROTEASE inhibitor CARFILZOMIB CARFILZOMIB 47763 32609 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME DIETHYL-2-DODECYLIDENEMALONATE CHEMBL1797708 21292492 47765 32610 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME IFN 2499691 47766 32611 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME flibanserin FLIBANSERIN 47767 32612 POU2F2 5452 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LINAGLIPTIN LINAGLIPTIN 23073734 47768 32613 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME U-73122 CHEMBL1256678 47769 32614 APOE 348 DRUGGABLE GENOME GINKGO BILOBA 12684092 47770 32615 KCNT2 343450 ION CHANNEL, DRUGGABLE GENOME phorbol 12-myristate 13-acetate 47771 32616 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 348353643 47772 32617 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DNDI1417254 CHEMBL2094567 47773 32618 MPHOSPH8 54737 NA R(-)-APOCODEINE HCL CHEMBL1256735 47774 32619 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Lapatinib LAPATINIB 27108243 47775 32620 CDC42BPA 8476 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ALSTERPAULLONE ALSTERPAULLONE 47778 32621 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUOCINONIDE FLUOCINONIDE 47781 32622 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DNDI1417132 CHEMBL1492017 47782 32623 UBE2N 7334 ENZYME, DRUGGABLE GENOME TCMDC-124495 CHEMBL532452 47783 32624 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROMETHAZINE HYDROCHLORIDE PROMETHAZINE HYDROCHLORIDE 47784 32625 PDE3A 5139 ENZYME, DRUGGABLE GENOME AMRINONE INAMRINONE 47785 32626 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Staurosporine STAUROSPORINE 47786 32627 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE UB-311 24476230 47787 32628 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME rituximab RITUXIMAB 47788 32629 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SANGUINARIUM SANGUINARIUM 47789 32630 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE THALIDOMIDE THALIDOMIDE 47790 32631 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-49789 CHEMBL469309 47791 32632 FAAH2 158584 DRUGGABLE GENOME, ENZYME inhibitor 178101919 47793 32633 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ICI-199,441 ICI-199,441 47794 32634 HTT 3064 DRUGGABLE GENOME D-TRYPTOPHAN D-TRYPTOPHAN 47796 32635 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Glipizide GLIPIZIDE 47797 32636 BRDT 676 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE MIDAZOLAM MIDAZOLAM 22137933 47798 32637 ALOX15 246 ENZYME, DRUGGABLE GENOME CITRONELLOL CITRONELLOL 47800 32638 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR NEUROTROPHIC FACTOR 16716308 47801 32639 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 135650390 INDOMETHACIN 47803 32640 TUBA4A 7277 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 47805 32641 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor CHEMBL3544940 G1T28-1 47807 32642 SERPINA5 5104 PROTEASE INHIBITOR, ENZYME, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE HEPARIN HEPARIN 8136018 47808 32643 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Enzastaurin ENZASTAURIN 47809 32644 TUBA1B 10376 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 47810 32645 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TYRPHOSTIN AG-1478 TYRPHOSTIN AG-1478 47813 32646 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GITOXIGENIN GITOXIGENIN 47814 32647 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102928 CHEMBL1818218 47819 32648 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Dasatinib DASATINIB 47820 32649 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE CEFACLOR CEFACLOR 47821 32650 MAPT 4137 DRUGGABLE GENOME GNF-PF-1644 CHEMBL600734 47822 32651 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR acebutolol ACEBUTOLOL 47823 32652 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000113257 CHEMBL528694 47824 32653 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL3545176 DB959 47825 32654 HDAC11 79885 DRUGGABLE GENOME, ENZYME ROMIDEPSIN ROMIDEPSIN 47826 32655 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE DOX 15792348 47827 32656 XDH 7498 DRUGGABLE GENOME, ENZYME Azaindole derivative 3 47828 32657 BAZ2B 29994 NA 2',3,4-TRIHYDROXYCHALCONE CHEMBL339587 47830 32658 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor LEE011 RIBOCICLIB 47831 32659 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 47835 32660 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PYRAZOPHOS PYRAZOPHOS 47836 32661 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor 178103398 ACETAZOLAMIDE 47837 32662 ALDH1A1 216 DRUGGABLE GENOME, ENZYME KAINIC ACID KAINIC ACID 47838 32663 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RG-2833 47839 32664 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME QUERCETAGETIN QUERCETAGETIN 25190466 47842 32665 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR gemcitabine GEMCITABINE 22838950 47843 32666 TUBB4B 10383 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 47845 32667 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL1421 DASATINIB 47846 32668 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000082806 CHEMBL494668 47847 32669 RRM2B 50484 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL1750 CLOFARABINE 47848 32670 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME TRIMETHIDINIUM TRIMETHIDINIUM 47849 32671 HTT 3064 DRUGGABLE GENOME SJ000044511 CHEMBL592124 47852 32672 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 3-oxo-2,3-dihydro-1H-indazole-4-carboxamide derivative 4 47853 32673 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Imidazo pyridine derivative 2 47855 32674 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE JNJ-54175446 JNJ-54175446 47856 32675 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PROCATEROL PROCATEROL 47858 32676 MAPT 4137 DRUGGABLE GENOME NSC-69187 CHEMBL19954 47860 32677 ROR2 4920 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CELL SURFACE, ENZYME CCT301-38 (targeting ROR2) 47861 32678 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 COLCHICINE COLCHICINE 22931300 47862 32679 BAZ2B 29994 NA CEFOTIAM HYDROCHLORIDE CEFOTIAM HYDROCHLORIDE 47863 32680 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 2 47864 32681 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TAMOXIFEN TAMOXIFEN 47865 32682 EIF2AK2 5610 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR IL-3 7519779 47866 32683 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL3707357 BROLUCIZUMAB 47868 32684 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROTHIOFOS PROTHIOFOS 47869 32685 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GYKI-52466 GYKI-52466 47870 32686 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ETHACRYNIC ACID ETHACRYNIC ACID 47871 32687 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL378544 VINBLASTINE SULFATE 47872 32688 ALDH5A1 7915 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2105613 DIVALPROEX SODIUM 47873 32689 CA7 766 DRUGGABLE GENOME, ENZYME activator 178100344 HISTIDINE 47874 32690 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CUPRESSUFLAVONE CUPRESSUFLAVONE 47875 32691 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME LAUROGUADINE LAUROGUADINE 47878 32692 MAPT 4137 DRUGGABLE GENOME MMV006319 CHEMBL579105 47880 32693 GLS 2744 ENZYME COUMESTROL COUMESTROL 47881 32694 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SB-415286 CHEMBL322970 47883 32695 ATAD5 79915 NA GNF-PF-4463 CHEMBL584520 47884 32696 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE KINASE INHIBITOR 14521590 47885 32697 GPER1 2852 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR antagonist 178100354 47889 32698 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (-)-ASARININ CHEMBL1572261 47895 32699 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE RG3638 47896 32700 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IODOPHTHALEIN IODOPHTHALEIN 47897 32701 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 47898 32702 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ADJUVANT CHEMOTHERAPY 26899019 47899 32703 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME N-METHYL-D-ASPARTIC ACID (NMDA) N-METHYL-D-ASPARTIC ACID (NMDA) 47902 32704 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME GEMCITABINE GEMCITABINE 26057002 47903 32705 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-127133 CHEMBL1172911 22524450 47905 32706 ORAI1 84876 TRANSCRIPTION FACTOR, ION CHANNEL, TRANSPORTER RP4010 47906 32707 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1201146 NORETHINDRONE ACETATE 47907 32708 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE CAMPTOTHECIN CAMPTOTHECIN 14973057 47909 32709 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BENZODODECINIUM CHLORIDE BENZODODECINIUM CHLORIDE 47910 32710 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200977 MILRINONE LACTATE 47911 32711 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 47912 32712 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 4,2',4',6'-TETRAHYDROXYCHALCONE 4,2',4',6'-TETRAHYDROXYCHALCONE 47914 32713 ENO2 2026 CELL SURFACE TRIIODOTHYRONINE LIOTHYRONINE SODIUM 3455610 47915 32714 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Flibanserin FLIBANSERIN 47916 32715 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Masoprocol MASOPROCOL 47917 32716 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DAZOMET DAZOMET 47918 32717 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROPOXYPHENE PROPOXYPHENE 47921 32718 LTA 4049 DRUGGABLE GENOME carbamazepine CARBAMAZEPINE 11294926 47922 32719 TUBA1C 84790 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 47923 32720 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor 178101880 47924 32721 NBEA 26960 KINASE antidepressants 47925 32722 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Gefitinib GEFITINIB 47926 32723 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME inhibitor AZD6244 SELUMETINIB 47928 32724 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TYRPHOSTIN 25 TYRPHOSTIN 25 47929 32725 NUAK1 9891 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 310264757 47930 32726 KDM4A 9682 DRUGGABLE GENOME, ENZYME COLCHICEINE COLCHICEINE 47932 32727 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102758 47933 32728 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL2107358 OBATOCLAX MESYLATE 47934 32729 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650013 BNTX 47937 32730 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-38 47941 32731 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2043437 GLASDEGIB 47942 32732 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545155 JI-101 47943 32733 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL270995 BRIVANIB ALANINATE 47946 32734 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL193240 ROFLUMILAST 47947 32735 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor VEMURAFENIB VEMURAFENIB 47948 32736 CBX1 10951 NA BI-87E7 CHEMBL523200 47949 32737 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BN-AO-014 47950 32738 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102322 TANDUTINIB 47954 32739 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 47957 32740 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 47958 32741 TH 7054 ENZYME, DRUGGABLE GENOME DHEA PRASTERONE 8704732 47959 32742 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 252166736 47963 32743 PMEL 6490 DRUGGABLE GENOME HMBA 11310793 47965 32744 AAK1 22848 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME inhibitor 384403682 47966 32745 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL448 PENTOBARBITAL 47968 32746 MPHOSPH8 54737 NA IDARUBICIN IDARUBICIN 47969 32747 RCE1 9986 ENZYME, PROTEASE, DRUGGABLE GENOME SJ000293754 CHEMBL486706 47970 32748 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 178101884 GSK-690693 47971 32749 RPSA 3921 NA DOXORUBICIN DOXORUBICIN 11493465 47972 32750 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME 8-METHOXYPSORALEN METHOXSALEN 15711930 47974 32751 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL288441 BOSUTINIB 47975 32752 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor PAZOPANIB PAZOPANIB 47977 32753 TYMP 1890 GROWTH FACTOR, DRUGGABLE GENOME MPA PROGESTERONE 12711006 47978 32754 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR KAMEBANIN KAMEBANIN 47980 32755 CD47 961 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE TTI-621 47981 32756 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 7,8,3'-TRIHYDROXYFLAVONE CHEMBL225513 47982 32757 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE LY2801653 26757360,23275061,27694386 47985 32758 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE SB-220025 SB-220025 47986 32759 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200694 SEVOFLURANE 47988 32760 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ISOPROPAMIDE ISOPROPAMIDE 47989 32761 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE ALPHA-TOCOPHEROL VITAMIN E 14871472 47990 32762 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-339578 CHEMBL353764 47991 32763 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME hmg coa reductase inhibitors 25084202 47992 32764 KMO 8564 DRUGGABLE GENOME, ENZYME Benzene sulfonamide derivative 3 47993 32765 KDM4A 9682 DRUGGABLE GENOME, ENZYME MMV000704 CHEMBL582478 47994 32766 ARSA 410 DRUGGABLE GENOME, ENZYME 3,5-DINITROCATECHOL (OR-486) 3,5-DINITROCATECHOL (OR-486) 47995 32767 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 testosterone TESTOSTERONE 9187528 47997 32768 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 404859028 47999 32769 TARDBP 23435 TUMOR SUPPRESSOR DNDI1417560 CHEMBL1373255 48000 32770 GMNN 51053 DRUGGABLE GENOME GNF-PF-5134 CHEMBL602969 48001 32771 PTGS2 5743 DRUGGABLE GENOME, ENZYME Aminosalicylic Acid 48002 32772 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL315985 ESLICARBAZEPINE 48003 32773 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ATROPINE ATROPINE 48004 32774 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THEOPHYLLINE THEOPHYLLINE 48005 32775 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME ENOXAPARIN ENOXAPARIN 48006 32776 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SB-203580 SB-203580 25692815,19301816,17659871 48007 32777 KDM4A 9682 DRUGGABLE GENOME, ENZYME ERBSTATIN ERBSTATIN 48008 32778 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME E927A E927A 48010 32779 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL2159122 ELUXADOLINE 48012 32780 SMG1 23049 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DNA REPAIR ApoC-III 48013 32781 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME QUISQUALATE QUISQUALATE 48014 32782 GAL 51083 DRUGGABLE GENOME heroin DIACETYLMORPHINE 48016 32783 CCNA2 890 DRUGGABLE GENOME, KINASE TNF-ALPHA 15965500 48017 32784 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BROMUCONAZOLE BROMUCONAZOLE 48021 32785 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RETINOIDS 11223164,9417874,8839862,9334253,10441468 48022 32786 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ENTRECTINIB ENTRECTINIB 48025 32787 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER tipifarnib TIPIFARNIB 15122075 48026 32788 FES 2242 ENZYME, DRUGGABLE GENOME, KINASE, TYROSINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 48027 32789 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Beta blocking agents, non-selective 48028 32790 UBE2N 7334 ENZYME, DRUGGABLE GENOME SJ000160630 CHEMBL591404 48029 32791 HBB 3043 DRUGGABLE GENOME, ENZYME ELLIPTECINE ELLIPTECINE 48030 32792 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 375973268 48032 32793 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-747261 CHEMBL593366 48036 32794 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX PROTOAPIGENONE PROTOAPIGENONE 48037 32795 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MCP-1 16614397 48038 32796 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING TCMDC-125182 CHEMBL588143 48039 32797 GMNN 51053 DRUGGABLE GENOME CLOTRIMAZOLE CLOTRIMAZOLE 48040 32798 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL1684984 PA-799 48041 32799 RGS5 8490 NA irinotecan IRINOTECAN 25069475 48042 32800 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME OXYTOCIN OXYTOCIN 15590985 48043 32801 P2RX4 5025 ION CHANNEL, DRUGGABLE GENOME agonist 135651446 ADENOSINE TRIPHOSPHATE 48044 32802 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEXBUDESONIDE DEXBUDESONIDE 48045 32803 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor 310264693 ACALABRUTINIB 48047 32804 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIFENOCONAZOLE DIFENOCONAZOLE 48048 32805 ATAD5 79915 NA ALPHA,BETA-DEHYDROCURVULARIN CHEMBL482050 48051 32806 ALOX15 246 ENZYME, DRUGGABLE GENOME GNF-PF-5114 CHEMBL601952 48052 32807 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING CRIDANIMOD CRIDANIMOD 48053 32808 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure3-Lycojaponicumin A 48056 32809 GMNN 51053 DRUGGABLE GENOME BI-87E7 CHEMBL523200 48057 32810 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Piperidinyl triazole derivative 2 48062 32811 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 3 48064 32812 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYDROCORTISONE VALERATE HYDROCORTISONE VALERATE 48067 32813 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650689 NALTRINDOLE 48069 32814 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AG-494 CHEMBL56731 48072 32815 CBX1 10951 NA PHENOXYBENZAMINE PHENOXYBENZAMINE 48075 32816 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEFAZOLIN CEFAZOLIN 48076 32817 TUBB4B 10383 DRUGGABLE GENOME ABT-751 ABT-751 25468039 48078 32818 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor SORAFENIB SORAFENIB 48079 32819 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME NEFAZODONE NEFAZODONE 48081 32820 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER pantoprazole PANTOPRAZOLE 15976989 48082 32821 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME BESTATIN 12554354 48083 32822 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Dendritic cell vaccine 48084 32823 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200959 METHDILAZINE 48085 32824 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist 381118896 48086 32825 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 363894179 48087 32826 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000089001 CHEMBL591618 48088 32827 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR SAQUINAVIR SAQUINAVIR 15388451 48089 32828 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565731 48091 32829 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR LETROZOLE LETROZOLE 25524798 48092 32830 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PHA-767491 CHEMBL225519 48093 32831 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME (+)-THALIPORPHINE CHEMBL1397308 48094 32832 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103499 48096 32833 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE FENOTEROL FENOTEROL 48097 32834 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE amodiaquine AMODIAQUINE 48099 32835 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DES DIETHYLSTILBESTROL 15545218 48100 32836 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME XL999 48101 32837 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING BML-210 CHEMBL324053 16921367 48102 32838 SMN1 6606 DRUGGABLE GENOME CID 926663 CHEMBL265686 48104 32839 CBX1 10951 NA TRIFLUOPERAZINE TRIFLUOPERAZINE 48105 32840 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NINTEDANIB NINTEDANIB 48108 32841 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Temozolomide TEMOZOLOMIDE 25910950,26846818 48111 32842 BCHE 590 DRUGGABLE GENOME, ENZYME PHENOTHIAZINE PHENOTHIAZINE 12443046 48113 32843 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TERAZOSIN TERAZOSIN 22931300 48114 32844 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-95397 CHEMBL429095 48115 32845 MYD88 4615 CLINICALLY ACTIONABLE IBRUTINIB IBRUTINIB 25853747 48118 32846 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE EMODIC ACID EMODIC ACID 48120 32847 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565877 48121 32848 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GIMESTAT GIMERACIL 48122 32849 MPHOSPH8 54737 NA SANGUINARIUM CHLORIDE SANGUINARIUM CHLORIDE 48124 32850 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DIPHENHYDRAMINE DIPHENHYDRAMINE 48126 32851 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CROMOLYN CROMOLYN 22931300 48128 32852 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME ENCORAFENIB ENCORAFENIB 31566309,28363909,29573941 48129 32853 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Teneligliptin TENELIGLIPTIN 48131 32854 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL2109613 PF-04236921 48132 32855 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR CID2350207 CHEMBL259615 48133 32856 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 135651469 48134 32857 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME nevirapine NEVIRAPINE 20017669,23774940,19228205,17638512,20625352,27195527,21824325,11470993,21860339,15864119,28689274,22354160,21505298 48135 32858 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 8,2'-DIMETHOXYFLAVONE 8,2'-DIMETHOXYFLAVONE 48136 32859 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE OUABAIN OUABAIN 48137 32860 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE TG003 48140 32861 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650054 CARAZOLOL 48141 32862 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545133 JNJ-26483327 48142 32863 MAPT 4137 DRUGGABLE GENOME S(+)-ISOPROTERENOL-BITARTRATE CHEMBL1257092 48143 32864 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME GW9662 CHEMBL375270 48144 32865 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme25-2 48146 32866 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME GO-6976 GO-6976 48147 32867 XDH 7498 DRUGGABLE GENOME, ENZYME Azaindole derivative 5 48150 32868 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE Biphenyl carboxylic acid derivative 2 48151 32869 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME L-CYSTEINESULPHINIC ACID CHEMBL1160508 48153 32870 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME VEGF 15947259 48154 32871 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR eribulin ERIBULIN 48155 32872 NDUFA12 55967 ENZYME inhibitor CHEMBL3545320 ME-344 48156 32873 ATAD5 79915 NA NSC-353720 CHEMBL1408276 48157 32874 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR TYRPHOSTIN AG-835 CHEMBL261557 48158 32875 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Lenvatinib LENVATINIB 26169970 48159 32876 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME PMID27539678-Compound-17 48162 32877 TSPO 706 DRUGGABLE GENOME ZOLPIDEM ZOLPIDEM 48163 32878 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER HISTONE DEACETYLASE INHIBITOR 16223781 48164 32879 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DOXERCALCIFEROL DOXERCALCIFEROL 48167 32880 MBNL1 4154 DRUGGABLE GENOME NSC-95397 CHEMBL429095 48168 32881 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME BENZAMIL BENZAMIL 48171 32882 NDUFA3 4696 ENZYME inhibitor CHEMBL3545320 ME-344 48172 32883 PTGS2 5743 DRUGGABLE GENOME, ENZYME (R)-IBUPROPHEN (R)-IBUPROPHEN 20143779 48173 32884 HBB 3043 DRUGGABLE GENOME, ENZYME PolyHeme 18523531 48176 32885 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Trabectedin TRABECTEDIN 26036639 48178 32886 MARCHF8 220972 ENZYME H1N1 pandemic influenza A vaccine 48179 32887 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545324 RG-7666 48180 32888 SV2A 9900 DRUGGABLE GENOME, TRANSPORTER SELETRACETAM SELETRACETAM 48181 32889 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IBUDILAST IBUDILAST 48182 32890 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CETRIMONIUM BROMIDE CETRIMONIUM BROMIDE 48183 32891 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE RG-1530 RG-1530 48184 32892 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CHF 5407 48185 32893 GMNN 51053 DRUGGABLE GENOME GNF-PF-4786 CHEMBL602363 48186 32894 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CAULIBUGULONE C CAULIBUGULONE C 48188 32895 TUBB 203068 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 48189 32896 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178102295 AFATINIB 48190 32897 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651109 48191 32898 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-Table1Example4 48193 32899 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR IBUPROFEN IBUPROFEN 15217953 48194 32900 ATXN2 6311 NA DNDI1417076 CHEMBL1526167 48196 32901 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL TEMAZEPAM TEMAZEPAM 48197 32902 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PEG-IRINOTECAN 48198 32903 ATAD5 79915 NA TOLONIUM CHLORIDE TOLONIUM CHLORIDE 48199 32904 TOP2B 7155 DRUGGABLE GENOME, ENZYME DAUNORUBICIN DAUNORUBICIN 48202 32905 BAZ2B 29994 NA NIFEDIPINE NIFEDIPINE 48203 32906 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103101 48205 32907 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Carbamide derivative 5 48206 32908 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 650707 CHEMBL408653 48207 32909 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1513 IRBESARTAN 48211 32910 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SR-2640 SR-2640 48212 32911 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-11 48213 32912 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 328083488 CHEMBL401930 48215 32913 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Sulfadiazine SULFADIAZINE 48216 32914 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME (RS)-ROSCOVITINE (RS)-ROSCOVITINE 48217 32915 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SIGNAL TRANSDUCTION INHIBITORS 16926049 48220 32916 ADK 132 DRUGGABLE GENOME, ENZYME, KINASE DACARBAZINE DACARBAZINE 6317371 48222 32917 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX LOBARIC ACID LOBARIC ACID 48223 32918 DGAT1 8694 ENZYME, DRUGGABLE GENOME Pyridine-carboximide derivative 1 48225 32919 PSMB3 5691 PROTEASE, DRUGGABLE GENOME inhibitor CARFILZOMIB CARFILZOMIB 48226 32920 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 4-HYDROXYFLAVONOL CHEMBL272682 48227 32921 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHENYLBUTYRYLHYDROXAMIC ACID PHENYLBUTYRYLHYDROXAMIC ACID 21874153 48230 32922 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR BORTEZOMIB BORTEZOMIB 15813915 48232 32923 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME MYRICETIN MYRICETIN 48233 32924 KDM4A 9682 DRUGGABLE GENOME, ENZYME MIFEPRISTONE MIFEPRISTONE 48234 32925 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650495 48235 32926 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLOROXYLENOL CHLOROXYLENOL 48236 32927 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor CHEMBL574737 UCN-01 48239 32928 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE VINCLOZOLIN VINCLOZOLIN 48240 32929 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ENOXIMONE ENOXIMONE 48242 32930 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME Topical ruxolitinib 48243 32931 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GW7074 CHEMBL72365 48244 32932 MAP3K14 9020 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE inhibitor 249565854 48246 32933 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE IMATINIB IMATINIB 48248 32934 KDM4A 9682 DRUGGABLE GENOME, ENZYME inhibitor 252827402 48249 32935 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME VALINOMYCIN VALINOMYCIN 6129560 48250 32936 GLS 2744 ENZYME PMID30273516-Compound-13 48253 32937 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4-NONYLPHENOL 4-NONYLPHENOL 48254 32938 CLDN18 51208 KINASE, DRUGGABLE GENOME Claudiximab ZOLBETUXIMAB 48256 32939 POLK 51426 DNA REPAIR, ENZYME IRIGINOL HEXAACEATATE IRIGINOL HEXAACEATATE 48257 32940 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Leucovorin LEUCOVORIN 27626067 48258 32941 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 48259 32942 GPR183 1880 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178101172 48262 32943 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565601 ONVANSERTIB 48263 32944 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 3-METHYLCHOLANTHRENE 3-METHYLCHOLANTHRENE 48264 32945 GALNT14 79623 ENZYME cisplatin CISPLATIN 31611591,21635146 48266 32946 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME TCMDC-123730 CHEMBL530280 48267 32947 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651191 48268 32948 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER CEFACLOR CEFACLOR 22166395 48269 32949 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1,2-BENZANTHRACENE CHEMBL1873684 48270 32950 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ENTINOSTAT ENTINOSTAT 48271 32951 UMPS 7372 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE 5-FLUORO-6-AMIDO-UMP CHEMBL1164954 20452222 48272 32952 BAZ2B 29994 NA GNF-PF-5007 CHEMBL1989853 48274 32953 PDE4D 5144 DRUGGABLE GENOME, ENZYME MK-0873 MK-0873 48276 32954 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 381744930 48278 32955 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GNF-PF-2391 CHEMBL577415 48280 32956 UGT2B7 7364 DRUGGABLE GENOME ticagrelor TICAGRELOR 25935875 48281 32957 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 252827451 SAR-260301 48282 32958 MYB 4602 CLINICALLY ACTIONABLE DOXORUBICIN DOXORUBICIN 15001837 48285 32959 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIAMTERENE TRIAMTERENE 48286 32960 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ALPELISIB ALPELISIB 25002028 48287 32961 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1246786 CHEMBL1863271 48288 32962 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ZERANOL ZERANOL 48289 32963 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING HINOKITIOL HINOKITIOL 48290 32964 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE A-443654 A-443654 19465931 48291 32965 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 385612248 48292 32966 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Micardis telmisartan 48293 32967 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Oxetane 3,3-dicarboxamide compound 1 48295 32968 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Sunitinib SUNITINIB 27149458 48296 32969 PDGFA 5154 GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE inhibitor SUNITINIB SUNITINIB 48297 32970 SOD1 6647 ENZYME, DRUGGABLE GENOME TETRACYCLINE TETRACYCLINE 48299 32971 AMH 268 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RETINOIC ACID 8326606,7815634 48300 32972 PCSK2 5126 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 252166858 48301 32973 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SARALASIN SARALASIN 48302 32974 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PINDOLOL PINDOLOL 48303 32975 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651886 SOMATOSTATIN 48304 32976 EPHB4 2050 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE KD019 TESEVATINIB 48305 32977 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE DNDI1417467 CHEMBL1997335 48306 32978 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-95397 CHEMBL429095 48307 32979 COMT 1312 DRUGGABLE GENOME, ENZYME buprenorphine BUPRENORPHINE 30549211 48308 32980 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE THIDIAZURON THIDIAZURON 48309 32981 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SERTRALINE SERTRALINE 16680159 48312 32982 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME CHINIOFON CHINIOFON 48313 32983 HPSE 10855 ENZYME, DRUGGABLE GENOME PG545 48315 32984 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FIDUXOSIN HYDROCHLORIDE FIDUXOSIN HYDROCHLORIDE 48317 32985 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VACCINE 17120728 48320 32986 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER COTI-2 48321 32987 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PROTEASOME INHIBITOR 12532325 48325 32988 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME RAPAMYCIN SIROLIMUS 26619011,24631838 48328 32989 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE Nivocasan NIVOCASAN 48329 32990 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Pegloticase PEGLOTICASE 48330 32991 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SOTALOL SOTALOL 22931300 48332 32992 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 178100878 48333 32993 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME 4-METHYLDAPHNETIN 4-METHYLDAPHNETIN 48334 32994 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 252827367 OZANIMOD 48335 32995 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME PURPUROGALLIN PURPUROGALLIN 48336 32996 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE 7-HYDROXY ISOFLAVONE 7-HYDROXY ISOFLAVONE 48337 32997 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME GALLINAMIDE A GALLINAMIDE A 24364476 48338 32998 GSTM1 2944 DRUGGABLE GENOME, ENZYME CHLORAMBUCIL CHLORAMBUCIL 15044619 48340 32999 TUBA1A 7846 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 48341 33000 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 prasugrel PRASUGREL 48342 33001 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178100243 VALDECOXIB 48343 33002 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3545202 BERZOSERTIB 48344 33003 MPI 4351 ENZYME, DRUGGABLE GENOME NSC-66209 CHEMBL175266 48346 33004 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor XL147 PILARALISIB 48352 33005 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR IOXYNIL IOXYNIL 48354 33006 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MYRICETIN MYRICETIN 48355 33007 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Benzotriazole derivative 1 48358 33008 KDM4A 9682 DRUGGABLE GENOME, ENZYME PURPURIN PURPURIN 48361 33009 FOSL1 8061 TRANSCRIPTION FACTOR TPA ALTEPLASE 7761434 48362 33010 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-1134 CHEMBL600694 48363 33011 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 tamsulosin TAMSULOSIN 9187528 48364 33012 KRT19 3880 DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 15793288 48365 33013 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CHEMBL1743025 GANTENERUMAB 48369 33014 FGA 2243 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, FIBRINOGEN abciximab ABCIXIMAB 20938371 48370 33015 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Indol-5-ol derivative 1 48371 33016 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COLUBRINIC ACID COLUBRINIC ACID 18842418 48372 33017 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-4576 CHEMBL527336 48374 33018 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER R-FLURBIPROFEN 15710360 48378 33019 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME DABIGATRAN DABIGATRAN 48379 33020 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL452 CLONAZEPAM 48380 33021 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Ipratropium IPRATROPIUM 48383 33022 MUC2 4583 DRUGGABLE GENOME PD-98059 CHEMBL35482 12391274 48384 33023 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME SELICICLIB SELICICLIB 48385 33024 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME activator 178104015 48386 33025 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-F2 48387 33026 ATAD5 79915 NA NSC-656158 CHEMBL280099 48388 33027 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AG-528 CHEMBL56542 48389 33028 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR PD-0325901 PD-0325901 26267534,26582713 48390 33029 POLI 11201 DNA REPAIR PROTOPORPHYRIN DISODIUM PROTOPORPHYRIN DISODIUM 48391 33030 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHA-793887 PHA-793887 48392 33031 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME 178101401 48393 33032 S100A4 6275 NA DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 48394 33033 TUBB4B 10383 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 48398 33034 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LEVOPROPOXYPHENE NAPSYLATE ANHYDROUS LEVOPROPOXYPHENE NAPSYLATE 48399 33035 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-4325 CHEMBL598263 48400 33036 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Calcipotriol CALCIPOTRIOL 48401 33037 SCD 6319 DRUGGABLE GENOME, ENZYME ROSIGLITAZONE ROSIGLITAZONE 15855323 48402 33038 BCHE 590 DRUGGABLE GENOME, ENZYME Plasma derived human butyrylcholinesterase 48403 33039 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102642 48404 33040 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CYCLOSPORINE CYCLOSPORINE 48405 33041 KDM4A 9682 DRUGGABLE GENOME, ENZYME 4-METHYL-[1,10]PHENANTHROLINE CHEMBL316589 48407 33042 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE axitinib AXITINIB 25686603 48412 33043 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIXANTHOGEN DIXANTHOGEN 48413 33044 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MECLOFENAMATE SODIUM MECLOFENAMATE SODIUM 48415 33045 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE isoproterenol ISOPROTERENOL 11586955 48416 33046 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME OXYPHENBUTAZONE OXYPHENBUTAZONE 48417 33047 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417181 CHEMBL1537417 48418 33048 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME (-)-Phenserine 48422 33049 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE isoniazid ISONIAZID 22151084 48423 33050 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME AVX701 48425 33051 ALB 213 TRANSPORTER, DRUGGABLE GENOME EVANS BLUE 48427 33052 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Atezolizumab ATEZOLIZUMAB 48428 33053 ALOX15 246 ENZYME, DRUGGABLE GENOME ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 48429 33054 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4590 CHEMBL529361 48430 33055 NOTCH2 4853 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE inhibitor PF-03084014 NIROGACESTAT 48431 33056 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651538 48432 33057 NDUFA2 4695 ENZYME inhibitor CHEMBL3545320 ME-344 48433 33058 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 3-phenyl isoquinolin-1(2H) derivative 2 48436 33059 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER 6-DESOXYCODEINE CHEMBL408422 18311899 48437 33060 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SEMAXANIB SEMAXANIB 48438 33061 PTPRZ1 5803 PROTEIN PHOSPHATASE, DRUGGABLE GENOME PMA 10809755 48439 33062 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Galcanezumab GALCANEZUMAB 48441 33063 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TRASTUZUMAB TRASTUZUMAB 48442 33064 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME PMID27998201-Compound-12 48444 33065 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME BETA-INTERFERON 2491749 48445 33066 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ACROLEIN ACROLEIN 48447 33067 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-51 48448 33068 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE AFURESERTIB HYDROCHLORIDE 48449 33069 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE OCHROMYCINONE OCHROMYCINONE 18006313 48450 33070 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE AMITRIPTYLINE AMITRIPTYLINE 12856820 48455 33071 CD74 972 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE antagonist CHEMBL1743040 MILATUZUMAB 48456 33072 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR EPINEPHRINE EPINEPHRINE 48461 33073 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 178100398 48462 33074 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OXYPHENCYCLIMINE OXYPHENCYCLIMINE 48463 33075 NAMPT 10135 DRUGGABLE GENOME inhibitor CHEMBL190412 TEGLARINAD CHLORIDE 48464 33076 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650631 48465 33077 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SOLIFENACIN SOLIFENACIN 48466 33078 POLK 51426 DNA REPAIR, ENZYME SULFOBROMOPHTHALEIN SULFOBROMOPHTHALEIN 48467 33079 HERC2 8924 DNA REPAIR, ENZYME NERATINIB NERATINIB 23220880 48468 33080 XDH 7498 DRUGGABLE GENOME, ENZYME AZITHROMYCIN AZITHROMYCIN 14730107 48469 33081 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 249565740 AMG-900 48470 33082 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR 7,12-DIMETHYL-BENZO[A]ANTHRACENE CHEMBL329673 48472 33083 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 315661346 48473 33084 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX TAZAROTENE TAZAROTENE 48474 33085 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200903 SECOBARBITAL SODIUM 48475 33086 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TYRPHOSTIN AG-835 CHEMBL261557 48478 33087 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME PF-562271 PF-00562271 48480 33088 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124857 CHEMBL546580 48482 33089 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-62 48483 33090 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SULCONAZOLE NITRATE SULCONAZOLE NITRATE 48484 33091 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AZD8329 48485 33092 ALB 213 TRANSPORTER, DRUGGABLE GENOME PYROGALLOL PYROGALLOL 20598557 48486 33093 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME METARAMINOL METARAMINOL 22931300 48487 33094 CSNK2A2 1459 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME, TRANSCRIPTION FACTOR inhibitor 249565820 48489 33095 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135650111 CLOMIPRAMINE 48490 33096 MPHOSPH8 54737 NA SURAMIN SURAMIN 48491 33097 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Pyridine derivative 18 48494 33098 AKR1B1 231 DRUGGABLE GENOME, ENZYME PMID30124346-Compound-60TABLE5 48495 33099 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Pembrolizumab PEMBROLIZUMAB 28514312 48498 33100 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 340590233 48499 33101 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DEOXIEPINEPHRINE DEOXIEPINEPHRINE 48500 33102 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TAMOXIFEN TAMOXIFEN 48501 33103 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1079175 MK-2206 48502 33104 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor MEK162 BINIMETINIB 48504 33105 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME pazopanib PAZOPANIB 25504632 48505 33106 TDO2 6999 ENZYME, DRUGGABLE GENOME Indazole derivative 3 48506 33107 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RALOXIFENE RALOXIFENE 24456369 48507 33108 TAC1 6863 DRUGGABLE GENOME CHLORHEXIDINE CHLORHEXIDINE 14631229 48508 33109 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME CRYPTOLEPINE HYDROCHLORIDE CRYPTOLEPINE HYDROCHLORIDE 23507189 48511 33110 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR fluorouracil FLUOROURACIL 21057378,23314736,28796378 48512 33111 PROS1 5627 DRUGGABLE GENOME avatrombopag AVATROMBOPAG 48514 33112 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 381118815 48515 33113 NOS2 4843 DRUGGABLE GENOME, ENZYME inhibitor 178101795 1400W 48516 33114 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 6-METHYLFLAVONE 6-METHYLFLAVONE 48517 33115 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651021 48518 33116 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 328083483 PF-00562271 48519 33117 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE SUBEROYLANILIDE HYDROXAMIC ACID 16144943 48520 33118 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1161 MOMETASONE FUROATE 48521 33119 APOE 348 DRUGGABLE GENOME RETINOIC ACID 3468509 48522 33120 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor XL765 48523 33121 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME STREPTOZOTOCIN STREPTOZOCIN 8171758 48524 33122 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-A10 48526 33123 SCTR 6344 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME SECRETIN SECRETIN 48527 33124 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE TCMDC-125543 CHEMBL546170 48528 33125 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor 178103252 SELEGILINE 48530 33126 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RESMETHRIN RESMETHRIN 48532 33127 KLC3 147700 NA oxaliplatin OXALIPLATIN 19434073,22188361,29662106,22026922,21449681 48533 33128 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (+)-3-DEOXYTHYSANONE CHEMBL593570 19783445 48534 33129 AKR1C4 1109 DRUGGABLE GENOME, ENZYME exemestane EXEMESTANE 27111237 48535 33130 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME FLUVOXAMINE FLUVOXAMINE 48537 33131 XDH 7498 DRUGGABLE GENOME, ENZYME Fused heterocyclic compound 5 48538 33132 DMD 1756 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME DYSTROPHIN 48539 33133 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 3',4' DICHLOROBENZAMIL 3',4' DICHLOROBENZAMIL 48540 33134 ALOX15 246 ENZYME, DRUGGABLE GENOME ZAPRINAST ZAPRINAST 48542 33135 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201454 ALSEROXYLON 48543 33136 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PMID26924192-Compound-104 48545 33137 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-18 48546 33138 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102667 48549 33139 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor BELINOSTAT BELINOSTAT 48551 33140 PSMC3 5702 NA inhibitor CHEMBL325041 BORTEZOMIB 48553 33141 HSPA8 3312 TUMOR SUPPRESSOR ADENOSINE DIPHOSPHATE ADENOSINE DIPHOSPHATE 48554 33142 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME DNDI1417548 CHEMBL2094789 48555 33143 KDM4A 9682 DRUGGABLE GENOME, ENZYME 2-ANILINOPYRIDINE CHEMBL555260 48556 33144 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME ospemifene OSPEMIFENE 48558 33145 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL3707315 D-3263 48559 33146 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE egfr inhibitors 18006781,23959273,16788380,22158333 48560 33147 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY POLYETHYLENE GLYCOL 6667021 48562 33148 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-23 48563 33149 MAP3K5 4217 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545429 SELONSERTIB 48564 33150 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic-carboxamide derivative 1 48565 33151 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME HUMAN CHORIONIC GONADOTROPIN 17049229 48566 33152 PTGS1 5742 ENZYME, DRUGGABLE GENOME KETOROLAC KETOROLAC 48567 33153 FAAH 2166 ENZYME, DRUGGABLE GENOME PHENMEDIPHAM PHENMEDIPHAM 19850474 48568 33154 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650381 IMETIT 48570 33155 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Lintopride LINTOPRIDE 48572 33156 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE 3-NITROPROPIONIC ACID CHEMBL451226 48573 33157 TET2 54790 CLINICALLY ACTIONABLE, ENZYME hydrochlorothiazide HYDROCHLOROTHIAZIDE 48575 33158 RACGAP1 29127 NA NSC-60340 CHEMBL1534034 48576 33159 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE ILORASERTIB ILORASERTIB 48577 33160 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENTICLOR FENTICLOR 48578 33161 GGCX 2677 DRUGGABLE GENOME, ENZYME inhibitor 178103541 ANISINDIONE 48579 33162 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DASATINIB DASATINIB 20956938 48581 33163 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor XL647 TESEVATINIB 48582 33164 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL IBUTILIDE IBUTILIDE 48583 33165 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL3707402 PF-06372865 48584 33166 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE CEFUROXIME CEFUROXIME 22166395 48585 33167 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 risperidone RISPERIDONE 48586 33168 GAPVD1 26130 NA interferon beta-1a 27001119 48588 33169 SLC29A2 3177 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE TECADENOSON TECADENOSON 23388705 48591 33170 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 354702227 MOFEGILINE 48594 33171 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-62406 CHEMBL1332182 48596 33172 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER HALOPERIDOL HALOPERIDOL 16476148 48598 33173 GC 2638 DRUGGABLE GENOME Pirsidomine PIRSIDOMINE 48599 33174 ACP1 52 ENZYME, DRUGGABLE GENOME, PROTEIN PHOSPHATASE TCMDC-125603 CHEMBL528734 48600 33175 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE SULINDAC SULINDAC 30683736 48601 33176 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor PKI-587 GEDATOLISIB 48602 33177 SLC28A1 9154 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE URIDINE URIDINE 10455109 48603 33178 BCHE 590 DRUGGABLE GENOME, ENZYME ECHOTHIOPHATE IODIDE 48605 33179 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR CID 2056784 CHEMBL261123 48607 33180 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SA-237 SATRALIZUMAB 23575266 48608 33181 GMNN 51053 DRUGGABLE GENOME TCMDC-123811 CHEMBL587433 48610 33182 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE TIROFIBAN TIROFIBAN 48611 33183 FOXO1 2308 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR epirubicin EPIRUBICIN 48613 33184 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR OXYCARBOXIN OXYCARBOXIN 48615 33185 TUBA4A 7277 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 48616 33186 SLC16A3 9123 DRUGGABLE GENOME, TRANSPORTER STZ STREPTOZOCIN 12611763 48617 33187 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200478 DYCLONINE HYDROCHLORIDE 48619 33188 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME blocker 178103079 48621 33189 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW305074X GW305074X 48623 33190 HTT 3064 DRUGGABLE GENOME TDR78109 CHEMBL1304363 48624 33191 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME ABT-348 ILORASERTIB 48625 33192 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BEZ235 DACTOLISIB 26272063,23629727,25673820,23475782,26206338,24939055,19029981,26232337,22662154 48626 33193 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME phorbol 12-myristate 13-acetate 48627 33194 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1200705 HYDROXYAMPHETAMINE HYDROBROMIDE 48629 33195 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-D1 48630 33196 ATXN2 6311 NA DNDI1417932 CHEMBL1334191 48631 33197 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL52885 ENMD-981693 48632 33198 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE SD-093 15289325 48634 33199 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PF-05212384 GEDATOLISIB 17314276,14737113,21325073 48636 33200 SMN2 6607 DRUGGABLE GENOME CID 5310655 CHEMBL408563 48637 33201 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR PROGESTERONE PROGESTERONE 16954335 48638 33202 ALOX15 246 ENZYME, DRUGGABLE GENOME NONIVAMIDE NONIVAMIDE 48639 33203 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 310264762 48640 33204 MAOB 4129 DRUGGABLE GENOME, ENZYME 5-(2-PHENYLETHYL)ISATIN CHEMBL1642672 21134756 48641 33205 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID29757691-Compound-8a 48642 33206 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE lovastatin LOVASTATIN 18695978,15284534 48643 33207 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MERADIMATE MERADIMATE 48645 33208 CTSV 1515 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 252166762 CITIBRASINE 48649 33209 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE WORTMANNIN WORTMANNIN 15683719 48650 33210 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL3545351 AV-101 48653 33211 HTT 3064 DRUGGABLE GENOME HEXACHLOROPHENE HEXACHLOROPHENE 48654 33212 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RIMCAZOLE RIMCAZOLE 48655 33213 PTGS1 5742 ENZYME, DRUGGABLE GENOME KETOROLAC KETOROLAC 48656 33214 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GS-39783 GS-39783 48657 33215 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ERLOTINIB ERLOTINIB 21258250,15696205,19794967,23313110,21969500,21862683 48658 33216 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SNS-314 SNS-314 48659 33217 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ALDESLEUKIN ALDESLEUKIN 48660 33218 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR PD0325901 48661 33219 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GLABROL GLABROL 48662 33220 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR FLUOXASTROBIN FLUOXASTROBIN 48664 33221 ATXN2 6311 NA DNDI1416975 CHEMBL1415851 48665 33222 REV3L 5980 DRUGGABLE GENOME, DNA DIRECTED RNA POLYMERASE cisplatin CISPLATIN 48667 33223 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE TDR77593 CHEMBL1510164 48670 33224 POLRMT 5442 NA 2',2'-DIFLUORODEOXYCYTIDINE 5'-TRIPHOSPHATE 2',2'-DIFLUORODEOXYCYTIDINE 5'-TRIPHOSPHATE 25667954 48671 33225 DPYSL2 1808 NA LACOSAMIDE ERLOSAMIDE 48672 33226 ABHD6 57406 PHOSPHOLIPASE, ENZYME Pyrazole derivative 82 48675 33227 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PMID30124346-Compound-LDT66 48676 33228 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME LINIFANIB LINIFANIB 48677 33229 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR lithium LITHIUM 21781277,23021822,21047205,24885933 48683 33230 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TOPOTECAN HYDROCHLORIDE TOPOTECAN HYDROCHLORIDE 48684 33231 AKR1B1 231 DRUGGABLE GENOME, ENZYME inhibitor 178103987 SORBINIL 48687 33232 BAZ2B 29994 NA GNF-PF-107 CHEMBL578675 48688 33233 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PREDNISOLONE ACETATE PREDNISOLONE ACETATE 48690 33234 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE LESTAURTINIB LESTAURTINIB 24162815 48691 33235 TUBA3C 7278 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 48693 33236 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ROSIGLITAZONE ROSIGLITAZONE 11699047 48695 33237 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL3545264 LY-2874455 48696 33238 HSPB2 3316 KINASE DIFFERENTIATION INDUCER 9332492 48697 33239 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125813 CHEMBL580076 48698 33240 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1522 ESZOPICLONE 48699 33241 CD47 961 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE CC-90002 48700 33242 CSF1 1435 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ACTINOMYCIN D 3265472,9419789 48701 33243 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX PYROCATECHOL VIOLET PYROCATECHOL VIOLET 16759101 48702 33244 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HYDRALAZINE HYDRALAZINE 22931300 48703 33245 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650587 METHOXAMINE 48704 33246 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME SURAMIN SURAMIN 48706 33247 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID25991433-Compound-A1 48707 33248 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 328083469 48708 33249 IL1B 3553 KINASE, DRUGGABLE GENOME inhibitor CHEMBL1201830 RILONACEPT 48710 33250 L1CAM 3897 CELL SURFACE, DRUGGABLE GENOME, KINASE CD171 specific CAR T cells expressing EGFRt 48711 33251 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 2,7-BIS[3-(ETHYLAMINO)PROPIONAMIDO]ANTHRAQUINONE CHEMBL481161 18571928 48712 33252 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME PRAVASTATIN PRAVASTATIN 16678544 48714 33253 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME GW-796406 48715 33254 ALOX15B 247 DRUGGABLE GENOME, ENZYME NSC-172033 CHEMBL238624 48719 33255 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR ORAL CONTRACEPTIVE 8392873 48720 33256 DNER 92737 NA Pyrimido-indole derivative 3 48721 33257 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE KU-0058948 CHEMBL380648 19354255 48722 33258 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME CYCLOSPORINE CYCLOSPORINE 21488686 48723 33259 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE PROGESTIN PROGESTERONE 12529413 48724 33260 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME VORINOSTAT VORINOSTAT 19344175,19966789,26211462,23622981,22260166,20491440,21548582,19084294 48725 33261 PTGS2 5743 DRUGGABLE GENOME, ENZYME Lumiracoxib LUMIRACOXIB 48728 33262 ANXA5 308 KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER BETA-LAPACHONE LAPACHONE 11474117 48729 33263 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 2'-HYDROXY-2,3,4',6',TETRAMETHOXYCHALCONE CHEMBL1254091 20813535 48730 33264 SRD5A1 6715 DRUGGABLE GENOME LY-266111 CHEMBL29166 48731 33265 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565830 GSK-579289A 48733 33266 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TELENZEPINE TELENZEPINE 48736 33267 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME Prasugrel PRASUGREL 48737 33268 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BML-210 CHEMBL324053 16921367 48738 33269 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 48739 33270 TAT 6898 ENZYME GENISTEIN GENISTEIN 9128187 48741 33271 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLOTRIMAZOLE CLOTRIMAZOLE 22931300 48743 33272 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME NEU-2000 48744 33273 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE ALSTERPAULLONE ALSTERPAULLONE 48745 33274 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 375973268 48746 33275 IL1B 3553 KINASE, DRUGGABLE GENOME NICARDIPINE NICARDIPINE 1888883 48747 33276 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE activator 135650716 48748 33277 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 135649932 PLERIXAFOR 48749 33278 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ARACHIDONIC ACID ARACHIDONIC ACID 48750 33279 RGS12 6002 DRUGGABLE GENOME SANGUINARINE SULFATE SANGUINARINE SULFATE 48751 33280 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME allosteric modulator 385612232 MITAPIVAT 48752 33281 ATXN2 6311 NA TCMDC-125185 CHEMBL580819 48753 33282 GSTT1 2952 DRUGGABLE GENOME etoposide ETOPOSIDE 48755 33283 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER 1,3-BIS(3-CHLOROPHENYL)UREA CHEMBL1417470 48756 33284 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 348353643 48757 33285 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PS433540 48758 33286 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor LY2835219 ABEMACICLIB 48759 33287 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL blocker 135652748 48762 33288 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Ipilimumab IPILIMUMAB 48763 33289 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SCOPOLETIN SCOPOLETIN 48764 33290 POLI 11201 DNA REPAIR SLAZINIC ACID SLAZINIC ACID 48765 33291 ALPI 248 DRUGGABLE GENOME, ENZYME DNDI1417368 CHEMBL2094652 48766 33292 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DEMETHOXYCURCUMIN DEMETHOXYCURCUMIN 48767 33293 ETS2 2114 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR carboplatin CARBOPLATIN 31616045 48768 33294 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TEGAFUR TEGAFUR 8521418 48769 33295 FAAH 2166 ENZYME, DRUGGABLE GENOME PF-04457845 PF-04457845 48770 33296 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-52 48771 33297 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME HISPIDIN HISPIDIN 48773 33298 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GNF-PF-5510 CHEMBL578741 48774 33299 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PLERIXAFOR PLERIXAFOR 17715128,19451305,17958344,26191361 48775 33300 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TETRAIDOFLUORESCEIN TETRAIDOFLUORESCEIN 48777 33301 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-54 48780 33302 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Tisagenlecleucel TISAGENLECLEUCEL 48782 33303 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ZUCAPSAICIN ZUCAPSAICIN 48783 33304 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TGF-BETA 2 15223827 48784 33305 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 328083488 CHEMBL401930 48785 33306 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist CHEMBL2181927 FINERENONE 48786 33307 ATXN2 6311 NA TCMDC-125567 CHEMBL530049 48788 33308 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-5029 CHEMBL600360 48789 33309 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-G4 48790 33310 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL atenolol ATENOLOL 20031608 48792 33311 SIRT6 51548 TRANSCRIPTION FACTOR, ENZYME allosteric modulator 381118833 48794 33312 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR PROTEASOME INHIBITOR 10871842,15994939 48796 33313 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME MGCD-0103 MOCETINOSTAT 48798 33314 NDUFA8 4702 ENZYME inhibitor CHEMBL3545320 ME-344 48799 33315 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BENZO[B]FLUORANTHENE BENZO[B]FLUORANTHENE 48800 33316 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3545274 MK-6913 48801 33317 CP 1356 DRUGGABLE GENOME, ENZYME ISOFLAVONE ISOFLAVONE 15754123 48802 33318 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme9EHT1610 48803 33319 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PINOSYLVIN METHYL ETHER PINOSYLVIN METHYL ETHER 48806 33320 CCNA2 890 DRUGGABLE GENOME, KINASE 3-DEOXYADENOSINE 11566717 48808 33321 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651361 48811 33322 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Paclitaxel PACLITAXEL 28514312 48812 33323 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL2220486 LUCITANIB 48816 33324 EPHX2 2053 DRUGGABLE GENOME, ENZYME inhibitor 387065576 48817 33325 BRCA2 675 CLINICALLY ACTIONABLE INIPARIB INIPARIB 21508395 48818 33326 CTSA 5476 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 223366214 48819 33327 PTK6 5753 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL24828 VANDETANIB 48822 33328 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Fused benzoheterocycle amide derivative 2 48823 33329 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE CEDIRANIB CEDIRANIB 48824 33330 ATAD5 79915 NA SJ000149318 CHEMBL600662 48825 33331 GPER1 2852 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR agonist 135651381 48829 33332 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 315661218 GLESATINIB 48830 33333 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CARBAMAZEPINE CARBAMAZEPINE 22931300 48832 33334 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178103794 MELOXICAM 48834 33335 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyrimidine derivative 7 48835 33336 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME cyclophosphamide CYCLOPHOSPHAMIDE 48836 33337 POLI 11201 DNA REPAIR MITOXANTRONE MITOXANTRONE 48837 33338 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE OLIVOMYCIN I OLIVOMYCIN I 19535252 48838 33339 BAZ2B 29994 NA 2-PYRIDYLCARBOXALDEHYDE ISONICOTINOYLHYDRAZONE CHEMBL401362 48839 33340 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Pyrrolidine derivative 12 48840 33341 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW621431X GW621431X 48841 33342 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 4'-DEMETHYLEPIPODOPHYLLOTOXIN 4'-DEMETHYLEPIPODOPHYLLOTOXIN 48842 33343 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135650654 48843 33344 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2105754 TRELAGLIPTIN SUCCINATE 48845 33345 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 348353615 48846 33346 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 (R)-FELODIPINE (R)-FELODIPINE 48847 33347 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL686 MEFENAMIC ACID 48850 33348 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Ponatinib PONATINIB 24552773,21482694,22301675,25239608 48851 33349 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Salicylic acid derivative 4 48852 33350 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL2108018 ADECATUMUMAB 48853 33351 RAPGEF3 10411 ENZYME GNF-PF-1947 CHEMBL585591 48856 33352 CPB2 1361 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166856 48858 33353 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 223366122 MOMELOTINIB 48859 33354 ILKAP 80895 KINASE hydrochlorothiazide HYDROCHLOROTHIAZIDE 48860 33355 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR U-69593 U-69593 24613457 48861 33356 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE ZONISAMIDE ZONISAMIDE 48862 33357 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE GSK2141795 UPROSERTIB 24735930,24978597,23795919,26429956 48864 33358 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TELITHROMYCIN TELITHROMYCIN 48865 33359 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR BITHIONOL BITHIONOL 48866 33360 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL3545169 AZD1305 48870 33361 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME activator 223366036 48871 33362 EEF2 1938 DRUGGABLE GENOME, KINASE VB4-845 OPORTUZUMAB MONATOX 48872 33363 TUBB 203068 DRUGGABLE GENOME CKD-516 48873 33364 ABAT 18 DRUGGABLE GENOME, ENZYME VIGABATRIN VIGABATRIN 48874 33365 GRB2 2885 NA ANTINEOPLASTIC 10403397 48875 33366 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135649939 AMITRIPTYLINE 48876 33367 CFL1 1072 KINASE CLOTRIMAZOLE CLOTRIMAZOLE 16680159 48878 33368 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 178102615 48879 33369 MYB 4602 CLINICALLY ACTIONABLE G4460 48880 33370 ACE2 59272 ENZYME, TRANSPORTER, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, CELL SURFACE, PROTEASE LISINOPRIL LISINOPRIL 48881 33371 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PI3K/BET INHIBITOR LY294002 15324695 48885 33372 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Danaparoid DANAPAROID 48886 33373 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TCMDC-124570 CHEMBL546475 48887 33374 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CISPLATIN CISPLATIN 9935158 48888 33375 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE NEU-2000 48889 33376 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-8 48890 33377 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-E3 48891 33378 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE lidocaine / prilocaine 48892 33379 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor PF03084014 48893 33380 POLI 11201 DNA REPAIR HYDROXYSTILBAMIDINE HYDROXYSTILBAMIDINE 48895 33381 CXCL8 3576 DRUGGABLE GENOME ANTIDEPRESSANTS 11418279 48896 33382 GUCY1A1 2982 ENZYME, DRUGGABLE GENOME activator CHEMBL6622 ISOSORBIDE DINITRATE 48898 33383 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE daunorubicin DAUNORUBICIN 48899 33384 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 67S 48901 33385 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME inhibitor 135651334 48903 33386 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GNF-PF-3996 CHEMBL584458 48904 33387 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR IFN ALPHA-2B 12567763 48905 33388 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor DOVITINIB DOVITINIB 48907 33389 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE HM-5016504 48908 33390 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100322 DERENOFYLLINE 48909 33391 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-32 48910 33392 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE allosteric modulator 329968374 TOLIMIDONE 48911 33393 GABPA 2551 TRANSCRIPTION FACTOR DOX 17081560 48912 33394 ITGB5 3693 CELL SURFACE, DRUGGABLE GENOME CILENGITIDE CILENGITIDE 48913 33395 HTT 3064 DRUGGABLE GENOME DNDI1417614 CHEMBL1567571 48914 33396 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor XL-765 VOXTALISIB 48916 33397 SMN2 6607 DRUGGABLE GENOME DIBENZOYLMETHANE DIBENZOYLMETHANE 48917 33398 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CISAPRIDE CISAPRIDE 48918 33399 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102337 SORAFENIB 48919 33400 ATAD5 79915 NA NSC-234945 CHEMBL260311 48920 33401 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RIFAMPICIN RIFAMPIN 22931300,26291341 48922 33402 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652286 48923 33403 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135649930 TAMIBAROTENE 48925 33404 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE DOVITINIB DOVITINIB 48926 33405 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 223366074 BRIGATINIB 48927 33406 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME (D)-SERINE (D)-SERINE 48928 33407 MARCHF8 220972 ENZYME AFO-18 48929 33408 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 1540545 CHEMBL259784 48930 33409 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 48931 33410 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE LINIFANIB LINIFANIB 48932 33411 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417032 CHEMBL1523974 48934 33412 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME DORAMAPIMOD DORAMAPIMOD 48935 33413 TNNI2 7136 NA activator CHEMBL3039529 TIRASEMTIV 48936 33414 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SP-600125 SP-600125 48937 33415 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 252166687 48939 33416 FABP4 2167 DRUGGABLE GENOME inhibitor 252827446 48940 33417 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE DIMIRACETAM DIMIRACETAM 48942 33418 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ERLOTINIB ERLOTINIB 48947 33419 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DOXACURIUM CHLORIDE 48949 33420 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SALAGEN SALAGEN 48950 33421 IL23A 51561 DRUGGABLE GENOME Tildrakizumab TILDRAKIZUMAB 48951 33422 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650784 OXYBUTYNIN 48952 33423 ATXN2 6311 NA CALCIMYCIN CALCIMYCIN 48953 33424 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME fenofibrate FENOFIBRATE 19207029,23119086 48956 33425 BAZ2B 29994 NA MIANSERIN HYDROCHLORIDE MIANSERIN HYDROCHLORIDE 48957 33426 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ETHINYL ESTRADIOL ETHINYL ESTRADIOL 48959 33427 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 187051793 GIVINOSTAT 48960 33428 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE E7449 2X-121 48961 33429 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 135651472 DIETHYLSTILBESTROL 48962 33430 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Diaryl amine derivative 2 48963 33431 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 310264782 48964 33432 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VACCINE 15328177 48965 33433 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL919 FOSPHENYTOIN SODIUM 48966 33434 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PICTILISIB PICTILISIB 48968 33435 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR NIS793 NIS-793 48969 33436 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME DOXORUBICIN DOXORUBICIN 11589785 48971 33437 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME ANTI-INFLAMMATORY DRUGS 16550006 48974 33438 MAPT 4137 DRUGGABLE GENOME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 48977 33439 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME KW-5092 48978 33440 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME Calcineurin inhibitors 23426640 48980 33441 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651467 48981 33442 PRKAA2 5563 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME METFORMIN HYDROCHLORIDE METFORMIN HYDROCHLORIDE 23490148 48982 33443 PSMD2 5708 NA inhibitor CHEMBL451887 CARFILZOMIB 48983 33444 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-155693 CHEMBL68096 48984 33445 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ELETRIPTAN ELETRIPTAN 48985 33446 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 5-FU FLUOROURACIL 12904931 48986 33447 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PF-3758309 PF-03758309 48987 33448 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL593430 ATAGABALIN 48988 33449 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME KENPAULLONE KENPAULLONE 48990 33450 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545381 PLX-7486 48991 33451 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor PCI-24781 ABEXINOSTAT 48992 33452 GBA 2629 DRUGGABLE GENOME, ENZYME MIGALASTAT MIGALASTAT 48993 33453 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124317 CHEMBL586937 48995 33454 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 385612219 BREPOCITINIB 48996 33455 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CLOSANTEL CLOSANTEL 48997 33456 HMOX1 3162 ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Stannsoporfin STANNSOPORFIN 48998 33457 FAAH 2166 ENZYME, DRUGGABLE GENOME URB597 URB-597 19386497,23287055,21666860 48999 33458 GJA1 2697 ION CHANNEL VITAMIN C 16448880 49000 33459 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL932 DIPYRIDAMOLE 49001 33460 ATAD5 79915 NA HISPIDULIN HISPIDULIN 49002 33461 KHSRP 8570 NA GO-Y030 CHEMBL598509 49006 33462 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DESOXYCORTICOSTERONE PIVALATE DESOXYCORTICOSTERONE PIVALATE 49007 33463 CDK16 5127 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3544942 RONICICLIB 49008 33464 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME ISOQUINOLINE-1,3(2H,4H)-DIONE CHEMBL1210769 49009 33465 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545301 HMPL-523 49011 33466 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CYPROTERONE CYPROTERONE 22931300 49012 33467 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-37 49013 33468 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102316 CHEMBL1908395 49015 33469 ATAD5 79915 NA KN-62 CHEMBL28324 49016 33470 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ISOPROTERENOL HYDROCHLORIDE ISOPROTERENOL HYDROCHLORIDE 49017 33471 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE FENTICLOR FENTICLOR 49019 33472 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CYT007-TNFQB 49020 33473 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME TAMATINIB R-406 49021 33474 HSPA1A 3303 DRUGGABLE GENOME carbamazepine CARBAMAZEPINE 16538175 49022 33475 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 348353626 PF-06650833 49024 33476 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE INDOXACARB INDOXACARB 49025 33477 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650625 MOSAPRIDE 49026 33478 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL235191 TACEDINALINE 49027 33479 MAP2K5 5607 KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor DABRAFENIB MESYLATE 49028 33480 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor DANUSERTIB DANUSERTIB 49029 33481 ADD1 118 KINASE torasemide TORSEMIDE 20877298 49030 33482 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-4459 CHEMBL585502 49032 33483 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE HYCANTHONE HYCANTHONE 49035 33484 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE ABIRATERONE ABIRATERONE 49038 33485 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR UR-63325 UR-63325 49040 33486 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ANTIBIOTIC ANTIBIOTIC 8096833 49041 33487 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME leucovorin LEUCOVORIN 18267032,20385995,20078613 49042 33488 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BROMOXYNIL BROMOXYNIL 49044 33489 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TYRPHOSTIN A9 TYRPHOSTIN A9 49048 33490 TRBC1 28639 KINASE, TRANSCRIPTION FACTOR, EXTERNAL SIDE OF PLASMA MEMBRANE TRBC1 49050 33491 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1689 TOLAZOLINE HYDROCHLORIDE 49052 33492 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME antidepressants 9918137,20531370,1346258,15252821,14716707,18359183,14520122,8867869,15116051,8181196,8941025,17721180,17667959,15115913,12360109,14646691,15205367,11682257,16024198,16361630,17008819,27023676,10460069,9585799,16871470 49053 33493 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2,3,4-TRIHYDROXYBENZALDEHYDE CHEMBL254077 49056 33494 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID27744724-Compound-10 49057 33495 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL TEMAZEPAM TEMAZEPAM 49058 33496 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 49059 33497 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3545165 AFACIFENACIN 49061 33498 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE Refametinib REFAMETINIB 49063 33499 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor BELINOSTAT BELINOSTAT 49065 33500 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE SAR 1118 49066 33501 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME BENZYL CAFFEATE BENZYL CAFFEATE 25314129 49067 33502 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PWT33597 49069 33503 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774822-Compound-Figure11Example5 49070 33504 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE capecitabine CAPECITABINE 27738344,18245544,17700593,24167597,29845393,27864592,18299612,20819423,27995989,19384296,29134491,23314736,20638924,25331073,20385995,27557140,26967565,23407049,26014925,23736036 49072 33505 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE RG-1530 RG-1530 49073 33506 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR cisplatin CISPLATIN 21430602 49076 33507 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL inverse agonist CHEMBL2107801 RESEQUINIL 49077 33508 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102667 49079 33509 KMO 8564 DRUGGABLE GENOME, ENZYME Pyrimidine benzenesulfonamide derivative 1 49080 33510 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Pertuzumab PERTUZUMAB 49081 33511 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER APOMORPHINE APOMORPHINE 49083 33512 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME IRX4204 49084 33513 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE ACIVICIN ACIVICIN 1596574,1997162 49085 33514 KDM4A 9682 DRUGGABLE GENOME, ENZYME FAMOTIDINE FAMOTIDINE 49086 33515 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Raloxifene RALOXIFENE 49087 33516 PDE4B 5142 DRUGGABLE GENOME, ENZYME ENPROFYLLINE ENPROFYLLINE 49089 33517 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 381118818 49091 33518 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE inhibitor 385612233 49092 33519 ALOX15 246 ENZYME, DRUGGABLE GENOME TCMDC-124536 CHEMBL580851 49093 33520 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor JNJ38877605 49094 33521 DHFR 1719 DRUGGABLE GENOME, ENZYME AMETHOPTERIN METHOTREXATE 9129 49097 33522 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR RUXOLITINIB RUXOLITINIB 27518686 49098 33523 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SORAFENIB SORAFENIB 49099 33524 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PRAZOSIN PRAZOSIN 49100 33525 POLK 51426 DNA REPAIR, ENZYME TYRPHOSTIN 47 TYRPHOSTIN 47 49102 33526 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE PROTOPORPHYRIN DISODIUM PROTOPORPHYRIN DISODIUM 49103 33527 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ILORASERTIB ILORASERTIB 49104 33528 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GBR-12909 VANOXERINE 49105 33529 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE RIBOCICLIB RIBOCICLIB 25002028 49107 33530 TSPO 706 DRUGGABLE GENOME PMID27599163-Compound-75 49108 33531 PDE4B 5142 DRUGGABLE GENOME, ENZYME PAPAVERINE PAPAVERINE 49109 33532 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE ZYC300 49111 33533 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 propafenone PROPAFENONE 9187528 49112 33534 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZD-3514 AZD3514 49113 33535 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE PAN-AKT KINASE INHIBITOR GSK690693 24335962 49114 33536 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE ILORASERTIB ILORASERTIB 49118 33537 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178103999 VILAZODONE 49120 33538 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME RESERPINE RESERPINE 10700389 49121 33539 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PF3644022 26140595 49123 33540 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649710 49125 33541 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE CHLOROTHIAZIDE CHLOROTHIAZIDE 49126 33542 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Paclitaxel PACLITAXEL 28514312 49128 33543 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL108 CARBAMAZEPINE 49129 33544 TMEM97 27346 NA Fused aryl carbocycle derivative 8 49130 33545 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor PX-866 SONOLISIB 49131 33546 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651413 SEROTONIN 49132 33547 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR SENNOSIDE B SENNOSIDE B 49134 33548 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE PEGINTERFERON ALFA-2A 49135 33549 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ANTIAROL ANTIAROL 49136 33550 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME BOS172722 49137 33551 DHFR 1719 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL34259 METHOTREXATE 49138 33552 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME RETIGABINE EZOGABINE 49142 33553 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 405560505 49144 33554 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE MOTESANIB MOTESANIB 49145 33555 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL661 ALPRAZOLAM 49146 33556 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ROTENONE ROTENONE 49147 33557 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME AZQ DIAZIQUONE 8943236 49148 33558 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME HUMAN CHORIONIC GONADOTROPIN 9530505 49149 33559 ACACA 31 ENZYME, DRUGGABLE GENOME allosteric modulator 404859092 FIRSOCOSTAT 49150 33560 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE fulvestrant FULVESTRANT 49152 33561 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME cabozantinib CABOZANTINIB 27525386 49154 33562 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENTOLAMINE MESYLATE PHENTOLAMINE MESYLATE 49155 33563 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DEXFENFLURAMINE DEXFENFLURAMINE 49156 33564 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker 223366054 ABT-639 49157 33565 GMNN 51053 DRUGGABLE GENOME NSC-724440 CHEMBL515617 49158 33566 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Xatral ALFUZOSIN HYDROCHLORIDE 49161 33567 MPHOSPH8 54737 NA METHYLDOPA METHYLDOPA 49163 33568 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101454 SILDENAFIL 49164 33569 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME avatrombopag AVATROMBOPAG 49165 33570 NDUFB11 54539 ENZYME inhibitor CHEMBL3545320 ME-344 49166 33571 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR sparsentan SPARSENTAN 49167 33572 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL979 MEPROBAMATE 49168 33573 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE BREFELDIN A BREFELDIN A 49169 33574 TNFRSF18 8784 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME TRX-518 TRX-518 49170 33575 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-56452 CHEMBL1358137 49171 33576 RPS19 6223 NA VITAMIN A 12175513 49172 33577 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 187051799 DACINOSTAT 49174 33578 IGFBP5 3488 DRUGGABLE GENOME TGFBETA1 16214131 49175 33579 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Bazedoxifene BAZEDOXIFENE 49176 33580 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL487 DROLOXIFENE 49177 33581 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR LGD1069 BEXAROTENE 17027148 49178 33582 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GW405833 CHEMBL73711 49179 33583 NR1D2 9975 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 310264684 49180 33584 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651563 49181 33585 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE SP-600125 SP-600125 49182 33586 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-4 49184 33587 ST14 6768 ENZYME, DRUGGABLE GENOME, PROTEASE SURAMIN SURAMIN 15590895 49185 33588 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178103660 HYDROCODONE 49186 33589 TUBB3 10381 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 49187 33590 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME fenofibrate FENOFIBRATE 49188 33591 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor BELINOSTAT BELINOSTAT 49189 33592 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (S)-FLUOXETINE CHEMBL1169388 49190 33593 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PYRONIN Y PYRONIN Y 49191 33594 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE PMID29130358-Compound-Figure18(14a) 49192 33595 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Cetuximab CETUXIMAB 49193 33596 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE DEFEROXAMINE DEFEROXAMINE 24074025 49194 33597 ATP5F1E 514 TRANSPORTER methotrexate METHOTREXATE 26307125 49195 33598 MAOA 4128 DRUGGABLE GENOME, ENZYME N-(2-phenylcyclopropyl) amino acid derivative 3 49196 33599 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE midazolam MIDAZOLAM 24214410,25979262,28986606,23327575 49197 33600 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE AG-555 CHEMBL53898 49201 33601 CP 1356 DRUGGABLE GENOME, ENZYME OESTRADIOL ESTRADIOL 6446099 49202 33602 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME VX-702 VX-702 49203 33603 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator 178103425 FONDAPARINUX 49204 33604 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER COLCHICINE COLCHICINE 49205 33605 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR CLOFIBRATE CLOFIBRATE 49206 33606 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DAPH DAPH 49207 33607 ARHGEF28 64283 NA methylphenidate METHYLPHENIDATE 29382897 49211 33608 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME PYRONIN Y PYRONIN Y 49212 33609 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-40 49213 33610 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE DIPYRIDAMOLE DIPYRIDAMOLE 49215 33611 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DICOFOL DICOFOL 49216 33612 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 178100443 BARDOXOLONE METHYL 49221 33613 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545426 CC-115 49225 33614 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2010077680 109 49227 33615 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME BMS-986165 49228 33616 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME MV-CEA 49229 33617 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE doxorubicin DOXORUBICIN 22016816 49231 33618 GLA 2717 ENZYME, DRUGGABLE GENOME IODOACETAMIDE IODOACETAMIDE 49232 33619 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL17350 TRAXOPRODIL 49235 33620 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HEXADECYLTRIMETHYLAMMONIUM CHLORIDE HEXADECYLTRIMETHYLAMMONIUM CHLORIDE 49236 33621 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL MIDAZOLAM MIDAZOLAM 49238 33622 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor AZD4547 49239 33623 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PHENOXYBENZAMINE PHENOXYBENZAMINE 49240 33624 PSMD4 5710 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 49241 33625 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000114740 CHEMBL592068 49242 33626 TAT 6898 ENZYME METHOTREXATE METHOTREXATE 1967611 49243 33627 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Afatinib AFATINIB 27694386 49245 33628 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME SULINDAC SULINDAC 16707021,16950207 49246 33629 SLC38A1 81539 TRANSPORTER 178101264 49247 33630 ERAP1 51752 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 348353641 49248 33631 MPHOSPH8 54737 NA DISULFIRAM DISULFIRAM 49249 33632 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME BARASERTIB BARASERTIB 49250 33633 FZD6 8323 CELL SURFACE, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651916 49252 33634 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE IMATINIB IMATINIB 49254 33635 BCHE 590 DRUGGABLE GENOME, ENZYME TRIAMCINOLONE TRIAMCINOLONE 7937594 49255 33636 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SOTRASTAURIN SOTRASTAURIN 49256 33637 MAOA 4128 DRUGGABLE GENOME, ENZYME AphanamgrandiolA 49258 33638 PLCG1 5335 ENZYME, KINASE, PHOSPHOLIPASE, DRUGGABLE GENOME PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER 49259 33639 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME activator 178101926 49260 33640 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE MLN0128 SAPANISERTIB 26272063,27974663 49261 33641 IL23A 51561 DRUGGABLE GENOME BI 655066 49263 33642 TUBB3 10381 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 49264 33643 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 381118813 RUPATADINE 49265 33644 IL1B 3553 KINASE, DRUGGABLE GENOME CANAKINUMAB CANAKINUMAB 49266 33645 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER VERAPAMIL VERAPAMIL 9862768,1671173 49269 33646 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR CUDC-101 CUDC-101 49270 33647 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SULFADOXINE SULFADOXINE 22931300 49272 33648 GMNN 51053 DRUGGABLE GENOME GNF-PF-3407 CHEMBL602990 49274 33649 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2-TERT-BUTYLPHENOL CHEMBL108851 49278 33650 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651018 CHEMBL112816 49280 33651 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE 178101745 49281 33652 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE HER-2/HER-1 vaccine 49283 33653 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL526 PROPOFOL 49284 33654 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SELUMETINIB SELUMETINIB 31151904 49285 33655 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CHLORPROPAMIDE CHLORPROPAMIDE 22931300 49286 33656 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BYL719 ALPELISIB 49287 33657 KDM4A 9682 DRUGGABLE GENOME, ENZYME GALLAMINE TRIETHIODIDE GALLAMINE TRIETHIODIDE 49288 33658 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-1232 CHEMBL601822 49291 33659 ATP6V1B2 526 ENZYME, TRANSPORTER inhibitor 252827539 ENOXACIN 49292 33660 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME DOPAMINE DOPAMINE 49294 33661 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Peptide analog 44 49297 33662 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor 178102320 ENZASTAURIN 49298 33663 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR DOX 12883037 49301 33664 RAPGEF3 10411 ENZYME PHYSODIC ACID PHYSODIC ACID 49303 33665 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE HPP-607 49305 33666 PSMA4 5685 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL3545432 IXAZOMIB CITRATE 49307 33667 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME GSK-269962A GSK-269962A 49308 33668 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BOPINDOLOL BOPINDOLOL 49310 33669 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 49312 33670 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME COLCHICINE COLCHICINE 6651778 49313 33671 CYB5R4 51167 DRUGGABLE GENOME isosorbide mononitrate 49314 33672 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE Belerofon 49315 33673 ATAD5 79915 NA 1,2-DIMETHOXY-ANTHRAQUINONE CHEMBL52884 49316 33674 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-MERCAPTOBENZOTHIAZOLE 2-MERCAPTOBENZOTHIAZOLE 49318 33675 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ANTISERUM 15554359 49319 33676 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1014 CANDESARTAN CILEXETIL 49323 33677 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 49324 33678 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE pembrolizumab PEMBROLIZUMAB 49325 33679 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL2364619 METHYLSAMIDORPHAN 49326 33680 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DOVITINIB DOVITINIB 27932416,21119661 49328 33681 PDE10A 10846 ENZYME, DRUGGABLE GENOME AMG 579 49329 33682 KCNH6 81033 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL2107762 NERISPIRDINE 49331 33683 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL3707317 LOREDIPLON 49333 33684 PSMB4 5692 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL371405 MARIZOMIB 49335 33685 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR MRT-92 25636740 49336 33686 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker 223366053 49338 33687 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR CS-038 49339 33688 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3545006 PWT-33587 49340 33689 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME LINIFANIB LINIFANIB 49341 33690 FKBP4 2288 DRUGGABLE GENOME RAPAMYCIN SIROLIMUS 1700475 49342 33691 ATAD5 79915 NA TDR77225 CHEMBL1353528 49344 33692 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL antagonist CHEMBL3707318 GRC-17536 49346 33693 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL856 PRIMIDONE 49347 33694 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RETINOL RETINOL 49348 33695 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SALMETEROL SALMETEROL 49349 33696 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE DEXAMETHASONE DEXAMETHASONE 8145726 49350 33697 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-124506 CHEMBL579640 49352 33698 CHRNA5 1138 DRUGGABLE GENOME, ION CHANNEL ethanol ALCOHOL 49353 33699 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1201026 ALBUTEROL SULFATE 49354 33700 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL2108658 TREMELIMUMAB 49356 33701 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME HESPERETIN HESPERETIN 22429094 49357 33702 P2RX4 5025 ION CHANNEL, DRUGGABLE GENOME agonist 178100916 49361 33703 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME DNDI1417467 CHEMBL1997335 49362 33704 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PRACTOLOL PRACTOLOL 49363 33705 MLH1 4292 CLINICALLY ACTIONABLE, DRUGGABLE GENOME N/A 22810696 49364 33706 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FLUCONAZOLE FLUCONAZOLE 22931300 49365 33707 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME INNO-206 ALDOXORUBICIN 49368 33708 PDE4A 5141 DRUGGABLE GENOME, ENZYME Piclamilast PICLAMILAST 49369 33709 PSMA8 143471 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL451887 CARFILZOMIB 49370 33710 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-3352 CHEMBL600306 49371 33711 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CLOFIBRATE CLOFIBRATE 16680159 49372 33712 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme9EHT5372 49374 33713 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Cisplatin CISPLATIN 27040853,28652249 49378 33714 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-125034 CHEMBL239439 49379 33715 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE antibody 178103471 MUROMONAB-CD3 49380 33716 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DINOPROST TROMETHAMINE 49381 33717 CRBN 51185 ENZYME, DRUG RESISTANCE 340590248 IBERDOMIDE 49383 33718 SLC14A1 6563 TRANSPORTER inhibitor 252827538 49384 33719 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker 384403636 49386 33720 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-43 49387 33721 PRLR 5618 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, KINASE SOMATROPIN RECOMBINANT 49389 33722 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE Peptide analog 70 49390 33723 ADK 132 DRUGGABLE GENOME, ENZYME, KINASE BLEOMYCIN BLEOMYCIN 6317371 49391 33724 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE SKI-758 CHEMBL219557 49394 33725 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE MASITINIB MASITINIB 49395 33726 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR ALPHA-TOCOPHEROL VITAMIN E 12023009 49396 33727 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME VITAMIN E 16006884 49397 33728 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HYDROXYCHLOROQUINE HYDROXYCHLOROQUINE 10848718 49398 33729 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PS-341 BORTEZOMIB 49399 33730 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651309 49401 33731 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE LAUROGUADINE LAUROGUADINE 49402 33732 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor NINTEDANIB NINTEDANIB 49403 33733 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AURAPTENE AURAPTENE 49405 33734 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME MG-132 MG-132 24321833,18801655 49406 33735 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME COBIMETINIB COBIMETINIB 25037139,27480103,25265494,23934108 49407 33736 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE RADIOSUMIN B RADIOSUMIN B 11374973 49408 33737 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-2413 CHEMBL578515 49411 33738 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 249565708 49412 33739 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE QUINAPRIL QUINAPRIL 9370386 49414 33740 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME XEN007 49415 33741 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102263 49416 33742 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORMIDAZOLE CHLORMIDAZOLE 49417 33743 LSS 4047 ENZYME, DRUGGABLE GENOME inhibitor 178103324 49418 33744 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE WEHI-539 27974663 49420 33745 GMNN 51053 DRUGGABLE GENOME KAMEBANIN KAMEBANIN 49421 33746 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 49422 33747 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Triprolidine TRIPROLIDINE 49423 33748 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Buclizine BUCLIZINE 49426 33749 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2219421 RECILISIB 49427 33750 MPHOSPH8 54737 NA CISPLATIN CISPLATIN 49428 33751 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR SPIRONOLACTONE SPIRONOLACTONE 49429 33752 PDE4B 5142 DRUGGABLE GENOME, ENZYME AN-2898 49430 33753 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL3545113 PX-102 49431 33754 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CYCLOHEXIMIDE CYCLOHEXIMIDE 49432 33755 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME GENISTEIN GENISTEIN 49433 33756 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TRIIODOTHYRONINE (T3) 49435 33757 SMN2 6607 DRUGGABLE GENOME 2-(STYRYL)-BENZIMIDAZOLE CHEMBL473721 49436 33758 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 49437 33759 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE CHEMBL1255944 49439 33760 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME PROTRIPTYLINE PROTRIPTYLINE 49440 33761 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME THIRAM THIRAM 49443 33762 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME TAE-684 TAE-684 49446 33763 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Bisphosphonates 10692979,12608943,18443790,19020788,15739035,12162507 49447 33764 MBNL1 4154 DRUGGABLE GENOME EPINEPHRINE BITARTRATE EPINEPHRINE BITARTRATE 49448 33765 CA2 760 DRUGGABLE GENOME, ENZYME PHENOL PHENOL 49450 33766 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CHEMBL591 ETHCHLORVYNOL 49451 33767 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME fosphenytoin FOSPHENYTOIN 49453 33768 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-37136 CHEMBL1370674 22524450 49454 33769 AKR1C3 8644 ENZYME, DRUGGABLE GENOME inhibitor 381745025 49455 33770 RACGAP1 29127 NA MORACIN M MORACIN M 49457 33771 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103571 49458 33772 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ZIDOVUDINE ZIDOVUDINE 22931300 49459 33773 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650779 ASENAPINE 49460 33774 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME OMS405 OMS405 49462 33775 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME FLAVOXATE FLAVOXATE 49463 33776 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LEUCINE LEUCINE 22931300 49464 33777 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME TEMAZEPAM TEMAZEPAM 49466 33778 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE EGF816 26825170 49467 33779 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650096 CIGLITAZONE 49468 33780 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR GSK8062 CHEMBL476302 21256005 49469 33781 MAPT 4137 DRUGGABLE GENOME SJ000113972 CHEMBL591137 49470 33782 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-124447 CHEMBL587229 49472 33783 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-31 49474 33784 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR antagonist 375973247 MIRICORILANT 49475 33785 HTT 3064 DRUGGABLE GENOME GNF-PF-4418 CHEMBL604321 49478 33786 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME PI-103 PI-103 49479 33787 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BMS-182874 BMS-182874 49480 33788 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ACACETIN ACACETIN 25190466 49481 33789 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Citalopram CITALOPRAM 49482 33790 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AT13387 49484 33791 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE NVP-AEW541 AEW-541 27196766 49485 33792 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Glyburide GLYBURIDE 49486 33793 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME methadone METHADONE 29333880 49487 33794 NFKBIA 4792 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME WEDELOLACTONE WEDELOLACTONE 22926226 49488 33795 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Gemigliptin GEMIGLIPTIN 49490 33796 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CRIZOTINIB CRIZOTINIB 49492 33797 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NORGESTIMATE NORGESTIMATE 49493 33798 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-93392 CHEMBL53738 49494 33799 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PURPURIN PURPURIN 49495 33800 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME SILIBININ SILIBININ 23401473 49497 33801 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TESTOSTERONE TESTOSTERONE 49498 33802 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TOPOTECAN TOPOTECAN 49499 33803 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE clozapine CLOZAPINE 11266078 49500 33804 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Carbamide derivative 11 49501 33805 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME 6,4'-DIHYDROXYFLAVONE CHEMBL484663 49502 33806 ABHD6 57406 PHOSPHOLIPASE, ENZYME PMID29053063-Compound-11c 49504 33807 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FLUDROCORTISONE FLUDROCORTISONE 49505 33808 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1201733 PAZOPANIB HYDROCHLORIDE 49507 33809 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL16 PHENYTOIN 49508 33810 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ZEARALENONE ZEARALENONE 49510 33811 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 vilazodone VILAZODONE 21951984 49511 33812 ATAD5 79915 NA NOCODAZOLE NOCODAZOLE 49513 33813 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR medroxyprogesterone MEDROXYPROGESTERONE ACETATE 9860300 49514 33814 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE NSC-88165 CHEMBL1709259 49515 33815 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME EUFLAVINE EUFLAVINE 49516 33816 SMN2 6607 DRUGGABLE GENOME CHRYSIN CHRYSIN 49517 33817 RAB9A 9367 ENZYME, DRUGGABLE GENOME SJ000201287 CHEMBL590900 49518 33818 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CLONAZEPAM CLONAZEPAM 49519 33819 GMNN 51053 DRUGGABLE GENOME THIOTEPA THIOTEPA 49520 33820 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME SNS-032 BMS-387032 49522 33821 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SERTRALINE HYDROCHLORIDE SERTRALINE HYDROCHLORIDE 49523 33822 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PAROXETINE HYDROCHLORIDE PAROXETINE HYDROCHLORIDE 49525 33823 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHLORHEXIDINE CHLORHEXIDINE 49526 33824 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE orciprenaline METAPROTERENOL 49527 33825 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 374883889 49528 33826 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RO-046790 CHEMBL433461 49529 33827 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TAMATINIB R-406 49530 33828 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TAMATINIB R-406 49531 33829 TMEM97 27346 NA Fused aryl carbocycle derivative 1 49532 33830 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL1879463 DACTOLISIB 49533 33831 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE LAPATINIB LAPATINIB 49534 33832 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1133 OXYBUTYNIN CHLORIDE 49536 33833 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME THIETHYLPERAZINE THIETHYLPERAZINE 49538 33834 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR KEYHOLE LIMPET HEMOCYANIN 17093201 49539 33835 GMNN 51053 DRUGGABLE GENOME GNF-PF-3725 CHEMBL598695 49540 33836 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR CI-1040 CI-1040 49541 33837 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MMV085203 CHEMBL586031 49542 33838 TSPO 706 DRUGGABLE GENOME Quinoline carboxamide derivative 9 49544 33839 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR TOREMIFENE CITRATE TOREMIFENE CITRATE 49545 33840 FANCA 2175 CLINICALLY ACTIONABLE, DNA REPAIR CISPLATIN CISPLATIN 26181256 49546 33841 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE AM-101 ESKETAMINE HYDROCHLORIDE 49547 33842 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1889140 ROPIVACAINE HYDROCHLORIDE 49549 33843 RNASE1 6035 DRUGGABLE GENOME CYTIDINE 3'-PHOSPHATE CHEMBL258728 18226913 49550 33844 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DAUNORUBICIN DAUNORUBICIN 22260166 49551 33845 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Pertuzumab PERTUZUMAB 49552 33846 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RO-106-9920 CHEMBL271023 49553 33847 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor BMS-690514 BMS-690514 49555 33848 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SB-205384 CHEMBL1256667 49556 33849 TNNT2 7139 DRUGGABLE GENOME TIRAMSETIV 49557 33850 KLK1 3816 PROTEASE, DRUGGABLE GENOME, ENZYME ECALLANTIDE ECALLANTIDE 49558 33851 F12 2161 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 178103167 49560 33852 HPSE 10855 ENZYME, DRUGGABLE GENOME HEPARIN HEPARIN 49561 33853 BAZ2B 29994 NA NSC-632536 CHEMBL1367933 49562 33854 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 49564 33855 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 404859073 49565 33856 GAPDH 2597 DRUGGABLE GENOME, ENZYME ANESTHETICS 17194030 49566 33857 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565840 49569 33858 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TOPOTECAN TOPOTECAN 49570 33859 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE BORTEZOMIB BORTEZOMIB 20578819 49571 33860 GLS 2744 ENZYME METHOTREXATE METHOTREXATE 15511236 49572 33861 TMEM97 27346 NA PMID30185082-Compound-14 49573 33862 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME ALISERTIB ALISERTIB 49574 33863 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE HF-0299 49575 33864 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE SORAFENIB SORAFENIB 49578 33865 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SB-744185 CHEMBL490417 21053897 49579 33866 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE HP-184 NERISPIRDINE 49580 33867 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE CLIOXANIDE CLIOXANIDE 49581 33868 CYP27B1 1594 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 5-AZA-2'-DEOXYCYTIDINE 15860259 49582 33869 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE AZD8835 AZD-8835 26839307 49583 33870 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody MM111 49584 33871 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PF-04236921 PF-04236921 49585 33872 NFKBIA 4792 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME DIOSCIN DIOSCIN 23621869 49586 33873 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ZAFIRLUKAST ZAFIRLUKAST 22931300 49587 33874 SMN1 6606 DRUGGABLE GENOME METHOXYVONE METHOXYVONE 49589 33875 PROS1 5627 DRUGGABLE GENOME Avatrombopag AVATROMBOPAG 49590 33876 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651526 NOREPINEPHRINE BITARTRATE 49591 33877 POLI 11201 DNA REPAIR SALIRASIB SALIRASIB 49592 33878 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AZELASTINE HYDROCHLORIDE AZELASTINE HYDROCHLORIDE 49593 33879 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650031 LEVOBUNOLOL 49594 33880 MEX3C 51320 ENZYME Bisphosphonates 49596 33881 ALOX15 246 ENZYME, DRUGGABLE GENOME 4',6,7-TRIHYDROXYISOFLAVAN CHEMBL8328 17869117 49597 33882 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417777 CHEMBL1412002 49598 33883 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROCHLORAZ PROCHLORAZ 49600 33884 BAZ2B 29994 NA NSC-92207 CHEMBL139935 49601 33885 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CIANIDANOL CIANIDANOL 49602 33886 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417111 CHEMBL2094456 49604 33887 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Ruxolitinib derivative 2 49606 33888 TFF2 7032 DRUGGABLE GENOME Gabexate GABEXATE 49607 33889 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PSAMMAPLIN A PSAMMAPLIN A 25884112 49608 33890 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Atezolizumab ATEZOLIZUMAB 49609 33891 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL3545378 MK-6592 49610 33892 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Benzimidazole derivative 7 49611 33893 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR LEE011 RIBOCICLIB 49612 33894 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL2103803 DAROTROPIUM BROMIDE 49613 33895 POLI 11201 DNA REPAIR 2-METHOXY-1,4-NAPHTHOQUINONE 2-METHOXY-1,4-NAPHTHOQUINONE 49616 33896 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1201048 DROMOSTANOLONE PROPIONATE 49617 33897 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651332 49618 33898 KCNA7 3743 ION CHANNEL, DRUGGABLE GENOME blocker 135650872 QUINIDINE 49620 33899 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME OCINAPLON OCINAPLON 49621 33900 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME TG101348 FEDRATINIB 49623 33901 CXCL8 3576 DRUGGABLE GENOME DANAZOL DANAZOL 16161451 49624 33902 GC 2638 DRUGGABLE GENOME Erythrityl Tetranitrate 49625 33903 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE MUROMONAB MUROMONAB-CD3 49626 33904 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1170 TESTOSTERONE PROPIONATE 49628 33905 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PIPLARTINE PIPLARTINE 49629 33906 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR DOCOSATETRA-7Z,10Z,13Z,16Z-ENOYL ETHANOLAMIDE CHEMBL321585 49630 33907 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME TAMATINIB R-406 49631 33908 MAPT 4137 DRUGGABLE GENOME SHIKONIN SHIKONIN 49632 33909 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE QUERCETIN QUERCETIN 49634 33910 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR calcipotriol CALCIPOTRIOL 17274004,21651652,10707958,9933478,21418277,15295697,15861036,15739035,17763859,20716226,20500803,15864137,19647104 49635 33911 GMNN 51053 DRUGGABLE GENOME TCMDC-124317 CHEMBL586937 49636 33912 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TETRAHYDROGAMBOGIC ACID TETRAHYDROGAMBOGIC ACID 49639 33913 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE QUERCETIN QUERCETIN 49640 33914 HDAC11 79885 DRUGGABLE GENOME, ENZYME PMID29671355-Compound-62 49641 33915 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 cisplatin CISPLATIN 49642 33916 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME FULVESTRANT FULVESTRANT 23448346 49643 33917 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME 178101283 49645 33918 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NEPAPRAZOLE NEPAPRAZOLE 49648 33919 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 49650 33920 SLC34A2 10568 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME antibody 252166615 49652 33921 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IPRATROPIUM IPRATROPIUM 22931300 49654 33922 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE DEPHOSTATIN DEPHOSTATIN 49655 33923 GEM 2669 NA Lirilumab LIRILUMAB 49659 33924 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SILIBININ SILIBININ 49660 33925 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE antibody LBY135 49661 33926 ATXN2 6311 NA GNF-PF-2968 CHEMBL582473 49662 33927 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENORILATE BENORILATE 49663 33928 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL LIDOCAINE LIDOCAINE 49664 33929 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME PF-06700841 BREPOCITINIB 49665 33930 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING BUTINOLINE BUTINOLINE 49666 33931 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR BELIMUMAB BELIMUMAB 49668 33932 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME PMID26293650-Compound-34 49669 33933 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME desvenlafaxine DESVENLAFAXINE 29327975 49670 33934 KDM4A 9682 DRUGGABLE GENOME, ENZYME KETOCONAZOLE KETOCONAZOLE 49671 33935 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Withacnistin 24983364 49672 33936 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME MILNACIPRAN MILNACIPRAN 49673 33937 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000024939 CHEMBL590691 49674 33938 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL419667 RELCOVAPTAN 49676 33939 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 178103304 GALANTAMINE 49678 33940 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL312443 GABOXADOL 49679 33941 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FTI-276 CHEMBL54044 49681 33942 PSMB9 5698 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL371405 MARIZOMIB 49682 33943 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME CAR-T cells targeting MucI 49683 33944 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR TRIAMCINOLONE TRIAMCINOLONE 49686 33945 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHYLTESTOSTERONE METHYLTESTOSTERONE 49687 33946 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME 1,4-BIS(2,6-DIFLUOROPHENYLSULFONYL)PIPERAZINE CHEMBL1093369 49688 33947 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IL-6 18566435 49689 33948 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME paclitaxel PACLITAXEL 30520341 49691 33949 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME CEA/MUC-1/VF/TRICOM 49693 33950 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ELLIPTECINE ELLIPTECINE 49694 33951 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE OBLIMERSEN OBLIMERSEN 49695 33952 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Salmeterol SALMETEROL 49696 33953 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1731 CHEMBL581251 49697 33954 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ALSTERPAULLONE ALSTERPAULLONE 49702 33955 GMNN 51053 DRUGGABLE GENOME TCMDC-124570 CHEMBL546475 49703 33956 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PROTRIPTYLINE PROTRIPTYLINE 49705 33957 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME sorafenib SORAFENIB 20124951 49707 33958 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME TCMDC-125221 CHEMBL546649 49708 33959 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME LEUCETTAMINE B LEUCETTAMINE B 22998443 49709 33960 TNFRSF1B 7133 DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 25850964,18565259,25537528,22129793 49710 33961 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 249565645 MK-2461 49711 33962 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-633825 CHEMBL237571 49712 33963 GAL 51083 DRUGGABLE GENOME IMMUNOTOXIN 9189270 49713 33964 MAPT 4137 DRUGGABLE GENOME SB-204741 CHEMBL323356 49715 33965 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (R)-NITRENDIPINE (R)-NITRENDIPINE 49717 33966 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE NSC-93401 CHEMBL452954 49718 33967 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME SULOCHRIN SULOCHRIN 49719 33968 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL220492 TOPIRAMATE 49720 33969 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE Anti-HER3/EGFR DAF 49721 33970 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 363894217 VORUCICLIB 49722 33971 MAP2K6 5608 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE, TUMOR SUPPRESSOR inhibitor 135652717 STAUROSPORINE 49723 33972 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE FORETINIB FORETINIB 49725 33973 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2028852 ICATIBANT ACETATE 49726 33974 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IIE AESCULIOSIDE IIE 20371180 49728 33975 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR MANNITOL MANNITOL 8670069 49729 33976 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651310 49730 33977 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051794 49731 33978 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Macrolactam derivative 4 49732 33979 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HYDROXYZINE PAMOATE HYDROXYZINE PAMOATE 49733 33980 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PHENYLBUTANOIC ACID PHENYLBUTANOIC ACID 24044874 49734 33981 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200561 DOXAZOSIN MESYLATE 49736 33982 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL3137314 ESUBERAPROST 49737 33983 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME FLUOROURACIL FLUOROURACIL 24708484 49738 33984 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER Enzastaurin ENZASTAURIN 49739 33985 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545385 WX-037 49741 33986 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Maleimides derivative 1 49742 33987 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BR-4628 49743 33988 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor XL820 49744 33989 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist 135650259 FEXARAMINE 49745 33990 CBX1 10951 NA LERCANIDIPINE LERCANIDIPINE 49746 33991 GMNN 51053 DRUGGABLE GENOME AMIODARONE AMIODARONE 49747 33992 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GAMMA-AMINOBUTYRIC ACID GAMMA-AMINOBUTYRIC ACID 49748 33993 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MICONAZOLE MICONAZOLE 49749 33994 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1319 CHEMBL235891 49751 33995 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE CENISERTIB CENISERTIB 49753 33996 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR LOTEPREDNOL ETABONATE 49754 33997 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE FX125L 49755 33998 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Anti-CD19/20-CAR vector-transduced T cells 49756 33999 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE GSK2646264 49757 34000 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 135651471 DEXAMETHASONE 49758 34001 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE fluoxetine FLUOXETINE 18695978 49759 34002 APH1B 83464 PROTEASE, DRUGGABLE GENOME MK-0752 MK-0752 49761 34003 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL98 VORINOSTAT 49763 34004 BCHE 590 DRUGGABLE GENOME, ENZYME IRINOTECAN IRINOTECAN 11345644 49766 34005 PPID 5481 DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING, KINASE US8901295, F609 49767 34006 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME CART-19/BCMA 49768 34007 BAZ2B 29994 NA DNDI1417099 CHEMBL1565444 49769 34008 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-3464 CHEMBL602213 49772 34009 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2,3-DICHLORO-PROPENE CHEMBL156075 49774 34010 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE DASATINIB DASATINIB 49777 34011 DUSP6 1848 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE RETINOIC ACID 11104676 49779 34012 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL3544960 AT-13148 49780 34013 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ZOSUQUIDAR ZOSUQUIDAR 49781 34014 POLK 51426 DNA REPAIR, ENZYME IDARUBICIN IDARUBICIN 49782 34015 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME LENALIDOMIDE LENALIDOMIDE 49783 34016 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE DISULFIRAM DISULFIRAM 49784 34017 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PHENYLBUTYRYLHYDROXAMIC ACID PHENYLBUTYRYLHYDROXAMIC ACID 21874153 49785 34018 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL3545319 EDICOTINIB 49787 34019 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 249565858 49788 34020 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR ILORASERTIB ILORASERTIB 49789 34021 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor 363894146 49792 34022 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651218 49795 34023 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME 2-METHOXYESTRADIOL 2-METHOXYESTRADIOL 17012370 49796 34024 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 OCTADEC-17-YNOIC ACID CHEMBL182310 49798 34025 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE US9040714, 155 49799 34026 GPR132 29933 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102204 49802 34027 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2014152663 701 49805 34028 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist CHEMBL1509 DROSPIRENONE 49811 34029 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR THIOPHANATE METHYL THIOPHANATE METHYL 49813 34030 POLK 51426 DNA REPAIR, ENZYME DIOTYROSINE DIOTYROSINE 49816 34031 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR CETRIMONIUM BROMIDE CETRIMONIUM BROMIDE 49818 34032 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE TANNIC ACID TANNIC ACID 49819 34033 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565637 BMS-911543 49820 34034 EPHB2 2048 KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL24828 VANDETANIB 49822 34035 BAZ2B 29994 NA DNDI1416934 CHEMBL1989750 49823 34036 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Quinoxaline derivative 5 49829 34037 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 381118836 49831 34038 XRCC5 7520 KINASE HYDROGEN PEROXIDE 11121725 49832 34039 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR 9-AMINOCAMPTOTHECIN 9-AMINOCAMPTOTHECIN 49833 34040 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LIOTHYRONINE LIOTHYRONINE 49836 34041 POLI 11201 DNA REPAIR INDIUM CHLORIDE INDIUM CHLORIDE 49837 34042 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE METHADYL ACETATE 49838 34043 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme2WO2012/098065upper 49841 34044 PACSIN2 11252 KINASE, TRANSPORTER mercaptopurine MERCAPTOPURINE 22846425,27452984 49842 34045 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR BIAFINE 9449167 49845 34046 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DICHLOROPHEN DICHLOROPHEN 49846 34047 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE CHEMOPREVENTIVE 12894495 49849 34048 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor GIVINOSTAT GIVINOSTAT 49850 34049 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ERLOTINIB ERLOTINIB 49851 34050 TMEM97 27346 NA Aryl azepine derivative 1 49852 34051 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ICILLIN ICILLIN 49855 34052 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PWT33597 49856 34053 GMNN 51053 DRUGGABLE GENOME CAPSAZEPINE CAPSAZEPINE 49860 34054 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME SP-54 PENTOSAN POLYSULFATE SODIUM 1384503 49861 34055 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 363894199 49862 34056 COL11A1 1301 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 49865 34057 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ISOPROTERENOL ISOPROTERENOL 11358333,14734046,10784181 49866 34058 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME FR-122047 FR-122047 49870 34059 BAZ2B 29994 NA DNDI1417739 CHEMBL487356 49872 34060 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TAK-715 TAK-715 49873 34061 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GENE THERAPY VECTORS 18449215 49874 34062 PRKCH 5583 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL608533 MIDOSTAURIN 49875 34063 BAZ2B 29994 NA NSC-19803 CHEMBL522983 49881 34064 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MECARBAM MECARBAM 49882 34065 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE STILONIUM IODIDE STILONIUM IODIDE 49883 34066 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-29 49884 34067 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DOXORUBICIN DOXORUBICIN 16905201,15557793 49885 34068 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-71033 CHEMBL116548 49886 34069 PPP1CA 5499 KINASE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE DEMETHYL-CANTHARIDIN DEMETHYL-CANTHARIDIN 49887 34070 MT1H 4496 NA SELENIUM 3309208 49888 34071 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME FLUOROURACIL FLUOROURACIL 20921465 49889 34072 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-69187 CHEMBL19954 49890 34073 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE LINIFANIB LINIFANIB 49891 34074 TSPO 706 DRUGGABLE GENOME Benzothiazepine analog 1 49892 34075 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE DIAZEPAM DIAZEPAM 12020046 49893 34076 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 178103952 PALBOCICLIB 49898 34077 MAPT 4137 DRUGGABLE GENOME PTI-80 49899 34078 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE 681640 CHEMBL379975 49904 34079 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor TRAMETINIB TRAMETINIB 49905 34080 AOX1 316 DRUGGABLE GENOME allopurinol ALLOPURINOL 27798726 49907 34081 CA2 760 DRUGGABLE GENOME, ENZYME DORZOLAMIDE DORZOLAMIDE 10536879 49908 34082 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PSEUDOEPHEDRINE PSEUDOEPHEDRINE 49910 34083 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE DASATINIB DASATINIB 49911 34084 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR SNS-314 SNS-314 49914 34085 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2177390 IPATASERTIB 49915 34086 POLK 51426 DNA REPAIR, ENZYME STREPTONIGRIN STREPTONIGRIN 49917 34087 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1504 TRIAMCINOLONE ACETONIDE 49919 34088 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Dabigatran DABIGATRAN 49921 34089 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PROSTAGLANDIN D2 PROSTAGLANDIN D2 23566516 49922 34090 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 9Z-RETINOIC ACID CHEMBL451158 18760926,20673632 49923 34091 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor 178101964 TRANYLCYPROMINE 49924 34092 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CUDC-101 CUDC-101 49926 34093 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME MESALAMINE MESALAMINE 49929 34094 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200769 TRIPELENNAMINE CITRATE 49930 34095 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE E75 49931 34096 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL484785 CRISABOROLE 49932 34097 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER NSC-73753 CHEMBL1506226 49934 34098 SAE1 10055 ENZYME, DRUGGABLE GENOME BETULINIC ACID BETULINIC ACID 49935 34099 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME YKP-10A SOLRIAMFETOL 49936 34100 DNER 92737 NA Isoxazole-based bicyclic compound 16 49938 34101 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 1,2-NAPHTHOQUINONE 1,2-NAPHTHOQUINONE 49940 34102 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102734 49943 34103 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000113372 CHEMBL589912 49944 34104 ALOX15B 247 DRUGGABLE GENOME, ENZYME TRICETIN TRICETIN 49946 34105 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator CHEMBL1201534 DANAPAROID SODIUM 49947 34106 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 49948 34107 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor FORETINIB FORETINIB 49949 34108 BAZ2B 29994 NA GNF-PF-3996 CHEMBL584458 49950 34109 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-1083 CHEMBL530361 49951 34110 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PF-04217903 PF-04217903 27659046 49954 34111 GMNN 51053 DRUGGABLE GENOME 2-METHOXYESTRADIOL 2-METHOXYESTRADIOL 49955 34112 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME PRAZEPAM PRAZEPAM 49956 34113 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE CETUXIMAB CETUXIMAB 21900593 49958 34114 APOE 348 DRUGGABLE GENOME CYTOKINES 9617572,10686578 49960 34115 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENOXYBENZAMINE HYDROCHLORIDE PHENOXYBENZAMINE HYDROCHLORIDE 49964 34116 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650115 CLOZAPINE 49967 34117 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLEMIZOLE CLEMIZOLE 49968 34118 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor 252166525 TALAZOPARIB 49969 34119 DUSP3 1845 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE GNF-PF-159 CHEMBL599924 49970 34120 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR AUTOANTIGEN 15084273 49971 34121 POLK 51426 DNA REPAIR, ENZYME QUINACRINE QUINACRINE 49972 34122 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME LTB4 49973 34123 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME TENOVIN-1 CHEMBL1436543 22304848 49974 34124 ANO1 55107 ION CHANNEL blocker 135650270 FLUOXETINE 49975 34125 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHACHOLINE CHLORIDE METHACHOLINE CHLORIDE 49976 34126 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME vemurafenib VEMURAFENIB 49977 34127 SIRT3 23410 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME 4-METHYLNICOTINAMIDE CHEMBL1501622 22835719 49979 34128 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist CHEMBL464 ETRETINATE 49982 34129 EML4 27436 CLINICALLY ACTIONABLE, KINASE TAE684 25228534 49985 34130 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME SNS-314 SNS-314 49986 34131 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-21 49988 34132 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME ENTRECTINIB ENTRECTINIB 49989 34133 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE agonist 178101670 49991 34134 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME NEVIRAPINE NEVIRAPINE 21189339 49993 34135 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME FR901228 ROMIDEPSIN 14767553 49994 34136 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR ROTTLERIN ROTTLERIN 22093759 49995 34137 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME PMID25435179-Compound-WO2012106509CAY10602 49996 34138 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-66209 CHEMBL175266 49998 34139 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME PHORBOL MYRISTATE ACETATE PHORBOL MYRISTATE ACETATE 24794745 49999 34140 EGLN2 112398 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3544988 DAPRODUSTAT 50001 34141 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE OPIOID 10232386 50002 34142 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GOSSYPOL GOSSYPOL 50004 34143 PCBD1 5092 ENZYME ANTISERUM 10403117 50005 34144 CA12 771 DRUGGABLE GENOME zonisamide ZONISAMIDE 21278619 50007 34145 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-61 50008 34146 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME MGCD-0103 MOCETINOSTAT 50009 34147 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 340590266 GDC-0077 50010 34148 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Dihydroisoxazole derivative 2 50011 34149 SMN1 6606 DRUGGABLE GENOME 6-AZAURIDINE 6-AZAURIDINE 50012 34150 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Hydroxamate analog 1 50013 34151 FKBP5 2289 DRUGGABLE GENOME fluoxetine FLUOXETINE 20709156,15565110 50014 34152 TH 7054 ENZYME, DRUGGABLE GENOME VITAMIN E 11172767 50017 34153 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125602 CHEMBL580183 50018 34154 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 terfenadine TERFENADINE 9187528 50019 34155 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4325 CHEMBL598263 50020 34156 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BAICALEIN BAICALEIN 50021 34157 MTR 4548 ENZYME, DRUGGABLE GENOME carboplatin CARBOPLATIN 21605004,29662106,19159907 50022 34158 CEACAM6 4680 CELL SURFACE, DRUGGABLE GENOME ANTISERUM 6388310 50023 34159 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE OPIOID 14504158 50024 34160 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 249565835 50027 34161 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR HOMIDIUM BROMIDE HOMIDIUM BROMIDE 50028 34162 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR RESMINOSTAT RESMINOSTAT 50031 34163 MSH6 2956 CLINICALLY ACTIONABLE, DNA REPAIR TEMOZOLOMIDE TEMOZOLOMIDE 17404084 50032 34164 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor 178103103 AVAGACESTAT 50033 34165 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ESTRADIOL ESTRADIOL 50034 34166 HTT 3064 DRUGGABLE GENOME VANDETANIB VANDETANIB 50035 34167 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE doxorubicin DOXORUBICIN 50036 34168 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR antagonist 223366066 GDC-0152 50038 34169 DHFR 1719 DRUGGABLE GENOME, ENZYME inhibitor 223365948 TRIMETREXATE 50039 34170 TXNRD1 7296 DRUGGABLE GENOME Disulfide compound 2 50040 34171 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR CARBAMAZEPINE CARBAMAZEPINE 50042 34172 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE COLCHICINE COLCHICINE 16239226 50043 34173 PSME1 5720 NA inhibitor CARFILZOMIB CARFILZOMIB 50044 34174 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ropivacaine ROPIVACAINE 9187528 50045 34175 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME IFN 15342387 50046 34176 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PHT-427 20197390,20418756 50047 34177 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR VISMODEGIB VISMODEGIB 19726788,25759020 50048 34178 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL2364614 LIAFENSINE 50049 34179 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 50052 34180 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL3545085 XL-228 50053 34181 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TESMILIFENE TESMILIFENE 50055 34182 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FEPRAZONE FEPRAZONE 50057 34183 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SOFALCONE SOFALCONE 50059 34184 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GDC-0941 PICTILISIB 27020857 50060 34185 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE LANATOSIDE C LANATOSIDE C 50061 34186 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME fexofenadine FEXOFENADINE 21280267 50063 34187 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE Ac-YVAD-FMK 50065 34188 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MRS-1220 CHEMBL88147 50068 34189 POLK 51426 DNA REPAIR, ENZYME HAEMATOXYLIN HAEMATOXYLIN 50069 34190 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMSG 7588311 50070 34191 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE CISPLATIN CISPLATIN 15225672 50073 34192 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BGT226 BGT-226 50074 34193 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DISULFIRAM DISULFIRAM 50075 34194 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor BORTEZOMIB BORTEZOMIB 50076 34195 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL507361 PD-0325901 50077 34196 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor 178101944 ROLIPRAM 50079 34197 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Bromodiphenhydramine BROMODIPHENHYDRAMINE 50080 34198 RIPOR2 9750 NA Drugs For Treatment Of Tuberculosis 30720667 50081 34199 PTGES 9536 DRUGGABLE GENOME, ENZYME Benzamide derivative 18 50086 34200 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL ISO-IANTHERAN A ISO-IANTHERAN A 17941622 50087 34201 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-3542 CHEMBL598477 50088 34202 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651289 50089 34203 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 187051816 CHEMBL2153434 50090 34204 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AST-487 AST-487 50091 34205 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1370561 AMINOPHYLLINE 50092 34206 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE MENTHOL MENTHOL 50093 34207 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE THIETHYLPERAZINE MALATE THIETHYLPERAZINE MALATE 50095 34208 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Metformin arginine-hemisuccinimide 50097 34209 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE 8-AZAGUANINE 8-AZAGUANINE 50098 34210 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 354702286 50099 34211 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody IPILIMUMAB IPILIMUMAB 50100 34212 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417013 CHEMBL1452227 50104 34213 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Paracetamol, combinations excl. Psycholeptics (Vicks MediNait Sirup) 50105 34214 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PSORALEN PSORALEN 50106 34215 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE KEPONE KEPONE 50108 34216 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE SCY-635 SCY 635 50113 34217 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BN-CB-045 50115 34218 PDE4C 5143 DRUGGABLE GENOME, ENZYME CS-W011402 50117 34219 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ATORVASTATIN CALCIUM ATORVASTATIN CALCIUM 50118 34220 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist 187051765 50119 34221 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist,allosteric modulator 329968434 50121 34222 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME AM-111 BRIMAPITIDE, C-TERMINAL ACID 50123 34223 PAK2 5062 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 329968394 50124 34224 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 3 50125 34225 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CAROTENOID 15657364 50126 34226 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE KTN0073-IgG1 27550450 50127 34227 MAPT 4137 DRUGGABLE GENOME 2,5-BIS(4-ISOPROPYLSTYRYL)PYRAZINE CHEMBL2181040 22913544 50129 34228 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME AR-A014418 CHEMBL259850 50130 34229 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Antibodie derivative 7 50131 34230 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Olaparib OLAPARIB 20739657,26510020,28363999,26282658 50133 34231 PDE7B 27115 DRUGGABLE GENOME, ENZYME inhibitor 178101953 50134 34232 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antibody 354702274 ISCALIMAB 50135 34233 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE FLUFENAMIC ACID FLUFENAMIC ACID 50137 34234 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 178102342 FEDRATINIB 50139 34235 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103096 APRATASTAT 50142 34236 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME sorafenib SORAFENIB 28362716 50143 34237 DCPS 28960 ENZYME, DRUGGABLE GENOME RG3039 50145 34238 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Quinoline derivative 12 50148 34239 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor XL820 50150 34240 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME Oxotetrahydro-2-H-furo[3.2-b]pyrrol-4(5-H)-yl derivative 1 50153 34241 HPRT1 3251 DRUGGABLE GENOME, ENZYME MERCAPTOPURINE MERCAPTOPURINE 50154 34242 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 187051799 DACINOSTAT 50155 34243 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor LAPATINIB LAPATINIB 50156 34244 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ETHYNODIOL DIACETATE 50157 34245 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL27759 ENTINOSTAT 50159 34246 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE TCMDC-124224 CHEMBL580421 50160 34247 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME INTERLEUKIN-1 10666367 50161 34248 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME KETOCONAZOLE KETOCONAZOLE 22931300 50162 34249 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE PALBOCICLIB PALBOCICLIB 50163 34250 AQP1 358 ION CHANNEL, DRUGGABLE GENOME inhibitor 135650790 50164 34251 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE PHENETHYLISOTHIOCYANATE PHENETHYLISOTHIOCYANATE 22607231 50165 34252 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE NSC-71033 CHEMBL116548 50166 34253 ALDH1A1 216 DRUGGABLE GENOME, ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 29938344,10469894,18854779,15237855 50167 34254 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OLOMOUCINE OLOMOUCINE 50168 34255 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR MK-2206 MK-2206 50169 34256 CA2 760 DRUGGABLE GENOME, ENZYME Ethinamate ETHINAMATE 50170 34257 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME NIRAPARIB NIRAPARIB 50171 34258 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME TAE-684 TAE-684 50172 34259 CA1 759 DRUGGABLE GENOME, ENZYME Salicyclic acid 50173 34260 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE carboplatin CARBOPLATIN 22370314,20573926,19692680,22581822,21783417,22285168,21900837,20022809 50174 34261 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-66209 CHEMBL175266 50175 34262 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME INDOMETHACIN INDOMETHACIN 17270149 50178 34263 SMN2 6607 DRUGGABLE GENOME DNDI1417260 CHEMBL2094573 50180 34264 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1095 ETHOTOIN 50181 34265 F11 2160 DRUGGABLE GENOME, PROTEASE, ENZYME ISIS-FXIRX 50182 34266 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178102299 BRIVANIB 50184 34267 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME anthracyclines and related substances 24021215 50187 34268 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor CHEMBL3545332 CEP-2563 50189 34269 FFAR4 338557 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651531 50190 34270 MAOB 4129 DRUGGABLE GENOME, ENZYME Ladostigil LADOSTIGIL 50191 34271 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 252827435 50192 34272 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR (R)-mequitazine (incontinence/respiratory disease), Pierre Fabre 50197 34273 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL494089 GSK-690693 50198 34274 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PRED 10050715 50200 34275 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565795 50201 34276 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Carfentanil CARFENTANIL 50203 34277 ABCB4 5244 TRANSPORTER, DRUGGABLE GENOME, ENZYME, ABC TRANSPORTER MITOMYCIN-C 11167651 50204 34278 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME PYRITHIONE PYRITHIONE 50205 34279 BAZ2B 29994 NA GNF-PF-3125 CHEMBL534288 50206 34280 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649655 50207 34281 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR GSK221149 RETOSIBAN 50208 34282 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER indinavir INDINAVIR 50209 34283 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BMS-770767 50210 34284 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE KD-025 CHEMBL2005186 50212 34285 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor AEE788 AEE-788 50213 34286 CBX1 10951 NA PD-169316 PD-169316 50215 34287 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TRICHOSTATIN TRICHOSTATIN 21055848,16921367,19966789,19385600 50217 34288 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME 3K3A-APC 50218 34289 NOS1 4842 DRUGGABLE GENOME, ENZYME TIRAPAZAMINE TIRAPAZAMINE 10213502 50219 34290 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR US9359293, TB 50221 34291 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-377852 CHEMBL1466186 50222 34292 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DICHLORODIMETHYLSTANNANE DICHLORODIMETHYLSTANNANE 50223 34293 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Trametinib TRAMETINIB 27338794 50225 34294 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE AMT-011 50226 34295 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor TANESPIMYCIN TANESPIMYCIN 50227 34296 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME AZD-1775 ADAVOSERTIB 50228 34297 MAPT 4137 DRUGGABLE GENOME GENTIAN VIOLET GENTIAN VIOLET 50229 34298 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-130813 CHEMBL463783 50230 34299 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME RAC-GONIOTHALAMIN CHEMBL1170485 50232 34300 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ERBSTATIN ERBSTATIN 50234 34301 FMO3 2328 ENZYME, DRUGGABLE GENOME itopride ITOPRIDE 25224784 50235 34302 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME TEMOLOZOMIDE 50237 34303 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW782612X GW782612X 50238 34304 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 187051823 50239 34305 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME CEDIRANIB CEDIRANIB 50241 34306 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL107 COLCHICINE 50242 34307 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 328083525 NEMIRALISIB 50243 34308 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GENTAMICIN GENTAMICIN 22931300 50244 34309 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 354702301 50245 34310 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GW7647 GW7647 50246 34311 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545026 FAMITINIB 50250 34312 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 249565619 PF-04691502 50252 34313 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-24 50253 34314 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652025 50254 34315 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MM-111 MM-111 50256 34316 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME DIETHYL-2-TRIDECYLMALONATE CHEMBL1797711 21292492 50257 34317 MYO9B 4650 NA CAPTOPRIL CAPTOPRIL 10052650 50258 34318 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 5 50261 34319 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AG 879 15526167 50262 34320 HSPA9 3313 NA MKT-077 CHEMBL33859 11156371 50264 34321 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PONATINIB PONATINIB 31937621 50266 34322 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 cyclophosphamide CYCLOPHOSPHAMIDE 12386121,19702528,19442086,11038165,14704462,8886611 50267 34323 CBX1 10951 NA AG-538 CHEMBL56393 50268 34324 LUM 4060 DRUGGABLE GENOME FAS LIGAND 15051477 50269 34325 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE VALNEMULIN VALNEMULIN 50270 34326 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE sulfamethoxazole / trimethoprim 26086150 50272 34327 EIF4G1 1981 NA INSULIN INSULIN 8521827 50273 34328 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RUCAPARIB RUCAPARIB 50274 34329 KDM4A 9682 DRUGGABLE GENOME, ENZYME GW7647 GW7647 50275 34330 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 29 50276 34331 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL3039508 NALDEMEDINE TOSYLATE 50277 34332 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor 178101942 50278 34333 TOP2B 7155 DRUGGABLE GENOME, ENZYME Ciprofloxacin+dexamethasone 50279 34334 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE IRINOTECAN IRINOTECAN 16799812 50281 34335 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-4029 CHEMBL596633 50282 34336 POLK 51426 DNA REPAIR, ENZYME LINOLENIC ACID LINOLENIC ACID 50283 34337 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 363894135 MERESTINIB 50285 34338 KRT20 54474 NA CISPLATIN CISPLATIN 15017198 50286 34339 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR ACRIDINE ACRIDINE 16950763 50287 34340 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000018298 CHEMBL591412 50289 34341 NDUFC2 4718 ENZYME inhibitor CHEMBL3545320 ME-344 50291 34342 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200750 PROMETHAZINE HYDROCHLORIDE 50292 34343 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME trametinib TRAMETINIB 50293 34344 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200773 TOCAINIDE HYDROCHLORIDE 50295 34345 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE PF-06463922 LORLATINIB 25749034 50298 34346 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE BI-811283 BI-811283 22350019 50299 34347 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW827099X GW827099X 50302 34348 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR inhibitor 249565817 50305 34349 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Antibodie derivative 2 50306 34350 POLB 5423 DNA REPAIR, DRUGGABLE GENOME METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 50307 34351 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BELINOSTAT BELINOSTAT 50308 34352 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Serabelisib SERABELISIB 50309 34353 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor NINTEDANIB NINTEDANIB 50310 34354 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 135650211 DROSPIRENONE 50311 34355 ATP10A 57194 ENZYME, TRANSPORTER duloxetine DULOXETINE 29407288 50312 34356 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME WEHI-539 27974663 50313 34357 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545075 LAROTRECTINIB 50314 34358 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FIPEXIDE HYDROCHLORIDE FIPEXIDE HYDROCHLORIDE 50317 34359 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL371405 MARIZOMIB 50319 34360 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME antagonist CHEMBL928 DANTROLENE SODIUM 50322 34361 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-38a 50326 34362 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE GSI-136 GSI-136 50328 34363 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME inhibitor 178101344 50329 34364 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME MAGNESIUM CHLORIDE 8747488 50330 34365 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL antidepressants 19924111,17671280,23394390 50331 34366 ALPL 249 ENZYME, DRUGGABLE GENOME GNF-PF-1609 CHEMBL600956 50332 34367 GBA 2629 DRUGGABLE GENOME, ENZYME Velaglucerase alfa 50333 34368 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor 249565816 50334 34369 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME OXAZEPAM OXAZEPAM 50336 34370 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TONABERSAT TONABERSAT 50339 34371 SLC4A1 6521 ENZYME, TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME metoprolol METOPROLOL 50341 34372 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-2356 CHEMBL601547 50342 34373 ITPR2 3709 ION CHANNEL, DRUGGABLE GENOME antagonist 135652750 50343 34374 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-693571 CHEMBL1287983 50344 34375 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TERAZOSIN TERAZOSIN 22931300 50346 34376 CHRNA5 1138 DRUGGABLE GENOME, ION CHANNEL Drugs used in nicotine dependence 25950378 50347 34377 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HYMECROMONE HYMECROMONE 50349 34378 MPI 4351 ENZYME, DRUGGABLE GENOME SJ000029642 CHEMBL591126 50351 34379 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE AI-850 50352 34380 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER GNF-PF-321 CHEMBL581044 50355 34381 POLB 5423 DNA REPAIR, DRUGGABLE GENOME 2-HYDROXYPHENAZINE 5,10-DIOXIDE CHEMBL179611 50356 34382 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BETA-CCM BETA-CCM 50358 34383 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE ATRA TRETINOIN 10837916 50359 34384 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE LENVATINIB LENVATINIB 50360 34385 POLK 51426 DNA REPAIR, ENZYME (-)-EPICATECHIN (-)-EPICATECHIN 50361 34386 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PMID29130358-Compound-Figure13(4) 50362 34387 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE IPATASERTIB IPATASERTIB 22934575 50364 34388 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR DHT ANDROSTANOLONE 11181522 50365 34389 GMNN 51053 DRUGGABLE GENOME (R)-EDELFOSINE (R)-EDELFOSINE 50367 34390 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TICLOPIDINE TICLOPIDINE 22931300 50368 34391 ST14 6768 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 405067326 50369 34392 ATF3 467 TRANSCRIPTION FACTOR PROGESTERONE PROGESTERONE 15674352 50370 34393 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME GEFITINIB GEFITINIB 50373 34394 PPIA 5478 DRUGGABLE GENOME, ENZYME CSA CYCLOSPORINE 12207006 50374 34395 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Metadoxine 50376 34396 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2108038 MATUZUMAB 50377 34397 NDUFS4 4724 ENZYME inhibitor CHEMBL3545135 NV-128 50378 34398 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NSC-176327 CHEMBL363332 50379 34399 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE DECITABINE DECITABINE 22124213 50380 34400 SCD 6319 DRUGGABLE GENOME, ENZYME Aramchol ARAMCHOL 50383 34401 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3545194 LGH-447 50389 34402 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SULFAPYRIDINE SULFAPYRIDINE 50391 34403 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR PHA-767491 CHEMBL225519 50392 34404 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 187051825 50393 34405 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL940 GABAPENTIN 50394 34406 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-14 50395 34407 TSPO 706 DRUGGABLE GENOME Bidentate pyrazolopyrimidine acetamide analog 1 50396 34408 MAOA 4128 DRUGGABLE GENOME, ENZYME MOCLOBEMIDE MOCLOBEMIDE 21680183 50397 34409 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID29757691-Compound-8c 50398 34410 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor SELICICLIB SELICICLIB 50400 34411 PRKACB 5567 ENZYME, KINASE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 135652717 STAUROSPORINE 50402 34412 NDUFS7 374291 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 50403 34413 ALDH1A1 216 DRUGGABLE GENOME, ENZYME AVOCADYNE ACETATE AVOCADYNE ACETATE 50404 34414 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 18 50405 34415 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE genistein GENISTEIN 27261451 50406 34416 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Binimetinib BINIMETINIB 27307593,23414587,28152546,26577700 50407 34417 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE SOTRASTAURIN SOTRASTAURIN 50410 34418 PDE4A 5141 DRUGGABLE GENOME, ENZYME Roflumilast ROFLUMILAST 50412 34419 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3-HYDROXYBENZYLHYDRAZINE DIHYDROCHLORIDE 50413 34420 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME TRICHOSTATIN TRICHOSTATIN 21055848,16921367,18054239,19966789,22280363,19385600 50415 34421 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PILOCARPINE NITRATE PILOCARPINE NITRATE 50416 34422 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME RIVAROXABAN RIVAROXABAN 50417 34423 ALOX15 246 ENZYME, DRUGGABLE GENOME CID 887167 CHEMBL260342 50419 34424 USP1 7398 DNA REPAIR, PROTEASE, ENZYME MECETRONIUM MECETRONIUM 50420 34425 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CURCUMIN CURCUMIN 50424 34426 TNFRSF25 8718 DRUGGABLE GENOME 178101764 50427 34427 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3545083 RGB-286638 50431 34428 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME KPT-185 27680702 50432 34429 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor DINACICLIB DINACICLIB 50433 34430 TUBA1A 7846 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 50435 34431 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR DALTEPARIN DALTEPARIN 17057417 50436 34432 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME DIMETHYL SULFOXIDE 3856429 50437 34433 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE KENPAULLONE KENPAULLONE 50439 34434 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BLY719 50440 34435 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE DEZOCINE DEZOCINE 50444 34436 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 348353622 50445 34437 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME N-OXALYLGLYCINE N-OXALYLGLYCINE 19359167 50446 34438 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 187051793 GIVINOSTAT 50447 34439 HTT 3064 DRUGGABLE GENOME APH-0812 50448 34440 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 9 50449 34441 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME E319 E319 50450 34442 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CINOLAZEPAM CINOLAZEPAM 50452 34443 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE SP-600125 SP-600125 50459 34444 TMEM97 27346 NA Piperazine derivative 7 50460 34445 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE NSC-50688 CHEMBL1456848 50463 34446 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SAR-389644 50464 34447 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CHEMBL1341 METHOXYFLURANE 50465 34448 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1201467 SYNTHETIC CONJUGATED ESTROGENS, B 50467 34449 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME Ace Inhibitors, Plain 21052031 50468 34450 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PURPUROGALLIN PURPUROGALLIN 50469 34451 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GALLAMINE GALLAMINE 50471 34452 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ALPHA-NAPHTHOFLAVONE ALPHA-NAPHTHOFLAVONE 50473 34453 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1201749 DIFLUPREDNATE 50474 34454 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ZM-447439 CHEMBL202721 50476 34455 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 phenytoin PHENYTOIN 12386121,19702528,19442086,11038165,14704462,8886611 50477 34456 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LURTOTECAN LURTOTECAN 50478 34457 PRKAB1 5564 ENZYME, KINASE, DRUGGABLE GENOME METFORMIN HYDROCHLORIDE 50480 34458 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE FF-284 26438159,25169980 50481 34459 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201562 INTERFERON BETA-1A 50482 34460 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BKM120 BUPARLISIB 26715098,26909613,22159814,27974663,24470511,23940356,28539475,26098748,26013318,28119489 50483 34461 PEMT 10400 ENZYME CHEMBL2109364 AR-20.5 50485 34462 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME DOCETAXEL DOCETAXEL 10687988,15864591 50486 34463 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE QUESTIOMYCIN B QUESTIOMYCIN B 50487 34464 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME EPIRUBICIN HYDROCHLORIDE EPIRUBICIN HYDROCHLORIDE 50488 34465 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RHODOMYRTOXIN B RHODOMYRTOXIN B 50490 34466 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-47 50494 34467 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHENETHYL ISOCYANATE PHENETHYL ISOCYANATE 23371965 50495 34468 PTGS1 5742 ENZYME, DRUGGABLE GENOME SALICYLIC ACID 50496 34469 PTGS2 5743 DRUGGABLE GENOME, ENZYME TIAPROFENIC ACID 50497 34470 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 223366169 BMS-582949 50498 34471 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE BETA-ADRENERGIC ANTAGONIST 10381893 50499 34472 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME RESERPINE RESERPINE 50500 34473 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Isoindoline derivative 5 50502 34474 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME N-METHYL-N-NITROSOUREA 2415236 50505 34475 ATP2C1 27032 ENZYME, TRANSPORTER, DRUGGABLE GENOME ENFLURANE ENFLURANE 50506 34476 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 losigamone LOSIGAMONE 12386121,19702528,19442086,11038165,14704462,8886611 50508 34477 GADD45A 1647 DNA REPAIR, TUMOR SUPPRESSOR, KINASE CHELATORS 10397746 50509 34478 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 clarithromycin CLARITHROMYCIN 9951426,9187528 50510 34479 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER lamivudine LAMIVUDINE 23996099 50511 34480 MYLK 4638 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE ME-3407 50512 34481 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME DIPHENYLUREA DIPHENYLUREA 50514 34482 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DIMENHYDRINATE DIMENHYDRINATE 50515 34483 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CAR-T cells recognizing EpCAM 50516 34484 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR LORATADINE LORATADINE 50518 34485 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME blocker 178100936 50522 34486 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650115 CLOZAPINE 50523 34487 TPK1 27010 KINASE, ENZYME ANTIMETABOLITE 228770 50524 34488 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist CHEMBL3833307 SATRALIZUMAB 50525 34489 PDE4B 5142 DRUGGABLE GENOME, ENZYME Revamilast REVAMILAST 50526 34490 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VB6-845 CITATUZUMAB BOGATOX 50528 34491 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME EBSELEN EBSELEN 50529 34492 NUDT15 55270 ENZYME, CLINICALLY ACTIONABLE mercaptopurine MERCAPTOPURINE 27530327,26503813,28146264,27558924,29967377,30035323,29923122,28659275,27381176,26590936,27193222,26878724,30048756,28445187,26033531,27416873,26076924,27604507,26735160,27577869,30101994,27095468 50530 34493 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ZINC 00387478 CHEMBL1668301 21419531 50531 34494 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Imidazo[1,2-b]pyridazine derivative 2 50532 34495 TAC1 6863 DRUGGABLE GENOME RESERPINE RESERPINE 6174352,6183051 50534 34496 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR PU-H71 PU-H71 50535 34497 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651003 50536 34498 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Trastuzumab-DM1 ADO-TRASTUZUMAB EMTANSINE 50538 34499 MAPT 4137 DRUGGABLE GENOME GNF-PF-4283 CHEMBL606166 50539 34500 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PYROGALLOL PYROGALLOL 50540 34501 POLK 51426 DNA REPAIR, ENZYME NSC-19803 CHEMBL522983 50541 34502 RPS6KB2 6199 DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME, KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545134 LY-2780301 50542 34503 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135649989 BEZAFIBRATE 50543 34504 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE OXYTETRACYCLINE HYDROCHLORIDE OXYTETRACYCLINE HYDROCHLORIDE 50544 34505 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE CISPLATIN CISPLATIN 28490518 50545 34506 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652340 CHEMBL446325 50546 34507 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-34 50547 34508 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CHLORHEXIDINE HYDROCHLORIDE CHLORHEXIDINE HYDROCHLORIDE 50548 34509 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CENISERTIB CENISERTIB 50550 34510 IFNG 3458 DRUGGABLE GENOME THROMBIN THROMBIN 9731747 50552 34511 COL18A1 80781 DRUGGABLE GENOME CAMPTOTHECIN CAMPTOTHECIN 15069724 50553 34512 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DANTROLENE DANTROLENE 22931300 50554 34513 MMP15 4324 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103981 ILOMASTAT 50555 34514 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DEOXYSAPPANONE B TRIMETHYL ETHER DEOXYSAPPANONE B TRIMETHYL ETHER 50556 34515 CD63 967 CELL SURFACE, DRUGGABLE GENOME, KINASE NONSTEROIDAL ANTI-INFLAMMATORY DRUGS 15608437 50559 34516 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME LEUCOVORIN LEUCOVORIN 11237386 50560 34517 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR HISPIDIN HISPIDIN 50561 34518 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME NSC-748113 CHEMBL2063687 22283430 50562 34519 EHMT1 79813 ENZYME, DRUGGABLE GENOME inhibitor 178103593 CHEMBL569864 50563 34520 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL274654 ORANTINIB 50564 34521 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Dacomitinib DACOMITINIB 26561558,25939761 50565 34522 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PERGOLIDE MESYLATE PERGOLIDE MESYLATE 50566 34523 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE VELIPARIB VELIPARIB 50568 34524 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME IPILIMUMAB IPILIMUMAB 50569 34525 EPHX2 2053 DRUGGABLE GENOME, ENZYME GSK2256294 50572 34526 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR R-1487 R-1487 50573 34527 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME BMS-204493 CHEMBL472172 19216008,18702457 50574 34528 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000069305 CHEMBL603739 50575 34529 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Aminopyrimidine derivative 6 50577 34530 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CISPLATIN CISPLATIN 50578 34531 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX AROMATICIN AROMATICIN 50579 34532 SLC22A11 55867 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor CHEMBL897 PROBENECID 50583 34533 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Pyrimethamine PYRIMETHAMINE 50584 34534 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR CEFOTAXIME SODIUM CEFOTAXIME SODIUM 50586 34535 CBX1 10951 NA NSC-3323 CHEMBL1270169 50588 34536 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME STAUROSPORINE STAUROSPORINE 22705001 50589 34537 BAZ2B 29994 NA TCMDC-125319 CHEMBL527586 50591 34538 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-15 50592 34539 GSTM1 2944 DRUGGABLE GENOME, ENZYME taxanes 27785604 50593 34540 KAT2B 8850 ENZYME, DRUGGABLE GENOME inhibitor 187051809 50594 34541 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME SP-600125 SP-600125 50596 34542 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GLAUCINE METHIODIDE GLAUCINE METHIODIDE 50598 34543 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Trastuzumab emtansine 50600 34544 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE cyanocobalamin CYANOCOBALAMIN 29662106,20634689,19307503 50603 34545 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORPROMAZINE HYDROCHLORIDE CHLORPROMAZINE HYDROCHLORIDE 50605 34546 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NLG802 50607 34547 RGS4 5999 DRUGGABLE GENOME olanzapine OLANZAPINE 50608 34548 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME EFAVIRENZ EFAVIRENZ 17041008 50609 34549 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR STILONIUM IODIDE STILONIUM IODIDE 50610 34550 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE GW441756X GW441756X 50612 34551 NCOA3 8202 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, ENZYME TCMDC-137788 CHEMBL587564 50613 34552 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MOMETASONE FUROATE MOMETASONE FUROATE 50615 34553 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3544963 DS-3078A 50616 34554 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER grapefruit juice 50618 34555 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 249565689 50619 34556 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-27 50621 34557 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME AVOBENZONE AVOBENZONE 50622 34558 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651569 50625 34559 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SALBUTAMOL ALBUTEROL 50627 34560 SOAT1 6646 DRUGGABLE GENOME TESTOSTERONE TESTOSTERONE 2765620 50628 34561 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IDARUBICIN IDARUBICIN 50629 34562 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL254760 MGCD-265 50631 34563 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 249565800 50633 34564 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SULFINPYRAZONE SULFINPYRAZONE 50634 34565 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor GIVINOSTAT GIVINOSTAT 50635 34566 POLK 51426 DNA REPAIR, ENZYME HYPERICIN HYPERICIN 50636 34567 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-74429 CHEMBL1269022 50637 34568 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME METHYL 4-(3-METHOXYBENZAMIDO)BENZOATE CHEMBL1214407 50638 34569 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HARMINE HYDROCHLORIDE HARMINE HYDROCHLORIDE 50640 34570 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR OMEPRAZOLE OMEPRAZOLE 11100337 50641 34571 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DOPAMINE DOPAMINE 50642 34572 TESK2 10420 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TYROSINE KINASE inhibitor 249565797 50643 34573 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR antagonist 381745028 50644 34574 GMNN 51053 DRUGGABLE GENOME AZELNIDIPINE AZELNIDIPINE 50645 34575 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE DOVITINIB DOVITINIB 24124571 50646 34576 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 24 50647 34577 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 223366060 50648 34578 CBX1 10951 NA NSC-102742 CHEMBL1519374 50649 34579 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE SNS-314 SNS-314 50650 34580 RAC1 5879 CLINICALLY ACTIONABLE, KINASE, DRUG RESISTANCE PLX4720 PLX-4720 31257073 50652 34581 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE iOWH032 IOWH-032 50654 34582 ATXN2 6311 NA TCMDC-123920 CHEMBL1606 50656 34583 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 385612201 50657 34584 MAPT 4137 DRUGGABLE GENOME STAUROSPORINE AGLYCON STAUROSPORINE AGLYCON 50659 34585 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL98 VORINOSTAT 50663 34586 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PF-885706 50664 34587 MAPT 4137 DRUGGABLE GENOME ELLIPTECINE ELLIPTECINE 50665 34588 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE pitrakinra PITRAKINRA 50667 34589 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME leucovorin LEUCOVORIN 20125120,25955730 50668 34590 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL OCINAPLON OCINAPLON 50669 34591 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENAZINE PHENAZINE 50670 34592 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE CYCLOHEXIMIDE CYCLOHEXIMIDE 15974627 50671 34593 MAPT 4137 DRUGGABLE GENOME BAICALEIN BAICALEIN 50673 34594 CTH 1491 ENZYME inhibitor 252827517 AMINOETHOXYVINYLGLYCINE 50674 34595 TUBA1C 84790 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 50675 34596 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 10 50676 34597 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-5134 CHEMBL602969 50677 34598 BAZ2B 29994 NA GNF-PF-628 CHEMBL1448140 50679 34599 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-PYRIDYLKETONE BENZOYL HYDRAZONE CHEMBL252151 50681 34600 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE FGF-1 FIBROBLAST GROWTH FACTOR-1 16682955 50685 34601 ADH7 131 DRUGGABLE GENOME, ENZYME anthracyclines and related substances 23441093,21900104 50687 34602 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103736 FENOPROFEN CALCIUM 50688 34603 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME BETAMETHASONE BETAMETHASONE 50689 34604 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-123528 CHEMBL529138 50690 34605 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL744 RILUZOLE 50691 34606 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALCIPOTRIOL CALCIPOTRIOL 50692 34607 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PENTACHLORONITROBENZENE PENTACHLORONITROBENZENE 50693 34608 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE SP-600125 SP-600125 23498914 50697 34609 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor ROMIDEPSIN ROMIDEPSIN 50701 34610 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor PWT33597 50702 34611 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Panitumumab PANITUMUMAB 26341920 50703 34612 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME haloperidol HALOPERIDOL 27023437 50704 34613 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE IODOQUINOL IODOQUINOL 50707 34614 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Etoposide ETOPOSIDE 23536011 50709 34615 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitory allosteric modulator MK2206 MK-2206 50710 34616 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME Efavirenz EFAVIRENZ 50711 34617 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL2108675 DUPILUMAB 50714 34618 NCOA3 8202 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, ENZYME METHOTREXATE METHOTREXATE 50716 34619 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CPT-11 IRINOTECAN HYDROCHLORIDE 10639573 50718 34620 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-44 50719 34621 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME tafamidis TAFAMIDIS 50720 34622 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Benzonaphthyridine derivative 1 50721 34623 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Sunitinib SUNITINIB 50722 34624 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 178103585 ROMIDEPSIN 50723 34625 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME GLUCOCORTICOID 12123742 50725 34626 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CENTAUREIDIN CENTAUREIDIN 50727 34627 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PRAZOSIN PRAZOSIN 50728 34628 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE NSC-319994 CHEMBL1329443 50729 34629 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL1743044 NAMILUMAB 50730 34630 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE BEAUVERICIN BEAUVERICIN 16297711 50731 34631 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 50732 34632 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL571948 Y-39983 50733 34633 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROCHLORPERAZINE EDISYLATE PROCHLORPERAZINE EDISYLATE 50735 34634 ATAD5 79915 NA OXOPURPUREINE OXOPURPUREINE 50736 34635 GCLM 2730 ENZYME MELATONIN MELATONIN 10515588 50738 34636 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antidepressants 50740 34637 POLI 11201 DNA REPAIR (+)-TAXIFOLIN (+)-TAXIFOLIN 50741 34638 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PROPRANOLOL PROPRANOLOL 14744938 50744 34639 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SORAFENIB SORAFENIB 50746 34640 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BMS-204493 CHEMBL472172 18702457 50752 34641 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE methamphetamine METHAMPHETAMINE 16402083 50753 34642 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 384403638 50755 34643 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PALBOCICLIB PALBOCICLIB 50756 34644 MAOB 4129 DRUGGABLE GENOME, ENZYME ISOCARBOXAZID ISOCARBOXAZID 50757 34645 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR ATORVASTATIN ATORVASTATIN 15792677 50758 34646 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER sparfloxacin SPARFLOXACIN 50759 34647 CXCL8 3576 DRUGGABLE GENOME LEFLUNOMIDE LEFLUNOMIDE 10902750 50760 34648 VKORC1 79001 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200879 WARFARIN SODIUM 50761 34649 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-2059 CHEMBL601968 50762 34650 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Deutetrabenazine DEUTETRABENAZINE 50766 34651 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor 178103151 50767 34652 PSMD7 5713 PROTEASE CARFILZOMIB CARFILZOMIB 24524217 50768 34653 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE CEDIRANIB CEDIRANIB 50769 34654 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME ezetimibe / simvastatin 50770 34655 RGS4 5999 DRUGGABLE GENOME D-ALANINE D-ALANINE 50771 34656 IL1B 3553 KINASE, DRUGGABLE GENOME CYT-013-IL1bQb 50772 34657 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2029988 CEP-32496 50773 34658 UGT1A6 54578 ENZYME, DRUGGABLE GENOME DICLOFENAC DICLOFENAC 8511777 50774 34659 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MYRICETIN MYRICETIN 50775 34660 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AT13148 AT-13148 22781553 50776 34661 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 187051774 ALVIMOPAN 50777 34662 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE carboplatin CARBOPLATIN 26033044 50778 34663 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Carboxamide derivative 7 50779 34664 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1084172 VILANTEROL TRIFENATATE 50780 34665 TSPO 706 DRUGGABLE GENOME Bidentate pyrazolopyrimidine acetamide analog 3 50781 34666 CA12 771 DRUGGABLE GENOME ACETAZOLAMIDE ACETAZOLAMIDE 50782 34667 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AY-9944 CHEMBL1513392 50783 34668 ATP2C1 27032 ENZYME, TRANSPORTER, DRUGGABLE GENOME SEVOFLURANE SEVOFLURANE 50784 34669 IDE 3416 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, ENZYME, PROTEASE N-(4-NITROPHENYL)ANTHRANILIC ACID CHEMBL1574420 50785 34670 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME hmg coa reductase inhibitors 27839692 50787 34671 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PMID27376512-Compound-Figure3CN 50788 34672 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE ERLOTINIB ERLOTINIB 50790 34673 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178102316 CHEMBL1908395 50792 34674 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME E-64C E-64C 50794 34675 GMNN 51053 DRUGGABLE GENOME NSC-172614 CHEMBL1317506 50798 34676 PSMD13 5719 NA inhibitor BORTEZOMIB BORTEZOMIB 50799 34677 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE CWP232291 50805 34678 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 354702283 50806 34679 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE GS-9411 50807 34680 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER PMEA 12695538,10470083 50808 34681 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE POSIPHEN PHENSERINE, (+)- 50810 34682 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor AS703569 CENISERTIB 50811 34683 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIPYRIDAMOLE DIPYRIDAMOLE 50812 34684 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE 1R,9S-HYDRASTINE 1R,9S-HYDRASTINE 50814 34685 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME carbamazepine CARBAMAZEPINE 21738081 50817 34686 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Larotrectinib LAROTRECTINIB 50818 34687 GMNN 51053 DRUGGABLE GENOME GNF-PF-4291 CHEMBL585462 50819 34688 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 50820 34689 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 387065596 50821 34690 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200715 HEXYLCAINE HYDROCHLORIDE 50822 34691 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heteroaryl-carboxamide derivative 7 50823 34692 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RANITIDINE RANITIDINE 22931300 50825 34693 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HYDRASTININE HYDRASTININE 50827 34694 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE HYDROQUINONE HYDROQUINONE 50828 34695 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GLIQUIDONE GLIQUIDONE 50829 34696 CES1 1066 DRUGGABLE GENOME, ENZYME enalapril ENALAPRIL 25919042 50830 34697 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-2713 CHEMBL578719 50831 34698 LGALS3 3958 CELL SURFACE, DRUGGABLE GENOME Antibiotics 25869013 50832 34699 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE MGCD265 GLESATINIB 50833 34700 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PHENOTHIAZINE PHENOTHIAZINE 16750172 50834 34701 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TETRABROMOBENZOTRIAZOLE TETRABROMOBENZOTRIAZOLE 50836 34702 CDKN3 1033 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, TUMOR SUPPRESSOR, ENZYME, KINASE inhibitor CHEMBL488436 AZD-5438 50837 34703 BAZ2B 29994 NA PROPIDIUM PROPIDIUM 50838 34704 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX RETINOIC ACID 7521842 50840 34705 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Azaindole derivative 1 50843 34706 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE CAR-T cells targeting Glypican-3 (GPC3) 50844 34707 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 363894209 PAMAPIMOD 50847 34708 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Pratosartan PRATOSARTAN 50848 34709 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE OXALIPLATIN OXALIPLATIN 50849 34710 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 315661258 RIPRETINIB 50850 34711 TRIT1 54802 NA 5-AZACYTIDINE AZACITIDINE 2479825 50851 34712 ACP3 55 ENZYME, DRUGGABLE GENOME MVI-816 50853 34713 AKR1C3 8644 ENZYME, DRUGGABLE GENOME NSAIDS 12543809 50854 34714 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DISULFIRAM DISULFIRAM 50855 34715 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Afeletecan AFELETECAN 21547368 50856 34716 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE dolutegravir DOLUTEGRAVIR 50858 34717 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME CHLORFENAPYR CHLORFENAPYR 50860 34718 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Isoquinoline derivative 4 50861 34719 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DOCETAXEL DOCETAXEL 10639573 50862 34720 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TRIPROLIDINE TRIPROLIDINE 50864 34721 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL1201733 PAZOPANIB HYDROCHLORIDE 50866 34722 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HYDROCORTISONE HYDROCORTISONE 14705237,1647304 50867 34723 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL482968 ENMD-2076 50868 34724 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Regorafenib REGORAFENIB 21170960,23629727,25838391 50869 34725 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CGS-12066A MALEATE CHEMBL1256689 50871 34726 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 2877750 50873 34727 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PMID25726713-Compound-50 50875 34728 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR NSC-95397 CHEMBL429095 50877 34729 TUBA4A 7277 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 50878 34730 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor SOPHORETIN QUERCETIN 50879 34731 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME EMEDASTINE EMEDASTINE 50880 34732 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650882 RAGAGLITAZAR 50882 34733 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME TAE-684 TAE-684 50883 34734 POLK 51426 DNA REPAIR, ENZYME GNF-PF-254 CHEMBL461579 50884 34735 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME ENTRECTINIB ENTRECTINIB 50887 34736 FST 10468 DRUGGABLE GENOME ANTICOAGULANT 15128279 50888 34737 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor AT9283 AT-9283 50889 34738 HSPA8 3312 TUMOR SUPPRESSOR ATRA TRETINOIN 8578578 50891 34739 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VB-111 OFRANERGENE OBADENOVEC 50895 34740 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ORTHOTOLIDINE ORTHOTOLIDINE 50898 34741 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE TAMATINIB R-406 50899 34742 ADM 133 DRUGGABLE GENOME, HORMONE ACTIVITY paroxetine PAROXETINE 19636336 50900 34743 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565732 50901 34744 LANCL2 55915 NA 384403643 50905 34745 RBP4 5950 DRUGGABLE GENOME US9434727, 40 50906 34746 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GEFITINIB GEFITINIB 50908 34747 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GRISEOFULVIN GRISEOFULVIN 50909 34748 ATXN2 6311 NA TCMDC-124063 CHEMBL534535 50910 34749 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme9EHT5372 50912 34750 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TETRACYCLINE TETRACYCLINE 22931300 50913 34751 SV2A 9900 DRUGGABLE GENOME, TRANSPORTER Levetiracetam LEVETIRACETAM 50915 34752 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME gemcitabine GEMCITABINE 50919 34753 PDE3A 5139 ENZYME, DRUGGABLE GENOME Oxtriphylline OXTRIPHYLLINE 50920 34754 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME 4-(4-AMINOPHENYL)BUTANOIC ACID CHEMBL1650245 24044874 50923 34755 TAC1 6863 DRUGGABLE GENOME BUTYRATE 17187013 50926 34756 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TOPOISOMERASE INHIBITORS 2553992 50927 34757 TUBB6 84617 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 50928 34758 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL551064 AEW-541 50929 34759 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CLOPIDOGREL CLOPIDOGREL 50930 34760 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor LGX818 ENCORAFENIB 50933 34761 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME N/A 50935 34762 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (S)-NITRENDIPINE (S)-NITRENDIPINE 50936 34763 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AMIODARONE AMIODARONE 50938 34764 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CENISERTIB CENISERTIB 50939 34765 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 381118896 50940 34766 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE agonist CHEMBL1743003 CONATUMUMAB 50942 34767 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MORICIZINE HYDROCHLORIDE MORICIZINE HYDROCHLORIDE 50943 34768 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL488436 AZD-5438 50945 34769 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Plasminogen concentrate 50946 34770 FAAH2 158584 DRUGGABLE GENOME, ENZYME inhibitor 381744930 50947 34771 RAPGEF3 10411 ENZYME PYROGALLOL RED PYROGALLOL RED 50948 34772 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE TOZASERTIB TOZASERTIB 50949 34773 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE SORAFENIB SORAFENIB 50950 34774 PRMT6 55170 ENZYME, METHYL TRANSFERASE inhibitor 315661318 50951 34775 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE THIRAM THIRAM 50952 34776 TXNRD1 7296 DRUGGABLE GENOME Spermidine SPERMIDINE 50953 34777 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545139 PS-516895 50955 34778 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL539843 VAPITADINE DIHYDROCHLORIDE 50956 34779 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 2-MERCAPTOBENZIMIDAZOLE 2-MERCAPTOBENZIMIDAZOLE 50958 34780 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME B-RAF/VEGFR-2 INHIBITOR RAF265 25199829 50960 34781 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME PACLITAXEL PACLITAXEL 9588740 50961 34782 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METIPRANOLOL METIPRANOLOL 50962 34783 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR GSK-557296 EPELSIBAN 50965 34784 IL6ST 3572 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE RALOXIFENE RALOXIFENE 24456369 50966 34785 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PERVILLEINE F PERVILLEINE F 11754602 50967 34786 PGRMC1 10857 NA OPC-14523 50970 34787 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32o 50972 34788 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR ILORASERTIB ILORASERTIB 50973 34789 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TANSHINONE I TANSHINONE I 50975 34790 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor PANOBINOSTAT PANOBINOSTAT 50976 34791 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOFISOPAM TOFISOPAM 50977 34792 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 178101154 50981 34793 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 178102309 PICTILISIB 50982 34794 ESRRG 2104 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DIETHYLSTILBESTROL DIETHYLSTILBESTROL 12579585 50983 34795 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE ESTRADIOL BENZOATE 18084728 50984 34796 USP1 7398 DNA REPAIR, PROTEASE, ENZYME AMARANTH AMARANTH 50986 34797 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 9389690 50987 34798 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrrolo-pyridone derivative 1 50989 34799 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE digoxin DIGOXIN 22543981 50990 34800 LTB 4050 DRUGGABLE GENOME abacavir ABACAVIR 50991 34801 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR FULVESTRANT FULVESTRANT 17029634 50993 34802 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-2812 CHEMBL125044 50994 34803 ATXN2 6311 NA DNDI1417420 CHEMBL1546223 50995 34804 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101492 PAROXETINE 50997 34805 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE inhibitor PF-03084014 NIROGACESTAT 50998 34806 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Tagraxofusp TAGRAXOFUSP 50999 34807 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor BAY1000394 51000 34808 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME METHYLDOPA METHYLDOPA 51005 34809 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE M-COPA 27197184 51006 34810 NDUFA5 4698 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 51007 34811 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL3707396 EVT401 51008 34812 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BACLOFEN BACLOFEN 51012 34813 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME partial agonist CHEMBL2103991 BALAGLITAZONE 51014 34814 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DYDROGESTERONE DYDROGESTERONE 51016 34815 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CLOBAZAM CLOBAZAM 51018 34816 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RHODAMINE RHODAMINE 51019 34817 ALOX15B 247 DRUGGABLE GENOME, ENZYME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 51021 34818 FURIN 5045 ENZYME, PROTEASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 252166868 51022 34819 PMEL 6490 DRUGGABLE GENOME GPA-TriMAR-T cells 51025 34820 ATXN2 6311 NA BROMOENOL LACTONE BROMOENOL LACTONE 51026 34821 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ESCITALOPRAM ESCITALOPRAM 51027 34822 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NUTLIN-3A 17671205 51028 34823 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor CARFILZOMIB CARFILZOMIB 51029 34824 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1113 AMOXAPINE 51030 34825 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 315661176 51031 34826 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL495727 AT-9283 51032 34827 RGS4 5999 DRUGGABLE GENOME PODOCARIC ACID PODOCARIC ACID 51033 34828 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor SNS-032 BMS-387032 51034 34829 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR MIFEPRISTONE MIFEPRISTONE 51035 34830 MPHOSPH8 54737 NA SURAMIN HEXASODIUM SURAMIN HEXASODIUM 51036 34831 TH 7054 ENZYME, DRUGGABLE GENOME OPIATE 1849802 51037 34832 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DIENOGEST DIENOGEST 51039 34833 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME DM-99 51040 34834 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME OSI-027 OSI-027 21673091,26725216 51041 34835 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SCANDENIN SCANDENIN 51042 34836 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 385612183 51043 34837 CBX1 10951 NA GNF-PF-4283 CHEMBL606166 51044 34838 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 51046 34839 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL2103852 CROLIBULIN 51047 34840 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME TCMDC-125758 CHEMBL546797 51048 34841 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 11 51049 34842 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME blocker 178101137 51053 34843 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-747261 CHEMBL593366 51054 34844 EPAS1 2034 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX HALICLONADIAMINE HALICLONADIAMINE 22928967 51055 34845 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ISOQUERCETIN ISOQUERCETIN 51057 34846 ALOX5 240 DRUGGABLE GENOME, ENZYME ZILEUTON ZILEUTON 24697244,19492852,25686392 51058 34847 CDC42BPA 8476 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565832 51060 34848 ALDH1A1 216 DRUGGABLE GENOME, ENZYME thiotepa THIOTEPA 18854779 51061 34849 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ALTENUSIN ALTENUSIN 51062 34850 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1628502 GABAPENTIN ENACARBIL 51064 34851 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE S-222611 S-222611 24837299,25434923 51066 34852 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ARACHIDONIC ACID ARACHIDONIC ACID 51070 34853 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY 13-CIS-RETINOIC ACID 17006844 51071 34854 SERPINH1 871 PROTEASE INHIBITOR, DRUGGABLE GENOME ANTISENSE OLIGONUCLEOTIDES 9714184 51072 34855 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HISPIDIN HISPIDIN 51075 34856 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL521851 PICTILISIB 51077 34857 IKBKG 8517 KINASE, DRUGGABLE GENOME sulfadoxine SULFADOXINE 51078 34858 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE dapsone DAPSONE 12387962,20599264,18349424,24372186,20701405,15183620 51079 34859 DPP9 91039 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 363894200 TENELIGLIPTIN 51080 34860 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TRIMEPRAZINE METHYLPROMAZINE 51081 34861 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178100241 CELECOXIB 51085 34862 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME HUMAN CHORIONIC GONADOTROPIN 11585432 51086 34863 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C8 51087 34864 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103089 LY-2886721 51091 34865 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID25416646-Compound-Figure5-C 51092 34866 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 4-PHENYLPHENOL CHEMBL73380 51093 34867 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME CEPHALOCHROMIN CEPHALOCHROMIN 51094 34868 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 223366076 51098 34869 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 178103565 51099 34870 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 51100 34871 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE talazoparib TALAZOPARIB 51102 34872 POLK 51426 DNA REPAIR, ENZYME ACRISORCIN ACRISORCIN 51103 34873 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ANISOMYCIN ANISOMYCIN 51105 34874 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 L-765314 L-765314 51106 34875 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE NILOTINIB NILOTINIB 20537386,19075254,18191450,25686603,19652056,16772610 51107 34876 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER fentanyl FENTANYL 29601950,22277678,27883323,17192767,19514130,23557865 51108 34877 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 223366126 DUVELISIB 51110 34878 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1255654 TETRACAINE HYDROCHLORIDE 51111 34879 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SPIRADOLINE SPIRADOLINE 51113 34880 KDM4A 9682 DRUGGABLE GENOME, ENZYME GARCINONE E GARCINONE E 51115 34881 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE TGFBETA1 8900367 51116 34882 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LOTEPREDNOL ETABONATE LOTEPREDNOL ETABONATE 51118 34883 PSENEN 55851 DRUGGABLE GENOME NIC5-15 METHYLINOSITOL 51119 34884 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL2035187 PACRITINIB 51120 34885 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL705 ALITRETINOIN 51122 34886 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650290 51123 34887 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER APG-115 51124 34888 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Flavonoid derivative 5 51125 34889 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (S)-ROSCOVITINE (S)-ROSCOVITINE 51126 34890 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-21 51128 34891 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CETUXIMAB CETUXIMAB 23729478 51129 34892 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE GSK2126458 OMIPALISIB 22733540 51131 34893 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SULFORAPHANE SULFORAPHANE 20395150 51132 34894 IL1B 3553 KINASE, DRUGGABLE GENOME FLUTICASONE PROPIONATE 11943316 51135 34895 PDE3A 5139 ENZYME, DRUGGABLE GENOME Cilostazol CILOSTAZOL 51137 34896 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL3545063 OSIMERTINIB MESYLATE 51138 34897 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 178101155 51140 34898 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 1540951 CHEMBL259421 51141 34899 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PHENMEDIPHAM PHENMEDIPHAM 51143 34900 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE VANDETANIB VANDETANIB 51144 34901 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RO-0505082 CHEMBL2164761 51146 34902 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME ERYTHROPOIESIS-STIMULATING AGENT 51147 34903 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME lamivudine LAMIVUDINE 23089673 51149 34904 HTT 3064 DRUGGABLE GENOME DAC-060 22416777 51150 34905 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE modulator CHEMBL190083 TARENFLURBIL 51152 34906 DCN 1634 DRUGGABLE GENOME IFN 12707320 51153 34907 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME COLCHICINE COLCHICINE 9667638,17291686 51154 34908 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE DP-b99 51156 34909 PON2 5445 DRUGGABLE GENOME, ENZYME antidepressants 51157 34910 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE URACIL URACIL 1682063 51158 34911 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME antagonist 223366062 AT-406 51159 34912 LDHA 3939 DRUGGABLE GENOME TETRAHYDRO-NAD CHEMBL2058994 22417091 51160 34913 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL2146146 ATROPINE SULFATE 51162 34914 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME [14C]-TACRINE MONOHYDRATE MONOHYDROCHLORIDE CHEMBL1337960 51163 34915 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ELLAGIC ACID ELLAGIC ACID 51164 34916 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR VE-821 25593184 51165 34917 HBEGF 1839 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME U3-1565 51166 34918 MAPT 4137 DRUGGABLE GENOME HEMATOXYLIN HEMATOXYLIN 51167 34919 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE paclitaxel PACLITAXEL 21151855 51169 34920 GMNN 51053 DRUGGABLE GENOME 2-(STYRYL)-BENZIMIDAZOLE CHEMBL473721 51171 34921 PTGS1 5742 ENZYME, DRUGGABLE GENOME Gamma-Homolinolenic acid 51173 34922 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME H-89 CHLORIDE CHEMBL1315166 51174 34923 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE PEG-INTERFERON ALFACON-1 51176 34924 S100B 6285 DRUGGABLE GENOME, KINASE PHENOTHIAZINE PHENOTHIAZINE 6947252 51179 34925 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE BGC20-1531 51180 34926 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-415286 CHEMBL322970 51181 34927 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR ANESTHETICS 11942866 51183 34928 ABAT 18 DRUGGABLE GENOME, ENZYME inhibitor 252166496 CPP-115 51184 34929 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-(STYRYL)-BENZIMIDAZOLE CHEMBL473721 51185 34930 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR METHYLPREDNISOLONE METHYLPREDNISOLONE 51186 34931 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PAPAVERINE HYDROCHLORIDE PAPAVERINE HYDROCHLORIDE 51187 34932 TMEM97 27346 NA PMID28051882-Compound-XIV 51189 34933 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OXYPHENBUTAZONE OXYPHENBUTAZONE 51190 34934 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE MK-2206 MK-2206 51192 34935 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-123927 CHEMBL531268 51193 34936 MAOB 4129 DRUGGABLE GENOME, ENZYME SELEGILINE SELEGILINE 21680183,23631427 51194 34937 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL576982 QUIZARTINIB 51195 34938 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER inhibitor CHEMBL348475 TARIQUIDAR 51196 34939 AQP9 366 ION CHANNEL FLUTAMIDE FLUTAMIDE 12021052 51198 34940 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antineoplastic agents 21487324 51199 34941 NEK6 10783 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565885 51200 34942 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200491 EPINASTINE HYDROCHLORIDE 51202 34943 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3352 CHEMBL600306 51203 34944 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIAMCINOLONE ACETONIDE TRIAMCINOLONE ACETONIDE 51204 34945 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME INSULIN INSULIN 51205 34946 PRLR 5618 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, KINASE agonist 178101594 51206 34947 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ELOMOTECAN HYDROCHLORIDE 51208 34948 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIDANOSINE DIDANOSINE 51209 34949 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR MERCURIC CHLORIDE MERCURIC CHLORIDE 51210 34950 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-107022 CHEMBL1601846 51211 34951 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE carboplatin CARBOPLATIN 31616045 51212 34952 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 405560505 51214 34953 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME activator 178101022 51217 34954 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME CARBAMAZEPINE CARBAMAZEPINE 14977870 51218 34955 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME GSK683699 51220 34956 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL521 IBUPROFEN 51222 34957 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR TCMDC-123723 CHEMBL525103 51223 34958 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME ceftriaxone CEFTRIAXONE 29873816 51224 34959 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME 5-METHYLFURMETHIDE CHEMBL92387 51225 34960 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 6 51226 34961 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE ENMD-1198 51227 34962 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR LXH 254 51229 34963 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-4853 CHEMBL599957 51230 34964 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565621 MILCICLIB 51231 34965 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1201604 TOSITUMOMAB 51233 34966 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ARSENIC TRIOXIDE 16711005 51236 34967 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL allosteric modulator 135651250 51239 34968 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-47c 51241 34969 PDE4A 5141 DRUGGABLE GENOME, ENZYME TADALAFIL TADALAFIL 51243 34970 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor SORAFENIB SORAFENIB 51244 34971 HSD3B7 80270 ENZYME, DRUGGABLE GENOME cholic acid 51245 34972 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME TCMDC-124321 CHEMBL526952 51247 34973 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PKI-179 PKI-179 20797855 51248 34974 HSPA4 3308 NA BORTEZOMIB BORTEZOMIB 16846475 51250 34975 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NRP290 51256 34976 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178100710 51257 34977 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BMS-695735 CHEMBL459729 51258 34978 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER valproic acid 21747585,20417680,18812236 51260 34979 CANX 821 NA MPO MYELOPEROXIDASE 11818449 51261 34980 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MEPRYLCAINE MEPRYLCAINE 51263 34981 PPP2CA 5515 PROTEIN PHOSPHATASE, ENZYME, KINASE LB-100 LB-100 51264 34982 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Carbamide derivative 4 51265 34983 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR EPHEDRINE EPHEDRINE 51266 34984 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ephedrine EPHEDRINE 26771271,25730298 51270 34985 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3545322 PANULISIB 51271 34986 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000200944 CHEMBL600173 51272 34987 SMN2 6607 DRUGGABLE GENOME PIFITHRIN-ALPHA CHEMBL198759 51273 34988 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178103129 51276 34989 THOP1 7064 DRUGGABLE GENOME, PROTEASE Icofungipen ICOFUNGIPEN 51278 34990 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme8NCGC-00185981 51279 34991 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PYRITHIONE PYRITHIONE 51280 34992 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LAPATINIB LAPATINIB 26619011,24516025,25157968,22046346,23220880,16397024,26243863 51281 34993 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist CHEMBL464 ETRETINATE 51282 34994 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME QUINALIZARIN QUINALIZARIN 51283 34995 TMEM97 27346 NA PMID30185082-Compound-55 51284 34996 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME LOMETREXOL LOMETREXOL 20085328 51287 34997 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR THIORIDAZINE THIORIDAZINE 51288 34998 PDE10A 10846 ENZYME, DRUGGABLE GENOME Pyrido[3,2-e][1,2,4]triazolo[4,3-a]pyrazine derivative 1 51289 34999 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 4,4'-DIMETHOXYDALBERGIONE 4,4'-DIMETHOXYDALBERGIONE 51290 35000 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 249565577 FAMITINIB 51291 35001 MTTP 4547 DRUGGABLE GENOME SLx-4090 SLX-4090 51292 35002 ZDHHC7 55625 NA methylphenidate METHYLPHENIDATE 29382897 51293 35003 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1194 PRILOCAINE 51295 35004 GMNN 51053 DRUGGABLE GENOME ACETOMENAPHTHONE ACETOMENAPHTHONE 51296 35005 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME FLUDIAZEPAM FLUDIAZEPAM 51300 35006 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DULOXETINE DULOXETINE 51301 35007 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE STAUROSPORINE STAUROSPORINE 51303 35008 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 404859082 51305 35009 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 51307 35010 KDM4A 9682 DRUGGABLE GENOME, ENZYME PMID27019002-Compound-21b 51309 35011 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650251 FARGLITAZAR 51310 35012 TET2 54790 CLINICALLY ACTIONABLE, ENZYME Decitabine DECITABINE 25224413 51312 35013 BAZ2B 29994 NA GARCINONE E GARCINONE E 51313 35014 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Neratinib NERATINIB 26243863 51315 35015 ATXN2 6311 NA DNDI1417692 CHEMBL1481509 51317 35016 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135649816 CHEMBL64716 51319 35017 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ISOPIMARIC ACID ISOPIMARIC ACID 21793559 51320 35018 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME URIDINE URIDINE 10763851 51321 35019 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL288441 BOSUTINIB 51322 35020 CRY1 1407 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR lithium LITHIUM 51323 35021 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PYRACLOSTROBIN PYRACLOSTROBIN 51325 35022 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL2105719 DACOMITINIB 51326 35023 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME CAPIVASERTIB CAPIVASERTIB 26490311 51328 35024 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CI-1040 CI-1040 51330 35025 TARDBP 23435 TUMOR SUPPRESSOR ISOQUINOLINE-1,3(2H,4H)-DIONE CHEMBL1210769 51331 35026 CADM2 253559 NA ethanol ALCOHOL 32451486 51332 35027 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 252827499 51333 35028 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CHONDROITIN SULFATE 18006074 51336 35029 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL1232583 INDEGLITAZAR 51340 35030 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IDAZOXAN IDAZOXAN 51341 35031 PTK6 5753 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, ENZYME DASATINIB DASATINIB 51342 35032 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-31 51343 35033 MAOB 4129 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 2 51344 35034 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ESTRADIOL ESTRADIOL 51345 35035 ACP1 52 ENZYME, DRUGGABLE GENOME, PROTEIN PHOSPHATASE PYRIMETHAMINE PYRIMETHAMINE 51346 35036 ABHD6 57406 PHOSPHOLIPASE, ENZYME Pyrazole derivative 81 51347 35037 MPHOSPH8 54737 NA FPL-64176 CHEMBL93655 51348 35038 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651359 ZIPRASIDONE 51349 35039 XDH 7498 DRUGGABLE GENOME, ENZYME Fused heterocyclic compound 6 51350 35040 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TOLONIUM CHLORIDE TOLONIUM CHLORIDE 51351 35041 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CAPSAICIN CAPSAICIN 2492344 51352 35042 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545063 OSIMERTINIB MESYLATE 51353 35043 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL3707402 PF-06372865 51354 35044 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 inhibitor 404859006 VOXELOTOR 51355 35045 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR THYROGLOBULIN THYROGLOBULIN 8895887 51356 35046 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MITOTANE MITOTANE 51357 35047 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL blocker 135652058 51358 35048 KEAP1 9817 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING 385612247 51360 35049 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME LATREPIRDINE LATREPIRDINE 51364 35050 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE PAZOPANIB PAZOPANIB 51367 35051 MDH2 4191 NA ANTIOXIDANT 15225672 51368 35052 GNA11 2767 CLINICALLY ACTIONABLE MEK162 BINIMETINIB 24141786,27507190 51369 35053 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ADL7445 51370 35054 GMNN 51053 DRUGGABLE GENOME MECLOFENAMATE SODIUM MECLOFENAMATE SODIUM 51371 35055 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME AZ628 CHEMBL2144069 23398453 51372 35056 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE CEP-11981 CEP-11981 22148921 51374 35057 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME METHYLPHENIDATE METHYLPHENIDATE 10831022 51375 35058 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME AURANOFIN AURANOFIN 51376 35059 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME KAEMPFEROL KAEMPFEROL 51377 35060 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MEPHOBARBITAL MEPHOBARBITAL 51382 35061 IFNGR2 3460 CLINICALLY ACTIONABLE, DRUGGABLE GENOME INTERFERON GAMMA-1B 51385 35062 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME HARMINE HARMINE 22998443 51387 35063 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE KU-0058948 CHEMBL380648 51388 35064 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSAID 16945925 51389 35065 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME SP-600125 SP-600125 51391 35066 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME PMID17935984C1 51392 35067 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE inhibitor CHEMBL269732 TACROLIMUS 51393 35068 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor RIDAFOROLIMUS RIDAFOROLIMUS 51395 35069 GMNN 51053 DRUGGABLE GENOME ETOPOSIDE ETOPOSIDE 51397 35070 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME PMID27998201-Compound-13 51399 35071 LPAR2 9170 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE OCTREOTIDE OCTREOTIDE 18624922 51402 35072 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 363894214 SITRAVATINIB 51403 35073 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR INAMRINONE INAMRINONE 51409 35074 TNC 3371 DRUGGABLE GENOME, FIBRINOGEN F-16-IL-2 fusion protein 51410 35075 CDH3 1001 DRUGGABLE GENOME PF-06671008 PF-06671008 51411 35076 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PSAMMAPLIN A PSAMMAPLIN A 25884112 51412 35077 AMACR 23600 ENZYME ibuprofen IBUPROFEN 25502615 51414 35078 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR US10040779, Example 1 51415 35079 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE GPC3-CART cells 51416 35080 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651302 51417 35081 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 51420 35082 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME activator 135652731 51422 35083 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Neratinib NERATINIB 51423 35084 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-8 51424 35085 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME 178101458 51425 35086 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE (R)-BICALUTAMIDE (R)-BICALUTAMIDE 25121586 51427 35087 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BENZPIPERYLON BENZPIPERYLON 51429 35088 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR ROMIDEPSIN ROMIDEPSIN 51431 35089 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME venetoclax VENETOCLAX 51432 35090 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME cobimetinib COBIMETINIB 22084396 51434 35091 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody 310264712 MM-111 51435 35092 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201167 CARVEDILOL PHOSPHATE 51438 35093 CA2 760 DRUGGABLE GENOME, ENZYME BUTYLATEDHYDROXYTOLUENE 51440 35094 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor CHEMBL197672 EMRICASAN 51443 35095 BTN3A1 11119 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, B30_2 SPRY DOMAIN 340590246 51445 35096 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ARABINOFURANOSYLCYTOSINE 1394224 51446 35097 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL antagonist 135650843 51447 35098 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRETAZICAR TRETAZICAR 51449 35099 HSPB1 3315 DRUGGABLE GENOME RHAMNETIN RHAMNETIN 19296652 51450 35100 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CANERTINIB CANERTINIB 51451 35101 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178101149 51454 35102 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DOVITINIB DOVITINIB 51456 35103 TGFBR2 7048 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME agonist 348353672 51457 35104 NPC1L1 29881 DRUGGABLE GENOME, TRANSPORTER Ezetimibe EZETIMIBE 51459 35105 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker 384403636 51460 35106 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE FGF-6 16617195 51461 35107 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Oxaliplatin OXALIPLATIN 21468686 51462 35108 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor BAY869766 51463 35109 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE CYC-116 CYC-116 20462263 51465 35110 PTGS2 5743 DRUGGABLE GENOME, ENZYME Curcumin CURCUMIN 51466 35111 CD9 928 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE IL-5 10704064 51468 35112 CYB5R2 51700 DRUGGABLE GENOME isosorbide dinitrate 51472 35113 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ENTINOSTAT ENTINOSTAT 20452226,19966789,18381238,20491440,22321215 51473 35114 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NSC-632536 CHEMBL1367933 51474 35115 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BENZO(K)FLUORANTHENE BENZO(K)FLUORANTHENE 51475 35116 COL4A3 1285 KINASE, DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 51476 35117 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL166863 POLMACOXIB 51477 35118 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LY-294002 LY-294002 51478 35119 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651289 51480 35120 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME SITAGLIPTIN SITAGLIPTIN 51481 35121 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178101057 51483 35122 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor XL228 XL-228 51485 35123 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 178103585 ROMIDEPSIN 51486 35124 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE NI-0801 NI-0801 51487 35125 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME inhibitor SELUMETINIB SELUMETINIB 51488 35126 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LAUROGUADINE LAUROGUADINE 51490 35127 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Neratinib NERATINIB 51493 35128 KDM4A 9682 DRUGGABLE GENOME, ENZYME CLIOQUINOL CLIOQUINOL 51494 35129 CARM1 10498 ENZYME, METHYL TRANSFERASE, DRUGGABLE GENOME inhibitor 310264736 51496 35130 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL PHENYTOIN PHENYTOIN 51497 35131 HPD 3242 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1337 NITISINONE 51498 35132 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL activator CHEMBL222460 BMS-223131 51501 35133 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER KETOCONAZOLE KETOCONAZOLE 51502 35134 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER citalopram CITALOPRAM 24192121,18215618,26704739,22641028,21546862 51504 35135 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NITAZOXANIDE NITAZOXANIDE 51505 35136 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE IRINOTECAN IRINOTECAN 25601188 51506 35137 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE ACTINOMYCIN D 10383144 51508 35138 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33b 51509 35139 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME 6-AZAURIDINE 6-AZAURIDINE 51510 35140 GMNN 51053 DRUGGABLE GENOME DNDI1416969 CHEMBL1453126 51512 35141 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Mercaptopurine MERCAPTOPURINE 28151717 51513 35142 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR TAMOXIFEN CITRATE TAMOXIFEN CITRATE 51514 35143 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR 13-CIS-RETINOIC ACID 9815590 51517 35144 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor CHEMBL608533 MIDOSTAURIN 51518 35145 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NSC-119889 CHEMBL516616 51519 35146 PTGS1 5742 ENZYME, DRUGGABLE GENOME TOLMETIN TOLMETIN 51520 35147 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE OSIMERTINIB OSIMERTINIB 31825714,32193290,31254668,24893891,27959700,25923549,26729184,28202511,25939061,26720284 51521 35148 C1S 716 ENZYME, PROTEASE, DRUGGABLE GENOME TS01 51525 35149 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor BIBW2992 CHEMBL2347958 51526 35150 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ETONOGESTREL ETONOGESTREL 51528 35151 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR GM-CSF REGRAMOSTIM 51529 35152 ATXN2 6311 NA FENDILINE HYDROCHLORIDE FENDILINE HYDROCHLORIDE 51530 35153 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DOVITINIB DOVITINIB 51531 35154 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BISPHENOL A BISPHENOL A 51533 35155 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME MINOCYCLINE HYDROCHLORIDE MINOCYCLINE HYDROCHLORIDE 51534 35156 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME BROMAZEPAM BROMAZEPAM 51535 35157 SLC9A3 6550 DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE, EXCHANGER AZD1772//RDX5791 51536 35158 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PLERIXAFOR PLERIXAFOR 51537 35159 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545285 XL-999 51540 35160 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102605 CHEMBL406375 51542 35161 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-107022 CHEMBL1601846 51544 35162 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR GENTIAN VIOLET GENTIAN VIOLET 51545 35163 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME KD-025 CHEMBL2005186 51546 35164 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Altrakincept 51547 35165 YY1 7528 TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR ANTISERUM 10514482 51548 35166 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyrrolo-pyrimidine derivative 10 51549 35167 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TCMDC-123869 CHEMBL546597 51551 35168 ABCB4 5244 TRANSPORTER, DRUGGABLE GENOME, ENZYME, ABC TRANSPORTER anthracyclines and related substances 23441093,21900104 51552 35169 IRAK3 11213 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565893 51554 35170 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE PROPYLTHIOURACIL PROPYLTHIOURACIL 51555 35171 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TAZAROTENE TAZAROTENE 51556 35172 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor PANOBINOSTAT PANOBINOSTAT 51557 35173 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Peg-G-CSF 51558 35174 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 178103589 RICOLINOSTAT 51559 35175 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR ADRIAMYCIN ADRIAMYCIN 10203574 51560 35176 MEG3 55384 NA radiotherapy 51561 35177 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PD-169316 PD-169316 51562 35178 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-4464 CHEMBL600692 51563 35179 PTGS2 5743 DRUGGABLE GENOME, ENZYME CURCUMIN PYRAZOLE CURCUMIN PYRAZOLE 24920381 51564 35180 FAAH 2166 ENZYME, DRUGGABLE GENOME TETRAHYDROCANNABINOL DRONABINOL 16886056 51568 35181 MYO9B 4650 NA FELODIPINE FELODIPINE 2833901 51569 35182 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE L-TRIIODOTHYRONINE 1322573 51571 35183 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER VP-16 ETOPOSIDE PHOSPHATE 7671247 51572 35184 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor REGORAFENIB REGORAFENIB 51573 35185 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Enbrel ENBREL 51574 35186 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SULFADOXINE SULFADOXINE 22931300 51575 35187 BSG 682 DRUGGABLE GENOME, TRANSPORTER Gavilimomab GAVILIMOMAB 51578 35188 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CHLORHEXIDINE CHLORHEXIDINE 51579 35189 ATAD5 79915 NA PIFITHRIN-ALPHA CHEMBL198759 51581 35190 MYLIP 29116 ENZYME atorvastatin ATORVASTATIN 25171759 51582 35191 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3182621 AZD-8330 51583 35192 NDUFA10 4705 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 51584 35193 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL2326966 SF-1126 51585 35194 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE AZD-1152-HQPA AZD-1152-HQPA 51586 35195 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor SNS-314 SNS-314 51587 35196 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL522892 DOVITINIB 51588 35197 POLL 27343 NA HYMENOIC ACID HYMENOIC ACID 18364258 51589 35198 MAP3K11 4296 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL290352 CEP-1347 51591 35199 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PIPERONYL BUTOXIDE PIPERONYL BUTOXIDE 51592 35200 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR CISPLATIN CISPLATIN 16980606,16807441,17229776 51594 35201 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CILOSTAZOL CILOSTAZOL 51595 35202 SMN2 6607 DRUGGABLE GENOME SU-4312 CHEMBL328710 51596 35203 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID28048944-Compound-7 51597 35204 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Anatibant ANATIBANT 51598 35205 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL490665 NALFURAFINE HYDROCHLORIDE 51599 35206 POLD1 5424 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME inhibitor CHEMBL1750 CLOFARABINE 51600 35207 ITPKC 80271 ENZYME, KINASE Immunoglobulins 21987091 51601 35208 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX PERUVOSIDE PERUVOSIDE 51602 35209 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE MITOMYCIN-C 15613449 51603 35210 SF3B3 23450 DRUGGABLE GENOME PLA D PLA D 17643112 51604 35211 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Macrolactam derivative 1 51605 35212 USP1 7398 DNA REPAIR, PROTEASE, ENZYME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 51610 35213 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1743054 OZORALIZUMAB 51613 35214 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DESOXYCORTICOSTERONE ACETATE DESOXYCORTICOSTERONE ACETATE 51614 35215 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TPCK TPCK 51616 35216 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor 178103127 51617 35217 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-7 51621 35218 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYPROTERONE CYPROTERONE 51622 35219 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME PROTOPORPHYRIN DISODIUM PROTOPORPHYRIN DISODIUM 51623 35220 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CLADRIBINE CLADRIBINE 51624 35221 DGAT1 8694 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2364624 PRADIGASTAT 51625 35222 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MEM 1003 51626 35223 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE BMS-777607 BMS-777607 51627 35224 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545300 CP-459632 51628 35225 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1237065 TRAMADOL HYDROCHLORIDE 51629 35226 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ARG098 51633 35227 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE rucaparib RUCAPARIB 51634 35228 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650156 DADLE 51635 35229 ARAP2 116984 NA Tumor necrosis factor alpha (TNF-alpha) inhibitors 51636 35230 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER VOACAMINE VOACAMINE 24720452 51637 35231 TGFA 7039 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME cetuximab CETUXIMAB 51638 35232 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE V934/V935 51639 35233 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE activator CHEMBL2109084 DESMOTEPLASE 51641 35234 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE metabutethamine METABUTETHAMINE 51642 35235 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER WIN-62577 CHEMBL1256845 51643 35236 APRT 353 ENZYME, DRUGGABLE GENOME HYDROGEN PEROXIDE 10213488 51644 35237 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL3545035 REVEXEPRIDE 51645 35238 CA2 760 DRUGGABLE GENOME, ENZYME TOPIRAMATE TOPIRAMATE 51646 35239 POLK 51426 DNA REPAIR, ENZYME NSC-107022 CHEMBL1601846 51647 35240 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545248 DS-7423 51649 35241 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor CHEMBL2364611 GALUNISERTIB 51650 35242 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1628502 GABAPENTIN ENACARBIL 51651 35243 ATXN2 6311 NA SB-242084 SB-242084 51653 35244 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 gliclazide GLICLAZIDE 24442125 51654 35245 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 340590266 GDC-0077 51655 35246 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 135651721 51656 35247 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650806 51657 35248 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Crizotinib CRIZOTINIB 51659 35249 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIPYRIDYL DIPYRIDYL 51660 35250 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME HOE-33342 CHEMBL343002 51661 35251 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KD3010 KD3010 51662 35252 APC 324 CLINICALLY ACTIONABLE MF tricyclic 23843721 51663 35253 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CETUXIMAB CETUXIMAB 22199315 51664 35254 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE CHEMBL2010601 IVACAFTOR 51665 35255 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Sapanisertib SAPANISERTIB 25261369 51666 35256 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200602 51667 35257 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME PMID28270021-Compound-WO2015042088Example4 51668 35258 RACGAP1 29127 NA GNF-PF-3996 CHEMBL584458 51669 35259 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-47 51670 35260 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MGCD265 GLESATINIB 51671 35261 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR PALBOCICLIB PALBOCICLIB 51674 35262 HDAC11 79885 DRUGGABLE GENOME, ENZYME SUBEROHYDROXAMIC ACID SUBEROHYDROXAMIC ACID 16921367 51675 35263 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME PESUDOGINSENOSIDE RP1 METHYL ESTER PESUDOGINSENOSIDE RP1 METHYL ESTER 20951582 51677 35264 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE ANTITHYMOCYTE GLOBULIN 51678 35265 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PMID27774824-Compound-Figure2Example4 51679 35266 PBK 55872 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, ENZYME SP-600125 SP-600125 51680 35267 SLC25A4 291 DRUGGABLE GENOME, TRANSPORTER inhibitor 178101293 51681 35268 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Cyclopentane carboxamide derivative 1 51683 35269 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL3545252 DOCETAXEL 51686 35270 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME 4-IPOMEANOL CHEMBL1743358 1976855 51687 35271 SIRT5 23408 ENZYME CEFIXIME CEFIXIME 51688 35272 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE TOZASERTIB TOZASERTIB 51689 35273 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135649650 51690 35274 DDB1 1642 DNA REPAIR inhibitor CHEMBL468 THALIDOMIDE 51691 35275 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Isoquinoline sulfonamide derivative 2 51693 35276 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Arformoterol ARFORMOTEROL 51698 35277 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Quinazoline derivative 1 51699 35278 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 51700 35279 EPHA3 2042 ENZYME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody 310264706 51701 35280 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Nivolumab NIVOLUMAB 51702 35281 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Serdemetan SERDEMETAN 21831953 51703 35282 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME DNDI1417156 CHEMBL1504679 51705 35283 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Sunitinib SUNITINIB 19164557,19861435,25594040,18955458,25239608,23582185,26772734 51706 35284 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103981 ILOMASTAT 51707 35285 TUBA3D 113457 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 51711 35286 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AFATINIB AFATINIB 24685132 51713 35287 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL Nitrendipine NITRENDIPINE 51714 35288 PSMB4 5692 DRUGGABLE GENOME, PROTEASE inhibitor BORTEZOMIB BORTEZOMIB 51716 35289 MAPT 4137 DRUGGABLE GENOME NSC-66209 CHEMBL175266 51717 35290 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-11 51719 35291 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHOLECALCIFEROL CHOLECALCIFEROL 51720 35292 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 187051755 51722 35293 POLK 51426 DNA REPAIR, ENZYME 5,7,3',5'-TETRAHYDROXYFLAVANONE CHEMBL307893 51723 35294 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER ABACAVIR ABACAVIR 17172311 51724 35295 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135650657 51725 35296 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PYRILAMINE PYRILAMINE 22931300 51726 35297 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3702 CHEMBL598268 51727 35298 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE STREPTOKINASE STREPTOKINASE 51729 35299 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Piroxicam PIROXICAM 51730 35300 ITPR1 3708 ION CHANNEL, KINASE, DRUGGABLE GENOME, TRANSPORTER activator 178101040 51731 35301 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE NERVIANO NERVIANO 20621725 51732 35302 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-732881 CHEMBL261129 51733 35303 SERPINA5 5104 PROTEASE INHIBITOR, ENZYME, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE carboplatin CARBOPLATIN 31616045 51734 35304 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AU105 51735 35305 NQO2 4835 DRUGGABLE GENOME, ENZYME IMATINIB IMATINIB 22494098 51736 35306 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Goserelin GOSERELIN 51737 35307 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-1134 CHEMBL600694 51738 35308 RGS16 6004 NA s2901 51739 35309 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR CYC-116 CYC-116 51741 35310 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 404859142 51742 35311 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE carbamazepine CARBAMAZEPINE 12083967 51743 35312 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR BECLOMETHASONE DIPROPIONATE 51744 35313 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ERGOCALCIFEROL ERGOCALCIFEROL 51746 35314 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE MEMANTINE MEMANTINE 51748 35315 ENTPD2 954 ENZYME inhibitor 315661118 CHEMBL469212 51749 35316 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SGX523 51750 35317 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ADRIAMYCIN ADRIAMYCIN 2897875 51751 35318 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME RESMINOSTAT RESMINOSTAT 51752 35319 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Amidopyrazole derivative 4 51753 35320 HP 3240 DRUGGABLE GENOME, PROTEASE, ENZYME STREPTOZOTOCIN STREPTOZOCIN 16713232 51754 35321 BAZ2B 29994 NA TCMDC-124544 CHEMBL531322 51755 35322 COL18A1 80781 DRUGGABLE GENOME HEPARAN SULFATE 14585835 51756 35323 PDE10A 10846 ENZYME, DRUGGABLE GENOME inhibitor 252827416 51758 35324 HNMT 3176 ENZYME, DRUGGABLE GENOME Diphenhydramine DIPHENHYDRAMINE 51760 35325 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200617 RIMEXOLONE 51761 35326 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME TEMAZEPAM TEMAZEPAM 51763 35327 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE salbutamol ALBUTEROL 23126384,29053759,15500895,19800676,24279851,18156033 51764 35328 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Tamoxifen TAMOXIFEN 51765 35329 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL1094 FELBAMATE 51767 35330 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SALINE SODIUM CHLORIDE 9603077 51769 35331 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME PD-98059 CHEMBL35482 51771 35332 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201640 INSULIN ZINC SUSP EXTENDED BEEF 51772 35333 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL460702 BMS-777607 51773 35334 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE TOZASERTIB TOZASERTIB 51774 35335 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 51776 35336 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME VALDECOXIB VALDECOXIB 16707021 51778 35337 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CHLORPYRIFOS CHLORPYRIFOS 51779 35338 TCN1 6947 DRUGGABLE GENOME CYANOCOBALAMIN CYANOCOBALAMIN 2876185 51781 35339 PTGS2 5743 DRUGGABLE GENOME, ENZYME MESALAMINE MESALAMINE 51782 35340 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX OSAJIN OSAJIN 51783 35341 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3545420 AG-24322 51788 35342 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR capecitabine CAPECITABINE 25026457 51789 35343 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200715 HEXYLCAINE HYDROCHLORIDE 51790 35344 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 310264733 FIMEPINOSTAT 51791 35345 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SNS-314 SNS-314 51792 35346 ATAD5 79915 NA RESERPINE RESERPINE 51795 35347 TUBB2B 347733 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 51799 35348 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SU-6656 CHEMBL605003 51800 35349 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CALOTHRIXIN A CALOTHRIXIN A 19203291 51802 35350 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FERBAM FERBAM 51803 35351 SLC22A3 6581 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER ANTIDEPRESSANT DRUGS 15121658 51804 35352 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR THIOPERAMIDE THIOPERAMIDE 19053770,20192225 51805 35353 SLPI 6590 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR CYTOKINES 11385113 51806 35354 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor CHEMBL1046 AMINOCAPROIC ACID 51809 35355 RGS4 5999 DRUGGABLE GENOME DEQUALINIUM DEQUALINIUM 51810 35356 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR XL418 XL-418 51811 35357 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR methadone METHADONE 23651024 51813 35358 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL12 DIAZEPAM 51814 35359 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER GNF-PF-1731 CHEMBL581251 51815 35360 DHODH 1723 DRUGGABLE GENOME, ENZYME Teriflunomide TERIFLUNOMIDE 51818 35361 SLC36A1 206358 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 135651515 TRYPTOPHAN 51819 35362 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DOPAMINE HYDROCHLORIDE DOPAMINE HYDROCHLORIDE 51821 35363 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME LORAZEPAM LORAZEPAM 51824 35364 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1201729 DRONEDARONE HYDROCHLORIDE 51825 35365 PSMD12 5718 NA inhibitor CHEMBL325041 BORTEZOMIB 51826 35366 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR inhibitor CHEMBL2108431 METELIMUMAB 51827 35367 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHOXYCHLOR METHOXYCHLOR 51829 35368 KDM4A 9682 DRUGGABLE GENOME, ENZYME LAVENDUSTIN C LAVENDUSTIN C 51830 35369 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUTICASONE FLUTICASONE 51832 35370 ANGPT1 284 KINASE, DRUGGABLE GENOME, FIBRINOGEN AMG 386 51833 35371 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8889696, Staurosporine 51834 35372 BAP1 8314 PROTEASE, TUMOR SUPPRESSOR, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE EVEROLIMUS EVEROLIMUS 27751729 51837 35373 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL220492 TOPIRAMATE 51839 35374 NOS2 4843 DRUGGABLE GENOME, ENZYME ECG 12081242 51843 35375 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR WEDELOLACTONE WEDELOLACTONE 22926226 51844 35376 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 328083472 51845 35377 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME bilirubin BILIRUBIN 21813404,10353933,20693308,22805420,17000907,7565971,20562445,12816916,10836148,9630669,18518849,10190918,10748067,15712364,9765507,10091406,4897277,11929814,11401924,15111762,16609363,3306242,19830808,12386134,15179405,9784835,17898154,17949292,12181419,8027054,22559977,1898728,10706110,12891498,11013440,15986396 51850 35378 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MB07811 MB07811 51853 35379 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TRAVOPROST TRAVOPROST 51854 35380 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME GIVINOSTAT GIVINOSTAT 51856 35381 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE GSK269962A 51857 35382 TAT 6898 ENZYME URIDINE URIDINE 6161802 51858 35383 TUBB 203068 DRUGGABLE GENOME Albendazole ALBENDAZOLE 51859 35384 ARSA 410 DRUGGABLE GENOME, ENZYME NBQX NBQX 51860 35385 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR GEMCITABINE GEMCITABINE 16980606,17229776 51862 35386 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR PLATINUM PLATINUM 8996528 51863 35387 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME NN5401 51864 35388 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PMID25416646-Compound-Figure5-C 51865 35389 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME PROTEASE INHIBITORS 12554354 51867 35390 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178100513 SUFENTANIL 51868 35391 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME (S)-MAP4 HCL CHEMBL1256510 51869 35392 POLK 51426 DNA REPAIR, ENZYME LAVENDUSTIN A LAVENDUSTIN A 51870 35393 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CEFUROXIME SODIUM CEFUROXIME SODIUM 51871 35394 POLA2 23649 NA DACARBAZINE DACARBAZINE 51873 35395 ACLY 47 ENZYME, DRUGGABLE GENOME GLUCAGON GLUCAGON 489538 51874 35396 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor BAY80-6946 COPANLISIB 51875 35397 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR BETAMETHASONE BETAMETHASONE 51877 35398 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME APICIDIN APICIDIN 19705846,17956988 51879 35399 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 10 51880 35400 MAPT 4137 DRUGGABLE GENOME LAVENDUSTIN A LAVENDUSTIN A 51881 35401 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME AZD-1080 AZD-1080 51883 35402 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 315661272 ZYKLOPHIN 51884 35403 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME FTI 16818651 51885 35404 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE GONIOTHALAMIN GONIOTHALAMIN 25305718 51886 35405 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER inhibitor BORTEZOMIB BORTEZOMIB 51887 35406 FANCD2 2177 CLINICALLY ACTIONABLE DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 23026082 51889 35407 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE Buparlisib BUPARLISIB 51890 35408 HMBS 3145 ENZYME givosiran GIVOSIRAN 51891 35409 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME 2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE CHEMBL412603 51892 35410 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Trastuzumab TRASTUZUMAB 27626067 51894 35411 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652502 51895 35412 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102573 51896 35413 ABCB4 5244 TRANSPORTER, DRUGGABLE GENOME, ENZYME, ABC TRANSPORTER Benzquinamide BENZQUINAMIDE 51897 35414 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-26 51901 35415 BMPR2 659 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, CELL SURFACE inhibitor 249565835 51902 35416 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME YSCMA 51904 35417 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME ANTHRACYCLINES 8069262 51906 35418 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER Tetrabenazine TETRABENAZINE 51907 35419 CGA 1081 DRUGGABLE GENOME, HORMONE ACTIVITY 9-CIS-RETINOIC ACID 8070357 51911 35420 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 328083473 CHEMBL1951415 51912 35421 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8921389, 1 51913 35422 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 178103353 51914 35423 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME activator 53801065 NIFEDIPINE 51915 35424 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISOFLAVONES 16380645 51916 35425 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TAK-285 TAK-285 25594012,18441328,23983820 51917 35426 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IPRONIAZID SULFATE IPRONIAZID SULFATE 51918 35427 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE tolazamide TOLAZAMIDE 51920 35428 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THIRAM THIRAM 51922 35429 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SENNOSIDE B SENNOSIDE B 51923 35430 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME DENILEUKIN DIFTITOX 51926 35431 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MONOBENZONE MONOBENZONE 51927 35432 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER rivaroxaban RIVAROXABAN 27893182 51928 35433 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NELFINAVIR MESYLATE NELFINAVIR MESYLATE 51930 35434 PSMD11 5717 KINASE inhibitor BORTEZOMIB BORTEZOMIB 51933 35435 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME agonist CHEMBL1963684 PEGINESATIDE ACETATE 51934 35436 CST3 1471 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR RIBAVIRIN RIBAVIRIN 18637076 51935 35437 RACGAP1 29127 NA PHENIDONE PHENIDONE 51938 35438 SMARCB1 6598 CLINICALLY ACTIONABLE TAZEMETOSTAT TAZEMETOSTAT 29650362,23620515 51939 35439 MARCHF8 220972 ENZYME CAF-01 23720661 51941 35440 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 51943 35441 ALOX15B 247 DRUGGABLE GENOME, ENZYME SANGUINARIUM SANGUINARIUM 51944 35442 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 385612197 51945 35443 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TALAZOPARIB TALAZOPARIB 31852834 51946 35444 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor 178103626 ZONISAMIDE 51948 35445 CP 1356 DRUGGABLE GENOME, ENZYME ISOPROTERENOL ISOPROTERENOL 12557918 51949 35446 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor POZIOTINIB POZIOTINIB 51951 35447 KDM4A 9682 DRUGGABLE GENOME, ENZYME L-NOREPINEPHRINE L-NOREPINEPHRINE 51953 35448 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME NVP-AEW541 AEW-541 26577700 51954 35449 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AZAMETHIPHOS AZAMETHIPHOS 51955 35450 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545361 ROGARATINIB 51957 35451 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 diclofenac DICLOFENAC 23959274,25994031,23400009,20814155,8417277,17681167 51958 35452 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PIOGLITAZONE HYDROCHLORIDE PIOGLITAZONE HYDROCHLORIDE 51960 35453 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 354702263 51961 35454 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ETONOGESTREL ETONOGESTREL 51962 35455 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE lopinavir LOPINAVIR 22027652,19842932,26287941 51963 35456 MAOB 4129 DRUGGABLE GENOME, ENZYME Safinamide SAFINAMIDE 51964 35457 SLC28A2 9153 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME protease inhibitors 26071337 51965 35458 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE 11C-6-Me-BTA-1 51966 35459 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR APIGENIN APIGENIN 51967 35460 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME VORINOSTAT VORINOSTAT 51968 35461 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE ABBV-2222 GALICAFTOR 51970 35462 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HYDROCORTISONE VALERATE HYDROCORTISONE VALERATE 51972 35463 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor GIVINOSTAT GIVINOSTAT 51973 35464 IL17RA 23765 DRUGGABLE GENOME antibody 187051841 BRODALUMAB 51974 35465 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME CAMBINOL CAMBINOL 51978 35466 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL 9-CIS-RETINOIC ACID 18404486 51980 35467 NEK4 6787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 51981 35468 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER NICOTINE NICOTINE 16191663 51982 35469 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GEFITINIB GEFITINIB 16818711 51983 35470 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GW441756X GW441756X 51984 35471 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 5,7-DIMETHOXYISOFLAVONE 5,7-DIMETHOXYISOFLAVONE 51985 35472 BAZ2B 29994 NA NSC-107022 CHEMBL1601846 51986 35473 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 51987 35474 PTGS2 5743 DRUGGABLE GENOME, ENZYME PIROXICAM PIROXICAM 51988 35475 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CF102 NAMODENOSON 51990 35476 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CHEMBL1102 GLUTETHIMIDE 51992 35477 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DICYCLOMINE DICYCLOMINE 51993 35478 PDE3A 5139 ENZYME, DRUGGABLE GENOME THEOPHYLLINE THEOPHYLLINE 51996 35479 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CH5132799 PA-799 25231405,21558396 51998 35480 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME ABT-263 NAVITOCLAX 27659046 51999 35481 CPA6 57094 DRUGGABLE GENOME, PROTEASE, ENZYME metformin METFORMIN 29650774 52000 35482 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE LINIFANIB LINIFANIB 52002 35483 POLI 11201 DNA REPAIR DNDI1417614 CHEMBL1567571 52003 35484 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Velimogene aliplasmid 52004 35485 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417400 CHEMBL1362503 52005 35486 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME OXAPIUM OXAPIUM 52007 35487 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor BMS-690514 BMS-690514 52008 35488 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME inhibitor 178103583 52011 35489 IL1B 3553 KINASE, DRUGGABLE GENOME Canakinumab CANAKINUMAB 52013 35490 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist CHEMBL75133 IRX-4204 52015 35491 RORA 6095 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE agonist 178100434 52016 35492 ALDH1A1 216 DRUGGABLE GENOME, ENZYME EPHEDRINE SULFATE EPHEDRINE SULFATE 52017 35493 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3545366 VOXTALISIB 52019 35494 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MM-111 MM-111 52020 35495 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME O6-[3-(AMINOMETHYL)BENZYL]GUANINE CHEMBL485756 22932317,18973327 52021 35496 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor GEFITINIB GEFITINIB 52023 35497 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2205230 TAK-441 52024 35498 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GEMCITABINE GEMCITABINE 24915778,21862683 52025 35499 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PKI-587 GEDATOLISIB 52026 35500 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AFLOQUALONE AFLOQUALONE 52027 35501 PTGES 9536 DRUGGABLE GENOME, ENZYME TNF-ALPHA 12130559 52028 35502 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CID 667285 CHEMBL267160 52030 35503 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR GNF-PF-2301 CHEMBL578061 52032 35504 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME TG-100435 CHEMBL230686 17113292 52033 35505 ALOX5 240 DRUGGABLE GENOME, ENZYME MK-866 12967948 52035 35506 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ARRY-614 PEXMETINIB 52037 35507 ALB 213 TRANSPORTER, DRUGGABLE GENOME AMODIAQUINE HYDROCHLORIDE AMODIAQUINE HYDROCHLORIDE 22658498 52040 35508 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor TRAMETINIB TRAMETINIB 52041 35509 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Vitamin A 52043 35510 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565590 CHEMBL1236539 52044 35511 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME ANTISENSE OLIGONUCLEOTIDES 10843995 52045 35512 PTGS2 5743 DRUGGABLE GENOME, ENZYME ROFECOXIB ROFECOXIB 52047 35513 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PERHEXILINE PERHEXILINE 22931300 52048 35514 XPO1 7514 CLINICALLY ACTIONABLE, KINASE KPT-330 SELINEXOR 24631834 52049 35515 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 249565599 52053 35516 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME TCMDC-125758 CHEMBL546797 52055 35517 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME GNF-PF-3352 CHEMBL600306 52057 35518 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-METHOXYPHENAZINE CHEMBL1420181 52058 35519 SCD 6319 DRUGGABLE GENOME, ENZYME Isoxyl 52059 35520 BCHE 590 DRUGGABLE GENOME, ENZYME JES-9501 52060 35521 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GALLIC ACID GALLIC ACID 52061 35522 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-17 52062 35523 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 5-FLUOROURACIL FLUOROURACIL 12845662 52063 35524 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE SORAFENIB SORAFENIB 52064 35525 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME dabrafenib DABRAFENIB 52066 35526 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135651244 TERBUTALINE 52068 35527 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MLN-8054 MLN-8054 52069 35528 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CHLOROTRIANISENE CHLOROTRIANISENE 52070 35529 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE M2698 MSC-2363318A 52072 35530 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PD-325901 52073 35531 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CZ-48 52074 35532 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE RX-0201 ARCHEXIN 52075 35533 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME CYCLIC CRYPEVEIC CYCLIC CRYPEVEIC 21545152 52076 35534 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE GW441756X GW441756X 52077 35535 SMN1 6606 DRUGGABLE GENOME VALPROIC ACID 14595654 52078 35536 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MRS-2179 CHEMBL129841 52079 35537 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CPUY201112 26743233 52080 35538 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME METHOTREXATE METHOTREXATE 52081 35539 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SB-242235 SB-242235 52084 35540 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL846 CALCITRIOL 52090 35541 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME TIDEGLUSIB TIDEGLUSIB 52091 35542 CCL5 6352 CELL SURFACE, ENZYME, KINASE, DRUGGABLE GENOME FLUTICASONE PROPIONATE 14556981 52092 35543 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ADINAZOLAM ADINAZOLAM 52093 35544 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 348353623 52094 35545 XRCC4 7518 KINASE fluorouracil FLUOROURACIL 28796378 52095 35546 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR CORTICOSTEROIDS 17013807 52096 35547 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR QAW-039 FEVIPIPRANT 52097 35548 DGAT1 8694 ENZYME, DRUGGABLE GENOME PMID25470667-Compound-BAY744113 52098 35549 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE IMATINIB IMATINIB 18191450 52099 35550 PSMD6 9861 NA inhibitor BORTEZOMIB BORTEZOMIB 52100 35551 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME DICUMAROL DICUMAROL 9343371 52102 35552 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME HALAZEPAM HALAZEPAM 52106 35553 TLK2 11011 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME GF109203X 27694828 52107 35554 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR interferons 27139837 52108 35555 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist,antagonist 135650190 52109 35556 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL981 FENOFIBRIC ACID 52110 35557 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Alitretinoin ALITRETINOIN 52111 35558 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME HUMAN CHORIONIC GONADOTROPIN 9764349,15388676 52112 35559 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ISOXABEN ISOXABEN 52114 35560 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ANTITHYMOCYTE GLOBULIN 52115 35561 IFNGR1 3459 DRUGGABLE GENOME, CLINICALLY ACTIONABLE IFN-GAMMA INTERFERON GAMMA-1B 52116 35562 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AC0010MA ABIVERTINIB MALEATE 27573423 52119 35563 PTGS2 5743 DRUGGABLE GENOME, ENZYME Valdecoxib VALDECOXIB 52122 35564 PRMT6 55170 ENZYME, METHYL TRANSFERASE inhibitor 336446915 52124 35565 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Ace Inhibitors, Plain 23407050,18347611 52125 35566 FDFT1 2222 DRUGGABLE GENOME, ENZYME LOVASTATIN LOVASTATIN 7685352 52126 35567 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME VALPROIC ACID 6138013 52127 35568 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DESOXIMETASONE DESOXIMETASONE 52128 35569 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER PILOCARPINE PILOCARPINE 15860570 52129 35570 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102588 52130 35571 GZMA 3001 PROTEASE, DRUGGABLE GENOME, ENZYME ANTIVIRAL 12820184 52132 35572 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING SERGEOLIDE SERGEOLIDE 19199792 52133 35573 PSCA 8000 DRUGGABLE GENOME BPX-601 52134 35574 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME SLV-334 SLV-334 52135 35575 KDM4A 9682 DRUGGABLE GENOME, ENZYME FLUSPIRILENE FLUSPIRILENE 52136 35576 PDE4D 5144 DRUGGABLE GENOME, ENZYME DYPHYLLINE DYPHYLLINE 52137 35577 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL14762 SELICICLIB 52138 35578 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000044417 CHEMBL609438 52139 35579 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 252166521 DECERNOTINIB 52140 35580 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1021 NEPAFENAC 52141 35581 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051817 52143 35582 CA9 768 DRUGGABLE GENOME, ENZYME Girentuximab I-124 52144 35583 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE ceftriaxone CEFTRIAXONE 29873816 52145 35584 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME Sodium bicarbonate 52147 35585 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE BAN2401 BAN2401 52148 35586 KDM4A 9682 DRUGGABLE GENOME, ENZYME OMEPRAZOLE MAGNESIUM OMEPRAZOLE MAGNESIUM 52149 35587 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AM-251 CHEMBL285932 52150 35588 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME ibuprofen IBUPROFEN 26122864,18216720,15289789,25502615,30562214,18694831,19480553 52152 35589 TLR7 51284 DRUGGABLE GENOME CPG 52364 52154 35590 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE BLEOMYCIN BLEOMYCIN 14559807 52156 35591 ZEB1 6935 TRANSCRIPTION FACTOR, DRUG RESISTANCE OXALIPLATIN OXALIPLATIN 29151941 52157 35592 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Aryl carboxamide derivative 1 52158 35593 CA2 760 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL166863 POLMACOXIB 52159 35594 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME GNF-PF-4328 CHEMBL597452 52160 35595 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER LY333531 52161 35596 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE ENTRECTINIB ENTRECTINIB 52162 35597 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1534525 MIBEFRADIL DIHYDROCHLORIDE 52163 35598 MAPT 4137 DRUGGABLE GENOME CYSTEAMINE HYDROCHLORIDE CYSTEAMINE HYDROCHLORIDE 52164 35599 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME CANERTINIB CANERTINIB 52165 35600 MAOA 4128 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 1 52166 35601 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor DANUSERTIB DANUSERTIB 52167 35602 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE PHA-767491 CHEMBL225519 52168 35603 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649901 52170 35604 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE PENTACHLOROPHENOL PENTACHLOROPHENOL 52172 35605 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 249565687 52173 35606 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ANGUSTIBALIN ANGUSTIBALIN 52174 35607 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200382 BEPRIDIL HYDROCHLORIDE 52175 35608 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 3 52177 35609 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR DICHLOROPHEN DICHLOROPHEN 52179 35610 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME BITHIONOL BITHIONOL 52181 35611 APCS 325 TRANSPORTER, DRUGGABLE GENOME CPHPC MIRIDESAP 52182 35612 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 315661262 52184 35613 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 7-NITROINDAZOLE 7-NITROINDAZOLE 52185 35614 HTT 3064 DRUGGABLE GENOME ISOVELLERAL ISOVELLERAL 52187 35615 CLK3 1198 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 249565735 52191 35616 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 4 52192 35617 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PDGF-BB 52194 35618 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE ALPHA-NAPHTHOFLAVONE ALPHA-NAPHTHOFLAVONE 23600958 52195 35619 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL3545019 MBX-8025 52196 35620 BRD7 29117 ENZYME inhibitor 336446908 52198 35621 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 sorafenib SORAFENIB 28362716 52199 35622 ATP2C1 27032 ENZYME, TRANSPORTER, DRUGGABLE GENOME DESFLURANE DESFLURANE 52200 35623 POLK 51426 DNA REPAIR, ENZYME CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 52201 35624 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE CEDIRANIB CEDIRANIB 52202 35625 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1256958 EPINEPHRINE BITARTRATE 52203 35626 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME THIETHYLPERAZINE THIETHYLPERAZINE 52206 35627 TUBB6 84617 DRUGGABLE GENOME ABT-751 ABT-751 25468039 52207 35628 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME GMI-1359 52208 35629 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200635 HYDROCORTAMATE HYDROCHLORIDE 52209 35630 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUOROMETHOLONE FLUOROMETHOLONE 52211 35631 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR AZD9496 AZD-9496 52212 35632 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE FRUQUINTINIB FRUQUINTINIB 52217 35633 KMO 8564 DRUGGABLE GENOME, ENZYME Cyclopropane 1-carboxylic acid derivative 5 52218 35634 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE TRANEXAMIC ACID 52220 35635 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME BI-836880 52221 35636 PRDX1 5052 ENZYME HYDROGEN PEROXIDE 14765133 52222 35637 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-3641 CHEMBL599098 52224 35638 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME imatinib IMATINIB 21633340 52225 35639 USP1 7398 DNA REPAIR, PROTEASE, ENZYME 3,4-DICHLOROISOCOUMARIN CHEMBL24983 52226 35640 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650020 52227 35641 ATAD5 79915 NA TCMDC-125756 CHEMBL536599 52229 35642 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Regorafenib REGORAFENIB 23629727,25838391 52230 35643 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE ILORASERTIB ILORASERTIB 52231 35644 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CATECHOL CATECHOL 52232 35645 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CATECHOL CATECHOL 52233 35646 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1201109 DESONIDE 52236 35647 FGFRL1 53834 KINASE, DRUGGABLE GENOME brivanib BRIVANIB 20124951 52237 35648 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor CHEMBL3545425 BAY-1161909 52239 35649 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME METFORMIN HYDROCHLORIDE METFORMIN HYDROCHLORIDE 23490148 52241 35650 ARNT 405 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TCDD 9787404,11026553,9579024,14687977 52243 35651 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-27 52244 35652 CFL1 1072 KINASE FENOFIBRATE FENOFIBRATE 16680159 52245 35653 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HEXYLRESORCINOL HEXYLRESORCINOL 52246 35654 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL inhibitor 381118871 52249 35655 SGMS2 166929 KINASE, ENZYME inhibitor 252827491 52252 35656 CXCL8 3576 DRUGGABLE GENOME ABX-IL8 ABX-IL8 52253 35657 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE HARMINE HARMINE 22998443 52255 35658 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX PMID27336223-Compound-13 52256 35659 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME HELIOMYCIN HELIOMYCIN 52259 35660 NOS1 4842 DRUGGABLE GENOME, ENZYME ANTIBIOTICS 14730107 52260 35661 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NONYL 4-HYDROXYBENZOATE NONYL 4-HYDROXYBENZOATE 52265 35662 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051825 52266 35663 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME MSX-122 MSX-122 52267 35664 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SYL040012 BAMOSIRAN 52270 35665 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651539 DINOPROSTONE 52271 35666 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE METHIMAZOLE METHIMAZOLE 52272 35667 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-5052 CHEMBL601367 52275 35668 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor 178103722 CHLORTHALIDONE 52276 35669 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME PHYSODIC ACID PHYSODIC ACID 52277 35670 HTT 3064 DRUGGABLE GENOME ANGUIDIN ANGUIDIN 52278 35671 RAC2 5880 NA doxorubicin DOXORUBICIN 21048526 52279 35672 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 328083472 52281 35673 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MVAp53 52282 35674 HLA-DQA1 3117 CLINICALLY ACTIONABLE interferon beta-1a 21502966 52284 35675 SCTR 6344 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Secretin SECRETIN 52287 35676 PSMA5 5686 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL451887 CARFILZOMIB 52288 35677 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor CHEMBL2109540 ALIROCUMAB 52291 35678 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE OXOGLAUCINE OXOGLAUCINE 52294 35679 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME inhibitor 178103441 OXIGLUTATIONE 52295 35680 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME VBY-129 52297 35681 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IIIA AESCULIOSIDE IIIA 20371180 52298 35682 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DIFFERENTIATION AGENTS 10921005 52299 35683 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545117 AVE-9940 52300 35684 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME EPIRUBICIN EPIRUBICIN 52301 35685 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Icotinib hydrochloride 52302 35686 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Re-188-P-2045 52303 35687 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-39 52306 35688 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-19 52308 35689 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR SOTRASTAURIN SOTRASTAURIN 52309 35690 PDE7B 27115 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200875 FLAVOXATE HYDROCHLORIDE 52310 35691 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL1645462 AC-480 52311 35692 CCL21 6366 DRUGGABLE GENOME CHEMOKINES 11286540,11163192,10496316,12209625,14707047,15919372,11929789,10790423,15358618,10925282,12580544 52312 35693 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME CGS-15943 CGS-15943 52313 35694 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CYSTAMINE CYSTAMINE 52316 35695 CD47 961 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Hu5F9-G4 MAGROLIMAB 52317 35696 LCAT 3931 ENZYME, TRANSPORTER, DRUGGABLE GENOME STREPTOZOTOCIN STREPTOZOCIN 18436977 52318 35697 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TROGLITAZONE TROGLITAZONE 11344222 52319 35698 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 381118807 52320 35699 PPA2 27068 ENZYME risperidone RISPERIDONE 52321 35700 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZINC 02058890 CHEMBL1738936 22047606 52322 35701 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Imatinib IMATINIB 52323 35702 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR TAE-684 TAE-684 52324 35703 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103004 RIVAROXABAN 52326 35704 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME Intravenous glibenclamide 52327 35705 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE Ivacaftor IVACAFTOR 52328 35706 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NIALAMIDE NIALAMIDE 52329 35707 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR 4-(4-AMINOPHENYL)BUTANOIC ACID CHEMBL1650245 24044874 52331 35708 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE WARFARIN WARFARIN 14723717 52332 35709 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Adenosine ADENOSINE 52333 35710 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE FENOFIBRATE FENOFIBRATE 12606523 52335 35711 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR MELATONIN MELATONIN 9649124 52339 35712 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Vistusertib VISTUSERTIB 25805799 52340 35713 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE WIN-55212-2 WIN-552122 52341 35714 HSP90B1 7184 DRUGGABLE GENOME inhibitor 381118828 52342 35715 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE SAPONIN 11090099 52344 35716 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-62 52345 35717 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE PMID29130358-Compound-SB-3CT 52346 35718 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CRIZOTINIB CRIZOTINIB 21791641 52347 35719 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE GW843682X GW843682X 52348 35720 CALR 811 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PEGINTERFERON ALFA-2A 26486786 52349 35721 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2096642 INAMRINONE LACTATE 52350 35722 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR MART1 15665624 52351 35723 APC 324 CLINICALLY ACTIONABLE CCT070535 20610623 52354 35724 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor CHEMBL98 VORINOSTAT 52355 35725 CXCL8 3576 DRUGGABLE GENOME MEDROXYPROGESTERONE ACETATE 15914533 52356 35726 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR TRP-2 15603192 52357 35727 KDM4A 9682 DRUGGABLE GENOME, ENZYME DIOTYROSINE DIOTYROSINE 52358 35728 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MK2206 MK-2206 27026198 52359 35729 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL513909 BI-2536 52360 35730 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Dasatinib DASATINIB 28416483 52361 35731 MSH5 4439 NA gemcitabine GEMCITABINE 31616045 52362 35732 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME FLOVAGATRAN 52365 35733 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor 178103253 LAZABEMIDE 52367 35734 GMNN 51053 DRUGGABLE GENOME TCMDC-124022 CHEMBL548017 52369 35735 POLK 51426 DNA REPAIR, ENZYME FRAXETIN FRAXETIN 52370 35736 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME inhibitor 336446963 52372 35737 SMN2 6607 DRUGGABLE GENOME CID 695758 CHEMBL260028 52373 35738 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME SODIUM TETRADECYL SULFATE 52375 35739 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL101253 VATALANIB 52376 35740 LAG3 3902 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE BMS-986016 RELATLIMAB 25755681 52377 35741 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME inhibitor 249565695 52380 35742 HTT 3064 DRUGGABLE GENOME GNF-PF-1319 CHEMBL235891 52382 35743 PTPRD 5789 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE JSI-124 26267899 52385 35744 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CHF-4227 CHF4227 52386 35745 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GNF-PF-2133 CHEMBL578883 52387 35746 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME pyrazinamide PYRAZINAMIDE 28389387 52388 35747 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1428 NIMODIPINE 52389 35748 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-CINNAMAMIDOBENZAMIDE CHEMBL1522743 52390 35749 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166854 52391 35750 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TAZAROTENE TAZAROTENE 52392 35751 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-38a 52393 35752 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID25991433-Compound-J2 52394 35753 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER VM-26 TENIPOSIDE 9865734 52395 35754 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME MGCD-0103 MOCETINOSTAT 52396 35755 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KOS-2484 52398 35756 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Quinoline derivative 13 52399 35757 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103891 TRIPELENNAMINE 52401 35758 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651552 52403 35759 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE CP-609,754 52405 35760 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME DAPH DAPH 52406 35761 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201627 INSULIN SUSP ISOPHANE SEMISYNTHETIC PURIFIED HUMAN 52408 35762 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-5 52409 35763 PML 5371 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Tretinoin TRETINOIN 52410 35764 CHD4 1108 ENZYME, CLINICALLY ACTIONABLE vorinostat VORINOSTAT 26296641 52414 35765 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 340590210 52415 35766 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME S-707106 52417 35767 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL270995 BRIVANIB ALANINATE 52418 35768 TUBB2B 347733 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 52419 35769 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE TOZASERTIB TOZASERTIB 52420 35770 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 52423 35771 KMO 8564 DRUGGABLE GENOME, ENZYME Cyclopropane 1-carboxylic acid derivative 7 52425 35772 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR ASPIRIN ASPIRIN 10688535 52426 35773 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Dacomitinib DACOMITINIB 22135232,18606718,25899785,22761403,28363995 52428 35774 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX MORPHINE MORPHINE 10719211 52430 35775 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME dabrafenib DABRAFENIB 52433 35776 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565889 52434 35777 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor LINSITINIB LINSITINIB 52435 35778 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME agonist 178101085 N-METHYL-D-ASPARTIC ACID (NMDA) 52436 35779 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME lamivudine LAMIVUDINE 52439 35780 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZOFURAN BENZOFURAN 52440 35781 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102926 BENZOQUINONE 52441 35782 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Eribulin ERIBULIN 52442 35783 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201063 PROPAFENONE HYDROCHLORIDE 52444 35784 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor CHEMBL362558 LY-2090314 52447 35785 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HER2-CAR T Cells 52448 35786 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor 178103434 METHAZOLAMIDE 52449 35787 SMN1 6606 DRUGGABLE GENOME SELICICLIB SELICICLIB 52450 35788 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME Azaindazole amide derivative 1 52453 35789 PDHB 5162 ENZYME CPI-613 52454 35790 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER CEFOXITIN CEFOXITIN 22166395 52455 35791 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 249565845 52457 35792 TARDBP 23435 TUMOR SUPPRESSOR SCH-53020 CHEMBL66279 52458 35793 STK4 6789 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 310264738 CERDULATINIB 52459 35794 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Carbetocin CARBETOCIN 52461 35795 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME SCHEMBL15295829 52462 35796 POLI 11201 DNA REPAIR EUPAFOLIN EUPAFOLIN 52463 35797 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME LITHIUM LITHIUM 2888503 52464 35798 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SOPHORIDINE SOPHORIDINE 21807514 52465 35799 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252166849 52466 35800 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE CELL SURFACE ANTIGENS 16129046 52468 35801 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SENNOSIDE B SENNOSIDE B 52469 35802 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist CHEMBL2110618 MINOPAFANT 52471 35803 FNTA 2339 ENZYME, DRUGGABLE GENOME CP-609,754 52473 35804 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1416988 CHEMBL1389794 52474 35805 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CHLOROTHALONIL CHLOROTHALONIL 52475 35806 GAPDH 2597 DRUGGABLE GENOME, ENZYME GNF-PF-67 CHEMBL578512 52476 35807 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR GW441756X GW441756X 52477 35808 SMN1 6606 DRUGGABLE GENOME CID 3238892 CHEMBL261118 52480 35809 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AG-024322 AG-24322 52481 35810 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-632536 CHEMBL1367933 52482 35811 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ZIRAM ZIRAM 52483 35812 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652494 52484 35813 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR BETAMETHASONE BETAMETHASONE 52486 35814 HMGCR 3156 ENZYME, DRUGGABLE GENOME pravastatin PRAVASTATIN 17563401,18815589,18332269,16103896,18261733,15199031 52487 35815 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Gefitinib GEFITINIB 52489 35816 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NIFEDIPINE NIFEDIPINE 52490 35817 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CARBENDAZIM CARBENDAZIM 52491 35818 HTT 3064 DRUGGABLE GENOME AZACITIDINE AZACITIDINE 52495 35819 PLEKHA6 22874 NA haloperidol HALOPERIDOL 27023437 52496 35820 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650807 52498 35821 PSMD1 5707 NA BORTEZOMIB BORTEZOMIB 24524217 52499 35822 POLI 11201 DNA REPAIR STICTIC ACID STICTIC ACID 52500 35823 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CLOMIFENE CLOMIPHENE 52501 35824 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ARTEANNUIN B ARTEANNUIN B 52503 35825 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR CC-930 TANZISERTIB 52504 35826 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 52506 35827 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 354702204 DEZAPELISIB 52507 35828 GAD1 2571 DRUGGABLE GENOME, ENZYME inhibitor 178101950 52508 35829 XDH 7498 DRUGGABLE GENOME, ENZYME ANTICARCINOGENIC 15686439 52509 35830 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Panitumumab PANITUMUMAB 52510 35831 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor PX-866 SONOLISIB 52512 35832 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 404859045 52513 35833 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Pazopanib PAZOPANIB 26646755,25669829 52514 35834 DHFR 1719 DRUGGABLE GENOME, ENZYME L-MDAM 52516 35835 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME AMLEXANOX AMLEXANOX 52518 35836 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GSK-269962A GSK-269962A 52519 35837 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE THIOGUANINE THIOGUANINE 52520 35838 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Temsirolimus TEMSIROLIMUS 27893038,22271473,22245973,25527417,21216929,21289267,27016228 52522 35839 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME SAXAGLIPTIN SAXAGLIPTIN 52523 35840 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor BMN673 52524 35841 TARDBP 23435 TUMOR SUPPRESSOR STILONIUM IODIDE STILONIUM IODIDE 52525 35842 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GDC-0980 APITOLISIB 26951309 52526 35843 COMT 1312 DRUGGABLE GENOME, ENZYME quetiapine QUETIAPINE 26282453 52527 35844 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE LAMIVUDINE LAMIVUDINE 17172311 52528 35845 NCAM1 4684 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CAR-T cells targeting CD56 52531 35846 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR 5-FLUOROINDOLE-2-CARBOXYLIC ACID 5-FLUOROINDOLE-2-CARBOXYLIC ACID 52532 35847 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BENZO[E]PYRENE BENZO[E]PYRENE 52534 35848 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-57 52536 35849 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME EP42675 52537 35850 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3360203 PILARALISIB 52538 35851 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR APIGENIN APIGENIN 52539 35852 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565855 52540 35853 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 375973251 52541 35854 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PHENYLBUTANOIC ACID PHENYLBUTANOIC ACID 24044874 52542 35855 UGGT2 55757 NA hydrochlorothiazide HYDROCHLOROTHIAZIDE 52543 35856 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-860 CHEMBL593254 52544 35857 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103674 PREDNISONE 52548 35858 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR FENOFIBRATE FENOFIBRATE 52549 35859 GPER1 2852 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR agonist 135651382 52550 35860 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200795 CLEMASTINE FUMARATE 52551 35861 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Bepotastine BEPOTASTINE 52552 35862 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 52553 35863 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-317605 CHEMBL1312050 52554 35864 MAP3K1 4214 CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor CHEMBL1097999 E-6201 52555 35865 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME 1,5-di-substituted pyridine derivative 1 52556 35866 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR G1T28-1 G1T28-1 52557 35867 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR METHYLENE BLUE CHLORIDE HYDRATE METHYLENE BLUE 52559 35868 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CYTARABINE CYTARABINE 52560 35869 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE AVAPRITINIB AVAPRITINIB 30274985 52561 35870 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VANDETANIB VANDETANIB 52562 35871 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651616 52563 35872 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL635 PREDNISONE 52565 35873 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 404859081 52567 35874 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DYDROGESTERONE DYDROGESTERONE 52568 35875 KDM4A 9682 DRUGGABLE GENOME, ENZYME OLEIC ACID OLEIC ACID 52569 35876 ATXN2 6311 NA CLEMASTINE FUMARATE CLEMASTINE FUMARATE 52570 35877 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER XR9051 52571 35878 KDM4A 9682 DRUGGABLE GENOME, ENZYME DOCEBENONE DOCEBENONE 52572 35879 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL NITRAZEPAM NITRAZEPAM 52574 35880 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME RIFAMPIN RIFAMPIN 15771232 52575 35881 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3,6-DIMETHOXYFLAVONE 3,6-DIMETHOXYFLAVONE 52577 35882 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TOLFENAMIC ACID TOLFENAMIC ACID 52578 35883 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PALBOCICLIB PALBOCICLIB 52580 35884 GLS 2744 ENZYME SANGUINARIUM SANGUINARIUM 52581 35885 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Atezolizumab ATEZOLIZUMAB 52582 35886 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-123869 CHEMBL546597 52583 35887 RCE1 9986 ENZYME, PROTEASE, DRUGGABLE GENOME LEVOFLOXACIN LEVOFLOXACIN 52584 35888 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE HIRSUTINOLIDE-13-OACETATE CHEMBL2062869 26331426 52586 35889 CBX1 10951 NA WIN-552122 WIN-552122 52588 35890 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE GNF-PF-3501 CHEMBL581910 52592 35891 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650297 SOBETIROME 52593 35892 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 387065614 52595 35893 POLA1 5422 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, DNA REPAIR NELARABINE NELARABINE 52596 35894 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CAMPHOR CAMPHOR 52597 35895 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY HEXAMETHYLENEBISACETAMIDE HEXAMETHYLENEBISACETAMIDE 10650339 52598 35896 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102228 52599 35897 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivative 1 52600 35898 TUBA4A 7277 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 52603 35899 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist 178100798 52604 35900 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME CARBOPLATIN CARBOPLATIN 15347474 52606 35901 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BETAHISTINE BETAHISTINE 52607 35902 GMNN 51053 DRUGGABLE GENOME TCMDC-123605 CHEMBL547285 52609 35903 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 EMODIN EMODIN 52610 35904 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME RUTAECARPINE RUTAECARPINE 52611 35905 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME valproic acid 23407051 52612 35906 PTGS2 5743 DRUGGABLE GENOME, ENZYME KETOROLAC KETOROLAC 52614 35907 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME THIOLACTOMYCIN THIOLACTOMYCIN 52615 35908 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE RQ-00000007 (oral) 52616 35909 HLA-DQB1 3119 CLINICALLY ACTIONABLE acetaminophen ACETAMINOPHEN 21545408 52617 35910 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE LITHIUM LITHIUM 15286700 52618 35911 BAZ2B 29994 NA BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 52621 35912 XDH 7498 DRUGGABLE GENOME, ENZYME HYPOXANTHINE HYPOXANTHINE 15632148 52624 35913 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BROMOCRIPTINE BROMOCRIPTINE 52625 35914 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AMBAZONE AMBAZONE 52626 35915 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DEFEROXAMINE DEFEROXAMINE 15780758 52629 35916 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME Dasatinib DASATINIB 27231123 52630 35917 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-39 52631 35918 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178100975 52632 35919 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME EPINEPHRINE EPINEPHRINE 52633 35920 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FENOLDOPAM FENOLDOPAM 52634 35921 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME TOLONIUM CHLORIDE TOLONIUM CHLORIDE 52635 35922 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME MAGNESIUM SULFATE 11336444 52636 35923 BCHE 590 DRUGGABLE GENOME, ENZYME Hexafluronium bromide 52638 35924 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME BYAKANGELICIN BYAKANGELICIN 22222157 52639 35925 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR antibody FRESOLIMUMAB FRESOLIMUMAB 52641 35926 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor NAVITOCLAX NAVITOCLAX 52642 35927 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Aminopyrimidine derivative 10 52643 35928 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME STAUROSPORINE STAUROSPORINE 1356124 52644 35929 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650209 52645 35930 TARDBP 23435 TUMOR SUPPRESSOR DNDI1416975 CHEMBL1415851 52647 35931 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE RECOMBINANT INTERLEUKIN 3491626 52651 35932 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 135652732 52652 35933 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102475 52653 35934 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-P1 52654 35935 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME DOCETAXEL DOCETAXEL 15641988 52655 35936 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-659162 CHEMBL471005 52656 35937 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-3792 CHEMBL582983 52658 35938 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR TRICHOSTATIN TRICHOSTATIN 21055848,16921367,19966789,19385600 52659 35939 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME brivanib BRIVANIB 20124951 52660 35940 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178101750 SEMAXANIB 52663 35941 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417025 CHEMBL1320453 52666 35942 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-353720 CHEMBL1408276 52667 35943 PMEL 6490 DRUGGABLE GENOME Multi-epitope peptide melanoma vaccine 22495394 52669 35944 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR I3C 11948137 52670 35945 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE LEPIRUDIN LEPIRUDIN 15894352 52671 35946 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody TREMELIMUMAB TREMELIMUMAB 52672 35947 SFTPA1 653509 DRUGGABLE GENOME CGS 20267 12519892 52673 35948 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2079588 TELATINIB 52674 35949 HMGCR 3156 ENZYME, DRUGGABLE GENOME PMID27537201-Compound-Figure15b 52676 35950 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL154 NAPROXEN 52678 35951 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR GEMTUZUMAB OZOGAMICIN 12576328 52679 35952 SOD2 6648 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE paclitaxel PACLITAXEL 25495407 52680 35953 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PHENYL ISATIN PHENYL ISATIN 52682 35954 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 1,2-NAPHTHOQUINONE 1,2-NAPHTHOQUINONE 52683 35955 FCGR2A 2212 CLINICALLY ACTIONABLE, DRUGGABLE GENOME trastuzumab TRASTUZUMAB 18347005,21109570 52685 35956 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651739 52686 35957 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME RHAMNETIN RHAMNETIN 24397781 52687 35958 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR LOTEPREDNOL ETABONATE 52689 35959 SMARCB1 6598 CLINICALLY ACTIONABLE PANOBINOSTAT PANOBINOSTAT 26920892 52690 35960 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antagonist CHEMBL1743049 OLARATUMAB 52691 35961 ME3 10873 ENZYME GLUTACONATE GLUTACONATE 19595601 52692 35962 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-AMINOBIPHENYL CHEMBL296021 52694 35963 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178103923 VORTIOXETINE 52695 35964 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE talinolol TALINOLOL 18334920 52697 35965 CDK16 5127 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL445813 AT-7519 52698 35966 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EFAROXAN EFAROXAN 52699 35967 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL967 TEMAZEPAM 52701 35968 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651180 52704 35969 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIBENZOYLMETHANE DIBENZOYLMETHANE 52705 35970 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE eplerenone EPLERENONE 23788015 52706 35971 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER HEXACHLOROPHENE HEXACHLOROPHENE 52707 35972 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL2079588 TELATINIB 52708 35973 KDM4A 9682 DRUGGABLE GENOME, ENZYME 4'-EPICHAETOVIRIDIN A CHEMBL1306556 52710 35974 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME PD-0166285 PD-0166285 52712 35975 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545110 RIBOCICLIB 52713 35976 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ANTIMYCIN A ANTIMYCIN A 52714 35977 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650905 RIZATRIPTAN 52715 35978 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR RECOMBINANT INTERLEUKIN 1368117 52717 35979 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE AMINOPTERIN AMINOPTERIN 11410244 52718 35980 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR benazepril BENAZEPRIL 17261659,25143324 52720 35981 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME NALTREXONE NALTREXONE 16716514 52721 35982 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PIMARIC ACID PIMARIC ACID 24799257 52723 35983 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE CHONDROITIN 9409221 52724 35984 PPP1R18 170954 ENZYME gemcitabine GEMCITABINE 31616045 52726 35985 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650993 52728 35986 PPIA 5478 DRUGGABLE GENOME, ENZYME VOCLOSPORIN VOCLOSPORIN 52729 35987 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME MPC-0920 52732 35988 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor TIVOZANIB TIVOZANIB 52733 35989 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME ICA-105665 52734 35990 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 19839593 52735 35991 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR ALSTERPAULLONE ALSTERPAULLONE 52738 35992 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 7 52739 35993 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Peptide analog 51 52741 35994 APOE 348 DRUGGABLE GENOME PLANT STEROL 16677856 52742 35995 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 24524217 52743 35996 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650186 DIMAPRIT 52745 35997 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-218795 CHEMBL9843 52747 35998 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL548 DINOPROSTONE 52748 35999 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE GNF-PF-1577 CHEMBL600315 52749 36000 RRM2B 50484 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL467 HYDROXYUREA 52750 36001 LRMDA 83938 NA tamoxifen TAMOXIFEN 22180457 52752 36002 ABCA1 19 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CSA CYCLOSPORINE 15084924 52753 36003 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE IMATINIB MESYLATE 15650049,15201427,27073655,21969494,27687311 52755 36004 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX NAC ACETYLCYSTEINE 8647183 52756 36005 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME methotrexate METHOTREXATE 28525903,11477075,25098908,23233662,19901119,21317831,23652803,24712521,29683944,25999454 52757 36006 POLB 5423 DNA REPAIR, DRUGGABLE GENOME AG-808 CHEMBL68534 52758 36007 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE 1,4-DIMETHOXYANTHRAQUINONE 1,4-DIMETHOXYANTHRAQUINONE 52760 36008 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-26 52761 36009 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME GSK2606414 CHEMBL2171124 22827572 52762 36010 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GLUCOCORTICOID 16785155 52763 36011 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 52765 36012 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL384304 RG-547 52767 36013 SLC9A3 6550 DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE, EXCHANGER inhibitor CHEMBL3301627 TENAPANOR HYDROCHLORIDE 52768 36014 MAPT 4137 DRUGGABLE GENOME TYRPHOSTIN A9 TYRPHOSTIN A9 52771 36015 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME VX-15 PEPINEMAB 52772 36016 FAAH 2166 ENZYME, DRUGGABLE GENOME V158866 52773 36017 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME antibody 252166891 BEGELOMAB 52774 36018 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124536 CHEMBL580851 52776 36019 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CHLORPROTHIXENE CHLORPROTHIXENE 52777 36020 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CEFACLOR CEFACLOR 52778 36021 BAZ2B 29994 NA EUPAFOLIN EUPAFOLIN 52780 36022 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE TRAMETINIB TRAMETINIB 52781 36023 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL inhibitor 135652003 52783 36024 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor CHEMBL1421 DASATINIB 52784 36025 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME IP10 C8 52785 36026 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME SRT2379 52787 36027 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLORPYRIFOS CHLORPYRIFOS 52788 36028 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME Bryostatin-1 52790 36029 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Quinoline and quinazoline derivative 7 52792 36030 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSAIDS 16997128 52793 36031 EIF4E 1977 DRUGGABLE GENOME RAPAMYCIN SIROLIMUS 10516161,8816458,10477262,15292274,14581487,9867830 52794 36032 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RABEPRAZOLE SODIUM RABEPRAZOLE SODIUM 52795 36033 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649763 52797 36034 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME CATECHOL CATECHOL 52798 36035 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LAROPIPRANT LAROPIPRANT 52799 36036 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 dextromethorphan DEXTROMETHORPHAN 9187528 52800 36037 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE NERATINIB NERATINIB 26619011,24516025,25157968,22046346,23220880,16397024,26243863 52803 36038 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME BRYOSTATIN BRYOSTATIN 52804 36039 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Erlotinib ERLOTINIB 52807 36040 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL DENUFOSOL DENUFOSOL 52808 36041 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL3545156 KW-2450 52809 36042 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 363894211 PEXMETINIB 52810 36043 GAA 2548 DRUGGABLE GENOME, ENZYME GNF-PF-1295 CHEMBL579837 52811 36044 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 boceprevir BOCEPREVIR 52813 36045 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BUPARLISIB BUPARLISIB 25672916 52814 36046 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME ORPHENADRINE ORPHENADRINE 52815 36047 CD44 960 DRUGGABLE GENOME, CELL SURFACE HYALURONAN HYALURONAN 52818 36048 GTF2B 2959 TRANSCRIPTION FACTOR STEROID HORMONE 1517211 52820 36049 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102424 52822 36050 HTT 3064 DRUGGABLE GENOME SJ000047240 CHEMBL590706 52824 36051 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALPHA-TERTHIENYL ALPHA-TERTHIENYL 52827 36052 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW874091X GW874091X 52828 36053 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE DAIDZIN DAIDZIN 52829 36054 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4832 CHEMBL601137 52831 36055 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE OSI-632 OSI-632 52833 36056 PSMB10 5699 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL325041 BORTEZOMIB 52834 36057 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL inhibitor 405560464 52835 36058 BAZ2B 29994 NA NSC-111847 CHEMBL1984884 52836 36059 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-2755 CHEMBL600738 52838 36060 BAZ2B 29994 NA AFIMOXIFENE AFIMOXIFENE 52840 36061 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1480 FELODIPINE 52841 36062 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Pembrolizumab PEMBROLIZUMAB 26645196 52842 36063 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR SP-600125 SP-600125 52847 36064 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID25656651-Compound-28b 52848 36065 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Zarnestra TIPIFARNIB 52849 36066 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-15 52850 36067 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE CHEMBL502774 52853 36068 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 385612221 52854 36069 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME antibody BEVACIZUMAB BEVACIZUMAB 52856 36070 MAPT 4137 DRUGGABLE GENOME CIS-RESVERATROL CIS-RESVERATROL 52857 36071 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ACTINONIN ACTINONIN 52859 36072 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME (RS)-ROSCOVITINE (RS)-ROSCOVITINE 52863 36073 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE BAN2401 BAN2401 52864 36074 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 4-TERT-BUTYLCATECHOL CHEMBL220845 52870 36075 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565693 52872 36076 PPIB 5479 ENZYME, DRUGGABLE GENOME CYCLOSPORIN A 9841882 52873 36077 TARDBP 23435 TUMOR SUPPRESSOR SJ000260214 CHEMBL602740 52874 36078 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TRAIL 15367674 52875 36079 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PREDNISONE PREDNISONE 8976974 52877 36080 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MAPROTILINE HYDROCHLORIDE MAPROTILINE HYDROCHLORIDE 52878 36081 FMO3 2328 ENZYME, DRUGGABLE GENOME anthracyclines and related substances 23441093,21900104 52880 36082 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 249565741 MK-5108 52881 36083 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ACRIFLAVINE CHLORIDE ACRIFLAVINE 52882 36084 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE allosteric modulator 135649681 52883 36085 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE PEMETREXED PEMETREXED 23645741,23060591,21367480,26502926 52884 36086 RGS4 5999 DRUGGABLE GENOME NIFEDIPINE NIFEDIPINE 52885 36087 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 249565586 POZIOTINIB 52888 36088 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE VEMURAFENIB VEMURAFENIB 24265155 52889 36089 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 1,2-BENZANTHRACENE CHEMBL1873684 52890 36090 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME (S)-FELODIPINE (S)-FELODIPINE 52891 36091 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE TAXANES 7954398 52892 36092 SMN1 6606 DRUGGABLE GENOME NSC-93401 CHEMBL452954 52893 36093 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651511 52894 36094 NECTIN4 81607 DRUGGABLE GENOME ASG-22ME ENFORTUMAB VEDOTIN 52896 36095 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE PRALNACASAN PRALNACASAN 52897 36096 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125758 CHEMBL546797 52898 36097 LEPR 3953 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME atorvastatin ATORVASTATIN 19023160 52899 36098 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ACECLIDINE ACECLIDINE 52900 36099 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUPRENORPHINE BUPRENORPHINE 52902 36100 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE LAK CELLS 7947458,1380897,8128185,12202941,7908992,1968054,1379184,8641971 52903 36101 GLS 2744 ENZYME EBSELEN EBSELEN 52905 36102 EPHA3 2042 ENZYME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Ifabotuzumab 52906 36103 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100307 52908 36104 ATAD5 79915 NA ONONIN ONONIN 52909 36105 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME acetazolamide ACETAZOLAMIDE 21342230 52911 36106 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TCMDC-125758 CHEMBL546797 52912 36107 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME 4SC-202 DOMATINOSTAT 52914 36108 ABO 28 NA hormonal contraceptives for systemic use 28750087 52915 36109 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200799 TRAVOPROST 52917 36110 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2-METHOXY-5 (6)EPOXY-TETRAHYDROCARYOPHYLLENE 2-METHOXY-5 (6)EPOXY-TETRAHYDROCARYOPHYLLENE 52918 36111 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BIS(2-ETHYLHEXYL) PHTHALATE BIS(2-ETHYLHEXYL) PHTHALATE 52920 36112 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651064 SPIPERONE 52923 36113 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR N/A 52925 36114 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DITHIOLETHIONE DITHIOLETHIONE 52926 36115 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME GNF-PF-3964 CHEMBL599088 52927 36116 PSMC6 5706 NA inhibitor CHEMBL2103884 OPROZOMIB 52928 36117 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 252166602 NANATINOSTAT 52929 36118 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor XL147 PILARALISIB 52930 36119 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NSC-9037 CHEMBL1451216 52931 36120 VEGFB 7423 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR BEVACIZUMAB BEVACIZUMAB 52932 36121 NDUFA4 4697 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 52936 36122 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Entrectinib ENTRECTINIB 52937 36123 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL2103743 TOFACITINIB CITRATE 52938 36124 KDM4A 9682 DRUGGABLE GENOME, ENZYME FLUPHENAZINE HYDROCHLORIDE FLUPHENAZINE HYDROCHLORIDE 52939 36125 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1200598 DIETHYLSTILBESTROL DIPHOSPHATE 52941 36126 RNF43 54894 ENZYME, CLINICALLY ACTIONABLE RNF43-721 22977472 52942 36127 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Human coagulation factor X 52944 36128 DCAF4 26094 NA corticosteroids 22366774 52946 36129 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE A-1210477 27974663 52947 36130 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZD5363 CAPIVASERTIB 52948 36131 KEAP1 9817 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING DIMETHYL FUMARATE DIMETHYL FUMARATE 23647822 52949 36132 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 178100941 52950 36133 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PD-404182 CHEMBL595227 52951 36134 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-61 52953 36135 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE lamivudine LAMIVUDINE 52954 36136 TUBB4B 10383 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 52955 36137 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME DANTROLENE DANTROLENE 52958 36138 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DIMETHYLCURCUMIN DIMETHYLCURCUMIN 25753330 52959 36139 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE propofol PROPOFOL 18816295 52960 36140 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE NAVITOCLAX NAVITOCLAX 24749893 52961 36141 IL1A 3552 CELL SURFACE, DRUGGABLE GENOME IMMUNOSUPPRESSANT 1703047 52963 36142 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL41194 PRATOSARTAN 52964 36143 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Sarilumab SARILUMAB 52965 36144 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Oxazolyl methylthiothiazole derivative 1 52966 36145 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-668394 CHEMBL336095 52967 36146 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor VORINOSTAT VORINOSTAT 52968 36147 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME EDROPHONIUM EDROPHONIUM 52969 36148 NDUFA2 4695 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 52970 36149 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FURAZABOL FURAZABOL 52971 36150 CD3D 915 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE inhibitor CHEMBL1201608 MUROMONAB-CD3 52973 36151 ATAD5 79915 NA HARMALINE HARMALINE 52974 36152 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE XL-820 XL-820 52975 36153 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Selumetinib SELUMETINIB 52977 36154 GLA 2717 ENZYME, DRUGGABLE GENOME MIGALASTAT MIGALASTAT 52978 36155 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FRANGULIN B FRANGULIN B 20561793 52980 36156 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME WX-554 WX-554 52981 36157 AKR1B1 231 DRUGGABLE GENOME, ENZYME LIDORESTAT LIDORESTAT 52983 36158 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LANATOSIDE C LANATOSIDE C 52985 36159 CXCL8 3576 DRUGGABLE GENOME HYDROQUINONE HYDROQUINONE 52986 36160 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor SCH727965 DINACICLIB 52989 36161 BAZ2B 29994 NA DNDI1417809 CHEMBL1442783 52991 36162 POLB 5423 DNA REPAIR, DRUGGABLE GENOME QUERCETIN QUERCETIN 52992 36163 ATXN2 6311 NA XANTHOANGELOL F XANTHOANGELOL F 52993 36164 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649886 52994 36165 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor NKTR-102 ETIRINOTECAN PEGOL 52995 36166 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE GW843682X GW843682X 52997 36167 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME LU AA24493 52998 36168 MAPK7 5598 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 381118893 52999 36169 PTGS1 5742 ENZYME, DRUGGABLE GENOME ACETAMINOPHEN ACETAMINOPHEN 53000 36170 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GNF-PF-3537 CHEMBL601110 53001 36171 GHRL 51738 DRUGGABLE GENOME CELECOXIB CELECOXIB 18414388 53002 36172 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ENDO-ATROPINE ENDO-ATROPINE 25051097 53003 36173 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1232583 INDEGLITAZAR 53005 36174 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4864 CHEMBL583558 53006 36175 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME topiramate TOPIRAMATE 26524290 53008 36176 MAOA 4128 DRUGGABLE GENOME, ENZYME 8-[METHYL(4-PHENYLBUTYL)AMINO]CAFFEINE CHEMBL1927684 22055712 53009 36177 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME APICIDIN APICIDIN 19705846 53010 36178 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME RO5520985 53011 36179 ARNT 405 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR FUROSPONGOLIDE FUROSPONGOLIDE 18989978 53012 36180 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Azaindazole derivative 1 53013 36181 UBA2 10054 DRUGGABLE GENOME, ENZYME BETULINIC ACID BETULINIC ACID 53014 36182 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME XL765 53015 36183 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GW7074 CHEMBL72365 53017 36184 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 1,2,3,5-TETRACHLOROBENZENE CHEMBL44011 53018 36185 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 249565621 MILCICLIB 53019 36186 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL12 DIAZEPAM 53020 36187 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor REGORAFENIB REGORAFENIB 53022 36188 FCGR2A 2212 CLINICALLY ACTIONABLE, DRUGGABLE GENOME etanercept ETANERCEPT 24048425,27044681 53023 36189 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Indoline derivative 19 53025 36190 AQP1 358 ION CHANNEL, DRUGGABLE GENOME GLUCOCORTICOID 9374641 53026 36191 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Indole-based analog 13 53027 36192 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME ENTRECTINIB ENTRECTINIB 53028 36193 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 178103581 53029 36194 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX LARGAZOLE LARGAZOLE 53030 36195 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CENISERTIB CENISERTIB 53031 36196 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 385612183 53032 36197 ALOX15 246 ENZYME, DRUGGABLE GENOME (S)-PROMETHAZINE (S)-PROMETHAZINE 53033 36198 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135649795 ALENDRONIC ACID 53034 36199 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER MK-571 MK-571 19725578 53035 36200 TNC 3371 DRUGGABLE GENOME, FIBRINOGEN CHEMBL2109583 F16IL2 53036 36201 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME THERAPEUTIC TUMOR INFILTRATING LYMPHOCYTES 27959684 53037 36202 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GW7074 CHEMBL72365 53041 36203 GMNN 51053 DRUGGABLE GENOME GNF-PF-4276 CHEMBL605753 53042 36204 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE AMG 176 53043 36205 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME GALLIC ACID METHYL ESTER GALLIC ACID METHYL ESTER 53045 36206 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME SJ000082806 CHEMBL494668 53046 36207 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor AMG900 AMG-900 53047 36208 ALOX15 246 ENZYME, DRUGGABLE GENOME AG-494 CHEMBL56731 53048 36209 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MANGOSTIN MANGOSTIN 53049 36210 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124064 CHEMBL537045 53050 36211 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE allosteric modulator 178102170 CYCLIC ADENOSINE MONOPHOSPHATE 53051 36212 CSF3 1440 GROWTH FACTOR, DRUGGABLE GENOME Neugranin 25535738 53052 36213 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135649900 OTENZEPAD 53054 36214 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ARSENIC TRIOXIDE 53055 36215 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103892 TROPICAMIDE 53058 36216 MICB 4277 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE peginterferon alfa-2b 53060 36217 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE ACC-001 VANUTIDE CRIDIFICAR 53061 36218 TMEM167A 153339 NA Platinum compounds 28796378 53063 36219 ATAD5 79915 NA SB-205384 CHEMBL1256667 53064 36220 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-3416 CHEMBL579550 53065 36221 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1201466 ESTROGENS, CONJUGATED SYNTHETIC A 53067 36222 TUBB2A 7280 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 53068 36223 HR 55806 NUCLEAR HORMONE RECEPTOR ETS-6218 53069 36224 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178102585 DOVITINIB 53070 36225 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652114 53071 36226 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME PMID27774822-Compound-Figure11Example5 53072 36227 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR TCMDC-124242 CHEMBL529177 21488662 53073 36228 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL1684984 PA-799 53076 36229 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE SP-600125 SP-600125 53077 36230 RGS4 5999 DRUGGABLE GENOME DOCEBENONE DOCEBENONE 53079 36231 GLS 2744 ENZYME SURAMIN SURAMIN 53080 36232 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR enalapril ENALAPRIL 22706620,12522467 53083 36233 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200765 SIBUTRAMINE HYDROCHLORIDE 53086 36234 AKR1C3 8644 ENZYME, DRUGGABLE GENOME inhibitor 252827427 53087 36235 POLB 5423 DNA REPAIR, DRUGGABLE GENOME PICEATANNOL PICEATANNOL 53089 36236 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1240 PROPANTHELINE BROMIDE 53090 36237 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652248 53091 36238 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 4-HYDROXYBENZOHYDRAZIDE CHEMBL124267 53092 36239 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 178103946 TUBACIN 53093 36240 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME STREPTOZOTOCIN STREPTOZOCIN 6305526 53094 36241 NQO2 4835 DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 53095 36242 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE MLN1117 SERABELISIB 28490463 53097 36243 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL429876 CILENGITIDE 53099 36244 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PWT33597 53100 36245 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME ANTISENSE OLIGONUCLEOTIDES 9346938 53104 36246 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR TUMOR NECROSIS FACTOR 10683584 53106 36247 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE CHEMBL412603 53107 36248 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Benzamide derivative 13 53108 36249 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME NSC-628113 CHEMBL176599 53109 36250 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL494089 GSK-690693 53110 36251 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE V-950 22292124 53111 36252 IL10RB 3588 DRUGGABLE GENOME PEG-INTERFERON LAMBA 53112 36253 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR ACTINOMYCIN D 14635187 53115 36254 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL29919 ELPETRIGINE 53118 36255 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102781 53119 36256 PLD2 5338 ENZYME, DRUGGABLE GENOME inhibitor 252827439 53120 36257 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GITOXIN GITOXIN 53123 36258 CALR 811 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Alpha 2 Interferon 26486786 53124 36259 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE allosteric modulator 135652747 53126 36260 CTSZ 1522 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103092 ODANACATIB 53127 36261 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OLANZAPINE OLANZAPINE 53128 36262 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33o 53129 36263 HLA-DQA1 3117 CLINICALLY ACTIONABLE azathioprine AZATHIOPRINE 25217962 53132 36264 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 348353656 SOLCITINIB 53134 36265 CD14 929 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 24776844 53135 36266 BCL2L2 599 CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist 252166532 ABT 737 53136 36267 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 252166801 53138 36268 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ADAPALENE ADAPALENE 53139 36269 ATXN2 6311 NA TOLONIUM CHLORIDE TOLONIUM CHLORIDE 53140 36270 GMNN 51053 DRUGGABLE GENOME GNF-PF-1938 CHEMBL587728 53142 36271 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Sulfamic acid ester derivative 1 53143 36272 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NALOXONE NALOXONE 53145 36273 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MRS-1845 CHEMBL1256776 53147 36274 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2037511 EPELSIBAN 53148 36275 TSPO 706 DRUGGABLE GENOME Prazepam PRAZEPAM 53149 36276 ALOX5 240 DRUGGABLE GENOME, ENZYME inhibitor 178101979 ZILEUTON 53150 36277 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102334 53151 36278 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PIMOZIDE PIMOZIDE 53152 36279 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE LOPERAMIDE LOPERAMIDE 53153 36280 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 178101007 FELODIPINE 53156 36281 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 223366074 BRIGATINIB 53157 36282 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Fenofibrate FENOFIBRATE 53158 36283 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545134 LY-2780301 53159 36284 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME BYL719 ALPELISIB 53160 36285 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER NSC-228155 CHEMBL505670 53161 36286 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor NILOTINIB NILOTINIB 53164 36287 GMNN 51053 DRUGGABLE GENOME BIFONAZOLE BIFONAZOLE 53165 36288 AQP4 361 ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PHENYTOIN PHENYTOIN 18572411 53168 36289 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER vincristine VINCRISTINE 53169 36290 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 249565586 POZIOTINIB 53172 36291 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TPCK TPCK 53173 36292 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102756 53175 36293 FH 2271 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR DIETHYLDITHIOCARBAMATE DITIOCARB 1850448 53176 36294 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR perindopril PERINDOPRIL 20712529,8952600 53178 36295 GC 2638 DRUGGABLE GENOME ASA ASPIRIN 17555340 53180 36296 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME Debio 0827 53181 36297 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FLUSPIRILENE FLUSPIRILENE 53182 36298 OXSR1 9943 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565899 53183 36299 MAP3K11 4296 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565875 53185 36300 CA2 760 DRUGGABLE GENOME, ENZYME SULTHIAME SULTHIAME 53187 36301 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NELFINAVIR MESYLATE NELFINAVIR MESYLATE 53188 36302 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor SF1126 53190 36303 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ACYCLOVIR ACYCLOVIR 8683981 53191 36304 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR BLEOMYCIN BLEOMYCIN 16148050 53192 36305 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102911 53193 36306 LGR6 59352 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102183 53195 36307 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist CHEMBL2105648 PALOVAROTENE 53196 36308 PDE5A 8654 ENZYME, DRUGGABLE GENOME OSI-461 CP-461 53199 36309 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR HORMONES 1698537 53201 36310 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178103458 VORINOSTAT 53202 36311 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-24 53204 36312 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LOVASTATIN LOVASTATIN 53206 36313 ALOX15B 247 DRUGGABLE GENOME, ENZYME GNF-PF-321 CHEMBL581044 53207 36314 ALOX15 246 ENZYME, DRUGGABLE GENOME PYROGALLOL PYROGALLOL 53208 36315 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-27 53209 36316 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL agonist 178101000 53210 36317 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME PD173074 53211 36318 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ADAPALENE ADAPALENE 53213 36319 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PIRETANIDE PIRETANIDE 53214 36320 XPO1 7514 CLINICALLY ACTIONABLE, KINASE isoniazid ISONIAZID 22341855,29036176 53215 36321 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102261 53216 36322 APC 324 CLINICALLY ACTIONABLE Vandetanib VANDETANIB 20811697 53218 36323 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME disopyramide DISOPYRAMIDE 53219 36324 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CLOXYQUIN CLOXYQUIN 53220 36325 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DANAZOL DANAZOL 22931300 53223 36326 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR DIACEREIN DIACEREIN 53224 36327 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist 404859013 53226 36328 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL antagonist,activator 135652731 53227 36329 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 381118891 53228 36330 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-4029 CHEMBL596633 53230 36331 GMNN 51053 DRUGGABLE GENOME RAC-GONIOTHALAMIN CHEMBL1170485 53231 36332 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 chlorzoxazone CHLORZOXAZONE 9187528 53232 36333 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BROMOCRIPTINE MESYLATE BROMOCRIPTINE MESYLATE 53233 36334 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor AXITINIB AXITINIB 53235 36335 USP1 7398 DNA REPAIR, PROTEASE, ENZYME METHYLBENZETHONIUM CHLORIDE METHYLBENZETHONIUM CHLORIDE 53236 36336 CXCL8 3576 DRUGGABLE GENOME LANSOPRAZOLE LANSOPRAZOLE 17122965 53238 36337 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME COCAINE COCAINE 53239 36338 MAGEA1 4100 NA CAR-T cells targeting MAGE-A1 53241 36339 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE CA-170 53242 36340 USP1 7398 DNA REPAIR, PROTEASE, ENZYME MORIN MORIN 53243 36341 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 135651750 GALANIN 53244 36342 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE indacaterol INDACATEROL 53246 36343 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DEQUALINIUM DEQUALINIUM 53247 36344 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545413 FLUMATINIB 53249 36345 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR estradiol / progesterone 53250 36346 PTGES 9536 DRUGGABLE GENOME, ENZYME Benzamide derivative 15 53251 36347 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AFM24 53253 36348 ATXN2 6311 NA OXYPHENBUTAZONE OXYPHENBUTAZONE 53254 36349 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100324 53255 36350 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist 252166708 DANIRIXIN 53256 36351 KDM4A 9682 DRUGGABLE GENOME, ENZYME 3-HYDROXYANTHRANILIC ACID CHEMBL445304 53257 36352 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL2165191 AZD-6482 53258 36353 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME DIMETHYLPHENYLPIPERAZINIUM IODIDE DIMETHYLPHENYLPIPERAZINIUM IODIDE 53259 36354 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ENDOMORPHIN-1 ENDOMORPHIN-1 22724433 53260 36355 XRCC1 7515 CLINICALLY ACTIONABLE doxorubicin DOXORUBICIN 53261 36356 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1265 ADAPALENE 53262 36357 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178104006 BUDESONIDE 53263 36358 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME D-DOPA CHEMBL211670 53264 36359 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME activator 135650745 53265 36360 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-25 53266 36361 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Cisplatin CISPLATIN 25193512,26801247,27454289 53267 36362 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR antagonist 135649800 AFIMOXIFENE 53268 36363 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE GW441756X GW441756X 53271 36364 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME PF-562271 PF-00562271 53272 36365 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HERNIARIN HERNIARIN 53273 36366 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102738 53275 36367 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650293 FURTRETHONIUM 53276 36368 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL3545165 AFACIFENACIN 53278 36369 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME IL-6 17078027 53280 36370 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR RXDX 101 53281 36371 MBNL1 4154 DRUGGABLE GENOME MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 53282 36372 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SULFORAPHANE SULFORAPHANE 1549603 53284 36373 RAB9A 9367 ENZYME, DRUGGABLE GENOME RILUZOLE RILUZOLE 53285 36374 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ATROPINE ATROPINE 53286 36375 GGH 8836 PROTEASE, ENZYME, DRUGGABLE GENOME pemetrexed PEMETREXED 24732178 53287 36376 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LUTEOLIN LUTEOLIN 53289 36377 NAPEPLD 222236 ENZYME inhibitor 405560496 53290 36378 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME US8933228, 3 53293 36379 EPHX2 2053 DRUGGABLE GENOME, ENZYME inhibitor 375973267 53294 36380 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor GSK2636771 GSK-2636771 53296 36381 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 252166527 PEFICITINIB 53297 36382 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE CPH-102 53298 36383 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NISOLDIPINE NISOLDIPINE 53299 36384 ATXN2 6311 NA GNF-PF-2657 CHEMBL578944 53301 36385 MIA 8190 GROWTH FACTOR, DRUGGABLE GENOME LYMPHOKINE-ACTIVATED KILLER CELL 15386421 53302 36386 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135651318 53303 36387 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX CYTOSPORONE B CYTOSPORONE B 18690216 53305 36388 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMSACRINE AMSACRINE 22931300 53306 36389 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE HMPL-523 HMPL-523 53307 36390 GZMB 3002 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166850 53308 36391 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PD-0325901 PD-0325901 26272063,26267534,27488531,16273091,26573800 53309 36392 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME FLUPIRTINE MALEATE FLUPIRTINE MALEATE 53310 36393 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 53311 36394 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200395 ORPHENADRINE CITRATE 53313 36395 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL blocker 53801055 53314 36396 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL1742994 BRENTUXIMAB VEDOTIN 53315 36397 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SULFADIAZINE, SILVER SULFADIAZINE, SILVER 53316 36398 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME PAMOIC ACID PAMOIC ACID 53318 36399 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TCMDC-124307 CHEMBL546865 53319 36400 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Azaindazole amide derivative 1 53320 36401 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL545315 CANERTINIB DIHYDROCHLORIDE 53321 36402 XDH 7498 DRUGGABLE GENOME, ENZYME STN 9367530 53322 36403 APC 324 CLINICALLY ACTIONABLE JW55 22440753 53323 36404 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565641 LY-2090314 53325 36405 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor BMS-690514 BMS-690514 53327 36406 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BI-847325 25873592 53329 36407 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor PELITINIB PELITINIB 53330 36408 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME VEMURAFENIB VEMURAFENIB 21107323,23569304 53331 36409 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR ILORASERTIB ILORASERTIB 53332 36410 RICTOR 253260 CLINICALLY ACTIONABLE inhibitor OSI-027 OSI-027 53334 36411 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 252166685 53335 36412 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Dabigatran DABIGATRAN 27893182,27261537 53336 36413 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE PA-401 53338 36414 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PD173074 24122810,18757403 53339 36415 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 4,4'-THIODIANILINE 4,4'-THIODIANILINE 53340 36416 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AMG 747 53341 36417 SOCS1 8651 CLINICALLY ACTIONABLE, KINASE INSULIN INSULIN 18171911 53342 36418 HTT 3064 DRUGGABLE GENOME TERFENADINE TERFENADINE 53344 36419 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PENTAERYTHRITOL TETRANITRATE PENTAERYTHRITOL TETRANITRATE 53347 36420 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-10 53348 36421 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR Indazoletriazolephenyl derivative 2 53349 36422 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL3545085 XL-228 53350 36423 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DELTIBANT DELTIBANT 53351 36424 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1201163 SUFENTANIL CITRATE 53352 36425 POLK 51426 DNA REPAIR, ENZYME STICTIC ACID STICTIC ACID 53353 36426 CHURC1 91612 NA methylphenidate METHYLPHENIDATE 29382897 53354 36427 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-47 53355 36428 GMNN 51053 DRUGGABLE GENOME BENZBROMARONE BENZBROMARONE 53358 36429 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME dasatinib DASATINIB 24322003 53360 36430 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565856 53362 36431 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565941 53363 36432 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR AZQ DIAZIQUONE 8617583 53364 36433 LSS 4047 ENZYME, DRUGGABLE GENOME inhibitor 178103327 53365 36434 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor 135652702 ROTTLERIN 53366 36435 KCNH6 81033 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL113461 TEDISAMIL 53367 36436 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 26 53368 36437 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 clonazepam CLONAZEPAM 9187528 53369 36438 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TABIMORELIN TABIMORELIN 53371 36439 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE clindamycin CLINDAMYCIN 18695978 53372 36440 ADGRL3 23284 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME nicotine NICOTINE 53373 36441 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3545093 ZYH7 53375 36442 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE 681640 CHEMBL379975 53376 36443 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME PIPERINE PIPERINE 53377 36444 SRI 6717 NA ISOPROTERENOL ISOPROTERENOL 15754088 53378 36445 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652398 53379 36446 KCNH8 131096 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL284348 DALFAMPRIDINE 53380 36447 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR POTASSIUM DICHROMATE POTASSIUM DICHROMATE 53381 36448 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE IMGN289 24423618 53382 36449 ACY3 91703 NA atenolol ATENOLOL 28353407 53383 36450 DDB1 1642 DNA REPAIR inhibitor CHEMBL43452 POMALIDOMIDE 53384 36451 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME modulator CHEMBL93747 NETOGLITAZONE 53385 36452 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-95 53386 36453 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME GDC-0994 RAVOXERTINIB 25320010 53388 36454 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE PF-03084014 NIROGACESTAT 53389 36455 ADH1A 124 DRUGGABLE GENOME FOMEPIZOLE FOMEPIZOLE 53390 36456 FAAH 2166 ENZYME, DRUGGABLE GENOME Isoxazoline derivative 3 53392 36457 BAZ2B 29994 NA TCMDC-123916 CHEMBL493863 53393 36458 KIF11 3832 DRUGGABLE GENOME NSC-123138 CHEMBL409102 21344920 53395 36459 MAPT 4137 DRUGGABLE GENOME LUTEOLIN LUTEOLIN 53399 36460 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE FENTANYL FENTANYL 53400 36461 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135649700 53402 36462 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LIOTHYRONINE LIOTHYRONINE 53403 36463 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Aryl 1,2-diamine derivative 1 53404 36464 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 187051798 BELINOSTAT 53405 36465 BAZ2B 29994 NA GNF-PF-3756 CHEMBL597035 53408 36466 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ALICAFORSEN ALICAFORSEN 53409 36467 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR TEMSIROLIMUS TEMSIROLIMUS 16341243 53410 36468 HMGCR 3156 ENZYME, DRUGGABLE GENOME PMID27537201-Compound-Figure11 53412 36469 RGS4 5999 DRUGGABLE GENOME PROTOPORPHYRIN PROTOPORPHYRIN 53414 36470 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE Antiinflammatory agents, non-steroids 25096645 53415 36471 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-6 53416 36472 MAPK7 5598 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR XMD8-85 CHEMBL1673039 21412406 53417 36473 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME RBC 16192690 53421 36474 RAPGEF3 10411 ENZYME LOBARIC ACID LOBARIC ACID 53422 36475 MT1H 4496 NA HORMONES 15196976 53423 36476 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor MK5108 MK-5108 53424 36477 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-95397 CHEMBL429095 53426 36478 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHLORPYRIFOS-METHYL CHLORPYRIFOS-METHYL 53429 36479 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME AZELASTINE AZELASTINE 53430 36480 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR OX40 LIGAND 12496388 53431 36481 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DEXMEDETOMIDINE DEXMEDETOMIDINE 53432 36482 ALDH1A1 216 DRUGGABLE GENOME, ENZYME U-0124 CHEMBL97858 53433 36483 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME antibody 315661191 53434 36484 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201561 PEGINTERFERON ALFA-2B 53435 36485 MGLL 11343 DRUGGABLE GENOME, ENZYME Azetidinyl-piperazine derivative 2 53437 36486 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE FGFR INHIBITOR AZD4547 31027687 53438 36487 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR AC1LFGWU 53440 36488 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor SOPHORETIN QUERCETIN 53441 36489 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE REV-5901 REV-5901 53442 36490 PNPLA3 80339 ENZYME daunorubicin DAUNORUBICIN 28744905 53443 36491 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CAPECITABINE CAPECITABINE 24957073 53444 36492 SMN2 6607 DRUGGABLE GENOME nusinersen NUSINERSEN 53446 36493 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200654 BENOXINATE HYDROCHLORIDE 53447 36494 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GANCAONIN L GANCAONIN L 20022509 53449 36495 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL CROMOGLYCATE LISETIL HYDROCHLORIDE 53450 36496 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE prasugrel PRASUGREL 21828263 53451 36497 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DECA-1,9-DIENE CHEMBL31020 53452 36498 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME LC-150444 GEMIGLIPTIN 53453 36499 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER L-733060 CHEMBL27006 53454 36500 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Gemcitabine GEMCITABINE 26853339 53455 36501 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545382 R-348 53457 36502 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL2062267 HYDROCODONE BITARTRATE 53459 36503 TNFRSF1A 7132 CELL SURFACE, DRUGGABLE GENOME adalimumab ADALIMUMAB 22480748 53460 36504 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR GEMCITABINE GEMCITABINE 19543324,17131328,23038758,24647522,15217961,14977831,24595080 53461 36505 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL559 DEXTROTHYROXINE 53462 36506 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist CHEMBL1480 FELODIPINE 53465 36507 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR alpelisib ALPELISIB 53468 36508 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE BINIMETINIB BINIMETINIB 26925841 53469 36509 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SKIMMIANINE SKIMMIANINE 53470 36510 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 53472 36511 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME FGI-101-1A6 FGI-101-1A6 53474 36512 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PF-05230907 53475 36513 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME TAMATINIB R-406 53477 36514 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650832 PIRENZEPINE 53480 36515 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-102742 CHEMBL1519374 53481 36516 POLI 11201 DNA REPAIR RO-137410 CHEMBL275311 53482 36517 KLK4 9622 PROTEASE, DRUGGABLE GENOME, ENZYME LM-030 53484 36518 MAOB 4129 DRUGGABLE GENOME, ENZYME Piperonal PIPERONAL 53485 36519 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1416975 CHEMBL1415851 53488 36520 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR 17 BETA-ESTRADIOL 11498938 53489 36521 PNP 4860 ENZYME, DRUGGABLE GENOME Peldesine PELDESINE 53490 36522 CA1 759 DRUGGABLE GENOME, ENZYME LEVETIRACETAM LEVETIRACETAM 53492 36523 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1676 FLUTICASONE FUROATE 53493 36524 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME RO-0282750 CHEMBL1397270 53496 36525 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CARBETAPENTANE CARBETAPENTANE 53497 36526 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 315661253 53498 36527 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 178100433 53499 36528 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE LEUCOVORIN LEUCOVORIN 53500 36529 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102562 53501 36530 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 249565747 AEW-541 53502 36531 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL574737 UCN-01 53503 36532 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ACLIDINIUM ACLIDINIUM 53504 36533 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 6,4'-DIHYDROXYFLAVONE CHEMBL484663 53505 36534 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL565612 SOTRASTAURIN 53506 36535 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-123414 CHEMBL16751 53507 36536 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL325041 BORTEZOMIB 53508 36537 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME RG7129 53509 36538 CD9 928 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE STEROID HORMONE 17126340 53510 36539 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME ETHACRYNIC ACID 9155531 53511 36540 RACGAP1 29127 NA LASSBIO-1182 CHEMBL1173140 53512 36541 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652469 53513 36542 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE N/A 18648004,16384925,21343560,22869879,25111512,21714648,22689681,22180162,25652455,22753902,9746770 53514 36543 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR TROGLITAZONE TROGLITAZONE 17924870 53515 36544 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TETRAIDOFLUORESCEIN TETRAIDOFLUORESCEIN 53516 36545 GMNN 51053 DRUGGABLE GENOME TPCK TPCK 53518 36546 CXCL8 3576 DRUGGABLE GENOME DICHLORVOS DICHLORVOS 53519 36547 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GALLIC ACID GALLIC ACID 53520 36548 TYMSOS 494514 NA prednisone PREDNISONE 53522 36549 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TRN-157 53523 36550 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 404859010 53524 36551 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PHA-767491 CHEMBL225519 53525 36552 RALBP1 10928 TRANSPORTER, ABC TRANSPORTER vincristine VINCRISTINE 27180762 53527 36553 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME SUN-K0706 53528 36554 PDE10A 10846 ENZYME, DRUGGABLE GENOME inhibitor 252827415 53532 36555 STRAP 11171 KINASE ADJUVANT 15720808 53534 36556 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178103760 ETODOLAC 53535 36557 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33m 53536 36558 POLI 11201 DNA REPAIR AMENTOFLAVONE AMENTOFLAVONE 53539 36559 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CYT-107 53542 36560 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE AMPRENAVIR AMPRENAVIR 16433896 53543 36561 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME INSULIN INSULIN 8389451 53544 36562 TPM3 7170 KINASE, CLINICALLY ACTIONABLE MIDAZOLAM MIDAZOLAM 16738805 53546 36563 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE LENVATINIB LENVATINIB 53549 36564 ATP5F1D 513 TRANSPORTER DESFLURANE DESFLURANE 53550 36565 GALNS 2588 DRUGGABLE GENOME, ENZYME elosulfase alfa 53551 36566 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE CORONOPILIN CORONOPILIN 53553 36567 MPHOSPH8 54737 NA SU-4312 CHEMBL328710 53554 36568 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CLORAZEPATE CLORAZEPIC ACID 53555 36569 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE SELUMETINIB SELUMETINIB 25952648,24685132 53556 36570 FBXW7 55294 DNA REPAIR, CLINICALLY ACTIONABLE Temsirolimus TEMSIROLIMUS 24360397 53557 36571 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ETHACRYNIC ACID ETHACRYNIC ACID 53558 36572 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200443 MERETHOXYLLINE PROCAINE 53559 36573 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201729 DRONEDARONE HYDROCHLORIDE 53560 36574 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 letrozole LETROZOLE 11394901,16402128,15940289,16952495,19238117,18698229,12802030,16891249,10544257,15660270,20860463,11241319,15475735,16378601,18212800,15592323,9827545,20089352,11725533,19921195,15980104,11237731,19845430,10999944,20155256,16272956,17130279,11434509,12042667,15225612,15900015,21494765,10448083,30094551,20596643,11180041,12325023,12223434,12844137,19604090,11684323,15265511,15308589,21521021,16452582,19225447,11779172,12749606,18380793,14981342,17220563,17112802,21975350 53561 36575 NDUFB4 4710 ENZYME inhibitor CHEMBL3545135 NV-128 53563 36576 PLD1 5337 ENZYME, DRUGGABLE GENOME US9453017, 1 53564 36577 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BINIMETINIB BINIMETINIB 32822286,27167191 53565 36578 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL3545422 MIRANSERTIB 53567 36579 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME clavulanate CLAVULANIC ACID 53568 36580 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR PF-05212384 GEDATOLISIB 21325073 53570 36581 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CYCLOSPORINE CYCLOSPORINE 14550820,10515383 53571 36582 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-4156 CHEMBL585279 53574 36583 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor 178103558 BEGACESTAT 53575 36584 PI4K2A 55361 DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, ENZYME inhibitor 135651426 ADENOSINE 53578 36585 CTNNA3 29119 NA antidepressants 53580 36586 ACY3 91703 NA bisoprolol BISOPROLOL 28353407 53581 36587 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME TETRAIDOFLUORESCEIN TETRAIDOFLUORESCEIN 53583 36588 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BAZEDOXIFENE BAZEDOXIFENE 24456369 53584 36589 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL1231124 AZD-1480 53585 36590 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME NERVE GROWTH FACTOR 10713102 53586 36591 CA1 759 DRUGGABLE GENOME, ENZYME RESORCINOL RESORCINOL 26073005 53589 36592 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME JVS-100 53590 36593 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL2110725 VINFLUNINE 53591 36594 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME SELENOMETHIONINE SELENOMETHIONINE 12539231 53594 36595 PSMB7 5695 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL325041 BORTEZOMIB 53595 36596 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 178103212 DONEPEZIL 53596 36597 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Alpelisib ALPELISIB 27126994 53597 36598 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Levothyroxine LEVOTHYROXINE 53599 36599 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Radiotherapy 26853339,26363012 53600 36600 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE GW843682X GW843682X 53604 36601 TUBB4B 10383 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 53605 36602 RGS4 5999 DRUGGABLE GENOME GUANIDINONALTRINDOLE GUANIDINONALTRINDOLE 53607 36603 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE APIGENIN APIGENIN 53608 36604 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 681640 CHEMBL379975 53609 36605 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme4Bottom 53610 36606 MPHOSPH8 54737 NA SKF-83565 HYDROBROMIDE CHEMBL541585 53612 36607 GMNN 51053 DRUGGABLE GENOME TEROXIRONE TEROXIRONE 53613 36608 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL593430 ATAGABALIN 53615 36609 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Imidazo[4,5-c]pyridine derivative 1 53616 36610 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL2105712 AFATINIB DIMALEATE 53617 36611 PAK2 5062 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME allosteric modulator 310264717 53620 36612 MAPT 4137 DRUGGABLE GENOME LANSOPRAZOLE LANSOPRAZOLE 53621 36613 ALDH1A1 216 DRUGGABLE GENOME, ENZYME WIN-55212-2 WIN-552122 53622 36614 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650162 53623 36615 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL971 PENTOBARBITAL SODIUM 53624 36616 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DANTHRON DANTHRON 53627 36617 HIF1AN 55662 NA L-3,4-DEHYDROPROLINE CHEMBL78920 21665470 53628 36618 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ISOPROTERENOL ISOPROTERENOL 19464886,16680159 53629 36619 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME ALSTERPAULLONE ALSTERPAULLONE 53630 36620 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME PegCNTF 53631 36621 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE DHEA PRASTERONE 15501480 53632 36622 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TYRPHOSTIN A9 TYRPHOSTIN A9 53633 36623 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Saralasin Acetate 53635 36624 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL2104984 SODELGLITAZAR 53637 36625 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 4-(7-METHYLOCTYL)PHENOL CHEMBL503990 53641 36626 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME US8933228, Ref 2 53644 36627 SPSB2 84727 DRUGGABLE GENOME, B30_2 SPRY DOMAIN methylphenidate METHYLPHENIDATE 29382897 53645 36628 TFAP2A 7020 TRANSCRIPTION FACTOR INDINAVIR INDINAVIR 10996400 53646 36629 APOE 348 DRUGGABLE GENOME SOY PROTEIN 1902348 53647 36630 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor 328083471 53649 36631 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-4864 CHEMBL583558 53650 36632 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651406 53651 36633 SIK3 23387 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 178102305 DASATINIB 53653 36634 CA1 759 DRUGGABLE GENOME, ENZYME PHENOL PHENOL 53655 36635 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE DOCETAXEL DOCETAXEL 53660 36636 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1951575 VIDUPIPRANT 53664 36637 FAAH 2166 ENZYME, DRUGGABLE GENOME Pyrazole derivative 81 53666 36638 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR 870086 (topical, atopic dermatitis), GlaxoSmithKline 53667 36639 CXCR6 10663 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135651711 53669 36640 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 381118839 REVEFENACIN 53670 36641 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-123789 CHEMBL588859 53673 36642 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MENADIONE SODIUM BISULPHITE MENADIONE SODIUM BISULPHITE 53674 36643 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR bleomycin BLEOMYCIN 53677 36644 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL918 PHENACEMIDE 53678 36645 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AR-A014418 CHEMBL259850 53679 36646 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pembrolizumab PEMBROLIZUMAB 53680 36647 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME NG2-73 ADIPIPLON 53681 36648 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME blocker 135650617 DIZOCILPINE 53683 36649 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AVID100 53684 36650 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PKI-587 GEDATOLISIB 53685 36651 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 381118818 53686 36652 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR 22056021,20826716,16282176,26439803 53687 36653 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DESIPRAMINE DESIPRAMINE 53688 36654 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor DOVITINIB DOVITINIB 53689 36655 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR fluoxetine FLUOXETINE 20016225 53690 36656 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE GEFITINIB GEFITINIB 53691 36657 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EPITESTOSTERONE EPITESTOSTERONE 53692 36658 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR abemaciclib ABEMACICLIB 53693 36659 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Oleclumab OLECLUMAB 53694 36660 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651253 53695 36661 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Epoxysuccinate derivative 1 53696 36662 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME NSC-638080 CHEMBL136344 53697 36663 TOP2B 7155 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL68117 VOSAROXIN 53698 36664 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME MDX-1203 53700 36665 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 53704 36666 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR TOPOISOMERASE-II INHIBITOR 12874004 53705 36667 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PALIFERMIN PALIFERMIN 53709 36668 KDM4A 9682 DRUGGABLE GENOME, ENZYME CITRIC ACID CITRIC ACID 53710 36669 PAH 5053 DRUGGABLE GENOME, ENZYME activator 178101959 SAPROPTERIN 53711 36670 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GNF-PF-1852 CHEMBL533293 53712 36671 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MIFEPRISTONE MIFEPRISTONE 53713 36672 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE CHIR-99021 CHIR-99021 53714 36673 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME (RS)-ROSCOVITINE (RS)-ROSCOVITINE 53715 36674 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CAPECITABINE CAPECITABINE 23988873 53716 36675 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL2104954 BALAMAPIMOD 53717 36676 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MVA-BN-HER-2 53718 36677 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 310264764 53720 36678 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE blocker CHEMBL284348 DALFAMPRIDINE 53721 36679 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8536181, C14 53723 36680 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270010-Compound-Figure16-a 53724 36681 USP1 7398 DNA REPAIR, PROTEASE, ENZYME IDARUBICIN IDARUBICIN 53725 36682 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CHELERYTHRINE CHELERYTHRINE 53726 36683 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE RUCAPARIB RUCAPARIB 27908594 53727 36684 CASP2 835 PROTEASE, DRUGGABLE GENOME, ENZYME SPERMINE SPERMINE 18366176 53731 36685 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME US8481733, 95 53733 36686 TUBA1B 10376 DRUGGABLE GENOME CHEMBL492399 VERUBULIN 53734 36687 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE inhibitor CHEMBL1201584 ABCIXIMAB 53735 36688 FZD7 8324 G PROTEIN COUPLED RECEPTOR, KINASE antagonist 381745005 53736 36689 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE GOSSYPOL GOSSYPOL 53737 36690 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR LUCIDUMOL A LUCIDUMOL A 22014750 53738 36691 IMPDH2 3615 DRUGGABLE GENOME, ENZYME AVN-944 AVN-944 53739 36692 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-74859 CHEMBL477936 53740 36693 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR TRICIRIBINE TRICIRIBINE 53742 36694 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650726 53743 36695 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR INTERCALATING AGENT 2914585 53744 36696 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL3545134 LY-2780301 53745 36697 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DOVITINIB DOVITINIB 53747 36698 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE EPINEPHRINE EPINEPHRINE 53750 36699 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CO1686 24065731,25948633,27252416,25939061,27283993,26206867,27435396,25923550 53751 36700 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PKI-166 PKI-166 22018877 53754 36701 GMNN 51053 DRUGGABLE GENOME PIPLARTINE PIPLARTINE 53755 36702 LTB 4050 DRUGGABLE GENOME inhibitor CHEMBL1742988 BAMINERCEPT 53756 36703 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE 2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE 53757 36704 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor XL147 PILARALISIB 53758 36705 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor BELINOSTAT BELINOSTAT 53759 36706 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR ANGIOTENSIN CONVERTING ENZYME INHIBITOR 15770649 53761 36707 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 381118818 53763 36708 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Cetuximab CETUXIMAB 53764 36709 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 1-ETHYLPYRIDINIUM IODIDE CHEMBL539954 53765 36710 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TCMDC-125758 CHEMBL546797 53766 36711 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE R343 53767 36712 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR Birinapant BIRINAPANT 53768 36713 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE LESCOL LESCOL 53769 36714 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME 7-azaindole derivative 3 53770 36715 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Pyridine derivative 22 53773 36716 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Sorafenib SORAFENIB 53774 36717 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor NAVITOCLAX NAVITOCLAX 53775 36718 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PACRITINIB PACRITINIB 32226941 53778 36719 VKORC1 79001 DRUGGABLE GENOME, ENZYME TECARFARIN TECARFARIN 53779 36720 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GALLIC ACID GALLIC ACID 53782 36721 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE Thyrotropin Alfa 53784 36722 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME alirocumab ALIROCUMAB 53785 36723 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL agonist 178101048 53787 36724 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CSA CYCLOSPORINE 8212167 53788 36725 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME CGP-60474 CHEMBL300389 53789 36726 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist 135651388 53790 36727 DHFR 1719 DRUGGABLE GENOME, ENZYME PIRITREXIM PIRITREXIM 53793 36728 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME E-3810 RABEPRAZOLE SODIUM 53794 36729 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL TOPIRAMATE TOPIRAMATE 53795 36730 LGR5 8549 G PROTEIN COUPLED RECEPTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME fluorouracil FLUOROURACIL 25665511 53796 36731 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1416975 CHEMBL1415851 53797 36732 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL FLUDIAZEPAM FLUDIAZEPAM 53800 36733 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL3301610 ABEMACICLIB 53801 36734 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR ribavirin RIBAVIRIN 53806 36735 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYSTEAMINE CYSTEAMINE 53807 36736 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651245 TERFENADINE 53811 36737 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2011803494010 53812 36738 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417086 CHEMBL1224755 53813 36739 QRFPR 84109 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651879 53814 36740 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE LIDOCAINE LIDOCAINE 53815 36741 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRAMUSTINE ESTRAMUSTINE 53816 36742 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 328083485 OSI-930 53817 36743 USP1 7398 DNA REPAIR, PROTEASE, ENZYME 4-AMINO-[1,2]NAPHTHOQUINONE 4-AMINO-[1,2]NAPHTHOQUINONE 53818 36744 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TRICHOSTATIN TRICHOSTATIN 21055848,16921367,19966789,19385600 53820 36745 BCHE 590 DRUGGABLE GENOME, ENZYME inhibitor 310264772 PYRIDOSTIGMINE 53822 36746 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor CHEMBL3833309 ELENBECESTAT 53823 36747 TSPO 706 DRUGGABLE GENOME Chlordiazepoxide CHLORDIAZEPOXIDE 53824 36748 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-125544 CHEMBL533602 53826 36749 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Radiotherapy 27154916 53829 36750 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PROTEASOME INHIBITOR 15498850 53831 36751 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Tumor necrosis factor alpha (TNF-alpha) inhibitors 27670765 53833 36752 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE RESERPINE RESERPINE 7282227 53834 36753 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 310264679 53836 36754 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2011137219 38(5-7) 53837 36755 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 12 53838 36756 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME ERYTHROPOIETIN EPOETIN BETA 11023508 53839 36757 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME IL-8 14530367 53840 36758 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME LIDOCAINE LIDOCAINE 12401608 53845 36759 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 249565741 MK-5108 53846 36760 ALDH1A1 216 DRUGGABLE GENOME, ENZYME AMBUNOL AMBUNOL 53847 36761 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NITROBLUE TETRAZOLIUM CHLORIDE NITROBLUE TETRAZOLIUM CHLORIDE 53848 36762 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME FLUORESCEIN DIACETATE FLUORESCEIN DIACETATE 53849 36763 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR HYDROGEN PEROXIDE 11145585 53851 36764 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Isosteric imidazolyl pyrimidine derivative 1 53852 36765 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TERFENADINE TERFENADINE 53853 36766 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CARMINE CARMINE 53857 36767 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME NAC ACETYLCYSTEINE 12031897 53858 36768 KDM4A 9682 DRUGGABLE GENOME, ENZYME XANTHURENATE XANTHURENATE 53861 36769 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME NSC-677436 CHEMBL120580 16998480 53862 36770 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AZINPHOS-ETHYL AZINPHOS-ETHYL 53863 36771 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650087 53864 36772 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AG-34 CHEMBL80155 53865 36773 BAZ2B 29994 NA AG-490 CHEMBL56543 53866 36774 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 53867 36775 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TOZASERTIB TOZASERTIB 53868 36776 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE JNJ-7706621 JNJ-7706621 53871 36777 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME ANESTHETIC AGENT 9585305 53873 36778 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MERCAPTOPURINE MERCAPTOPURINE 22931300 53874 36779 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-49789 CHEMBL469309 53875 36780 HLA-G 3135 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME hmg coa reductase inhibitors 53876 36781 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 178101927 53877 36782 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROMAZINE HYDROCHLORIDE PROMAZINE HYDROCHLORIDE 53878 36783 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Indoline derivative 14 53879 36784 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ALOE-EMODIN ALOE-EMODIN 53882 36785 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PF-477736 PF-00477736 26140595 53883 36786 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GW441756X GW441756X 53884 36787 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor SB939 53885 36788 CBX1 10951 NA TAXIFOLIN TAXIFOLIN 53886 36789 GMNN 51053 DRUGGABLE GENOME DULOXETINE DULOXETINE 53887 36790 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 4-TERT-BUTYLCATECHOL CHEMBL220845 53888 36791 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PENTAMIDINE DIISETHIONATE PENTAMIDINE ISETHIONATE 53889 36792 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PIMASERTIB PIMASERTIB 53891 36793 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME rucaparib RUCAPARIB 53892 36794 GMNN 51053 DRUGGABLE GENOME DNDI1417519 CHEMBL1402376 53893 36795 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME inhibitor CARFILZOMIB CARFILZOMIB 53895 36796 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LINIFANIB LINIFANIB 53896 36797 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME SPERMINE TRIS-2-NAPG CHEMBL2347633 23434419 53897 36798 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLOZAPINE CLOZAPINE 22931300 53899 36799 NDUFA7 4701 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 53901 36800 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 374883878 ABROCITINIB 53903 36801 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650152 CYPROHEPTADINE 53904 36802 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DIGOXIN DIGOXIN 53906 36803 POLI 11201 DNA REPAIR MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 53910 36804 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor 252827505 CHEMBL2159511 53911 36805 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME THALIDOMIDE THALIDOMIDE 7876469 53912 36806 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1200853 DYDROGESTERONE 53915 36807 ALOX5 240 DRUGGABLE GENOME, ENZYME zileuton ZILEUTON 53918 36808 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166767 53919 36809 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL antagonist 135651219 SURAMIN 53920 36810 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1201825 RANIBIZUMAB 53922 36811 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 53923 36812 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200434 OXTRIPHYLLINE 53924 36813 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL3545094 ELOCALCITOL 53926 36814 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102332 VATALANIB 53928 36815 IL1B 3553 KINASE, DRUGGABLE GENOME RALOXIFENE RALOXIFENE 12773123 53929 36816 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Pimasertib PIMASERTIB 23629727 53930 36817 MAPT 4137 DRUGGABLE GENOME D-DOPA CHEMBL211670 53931 36818 PSORS1C1 170679 NA allopurinol ALLOPURINOL 21801394,29193002 53933 36819 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CID 3237815 CHEMBL410484 53935 36820 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME METHAPYRILENE METHAPYRILENE 53936 36821 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR UREA UREA 3342876 53937 36822 ADAMTS5 11096 DRUGGABLE GENOME, ENZYME, PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE TUMOR NECROSIS FACTOR 11520168 53938 36823 POLI 11201 DNA REPAIR AG-538 CHEMBL56393 53939 36824 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1152 PREDNISOLONE ACETATE 53941 36825 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME LY3009120 LY-3009120 26343583 53942 36826 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME blocker 135650114 CLOTRIMAZOLE 53943 36827 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE L-741626 CHEMBL445102 53944 36828 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MIDODRINE MIDODRINE 22931300 53945 36829 CCNA2 890 DRUGGABLE GENOME, KINASE SELICICLIB SELICICLIB 21080703 53946 36830 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID30259754-Compound-pyrrole[2,3-d]azepines 53947 36831 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Demcizumab DEMCIZUMAB 26855149 53948 36832 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1200980 ESTROPIPATE 53949 36833 CBX1 10951 NA RUFINAMIDE RUFINAMIDE 53951 36834 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE DOVITINIB DOVITINIB 53953 36835 MAPT 4137 DRUGGABLE GENOME VU001171 CHEMBL515763 53954 36836 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER MILTEFOSINE MILTEFOSINE 11355955 53955 36837 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 2,3,3',4',5'-PENTAMETHOXYCHALCONE CHEMBL608862 20813535 53956 36838 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PENFLURIDOL PENFLURIDOL 53959 36839 ATXN2 6311 NA NELFINAVIR MESYLATE NELFINAVIR MESYLATE 53962 36840 CBX1 10951 NA TAMOXIFEN TAMOXIFEN 53963 36841 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor PLX3397 PEXIDARTINIB 53964 36842 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE IMATINIB IMATINIB 53966 36843 CA2 760 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201162 DORZOLAMIDE HYDROCHLORIDE 53967 36844 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-67 CHEMBL578512 53968 36845 KDM4A 9682 DRUGGABLE GENOME, ENZYME AG-527 CHEMBL258767 53970 36846 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE MPDL-3280A ATEZOLIZUMAB 24829850 53971 36847 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR DIHYDROSPHINGOSINE 10022508 53973 36848 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Volasertib VOLASERTIB 26597303 53974 36849 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE 6,6-fused nitrogenous heterocyclic compound 1 53975 36850 CP 1356 DRUGGABLE GENOME, ENZYME DES DIETHYLSTILBESTROL 1533964 53976 36851 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME DP-4088 53977 36852 ALOX15B 247 DRUGGABLE GENOME, ENZYME ZM-449829 CHEMBL154580 53978 36853 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 53980 36854 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor 178101399 53981 36855 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Dabrafenib DABRAFENIB 27797976 53982 36856 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125472 CHEMBL587389 53983 36857 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE TENOFOVIR TENOFOVIR 17172311 53984 36858 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR CGP41251 10463595 53986 36859 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Everolimus EVEROLIMUS 53987 36860 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME PMID27774824-Compound-Figure9Example2up 53993 36861 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SHIKONIN SHIKONIN 53995 36862 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-2936 CHEMBL582503 53997 36863 KDM6B 23135 ENZYME inhibitor 374883847 53998 36864 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 315661280 NAZARTINIB 54000 36865 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 lumefantrine LUMEFANTRINE 54001 36866 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM BROMIDE 54002 36867 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL932 DIPYRIDAMOLE 54003 36868 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor CHEMBL445813 AT-7519 54004 36869 TOP2B 7155 DRUGGABLE GENOME, ENZYME Fluoroquinolone 54006 36870 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE carbamazepine CARBAMAZEPINE 24384557,21738081,18695978,25495409,26421491,23252947 54007 36871 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GW501516 GW501516 23566516 54009 36872 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE TST10088 54011 36873 GMNN 51053 DRUGGABLE GENOME RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 54012 36874 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER TCMDC-123650 CHEMBL580727 54013 36875 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LASALOCID A SODIUM LASALOCID A SODIUM 54014 36876 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200341 INDECAINIDE HYDROCHLORIDE 54015 36877 CDH2 1000 CELL SURFACE, DRUGGABLE GENOME Exherin 54017 36878 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor DABRAFENIB MESYLATE 54018 36879 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2216870 IDELALISIB 54019 36880 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AMENTOFLAVONE AMENTOFLAVONE 54020 36881 UGT1A7 54577 DRUGGABLE GENOME, ENZYME atazanavir ATAZANAVIR 17058217 54022 36882 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BETA-LAPACHONE LAPACHONE 54023 36883 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Dasatinib DASATINIB 21689725,18024392,25594040,18986703,19671763,17699867,16397263,23582185 54024 36884 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME BUTYRYLHYDROXAMIC ACID BUTYRYLHYDROXAMIC ACID 21874153 54025 36885 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX Alitretinoin ALITRETINOIN 54026 36886 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor 223366167 E-6201 54028 36887 RORA 6095 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE agonist 310264687 54029 36888 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 363894210 PANULISIB 54030 36889 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GW843682X GW843682X 54032 36890 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651130 54033 36891 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING NAFRONYL OXALATE NAFRONYL OXALATE 54034 36892 TYMSOS 494514 NA hydroxychloroquine HYDROXYCHLOROQUINE 18322994 54036 36893 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Talazoparib TALAZOPARIB 23881923 54038 36894 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 187051782 ARFORMOTEROL 54039 36895 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME ROMIDEPSIN ROMIDEPSIN 54041 36896 MAPT 4137 DRUGGABLE GENOME CARMINOMYCIN CARUBICIN 54044 36897 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME RO5520985 54045 36898 TMEM97 27346 NA Piperazinyl methyl quinazolinone derivative 2 54046 36899 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE FLUNARIZINE DIHYDROCHLORIDE FLUNARIZINE DIHYDROCHLORIDE 54048 36900 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor IMATINIB IMATINIB 54049 36901 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2108739 PLACULUMAB 54054 36902 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 14 54055 36903 PECAM1 5175 NA RESVERATROL RESVERATROL 15041740 54056 36904 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMA 1827816 54058 36905 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ANTI-CANCER AGENTS 8509220 54061 36906 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CINOBUFOTALIN CINOBUFOTALIN 54062 36907 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32p 54065 36908 PTGS2 5743 DRUGGABLE GENOME, ENZYME MECLOFENAMIC ACID 54066 36909 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GEMFIBROZIL GEMFIBROZIL 54067 36910 GMNN 51053 DRUGGABLE GENOME METERGOLINE METERGOLINE 54068 36911 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME CENISERTIB CENISERTIB 54069 36912 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1201150 SUMATRIPTAN SUCCINATE 54070 36913 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE SJ000032151 CHEMBL592600 54071 36914 HLA-DQA1 3117 CLINICALLY ACTIONABLE Drugs For Treatment Of Tuberculosis 12359646 54072 36915 TH 7054 ENZYME, DRUGGABLE GENOME STREPTOZOCIN STREPTOZOCIN 2568957 54073 36916 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103092 ODANACATIB 54074 36917 GATA4 2626 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE ANTHRACYCLINES 12527808 54075 36918 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE UROKINASE-TYPE PLASMINOGEN ACTIVATOR 11865026 54076 36919 HEBP1 50865 DRUGGABLE GENOME Chalcone derivative 2 54078 36920 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor GDC-0980 APITOLISIB 54079 36921 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CB7969312 CHEMBL599255 54080 36922 MAPT 4137 DRUGGABLE GENOME APIGENIN APIGENIN 54081 36923 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME BAY-613606 CHEMBL541400 54082 36924 CCL21 6366 DRUGGABLE GENOME CALDARET HYDRATE 54083 36925 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650119 54084 36926 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR EUPAFOLIN EUPAFOLIN 54085 36927 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE pemetrexed PEMETREXED 54086 36928 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SHIKONIN SHIKONIN 54087 36929 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545396 BMS-690514 54088 36930 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE SORAFENIB SORAFENIB 54089 36931 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX HALOFUGINONE HALOFUGINONE 11874485 54091 36932 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor AMG 208 54092 36933 MVK 4598 KINASE, ENZYME inhibitor 135651491 54093 36934 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PYRIDABEN PYRIDABEN 54095 36935 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALPHA-TOCOPHEROL VITAMIN E 17029404 54096 36936 ATAD5 79915 NA EMETINE HYDROCHLORIDE EMETINE HYDROCHLORIDE 54099 36937 PDE5A 8654 ENZYME, DRUGGABLE GENOME Tadalafil TADALAFIL 54100 36938 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME CARBAMAZEPINE CARBAMAZEPINE 12402220 54101 36939 BRCA2 675 CLINICALLY ACTIONABLE OLAPARIB OLAPARIB 31157963,23346317,26510020,30345884,25366685,19553641,32343890,28792849,25218906,28578601,21862407,30797618,32043779,24882434 54102 36940 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor PANOBINOSTAT PANOBINOSTAT 54103 36941 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME PMID27841036-Compound-37 54104 36942 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NORELGESTROMIN NORELGESTROMIN 54105 36943 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Renzapride RENZAPRIDE 54107 36944 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFACON-1 54109 36945 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL activator 135652724 VERATRIDINE 54110 36946 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL408513 BELINOSTAT 54111 36947 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE VITAMIN D 12193704 54113 36948 POLK 51426 DNA REPAIR, ENZYME AMARANTH AMARANTH 54118 36949 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ANILERIDINE ANILERIDINE 54120 36950 CCR10 2826 DRUGGABLE GENOME, CELL SURFACE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135651679 54121 36951 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Trastuzumab TRASTUZUMAB 54122 36952 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME EMODIN EMODIN 54123 36953 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ETOPOSIDE ETOPOSIDE 8823806,9485461,8870683,9494516,9426516 54125 36954 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Pembrolizumab PEMBROLIZUMAB 28039262 54126 36955 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PROGESTERONE PROGESTERONE 54127 36956 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME E-2609 ELENBECESTAT 54129 36957 ALDH1A1 216 DRUGGABLE GENOME, ENZYME doxorubicin DOXORUBICIN 29938344 54130 36958 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CLONAZEPAM CLONAZEPAM 54131 36959 EIF2AK2 5610 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 178102572 54133 36960 ADGRL3 23284 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME methylphenidate METHYLPHENIDATE 25229170,29230023,22851411,25989180,20157310,22486528 54134 36961 KHK 3795 KINASE, ENZYME, DRUGGABLE GENOME fructose FRUCTOSE 24915143 54135 36962 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 135651283 TROGLITAZONE 54136 36963 ICA1 3382 NA o-desmethyltramadol 30971809 54141 36964 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FERBAM FERBAM 54143 36965 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FANETIZOLE FANETIZOLE 54146 36966 IL1B 3553 KINASE, DRUGGABLE GENOME PENTOXIFYLLINE PENTOXIFYLLINE 8048000 54147 36967 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 135652555 54148 36968 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW784684X GW784684X 54152 36969 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 2056784 CHEMBL261123 54153 36970 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME activator 404859003 54155 36971 CA9 768 DRUGGABLE GENOME, ENZYME CHEMBL3707280 CG250 111IN 54156 36972 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33e 54157 36973 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649644 54159 36974 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR THIRAM THIRAM 54160 36975 STX11 8676 NA Emapalumab-lzsg EMAPALUMAB 54163 36976 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PERICIAZINE PERICIAZINE 17606915 54164 36977 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 54165 36978 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR Indazoletriazolephenyl derivative 1 54166 36979 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME PRAVASTATIN PRAVASTATIN 17622941 54167 36980 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200953 HYDROCORTISONE PROBUTATE 54168 36981 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 363894197 CT-7001 54169 36982 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME letermovir LETERMOVIR 31022310 54170 36983 COMT 1312 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL953 ENTACAPONE 54172 36984 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE METHYLPREDNISOLONE METHYLPREDNISOLONE 17220550 54173 36985 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME activator 135650218 54174 36986 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE 3-CHLOROBENZOPEROXOIC ACID CHEMBL458855 18595691 54175 36987 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME SPC-3042 54176 36988 POLI 11201 DNA REPAIR PENTAMIDINE DIISETHIONATE PENTAMIDINE ISETHIONATE 54178 36989 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME RACEMETIROSINE RACEMETYROSINE 54179 36990 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PROTUBOXEPIN A PROTUBOXEPIN A 22595423 54180 36991 ITGB6 3694 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE GLPG0187 GLPG-0187 54181 36992 NDUFA1 4694 ENZYME inhibitor CHEMBL3545135 NV-128 54182 36993 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME T3D-959 DB959 54184 36994 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE venetoclax VENETOCLAX 54185 36995 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650169 54186 36996 MAOA 4128 DRUGGABLE GENOME, ENZYME 5-(2-PHENYLETHYL)ISATIN CHEMBL1642672 21134756 54187 36997 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL507361 PD-0325901 54188 36998 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-US20130053382 36(3-5) 54191 36999 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL1234354 PF-04691502 54193 37000 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL2017974 BUPARLISIB 54196 37001 TYMP 1890 GROWTH FACTOR, DRUGGABLE GENOME SULFASALAZINE SULFASALAZINE 15269287 54197 37002 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1230065 BMS-582949 54199 37003 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ROCURONIUM BROMIDE ROCURONIUM BROMIDE 54200 37004 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BMS-986205 LINRODOSTAT 54201 37005 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE crizotinib CRIZOTINIB 22162641 54202 37006 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME MTOR KINASE INHIBITOR AZD8055 27279227 54205 37007 MAP3K10 4294 SERINE THREONINE KINASE, ENZYME, KINASE, DRUGGABLE GENOME PF-562271 PF-00562271 54206 37008 GLS 2744 ENZYME CB-839 TELAGLENASTAT 54207 37009 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME BUDESONIDE BUDESONIDE 7716352 54210 37010 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051799 DACINOSTAT 54212 37011 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Bicyclic heteroaryl amide derivative 1 54214 37012 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 223366146 DILMAPIMOD 54215 37013 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652468 54217 37014 TUBA3D 113457 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 54220 37015 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor AZD6244 SELUMETINIB 54221 37016 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE CARBIMAZOLE CARBIMAZOLE 54222 37017 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE EPINEPHRINE EPINEPHRINE 54223 37018 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651132 54224 37019 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Tripelennamine TRIPELENNAMINE 54226 37020 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Amlexanox AMLEXANOX 27287717 54227 37021 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US9434725, 285 54228 37022 GMNN 51053 DRUGGABLE GENOME SJ000032150 CHEMBL607140 54229 37023 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER efavirenz EFAVIRENZ 20662624,24497997,31628422,12545140,27045425,20860463,11809184,26774523,23734829,20720517,20625352,16267764,25303294,16912956 54231 37024 PSMC5 5705 TRANSCRIPTION FACTOR BINDING, PROTEASE inhibitor CHEMBL325041 BORTEZOMIB 54233 37025 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR LEAD DIACETATE TRIHYDRATE LEAD DIACETATE TRIHYDRATE 54234 37026 TSPO 706 DRUGGABLE GENOME PMID27599163-Compound-81 54235 37027 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor BMS-777607 BMS-777607 54238 37028 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor BAFETINIB BAFETINIB 54239 37029 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ARI-3037MO 54240 37030 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Trafermin TRAFERMIN 54242 37031 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR VAN-10-4-eluting stent 54243 37032 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 252827451 SAR-260301 54244 37033 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TETROQUINONE TETROQUINONE 54245 37034 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 6-OXIMOTRYPTANTHRIN CHEMBL308106 20373766 54248 37035 GLS 2744 ENZYME TCMDC-123723 CHEMBL525103 54249 37036 CD37 951 DRUGGABLE GENOME antibody 374883836 54250 37037 IL1B 3553 KINASE, DRUGGABLE GENOME antibody CANAKINUMAB CANAKINUMAB 54251 37038 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME JUGLONE JUGLONE 54252 37039 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE MGCD265 GLESATINIB 54253 37040 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL428647 PACLITAXEL 54255 37041 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE US9567304, Compound F-54 54256 37042 LPAR2 9170 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135649931 54257 37043 SMN1 6606 DRUGGABLE GENOME HOE-33342 CHEMBL343002 54258 37044 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME FLUDIAZEPAM FLUDIAZEPAM 54260 37045 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL ENFLURANE ENFLURANE 54264 37046 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-28620 CHEMBL1414990 22524450 54265 37047 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 10-(4-PYRIDYL)CAMPTOTHECIN CHEMBL1762593 21333532 54266 37048 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE 7-azaindole derivative 3 54267 37049 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DEXAMETHASONE DEXAMETHASONE 54268 37050 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME MLN8237 54270 37051 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE TOZASERTIB TOZASERTIB 54271 37052 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME DB-959 DB959 54272 37053 HEBP1 50865 DRUGGABLE GENOME 2-hydroxybenzamide derivative 1 54275 37054 ABHD6 57406 PHOSPHOLIPASE, ENZYME Piperazine carbamic compound 5 54276 37055 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Epoxysuccinate derivative 2 54277 37056 ITPA 3704 ENZYME azathioprine AZATHIOPRINE 26674571,16431304,21961091,18616518,18662289,15973722,19129747 54278 37057 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL240597 CHENODIOL 54279 37058 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CADMIUM ACETATE CADMIUM ACETATE 54280 37059 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor SORAFENIB TOSYLATE 54282 37060 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE inhibitor CHEMBL2109252 FORALUMAB 54283 37061 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651537 54284 37062 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LACTIC ACID LACTIC ACID 54285 37063 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZAPA ZAPA 54288 37064 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE Sorafenib SORAFENIB 54289 37065 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE METHOTREXATE METHOTREXATE 54290 37066 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 328083485 OSI-930 54291 37067 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Bavencio AVELUMAB 54292 37068 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME DICLOFENAC DICLOFENAC 9544613 54293 37069 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR MT203 NAMILUMAB 54294 37070 POLI 11201 DNA REPAIR GALUTEOLIN GALUTEOLIN 54295 37071 GMNN 51053 DRUGGABLE GENOME PROROXAN PROROXAN 54297 37072 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE NILOTINIB NILOTINIB 28720666,26424760,17372901,19671763,17699867 54298 37073 BRCA2 675 CLINICALLY ACTIONABLE Chlorambucil CHLORAMBUCIL 25193512 54299 37074 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SB-202190 SB-202190 54300 37075 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TAE-684 TAE-684 54301 37076 PDHX 8050 KINASE ANTIOXIDANT 14607783 54302 37077 CXCL8 3576 DRUGGABLE GENOME 13-CIS-RETINAL CHEMBL1579130 54303 37078 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHOLECALCIFEROL CHOLECALCIFEROL 54304 37079 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SANGUINARIUM SANGUINARIUM 54305 37080 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL970 HALAZEPAM 54306 37081 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 310264790 JNJ-42165279 54307 37082 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR YT-146 54308 37083 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL3545021 ANLOTINIB 54309 37084 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-125567 CHEMBL530049 54310 37085 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 178102310 54311 37086 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME docetaxel DOCETAXEL 25111199,24061601,26100253 54312 37087 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Tamsulosin TAMSULOSIN 54313 37088 MAPT 4137 DRUGGABLE GENOME DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 54314 37089 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE modulator CHEMBL3542265 LY2452473 54315 37090 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PURPUROGALLIN PURPUROGALLIN 54318 37091 HBB 3043 DRUGGABLE GENOME, ENZYME AES-103 AES-103 54319 37092 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL2103852 CROLIBULIN 54320 37093 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 cotinine COTININE 54322 37094 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1236962 OMIPALISIB 54323 37095 PSMC5 5705 TRANSCRIPTION FACTOR BINDING, PROTEASE BORTEZOMIB BORTEZOMIB 24524217 54324 37096 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME Ticlopidine TICLOPIDINE 54326 37097 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PS433540 54328 37098 SAA1 6288 DRUGGABLE GENOME IL-1RA ANAKINRA 1717568 54330 37099 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL2105682 EDOXABAN TOSYLATE 54334 37100 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 385612234 54335 37101 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME 178101232 54336 37102 CFB 629 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 404859157 54337 37103 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Dabigatran DABIGATRAN 32564268 54338 37104 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME TG-4010 54339 37105 NR2F2 7026 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME RESACTIN A RESACTIN A 54340 37106 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME ALVOCIDIB ALVOCIDIB 54341 37107 ALOX5 240 DRUGGABLE GENOME, ENZYME activator 178101873 54342 37108 HSPA4 3308 NA ENALAPRIL ENALAPRIL 12047041 54343 37109 HMGCR 3156 ENZYME, DRUGGABLE GENOME Atorvastatin lactole derivative 1 54344 37110 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ADEFOVIR DIPIVOXIL ADEFOVIR DIPIVOXIL 54345 37111 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE GNF-PF-1852 CHEMBL533293 54348 37112 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR antagonist 178102078 SULINDAC 54351 37113 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 336446964 54352 37114 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE METHYLPREDNISOLONE METHYLPREDNISOLONE 8976974 54353 37115 USP1 7398 DNA REPAIR, PROTEASE, ENZYME AC-55649 CHEMBL425027 54354 37116 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-28 54355 37117 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BCT303 54356 37118 SMN1 6606 DRUGGABLE GENOME AG-494 CHEMBL56731 54357 37119 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Cobimetinib COBIMETINIB 54359 37120 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 14-[(N-TETRADECYLAMIDO)SUCCINYL]DOXORUBICIN CHEMBL2023733 22276998 54360 37121 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Rizatriptan RIZATRIPTAN 54361 37122 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102609 54362 37123 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (R)-PROCYCLIDINE (R)-PROCYCLIDINE 54363 37124 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 54364 37125 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR STAUROSPORINE STAUROSPORINE 11035812 54365 37126 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor 178103971 IBUDILAST 54367 37127 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME INDIRUBIN-3'-MONOXIME CHEMBL1082552 16680159 54369 37128 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLOROTHALONIL CHLOROTHALONIL 54370 37129 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME inhibitor 249565876 54371 37130 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE DOXORUBICIN DOXORUBICIN 16749867 54372 37131 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME O6-BENZYLGUANINE 6-O-BENZYLGUANINE 7503788 54373 37132 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME RG-1530 RG-1530 54374 37133 TARDBP 23435 TUMOR SUPPRESSOR DNDI1417443 CHEMBL1553566 54375 37134 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR CYC-116 CYC-116 54377 37135 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME BAY-613606 CHEMBL541400 54378 37136 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME BISPECIFIC ANTIBODY 10928069 54379 37137 ATAD5 79915 NA WIN-62577 CHEMBL1256845 54381 37138 NUP107 57122 TRANSPORTER Platinum compounds 28562428 54382 37139 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 178102612 54384 37140 ATXN2 6311 NA SJ000114961 CHEMBL590168 54385 37141 ALOX5 240 DRUGGABLE GENOME, ENZYME TA-270 54386 37142 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL celecoxib CELECOXIB 22336956 54388 37143 BCHE 590 DRUGGABLE GENOME, ENZYME DONEPEZIL DONEPEZIL 15989517,16083542 54389 37144 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1240 PROPANTHELINE BROMIDE 54390 37145 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor PONATINIB PONATINIB 54392 37146 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3360203 PILARALISIB 54395 37147 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR OLSALAZINE OLSALAZINE 54396 37148 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR DEL-22379 DEL-22379 26267534 54397 37149 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR KAEMPFEROL KAEMPFEROL 25190466 54398 37150 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 1540545 CHEMBL259784 54399 37151 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME ICA-69673 19949402 54400 37152 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE irinotecan IRINOTECAN 16636344,23386248,12181437,18221820 54401 37153 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE Cycloserine CYCLOSERINE 54403 37154 ATXN2 6311 NA NIFEDIPINE NIFEDIPINE 54404 37155 PSMC5 5705 TRANSCRIPTION FACTOR BINDING, PROTEASE inhibitor CHEMBL3545432 IXAZOMIB CITRATE 54405 37156 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100670 54406 37157 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody CATUMAXOMAB CATUMAXOMAB 54407 37158 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178103844 PHENYLBUTAZONE 54408 37159 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE VINCRISTINE VINCRISTINE 12576455 54410 37160 F7 2155 ENZYME, DRUGGABLE GENOME, PROTEASE BAX-817 54412 37161 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME METHYLPHENIDATE METHYLPHENIDATE 54414 37162 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Pepticlere 54416 37163 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE IOPAMIDOL IOPAMIDOL 54417 37164 GMNN 51053 DRUGGABLE GENOME CHLOROXINE CHLOROXINE 54420 37165 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER G-CSF FILGRASTIM 7564516 54421 37166 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CHEMBL1102 GLUTETHIMIDE 54422 37167 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL inhibitor 135650057 CARVEDILOL 54423 37168 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME BDBM50011552 54424 37169 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 187051807 SCRIPTAID 54425 37170 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR STREPTOZOTOCIN STREPTOZOCIN 15016184,11937525 54426 37171 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-5029 CHEMBL600360 54427 37172 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL552212 LEXIBULIN 54428 37173 LAMA5 3911 DRUGGABLE GENOME RBC 9763582 54429 37174 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000044511 CHEMBL592124 54431 37175 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME BAY 94-9343 54432 37176 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102550 54433 37177 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Ace Inhibitors, Plain 22543981 54434 37178 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-13 54435 37179 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Epinephrine EPINEPHRINE 54436 37180 RBP4 5950 DRUGGABLE GENOME US8586571, 12 54437 37181 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE MUROMONAB MUROMONAB-CD3 54438 37182 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CYPROHEPTADINE CYPROHEPTADINE 54439 37183 CBX1 10951 NA SB-242084 SB-242084 54441 37184 GPD2 2820 DRUGGABLE GENOME HYDROGEN PEROXIDE 15209538 54443 37185 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MESALAMINE MESALAMINE 54444 37186 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GW501516 GW501516 23566516 54445 37187 SLC16A1 6566 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 252827471 54446 37188 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Vadimezan VADIMEZAN 54447 37189 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ANTITHYMOCYTE GLOBULIN 8970608,9389690 54448 37190 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GNF-PF-2298 CHEMBL578905 54449 37191 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR XP-23829 54450 37192 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650456 LEXACALCITOL 54451 37193 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME SORAFENIB SORAFENIB 54452 37194 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ENCLOMIPHENE ENCLOMIPHENE 54454 37195 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME SNS-314 SNS-314 54455 37196 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE MS417 26058079 54456 37197 CBX1 10951 NA AMBUNOL AMBUNOL 54457 37198 DNER 92737 NA PMID26924192-Compound-52 54458 37199 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GO-Y022 CHEMBL128729 23742639 54460 37200 ALOX15 246 ENZYME, DRUGGABLE GENOME 2-AMINOETHOXYDIPHENYL BORATE CHEMBL169233 54462 37201 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME MMV000704 CHEMBL582478 54463 37202 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHEMBL2068724 ACAMPROSATE CALCIUM 54464 37203 BRPF3 27154 DRUGGABLE GENOME 336446909 54465 37204 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135650768 54466 37205 SLC15A1 6564 DRUGGABLE GENOME, TRANSPORTER fluvastatin FLUVASTATIN 54467 37206 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 328083496 IPRAGLIFLOZIN 54468 37207 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE METHADONE METHADONE 54469 37208 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-9 54470 37209 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3544956 PYROTINIB 54471 37210 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ARFORMOTEROL ARFORMOTEROL 54472 37211 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE GEFITINIB GEFITINIB 23993328 54473 37212 HDC 3067 DRUGGABLE GENOME, ENZYME inhibitor 178101826 54474 37213 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME inhibitor CHEMBL3039522 BIRINAPANT 54475 37214 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE VENETOCLAX VENETOCLAX 31004028,30514704,31951646,32232486,31160589,31234236 54477 37215 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 VALERIAN VALERIAN 17214607 54479 37216 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER 7-DEOXYPACLITAXEL CHEMBL203365 16271474 54480 37217 PSMD2 5708 NA BORTEZOMIB BORTEZOMIB 24524217 54481 37218 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME RAC-ARISTOYUNNOLIN D CHEMBL2333543 54482 37219 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 135652187 54483 37220 SMN1 6606 DRUGGABLE GENOME 4-BENZYLOXYANILINE 4-BENZYLOXYANILINE 54485 37221 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 piroxicam PIROXICAM 16198655,17112811 54487 37222 HLA-DQB1 3119 CLINICALLY ACTIONABLE clavulanate CLAVULANIC ACID 10535882,30664875 54488 37223 POLI 11201 DNA REPAIR BETA-LAPACHONE LAPACHONE 54489 37224 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Esterified estrogens 54490 37225 GCLC 2729 DRUGGABLE GENOME, ENZYME ANTIOXIDANT 15485876 54491 37226 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-49 54492 37227 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LIPOSOMAL DOXORUBICIN 54493 37228 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE CI-1040 CI-1040 54494 37229 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AMPIROXICAM AMPIROXICAM 54496 37230 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME fludarabine FLUDARABINE 22584460 54497 37231 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Rituxan Hemotalogy/oncology 54498 37232 FUS 2521 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ATRA TRETINOIN 10691862 54500 37233 MDH2 4191 NA CISPLATIN CISPLATIN 15225672 54502 37234 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TETRABROMOBENZOTRIAZOLE TETRABROMOBENZOTRIAZOLE 54503 37235 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE LIPIDYL PSEUDOPTERANE A LIPIDYL PSEUDOPTERANE A 19061360 54504 37236 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ALVOCIDIB ALVOCIDIB 54505 37237 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME rosuvastatin ROSUVASTATIN 22331829,23930675,16784736,20207952,20679960,25630984,20130569,28322941,19474787,18617601 54506 37238 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 310264675 CUDC-101 54508 37239 IFI27 3429 NUCLEAR HORMONE RECEPTOR RETINOIDS 15086558 54509 37240 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE RESVERATROL RESVERATROL 16084059 54511 37241 BCL2L2 599 CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL2107358 OBATOCLAX MESYLATE 54512 37242 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650303 54514 37243 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME CAMPTOTHECIN CAMPTOTHECIN 16211302 54515 37244 IRF1-AS1 441108 NA hydrochlorothiazide HYDROCHLOROTHIAZIDE 31327267 54516 37245 GUCY2C 2984 DRUGGABLE GENOME, KINASE ISIS-GCCRrx 54517 37246 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CYC-116 CYC-116 54523 37247 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME activator 135652752 54524 37248 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 223366064 SARACATINIB 54525 37249 AKR1B1 231 DRUGGABLE GENOME, ENZYME CONTIGOSIDE B 54527 37250 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-102029 CHEMBL74913 54529 37251 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-6 54530 37252 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL27759 ENTINOSTAT 54531 37253 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ENMD-2076 ENMD-2076 54536 37254 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE AST-487 AST-487 54537 37255 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR CHONDROITIN 7974391 54538 37256 MAPT 4137 DRUGGABLE GENOME TCMDC-124422 CHEMBL527620 54539 37257 CBX1 10951 NA NAFTOPIDIL NAFTOPIDIL 54540 37258 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1082607 SALMETEROL XINAFOATE 54541 37259 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651393 54542 37260 TESK1 7016 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565798 54543 37261 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-14 54544 37262 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 363894180 54548 37263 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME PEGAPTANIB PEGAPTANIB SODIUM 54549 37264 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHENTOLAMINE PHENTOLAMINE 54552 37265 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE VER-49009 CHEMBL365617 54553 37266 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME yohimbine YOHIMBINE 15289791 54554 37267 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1614713 CC-401 54555 37268 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Bicyclic heteroaryl amide derivative 3 54556 37269 APBA1 320 NA NSC-180246 CHEMBL484640 54557 37270 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652255 LABRADIMIL 54559 37271 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME antisense oligonucleotide AFFINITAC APRINOCARSEN 54562 37272 DUSP1 1843 PROTEIN PHOSPHATASE, KINASE, DRUGGABLE GENOME salbutamol ALBUTEROL 20673984 54563 37273 PDHB 5162 ENZYME DEXLIPOTAM 54567 37274 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BETAXOLOL BETAXOLOL 54570 37275 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 404859126 BKT140 54573 37276 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME QUAZEPAM QUAZEPAM 54576 37277 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL568 OXAZEPAM 54578 37278 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GRACILIN A GRACILIN A 19601607 54579 37279 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 1 54581 37280 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR ALISERTIB ALISERTIB 54583 37281 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE PF-562271 PF-00562271 54584 37282 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR cyclophosphamide CYCLOPHOSPHAMIDE 19786980,22188361 54585 37283 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TRIFLUPROMAZINE TRIFLUPROMAZINE 54587 37284 DIABLO 56616 NA CASPASE INHIBITOR 12823542,15843890 54592 37285 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE DORSOMORPHIN DORSOMORPHIN 54593 37286 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER VINCA ALKALOIDS 11850258 54594 37287 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE GW441756X GW441756X 54595 37288 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Quinoline carboxamide derivative 1 54599 37289 NME1 4830 KINASE adefovir dipivoxil 54600 37290 NOS2 4843 DRUGGABLE GENOME, ENZYME inhibitor 252827417 54604 37291 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ARISTOLACTONE ARISTOLACTONE 54605 37292 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 329968397 CHEMBL494303 54607 37293 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE GDC-0973 COBIMETINIB 54608 37294 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DAUNORUBICIN DAUNORUBICIN 22260166 54609 37295 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE PTC299 54611 37296 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE allosteric modulator 252166534 54614 37297 NOS1 4842 DRUGGABLE GENOME, ENZYME epirubicin EPIRUBICIN 54615 37298 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 340590241 54616 37299 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE inhibitor 178103390 TACROLIMUS 54617 37300 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Indazoletriazolephenyl derivative 2 54619 37301 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor LY2940680 54620 37302 USP1 7398 DNA REPAIR, PROTEASE, ENZYME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 54621 37303 CD3D 915 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE inhibitor CHEMBL2109252 FORALUMAB 54622 37304 MBNL1 4154 DRUGGABLE GENOME NOREPINEPHRINE NOREPINEPHRINE 54624 37305 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 354702272 SELETALISIB 54625 37306 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200710 CLOMIPRAMINE HYDROCHLORIDE 54626 37307 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE IMATINIB IMATINIB 19755855,15928335,21818111,12944919,12949711,12660384,25658984,14504092,26130666,24132921,16954519,24456122 54627 37308 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME iloperidone ILOPERIDONE 23277250 54628 37309 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME PMID25399719-Compound-17 54629 37310 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 54631 37311 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR NPC-01 54632 37312 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545085 XL-228 54633 37313 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 9 54635 37314 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178102585 DOVITINIB 54637 37315 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TCMDC-125625 CHEMBL549208 54638 37316 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME GNF-PF-4068 CHEMBL584668 54639 37317 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1200436 OXANDROLONE 54640 37318 ABCC9 10060 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER Nicorandil NICORANDIL 54641 37319 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor SF1126 54642 37320 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE DOVITINIB DOVITINIB 54643 37321 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor PLX3397 PEXIDARTINIB 54645 37322 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CARTEOLOL CARTEOLOL 54646 37323 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 384403645 54647 37324 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE infliximab INFLIXIMAB 19005160,25823782,24048425,27044681 54648 37325 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Cetuximab CETUXIMAB 22586653,26296355,21900593,23948973,26243863 54650 37326 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SJ000281118 CHEMBL592561 54651 37327 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME ILORASERTIB ILORASERTIB 54652 37328 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 XANTHINE AMINE CONGENER XANTHINE AMINE CONGENER 54653 37329 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HARMALOL HARMALOL 54654 37330 SCNN1G 6340 ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE blocker CHEMBL1398126 AMILORIDE HYDROCHLORIDE 54655 37331 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PROTOPORPHYRIN PROTOPORPHYRIN 54656 37332 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TRICLOSAN TRICLOSAN 54658 37333 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME KENPAULLONE KENPAULLONE 54659 37334 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR THEONELLASTEROL E THEONELLASTEROL E 21428459 54660 37335 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ACETAMINOPHEN ACETAMINOPHEN 22931300 54661 37336 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-254 CHEMBL461579 54662 37337 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL272980 MOCETINOSTAT 54664 37338 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ENOBOSARM ENOBOSARM 54666 37339 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545365 ALTIRATINIB 54668 37340 KLC3 147700 NA cisplatin CISPLATIN 19434073,22188361,29662106,22026922,21449681 54670 37341 PRKAG2 51422 ENZYME, KINASE metformin METFORMIN 22722338 54671 37342 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 danazol DANAZOL 19923256 54672 37343 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 178102445 TREPROSTINIL 54674 37344 B4GALT2 8704 ENZYME aspirin ASPIRIN 54676 37345 IL1A 3552 CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL2109653 BERMEKIMAB 54677 37346 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE AZD-1152-HQPA AZD-1152-HQPA 54678 37347 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME BERKELEYACETAL C BERKELEYACETAL C 17970594 54679 37348 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME (E)-DIBENZYLIDENEACETONE CHEMBL17201 54680 37349 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ARISTOLOCHIC ACID ARISTOLOCHIC ACID 54681 37350 LGR4 55366 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100587 54687 37351 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER FAS LIGAND 14614330 54690 37352 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 Y-27632 Y-27632 54691 37353 POLK 51426 DNA REPAIR, ENZYME NSC-119889 CHEMBL516616 54692 37354 PTGS1 5742 ENZYME, DRUGGABLE GENOME NEPAFENAC NEPAFENAC 54693 37355 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CYTARABINE CYTARABINE 22931300 54694 37356 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ACACETIN ACACETIN 54695 37357 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME Methoxy polyethylene glycol-epoetin beta 54696 37358 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-123951 CHEMBL587849 54698 37359 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SERTINDOLE SERTINDOLE 54700 37360 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME antagonist 178100992 DANTROLENE 54701 37361 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DEBRISOQUIN DEBRISOQUIN 54702 37362 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Tubastatin A 25957812 54703 37363 NDUFB7 4713 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 54704 37364 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrazolo[4,3-c]pyridine derivative 2 54705 37365 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME EBSELEN EBSELEN 54707 37366 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ISOQUERCETIN ISOQUERCETIN 54708 37367 TAC1 6863 DRUGGABLE GENOME 8-MOP METHOXSALEN 9430496 54710 37368 FXYD2 486 DRUGGABLE GENOME, TRANSPORTER CYCLOTHIAZIDE CYCLOTHIAZIDE 54711 37369 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 clomipramine CLOMIPRAMINE 9187528 54713 37370 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME dapsone DAPSONE 29233746 54714 37371 PXN 5829 NA 1,2,4,5-BENZENETETRAAMINE TETRAHYDROCHLORIDE CHEMBL456559 18989950 54715 37372 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor DASATINIB DASATINIB 54716 37373 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Latanoprost LATANOPROST 54718 37374 GMNN 51053 DRUGGABLE GENOME SU-6656 CHEMBL605003 54723 37375 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MECHLORETHAMINE HYDROCHLORIDE MECHLORETHAMINE HYDROCHLORIDE 54724 37376 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ORSELLINIC ACID, ETHYL ESTER ORSELLINIC ACID, ETHYL ESTER 54727 37377 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CERIVASTATIN SODIUM CERIVASTATIN SODIUM 54728 37378 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR HYDROXYUREA HYDROXYUREA 54729 37379 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOCOPHEROL ACETATE TOCOPHEROL ACETATE 54730 37380 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE STREPTOZOTOCIN STREPTOZOCIN 16741044 54731 37381 AGBL4 84871 PROTEASE, DRUGGABLE GENOME ustekinumab USTEKINUMAB 27977334 54732 37382 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-125544 CHEMBL533602 54733 37383 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE ANTIOXIDANT 12633939 54736 37384 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1715 PIOGLITAZONE HYDROCHLORIDE 54737 37385 POLI 11201 DNA REPAIR NSC-155693 CHEMBL68096 54738 37386 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PYRAFLUFEN-ETHYL PYRAFLUFEN-ETHYL 54739 37387 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Aromatic bicyclic compound 6 54740 37388 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1200934 NORGESTIMATE 54741 37389 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER antidepressants 18215618,26704739,22641028 54743 37390 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR XL550 XL550 54744 37391 BAZ2B 29994 NA TCMDC-125536 CHEMBL528463 24304323 54748 37392 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME GENTAMICIN GENTAMICIN 9249592 54749 37393 ALPI 248 DRUGGABLE GENOME, ENZYME SULFURETIN SULFURETIN 54750 37394 ATP1B3 483 ENZYME, TRANSPORTER, DRUGGABLE GENOME inhibitor CHEMBL1751 DIGOXIN 54752 37395 ATAD5 79915 NA GNF-PF-3407 CHEMBL602990 54753 37396 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 223366154 54754 37397 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME OPIOIDS 10232386 54756 37398 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Unii-R228S06soh 54759 37399 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CH5132799 PA-799 21558396 54760 37400 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME PTC299 54762 37401 POLG 5428 ENZYME valproic acid 23448099,21357833,21686371,21455106,21038416,19054397,18208989,20138553 54763 37402 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker CHEMBL41355 EZOGABINE 54764 37403 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TYRPHOSTIN 1 TYRPHOSTIN 1 54766 37404 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE OSI-632 OSI-632 54768 37405 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR INSULIN INSULIN 9299565,16650607 54769 37406 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 sulfonamides, urea derivatives 29681852,24442125,19794412 54770 37407 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 6-9 54771 37408 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650115 CLOZAPINE 54772 37409 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BAICALEIN BAICALEIN 54774 37410 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 135651277 54776 37411 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME ITI-007 LUMATEPERONE 54777 37412 CYB5R3 1727 DRUGGABLE GENOME, ENZYME dapsone DAPSONE 54778 37413 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEFOTETAN CEFOTETAN 54779 37414 HLA-E 3133 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE methotrexate METHOTREXATE 54781 37415 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME BETAMETHASONE BETAMETHASONE 3896398 54783 37416 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-125561 CHEMBL526763 54784 37417 LIMK2 3985 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565799 54785 37418 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME MITONAFIDE MITONAFIDE 54787 37419 PLIN3 10226 NA GALSULFASE GALSULFASE 54788 37420 CDK14 5218 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME inhibitor CHEMBL3544942 RONICICLIB 54789 37421 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 178102337 SORAFENIB 54790 37422 PSMD1 5707 NA inhibitor CHEMBL2103884 OPROZOMIB 54793 37423 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 187051798 BELINOSTAT 54794 37424 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 310264763 54795 37425 RAPGEF3 10411 ENZYME GYROPHORIC ACID GYROPHORIC ACID 54797 37426 ILF3 3609 KINASE, TRANSCRIPTION FACTOR IL-2 ALDESLEUKIN 12504009 54798 37427 TSPO 706 DRUGGABLE GENOME TLN-4601 DIAZEPINOMICIN 54800 37428 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651540 54801 37429 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ILORASERTIB ILORASERTIB 54803 37430 ADK 132 DRUGGABLE GENOME, ENZYME, KINASE 2',3'-DIDEOXYINOSINE 3262616 54804 37431 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR VOLVALERENAL D VOLVALERENAL D 54805 37432 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-E2 54806 37433 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ZAPA ZAPA 54809 37434 PSMD7 5713 PROTEASE inhibitor CHEMBL451887 CARFILZOMIB 54810 37435 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL BIIB095 54813 37436 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 310264720 54814 37437 CLCN3 1182 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE, TRANSPORTER blocker 178101102 PHLORETIN 54816 37438 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE CRENOLANIB CRENOLANIB 15928335,15685537,22718859,16638875,15146165,12949711,26130666,25157968,24132921,14645423,16954519,18794084,22745105 54817 37439 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE EMZ701 54818 37440 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1201659 CHLORPHENIRAMINE POLISTIREX 54819 37441 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100386 CHEMBL234940 54820 37442 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200982 BUTABARBITAL SODIUM 54821 37443 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SH-1242 26645561 54822 37444 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103673 PENTOXIFYLLINE 54823 37445 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE INDACATEROL INDACATEROL 54824 37446 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME chlorpheniramine CHLORPHENIRAMINE 54826 37447 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2392545 TAK-960 54828 37448 PDE5A 8654 ENZYME, DRUGGABLE GENOME THEOPHYLLINE THEOPHYLLINE 54829 37449 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIHYDROERGOCRISTINE DIHYDROERGOCRISTINE 54831 37450 RACGAP1 29127 NA BAS 01152706 CHEMBL2002487 54832 37451 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CETYLPYRIDINIUM CETYLPYRIDINIUM 54833 37452 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Hydroxy amidine derivative 1 54834 37453 MAOB 4129 DRUGGABLE GENOME, ENZYME MOCLOBEMIDE MOCLOBEMIDE 21680183 54835 37454 PSMB3 5691 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL371405 MARIZOMIB 54836 37455 MUC2 4583 DRUGGABLE GENOME IFN 16504136 54837 37456 TARDBP 23435 TUMOR SUPPRESSOR DNDI1417085 CHEMBL1522984 54838 37457 DNER 92737 NA Isoxazole-based bicyclic compound 9 54840 37458 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DESOXIMETASONE DESOXIMETASONE 54842 37459 PRRC2A 7916 NA gemcitabine GEMCITABINE 31616045 54845 37460 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE DCCCyB 24900218 54846 37461 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 310264699 SAMOTOLISIB 54848 37462 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649720 CHEMBL1208085 54849 37463 MAOB 4129 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 1 54851 37464 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 252827442 SGI-1776 54853 37465 FBXW7 55294 DNA REPAIR, CLINICALLY ACTIONABLE Entinostat ENTINOSTAT 23274910 54855 37466 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545311 BRIGATINIB 54856 37467 SULT1C4 27233 ENZYME docetaxel DOCETAXEL 20038957 54857 37468 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Pyridostigmine PYRIDOSTIGMINE 54858 37469 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME EBSELEN EBSELEN 54862 37470 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR aspirin ASPIRIN 54863 37471 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE FENTANYL FENTANYL 54864 37472 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652213 54866 37473 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Everolimus EVEROLIMUS 27683183 54867 37474 TNFRSF1B 7133 DRUGGABLE GENOME etanercept ETANERCEPT 30075559 54869 37475 GMNN 51053 DRUGGABLE GENOME GNF-PF-108 CHEMBL578929 54872 37476 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL521851 PICTILISIB 54873 37477 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LEFLUNOMIDE LEFLUNOMIDE 54875 37478 NF2 4771 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, DRUG RESISTANCE, KINASE TEMSIROLIMUS TEMSIROLIMUS 25878190 54876 37479 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME AMD3100 PLERIXAFOR 11581376 54877 37480 CCNK 8812 KINASE cyclophosphamide CYCLOPHOSPHAMIDE 54880 37481 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CAFFEINE CAFFEINE 54881 37482 PGA3 643834 PROTEASE, DRUGGABLE GENOME, ENZYME SUCRALFATE SUCRALFATE 54883 37483 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME LEVONORDEFRIN LEVONORDEFRIN 54884 37484 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL TOPIRAMATE TOPIRAMATE 54885 37485 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3707183 QUINIDINE SULFATE 54887 37486 FST 10468 DRUGGABLE GENOME BRDU 16543675 54889 37487 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CHR-3996 NANATINOSTAT 54890 37488 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER anastrozole ANASTROZOLE 54893 37489 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW282974X GW282974X 54894 37490 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TCMDC-135909 CHEMBL453384 19284751 54895 37491 POLK 51426 DNA REPAIR, ENZYME PURPUROGALLIN PURPUROGALLIN 54896 37492 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE MK-1775 ADAVOSERTIB 28652249 54898 37493 SMN2 6607 DRUGGABLE GENOME N-(4-NITROPHENYL)ANTHRANILIC ACID CHEMBL1574420 54899 37494 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor XL228 XL-228 54901 37495 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NAPHTHOQUINONE NAPHTHOQUINONE 54902 37496 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR carbamazepine CARBAMAZEPINE 24384557,28837897 54904 37497 PSMA3 5684 PROTEASE, DRUGGABLE GENOME CARFILZOMIB CARFILZOMIB 24524217 54905 37498 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US8975409, Comparative compound B 54907 37499 AKR1C1 1645 DRUGGABLE GENOME, ENZYME 3,5-DIBROMOSALICYLIC ACID CHEMBL447448 19397269 54908 37500 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Testogen TDS 54909 37501 USP1 7398 DNA REPAIR, PROTEASE, ENZYME BITHIONOL BITHIONOL 54910 37502 GMNN 51053 DRUGGABLE GENOME PHENAMIL METHANESULFONATE PHENAMIL METHANESULFONATE 54911 37503 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 223366058 54914 37504 TXN2 25828 DRUGGABLE GENOME, THIOREDOXIN GAMBOGENIC ACID GAMBOGENIC ACID 22663155 54915 37505 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE TRANEXAMIC ACID 54916 37506 IL23A 51561 DRUGGABLE GENOME inhibitor CHEMBL2108681 TILDRAKIZUMAB 54918 37507 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DICYCLOMINE HYDROCHLORIDE DICYCLOMINE HYDROCHLORIDE 54919 37508 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NEVIRAPINE NEVIRAPINE 22931300 54920 37509 SMN1 6606 DRUGGABLE GENOME GNF-PF-1211 CHEMBL600968 54921 37510 IGF2R 3482 ENZYME, DRUGGABLE GENOME, CELL SURFACE Juvidex MANNOSE 6-PHOSPHATE 20927486 54922 37511 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER thioureidobutyronitrile 4-ISOTHIOUREIDOBUTYRONITRILE 54923 37512 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Five-and-six-membered heterocyclic compound 1 54924 37513 BAZ2B 29994 NA NSC-66209 CHEMBL175266 54925 37514 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE C5A 16634840 54926 37515 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE PMID29130358-Compound-LonimacranthoideVII 54927 37516 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR paclitaxel PACLITAXEL 25495407 54930 37517 KCNH6 81033 DRUGGABLE GENOME, ION CHANNEL activator 135650743 54931 37518 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ETHOPROPAZINE ETHOPROPAZINE 54932 37519 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR bimatoprost (free acid form) 54933 37520 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ACLIDINIUM ACLIDINIUM 54934 37521 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE COUMARIN COUMARIN 3160707 54935 37522 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE KTN3379 26064441 54936 37523 RAB27A 5873 ENZYME emapalumab EMAPALUMAB 54938 37524 DTYMK 1841 KINASE zidovudine ZIDOVUDINE 22960662 54939 37525 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR ACTINOMYCIN D 16616440 54940 37526 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ACECLIDINE ACECLIDINE 54941 37527 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME Platinum compounds 21940774 54942 37528 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NSC-748113 CHEMBL2063687 22283430 54943 37529 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE LINOLEIC ACID LINOLEIC ACID 54944 37530 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR RG-1530 RG-1530 54951 37531 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE PKI-402 CHEMBL589258 20371716 54953 37532 POLI 11201 DNA REPAIR BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 54954 37533 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator 178103452 TINZAPARIN 54955 37534 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 cisapride CISAPRIDE 9187528 54956 37535 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BRILLIANT GREEN OXALATE BRILLIANT GREEN OXALATE 54957 37536 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649956 ARIPIPRAZOLE 54959 37537 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-2B, RECOMBINANT 54960 37538 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR IL-10 INTERLEUKIN-10 16818766 54962 37539 TAC1 6863 DRUGGABLE GENOME MEXILETINE MEXILETINE 7686682 54964 37540 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MICONAZOLE MICONAZOLE 54965 37541 MAGEA3 4102 ENZYME, DRUGGABLE GENOME vaccine GSK1572932A ASTUPROTIMUT-R 54966 37542 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ANAZOLENE ANAZOLENE 54968 37543 GLS 2744 ENZYME PMID30273516-Compound-37 54970 37544 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR E319 E319 54971 37545 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME AR-42 AR-42 54974 37546 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE PMID27539678-Compound-4 54979 37547 ADAM17 6868 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, NEUTRAL ZINC METALLOPEPTIDASE, TRANSPORTER, ENZYME inhibitor 252166880 54983 37548 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME N-2-NAPHTHYLIMIDODICARBONIMIDIC DIAMIDE CHEMBL43078 54984 37549 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHRYSENE-1,4-DIONE CHEMBL421215 54985 37550 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ASCORBYL PALMITATE ASCORBYL PALMITATE 54987 37551 SMAD2 4087 KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX HYDROCORTISONE HYDROCORTISONE 16644034 54988 37552 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4746 CHEMBL584868 54990 37553 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CCG-50014 CHEMBL1917204 54991 37554 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUROGESTONE ACETATE FLUROGESTONE ACETATE 54992 37555 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR ACTINOMYCIN D 9851943 54993 37556 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 53801057 NIMODIPINE 54994 37557 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 178101928 54996 37558 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-neotuberostemonine 54997 37559 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CAULIBUGULONE C CAULIBUGULONE C 54998 37560 KCNJ3 3760 EXTERNAL SIDE OF PLASMA MEMBRANE, ION CHANNEL, DRUGGABLE GENOME CLOZAPINE CLOZAPINE 10780978 54999 37561 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102414 55001 37562 HTT 3064 DRUGGABLE GENOME Abexinostat ABEXINOSTAT 55003 37563 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000111875 CHEMBL590949 55004 37564 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 15 55005 37565 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DARBUFELONE MESYLATE DARBUFELONE MESYLATE 55007 37566 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL538943 VINORELBINE TARTRATE 55008 37567 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DIBUTYLDICHLOROSTANNANE DIBUTYLDICHLOROSTANNANE 55010 37568 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME methylphenidate METHYLPHENIDATE 27624150 55013 37569 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NONIVAMIDE NONIVAMIDE 55014 37570 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 249565930 55015 37571 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE 404859160 55016 37572 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TETRADECYLTHIOACETIC ACID TETRADECYLTHIOACETIC ACID 20036122 55017 37573 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolo[2,3-d]pyrimidine derivative 3 55019 37574 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER amprenavir AMPRENAVIR 55020 37575 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW795486X GW795486X 55021 37576 RAMP1 10267 DRUGGABLE GENOME, CELL SURFACE PRAMLINTIDE PRAMLINTIDE 55022 37577 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651383 55024 37578 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 310264765 PF-03893787 55025 37579 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DS-7423 DS-7423 24504419 55026 37580 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Doxorubicin DOXORUBICIN 26552700 55027 37581 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME ICA-105665 55028 37582 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ENZALUTAMIDE ENZALUTAMIDE 23779130,25184630 55030 37583 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Paclitaxel PACLITAXEL 26282658 55031 37584 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE AST-487 AST-487 55032 37585 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2-METHOXYESTRADIOL 2-METHOXYESTRADIOL 55033 37586 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ORTHO-PHTHALALDEHYDE ORTHO-PHTHALALDEHYDE 55034 37587 PABPC1 26986 NA DITOLYLGUANIDINE DITOLYLGUANIDINE 55035 37588 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DACOMITINIB DACOMITINIB 25899785 55036 37589 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Lapatinib LAPATINIB 55037 37590 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE IRINOTECAN IRINOTECAN 19775480 55038 37591 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CYC-116 CYC-116 55039 37592 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ALFADEX ALFADEX 55040 37593 KDM4A 9682 DRUGGABLE GENOME, ENZYME PURPUROGALLIN PURPUROGALLIN 55041 37594 RGS4 5999 DRUGGABLE GENOME METHYSERGIDE METHYSERGIDE 55043 37595 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Imidazo bicyclic iminium derivative 5 55044 37596 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Saxagliptin SAXAGLIPTIN 55045 37597 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor CHEMBL2109539 RG-7652 55048 37598 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME blinatumomab BLINATUMOMAB 55049 37599 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Ponatinib PONATINIB 22238366,26175911,26179511 55050 37600 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C18 55054 37601 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Nitroglycerin NITROGLYCERIN 55056 37602 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-302042 CHEMBL1600564 22524450 55057 37603 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 315661180 ZOTIRACICLIB 55058 37604 ATAD5 79915 NA BAY-11-7082 CHEMBL403183 55059 37605 ODC1 4953 DRUGGABLE GENOME, ENZYME VINCRISTINE VINCRISTINE 19006285 55060 37606 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME lomitapide LOMITAPIDE 55061 37607 GPI 2821 ENZYME, GROWTH FACTOR, DRUGGABLE GENOME FDG FLUDEOXYGLUCOSE-F18 10963181 55062 37608 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1835207 APRICOXIB 55063 37609 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME inhibitor 336446966 55064 37610 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor HESPERADIN HESPERADIN 19035792 55066 37611 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102901 SALIRASIB 55067 37612 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE ENILURACIL ENILURACIL 10692560 55069 37613 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178102700 CHEMBL295212 55070 37614 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME DM-199 RECOMBINANT HUMAN KALLIKREIN-1 55071 37615 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ERLOTINIB ERLOTINIB 55073 37616 TLR7 51284 DRUGGABLE GENOME agonist 178101746 RESIQUIMOD 55074 37617 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX SORBINIL SORBINIL 24819954 55075 37618 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2103878 ODELEPRAN 55076 37619 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME inhibitor 135652711 RIFAMPIN 55077 37620 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE capecitabine CAPECITABINE 55078 37621 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor 178101869 EHNA 55079 37622 GMNN 51053 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 55080 37623 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME atorvastatin ATORVASTATIN 19474787 55083 37624 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Nutlin-3a 21515735 55084 37625 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-67 CHEMBL578512 55085 37626 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor PERIFOSINE PERIFOSINE 55087 37627 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE valproic acid 12083967 55089 37628 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545397 ACALISIB 55090 37629 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISOEUGENITOL ISOEUGENITOL 55092 37630 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE NORDIHYDROGUAIARETIC ACID 17395008 55093 37631 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE LY2835219 ABEMACICLIB 55094 37632 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR PF3644022 26140595 55098 37633 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHLORPYRIFOS CHLORPYRIFOS 55099 37634 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651422 55102 37635 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ATEZOLIZUMAB ATEZOLIZUMAB 28525386 55103 37636 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 249565581 AFURESERTIB 55104 37637 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Alpelisib ALPELISIB 27659046 55105 37638 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1255840 NEBOGLAMINE 55107 37639 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US8524917, 60 55108 37640 BAZ2B 29994 NA SB-415286 CHEMBL322970 55109 37641 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor 385612197 55110 37642 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE agonist 178100991 (D)-SERINE 55112 37643 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CLOMIFENE CLOMIPHENE 55113 37644 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 374883857 55114 37645 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Selumetinib SELUMETINIB 24939055 55117 37646 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR epinephrine EPINEPHRINE 55118 37647 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BGB-283 LIFIRAFENIB 55119 37648 IL23R 149233 KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE Tumor necrosis factor alpha (TNF-alpha) inhibitors 26194362 55122 37649 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 348353623 55123 37650 BCAT2 587 ENZYME, TRANSPORTER inhibitor 315661170 55124 37651 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE OXALIPLATIN OXALIPLATIN 16101140 55125 37652 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CELECOXIB CELECOXIB 55127 37653 SEM1 7979 NA BORTEZOMIB BORTEZOMIB 24524217 55129 37654 CDA 978 ENZYME, DRUGGABLE GENOME GEMCITABINE GEMCITABINE 12477049 55130 37655 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR VX-702 VX-702 55133 37656 TH 7054 ENZYME, DRUGGABLE GENOME TRIAMTERENE TRIAMTERENE 6149469 55134 37657 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Crizotinib CRIZOTINIB 27595477,27343442,27694386,26779812,25971938,25971939,28514312,17483355,27149990,26483207,25232318,28765324,21266357,27393507,27283993,28522754,26432108,15494073,28396313 55135 37658 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME ZNCL2 8862750 55136 37659 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR METHYLTESTOSTERONE METHYLTESTOSTERONE 55137 37660 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME LAS38096 CHEMBL375293 55138 37661 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR NARINGENIN NARINGENIN 55139 37662 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 55140 37663 ALOX15 246 ENZYME, DRUGGABLE GENOME ZM-449829 CHEMBL154580 55143 37664 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Nutlin-3 NUTLIN-3 25964101,26494859,26883273 55145 37665 POLB 5423 DNA REPAIR, DRUGGABLE GENOME QUERCETIN DIHYDRATE QUERCETIN DIHYDRATE 55146 37666 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE PD-0166285 PD-0166285 55147 37667 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 178103954 ABEMACICLIB 55149 37668 PLCG1 5335 ENZYME, KINASE, PHOSPHOLIPASE, DRUGGABLE GENOME CEFIXIME CEFIXIME 55151 37669 MMP14 4323 PROTEASE, DRUGGABLE GENOME, ENZYME vaccine PRINOMASTAT PRINOMASTAT 55152 37670 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR CLOCORTOLONE CLOCORTOLONE 55154 37671 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1,5-NAPHTHALENEDIAMINE CHEMBL538965 55156 37672 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE CAMBINOL CAMBINOL 55157 37673 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-49789 CHEMBL469309 55158 37674 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR FLUSILAZOLE FLUSILAZOLE 55160 37675 TOP2B 7155 DRUGGABLE GENOME, ENZYME Fleroxacin FLEROXACIN 55161 37676 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ALACHLOR ALACHLOR 55162 37677 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Trastuzumab TRASTUZUMAB 55163 37678 PTGS2 5743 DRUGGABLE GENOME, ENZYME TOLMETIN TOLMETIN 55164 37679 SFTPA1 653509 DRUGGABLE GENOME NAC ACETYLCYSTEINE 10533675 55165 37680 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Pc4 (topical formulation 55166 37681 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135650440 55167 37682 FAP 2191 PROTEASE, CELL SURFACE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME BIBH 1 55169 37683 TACSTD2 4070 NA antibody 249565933 55170 37684 GLS 2744 ENZYME NSC-677438 CHEMBL118678 55171 37685 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200948 TRIMIPRAMINE MALEATE 55172 37686 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME agonist 178100991 (D)-SERINE 55173 37687 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 223366077 RGB-286638 55174 37688 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR PMID26924192-Compound-103 55176 37689 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME L-741626 CHEMBL445102 55177 37690 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR PF-477736 PF-00477736 26140595 55178 37691 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor 252166487 NIRAPARIB 55179 37692 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SK&F-82958 CHEMBL35354 55181 37693 ATXN2 6311 NA MIBEFRADIL MIBEFRADIL 55182 37694 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL3545355 CHF4227 55183 37695 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor LINIFANIB LINIFANIB 55184 37696 POLB 5423 DNA REPAIR, DRUGGABLE GENOME LOBARIC ACID LOBARIC ACID 55185 37697 VKORC1 79001 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL711 PHENINDIONE 55186 37698 UGT1A7 54577 DRUGGABLE GENOME, ENZYME CURCUMIN CURCUMIN 15845768 55187 37699 KDM4A 9682 DRUGGABLE GENOME, ENZYME HYDROXYZINE HYDROCHLORIDE HYDROXYZINE HYDROCHLORIDE 55188 37700 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR PIRENOXINE PIRENOXINE 55189 37701 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL1200976 IDARUBICIN HYDROCHLORIDE 55190 37702 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL378544 VINBLASTINE SULFATE 55191 37703 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE LEVOBUNOLOL LEVOBUNOLOL 55192 37704 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME N,N-HEXAMETHYLENEAMILORIDE N,N-HEXAMETHYLENEAMILORIDE 55193 37705 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL676 PAMIDRONATE DISODIUM 55195 37706 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME MAXY-G34 55196 37707 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE GO-6976 GO-6976 55198 37708 BRCA2 675 CLINICALLY ACTIONABLE Paclitaxel PACLITAXEL 55200 37709 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MGCD265 GLESATINIB 27694386,28765324,15494073 55201 37710 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 381118891 55202 37711 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL182066 RADIPRODIL 55203 37712 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2311030 ERGOLOID MESYLATES 55206 37713 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME LINIFANIB LINIFANIB 55208 37714 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE SNS-314 SNS-314 55210 37715 NUAK1 9891 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565727 55211 37716 GPER1 2852 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR agonist 135650370 FULVESTRANT 55212 37717 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 2093195 CHEMBL411085 55215 37718 ATXN2 6311 NA ISOVELLERAL ISOVELLERAL 55216 37719 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE E-3810 RABEPRAZOLE SODIUM 55217 37720 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PHENETHYLISOTHIOCYANATE PHENETHYLISOTHIOCYANATE 22607231 55218 37721 PTGS2 5743 DRUGGABLE GENOME, ENZYME TIAPROFENIC ACID 55219 37722 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 2,4-DIACETYL PHLOROGLUCINOL CHEMBL276139 55220 37723 PSMB3 5691 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL451887 CARFILZOMIB 55222 37724 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE ACETAZOLAMIDE ACETAZOLAMIDE 24074025 55223 37725 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650556 55224 37726 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 315661269 55225 37727 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CRIZOTINIB CRIZOTINIB 55226 37728 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME amoxicillin AMOXICILLIN 30664875 55227 37729 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2106068 ATRASENTAN HYDROCHLORIDE 55228 37730 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL blocker 178101137 55230 37731 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651738 55232 37732 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200790 METHYPRYLON 55233 37733 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HM-78136B 55236 37734 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL1751 DIGOXIN 55237 37735 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1628502 GABAPENTIN ENACARBIL 55238 37736 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 L-732138 L-732138 55239 37737 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor 363894146 55240 37738 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE AMG-714 AMG-714 55241 37739 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL445813 AT-7519 55243 37740 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-2713 CHEMBL578719 55244 37741 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Biricodar BIRICODAR 55245 37742 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE ABBV-3067 55246 37743 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME BEXAROTENE BEXAROTENE 55247 37744 KCND3 3752 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL113461 TEDISAMIL 55248 37745 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME 3,4,5,6-TETRACHLORO-[1,2]BENZOQUINONE CHEMBL364729 55250 37746 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 3-METHOXYCATECHOL 3-METHOXYCATECHOL 55251 37747 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE DORAMAPIMOD DORAMAPIMOD 55252 37748 PSENEN 55851 DRUGGABLE GENOME GSI-136 GSI-136 55254 37749 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Piperidinyl pyrazole derivative 4 55255 37750 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-42 55257 37751 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565786 55259 37752 TNFSF13 8741 DRUGGABLE GENOME inhibitor CHEMBL1742986 ATACICEPT 55260 37753 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100675 55261 37754 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Roclatan 55262 37755 NGFR 4804 CELL SURFACE, DRUGGABLE GENOME Cenegermin CENEGERMIN 55263 37756 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DESLORATADINE DESLORATADINE 55264 37757 EYA2 2139 DNA REPAIR BITHIONOLOXIDE BITHIONOLOXIDE 55265 37758 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650287 55266 37759 ALOX15B 247 DRUGGABLE GENOME, ENZYME inhibitor 381744945 55268 37760 ALOX15 246 ENZYME, DRUGGABLE GENOME N,N'-DIPHENYL-P-PHENYLENEDIAMINE N,N'-DIPHENYL-P-PHENYLENEDIAMINE 55270 37761 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL1201748 CABAZITAXEL 55271 37762 POLK 51426 DNA REPAIR, ENZYME NAVITOCLAX NAVITOCLAX 55272 37763 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-MTC-422 55274 37764 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME SaxaDapa FDC 55276 37765 CDKN1C 1028 CLINICALLY ACTIONABLE, KINASE HISTONE DEACETYLASE INHIBITOR 10667572 55279 37766 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR HOMIDIUM BROMIDE HOMIDIUM BROMIDE 55280 37767 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TRIMETREXATE TRIMETREXATE 55281 37768 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BIAPENEM BIAPENEM 55283 37769 SCNN1A 6337 DRUGGABLE GENOME, ION CHANNEL AMILORIDE AMILORIDE 55286 37770 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR TANSHINONE I TANSHINONE I 55287 37771 IL13RA2 3598 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ABT-308 CENDAKIMAB 55288 37772 NOS1 4842 DRUGGABLE GENOME, ENZYME doxorubicin DOXORUBICIN 21048526 55290 37773 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE agonist 178101085 N-METHYL-D-ASPARTIC ACID (NMDA) 55295 37774 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME LOMUSTINE LOMUSTINE 30782343 55297 37775 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 55298 37776 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TRIAMTERENE TRIAMTERENE 55301 37777 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE WITHAFERIN A WITHAFERIN A 24079846 55302 37778 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR HMG-COA REDUCTASE INHIBITOR 12953163 55303 37779 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE sorafenib SORAFENIB 22736425 55304 37780 KRT20 54474 NA DOXORUBICIN HYDROCHLORIDE 15017198 55305 37781 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE 55306 37782 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 55307 37783 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-41 55308 37784 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE HYDROMORPHONE HYDROMORPHONE 55309 37785 PTGS2 5743 DRUGGABLE GENOME, ENZYME NCX 4016 55310 37786 HPSE 10855 ENZYME, DRUGGABLE GENOME THROMBIN THROMBIN 1612123 55311 37787 DYRK2 8445 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID28766366-Compound-Scheme14BINDY 55312 37788 VKORC1L1 154807 DRUGGABLE GENOME, ENZYME WARFARIN WARFARIN 55313 37789 TUBA1A 7846 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 55314 37790 HIPK3 10114 SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME inhibitor 249565806 SILMITASERTIB 55316 37791 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-2B, RECOMBINANT 55318 37792 HSPG2 3339 KINASE, DRUGGABLE GENOME haloperidol HALOPERIDOL 27023437 55321 37793 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MM-302 GANCOTAMAB 26759238 55322 37794 MAOB 4129 DRUGGABLE GENOME, ENZYME EVT302 55325 37795 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-N1 55326 37796 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ESTRAMUSTINE ESTRAMUSTINE 15869997 55327 37797 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE 681640 CHEMBL379975 55328 37798 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor 178103187 55330 37799 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Indole carboxamide derivative 1 55331 37800 FKBP5 2289 DRUGGABLE GENOME bupropion BUPROPION 22947179 55332 37801 TUBB 203068 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 55334 37802 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE LETROZOLE LETROZOLE 12569569 55336 37803 PTGS1 5742 ENZYME, DRUGGABLE GENOME clopidogrel CLOPIDOGREL 22940005 55337 37804 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE PIMECROLIMUS PIMECROLIMUS 55338 37805 CBX1 10951 NA CALCIMYCIN CALCIMYCIN 55339 37806 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE allosteric modulator 315661242 55340 37807 TH 7054 ENZYME, DRUGGABLE GENOME inhibitor 178101807 55341 37808 POLI 11201 DNA REPAIR ISOVELLERAL ISOVELLERAL 55342 37809 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PSC 833 9446255 55343 37810 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DARGLITAZONE DARGLITAZONE 55345 37811 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE inhibitor CHEMBL1201182 TEMSIROLIMUS 55346 37812 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CARMINOMYCIN CARUBICIN 55347 37813 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist CHEMBL1201533 THYROTROPIN ALFA 55348 37814 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE MAPATUMUMAB MAPATUMUMAB 55349 37815 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE PAZOPANIB PAZOPANIB 55350 37816 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER LITHOCHOLIC ACID LITHOCHOLIC ACID 55352 37817 BAZ2B 29994 NA SJ000113107 CHEMBL589245 55353 37818 HBB 3043 DRUGGABLE GENOME, ENZYME 5-hydroxymethyl-2-furfural (sickle cell disease), AesRx LLC 55354 37819 POLR1G 10849 NA gemcitabine GEMCITABINE 55356 37820 BRCA2 675 CLINICALLY ACTIONABLE CISPLATIN CISPLATIN 29338080,25847936 55357 37821 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME LEVOMILNACIPRAN LEVOMILNACIPRAN 55358 37822 POLI 11201 DNA REPAIR 1-DEOXYRUBRALACTONE CHEMBL260980 18178092 55359 37823 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545401 X-82 55360 37824 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 249565584 DAPOXETINE 55362 37825 NCOR2 9612 NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GNF-PF-2893 CHEMBL312032 55365 37826 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1,3-DINITRO-NAPHTHALENE CHEMBL163970 55366 37827 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-WO2011127048 33 55368 37828 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME 3-HYDROXYPHTHALIC ANHYDRIDE CHEMBL2057864 22819190 55370 37829 MAPT 4137 DRUGGABLE GENOME AMENTOFLAVONE AMENTOFLAVONE 55371 37830 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135649888 55373 37831 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 lopinavir LOPINAVIR 55375 37832 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL1908397 KW-2449 55376 37833 NPR3 4883 DRUGGABLE GENOME ANX-042 23694773 55377 37834 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE TNF-ALPHA 8611631 55380 37835 PI4KA 5297 DRUGGABLE GENOME, ENZYME, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor 315661277 55381 37836 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 223366032 VISTUSERTIB 55382 37837 ABAT 18 DRUGGABLE GENOME, ENZYME T83193 55383 37838 EPHA3 2042 ENZYME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME KB004 55384 37839 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE ciprofloxacin CIPROFLOXACIN 20127091 55385 37840 MUTYH 4595 DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME cisplatin CISPLATIN 24533712 55386 37841 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MITOMYCIN MITOMYCIN 22931300 55388 37842 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE ERLOTINIB ERLOTINIB 16282176 55390 37843 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-134 CHEMBL578896 55392 37844 LIG3 3980 NA cisplatin CISPLATIN 24533712 55393 37845 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CORTICOSTEROIDS 9753488 55394 37846 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME EMODIC ACID EMODIC ACID 55397 37847 TUBA1C 84790 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 55398 37848 FAAH 2166 ENZYME, DRUGGABLE GENOME methamphetamine METHAMPHETAMINE 23556448,31789429 55399 37849 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME HPP-854 55401 37850 PRMT1 3276 ENZYME, METHYL TRANSFERASE STILBAMIDINE STILBAMIDINE 20666457 55402 37851 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 178100864 55403 37852 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DEMECLOCYCLINE HYDROCHLORIDE DEMECLOCYCLINE HYDROCHLORIDE 55404 37853 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650830 PIPAMPERONE 55408 37854 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR PTEROSTILBENE PTEROSTILBENE 55409 37855 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ISF35 55410 37856 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c][1,2,4]benzotriazine derivative 1 55412 37857 PDE7B 27115 DRUGGABLE GENOME, ENZYME inhibitor 178101509 DIPYRIDAMOLE 55413 37858 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUOXYMESTERONE FLUOXYMESTERONE 55415 37859 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 249565621 MILCICLIB 55416 37860 TNNC1 7134 DRUGGABLE GENOME PURPUROGALLIN PURPUROGALLIN 55417 37861 ALOX15B 247 DRUGGABLE GENOME, ENZYME GOSSYPOL GOSSYPOL 55418 37862 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody CETUXIMAB CETUXIMAB 55420 37863 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ABX-0401 55421 37864 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME FRAXETIN FRAXETIN 55422 37865 CD9 928 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE LIF 11950938 55423 37866 CXCL2 2920 DRUGGABLE GENOME STAUROSPORINE STAUROSPORINE 10354507 55424 37867 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-60339 CHEMBL1448793 55425 37868 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1090173 SD-0006 55426 37869 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME CSA CYCLOSPORINE 11827957 55427 37870 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME HAEMATOXYLIN HAEMATOXYLIN 55428 37871 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR GLYCITEIN GLYCITEIN 16038533 55429 37872 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER lamotrigine LAMOTRIGINE 55430 37873 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME FENOFIBRATE FENOFIBRATE 16680159 55431 37874 F11 2160 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103163 55433 37875 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL3545285 XL-999 55434 37876 POLK 51426 DNA REPAIR, ENZYME AG-537 CHEMBL67535 55436 37877 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Ridaforolimus RIDAFOROLIMUS 26187616 55437 37878 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 375973223 55438 37879 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME RUXOLITINIB RUXOLITINIB 29773603,25207766 55439 37880 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR imidapril IMIDAPRIL 25143324 55441 37881 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR lithium LITHIUM 20348464 55444 37882 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 55445 37883 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR PREMARIN PREMARIN 8888658 55446 37884 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR (E)-2-STYRYLCHROMONE CHEMBL388823 55447 37885 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-1319 CHEMBL235891 55448 37886 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE FASUDIL FASUDIL 55449 37887 SERPIND1 3053 DRUGGABLE GENOME, PROTEASE INHIBITOR ARDEPARIN 55450 37888 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE ALISERTIB ALISERTIB 55451 37889 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME Vincristine VINCRISTINE 55452 37890 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Benzothiazepine analog 12 55453 37891 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME RECOMBINANT ANTIHEMOPHILIC FACTOR 55454 37892 GMNN 51053 DRUGGABLE GENOME DIETHYLSTILBESTROL DIETHYLSTILBESTROL 55455 37893 PAK6 56924 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 178101884 GSK-690693 55456 37894 MAP3K5 4217 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, ENZYME hydroxyurea HYDROXYUREA 23556445 55457 37895 ARSA 410 DRUGGABLE GENOME, ENZYME BENZOXATHIAN BENZOXATHIAN 55458 37896 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK1023156A GSK-1023156A 55463 37897 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-10 55464 37898 PSMC4 5704 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 55465 37899 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-124317 CHEMBL586937 55468 37900 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TAZAROTENE TAZAROTENE 55469 37901 IL17RA 23765 DRUGGABLE GENOME Brodalumab BRODALUMAB 55470 37902 GMNN 51053 DRUGGABLE GENOME DNDI1417346 CHEMBL1490332 55471 37903 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 55472 37904 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CY-208243 CHEMBL313737 55474 37905 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ANAKINRA ANAKINRA 55475 37906 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME activator 178102130 GABAPENTIN 55476 37907 POLB 5423 DNA REPAIR, DRUGGABLE GENOME N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 55477 37908 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE ERYTHROPOIETIN EPOETIN BETA 10682118 55478 37909 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE KARANJIN KARANJIN 55482 37910 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME CAMPTOTHECIN CAMPTOTHECIN 9398050 55483 37911 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Indirubin derivative 2 55484 37912 MAPT 4137 DRUGGABLE GENOME TYRPHOSTIN 1 TYRPHOSTIN 1 55485 37913 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE JQ1 26552700 55486 37914 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-11 55488 37915 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME SLAZINIC ACID SLAZINIC ACID 55490 37916 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME BORTEZOMIB BORTEZOMIB 20875739 55491 37917 KDM3A 55818 ENZYME inhibitor 249565910 55493 37918 SERPIND1 3053 DRUGGABLE GENOME, PROTEASE INHIBITOR SULODEXIDE SULODEXIDE 55494 37919 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 252166561 55496 37920 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Abemaciclib ABEMACICLIB 27217383 55498 37921 PLCG1 5335 ENZYME, KINASE, PHOSPHOLIPASE, DRUGGABLE GENOME acetaminophen ACETAMINOPHEN 26398624 55499 37922 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE efavirenz EFAVIRENZ 20860463,20625352,24477223,16267764,15622315 55500 37923 LTA 4049 DRUGGABLE GENOME inhibitor CHEMBL1743056 PATECLIZUMAB 55501 37924 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BUTYRYLHYDROXAMIC ACID BUTYRYLHYDROXAMIC ACID 21874153 55502 37925 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PERHEXILINE PERHEXILINE 22931300 55503 37926 EIF4EBP1 1978 KINASE PACLITAXEL PACLITAXEL 15897904 55504 37927 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 405067318 55505 37928 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX CYNAROPICRIN CYNAROPICRIN 23232059 55506 37929 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Vitamin B-complex with vitamin C 55507 37930 TUBA3D 113457 DRUGGABLE GENOME CHEMBL492399 VERUBULIN 55508 37931 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER DAUNORUBICIN DAUNORUBICIN 10500777 55510 37932 ALOX15B 247 DRUGGABLE GENOME, ENZYME SJ000191886 CHEMBL601616 55511 37933 BAZ2B 29994 NA 2-HYDROXY-NAPHTHALDEHYDE THIOSEMICARBAZONE CHEMBL505209 55512 37934 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX (+)-TUBERIFERIN CHEMBL1940084 22153345 55514 37935 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRICIRIBINE TRICIRIBINE 55515 37936 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME umeclidinium UMECLIDINIUM 55516 37937 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-7387 CHEMBL119878 55517 37938 CREB1 1385 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ETHANOL ALCOHOL 11181917 55518 37939 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BIIB 028 55519 37940 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE aspirin ASPIRIN 28820077,23859572 55520 37941 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX POMIFERIN POMIFERIN 55521 37942 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR THYMIDINE THYMIDINE 16280359 55522 37943 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135652718 STRYCHNINE 55523 37944 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PROTOPORPHYRIN PROTOPORPHYRIN 55525 37945 GMNN 51053 DRUGGABLE GENOME GNF-PF-4337 CHEMBL277148 55526 37946 KDM4A 9682 DRUGGABLE GENOME, ENZYME DEOXYVASICINONE DEOXYVASICINONE 55528 37947 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE inhibitor RO4929097 RG-4733 55529 37948 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR AT13387 55531 37949 EPHA1 2041 DRUGGABLE GENOME, KINASE, TYROSINE KINASE inhibitor CHEMBL24828 VANDETANIB 55532 37950 POLI 11201 DNA REPAIR NOREPINEPHRINE NOREPINEPHRINE 55533 37951 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROPRANOLOL PROPRANOLOL 55534 37952 MARCHF8 220972 ENZYME Fendrix FENDRIX 55535 37953 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NARASIN NARASIN 55537 37954 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor PF-4691502 PF-04691502 55538 37955 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE agonist CHEMBL1201821 PALIFERMIN 55539 37956 CACNA2D3 55799 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL1628502 GABAPENTIN ENACARBIL 55540 37957 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650571 55541 37958 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL ARVERAPAMIL 55542 37959 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 252166878 FINERENONE 55543 37960 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652266 55544 37961 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ETONITAZENE ETONITAZENE 55546 37962 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker 135650376 55547 37963 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR S-PRAnt 55549 37964 GMNN 51053 DRUGGABLE GENOME GBR-12909 VANOXERINE 55551 37965 ATP1B1 481 DRUGGABLE GENOME, TRANSPORTER, ENZYME inhibitor CHEMBL3545057 ACETYLDIGITOXIN 55552 37966 QRFPR 84109 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 381744935 55553 37967 NEK4 6787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CYC-116 CYC-116 55554 37968 RICTOR 253260 CLINICALLY ACTIONABLE inhibitor AZD8055 AZD-8055 55556 37969 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DAUCOSTEROL SITOGLUSIDE 19716700 55557 37970 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Isochroman-4-ketone derivative 1 55558 37971 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 55561 37972 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE antagonist 178100872 ATOPAXAR 55562 37973 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MESO-HEXESTROL MESO-HEXESTROL 55563 37974 ATF2 1386 TRANSCRIPTION FACTOR STZ STREPTOZOCIN 12805110 55564 37975 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY TESTOSTERONE TESTOSTERONE 8404664 55565 37976 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CT-1578 CT-1578 22339472 55566 37977 ATAD5 79915 NA NSC-105827 CHEMBL171699 55567 37978 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650516 LEVONORGESTREL 55571 37979 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Sorafenib SORAFENIB 19139124,24317392,17229632,22665524,20372153,17699867,19461405,25363205,20970876 55573 37980 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SERTRALINE HYDROCHLORIDE SERTRALINE HYDROCHLORIDE 55575 37981 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651418 ALITRETINOIN 55576 37982 PMEL 6490 DRUGGABLE GENOME AE-08 55577 37983 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Pyrazolodiazepine derivative 1 55578 37984 PSMD7 5713 PROTEASE inhibitor BORTEZOMIB BORTEZOMIB 55579 37985 PSMD6 9861 NA inhibitor CHEMBL2103884 OPROZOMIB 55580 37986 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX 2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE CHEMBL201325 55583 37987 GDF15 9518 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR DICLOFENAC DICLOFENAC 15555568 55584 37988 CA1 759 DRUGGABLE GENOME, ENZYME TRICHLORMETHIAZIDE TRICHLORMETHIAZIDE 55585 37989 PRKG1 5592 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME SOTRASTAURIN SOTRASTAURIN 55587 37990 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1701 MEPERIDINE HYDROCHLORIDE 55588 37991 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR UNC1999 23614352 55589 37992 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME VINBLASTINE VINBLASTINE 8763853 55590 37993 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME cyclophosphamide CYCLOPHOSPHAMIDE 24533712 55591 37994 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE STROPHANTHIDIN STROPHANTHIDIN 55593 37995 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR Antiinflammatory agents, non-steroids 25096645 55594 37996 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 glibenclamide GLYBURIDE 24442125,16342679 55595 37997 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DIHYDROGAMBOGIC ACID DIHYDROGAMBOGIC ACID 55596 37998 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-48 55597 37999 IL1B 3553 KINASE, DRUGGABLE GENOME TT-301 TT-301 22131899 55598 38000 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME RELACATIB RELACATIB 55599 38001 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Copanlisib COPANLISIB 27672108,24170767 55600 38002 RGS4 5999 DRUGGABLE GENOME TYRPHOSTIN A9 TYRPHOSTIN A9 55601 38003 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL2106798 NERAMEXANE MESYLATE 55602 38004 PROM1 8842 CELL SURFACE, DRUGGABLE GENOME ICT-121 25691822 55607 38005 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE CEDIRANIB CEDIRANIB 55609 38006 USP1 7398 DNA REPAIR, PROTEASE, ENZYME OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 55611 38007 SMN1 6606 DRUGGABLE GENOME N-(4-NITROPHENYL)ANTHRANILIC ACID CHEMBL1574420 55613 38008 ANXA2 302 CELL SURFACE, DRUGGABLE GENOME N-ETHYLMALEIMIDE N-ETHYLMALEIMIDE 16408090 55614 38009 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200326 NICARDIPINE HYDROCHLORIDE 55615 38010 BRCA2 675 CLINICALLY ACTIONABLE VELIPARIB VELIPARIB 29338080 55616 38011 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME DIMETHYLPHENYLPIPERAZINIUM IODIDE DIMETHYLPHENYLPIPERAZINIUM IODIDE 55617 38012 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3268 CHEMBL582073 55619 38013 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME 681640 CHEMBL379975 55620 38014 RAMP1 10267 DRUGGABLE GENOME, CELL SURFACE agonist CHEMBL2105635 DAVALINTIDE 55622 38015 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650034 BURIMAMIDE 55623 38016 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NORSTICTIC ACID NORSTICTIC ACID 55624 38017 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CIGLITAZONE CIGLITAZONE 23566516 55625 38018 HAS3 3038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME anthracyclines and related substances 55628 38019 TXNRD1 7296 DRUGGABLE GENOME Binuclear gold(I) compound 3 55630 38020 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME MK-2578 55632 38021 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR antagonist 135650760 ONAPRISTONE 55633 38022 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME hmg coa reductase inhibitors 29210320 55635 38023 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME TCMDC-124266 CHEMBL124006 55636 38024 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Angiotensin II Antagonists 22543981 55637 38025 TUBB4B 10383 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 55638 38026 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 6-HYDROXYFLAVONE 6-HYDROXYFLAVONE 55641 38027 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROTEIN KINASE C INHIBITOR 7588324 55642 38028 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178103695 ATOMOXETINE 55644 38029 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL3544909 CALCIFEDIOL 55646 38030 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 178101606 DORSOMORPHIN 55647 38031 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE 381118909 TEZACAFTOR 55650 38032 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME NIFEDIPINE NIFEDIPINE 55651 38033 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651584 55652 38034 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BUTYLATED HYDROXYTOLUENE BUTYLATED HYDROXYTOLUENE 55654 38035 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRADIOL DIPROPIONATE ESTRADIOL DIPROPIONATE 55656 38036 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor CHEMBL3545022 ULIXERTINIB 55657 38037 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AM-630 CHEMBL181633 55658 38038 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 3,3',4,4',5'-PENTAMETHOXYCHALCONE CHEMBL190474 20813535 55659 38039 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL522302 VOFOPITANT 55663 38040 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SPHONDIN SPHONDIN 55666 38041 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Isoxazole derivative 2 55667 38042 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1615369 DABIGATRAN ETEXILATE MESYLATE 55668 38043 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GGF-2 55669 38044 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Atomoxetine ATOMOXETINE 55670 38045 KRT18 3875 DRUGGABLE GENOME IL-6 17213200 55671 38046 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolo[2,3-b]pyridine derivative 1 55673 38047 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR LGD-5552 CHEMBL259820 18032610 55676 38048 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565695 55677 38049 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor GIVINOSTAT GIVINOSTAT 55678 38050 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-12 55679 38051 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL1654 RISEDRONATE SODIUM 55680 38052 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BENZYL ISOTHIOCYANATE BENZYL ISOTHIOCYANATE 55684 38053 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE NADOLOL NADOLOL 55685 38054 POLI 11201 DNA REPAIR PENTAMIDINE ISETHIONATE PENTAMIDINE ISETHIONATE 55686 38055 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1743057 PEGSUNERCEPT 55687 38056 FKBP5 2289 DRUGGABLE GENOME nefazodone NEFAZODONE 18597649,21449676,20709156,19676097,15565110,23733030,17467808 55689 38057 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TOLFENAMIC ACID TOLFENAMIC ACID 55690 38058 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4-METHYLDAPHNETIN 4-METHYLDAPHNETIN 55693 38059 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Fremanezumab FREMANEZUMAB 55694 38060 BMPR1B 658 DRUGGABLE GENOME, CELL SURFACE, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 223366128 GALUNISERTIB 55696 38061 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME TAE-684 TAE-684 55697 38062 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE sevoflurane SEVOFLURANE 26771271 55698 38063 KDM4A 9682 DRUGGABLE GENOME, ENZYME PICEATANNOL PICEATANNOL 55703 38064 PTGS1 5742 ENZYME, DRUGGABLE GENOME Eicosapentaenoic acid/docosa-hexaenoic acid 55704 38065 TRIM24 8805 ENZYME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE inhibitor 252166607 55705 38066 APC 324 CLINICALLY ACTIONABLE Vantictumab VANTICTUMAB 22753465 55706 38067 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MINOCYCLINE HYDROCHLORIDE MINOCYCLINE HYDROCHLORIDE 55708 38068 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NISOLDIPINE NISOLDIPINE 22931300 55709 38069 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHYLEUGENOL METHYLEUGENOL 55710 38070 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000119988 CHEMBL589694 55711 38071 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE FLUOROURACIL FLUOROURACIL 55712 38072 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AZD-3199 AZD3199 25709399 55714 38073 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR HERBIMYCIN A 9933022 55715 38074 POLK 51426 DNA REPAIR, ENZYME METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE 55716 38075 MAOB 4129 DRUGGABLE GENOME, ENZYME 5-PHENOXYPHTHALIMIDE CHEMBL1813518 21778064 55719 38076 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE GM6001 55722 38077 PDE5A 8654 ENZYME, DRUGGABLE GENOME THEOPHYLLINE THEOPHYLLINE 55723 38078 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CLOBAZAM CLOBAZAM 55724 38079 UGT2B7 7364 DRUGGABLE GENOME flurbiprofen FLURBIPROFEN 21856293 55726 38080 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 363894214 SITRAVATINIB 55727 38081 PSMD1 5707 NA BORTEZOMIB BORTEZOMIB 55731 38082 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 223366055 55732 38083 PTGS2 5743 DRUGGABLE GENOME, ENZYME PARECOXIB PARECOXIB 55733 38084 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BCG BCG VACCINE 14742634 55736 38085 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRADIOL BENZOATE ESTRADIOL BENZOATE 55738 38086 TMEM97 27346 NA Isoindoline derivative 1 55739 38087 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TRANILAST TRANILAST 55740 38088 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE THIRAM THIRAM 55743 38089 GPR68 8111 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 404859019 55747 38090 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX LUTEOLIN LUTEOLIN 25190466 55748 38091 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AMONAFIDE AMONAFIDE 55749 38092 ALDH1A1 216 DRUGGABLE GENOME, ENZYME HAEMATOXYLIN HAEMATOXYLIN 55750 38093 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE donepezil DONEPEZIL 18695978 55751 38094 TNFRSF1A 7132 CELL SURFACE, DRUGGABLE GENOME 178101766 55752 38095 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178103951 DINACICLIB 55753 38096 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125587 CHEMBL532160 55755 38097 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME 2-alkyloxy-3-phenylethynyl-4a,5-dihydropyrido[2,3-b]pyrazine derivative 1 55756 38098 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE MM-151 25911688,26843189 55757 38099 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME FUROSEMIDE FUROSEMIDE 1446618 55759 38100 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1200890 OXYCODONE HYDROCHLORIDE 55762 38101 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME MMV006513 CHEMBL585622 55763 38102 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor 178103840 PHENELZINE 55764 38103 HR 55806 NUCLEAR HORMONE RECEPTOR Votucalis ophthalmic 55767 38104 HDC 3067 DRUGGABLE GENOME, ENZYME OMEPRAZOLE OMEPRAZOLE 8187977 55768 38105 LGR5 8549 G PROTEIN COUPLED RECEPTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 178100588 55769 38106 ATAD5 79915 NA GNF-PF-254 CHEMBL461579 55770 38107 ATAD5 79915 NA ANISOMYCIN ANISOMYCIN 55773 38108 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE HORMONES 10424406 55775 38109 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE TOZASERTIB TOZASERTIB 55777 38110 HBB 3043 DRUGGABLE GENOME, ENZYME QUINACRINE DIHYDROCHLORIDE QUINACRINE DIHYDROCHLORIDE 55779 38111 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SJ000113257 CHEMBL528694 55780 38112 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME VINBLASTINE VINBLASTINE 1371564 55785 38113 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-130813 CHEMBL463783 55787 38114 A2M 2 ENZYME, TRANSPORTER, DRUGGABLE GENOME, PROTEASE INHIBITOR PROSTAGLANDIN E1 6202298 55788 38115 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHELERYTHRINE CHELERYTHRINE 55789 38116 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME XR-9544 CHEMBL444075 26197160 55793 38117 KCNT2 343450 ION CHANNEL, DRUGGABLE GENOME Bisphosphonates 55795 38118 POLI 11201 DNA REPAIR DEOXYVASICINONE DEOXYVASICINONE 55796 38119 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME PMID27998201-Compound-24 55798 38120 GBA 2629 DRUGGABLE GENOME, ENZYME TCMDC-124482 CHEMBL529939 55802 38121 GMNN 51053 DRUGGABLE GENOME ZAFIRLUKAST ZAFIRLUKAST 55804 38122 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZ628 26351322 55805 38123 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Besipirdine BESIPIRDINE 55807 38124 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SNDX-275 ENTINOSTAT 55808 38125 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROROXAN HYDROCHLORIDE PROROXAN HYDROCHLORIDE 55809 38126 COL1A1 1277 CLINICALLY ACTIONABLE, DRUGGABLE GENOME COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 55810 38127 DHFR 1719 DRUGGABLE GENOME, ENZYME METHOTREXATE METHOTREXATE 8162600,6831441,7346712,1489988,944698 55811 38128 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GNF-PF-1500 CHEMBL577673 55812 38129 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PMID29130358-Compound-Figure16(9b) 55813 38130 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE C 82 55814 38131 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR D-DOPA CHEMBL211670 55815 38132 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE E319 E319 55816 38133 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 252166570 GSK-1070916 55818 38134 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 budesonide BUDESONIDE 9187528 55820 38135 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MAKALUVAMINE E MAKALUVAMINE E 8691207 55821 38136 BAZ2B 29994 NA FUSARIC ACID FUSARIC ACID 55822 38137 CDK16 5127 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1230607 PHA-793887 55824 38138 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME dantrolene DANTROLENE 55826 38139 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL TETRODOTOXIN TETRODOTOXIN 55828 38140 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ACEPROMAZINE ACEPROMAZINE 55829 38141 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SHP099 27362227 55830 38142 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GDC-0623 RG-7420 23934108 55831 38143 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME RECOMBINANT HUMAN THROMBIN 55832 38144 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650056 CARBACYCLIN 55833 38145 HBB 3043 DRUGGABLE GENOME, ENZYME FBS-0701 DEFERITAZOLE 55834 38146 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-123762 CHEMBL547483 55835 38147 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL1200515 DESERPIDINE 55836 38148 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DOFETILIDE DOFETILIDE 22931300 55844 38149 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR ETOPOSIDE ETOPOSIDE 22364746 55845 38150 POLR1G 10849 NA Platinum compounds 19203783 55846 38151 TOP1MT 116447 DRUGGABLE GENOME, ENZYME IRINOTECAN IRINOTECAN 55849 38152 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Osimertinib OSIMERTINIB 55850 38153 CXCL8 3576 DRUGGABLE GENOME C225 CETUXIMAB 10037173 55853 38154 MAPT 4137 DRUGGABLE GENOME GNF-PF-2357 CHEMBL578257 55854 38155 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PAPAVEROLINE PAPAVEROLINE 55855 38156 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 385612248 55856 38157 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1131 ACITRETIN 55857 38158 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL14762 SELICICLIB 55859 38159 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING PROTOPORPHYRIN PROTOPORPHYRIN 55861 38160 MYLK 4638 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565832 55864 38161 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE DOVITINIB DOVITINIB 55865 38162 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200927 DEXCHLORPHENIRAMINE MALEATE 55867 38163 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor MK5108 MK-5108 55870 38164 GMNN 51053 DRUGGABLE GENOME ETHYLESTRENOL ETHYLESTRENOL 55873 38165 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (S)-NOMIFENSINE CHEMBL51697 55874 38166 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AE37 55875 38167 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1201777 TAPENTADOL HYDROCHLORIDE 55876 38168 NOS2 4843 DRUGGABLE GENOME, ENZYME doxorubicin DOXORUBICIN 21048526 55878 38169 HSPB1 3315 DRUGGABLE GENOME ALBENDAZOLE ALBENDAZOLE 55879 38170 SMN2 6607 DRUGGABLE GENOME Nusinersen NUSINERSEN 55880 38171 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ERBB3 antibody 27196767 55881 38172 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Raltegravir RALTEGRAVIR 55882 38173 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 tolbutamide TOLBUTAMIDE 15284535,8742240,11875364,25994031,27339126,32531309 55883 38174 CFL1 1072 KINASE PATULIN PATULIN 16680159 55885 38175 EPHA3 2042 ENZYME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME KB-004 KB-004 55888 38176 MTTP 4547 DRUGGABLE GENOME pravastatin PRAVASTATIN 15136504 55890 38177 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor 384403679 55891 38178 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL501867 VINCRISTINE SULFATE 55893 38179 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FURFURAL FURFURAL 55894 38180 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME JNJ-7706621 JNJ-7706621 55897 38181 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME QUINACRINE QUINACRINE 55898 38182 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME TRAZODONE TRAZODONE 55900 38183 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 387065576 55901 38184 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME CAMPTOTHECIN CAMPTOTHECIN 17303082 55902 38185 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3133037 LEQ506 55903 38186 LTA 4049 DRUGGABLE GENOME inhibitor CHEMBL1742988 BAMINERCEPT 55904 38187 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LEVISOPRENALINE LEVISOPRENALINE 55907 38188 TPSAB1 7177 PROTEASE, DRUGGABLE GENOME, ENZYME THROMBIN THROMBIN 9020112 55908 38189 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER warfarin WARFARIN 25312789,29875668,22248286,29432897 55910 38190 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-747266 CHEMBL609570 55911 38191 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME GALANTAMINE GALANTAMINE 55912 38192 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR GW441756X GW441756X 55913 38193 TSPO 706 DRUGGABLE GENOME Quinazoline derivative 5 55914 38194 MAPT 4137 DRUGGABLE GENOME IDARUBICIN IDARUBICIN 55915 38195 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME METHYLDOPA (RACEMIC) METHYLDOPA (RACEMIC) 55916 38196 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR CARMINOMYCIN CARUBICIN 55917 38197 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AT7519 AT-7519 55920 38198 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 1-(4-HYDROXYPHENYL)MALEIMIDE CHEMBL565893 55921 38199 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-(4-METHOXYPHENYL)BENZO[D]THIAZOLE CHEMBL460508 55922 38200 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652263 55925 38201 GALT 2592 ENZYME Algenpantucel-L ALGENPANTUCEL-L 24343588 55926 38202 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE inhibitor 252166779 55927 38203 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COLCHICINE COLCHICINE 55929 38204 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 135651397 55930 38205 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME AG-1879 CHEMBL406845 55931 38206 ALDH5A1 7915 DRUGGABLE GENOME, ENZYME VALPROIC ACID VALPROIC ACID 11086726 55932 38207 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 384403651 55933 38208 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE SJ000018309 CHEMBL591363 55934 38209 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor ENZASTAURIN ENZASTAURIN 55935 38210 MUC2 4583 DRUGGABLE GENOME 5-AZADEOXYCYTIDINE DECITABINE 11368880 55936 38211 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178103790 LOPERAMIDE 55938 38212 SLC38A5 92745 TRANSPORTER 178101341 55940 38213 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Tiotropium TIOTROPIUM 55942 38214 ABAT 18 DRUGGABLE GENOME, ENZYME VALPROIC ACID 55944 38215 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME METHYLPHENIDATE METHYLPHENIDATE 55945 38216 ADAM10 102 ENZYME, CELL SURFACE, TRANSPORTER, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE inhibitor 252166769 55946 38217 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 310264694 AMG-337 55947 38218 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE BCG BCG VACCINE 10022737 55948 38219 GLS 2744 ENZYME CEFACLOR CEFACLOR 55951 38220 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Calcidiol CALCIFEDIOL 55952 38221 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OXADIAZON OXADIAZON 55953 38222 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 354702287 55954 38223 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-633 CHEMBL602408 55955 38224 THBD 7056 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME GINKGO BILOBA 17044640 55957 38225 GMNN 51053 DRUGGABLE GENOME CLOXYQUIN CLOXYQUIN 55958 38226 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PMID27376512-Compound-MTC-424 55961 38227 PSMA2 5683 DRUGGABLE GENOME, PROTEASE CARFILZOMIB CARFILZOMIB 24524217 55962 38228 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL SA4503 55964 38229 APC 324 CLINICALLY ACTIONABLE BEZ235 DACTOLISIB 26206338 55965 38230 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TDR78834 CHEMBL1507526 55966 38231 HBB 3043 DRUGGABLE GENOME, ENZYME HQK-1001 SODIUM 2,2-DIMETHYLBUTYRATE 55967 38232 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Neostigmine NEOSTIGMINE 55968 38233 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DEXAMETHASONE VALARATE DEXAMETHASONE VALARATE 55969 38234 POLI 11201 DNA REPAIR ERGOCORNINE ERGOCORNINE 55970 38235 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ENMD-2076 ENMD-2076 55971 38236 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BDBM50080570 55972 38237 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-4674 CHEMBL584452 55974 38238 MAPKAPK5 8550 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565857 55976 38239 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME DOVITINIB DOVITINIB 55978 38240 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652029 55979 38241 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 374883849 TRIFAROTENE 55980 38242 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-9 55981 38243 MBP 4155 CELL SURFACE INTERFERON BETA-1A 10932275 55984 38244 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652023 55986 38245 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor MK4827 NIRAPARIB 55987 38246 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Fesoterodine FESOTERODINE 55988 38247 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME S(+)-RACLOPRIDE L-TARTRATE CHEMBL1369632 55991 38248 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME ADAVOSERTIB ADAVOSERTIB 23270927,24305702 55992 38249 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3544998 LY-3007113 55993 38250 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4'-EPICHAETOVIRIDIN A CHEMBL1306556 55996 38251 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE allosteric modulator 310264748 55999 38252 TNKS2 80351 DRUGGABLE GENOME, ENZYME PMID27841036-Compound-37 56000 38253 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LIMONIN LIMONIN 56001 38254 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER GSK1614235 GSK-1614235 56002 38255 ATXN2 6311 NA MMV000634 CHEMBL602946 56003 38256 DPP7 29952 PROTEASE, ENZYME, DRUGGABLE GENOME BDBM50434165 56004 38257 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-58 56005 38258 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PYRAZINAMIDE PYRAZINAMIDE 22931300 56007 38259 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody RITUXIMAB RITUXIMAB 56008 38260 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENAZINE-1-CARBOXYLIC ACID PHENAZINE-1-CARBOXYLIC ACID 56009 38261 TUBB 203068 DRUGGABLE GENOME inhibitor 178103391 VINCRISTINE 56011 38262 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor GDC-0980 APITOLISIB 56012 38263 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649747 56013 38264 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist 381745013 56014 38265 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000029700 CHEMBL591864 56015 38266 PSMD8 5714 NA CARFILZOMIB CARFILZOMIB 24524217 56017 38267 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PHA-665752 PHA-665752 24165158,21266357,23542356 56018 38268 ALOX5 240 DRUGGABLE GENOME, ENZYME MELATONIN MELATONIN 10668425 56020 38269 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 329968436 56021 38270 BCHE 590 DRUGGABLE GENOME, ENZYME donepezil DONEPEZIL 18780301,27567841,27911294,17047484 56022 38271 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME PHENOXODIOL 56023 38272 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Dapsone DAPSONE 56024 38273 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR HOMATROPINE METHYLBROMIDE 56026 38274 UCP2 7351 TRANSPORTER, DRUGGABLE GENOME SALINE SODIUM CHLORIDE 10868951 56027 38275 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME IPRATROPIUM IPRATROPIUM 56028 38276 PTGS1 5742 ENZYME, DRUGGABLE GENOME SULINDAC SULINDAC 56029 38277 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1417529 CHEMBL1990783 56030 38278 ADH1B 125 DRUGGABLE GENOME, ENZYME FOMEPIZOLE FOMEPIZOLE 56031 38279 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME ASP8497 56033 38280 POLK 51426 DNA REPAIR, ENZYME ACRIFLAVINE CHLORIDE ACRIFLAVINE 56034 38281 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MERCAPTOPURINE MERCAPTOPURINE 22931300 56037 38282 TUBB2A 7280 DRUGGABLE GENOME ABT-751 ABT-751 25468039 56038 38283 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME EPINEPHRINE BITARTRATE EPINEPHRINE BITARTRATE 56040 38284 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME PRAZOSIN PRAZOSIN 23073734 56043 38285 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME TAMOXIFEN CITRATE TAMOXIFEN CITRATE 56044 38286 TSPO 706 DRUGGABLE GENOME Benzothiazepine analog 7 56047 38287 GMNN 51053 DRUGGABLE GENOME GR-127935 GR-127935 56048 38288 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL751 BROMFENAC SODIUM 56049 38289 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL117785 TETRABENAZINE 56050 38290 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Everolimus EVEROLIMUS 56051 38291 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME PMID27998201-Compound-12 56052 38292 GMNN 51053 DRUGGABLE GENOME NSC-95397 CHEMBL429095 56053 38293 TSC22D3 1831 NA CORTICOSTEROIDS 17208592 56055 38294 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL1201149 NALTREXONE HYDROCHLORIDE 56056 38295 COL6A1 1291 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 56057 38296 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL BUTETHAL BUTETHAL 56058 38297 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE methotrexate METHOTREXATE 16822847 56059 38298 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR TRICHOSTATIN A 17392473 56060 38299 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545300 CP-459632 56061 38300 TUBA1C 84790 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 56062 38301 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649923 56063 38302 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE AMG900 AMG-900 56064 38303 NFKBIA 4792 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PEPEROMIN E PEPEROMIN E 19559609 56065 38304 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TESAGLITAZAR TESAGLITAZAR 56066 38305 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PHENAZINE-2,3-DIAMINE CHEMBL274921 56068 38306 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME FAS LIGAND 15809706 56069 38307 CDK13 8621 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL3544942 RONICICLIB 56070 38308 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE VX-970 BERZOSERTIB 56072 38309 HMGCR 3156 ENZYME, DRUGGABLE GENOME Quinoline derivative 16 56073 38310 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Articaine ARTICAINE 56076 38311 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PYRROLIDINE DITHIOCARBAMATE PYRROLIDINE DITHIOCARBAMATE 56077 38312 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE DOVITINIB DOVITINIB 56078 38313 LIPC 3990 ENZYME, PHOSPHOLIPASE, LIPASE, DRUGGABLE GENOME ATORVASTATIN ATORVASTATIN 12547874 56081 38314 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME LY-2463665 56082 38315 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AEE-788 AEE-788 56083 38316 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE NIRAPARIB NIRAPARIB 56086 38317 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE morphine MORPHINE 32090339 56087 38318 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE AD-03 24353405 56089 38319 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Testosterone TESTOSTERONE 56090 38320 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 6,4'-DIMETHOXYFLAVONE 6,4'-DIMETHOXYFLAVONE 56092 38321 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 315661269 56093 38322 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MINOCYCLINE MINOCYCLINE 22931300 56094 38323 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME phenytoin PHENYTOIN 17638512 56095 38324 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-(PHENOXYMETHYL)BENZOTHIAZOLE 2-(PHENOXYMETHYL)BENZOTHIAZOLE 56096 38325 EZR 7430 CLINICALLY ACTIONABLE, KINASE RO 31-8220 9124348 56097 38326 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 385612188 56098 38327 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX BMS-204493 CHEMBL472172 19216008,18702457 56100 38328 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL FLURAZEPAM FLURAZEPAM 56102 38329 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TREQUINSIN HYDROCHLORIDE TREQUINSIN HYDROCHLORIDE 56103 38330 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PROMEGAPOIETIN 11602319 56105 38331 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME CAMPTOTHECIN CAMPTOTHECIN 9758415 56108 38332 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000240587 CHEMBL592834 56109 38333 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW828525X GW828525X 56110 38334 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME unspecified PD-1 antibody 26645196 56111 38335 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE FENTICLOR FENTICLOR 56112 38336 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FELBAMATE FELBAMATE 22931300 56113 38337 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-54 56114 38338 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1201119 LIOTHYRONINE SODIUM 56115 38339 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME ILORASERTIB ILORASERTIB 56116 38340 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201044 DAPIPRAZOLE HYDROCHLORIDE 56117 38341 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Navitoclax NAVITOCLAX 26474387 56118 38342 PDE1A 5136 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL932 DIPYRIDAMOLE 56119 38343 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Pidilizumab PIDILIZUMAB 56120 38344 SLC38A4 55089 TRANSPORTER 178100907 56121 38345 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor AS703569 CENISERTIB 56122 38346 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL189963 PALBOCICLIB 56125 38347 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE TAE-684 TAE-684 56126 38348 MAPT 4137 DRUGGABLE GENOME TCMDC-124022 CHEMBL548017 56128 38349 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME ERLOTINIB ERLOTINIB 56129 38350 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DIETHYLSTILBESTROL DIETHYLSTILBESTROL 22931300 56130 38351 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME INDIRUBIN SULFATE SU-9516 56132 38352 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE modulator CHEMBL2346976 AZD3514 56133 38353 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MIBEFRADIL DIHYDROCHLORIDE MIBEFRADIL DIHYDROCHLORIDE 56134 38354 PNPLA3 80339 ENZYME ethanol ALCOHOL 30132178 56135 38355 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL1822792 MK-2461 56136 38356 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL blocker 340590214 56137 38357 PRMT1 3276 ENZYME, METHYL TRANSFERASE NSC-47762 CHEMBL1092740 20666457 56138 38358 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 381118818 56140 38359 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 2'-METHOXYFORMONETIN 2'-METHOXYFORMONETIN 56141 38360 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE XMT-1522 56142 38361 KDM4A 9682 DRUGGABLE GENOME, ENZYME BROXYQUINOLINE BROXYQUINOLINE 56143 38362 GMNN 51053 DRUGGABLE GENOME BENZO[DEF]CHRYSENE BENZO[DEF]CHRYSENE 56144 38363 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME RO4987655 RO-4987655 26438159 56145 38364 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OLMESARTAN OLMESARTAN 56146 38365 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE gefitinib GEFITINIB 56147 38366 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROPARGITE PROPARGITE 56149 38367 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565690 CHEMBL188678 56150 38368 ZNF385D 79750 NA duloxetine DULOXETINE 29407288,28696415 56151 38369 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME PMID27998201-Compound-9 56152 38370 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-3641 CHEMBL599098 56153 38371 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME LOMATIN LOMATIN 56155 38372 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PF-06463922 LORLATINIB 28285684 56156 38373 APOE 348 DRUGGABLE GENOME NORETHISTERONE ACETATE 12398019 56158 38374 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AY-9944 CHEMBL1513392 56159 38375 GMNN 51053 DRUGGABLE GENOME CAPENSIN CAPENSIN 56161 38376 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TRIBUTYRIN TRIBUTYRIN 11593538 56162 38377 GPER1 2852 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR ESTRADIOL ESTRADIOL 16520733 56163 38378 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME VALPROIC ACID VALPROIC ACID 18294844,16921367,25304896 56164 38379 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE TIVOZANIB TIVOZANIB 56168 38380 GLA 2717 ENZYME, DRUGGABLE GENOME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 56169 38381 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 249565802 56170 38382 BAZ2B 29994 NA MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 56172 38383 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE URIDINE URIDINE 9030547 56173 38384 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME NSC-50690 CHEMBL1388703 56174 38385 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE PD-0166285 PD-0166285 56175 38386 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 56176 38387 POLK 51426 DNA REPAIR, ENZYME DIENOCHLOR DIENOCHLOR 56177 38388 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1558 PRAZOSIN HYDROCHLORIDE 56178 38389 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR THIORIDAZINE THIORIDAZINE 56179 38390 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 4-PHENOXY-BENZOIC ACID CHEMBL107518 22487179 56180 38391 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SPERMIDINE SPERMIDINE 56183 38392 PRNP 5621 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME BREFELDIN A BREFELDIN A 56184 38393 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME FLUTAMIDE FLUTAMIDE 7541862 56186 38394 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE RADIATION THERAPY 18386816 56187 38395 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CANDESARTAN CANDESARTAN 56188 38396 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TIOTIDINE TIOTIDINE 56189 38397 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE 17-AAG TANESPIMYCIN 16267832 56194 38398 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME XCT790 CHEMBL189753 56196 38399 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GW7647 GW7647 56197 38400 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE NSC-407228 CHEMBL74852 56199 38401 NOTCH3 4854 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Tarextumab TAREXTUMAB 56202 38402 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 404859044 56203 38403 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 223366031 56204 38404 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RESVERATROL RESVERATROL 15122319 56205 38405 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE TGAAC94 56210 38406 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE CYTOSINE ARABINOSIDE 2676043 56212 38407 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL3545252 DOCETAXEL 56213 38408 HEBP1 50865 DRUGGABLE GENOME Chalcone derivative 3 56214 38409 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR DOXORUBICIN DOXORUBICIN 12956904 56216 38410 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME olmesartan OLMESARTAN 18641915 56218 38411 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-402083 CHEMBL1546228 56219 38412 ENOSF1 55556 ENZYME AZT ZIDOVUDINE 15980332 56221 38413 KDM4A 9682 DRUGGABLE GENOME, ENZYME ISOPROPAMIDE IODIDE ISOPROPAMIDE IODIDE 56222 38414 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-93 56223 38415 CASP2 835 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178101981 56224 38416 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GLYBURIDE GLYBURIDE 26384286 56228 38417 PTK6 5753 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, ENZYME TAMATINIB R-406 56229 38418 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1531 ETONOGESTREL 56230 38419 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NONIVAMIDE NONIVAMIDE 56231 38420 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CODEINE CODEINE 18311899 56232 38421 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME A-77636 CHEMBL291143 56233 38422 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE INFLIXIMAB INFLIXIMAB 56234 38423 EEF2 1938 DRUGGABLE GENOME, KINASE LACTIMIDOMYCIN LACTIMIDOMYCIN 20118940 56236 38424 PDE3B 5140 ENZYME, DRUGGABLE GENOME RPL-554 56237 38425 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LACTOFEN LACTOFEN 56238 38426 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker CHEMBL3545352 P-1037 56241 38427 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL2103884 OPROZOMIB 56242 38428 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME 178100419 56243 38429 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 310264698 AMG-319 56244 38430 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME MLN2480 56247 38431 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CAMPTOTHECIN CAMPTOTHECIN 10777774 56249 38432 APC 324 CLINICALLY ACTIONABLE IWR-1 28179481 56250 38433 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 56251 38434 WNK3 65267 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME inhibitor 249565818 56256 38435 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 56258 38436 MPHOSPH8 54737 NA GNF-PF-5510 CHEMBL578741 56259 38437 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME LEVODOPA LEVODOPA 56260 38438 BRCA2 675 CLINICALLY ACTIONABLE Talazoparib TALAZOPARIB 26546619,23881923,28242752 56261 38439 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AZD8055 AZD-8055 25436981 56262 38440 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor CHEMBL3039507 SOTAGLIFLOZIN 56264 38441 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NXN-188 56266 38442 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HEXACHLOROPHENE HEXACHLOROPHENE 56268 38443 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ACETOCHLOR ACETOCHLOR 56269 38444 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME MUC1-Poly-ICLC 56270 38445 POLI 11201 DNA REPAIR APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 56271 38446 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650478 56272 38447 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME TCMDC-123912 CHEMBL106525 56275 38448 POLK 51426 DNA REPAIR, ENZYME PHANQUONE PHANQUONE 56276 38449 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE INSULIN INSULIN 8766822 56277 38450 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME BAS03450373 CHEMBL1576310 56279 38451 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-P1 56280 38452 SMN1 6606 DRUGGABLE GENOME 7-METHOXY-BAPTIGENIN CHEMBL583578 56281 38453 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102445 TREPROSTINIL 56282 38454 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME BAS-0338868 CHEMBL378903 56283 38455 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL1743005 DACETUZUMAB 56284 38456 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL969 PRAZEPAM 56285 38457 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE E927A E927A 56286 38458 POLI 11201 DNA REPAIR SJ000044511 CHEMBL592124 56287 38459 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL1200622 PARICALCITOL 56289 38460 TNNT3 7140 NA activator CHEMBL3039529 TIRASEMTIV 56291 38461 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 404859149 56292 38462 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ILORASERTIB ILORASERTIB 56293 38463 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TETANUS TOXOID 9694951 56294 38464 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE INOSITOL INOSITOL 1648562 56296 38465 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME OMIPALISIB OMIPALISIB 23431193 56297 38466 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 348353622 56298 38467 ICAM3 3385 DRUGGABLE GENOME PMA 7525295 56299 38468 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR 4-NONYLPHENOL 4-NONYLPHENOL 56300 38469 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SPHINX scaffold, 3 56301 38470 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE MODIFIED IFN-BETA 56303 38471 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CARVEDILOL CARVEDILOL 56305 38472 FKBP5 2289 DRUGGABLE GENOME antidepressants 18597649,21449676,20709156,19676097,15565110,23733030,17467808 56306 38473 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME GNF-PF-1656 CHEMBL579028 56307 38474 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL2103829 FAXELADOL 56309 38475 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 pioglitazone PIOGLITAZONE 28099407 56311 38476 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GW843682X GW843682X 56312 38477 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL1201008 IBANDRONATE SODIUM 56313 38478 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651527 56314 38479 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PYRITHIONE PYRITHIONE 56316 38480 ATAD5 79915 NA SIB-1893 CHEMBL88612 56317 38481 PTGS1 5742 ENZYME, DRUGGABLE GENOME NAPROXEN NAPROXEN 56318 38482 CXCL8 3576 DRUGGABLE GENOME PYROGALLOL PYROGALLOL 56320 38483 TARDBP 23435 TUMOR SUPPRESSOR T091317 T091317 56321 38484 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE HSP70 11821413 56322 38485 NDUFB7 4713 ENZYME inhibitor CHEMBL3545320 ME-344 56323 38486 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-22 56325 38487 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BAY-613606 CHEMBL541400 56327 38488 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ARACHIDONIC ACID ARACHIDONIC ACID 56328 38489 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DOMIPHEN BROMIDE DOMIPHEN BROMIDE 56329 38490 UBE2N 7334 ENZYME, DRUGGABLE GENOME SPERMINE TETRAHYDROCHLORIDE SPERMINE TETRAHYDROCHLORIDE 56332 38491 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Aceprometazine ACEPROMETAZINE 56334 38492 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR ERBSTATIN ERBSTATIN 56336 38493 MAPT 4137 DRUGGABLE GENOME U-0126 U-0126 56337 38494 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1318477 CHEMBL428064 56338 38495 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-11 56339 38496 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamate derivative 15 56341 38497 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TOSYL-L-LYSINE CHLOROMETHYL KETONE CHEMBL466465 56342 38498 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor 249565736 56344 38499 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE TAE-684 TAE-684 56345 38500 ATXN2 6311 NA GNF-PF-1969 CHEMBL601364 56346 38501 RGS4 5999 DRUGGABLE GENOME SB-415286 CHEMBL322970 56347 38502 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME RESVERATROL RESVERATROL 56348 38503 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME 6-HYDROXYMELATONIN CHEMBL127421 56349 38504 TUBB2B 347733 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 56352 38505 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-72 56353 38506 NTS 4922 DRUGGABLE GENOME RISPERIDONE RISPERIDONE 10991962 56354 38507 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHEMBL1102 GLUTETHIMIDE 56355 38508 ALOX5 240 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL876 MECLOFENAMATE SODIUM 56356 38509 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHLORAMPHENICOL CHLORAMPHENICOL 14576103 56359 38510 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor TIVANTINIB TIVANTINIB 56360 38511 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME flupenthixol E-FLUPENTIXOL 56361 38512 GRK2 156 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 249565823 56367 38513 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178101011 FLURBIPROFEN 56368 38514 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BI-69A11 26603897 56369 38515 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (+)-ELEUTHERIN CHEMBL594153 19783445 56370 38516 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Alpelisib ALPELISIB 27659046,27924459 56371 38517 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHEMBL591 ETHCHLORVYNOL 56372 38518 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SOTORASIB 31666701,31239544,31776128 56373 38519 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID29757691-Compound-8d 56375 38520 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-1919 CHEMBL576409 56377 38521 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE VEGFRECINE VEGFRECINE 56379 38522 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE KHELLIN KHELLIN 56380 38523 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ALFENTANIL ALFENTANIL 56381 38524 GMNN 51053 DRUGGABLE GENOME SJ000032081 CHEMBL590184 56382 38525 CHRNA5 1138 DRUGGABLE GENOME, ION CHANNEL Opium alkaloids and derivatives 20725741 56384 38526 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C10 56387 38527 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR methotrexate METHOTREXATE 24141364 56388 38528 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL58323 ERLOSAMIDE 56389 38529 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-254 CHEMBL461579 56390 38530 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CHLOROTRIANISENE CHLOROTRIANISENE 56391 38531 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ADRIAMYCIN ADRIAMYCIN 7723242 56393 38532 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY olanzapine OLANZAPINE 24624910 56395 38533 POLI 11201 DNA REPAIR ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 56397 38534 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Cytarabine CYTARABINE 18986703 56399 38535 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZEARALENONE ZEARALENONE 56400 38536 TARDBP 23435 TUMOR SUPPRESSOR NSC-139257 CHEMBL1256364 56401 38537 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME inhibitor 178103596 56403 38538 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651133 56404 38539 PDE4B 5142 DRUGGABLE GENOME, ENZYME CAFFEINE CAFFEINE 56405 38540 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR METHYLENE BLUE METHYLENE BLUE 56406 38541 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ADAPALENE ADAPALENE 56407 38542 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL628 PENTOXIFYLLINE 56409 38543 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1200444 PIRBUTEROL ACETATE 56410 38544 XDH 7498 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1164729 FEBUXOSTAT 56412 38545 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 5,7-DIHYDROXYISOFLAVONE 5,7-DIHYDROXYISOFLAVONE 56415 38546 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE PMID26882240-Compound-1 56416 38547 BAZ2B 29994 NA MICONAZOLE NITRATE MICONAZOLE NITRATE 56417 38548 DROSHA 29102 NA methotrexate METHOTREXATE 24614921 56419 38549 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE mycophenolic acid 24220207,25163792 56420 38550 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200794 OXYMORPHONE HYDROCHLORIDE 56422 38551 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor 178101857 CILOSTAMIDE 56423 38552 GMNN 51053 DRUGGABLE GENOME CID 94381 CHEMBL374632 56424 38553 GBA 2629 DRUGGABLE GENOME, ENZYME CIRSIMARITIN CIRSIMARITIN 56425 38554 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME LOMOFUNGIN LOMOFUNGIN 56426 38555 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME HARMALINE HARMALINE 56430 38556 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TAE-684 TAE-684 56431 38557 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR GALLIUM NITRATE 8788232 56433 38558 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL blocker,activator 178101120 RYANODINE 56435 38559 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ORYZALIN ORYZALIN 56438 38560 TUBB 203068 DRUGGABLE GENOME inhibitor 178103404 CABAZITAXEL 56440 38561 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER N6-BENZYLADENOSINE N6-BENZYLADENOSINE 56441 38562 BAZ2B 29994 NA REMACEMIDE HYDROCHLORIDE REMACEMIDE HYDROCHLORIDE 56442 38563 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125110 CHEMBL580816 56443 38564 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE FLUNARIZINE DIHYDROCHLORIDE FLUNARIZINE DIHYDROCHLORIDE 56444 38565 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE T091317 T091317 56446 38566 ALOX15B 247 DRUGGABLE GENOME, ENZYME inhibitor 252827408 56447 38567 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-47 56448 38568 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GMI-1070 RIVIPANSEL 20508165 56449 38569 HKDC1 80201 DRUGGABLE GENOME, KINASE CHLORHEXIDINE CHLORHEXIDINE 56452 38570 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL 1,2,4-triazole derivative 4 56453 38571 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 hydrocortisone HYDROCORTISONE 9187528 56455 38572 ATF2 1386 TRANSCRIPTION FACTOR fentanyl FENTANYL 30106255 56456 38573 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL223360 LINIFANIB 56458 38574 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-67 56459 38575 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE CHELATORS 9144774 56460 38576 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MIM-D3 TAVILERMIDE 23836957 56461 38577 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist 135651418 ALITRETINOIN 56462 38578 INPP5D 3635 DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 336446950 56464 38579 FAAH 2166 ENZYME, DRUGGABLE GENOME Aryl urea derivative 1 56465 38580 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE NSAID 12654560 56470 38581 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 363894219 BALAMAPIMOD 56472 38582 IL6ST 3572 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE antagonist CHEMBL3833307 SATRALIZUMAB 56473 38583 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIETHYLSTILBESTROL DIETHYLSTILBESTROL 56474 38584 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Rituximab RITUXIMAB 56477 38585 GMNN 51053 DRUGGABLE GENOME DIPHENOXYLATE HYDROCHLORIDE DIPHENOXYLATE HYDROCHLORIDE 56478 38586 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 252827414 56479 38587 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DESACETYL SALANNIN DESACETYL SALANNIN 56481 38588 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CAPTAN CAPTAN 56482 38589 HLA-DQB1 3119 CLINICALLY ACTIONABLE bucillamine BUCILLAMINE 56486 38590 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GR-55562 GR-55562 56487 38591 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE EGCG EPIGALOCATECHIN GALLATE 18591783 56488 38592 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER vecuronium VECURONIUM 56489 38593 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME TAMATINIB R-406 56490 38594 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR TYRPHOSTIN 23 TYRPHOSTIN 23 56491 38595 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE SYD985 TRASTUZUMAB DUOCARMAZINE 25589493,27256376 56493 38596 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE RG-1530 RG-1530 56495 38597 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE RXDX 101 56497 38598 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE DS-7423 DS-7423 24504419 56498 38599 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL1200782 DEXTROAMPHETAMINE ADIPATE 56500 38600 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR THROMBOLYTIC AGENT 11041123 56502 38601 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist 178100912 56503 38602 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OXPRENOLOL OXPRENOLOL 56504 38603 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CHEMBL2109391 MDX-447 56505 38604 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102290 AT-7519 56506 38605 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE BISACODYL BISACODYL 56507 38606 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 56508 38607 GMNN 51053 DRUGGABLE GENOME TCMDC-123764 CHEMBL533226 56512 38608 PDE4A 5141 DRUGGABLE GENOME, ENZYME OGLEMILAST OGLEMILAST 56513 38609 MAPT 4137 DRUGGABLE GENOME CATECHIN CATECHIN 56515 38610 RPS6KA6 27330 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME inhibitor 404859044 56517 38611 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3402762 TEPOTINIB 56518 38612 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME DITHIOLETHIONE DITHIOLETHIONE 56519 38613 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME U-50488 METHANE SULFONATE U-50488 METHANE SULFONATE 56520 38614 PDE4C 5143 DRUGGABLE GENOME, ENZYME ETAZOLATE ETAZOLATE 56522 38615 HDAC11 79885 DRUGGABLE GENOME, ENZYME BELINOSTAT BELINOSTAT 25937017 56523 38616 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CLM3 24423321 56524 38617 BMP2K 55589 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 223366123 BARICITINIB 56525 38618 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR inhibitor 249565917 56526 38619 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor OSI-027 OSI-027 56529 38620 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DNDI1267127 CHEMBL135115 56531 38621 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178103766 FROVATRIPTAN 56534 38622 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 252166595 BIMIRALISIB 56539 38623 YWHAE 7531 CLINICALLY ACTIONABLE INSULIN INSULIN 16216880 56541 38624 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565858 56542 38625 COL2A1 1280 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 56544 38626 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE SUNITINIB SUNITINIB 15928335,15685537,22718859,16638875,15146165,12949711,26130666,25157968,14645423,16954519,18794084,22745105 56545 38627 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SERTINDOLE SERTINDOLE 56546 38628 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Alkylating Agents 18652519 56547 38629 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE lidocaine and tetracaine 56548 38630 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124066 CHEMBL529741 56552 38631 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CAP7.1 56553 38632 PPT1 5538 ENZYME, DRUGGABLE GENOME LAMOTRIGINE LAMOTRIGINE 9151331 56554 38633 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME DIPLAMINE B DIPLAMINE B 18977148 56556 38634 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TCMDC-124166 CHEMBL528712 56557 38635 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 187051780 TAPENTADOL 56560 38636 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE CX-072 CX-072 56561 38637 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE MELATONIN MELATONIN 7629697 56562 38638 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-107 CHEMBL578675 56563 38639 BCHE 590 DRUGGABLE GENOME, ENZYME PMID29757691-Compound-2a-i 56566 38640 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR diuretics 22543981 56567 38641 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL932 DIPYRIDAMOLE 56568 38642 HSPA1A 3303 DRUGGABLE GENOME AIMPILA 56569 38643 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE RUTIN RUTIN 12423426 56574 38644 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR N-(3-CHLOROPHENYL)PICOLINAMIDE CHEMBL556667 56575 38645 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TOREMIFENE TOREMIFENE 56576 38646 RAC1 5879 CLINICALLY ACTIONABLE, KINASE, DRUG RESISTANCE ZU-3594419 CHEMBL562095 19527032 56578 38647 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CAPROSPINOL CAPROSPINOL 56580 38648 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Carbamide derivative 22 56581 38649 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE BGJ398 INFIGRATINIB 56582 38650 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103626 ZONISAMIDE 56587 38651 LEPR 3953 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME agonist CHEMBL2107857 METRELEPTIN 56588 38652 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 252166658 SPARSENTAN 56589 38653 IMPDH1 3614 ENZYME, DRUGGABLE GENOME inhibitor 178103438 56590 38654 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FLUCONAZOLE FLUCONAZOLE 22931300 56591 38655 PBK 55872 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, ENZYME GEFITINIB GEFITINIB 26745678 56594 38656 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING BENZENETHIOL BENZENETHIOL 56595 38657 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER lenalidomide LENALIDOMIDE 29177954 56596 38658 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR YM-598 NEBENTAN 21232046 56597 38659 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME ALVOCIDIB ALVOCIDIB 18469809 56598 38660 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SJ000113257 CHEMBL528694 56599 38661 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE CYC-116 CYC-116 56603 38662 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL482767 SNS-314 56604 38663 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROPRANOLOL PROPRANOLOL 56605 38664 SLC28A2 9153 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME inhibitor 252166693 56606 38665 BCHE 590 DRUGGABLE GENOME, ENZYME (-)-Phenserine 56607 38666 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8536181, C17 56610 38667 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME BENZO[DEF]CHRYSENE BENZO[DEF]CHRYSENE 14684315 56611 38668 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METHOTRIMEPRAZINE LEVOMEPROMAZINE 56613 38669 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME RG-1530 RG-1530 56614 38670 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE Trametinib TRAMETINIB 27821489 56615 38671 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DOMIPHEN BROMIDE DOMIPHEN BROMIDE 56616 38672 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor GDC-0068 IPATASERTIB 56618 38673 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL272980 MOCETINOSTAT 56619 38674 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR ORLISTAT ORLISTAT 11410822 56620 38675 VEGFC 7424 GROWTH FACTOR, TRANSPORTER, DRUGGABLE GENOME inhibitor SORAFENIB TOSYLATE 56621 38676 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DICHLORODIPHENYLDICHLOROETHYLENE DICHLORODIPHENYLDICHLOROETHYLENE 56622 38677 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 11 56624 38678 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME NIACIN NIACIN 56626 38679 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME FOLFOX 27002107 56627 38680 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1370561 AMINOPHYLLINE 56628 38681 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL3545133 JNJ-26483327 56630 38682 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Ethylestrenol ETHYLESTRENOL 56631 38683 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GR-103545 CHEMBL277863 56632 38684 NPEPPS 9520 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 252166871 ANTAQ 56633 38685 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Bezafibrate BEZAFIBRATE 56634 38686 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME PMA 7488650 56635 38687 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE CARBOGEN CARBOGEN 12915890 56636 38688 F2RL3 9002 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100719 56638 38689 NOS2 4843 DRUGGABLE GENOME, ENZYME inhibitor 178101930 56639 38690 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650195 56642 38691 POLI 11201 DNA REPAIR ZINC 03369470 CHEMBL599013 56645 38692 BUB1 699 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565792 56649 38693 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX CID 4101591 CHEMBL428789 56650 38694 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME MIDAZOLAM MIDAZOLAM 56652 38695 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-466317A GSK-466317A 56653 38696 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CID 1245272 CHEMBL408850 56654 38697 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651843 56655 38698 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Binimetinib BINIMETINIB 28514312 56656 38699 ATXN2 6311 NA SPHAEROPSIDIN A SPHAEROPSIDIN A 56657 38700 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ED-71 ELDECALCITOL 56658 38701 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME CSA CYCLOSPORINE 17031644 56659 38702 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 2-PHENYLPHENOL 2-PHENYLPHENOL 56663 38703 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000112730 CHEMBL591178 56665 38704 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ORPHENADRINE ORPHENADRINE 56666 38705 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051799 DACINOSTAT 56668 38706 MAOA 4128 DRUGGABLE GENOME, ENZYME CHF-3381 INDANTADOL 56669 38707 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME CLARITHROMYCIN CLARITHROMYCIN 18212111 56670 38708 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR oxycodone OXYCODONE 27472837 56671 38709 ABCC5 10057 DRUGGABLE GENOME, ABC TRANSPORTER, TRANSPORTER fluorouracil FLUOROURACIL 26352872 56673 38710 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE GDC-0068 IPATASERTIB 56675 38711 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178102587 56676 38712 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE ALDISIN ALDISIN 21696953 56677 38713 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL448 PENTOBARBITAL 56678 38714 BCHE 590 DRUGGABLE GENOME, ENZYME Isochroman-4-ketone derivative 1 56680 38715 POLI 11201 DNA REPAIR CEFUROXIME SODIUM CEFUROXIME SODIUM 56681 38716 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME HALOPERIDOL HALOPERIDOL 8851165 56683 38717 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CORTICOSTERONE CORTICOSTERONE 56684 38718 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HALOFANTRINE HYDROCHLORIDE HALOFANTRINE HYDROCHLORIDE 56687 38719 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME AST-487 AST-487 56688 38720 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE ONC201 ONC-201 26474387 56690 38721 PON1 5444 ENZYME, TRANSPORTER, DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 56691 38722 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HOMIDIUM BROMIDE HOMIDIUM BROMIDE 56692 38723 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2012832440110 56694 38724 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-3832 CHEMBL261693 56695 38725 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ETHACRYNIC ACID 8010986 56697 38726 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE LINIFANIB LINIFANIB 56698 38727 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 cocaine COCAINE 9187528 56699 38728 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUROCHLORIDONE FLUROCHLORIDONE 56700 38729 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Tricyclic heterocycle derivative 1 56701 38730 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE BOSUTINIB BOSUTINIB 56707 38731 HSPB2 3316 KINASE TAMOXIFEN TAMOXIFEN 9607585 56709 38732 DSP 1832 NA ENALAPRIL ENALAPRIL 10839195 56710 38733 GMNN 51053 DRUGGABLE GENOME TCMDC-124280 CHEMBL528492 56711 38734 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME N/A 26768652 56712 38735 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME TOZASERTIB TOZASERTIB 56715 38736 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME STILONIUM IODIDE STILONIUM IODIDE 56716 38737 E2F1 1869 TRANSCRIPTION FACTOR ETOPOSIDE ETOPOSIDE 9766655,16849574 56718 38738 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE ASN003 56719 38739 GUCA2A 2980 DRUGGABLE GENOME, ENZYME, HORMONE ACTIVITY LACTOSE LACTOSE, ANHYDROUS 11677212 56720 38740 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Ipilimumab IPILIMUMAB 56721 38741 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR NCG-C00093820-01 CHEMBL544115 56722 38742 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME IL-1 12606540 56725 38743 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ATOMOXETINE ATOMOXETINE 56727 38744 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME EGS-21 56731 38745 TXK 7294 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 249565852 56735 38746 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-51 56737 38747 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-42 56739 38748 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Thioguanine THIOGUANINE 56740 38749 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METHOTRIMEPRAZINE LEVOMEPROMAZINE 56741 38750 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 2,7-BIS[3-(PIPERAZINO)PROPIONAMIDO]ANTHRAQUINONE CHEMBL520095 18571928 56743 38751 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor HTS-466284 CHEMBL261454 19035792 56744 38752 ATAD5 79915 NA GNF-PF-860 CHEMBL593254 56745 38753 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TAE-684 TAE-684 56746 38754 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-9037 CHEMBL1451216 56747 38755 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME N-methylmethanesulfonamide derivative 1 56748 38756 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME PMID27539678-Compound-14 56749 38757 TUBB6 84617 DRUGGABLE GENOME CHEMBL2108628 PACLITAXEL POLIGLUMEX 56750 38758 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BAS-8770954 CHEMBL478324 19179076 56751 38759 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 HOMATROPINE METHYLBROMIDE HOMATROPINE METHYLBROMIDE 22931300 56752 38760 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE Plevitrexed (R)-isomer 56753 38761 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE FASUDIL FASUDIL 56754 38762 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 56755 38763 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DOXORUBICIN DOXORUBICIN 21388138,26211460,20170164,22276998 56756 38764 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-1737 CHEMBL531710 56757 38765 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor TOZASERTIB TOZASERTIB 19035792 56758 38766 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME SAR-114137 56760 38767 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR CISPLATIN CISPLATIN 28490518 56761 38768 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME 13-CIS RETINOIC ACID 17916375 56762 38769 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME GENTAMICIN GENTAMICIN 9792955 56764 38770 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-228357 CHEMBL14276 56765 38771 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Dabrafenib DABRAFENIB 56766 38772 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-21 56768 38773 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR DNDI1417467 CHEMBL1997335 56769 38774 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME YM443 56772 38775 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DOV 102,677 56773 38776 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE AZD-1775 ADAVOSERTIB 56775 38777 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 310264690 LAROTRECTINIB 56778 38778 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SCH-58261 SCH-58261 56780 38779 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR C326 56781 38780 MAPT 4137 DRUGGABLE GENOME TCMDC-124055 CHEMBL546576 56782 38781 CA1 759 DRUGGABLE GENOME, ENZYME activator 135651430 56783 38782 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BREFELDIN A BREFELDIN A 56785 38783 MAOB 4129 DRUGGABLE GENOME, ENZYME RG1577 56786 38784 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BGJ398 INFIGRATINIB 56789 38785 SCD 6319 DRUGGABLE GENOME, ENZYME VITAMIN A 12538081 56790 38786 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SKF-62604 CHEMBL346551 56791 38787 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 omeprazole OMEPRAZOLE 9187528 56792 38788 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL386630 TESTOSTERONE 56796 38789 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200409 LIDOCAINE HYDROCHLORIDE 56798 38790 APCS 325 TRANSPORTER, DRUGGABLE GENOME antibody 249565935 DEZAMIZUMAB 56799 38791 TXNRD1 7296 DRUGGABLE GENOME Terpyridineplatinum(II) complexe 3 56800 38792 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor GDC-0941 PICTILISIB 56805 38793 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Durvalumab DURVALUMAB 56807 38794 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Imidazo[1,2-b]pyridazine derivative 4 56809 38795 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-123579 CHEMBL533954 56810 38796 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652413 56811 38797 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MBL 15766398 56813 38798 DHODH 1723 DRUGGABLE GENOME, ENZYME Vidofludimus VIDOFLUDIMUS 56815 38799 GAL 51083 DRUGGABLE GENOME TRIIODOTHYRONINE LIOTHYRONINE SODIUM 12147214 56817 38800 ABAT 18 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL89598 VIGABATRIN 56818 38801 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR DNDI1417400 CHEMBL1362503 56819 38802 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ACID BLUE 129 ACID BLUE 129 56822 38803 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE OXYCODONE OXYCODONE 56824 38804 BAZ2B 29994 NA GNF-PF-4459 CHEMBL585502 56825 38805 EPHA3 2042 ENZYME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565821 56826 38806 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417400 CHEMBL1362503 56827 38807 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178103114 56828 38808 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME SB-204741 CHEMBL323356 56829 38809 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE CYCLOSPORIN 10679127 56830 38810 KDM4A 9682 DRUGGABLE GENOME, ENZYME DISULFIRAM DISULFIRAM 56831 38811 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 348353622 56832 38812 PDE5A 8654 ENZYME, DRUGGABLE GENOME DIPYRIDAMOLE DIPYRIDAMOLE 56834 38813 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL919 FOSPHENYTOIN SODIUM 56835 38814 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX TCMDC-123532 CHEMBL547833 56836 38815 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE 56837 38816 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4665 CHEMBL601744 56838 38817 HTT 3064 DRUGGABLE GENOME GNF-PF-77 CHEMBL602987 56839 38818 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Sirolimus SIROLIMUS 26144316,26882569 56841 38819 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE TANESPIMYCIN TANESPIMYCIN 23153200 56842 38820 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE XL-147 PILARALISIB 56843 38821 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE LEVOLEUCOVORIN LEVOLEUCOVORIN 25788273 56845 38822 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE NVP-BEZ235 DACTOLISIB 56846 38823 DNER 92737 NA Isoxazole-based bicyclic compound 14 56849 38824 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PICEATANNOL PICEATANNOL 56850 38825 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 135649908 56852 38826 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME inhibitor 328083483 PF-00562271 56853 38827 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 2',BETA-DIHYDROXYCHALCONE 2',BETA-DIHYDROXYCHALCONE 56854 38828 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE BAY 1436032 56855 38829 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 6'-IODONONIVAMIDE CHEMBL177809 56856 38830 C1S 716 ENZYME, PROTEASE, DRUGGABLE GENOME ANX005 56858 38831 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GDNF 15289335 56859 38832 DLL3 10683 NA AMG 119 56862 38833 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE AST-487 AST-487 56863 38834 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE HYPERTHERMIC INTRAPERITONEAL CHEMOTHERAPY 20942962 56864 38835 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ERLOTINIB ERLOTINIB 26619011,19455431,22452896,23102728,20068085,16707764,17653080,15710947,20479403,25668228,16912157,24893891,15728811,20573926,16258541,19692680,15118125,18227510,24658966,18199554,19922469,20033049,26515464,25923549,21783417,19692684,22753918,16187797,22452895,23945392,15329413,24636847,23816963,24729716,23816960,22285168,19096302,16204070,24894453,16043828,22215752,21194487,24065731,15118073,20022809,23948351,16115929,18458038,17332364,24623981,19147750,25157968,16011858,21430269,2302402,15737014,26720284,21670455,21233402,23242437,17177598,25923550,22588155,21531810,18303429,19671738 56865 38836 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650525 LISURIDE 56866 38837 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR Bevacizumab + Trastuzumab 56868 38838 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE GEFITINIB GEFITINIB 17463250 56869 38839 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE HEXACHLOROPHENE HEXACHLOROPHENE 56870 38840 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME OXATOMIDE OXATOMIDE 56874 38841 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER astemizole ASTEMIZOLE 56876 38842 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR EMODIN EMODIN 56879 38843 SMN1 6606 DRUGGABLE GENOME LOVASTATIN LOVASTATIN 56880 38844 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME YYDJCLCSBYCSCO-UHFFFAOYSA-N 56881 38845 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 3,3',4,4',5,5'-HEXAMETHOXYCHALCONE CHEMBL17442 20813535 56882 38846 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR THR-18 56883 38847 DDC 1644 ENZYME, DRUGGABLE GENOME RAPAMYCIN SIROLIMUS 16126007 56884 38848 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME TCMDC-125758 CHEMBL546797 56887 38849 TOP2B 7155 DRUGGABLE GENOME, ENZYME PYRAZOLOACRIDINE PYRAZOLOACRIDINE 56889 38850 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-P5 56890 38851 POLK 51426 DNA REPAIR, ENZYME PARAPLATIN CARBOPLATIN 56891 38852 ATXN2 6311 NA TCMDC-123916 CHEMBL493863 56892 38853 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103625 INDISULAM 56893 38854 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE clozapine CLOZAPINE 24725652 56894 38855 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE LEVALLORPHAN LEVALLORPHAN 56896 38856 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME allopurinol ALLOPURINOL 29341237,26810134,30924126 56898 38857 LTC4S 4056 ENZYME, DRUGGABLE GENOME US20160326143, 28 56899 38858 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME PAZOPANIB PAZOPANIB 56901 38859 MAPT 4137 DRUGGABLE GENOME FISETIN FISETIN 56904 38860 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME activator BEXAROTENE BEXAROTENE 56905 38861 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME FLUNARIZINE FLUNARIZINE 56907 38862 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PROPYLPARABEN PROPYLPARABEN 56910 38863 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE oxaliplatin OXALIPLATIN 24924344 56914 38864 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 381744936 56915 38865 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING CEFIXIME CEFIXIME 56917 38866 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DOXORUBICIN DOXORUBICIN 15465924 56918 38867 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Bicyclic hexapeptide derivative 1 56920 38868 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BRL-52537 CHEMBL71294 56923 38869 BCHE 590 DRUGGABLE GENOME, ENZYME inhibitor 178103211 PHYSOSTIGMINE 56924 38870 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor REFAMETINIB REFAMETINIB 56927 38871 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor AFATINIB AFATINIB 56928 38872 POLK 51426 DNA REPAIR, ENZYME CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 56929 38873 MAPT 4137 DRUGGABLE GENOME PROPYLENE GLYCOL MONOSTEARATE PROPYLENE GLYCOL MONOSTEARATE 56931 38874 TUBA1C 84790 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 56934 38875 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALPHA-2B 56935 38876 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1395 METHYLTESTOSTERONE 56937 38877 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SLAZINIC ACID SLAZINIC ACID 56938 38878 PKN1 5585 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 178102304 TOFACITINIB 56939 38879 F5 2153 DRUGGABLE GENOME ethinyl estradiol / norelgestromin 56941 38880 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Sirolimus SIROLIMUS 24813888 56942 38881 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-21 56943 38882 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Scriptaid SCRIPTAID 56944 38883 UGCG 7357 ENZYME, DRUGGABLE GENOME GZ402671 VENGLUSTAT 56946 38884 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32b 56948 38885 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NALTREXONE NALTREXONE 56949 38886 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR PROTEIN KINASE C INHIBITOR 9677306 56950 38887 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME olanzapine OLANZAPINE 19622037 56952 38888 CSMD1 64478 NA hydrochlorothiazide HYDROCHLOROTHIAZIDE 56953 38889 CGA 1081 DRUGGABLE GENOME, HORMONE ACTIVITY TESTOSTERONE TESTOSTERONE 1157041 56955 38890 NDUFA9 4704 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 56956 38891 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CO-1686 ROCILETINIB 56957 38892 AKR7A2 8574 DRUGGABLE GENOME, ENZYME doxorubicin DOXORUBICIN 20837989 56958 38893 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CC-486 56959 38894 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE DESIPRAMINE DESIPRAMINE 56960 38895 POLK 51426 DNA REPAIR, ENZYME AMPICILLIN SODIUM AMPICILLIN SODIUM 56964 38896 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FOSPIRATE FOSPIRATE 56965 38897 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AP32788 56966 38898 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZOQUINONE BENZOQUINONE 56967 38899 PARD3B 117583 NA oxaliplatin OXALIPLATIN 22310351 56968 38900 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 178101107 56969 38901 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Tranilast TRANILAST 56970 38902 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417484 CHEMBL1308677 56972 38903 SLC15A1 6564 DRUGGABLE GENOME, TRANSPORTER ACYCLOVIR ACYCLOVIR 12821497 56973 38904 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ANANDAMIDE ANANDAMIDE 56974 38905 ZFP36L2 678 TRANSCRIPTION FACTOR BUTYRATE 10367403 56975 38906 KMO 8564 DRUGGABLE GENOME, ENZYME Aryl pyrimidine derivative 2 56976 38907 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PYRACLOSTROBIN PYRACLOSTROBIN 56978 38908 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774824-Compound-Figure8Example22 56982 38909 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME 6-THIOGUANINE THIOGUANINE 1638685 56984 38910 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MGAH22 MARGETUXIMAB 56988 38911 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 187051762 GLYCOPYRROLATE 56990 38912 APC 324 CLINICALLY ACTIONABLE Vinorelbine VINORELBINE 22399804 56991 38913 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CHRYSENE-1,4-DIONE CHEMBL421215 56992 38914 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051807 SCRIPTAID 56993 38915 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE DEXANABINOL DEXANABINOL 56996 38916 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SAR125844 SAR-125844 25504634 57000 38917 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE ATL1102 57002 38918 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 135650129 EVATANEPAG 57003 38919 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545361 ROGARATINIB 57004 38920 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL206834 BAFETINIB 57005 38921 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SB-228357 CHEMBL14276 57009 38922 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ARBUTAMINE ARBUTAMINE 57010 38923 CDK12 51755 KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR, SERINE THREONINE KINASE Pembrolizumab PEMBROLIZUMAB 57013 38924 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ruxolitinib RUXOLITINIB 57014 38925 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200670 SARALASIN ACETATE 57015 38926 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PROPANIL PROPANIL 57018 38927 HTT 3064 DRUGGABLE GENOME TCMDC-125544 CHEMBL533602 57021 38928 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME BAY-613606 CHEMBL541400 57022 38929 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE 57023 38930 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME PAZOPANIB PAZOPANIB 57024 38931 ULK1 8408 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565893 57025 38932 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE NINTEDANIB NINTEDANIB 57026 38933 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL3545383 RG-7167 57027 38934 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE inhibitor 178103388 DIGITOXIN 57029 38935 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme27LeucettineL41 57030 38936 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CYC116 57031 38937 BCL2A1 597 DRUGGABLE GENOME US8937193-compound-6b 57032 38938 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE XL765 57033 38939 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PACLITAXEL PACLITAXEL 57034 38940 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GAMMA-CYHALOTHRIN GAMMA-CYHALOTHRIN 57035 38941 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE GW843682X GW843682X 57037 38942 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE NRM8499 57038 38943 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SP-600125 SP-600125 57040 38944 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200578 THEOPHYLLINE SODIUM GLYCINATE 57042 38945 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE sorafenib SORAFENIB 28362716 57043 38946 CDKN3 1033 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, TUMOR SUPPRESSOR, ENZYME, KINASE inhibitor CHEMBL445813 AT-7519 57045 38947 CBX1 10951 NA CLOROTEPINE CLOROTEPINE 57046 38948 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 1-BENZYLMALEIMIDE CHEMBL388979 57049 38949 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649964 57050 38950 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SNC-80 SNC-80 57051 38951 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE NERATINIB NERATINIB 57052 38952 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 315661180 ZOTIRACICLIB 57053 38953 ATAD5 79915 NA DNDI1417085 CHEMBL1522984 57054 38954 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4218 CHEMBL585269 57056 38955 TGFBR2 7048 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME irinotecan IRINOTECAN 27160286 57058 38956 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GYKI-52466 GYKI-52466 57059 38957 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AROMATICIN AROMATICIN 57060 38958 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (+)-EPITAXIFOLIN (+)-EPITAXIFOLIN 57064 38959 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE METHOTREXATE METHOTREXATE 8509220 57065 38960 CSPG4 1464 CELL SURFACE, DRUGGABLE GENOME TPA ALTEPLASE 18000864 57068 38961 TUBA1B 10376 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 57069 38962 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor 178102147 SULPIRIDE 57070 38963 MAOB 4129 DRUGGABLE GENOME, ENZYME 8-(3-CHLOROBENZYLOXY)CAFFEINE CHEMBL602260 20093036 57072 38964 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SGI-1776 SGI-1776 57073 38965 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR STANOLONE STANOLONE 57075 38966 SMN2 6607 DRUGGABLE GENOME PHENAMIL METHANESULFONATE PHENAMIL METHANESULFONATE 57076 38967 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL antagonist CHEMBL220492 TOPIRAMATE 57077 38968 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Abemaciclib ABEMACICLIB 57080 38969 NDUFAF1 51103 NA inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 57081 38970 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLOTIAZEPAM CLOTIAZEPAM 57082 38971 CAMK1 8536 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME LAUROGUADINE LAUROGUADINE 57083 38972 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CAMPTOTHECIN CAMPTOTHECIN 57084 38973 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-2755 CHEMBL600738 57086 38974 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-130 CHEMBL578890 57088 38975 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE TPA ALTEPLASE 12033920 57089 38976 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME DIMETHYLADENINE DIMETHYLADENINE 57090 38977 MAPT 4137 DRUGGABLE GENOME DNDI1417607 CHEMBL1588679 57093 38978 GPR68 8111 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 374883820 57094 38979 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL482968 ENMD-2076 57095 38980 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ANTIBIOTIC ANTIBIOTIC 10030847 57096 38981 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL2109544 CDP-860 57097 38982 MAPT 4137 DRUGGABLE GENOME ISOGINKGETIN ISOGINKGETIN 57098 38983 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178101785 57100 38984 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201167 CARVEDILOL PHOSPHATE 57101 38985 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME CALCIMYCIN CALCIMYCIN 57104 38986 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CYCLOSPORIN A 7907109,11555673 57106 38987 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Irbesartan IRBESARTAN 57107 38988 F5 2153 DRUGGABLE GENOME RECOMBINANT HUMAN THROMBIN 57108 38989 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650094 CICAPROST 57109 38990 PSMB9 5698 DRUGGABLE GENOME, PROTEASE, ENZYME BORTEZOMIB BORTEZOMIB 24524217 57110 38991 SLAMF7 57823 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ELOTUZUMAB ELOTUZUMAB 57111 38992 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME antagonist 135652741 57112 38993 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ZIDOVUDINE ZIDOVUDINE 22931300 57113 38994 MYB 4602 CLINICALLY ACTIONABLE TAXOL PACLITAXEL 15001837 57114 38995 CHRNA5 1138 DRUGGABLE GENOME, ION CHANNEL antagonist 178100837 57115 38996 FBXW7 55294 DNA REPAIR, CLINICALLY ACTIONABLE SIROLIMUS SIROLIMUS 18787170 57116 38997 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 249565683 BERZOSERTIB 57117 38998 MAPT 4137 DRUGGABLE GENOME (+)-THALIPORPHINE CHEMBL1397308 57118 38999 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME NGR-HTNF 57120 39000 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PIPERACETAZINE PIPERACETAZINE 57123 39001 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Erlotinib ERLOTINIB 27659046,15696205,18626007,16043828,27480147 57124 39002 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ENTRECTINIB ENTRECTINIB 57125 39003 GAA 2548 DRUGGABLE GENOME, ENZYME ACRIDONE ACRIDONE 57126 39004 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLORAZEPATE CLORAZEPIC ACID 57127 39005 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652433 VAPREOTIDE 57129 39006 PRKAG1 5571 ENZYME, KINASE SAPONARIN SAPONARIN 26471090 57130 39007 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE inhibitor 178103156 57132 39008 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-5114 CHEMBL601952 57135 39009 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TAE-684 TAE-684 57136 39010 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PALBOCICLIB PALBOCICLIB 57137 39011 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE COUMATE 57138 39012 FGD4 121512 NA paclitaxel PACLITAXEL 22843789 57139 39013 NDUFB5 4711 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 57140 39014 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-H2 57141 39015 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE LEVOBUNOLOL LEVOBUNOLOL 57142 39016 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545298 AZD-6918 57143 39017 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY HMBA 10450830 57144 39018 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135649664 57148 39019 ANGPTL3 27329 DRUGGABLE GENOME, FIBRINOGEN, CELL SURFACE, GROWTH FACTOR Evinacumab EVINACUMAB 57149 39020 BAZ2B 29994 NA SJ000113257 CHEMBL528694 57150 39021 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 57152 39022 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Fluorinated donepezil derivative 2 57153 39023 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HERNANDEZINE HERNANDEZINE 57154 39024 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ALPHA-CYPERMETHRIN ALPHA-CYPERMETHRIN 57156 39025 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CABOZANTINIB CABOZANTINIB 57157 39026 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME pazopanib PAZOPANIB 26546620 57158 39027 IL20 50604 DRUGGABLE GENOME NN-8226 57159 39028 RIPK2 8767 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 381118799 57161 39029 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL3544949 CTCE-9908 57162 39030 H2AW 92815 NA ALBUMIN ALBUMIN HUMAN 1989977 57163 39031 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PIRINIXIC ACID PIRINIXIC ACID 23171045,17228882,25497132 57165 39032 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SB-206553 CHEMBL297784 57166 39033 IL18 3606 DRUGGABLE GENOME TACROLIMUS TACROLIMUS 11061569 57167 39034 HPN 3249 DRUGGABLE GENOME, PROTEASE, CELL SURFACE BENTIROMIDE BENTIROMIDE 57170 39035 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE RO-410960 CHEMBL1256291 57171 39036 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ZIPRASIDONE ZIPRASIDONE 57173 39037 ALOX15 246 ENZYME, DRUGGABLE GENOME DIENESTROL DIENESTROL 57175 39038 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE activator 223366001 57178 39039 CACNB3 784 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ION CHANNEL celecoxib CELECOXIB 22336956 57179 39040 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-4325 CHEMBL598263 57181 39041 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3545058 DEXTROTHYROXINE SODIUM 57182 39042 CA2 760 DRUGGABLE GENOME, ENZYME CHLOROTHIAZIDE CHLOROTHIAZIDE 57185 39043 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE LOPERAMIDE LOPERAMIDE 57188 39044 NGFR 4804 CELL SURFACE, DRUGGABLE GENOME SPI-205 57189 39045 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 310264693 ACALABRUTINIB 57190 39046 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000154295 CHEMBL578502 57191 39047 ATAD5 79915 NA JNJ-1661010 CHEMBL460273 57193 39048 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW434756X GW434756X 57194 39049 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MMV667491 CHEMBL1437888 57195 39050 P2RX4 5025 ION CHANNEL, DRUGGABLE GENOME antagonist 135650843 57196 39051 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE GW441756X GW441756X 57197 39052 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME DS-3032 MILADEMETAN 57198 39053 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME CHEMBL1699 MEMANTINE HYDROCHLORIDE 57199 39054 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME CYCLOSPORIN A 17031644 57201 39055 DDB1 1642 DNA REPAIR inhibitor CHEMBL848 LENALIDOMIDE 57202 39056 TPM3 7170 KINASE, CLINICALLY ACTIONABLE SIMVASTATIN SIMVASTATIN 10720627 57203 39057 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ASP8273 NAQUOTINIB 57204 39058 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CID 5330286 57205 39059 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DIBENZ[A,H]ANTHRACENE DIBENZ[A,H]ANTHRACENE 57206 39060 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor 178101942 57208 39061 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-1399 CHEMBL578504 57211 39062 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 223365970 57212 39063 PTGS2 5743 DRUGGABLE GENOME, ENZYME oxaliplatin OXALIPLATIN 19219602 57215 39064 GABBR2 9568 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL BACLOFEN BACLOFEN 57217 39065 VKORC1 79001 DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 57218 39066 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 6 57219 39067 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TRITIOZINE TRITIOZINE 57221 39068 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL2104984 SODELGLITAZAR 57223 39069 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Olaparib OLAPARIB 57226 39070 TLR7 51284 DRUGGABLE GENOME antagonist CHEMBL1690 HYDROXYCHLOROQUINE SULFATE 57228 39071 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CH5132799 PA-799 21558396 57229 39072 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SR-2640 SR-2640 57230 39073 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 385612180 57232 39074 GMNN 51053 DRUGGABLE GENOME OXOPURPUREINE OXOPURPUREINE 57233 39075 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 57234 39076 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME HGS1029 57235 39077 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 404859075 57236 39078 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SB-203580 SB-203580 25692815 57238 39079 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR CURCUMIN CURCUMIN 16306131 57239 39080 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME BINIMETINIB BINIMETINIB 26544513 57240 39081 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (S)-ROSCOVITINE (S)-ROSCOVITINE 57241 39082 DHFR 1719 DRUGGABLE GENOME, ENZYME MTX METHOTREXATE 14679136,6831441,7057421,1533575 57242 39083 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-2356 CHEMBL601547 57243 39084 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BAY1082439 57245 39085 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 57246 39086 CTSF 8722 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103149 57247 39087 RGS4 5999 DRUGGABLE GENOME ziprasidone ZIPRASIDONE 57248 39088 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FOLINIC ACID 10470170 57249 39089 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 252166755 57250 39090 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL661 ALPRAZOLAM 57251 39091 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXABOLONE CIPIONATE OXABOLONE CIPIONATE 57252 39092 PPT1 5538 ENZYME, DRUGGABLE GENOME Plitidepsin PLITIDEPSIN 25867045 57253 39093 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DIDANOSINE DIDANOSINE 22931300 57255 39094 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MANGOSTIN MANGOSTIN 57256 39095 PTPRD 5789 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TEPROTUMUMAB TEPROTUMUMAB 23800680 57259 39096 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Pamidronate PAMIDRONIC ACID 57260 39097 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE ZM-447439 CHEMBL202721 57262 39098 COMT 1312 DRUGGABLE GENOME, ENZYME trihexyphenidyl TRIHEXYPHENIDYL 57263 39099 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR KP201 BENZHYDROCODONE HYDROCHLORIDE 57264 39100 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CEFONICID SODIUM CEFONICID SODIUM 57265 39101 MPHOSPH8 54737 NA DIAMIDE DIAMIDE 57266 39102 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER MIFEPRISTONE MIFEPRISTONE 57267 39103 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR SIGNAL TRANSDUCTION INHIBITORS 16525725 57268 39104 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor EMD1214063 57269 39105 GCLC 2729 DRUGGABLE GENOME, ENZYME CBDCA CARBOPLATIN 11911273 57270 39106 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-45 57271 39107 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 354702282 57272 39108 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER EDP-322 57274 39109 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 381745024 57275 39110 TARDBP 23435 TUMOR SUPPRESSOR 1,4-DIMETHOXYANTHRAQUINONE 1,4-DIMETHOXYANTHRAQUINONE 57276 39111 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BAICALEIN BAICALEIN 57277 39112 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201486 QUINIDINE POLYGALACTURONATE 57278 39113 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200875 FLAVOXATE HYDROCHLORIDE 57279 39114 TUBB 203068 DRUGGABLE GENOME PHOMOPSIN A PHOMOPSIN A 19072542 57280 39115 POLI 11201 DNA REPAIR IDARUBICIN IDARUBICIN 57281 39116 GMNN 51053 DRUGGABLE GENOME NSC-601359 CHEMBL1306524 57282 39117 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL3545279 EFATUTAZONE HYDROCHLORIDE 57284 39118 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIFLORASONE DIACETATE DIFLORASONE DIACETATE 57286 39119 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103518 LY-2811376 57287 39120 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME inhibitor CHEMBL1743063 RILOTUMUMAB 57288 39121 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHIDATHION METHIDATHION 57289 39122 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TANNIC ACID TANNIC ACID 57290 39123 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TOLTERODINE TOLTERODINE 57291 39124 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200790 METHYPRYLON 57294 39125 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE TNF-ALPHA 8995390,16754199,14764603 57295 39126 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR STANOLONE STANOLONE 57296 39127 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TKI258 DOVITINIB 57298 39128 FES 2242 ENZYME, DRUGGABLE GENOME, KINASE, TYROSINE KINASE inhibitor 187051779 LORLATINIB 57302 39129 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ALPRAZOLAM ALPRAZOLAM 57303 39130 GMNN 51053 DRUGGABLE GENOME TCMDC-124063 CHEMBL534535 57305 39131 HPSE 10855 ENZYME, DRUGGABLE GENOME TCMDC-125528 CHEMBL375673 23415087 57308 39132 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2110732 DACOMITINIB 57310 39133 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME ABT-165 57311 39134 ATAD5 79915 NA TRICHOSTATIN TRICHOSTATIN 57312 39135 NDUFV1 4723 ENZYME inhibitor CHEMBL3545135 NV-128 57313 39136 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL antagonist 135652741 57314 39137 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE ADENOVIRUS VECTOR 17536066 57315 39138 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR VU0365137 CHEMBL1084941 57316 39139 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 893238 CHEMBL473735 57317 39140 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist 178100902 57318 39141 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR Tricyclic benzimidazole derivative 1 57320 39142 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ANISOMYCIN ANISOMYCIN 57321 39143 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SP-600125 SP-600125 57323 39144 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME CER-001 57325 39145 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Bis-aminopyrimidine derivative 3 57326 39146 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE DNDI1417467 CHEMBL1997335 57327 39147 PSMA6 5687 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 57329 39148 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor GANETESPIB GANETESPIB 57330 39149 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200703 CHLORDIAZEPOXIDE HYDROCHLORIDE 57336 39150 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SPHAEROPSIDIN A SPHAEROPSIDIN A 57337 39151 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME MRS-1220 CHEMBL88147 57340 39152 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178101750 SEMAXANIB 57342 39153 CCHCR1 54535 NA nevirapine NEVIRAPINE 21810746 57344 39154 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE QUINOLINIC ACID QUINOLINIC ACID 57345 39155 BCHE 590 DRUGGABLE GENOME, ENZYME Indoline derivative 1 57346 39156 ATXN2 6311 NA GNF-PF-2243 CHEMBL600908 57348 39157 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PRIDINOL PRIDINOL 57349 39158 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-28 57350 39159 SENP2 59343 ENZYME, PROTEASE N-ETHYLMALEIMIDE N-ETHYLMALEIMIDE 22801642 57351 39160 SLC23A2 9962 TRANSPORTER 178101253 57353 39161 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1201470 HYDROCODONE POLISTIREX 57354 39162 MAPT 4137 DRUGGABLE GENOME BISINDOLYLMALEIMIDE IX BISINDOLYLMALEIMIDE IX 57355 39163 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE IL-18 16313368 57356 39164 POLI 11201 DNA REPAIR QUINACRINE QUINACRINE 57357 39165 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 404859025 57358 39166 KDM4A 9682 DRUGGABLE GENOME, ENZYME GR-127935 GR-127935 57359 39167 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE CARBIMAZOLE CARBIMAZOLE 57360 39168 POLK 51426 DNA REPAIR, ENZYME NSC-155693 CHEMBL68096 57362 39169 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 tenoxicam TENOXICAM 18992346,15229460 57363 39170 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135651449 57364 39171 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEQUALINIUM DEQUALINIUM 57366 39172 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GYKI-52895 CHEMBL1256984 57368 39173 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CEFADROXIL CEFADROXIL 22166395 57369 39174 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME LB-30870 57370 39175 EPHX2 2053 DRUGGABLE GENOME, ENZYME inhibitor 178100355 ZAFIRLUKAST 57378 39176 BMP7 655 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR thioguanine THIOGUANINE 26590194 57379 39177 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ALPHA-NAPHTHOFLAVONE ALPHA-NAPHTHOFLAVONE 57381 39178 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PH-011685 CHEMBL126804 57382 39179 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BORIC ACID BORIC ACID 57383 39180 SCNN1A 6337 DRUGGABLE GENOME, ION CHANNEL amiloride AMILORIDE 23788015 57384 39181 TUBA1B 10376 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 57385 39182 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME 681640 CHEMBL379975 57386 39183 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CAFFEINE CAFFEINE 22931300 57387 39184 KCNC2 3747 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL284348 DALFAMPRIDINE 57388 39185 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE OBOVATAL OBOVATAL 17428670 57390 39186 BAZ2B 29994 NA PROTOPORPHYRIN DISODIUM PROTOPORPHYRIN DISODIUM 57391 39187 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME BDBM50379214 57392 39188 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Flavonoid derivative 7 57393 39189 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE AMUVATINIB AMUVATINIB 57394 39190 ADH1C 126 ENZYME, DRUGGABLE GENOME cisplatin CISPLATIN 24533712 57395 39191 DOCK8 81704 NA carboplatin CARBOPLATIN 31616045 57398 39192 EPHX2 2053 DRUGGABLE GENOME, ENZYME AR9281 AR9281 57400 39193 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CARMOFUR CARMOFUR 57402 39194 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE NAV-2729 27265506 57403 39195 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NGI-1 27694802 57406 39196 PSMB3 5691 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL325041 BORTEZOMIB 57407 39197 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650448 57408 39198 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL52885 ENMD-981693 57409 39199 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL2107341 FISPEMIFENE 57412 39200 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE GNF-PF-4085 CHEMBL528181 57413 39201 BAZ2B 29994 NA TAMOXIFEN TAMOXIFEN 57414 39202 ALOX15 246 ENZYME, DRUGGABLE GENOME RELCOVAPTAN RELCOVAPTAN 57417 39203 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE DOVITINIB DOVITINIB 57418 39204 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 381118823 57419 39205 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR antagonist CHEMBL3544957 CORT 125134 57420 39206 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Pazopanib PAZOPANIB 23558953 57421 39207 PDE3A 5139 ENZYME, DRUGGABLE GENOME CILOSTAZOL CILOSTAZOL 57424 39208 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE lapatinib LAPATINIB 18681783,14990633,16467544,16377102,14990632,18784101,16257339,18003960,23022519,11255078,19339720,18316547,12648464,22594511 57425 39209 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650491 57426 39210 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Fluorouracil FLUOROURACIL 26432108 57427 39211 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR adalimumab ADALIMUMAB 24253594 57428 39212 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000112730 CHEMBL591178 57429 39213 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamate derivative 17 57430 39214 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE VATALANIB VATALANIB 57431 39215 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Clazosentan CLAZOSENTAN 57433 39216 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PHENFORMIN HYDROCHLORIDE PHENFORMIN HYDROCHLORIDE 57435 39217 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Azelastine AZELASTINE 57436 39218 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CHIR-99021 CHIR-99021 57440 39219 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR TG-C 57441 39220 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FENITROTHION FENITROTHION 57445 39221 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GW441756X GW441756X 57446 39222 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR KERACYANIN KERACYANIN 17360708 57448 39223 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 363894127 57449 39224 GMNN 51053 DRUGGABLE GENOME NICLOSAMIDE NICLOSAMIDE 57450 39225 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545177 AZD-0424 57452 39226 ATAD5 79915 NA SJ000018298 CHEMBL591412 57455 39227 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BENZQUINAMIDE BENZQUINAMIDE 57456 39228 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Quinazolinedione derivative 3 57457 39229 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NORBINALTORPHIMINE NORBINALTORPHIMINE 17702750 57459 39230 TSPO 706 DRUGGABLE GENOME ZALEPLON ZALEPLON 57460 39231 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME capecitabine CAPECITABINE 20125120,25955730 57461 39232 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR MOCETINOSTAT MOCETINOSTAT 23829483,26287310 57468 39233 CDA 978 ENZYME, DRUGGABLE GENOME TETRAHYDROURIDINE TETRAHYDROURIDINE 2932216 57470 39234 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE ceftriaxone CEFTRIAXONE 57471 39235 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor CHEMBL1201619 APROTININ 57475 39236 GUCY1A2 2977 ENZYME, DRUGGABLE GENOME activator CHEMBL136478 SODIUM NITROPRUSSIDE 57476 39237 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ANDROSTENEDIONE ANDROSTENEDIONE 57478 39238 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TCMDC-124336 CHEMBL527271 57479 39239 HIF1AN 55662 NA BAICALEIN BAICALEIN 21665470 57480 39240 BAZ2B 29994 NA TANSHINONE I TANSHINONE I 57482 39241 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2165191 AZD-6482 57485 39242 CBX1 10951 NA GW7074 CHEMBL72365 57488 39243 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-19 57492 39244 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-2243 CHEMBL600908 57493 39245 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME TAE-684 TAE-684 57495 39246 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor RUCAPARIB RUCAPARIB 57496 39247 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545052 FIMEPINOSTAT 57499 39248 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME VEMURAFENIB VEMURAFENIB 24265155,25037139,24987354,31513482,24345920,22798288,23533272,24508103,24576830,20818844,26989536,26687137,27480103,22356324,27460442,25265494,23715574,25515853,18287029,26287849,27048246,25524477,21639808,22281684,22180495,28002790,29320312,27729313,24112705,24997557 57501 39249 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME DOXORUBICIN DOXORUBICIN 7532928 57503 39250 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 nicardipine NICARDIPINE 9187528 57504 39251 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CIMETIDINE CIMETIDINE 11556524 57505 39252 BMPR1B 658 DRUGGABLE GENOME, CELL SURFACE, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 249565800 57507 39253 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Debio1347 DEBIO-1347 57508 39254 PCSK1 5122 DRUGGABLE GENOME, PROTEASE, ENZYME INSULIN INSULIN 7883951,7925129 57510 39255 GUCY2C 2984 DRUGGABLE GENOME, KINASE LINACLOTIDE LINACLOTIDE 57512 39256 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AMLODIPINE BESYLATE AMLODIPINE BESYLATE 57513 39257 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR TCMDC-125185 CHEMBL580819 57514 39258 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Cetuxmab 23792568 57515 39259 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Tazemetostat TAZEMETOSTAT 26676756 57516 39260 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL107 COLCHICINE 57517 39261 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME 5-AZA-2'-DEOXYCYTIDINE 18174247 57518 39262 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 178103211 PHYSOSTIGMINE 57521 39263 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-42 57522 39264 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SALICYLANILIDE SALICYLANILIDE 57523 39265 PDE4B 5142 DRUGGABLE GENOME, ENZYME CC-1088 CDC-801 57524 39266 IMPDH1 3614 ENZYME, DRUGGABLE GENOME MYCOPHENOLIC ACID 57525 39267 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Pyrrolo[1,2-c]pyrazole derivative 1 57527 39268 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME GNF-PF-3832 CHEMBL261693 57529 39269 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 (R)-NITRENDIPINE (R)-NITRENDIPINE 57530 39270 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 404859149 57534 39271 HMOX2 3163 ENZYME BETAMETHASONE BETAMETHASONE 11698254 57535 39272 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME AZD-8055 AZD-8055 23375793 57536 39273 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME CHEMBL1714 KETAMINE HYDROCHLORIDE 57537 39274 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 249565585 UPROSERTIB 57538 39275 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME IGN101 57540 39276 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2-AMINOETHOXYDIPHENYL BORATE CHEMBL169233 57541 39277 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200803 SOLIFENACIN SUCCINATE 57542 39278 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor E-3810 RABEPRAZOLE SODIUM 57544 39279 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LARGAZOLE LARGAZOLE 21420302,21936551,25203782,20491440 57546 39280 HBB 3043 DRUGGABLE GENOME, ENZYME THIOINOSINE THIOINOSINE 57547 39281 PSMC5 5705 TRANSCRIPTION FACTOR BINDING, PROTEASE inhibitor CHEMBL2103884 OPROZOMIB 57548 39282 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2062267 HYDROCODONE BITARTRATE 57549 39283 TUBA4A 7277 DRUGGABLE GENOME CHEMBL492399 VERUBULIN 57550 39284 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL514800 APREMILAST 57553 39285 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AMSACRINE HYDROCHLORIDE AMSACRINE HYDROCHLORIDE 57554 39286 IMPDH2 3615 DRUGGABLE GENOME, ENZYME mycophenolate mofetil 21996196,19770842,20679962,18444945,19617864,22960765 57555 39287 GAA 2548 DRUGGABLE GENOME, ENZYME SJ000124275 CHEMBL602150 57556 39288 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE BETA-LAPACHONE LAPACHONE 10075082 57557 39289 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE doxorubicin DOXORUBICIN 9333325,10954045 57558 39290 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-23 57560 39291 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CISPLATIN CISPLATIN 21458988 57564 39292 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ALTANSERIN ALTANSERIN 57566 39293 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TESTOSTERONE TESTOSTERONE 9681518 57568 39294 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 404859050 57569 39295 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Quinazolinone derivative 2 57571 39296 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL738 THIOPENTAL SODIUM 57572 39297 PTGES 9536 DRUGGABLE GENOME, ENZYME Benzimidazole derivative 12 57574 39298 TXNRD1 7296 DRUGGABLE GENOME Benzisoselenazolone difluorocytidine derivative 1 57575 39299 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-123532 CHEMBL547833 57576 39300 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CATUMAXOMAB CATUMAXOMAB 57579 39301 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1-HYDROXY-4-ETHOXYBENZENE 1-HYDROXY-4-ETHOXYBENZENE 57580 39302 SERPINA1 5265 DRUGGABLE GENOME, PROTEASE INHIBITOR Igmesine IGMESINE 57581 39303 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROPRANOLOL PROPRANOLOL 57583 39304 METAP2 10988 ENZYME, DRUGGABLE GENOME, KINASE, PROTEASE inhibitor CHEMBL2103847 TOSEDOSTAT 57584 39305 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PLUMBAGIN PLUMBAGIN 57585 39306 AKR1B1 231 DRUGGABLE GENOME, ENZYME SSR-125047 57586 39307 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME GO-6976 GO-6976 57589 39308 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE carboplatin CARBOPLATIN 26179145 57592 39309 ALOX15 246 ENZYME, DRUGGABLE GENOME JUGLONE JUGLONE 57596 39310 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor SUNITINIB SUNITINIB 57597 39311 SFTPA1 653509 DRUGGABLE GENOME OPC-14117 57601 39312 CES1 1066 DRUGGABLE GENOME, ENZYME PACTIMIBE PACTIMIBE 57606 39313 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE KRC-00509 26801760 57611 39314 GMNN 51053 DRUGGABLE GENOME TCMDC-125567 CHEMBL530049 57612 39315 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545141 RP-6530 57613 39316 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE CNTO-95 INTETUMUMAB 57614 39317 FZD1 8321 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, KINASE TCMDC-124051 CHEMBL464249 23453073 57615 39318 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE EMODIN EMODIN 14694444 57617 39319 APOE 348 DRUGGABLE GENOME atorvastatin ATORVASTATIN 16103896,19667110,20031582,17289397 57619 39320 XPNPEP1 7511 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL2103847 TOSEDOSTAT 57621 39321 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR LY-2090314 LY-2090314 57622 39322 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 24524217 57625 39323 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 14 57626 39324 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ENCLOMIPHENE CITRATE ENCLOMIPHENE CITRATE 57627 39325 KDM4A 9682 DRUGGABLE GENOME, ENZYME MMV085203 CHEMBL586031 57628 39326 CXCL2 2920 DRUGGABLE GENOME BFGF 15194436 57629 39327 MPHOSPH8 54737 NA 5-(N-METHYL-N-ISOBUTYL)AMILORIDE 5-(N-METHYL-N-ISOBUTYL)AMILORIDE 57630 39328 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor VORINOSTAT VORINOSTAT 57631 39329 CA12 771 DRUGGABLE GENOME inhibitor CHEMBL20 ACETAZOLAMIDE 57632 39330 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CAMPTOTHECIN CAMPTOTHECIN 57633 39331 ALOX15 246 ENZYME, DRUGGABLE GENOME EMBELIN EMBELIN 57634 39332 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER METHYL ROBUSTONE METHYL ROBUSTONE 57635 39333 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME SIROLIMUS SIROLIMUS 22955920 57636 39334 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-105 57637 39335 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LAUROGUADINE LAUROGUADINE 57639 39336 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE D-3263 D-3263 19680529 57640 39337 PTPN6 5777 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE 4-HYDRAZINYLBENZENESULFONIC ACID CHEMBL510966 19007293 57642 39338 XDH 7498 DRUGGABLE GENOME, ENZYME POTASSIUM OXONATE 16182482 57643 39339 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135651324 57644 39340 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE topoisomerase I inhibitors 18652519 57645 39341 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650280 57646 39342 IDE 3416 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, ENZYME, PROTEASE inhibitor 252166798 57647 39343 ALDH1A1 216 DRUGGABLE GENOME, ENZYME FENRETINIDE FENRETINIDE 57649 39344 SDHB 6390 ENZYME, CLINICALLY ACTIONABLE GENTAMYCIN CHEMBL329592 11477914 57654 39345 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1200382 BEPRIDIL HYDROCHLORIDE 57656 39346 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649792 57657 39347 TUBA1B 10376 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 57658 39348 ADK 132 DRUGGABLE GENOME, ENZYME, KINASE BUSULFAN BUSULFAN 6317371 57659 39349 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 57660 39350 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102571 57661 39351 BAZ2B 29994 NA DNDI1417221 CHEMBL1459280 57662 39352 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Pyrrolo[2,3-d]pyrimidine derivative 1 57663 39353 BCHE 590 DRUGGABLE GENOME, ENZYME inhibitor 178103215 RIVASTIGMINE 57664 39354 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ORTHO-PHTHALALDEHYDE ORTHO-PHTHALALDEHYDE 57665 39355 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE DIFFERENTIATING AGENTS 10532805 57667 39356 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME METHOXY POLYETHYLENE GLYCOL-EPOETIN BETA 57669 39357 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SENNOSIDE B SENNOSIDE B 57670 39358 GLS 2744 ENZYME CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 57671 39359 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1611 PHENYTOIN SODIUM 57673 39360 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME IDARUBICIN IDARUBICIN 57674 39361 DUSP3 1845 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE GNF-PF-67 CHEMBL578512 57675 39362 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ritodrine RITODRINE 57676 39363 RAB9A 9367 ENZYME, DRUGGABLE GENOME NILE RED NILE RED 57678 39364 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor GDC-0623 RG-7420 57679 39365 ATXN2 6311 NA GR-127935 GR-127935 57680 39366 TUBA1B 10376 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 57681 39367 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20120264760C80 57682 39368 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MAPROTILINE HYDROCHLORIDE MAPROTILINE HYDROCHLORIDE 57683 39369 PDE3A 5139 ENZYME, DRUGGABLE GENOME Tipelukast TIPELUKAST 57684 39370 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME RECOMBINANT PEGYLATED ACETYLCHOLINESTERASE 57687 39371 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 12 57689 39372 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FLUOXETINE HYDROCHLORIDE FLUOXETINE HYDROCHLORIDE 57690 39373 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ALRN-6924 57691 39374 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE antibody LY2875358 57692 39375 TUBA1B 10376 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 57694 39376 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL526 PROPOFOL 57695 39377 NCAM1 4684 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE FGLL 57696 39378 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE BIX-01294 CHEMBL569864 57697 39379 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME antibody FICLATUZUMAB FICLATUZUMAB 57698 39380 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-42 57699 39381 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Isoquinoline sulfonyl derivative 1 57700 39382 ANXA2 302 CELL SURFACE, DRUGGABLE GENOME WITHAFERIN A WITHAFERIN A 16408090 57702 39383 CRABP2 1382 NA BESTATIN METHYL ESTER BESTATIN METHYL ESTER 21515062 57704 39384 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE TOZASERTIB TOZASERTIB 57705 39385 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR FASUDIL FASUDIL 57706 39386 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME EQUILIN EQUILIN 57707 39387 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Palbociclib PALBOCICLIB 27488531,26369631 57711 39388 CXCL8 3576 DRUGGABLE GENOME D-ALPHA-TOCOPHEROL ACETATE 15150308 57712 39389 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME LGX818 ENCORAFENIB 57714 39390 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME LY3009104 57716 39391 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE GSI-136 GSI-136 57717 39392 MPI 4351 ENZYME, DRUGGABLE GENOME GNF-PF-2272 CHEMBL601757 57718 39393 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103489 57719 39394 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR citalopram CITALOPRAM 22965830,21338649,23733030,23619509,19236730,29748862,20016225 57720 39395 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SORAFENIB SORAFENIB 57721 39396 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE APRINDINE HYDROCHLORIDE APRINDINE HYDROCHLORIDE 57722 39397 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CLOBAZAM CLOBAZAM 57723 39398 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER NBI-98854 VALBENAZINE TOSYLATE 57724 39399 TSPYL1 7259 NA abiraterone ABIRATERONE 57725 39400 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545354 CAFUSERTIB 57726 39401 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE BGB-283 LIFIRAFENIB 26208524 57727 39402 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 252166684 57729 39403 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER Valbenazine Tosylate 57731 39404 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR INECALCITOL INECALCITOL 57732 39405 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RETRO-INVERSO PEPTIDE 11418697 57733 39406 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DOPAMINE DOPAMINE 57734 39407 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME DEL-22379 DEL-22379 26267534 57735 39408 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BECLOMETHASONE BECLOMETHASONE 22931300 57738 39409 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER ritonavir RITONAVIR 23996099 57741 39410 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ROTTLERIN ROTTLERIN 57742 39411 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME DNDI1417467 CHEMBL1997335 57744 39412 EYA2 2139 DNA REPAIR NSC-95397 CHEMBL429095 57745 39413 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PREDNISONE PREDNISONE 57747 39414 VEGFB 7423 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR antibody ZIV-AFLIBERCEPT AFLIBERCEPT 57748 39415 MPHOSPH8 54737 NA GR-127935 GR-127935 57749 39416 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4992 CHEMBL275177 57750 39417 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PMID29671355-Compound-44 57752 39418 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102325 PAZOPANIB 57753 39419 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Di-substituted piperidine derivative 2 57755 39420 MAPT 4137 DRUGGABLE GENOME NSC-50654 CHEMBL1372046 57756 39421 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 328083457 57757 39422 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME SURAMIN SURAMIN 57758 39423 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE regorafenib REGORAFENIB 57760 39424 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Nimotuzumab NIMOTUZUMAB 25185971 57761 39425 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DITHIAZANINE IODIDE DITHIAZANINE IODIDE 57763 39426 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ritonavir RITONAVIR 17324111,26174719,14600574,24997317,16355344,23996099,28718515,1655344,21288825,25151207,20504240,25622064,17148966,26857335 57764 39427 TRPC4 7223 ION CHANNEL, KINASE, DRUGGABLE GENOME, CELL SURFACE TRPC4 and TRPC5 inhibitor 57765 39428 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PD-0166285 PD-0166285 57767 39429 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHENYL SALICYLATE PHENYL SALICYLATE 57768 39430 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-AMINOANTHRACENE 2-AMINOANTHRACENE 57769 39431 KCNC2 3747 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker 135652463 57770 39432 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PACLITAXEL PACLITAXEL 25672916 57774 39433 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL118 CELECOXIB 57776 39434 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 esomeprazole ESOMEPRAZOLE 57778 39435 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545402 XL-820 57779 39436 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME blocker 135652058 57781 39437 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ZUCAPSAICIN ZUCAPSAICIN 57782 39438 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE ACARBOSE ACARBOSE 12065205 57783 39439 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL450940 PRINABEREL 57784 39440 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 223366211 CRENOLANIB 57785 39441 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CC-223 CC-223 57786 39442 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-21 57787 39443 RGS4 5999 DRUGGABLE GENOME GNF-PF-5510 CHEMBL578741 57788 39444 IL1R2 7850 DRUGGABLE GENOME GSK-1827771 57789 39445 TSPO 706 DRUGGABLE GENOME Imidazo[1,2-b]pyridazine acetamide derivative 4 57790 39446 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PKI-587 GEDATOLISIB 57791 39447 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME VALPROIC ACID 1972258 57792 39448 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-Figure3bIII 57793 39449 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME A-substituted phenylpropionic acid derivative 1 57796 39450 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CEFTRIAXONE CEFTRIAXONE 22166395 57797 39451 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR leucovorin LEUCOVORIN 21057378,23314736 57798 39452 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Five-membered heteroaromatic compound 2 57799 39453 IMPDH2 3615 DRUGGABLE GENOME, ENZYME inhibitor 178103448 RIBAVIRIN 57801 39454 SLC38A2 54407 TRANSPORTER 178101263 57803 39455 PRLR 5618 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, KINASE Prolanta 57804 39456 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor XL-765 VOXTALISIB 57805 39457 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PAMIDRONATE PAMIDRONIC ACID 57806 39458 ALOX15 246 ENZYME, DRUGGABLE GENOME CITRONELLYL ACETATE CITRONELLYL ACETATE 57808 39459 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1416917 CHEMBL1335833 57809 39460 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL TRIAZOLAM TRIAZOLAM 57811 39461 BAZ2B 29994 NA NAFRONYL OXALATE NAFRONYL OXALATE 57812 39462 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME ALSTERPAULLONE ALSTERPAULLONE 57813 39463 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE IMATINIB IMATINIB 16707477 57814 39464 CYP27A1 1593 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PHYTOSTEROLS 11398149 57816 39465 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL WIN-552122 WIN-552122 20346682 57817 39466 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 1207456-01-6 57818 39467 CCR7 1236 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR agonist 252166852 57819 39468 MAOB 4129 DRUGGABLE GENOME, ENZYME Indeloxazine INDELOXAZINE 57821 39469 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200813 ACEBUTOLOL HYDROCHLORIDE 57823 39470 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE Sulfatinib SURUFATINIB 57826 39471 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-1731 CHEMBL581251 57827 39472 HSPA4 3308 NA VERAPAMIL VERAPAMIL 12857801 57828 39473 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BGJ398 INFIGRATINIB 22837387,26015511,27535980,27870574 57829 39474 TARDBP 23435 TUMOR SUPPRESSOR PHENANTHROLINE PHENANTHROLINE 57834 39475 BCHE 590 DRUGGABLE GENOME, ENZYME mivacurium chloride 57837 39476 CTH 1491 ENZYME inhibitor 252827516 57838 39477 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1185 ZOLMITRIPTAN 57839 39478 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102665 57842 39479 CDH1 999 CLINICALLY ACTIONABLE, DRUGGABLE GENOME N/A 26182300,26380059 57844 39480 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME peginterferon alfa-2b 20812847 57845 39481 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1201156 NORTRIPTYLINE HYDROCHLORIDE 57846 39482 ACP5 54 ENZYME, DRUGGABLE GENOME TPA ALTEPLASE 1436243 57847 39483 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GARCINOLIC ACID GARCINOLIC ACID 57849 39484 OGA 10724 ENZYME, DRUGGABLE GENOME inhibitor 387065590 57850 39485 DIABLO 56616 NA UCN-01 UCN-01 12488556 57851 39486 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 olanzapine OLANZAPINE 23559402 57855 39487 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor X-82 X-82 57857 39488 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (S)-NIMODIPINE (S)-NIMODIPINE 57858 39489 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OXETHAZAINE OXETHAZAINE 57859 39490 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Vismodegib VISMODEGIB 57861 39491 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME LANREOTIDE LANREOTIDE 17051749 57862 39492 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROCYCLIDINE PROCYCLIDINE 57863 39493 ABAT 18 DRUGGABLE GENOME, ENZYME VIGABATRIN VIGABATRIN 57864 39494 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME HYDROCORTAMATE HYDROCORTAMATE 57867 39495 GAA 2548 DRUGGABLE GENOME, ENZYME 2',3,4-TRIHYDROXYCHALCONE CHEMBL339587 57869 39496 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT 57870 39497 BRCA2 675 CLINICALLY ACTIONABLE OLAPARIB OLAPARIB 57871 39498 EIF2AK4 440275 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565849 57872 39499 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650217 SEOCALCITOL 57874 39500 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545336 SAVOLITINIB 57875 39501 CXCL5 6374 DRUGGABLE GENOME hmg coa reductase inhibitors 18769620 57876 39502 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE PMID26882240-Compound-15 57877 39503 PDE4B 5142 DRUGGABLE GENOME, ENZYME THEOPHYLLINE THEOPHYLLINE 57878 39504 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME MIDAZOLAM MIDAZOLAM 22137933 57879 39505 MAPT 4137 DRUGGABLE GENOME GNF-PF-321 CHEMBL581044 57880 39506 NQO2 4835 DRUGGABLE GENOME, ENZYME doxorubicin DOXORUBICIN 29938344,21946896 57881 39507 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102286 QUIZARTINIB 57882 39508 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME thioguanosine triphosphate 26332308 57883 39509 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Cetuximab CETUXIMAB 25714871 57884 39510 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 310264763 57885 39511 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENARIMOL FENARIMOL 57889 39512 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL3545000 MK-2201 57890 39513 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1201065 THIAMYLAL SODIUM 57893 39514 MAPT 4137 DRUGGABLE GENOME NSC-60340 CHEMBL1534034 57894 39515 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME PMID27998201-Compound-9 57895 39516 F5 2153 DRUGGABLE GENOME eltrombopag ELTROMBOPAG 57896 39517 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178100981 57897 39518 KDM4A 9682 DRUGGABLE GENOME, ENZYME STREPTONIGRIN STREPTONIGRIN 57898 39519 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1200817 LEVOMETHADYL ACETATE HYDROCHLORIDE 57899 39520 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist CHEMBL3545173 IRX4310 57900 39521 RACGAP1 29127 NA ORTHOTOLIDINE ORTHOTOLIDINE 57901 39522 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME RA101495 ZILUCOPLAN 57902 39523 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CHEMBL3833344 GANCOTAMAB 57904 39524 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 252827463 57905 39525 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565754 57906 39526 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR SB-203580 SB-203580 57907 39527 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE RHTPO 11944912 57908 39528 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX DEXAMETHASONE DEXAMETHASONE 23219855 57909 39529 TNIK 23043 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE inhibitor 135652717 STAUROSPORINE 57910 39530 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Isoflavone derivative 4 57912 39531 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Angiotensin II Antagonists 22543981 57914 39532 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Estradiol ESTRADIOL 57915 39533 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE INAMRINONE INAMRINONE 57916 39534 EYA2 2139 DNA REPAIR SJ000032154 CHEMBL591876 57917 39535 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME Everolimus EVEROLIMUS 57920 39536 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PANOBINOSTAT PANOBINOSTAT 57921 39537 KDM4A 9682 DRUGGABLE GENOME, ENZYME RHEIN RHEIN 57922 39538 HTT 3064 DRUGGABLE GENOME NVP-LAQ824 DACINOSTAT 57924 39539 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE OMEPRAZOLE OMEPRAZOLE 57925 39540 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HYDROXYZINE PAMOATE HYDROXYZINE PAMOATE 57927 39541 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE FLUDARABINE FLUDARABINE 57928 39542 MAPT 4137 DRUGGABLE GENOME GNF-PF-521 CHEMBL580071 57933 39543 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE LY-411575 CHEMBL392068 23181502,19443228 57934 39544 KDM4A 9682 DRUGGABLE GENOME, ENZYME RESERPINE RESERPINE 57935 39545 ABI1 10006 CLINICALLY ACTIONABLE, KINASE dasatinib DASATINIB 57936 39546 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102321 57937 39547 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE allosteric modulator 405560349 57938 39548 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Tricyclic indole compound 13 57940 39549 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME FLUNARIZINE FLUNARIZINE 57941 39550 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2-ETHOXYCARBONYL-2-ETHOXYOXALOYLOXYDIHYDROCHRYSIN DIMETHYL ETHER 2-ETHOXYCARBONYL-2-ETHOXYOXALOYLOXYDIHYDROCHRYSIN DIMETHYL ETHER 57942 39551 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE SR-59230A CHEMBL1326499 57943 39552 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-Table1Example11 57945 39553 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME AT-7519 AT-7519 18656911 57947 39554 HSPG2 3339 KINASE, DRUGGABLE GENOME CSA CYCLOSPORINE 14974815 57948 39555 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-19 57949 39556 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE PACLITAXEL PACLITAXEL 9174131 57950 39557 ATXN2 6311 NA GNF-PF-3148 CHEMBL81782 57951 39558 TUBB2A 7280 DRUGGABLE GENOME CHEMBL2108628 PACLITAXEL POLIGLUMEX 57952 39559 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702260 DEBIO-1347 57953 39560 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR DIMETHYLADENINE DIMETHYLADENINE 57954 39561 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor DABRAFENIB DABRAFENIB 57956 39562 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR MESTRANOL MESTRANOL 57957 39563 HSPE1 3336 NA XToll 57958 39564 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000032149 CHEMBL600778 57959 39565 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME galantamine GALANTAMINE 23503455 57961 39566 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DESMOSTEROL DESMOSTEROL 23910990 57962 39567 TGFBR2 7048 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME inhibitor 249565874 57963 39568 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 57965 39569 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MEFENAMIC ACID MEFENAMIC ACID 57966 39570 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 252166588 ERTUGLIFLOZIN 57967 39571 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE LONIDAMINE LONIDAMINE 57968 39572 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE EPIRUBICIN EPIRUBICIN 14503796 57970 39573 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (+)-VENTILOQUINONE CHEMBL594257 19783445 57971 39574 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545000 MK-2201 57972 39575 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE SUNITINIB SUNITINIB 57975 39576 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GABAZINE GABAZINE 57976 39577 MARCHF8 220972 ENZYME Polyoxidonium 57977 39578 RGS5 8490 NA bevacizumab BEVACIZUMAB 25069475 57978 39579 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CEP-1347 CEP-1347 24044867 57979 39580 AKR1B1 231 DRUGGABLE GENOME, ENZYME ALO-1567 57980 39581 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652251 57981 39582 SCTR 6344 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL3039582 SECRETIN 57982 39583 MAOB 4129 DRUGGABLE GENOME, ENZYME MELATONIN MELATONIN 9726430 57984 39584 SMAD2 4087 KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX BLM BLEOMYCIN 17274978 57985 39585 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE PHENCYCLIDINE HYDROCHLORIDE PHENCYCLIDINE HYDROCHLORIDE 57986 39586 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CHEMBL1200789 TRICLOFOS SODIUM 57987 39587 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BENZYL ISOTHIOCYANATE BENZYL ISOTHIOCYANATE 57988 39588 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME XANTHOANGELOL B XANTHOANGELOL B 57989 39589 ATXN2 6311 NA IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 57990 39590 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IMMUNOSUPPRESSIVE 17571057 57992 39591 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DOMIPHEN BROMIDE DOMIPHEN BROMIDE 57993 39592 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650210 57995 39593 CA9 768 DRUGGABLE GENOME, ENZYME COUMATE 57996 39594 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tacrine TACRINE 58004 39595 PSMD3 5709 NA inhibitor CARFILZOMIB CARFILZOMIB 58005 39596 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor 178103944 APREMILAST 58007 39597 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME Pyridopyrimidine derivative 1 58008 39598 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORANIL CHLORANIL 58009 39599 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME MIDAZOLAM MIDAZOLAM 58010 39600 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PROGESTERONE PROGESTERONE 21315613 58011 39601 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME (S)APOMORPHINE (S)APOMORPHINE 58013 39602 EYA2 2139 DNA REPAIR GNF-PF-2272 CHEMBL601757 58014 39603 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE DITOLYLGUANIDINE DITOLYLGUANIDINE 58016 39604 ADAMTS4 9507 ENZYME, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE 1607004-34-1 58019 39605 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE quinine QUININE 407765 58020 39606 POLK 51426 DNA REPAIR, ENZYME PENICILLIOL B PENICILLIOL B 19223184 58021 39607 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE TCMDC-124307 CHEMBL546865 58022 39608 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 178102516 VEMURAFENIB 58023 39609 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING QUINAPRIL HYDROCHLORIDE QUINAPRIL HYDROCHLORIDE 58024 39610 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RIFAPENTINE RIFAPENTINE 58026 39611 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NIMUSTINE NIMUSTINE 58028 39612 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 178102619 58030 39613 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BI-847325 25873592 58033 39614 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-F2 58034 39615 PSMA6 5687 PROTEASE, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 24524217 58035 39616 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME ELLIPTECINE ELLIPTECINE 58038 39617 HTT 3064 DRUGGABLE GENOME PIRARUBICIN PIRARUBICIN 58039 39618 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DOPAMINE DOPAMINE 58040 39619 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 404859045 58041 39620 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565822 BALANOL 58042 39621 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME AG-538 CHEMBL56393 58043 39622 KDM4A 9682 DRUGGABLE GENOME, ENZYME QUINOLINIC ACID QUINOLINIC ACID 58044 39623 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651223 T091317 58045 39624 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-645827 CHEMBL95704 58046 39625 TAPBP 6892 TRANSPORTER aspirin ASPIRIN 23736108 58047 39626 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR REL-BENDIGOLE D CHEMBL1915269 21684166 58048 39627 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor BELINOSTAT BELINOSTAT 58051 39628 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME Apratastat APRATASTAT 58052 39629 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME METHOTRIMEPRAZINE LEVOMEPROMAZINE 58053 39630 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ZAPRINAST ZAPRINAST 58054 39631 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE CHEMBL502774 58056 39632 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DEXAMETHASONE DEXAMETHASONE 58057 39633 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Isoflavone derivative 7 58058 39634 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US8524917, 11 58061 39635 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE L-NOREPINEPHRINE L-NOREPINEPHRINE 58062 39636 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE DITHIAZANINE IODIDE DITHIAZANINE IODIDE 58063 39637 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE 1-O-ACETYLGEOPYXIN A CHEMBL1902074 58064 39638 HLA-E 3133 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE certolizumab pegol 58065 39639 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650300 GENISTEIN 58066 39640 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE inhibitor CHEMBL877 TRANEXAMIC ACID 58067 39641 NRP1 8829 DRUGGABLE GENOME ranibizumab RANIBIZUMAB 26426212 58068 39642 NDUFA6 4700 ENZYME inhibitor CHEMBL3545320 ME-344 58069 39643 POLK 51426 DNA REPAIR, ENZYME PLUMBAGIN PLUMBAGIN 58070 39644 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 404859077 58071 39645 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 58072 39646 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME LUTEOLIN LUTEOLIN 58073 39647 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor 178103420 ETHOXZOLAMIDE 58076 39648 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE BARASERTIB BARASERTIB 58079 39649 BAZ2B 29994 NA MMV006513 CHEMBL585622 58080 39650 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor SOPHORETIN QUERCETIN 58082 39651 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME inhibitor 178103581 58085 39652 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 sulfinpyrazone SULFINPYRAZONE 9187528 58086 39653 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-5052 CHEMBL601367 58088 39654 F13A1 2162 DRUGGABLE GENOME, ENZYME photodynamic therapy 58089 39655 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME SJ000262801 CHEMBL605077 58094 39656 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PURVALANOLA PURVALANOLA 58095 39657 MAPT 4137 DRUGGABLE GENOME SAPPANONE A TRIMETHYL ETHER SAPPANONE A TRIMETHYL ETHER 58098 39658 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649679 58099 39659 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL ESTAZOLAM ESTAZOLAM 58101 39660 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME RG-1530 RG-1530 58102 39661 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GSK961081 BATEFENTEROL 58103 39662 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-104 58104 39663 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME PLX7904 26466569 58105 39664 EPHA6 285220 DRUGGABLE GENOME, KINASE, TYROSINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 58111 39665 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 7,8,2'-TRIHYDROXYFLAVONE CHEMBL244707 58112 39666 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 315661124 ERDAFITINIB 58113 39667 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE SELUMETINIB SELUMETINIB 22425996 58116 39668 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME PMID27998201-Compound-17 58119 39669 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CAFFEINE CAFFEINE 22931300 58120 39670 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME IL-13 7743667 58121 39671 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME BERGAMOTTIN BERGAMOTTIN 22222157 58123 39672 ATXN2 6311 NA THIOMERSAL THIMEROSAL 58125 39673 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE TIMOLOL MALEATE 12219997 58128 39674 SLC12A2 6558 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178101539 BUMETANIDE 58132 39675 POLK 51426 DNA REPAIR, ENZYME ROBINETIN ROBINETIN 58133 39676 FNTA 2339 ENZYME, DRUGGABLE GENOME TIPIFARNIB TIPIFARNIB 58137 39677 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE Imatinib IMATINIB 17555450 58138 39678 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE MECASERMIN RINFIBATE 58139 39679 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C22 58141 39680 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200837 LEVOBETAXOLOL HYDROCHLORIDE 58143 39681 THY1 7070 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE THYMOSIN FRACTION 5 6141799 58144 39682 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME N-DESMETHYLCLOZAPINE N-DESMETHYLCLOZAPINE 58145 39683 NPC1L1 29881 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL1138 EZETIMIBE 58146 39684 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL RG7893 RG7893 58147 39685 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIPHENADIONE DIPHENADIONE 58148 39686 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE activator 354702240 PEMIGATINIB 58149 39687 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178102585 DOVITINIB 58150 39688 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CYC-116 CYC-116 58153 39689 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME GNF-PF-2301 CHEMBL578061 58154 39690 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME AGT-182 58157 39691 VIM 7431 DRUGGABLE GENOME DIMETHYL SULFOXIDE 6376521 58158 39692 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 348353671 58159 39693 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 midazolam MIDAZOLAM 25287072,19255940,9187528,26114223,23327575 58160 39694 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 10 58161 39695 CBX1 10951 NA DNDI1417941 CHEMBL2095095 58164 39696 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103490 58165 39697 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor PF-03814735 PF-03814735 58167 39698 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RIFAMYCIN SODIUM RIFAMYCIN SODIUM 58168 39699 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CID 94381 CHEMBL374632 58170 39700 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PROGESTERONE PROGESTERONE 14557489 58171 39701 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DEMECLOCYCLINE DEMECLOCYCLINE 58173 39702 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE JUGLONE JUGLONE 58175 39703 PSMB6 5694 DRUGGABLE GENOME, PROTEASE, ENZYME BORTEZOMIB BORTEZOMIB 24524217 58176 39704 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 carbamazepine CARBAMAZEPINE 12386121,19702528,19442086,11038165,14704462,8886611 58180 39705 TLR7 51284 DRUGGABLE GENOME GSK2245035 GSK-2245035 58181 39706 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SJ000079774 CHEMBL601192 58182 39707 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME agonist 178101620 EPOETIN BETA 58184 39708 SLC30A9 10463 TRANSPORTER, NUCLEAR HORMONE RECEPTOR aspirin ASPIRIN 58185 39709 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 223365926 BUTORPHANOL 58186 39710 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Doxorubicin DOXORUBICIN 27924459 58187 39711 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor DACOMITINIB DACOMITINIB 58189 39712 FTO 79068 ENZYME ethanol ALCOHOL 32451486 58190 39713 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL411907 SONOLISIB 58191 39714 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME imatinib IMATINIB 24293093 58192 39715 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER sirolimus SIROLIMUS 23073467,28676933 58193 39716 DEGS1 8560 ENZYME inhibitor 252827536 58194 39717 CD38 952 CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1743007 DARATUMUMAB 58195 39718 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR IL-9 17446528 58196 39719 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CARBOPROST TROMETHAMINE 58200 39720 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RS-16566 CHEMBL145725 58201 39721 GMNN 51053 DRUGGABLE GENOME APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 58202 39722 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201020 DISOPYRAMIDE PHOSPHATE 58204 39723 ME3 10873 ENZYME MALEIC ACID MALEIC ACID 19595601 58205 39724 PTGS2 5743 DRUGGABLE GENOME, ENZYME Meclofenamate Sodium 58206 39725 PTGS2 5743 DRUGGABLE GENOME, ENZYME Etodolac ETODOLAC 58208 39726 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE PACLITAXEL PACLITAXEL 18593940 58209 39727 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE E-3810 RABEPRAZOLE SODIUM 58211 39728 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BISPECIFIC ANTIBODIES 10048973 58212 39729 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BCMA CAR-T 58213 39730 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME dexamethasone DEXAMETHASONE 21228734 58214 39731 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 27 58216 39732 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649866 58220 39733 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor NINTEDANIB NINTEDANIB 58221 39734 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL428647 PACLITAXEL 58223 39735 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME IPRIFLAVONE IPRIFLAVONE 58225 39736 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID29324067-Compound-38 58226 39737 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651255 58229 39738 KDM4A 9682 DRUGGABLE GENOME, ENZYME DIOSMIN DIOSMIN 58230 39739 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL2110368 BETHANIDINE SULFATE 58231 39740 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR GNF-PF-2301 CHEMBL578061 58233 39741 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR PROTEIN KINASE INHIBITOR 1735464 58236 39742 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651568 58237 39743 CD55 1604 DRUGGABLE GENOME, CELL SURFACE RETINOIC ACID 15668483 58238 39744 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 58239 39745 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX R667 58240 39746 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME mirtazapine MIRTAZAPINE 22926595 58242 39747 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Ciprofibrate CIPROFIBRATE 58243 39748 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR dexamethasone DEXAMETHASONE 24141364 58244 39749 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME ISOKAEMPFERIDE ISOKAEMPFERIDE 58245 39750 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL2110725 VINFLUNINE 58246 39751 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER antipsychotics 22909202 58249 39752 ISG15 9636 ENZYME, DRUGGABLE GENOME inhibitor IRINOTECAN IRINOTECAN 58250 39753 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CYC-800 58252 39754 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-A2 58253 39755 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201643 INSULIN ZINC SUSP PROMPT PURIFIED PORK 58254 39756 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR lusutrombopag LUSUTROMBOPAG 58257 39757 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774822-Compound-Figure7Example63 58258 39758 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL57242 AZILSARTAN 58259 39759 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 58260 39760 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PSEUDOEPHEDRINE PSEUDOEPHEDRINE 58261 39761 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SANGUINARIUM SANGUINARIUM 58262 39762 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650592 58263 39763 MARCHF8 220972 ENZYME HEV-239 58264 39764 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TESTOSTERONE TESTOSTERONE 1846593 58265 39765 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE K252a 12118367 58266 39766 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIENOCHLOR DIENOCHLOR 58267 39767 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR AG-555 CHEMBL53898 58270 39768 CXCL8 3576 DRUGGABLE GENOME 1-O-ACETYLGEOPYXIN A CHEMBL1902074 58271 39769 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545052 FIMEPINOSTAT 58272 39770 PRKAR2B 5577 ENZYME, KINASE THEOPHYLLINE THEOPHYLLINE 2893795 58273 39771 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-62 58274 39772 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CHEMBL1102 GLUTETHIMIDE 58275 39773 TNNC1 7134 DRUGGABLE GENOME Dihydroxyaluminium 58276 39774 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME INDOMETHACIN INDOMETHACIN 18832692 58277 39775 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000002502 CHEMBL591630 58278 39776 LGR6 59352 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100587 58279 39777 CRKL 1399 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE GEFITINIB GEFITINIB 22586683 58282 39778 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE N/A 58283 39779 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CEFTRIAXONE CEFTRIAXONE 22931300 58285 39780 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 363894213 58286 39781 KMT5B 51111 DNA REPAIR, METHYL TRANSFERASE, ENZYME inhibitor 310264730 58287 39782 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 178102645 58288 39783 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CEFOXITIN CEFOXITIN 22166395 58289 39784 ARSA 410 DRUGGABLE GENOME, ENZYME DECAMETHONIUM DECAMETHONIUM 58290 39785 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist 187051788 PEGVISOMANT 58295 39786 F3 2152 DRUGGABLE GENOME, CELL SURFACE TT-173 58296 39787 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 381118814 58297 39788 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DX-8951F EXATECAN MESYLATE 10639573 58298 39789 KDM4A 9682 DRUGGABLE GENOME, ENZYME TANSHINONE I TANSHINONE I 58301 39790 TUBA3D 113457 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 58302 39791 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME (4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE (4-CHLOROPHENYL)(MORPHOLINO)METHANETHIONE 58303 39792 HEXA 3073 DRUGGABLE GENOME, ENZYME ECHINOMYCIN ECHINOMYCIN 58304 39793 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565834 58308 39794 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME XL281 58310 39795 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR UVB 16951152 58313 39796 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ABSCISIC ACID ABSCISIC ACID 58314 39797 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME HALAZEPAM HALAZEPAM 58315 39798 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR CAMPTOTHECIN CAMPTOTHECIN 10428835 58316 39799 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME STICTIC ACID STICTIC ACID 58318 39800 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME DIETHYL-2-PENTADECYLMALONATE CHEMBL1797713 21292492 58319 39801 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 381118858 58320 39802 KDM4A 9682 DRUGGABLE GENOME, ENZYME FANCHININ FANCHININ 58321 39803 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Englitazone sodium 58322 39804 F7 2155 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 178103166 58323 39805 TOP2B 7155 DRUGGABLE GENOME, ENZYME XR-5944 58324 39806 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PACLITAXEL PACLITAXEL 58325 39807 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE TRIFLUOPERAZINE TRIFLUOPERAZINE 7595077 58326 39808 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 336446957 58327 39809 CYP27A1 1593 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 cholic acid 58329 39810 BRDT 676 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE inhibitor 187051825 58330 39811 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME NITROGLYCERIN NITROGLYCERIN 8968066 58331 39812 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Progesterone PROGESTERONE 58332 39813 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME TAE-684 TAE-684 58333 39814 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE AZD5363 CAPIVASERTIB 26910118,22294718 58335 39815 ENPP2 5168 ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 315661228 58336 39816 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor AT9283 AT-9283 58337 39817 ALB 213 TRANSPORTER, DRUGGABLE GENOME WARFARIN WARFARIN 17560104 58338 39818 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE BRYOSTATIN BRYOSTATIN 58339 39819 CD248 57124 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Ontuxizumab ONTUXIZUMAB 58340 39820 RACGAP1 29127 NA PINORESINOL PINORESINOL 58341 39821 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME SAR 1118 58342 39822 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PAZOPANIB PAZOPANIB 58343 39823 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LOSARTAN LOSARTAN 58344 39824 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME JNK INHIBITOR VIII CHEMBL210618 58345 39825 ALOX5 240 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL704 MESALAMINE 58346 39826 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IOPHENOXIC ACID IOPHENOXIC ACID 58347 39827 DNER 92737 NA Isoxazole-based bicyclic compound 13 58348 39828 NOS2 4843 DRUGGABLE GENOME, ENZYME OPIATE 11715524 58349 39829 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-74429 CHEMBL1269022 58352 39830 KCNK5 8645 ION CHANNEL, DRUGGABLE GENOME activator 135650346 HALOTHANE 58354 39831 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME MIFEPRISTONE MIFEPRISTONE 58355 39832 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GEFITINIB GEFITINIB 58358 39833 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR CRYPTOCHINONE B CRYPTOCHINONE B 25127166 58360 39834 ATAD5 79915 NA NSC-636948 CHEMBL1998001 58361 39835 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE PIPERONYL BUTOXIDE PIPERONYL BUTOXIDE 58362 39836 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102310 58363 39837 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DOXYCYCLINE DOXYCYCLINE 58364 39838 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER MEDI1341 58366 39839 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CLOBAZAM CLOBAZAM 58367 39840 ACVR1B 91 SERINE THREONINE KINASE, CELL SURFACE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE US10030004, Compound 33 58368 39841 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652241 58375 39842 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW581744X GW581744X 58376 39843 ATXN2 6311 NA FANGCHINOLINE FANGCHINOLINE 58377 39844 E2F1 1869 TRANSCRIPTION FACTOR 5-FLUOROURACIL FLUOROURACIL 9766655 58378 39845 POLA1 5422 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, DNA REPAIR FLUDARABINE FLUDARABINE 58380 39846 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-58 58381 39847 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIROXICAM PIROXICAM 22931300 58383 39848 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor E-3810 RABEPRAZOLE SODIUM 58386 39849 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 58388 39850 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME DIPHENYLUREA DIPHENYLUREA 58389 39851 GLS 2744 ENZYME EVANS BLUE EVANS BLUE 58391 39852 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-125103 CHEMBL530281 58393 39853 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor VORINOSTAT VORINOSTAT 58394 39854 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME RXDX 101 58397 39855 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 paclitaxel PACLITAXEL 21151855,16890579,9187528,25398452 58400 39856 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PHENYLBUTYRYLHYDROXAMIC ACID PHENYLBUTYRYLHYDROXAMIC ACID 21874153 58401 39857 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL463981 BEGACESTAT 58402 39858 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE NSC-180246 CHEMBL484640 58403 39859 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PERSEITOL PERSEITOL 58404 39860 MAPT 4137 DRUGGABLE GENOME OMEPRAZOLE OMEPRAZOLE 58405 39861 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103648 DOXORUBICIN 58407 39862 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor BEZ235 DACTOLISIB 58408 39863 POLK 51426 DNA REPAIR, ENZYME DITHIAZANINE DITHIAZANINE 58409 39864 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Rasburicase RASBURICASE 58410 39865 HEXA 3073 DRUGGABLE GENOME, ENZYME TCMDC-124296 CHEMBL22148 25984755 58411 39866 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER aripiprazole ARIPIPRAZOLE 29443543 58412 39867 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ETHAMSYLATE ETHAMSYLATE 58413 39868 IL1B 3553 KINASE, DRUGGABLE GENOME etidronic acid 16257277 58414 39869 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565841 58415 39870 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME JNJ-42756493 ERDAFITINIB 28341788 58418 39871 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LEVOBUNOLOL LEVOBUNOLOL 58419 39872 IMPDH2 3615 DRUGGABLE GENOME, ENZYME mycophenolic acid 21996196,19770842,24220207,20679962,18444945,19617864,22960765 58420 39873 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 58421 39874 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIDANOSINE DIDANOSINE 22931300 58422 39875 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME Dihydrothieno [2,3-e]indazole derivative 2 58423 39876 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TAMOXIFEN TAMOXIFEN 11306479 58424 39877 ALOX15B 247 DRUGGABLE GENOME, ENZYME DIPYRIDAMOLE DIPYRIDAMOLE 58425 39878 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 375973233 58428 39879 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR EFAVIRENZ EFAVIRENZ 58429 39880 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME KX-02 KX2-361 58431 39881 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 178102628 58432 39882 MAPT 4137 DRUGGABLE GENOME PATULIN PATULIN 58434 39883 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER cyanocobalamin CYANOCOBALAMIN 58435 39884 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 5,8,11,14-EICOSATETRAYNOIC ACID CHEMBL458328 58436 39885 ATAD2 29028 NUCLEAR HORMONE RECEPTOR, ENZYME inhibitor 252166840 58437 39886 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GS-9820 ACALISIB 58438 39887 COMT 1312 DRUGGABLE GENOME, ENZYME remifentanil REMIFENTANIL 28006928,23686330,21398039,23302985,26902643,29474345,23773341,25155931,25185591,19514130,28745577,27027462 58440 39888 HLA-G 3135 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME fluorouracil FLUOROURACIL 58441 39889 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 4-PHENYLIMIDAZOLE CHEMBL14145 24262887 58443 39890 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor 187051805 QUISINOSTAT 58444 39891 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PHA-665752 PHA-665752 26124204 58446 39892 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE AZD-1152-HQPA AZD-1152-HQPA 25036791 58447 39893 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE DIPYRIDAMOLE DIPYRIDAMOLE 1716731 58448 39894 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE CERITINIB CERITINIB 23837797 58450 39895 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Palbociclib PALBOCICLIB 22711607,27488531,21871868,20952405,22983396,26380006,26183925,23898052 58454 39896 MSH5 4439 NA carboplatin CARBOPLATIN 31616045 58456 39897 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR MIDAZOLAM MIDAZOLAM 22137933 58457 39898 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist CHEMBL3545392 MT-3995 58458 39899 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PAROXETINE HYDROCHLORIDE PAROXETINE HYDROCHLORIDE 58459 39900 SMN1 6606 DRUGGABLE GENOME THIABENDAZOLE THIABENDAZOLE 58460 39901 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051804 RESMINOSTAT 58461 39902 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 7-Veratraldehyde 58462 39903 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 381118877 TOMIVOSERTIB 58463 39904 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL XP13512 GABAPENTIN ENACARBIL 58465 39905 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 58466 39906 CDKL1 8814 TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565840 58467 39907 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 paclitaxel PACLITAXEL 16890579 58470 39908 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DICUMAROL DICUMAROL 58473 39909 ABAT 18 DRUGGABLE GENOME, ENZYME DP-VPA 58474 39910 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE agonist CHEMBL983 SUCCINYLCHOLINE CHLORIDE 58476 39911 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMIODARONE AMIODARONE 16537817 58478 39912 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE CHEMBL3544914 TEZACAFTOR 58480 39913 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME PSEUDOEPHEDRINE PSEUDOEPHEDRINE 58481 39914 FST 10468 DRUGGABLE GENOME RETINOIC ACIDS 1520319 58482 39915 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor VANDETANIB VANDETANIB 58483 39916 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33o 58484 39917 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CALOTHRIXIN B CALOTHRIXIN B 19203291 58485 39918 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME MLN8054 58486 39919 SLC22A5 6584 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME imatinib IMATINIB 28762371,23127916 58487 39920 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR GSK126 26936398,26360609,26304929,25605023 58488 39921 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NORADRENALINE NOREPINEPHRINE BITARTRATE 58489 39922 ALDH1A2 8854 DRUGGABLE GENOME, ENZYME RETINOIDS 11751205 58490 39923 MUC16 94025 DRUGGABLE GENOME OREGOVAMAB OREGOVOMAB 58491 39924 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Daniquidone DANIQUIDONE 58492 39925 POLI 11201 DNA REPAIR 4-AMINOPHENOL 4-AMINOPHENOL 58493 39926 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649943 ANATIBANT 58496 39927 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200600 FLUOROMETHOLONE 58497 39928 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 249565683 BERZOSERTIB 58498 39929 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME SJ000291864 CHEMBL592566 58499 39930 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 4'-HYDROXYPHENYL-BENZO[D]THIAZOLE CHEMBL47875 58500 39931 ALB 213 TRANSPORTER, DRUGGABLE GENOME DICLOFENAC DICLOFENAC 17560104 58501 39932 HTT 3064 DRUGGABLE GENOME GNF-PF-2906 CHEMBL579957 58502 39933 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 QUINIDINE QUINIDINE 22931300,19117415 58503 39934 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CYC-116 CYC-116 58504 39935 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER SIMVASTATIN SIMVASTATIN 15616150 58505 39936 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ALPRENOLOL ALPRENOLOL 2903243 58506 39937 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NICORANDIL NICORANDIL 58507 39938 LSS 4047 ENZYME, DRUGGABLE GENOME inhibitor 178103326 58508 39939 GC 2638 DRUGGABLE GENOME Nitric Oxide 58509 39940 CA2 760 DRUGGABLE GENOME, ENZYME Cyclothiazide CYCLOTHIAZIDE 58510 39941 RAB9A 9367 ENZYME, DRUGGABLE GENOME NSC-93401 CHEMBL452954 58511 39942 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist 135650520 BEXAROTENE 58512 39943 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BECLOMETHASONE BECLOMETHASONE 22931300 58513 39944 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE DEXAMETHASONE DEXAMETHASONE 29408328 58514 39945 TXNRD2 10587 DRUGGABLE GENOME Selective serotonin reuptake inhibitors 58515 39946 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR leflunomide LEFLUNOMIDE 21174621 58516 39947 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME MISTLETOE LECTIN 11690563 58517 39948 TAC1 6863 DRUGGABLE GENOME NALTREXONE NALTREXONE 7536308 58518 39949 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Epoprostenol EPOPROSTENOL 58521 39950 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor 178101536 TETRABENAZINE 58522 39951 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4'-METHOXYCHALCONE 4'-METHOXYCHALCONE 58523 39952 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL52885 ENMD-981693 58524 39953 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 249565816 58526 39954 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor PD0332991 PALBOCICLIB 58527 39955 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CANFOSFAMIDE CANFOSFAMIDE 58528 39956 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE AZD5363 CAPIVASERTIB 58529 39957 RAB9A 9367 ENZYME, DRUGGABLE GENOME TCMDC-125353 CHEMBL547924 58530 39958 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 5-NITRO-2-PHENYLPROPYLAMINOBENZOIC ACID [NPPB] 5-NITRO-2-PHENYLPROPYLAMINOBENZOIC ACID [NPPB] 58533 39959 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE CI-966 CHEMBL77287 58536 39960 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MODAFINIL MODAFINIL 22931300 58537 39961 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CUDC-101 CUDC-101 58538 39962 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417607 CHEMBL1588679 58542 39963 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TNF-ALPHA 7629160 58543 39964 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1200327 PENTAZOCINE LACTATE 58546 39965 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651512 58547 39966 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PMA 12919900 58548 39967 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BETA-LAPACHONE LAPACHONE 58552 39968 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 58553 39969 GMNN 51053 DRUGGABLE GENOME AMSACRINE HYDROCHLORIDE AMSACRINE HYDROCHLORIDE 58554 39970 DHFR 1719 DRUGGABLE GENOME, ENZYME Methotrexate Sodium 58555 39971 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME HYALURONAN HYALURONAN 58556 39972 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1743032 INTETUMUMAB 58558 39973 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor VOLASERTIB VOLASERTIB 58560 39974 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE KENPAULLONE KENPAULLONE 58562 39975 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR KENPAULLONE KENPAULLONE 58563 39976 SLC23A2 9962 TRANSPORTER Ursodeoxycholic acid 58564 39977 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ARSENIC TRIOXIDE 58565 39978 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME DIAZEPAM DIAZEPAM 58566 39979 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE MK-0752 MK-0752 58567 39980 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER NSC-50650 CHEMBL1561747 58569 39981 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE GS-9876 58572 39982 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME PHENYTOIN PHENYTOIN 15458527 58573 39983 HTT 3064 DRUGGABLE GENOME FASUDIL HYDROCHLORIDE FASUDIL HYDROCHLORIDE 58574 39984 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 58575 39985 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Sulfasalazine SULFASALAZINE 58577 39986 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GSK1210151A CHEMBL2017291 25559428 58578 39987 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VORINOSTAT VORINOSTAT 58579 39988 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1200807 NORELGESTROMIN 58581 39989 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-24 58582 39990 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GW441756X GW441756X 58584 39991 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652710 RAUWOLSCINE 58586 39992 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor DACOMITINIB DACOMITINIB 58587 39993 BAZ2B 29994 NA MK-886 CHEMBL29097 58588 39994 MAOB 4129 DRUGGABLE GENOME, ENZYME T83193 58589 39995 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ETHYLENEDIAMINE ETHYLENEDIAMINE 58590 39996 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CARMINOMYCIN CARUBICIN 58591 39997 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR obeticholic acid 58593 39998 IL13RA2 3598 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME MB-101 58595 39999 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE inhibitor CHEMBL2109621 ABITUZUMAB 58597 40000 SLC12A4 6560 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSPORTER inhibitor 178101310 58601 40001 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Tenecteplase TENECTEPLASE 58602 40002 CDK13 8621 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL488436 AZD-5438 58603 40003 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BMS-387032 BMS-387032 58605 40004 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CAPIVASERTIB CAPIVASERTIB 22294718 58608 40005 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL1096380 PLINABULIN 58610 40006 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 58611 40007 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TREQUINSIN HYDROCHLORIDE TREQUINSIN HYDROCHLORIDE 58613 40008 SMAD7 4092 KINASE TPA ALTEPLASE 15033458 58614 40009 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TYRPHOSTIN 25 TYRPHOSTIN 25 58618 40010 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CETIRIZINE DIHYDROCHLORIDE CETIRIZINE HYDROCHLORIDE 58619 40011 PRKAB2 5565 KINASE, ENZYME METFORMIN METFORMIN 26471090 58620 40012 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PICTILISIB PICTILISIB 27489350,23674493,23888070 58621 40013 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME Tricyclic isoxazoloquinazoline derivative 3 58622 40014 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166819 58624 40015 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 328083525 NEMIRALISIB 58627 40016 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-N3 58629 40017 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PMID27774822-Compound-Figure1Example20 58631 40018 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE AM-152 58633 40019 CLCA1 1179 DRUGGABLE GENOME TALNIFLUMATE TALNIFLUMATE 58635 40020 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE L-655240 CHEMBL362223 58636 40021 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 178100876 58639 40022 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 374883888 58641 40023 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor ICOTINIB ICOTINIB 58642 40024 REEP5 7905 NA paroxetine PAROXETINE 22795047 58643 40025 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651155 58646 40026 GJA1 2697 ION CHANNEL inhibitor 135650269 58647 40027 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9522888, 695 58648 40028 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ARRY-380 TUCATINIB 58649 40029 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 23 58651 40030 PSMD3 5709 NA CARFILZOMIB CARFILZOMIB 24524217 58652 40031 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Fasudil FASUDIL 58653 40032 POLB 5423 DNA REPAIR, DRUGGABLE GENOME S(+)-ISOPROTERENOL-BITARTRATE CHEMBL1257092 58654 40033 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ALITRETINOIN ALITRETINOIN 58655 40034 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE RAPAMYCIN SIROLIMUS 15683719 58656 40035 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GLUCOCORTICOID 6972103 58657 40036 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DOCEBENONE DOCEBENONE 58660 40037 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME flucloxacillin FLOXACILLIN 23596311,23132554,24731753,18637831,23291545,19696695,23032409,18256392,19483685,30664875 58661 40038 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Intravenous minocycline 58662 40039 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BINODENOSON BINODENOSON 58664 40040 PDE6A 5145 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL932 DIPYRIDAMOLE 58665 40041 CES1 1066 DRUGGABLE GENOME, ENZYME heroin DIACETYLMORPHINE 31837295 58666 40042 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Imatinib IMATINIB 27924459 58668 40043 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ERLOTINIB ERLOTINIB 17047074 58669 40044 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR THIOMERSAL THIMEROSAL 58670 40045 MAOA 4128 DRUGGABLE GENOME, ENZYME 1-PHENETHYLPIPERIDINE 1-PHENETHYLPIPERIDINE 22078410 58672 40046 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DIGOXIGENIN DIGOXIGENIN 58673 40047 POLI 11201 DNA REPAIR BISINDOLYLMALEIMIDE IX BISINDOLYLMALEIMIDE IX 58678 40048 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AURIN AURIN 58680 40049 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME olanzapine OLANZAPINE 23859574,20031235 58683 40050 SMN2 6607 DRUGGABLE GENOME CID 1225609 CHEMBL444376 58684 40051 NOS1 4842 DRUGGABLE GENOME, ENZYME NEUROTROPHIC FACTOR 9216986 58685 40052 KMO 8564 DRUGGABLE GENOME, ENZYME Benzene sulfonamide derivative 1 58687 40053 CA9 768 DRUGGABLE GENOME, ENZYME INDISULAM INDISULAM 58688 40054 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1356607 NOREPINEPHRINE BITARTRATE 58689 40055 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME METHIMAZOLE METHIMAZOLE 15504312 58690 40056 MAOB 4129 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 3 58691 40057 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201635 INSULIN SUSP ISOPHANE BEEF/PORK 58694 40058 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME IMATINIB IMATINIB 58696 40059 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 135650390 INDOMETHACIN 58697 40060 RAMP1 10267 DRUGGABLE GENOME, CELL SURFACE agonist CHEMBL3833353 PRAMLINTIDE ACETATE 58698 40061 RBX1 9978 DNA REPAIR, ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 58699 40062 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DHT ANDROSTANOLONE 12532336 58700 40063 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32d 58701 40064 RAPGEF3 10411 ENZYME ACID BLUE 129 ACID BLUE 129 58702 40065 VCAM1 7412 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 7694584 58704 40066 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178100902 58705 40067 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Trichostatin A 18483379,23498719 58706 40068 TLR7 51284 DRUGGABLE GENOME AZD-8848 AZD-8848 58707 40069 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417268 CHEMBL1517542 58709 40070 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antibody AVELUMAB AVELUMAB 58710 40071 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VERAPAMIL VERAPAMIL 58711 40072 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY VITAMIN D 6250216 58712 40073 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Five-membered heteroaromatic compound 3 58713 40074 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME PMID27998201-Compound-5 58714 40075 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GLYBURIDE GLYBURIDE 58716 40076 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SJ000293754 CHEMBL486706 58717 40077 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PAZOPANIB PAZOPANIB 27271022 58718 40078 NDUFA8 4702 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 58721 40079 GJA1 2697 ION CHANNEL Granexin gel 58722 40080 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 387065624 58723 40081 TOP1MT 116447 DRUGGABLE GENOME, ENZYME PEG-IRINOTECAN 58724 40082 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651367 ZOTEPINE 58725 40083 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-28 58726 40084 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE KINETIN RIBOSIDE KINETIN RIBOSIDE 58727 40085 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ECADOTRIL ECADOTRIL 58728 40086 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-20 58729 40087 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Topotecan TOPOTECAN 26826116 58731 40088 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650461 58732 40089 PYY 5697 DRUGGABLE GENOME, HORMONE ACTIVITY TYROSINE KINASE INHIBITOR 10970776 58733 40090 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MITOMYCIN MITOMYCIN 22931300 58734 40091 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ESTAZOLAM ESTAZOLAM 58735 40092 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1743088 VELTUZUMAB 58736 40093 NDUFA13 51079 ENZYME, TRANSCRIPTION FACTOR Flurpiridaz F 18 58738 40094 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CHEMBL1200789 TRICLOFOS SODIUM 58739 40095 ATXN2 6311 NA ENNIATIN B ENNIATIN B 58741 40096 BRD9 65980 ENZYME inhibitor 252166608 58742 40097 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 58747 40098 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BAS 8770945 CHEMBL478141 19179076 58748 40099 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GEFITINIB GEFITINIB 58750 40100 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 252166480 VELTUZUMAB 58752 40101 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 135651435 TRETINOIN 58753 40102 CA2 760 DRUGGABLE GENOME, ENZYME inhibitor 385612193 58754 40103 GMNN 51053 DRUGGABLE GENOME EBSELEN EBSELEN 58755 40104 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Phenylpyridine derivative 2 58756 40105 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32n 58757 40106 KDM4A 9682 DRUGGABLE GENOME, ENZYME TAMOXIFEN CITRATE TAMOXIFEN CITRATE 58758 40107 GPI 2821 ENZYME, GROWTH FACTOR, DRUGGABLE GENOME HEREGULIN 10667603 58759 40108 LAMB4 22798 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 58760 40109 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-39 58761 40110 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-1947 CHEMBL585591 58762 40111 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME TRIBUTYRIN TRIBUTYRIN 10629959 58763 40112 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BISOPROLOL BISOPROLOL 2903243 58765 40113 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER RG7935 PRASINEZUMAB 22355802 58766 40114 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE CHEMBL395091 ESKETAMINE 58767 40115 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VERAPAMIL VERAPAMIL 58768 40116 CLU 1191 CELL SURFACE, DRUGGABLE GENOME LUBIPROSTONE LUBIPROSTONE 58769 40117 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE VEMURAFENIB VEMURAFENIB 24265155,22180495 58770 40118 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Ruxolitinib RUXOLITINIB 58771 40119 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LGD-1550 58772 40120 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR INOSITOL INOSITOL 16286649 58773 40121 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor 187051821 OLAPARIB 58774 40122 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME DISULFIRAM DISULFIRAM 58775 40123 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER ALSEROXYLON ALSEROXYLON 58777 40124 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SHIKONIN SHIKONIN 58778 40125 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Saracatinib SARACATINIB 28416483 58780 40126 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TCMDC-124479 CHEMBL587259 58781 40127 GMNN 51053 DRUGGABLE GENOME TCMDC-125150 CHEMBL534244 58783 40128 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR THONZONIUM BROMIDE THONZONIUM BROMIDE 58784 40129 SPTLC3 55304 ENZYME inhibitor 178103276 MYRIOCIN 58787 40130 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1952329 SGI-1776 58789 40131 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 363894217 VORUCICLIB 58790 40132 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE VISILIZUMAB VISILIZUMAB 58791 40133 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 135649931 58795 40134 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE DOVITINIB DOVITINIB 58797 40135 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME amlodipine / atorvastatin / perindopril arginine 58798 40136 CCL2 6347 DRUGGABLE GENOME inhibitor CHEMBL1742999 CARLUMAB 58799 40137 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1417692 CHEMBL1481509 58800 40138 H3-3A 3020 CLINICALLY ACTIONABLE, DRUGGABLE GENOME AKT/ERK INHIBITOR ONC201 58801 40139 CA2 760 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL19 METHAZOLAMIDE 58802 40140 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL198877 AUS-131 58803 40141 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MURAGLITAZAR MURAGLITAZAR 58804 40142 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody PANITUMUMAB PANITUMUMAB 58805 40143 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 1058137-23-7 LUCITANIB 58806 40144 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IPCONAZOLE IPCONAZOLE 58807 40145 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME GENTAMICIN GENTAMICIN 14986132 58808 40146 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME EPOETIN ALFA 58809 40147 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HYDRALAZINE HYDROCHLORIDE HYDRALAZINE HYDROCHLORIDE 58810 40148 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PMID29671355-Compound-62 58811 40149 ATXN2 6311 NA GNF-PF-1339 CHEMBL600353 58812 40150 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE Tumor necrosis factor alpha (TNF-alpha) inhibitors 22480748 58813 40151 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CHELIDAMIC ACID CHELIDAMIC ACID 58814 40152 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR LC-1 20669221 58817 40153 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE BLZ-100 TOZULERISTIDE 58818 40154 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652096 58819 40155 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AMPHETAMINE AMPHETAMINE 9264312 58820 40156 BAD 572 KINASE, DRUGGABLE GENOME RUBOXISTAURIN RUBOXISTAURIN 18077363 58821 40157 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE Analgesics 25096645 58823 40158 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Trametinib TRAMETINIB 27488531 58824 40159 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SNS-314 SNS-314 58825 40160 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3544999 SAMOTOLISIB 58826 40161 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE IT-101 22081768 58828 40162 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 58829 40163 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Canfosfamide CANFOSFAMIDE 58830 40164 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-116702 CHEMBL1477383 58831 40165 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE QUERCETIN QUERCETIN 8759170 58832 40166 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist 252166709 58833 40167 KLK7 5650 ENZYME, PROTEASE, DRUGGABLE GENOME CASTANIN CASTANIN 58834 40168 PDF 64146 DRUGGABLE GENOME Pralatrexate PRALATREXATE 58835 40169 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER quinidine QUINIDINE 58837 40170 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PALIFERMIN PALIFERMIN 58839 40171 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545430 OLMUTINIB 58840 40172 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200413 TETRAHYDROZOLINE HYDROCHLORIDE 58842 40173 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME AT9283 AT-9283 58843 40174 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR partial agonist CHEMBL257978 DABUZALGRON 58847 40175 SMN1 6606 DRUGGABLE GENOME SU-6656 CHEMBL605003 58848 40176 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BW-373U86 CHEMBL25230 58850 40177 DNER 92737 NA ZEN-3694 58851 40178 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist 178100825 58854 40179 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651538 58855 40180 CA1 759 DRUGGABLE GENOME, ENZYME FERULIC ACID 58857 40181 AKR1A1 10327 ENZYME, DRUGGABLE GENOME doxorubicin DOXORUBICIN 21048526 58858 40182 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 dolutegravir DOLUTEGRAVIR 58859 40183 HTT 3064 DRUGGABLE GENOME MIRIPIRIUM MIRIPIRIUM 58860 40184 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE CHEMBL412603 58863 40185 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Sorafenib SORAFENIB 27992451 58864 40186 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Flavopiridol analog 1 58866 40187 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ZEARALENONE ZEARALENONE 58867 40188 ITPR3 3710 ION CHANNEL, DRUGGABLE GENOME antagonist 135652750 58869 40189 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LUCITANIB LUCITANIB 25193991 58870 40190 KDM4A 9682 DRUGGABLE GENOME, ENZYME N,N'-DIPHENYL-P-PHENYLENEDIAMINE N,N'-DIPHENYL-P-PHENYLENEDIAMINE 58872 40191 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR THYMOL IODIDE THYMOL IODIDE 58873 40192 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102922 METHYLGLYOXAL 58874 40193 MAOA 4128 DRUGGABLE GENOME, ENZYME SELEGILINE SELEGILINE 21680183 58876 40194 ENPP2 5168 ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING NSC-34937 CHEMBL1092743 20349977 58877 40195 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME TRIPHENYLSTANNANOL TRIPHENYLSTANNANOL 58878 40196 KDM4A 9682 DRUGGABLE GENOME, ENZYME TANSHINONE IIA TANSHINONE IIA 58879 40197 C1S 716 ENZYME, PROTEASE, DRUGGABLE GENOME antibody 354702279 SUTIMLIMAB 58880 40198 ZNF804A 91752 NA lithium LITHIUM 29121268 58881 40199 MAOA 4128 DRUGGABLE GENOME, ENZYME Isocarboxazid ISOCARBOXAZID 58882 40200 SLC22A3 6581 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER metformin METFORMIN 25920679,20859243,22722338 58885 40201 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 5-NITROACENAPHTHENE CHEMBL423081 58886 40202 PTGS1 5742 ENZYME, DRUGGABLE GENOME INDOMETHACIN INDOMETHACIN 23651359,20684598,22818041 58887 40203 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GUANFACINE GUANFACINE 58888 40204 PLEKHH2 130271 NA verapamil VERAPAMIL 27670767 58889 40205 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-62406 CHEMBL1332182 58890 40206 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 5-(N-METHYL-N-ISOBUTYL)AMILORIDE 5-(N-METHYL-N-ISOBUTYL)AMILORIDE 58891 40207 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker 178102358 58893 40208 PDE4D 5144 DRUGGABLE GENOME, ENZYME RESVERATROL RESVERATROL 58894 40209 MAP3K10 4294 SERINE THREONINE KINASE, ENZYME, KINASE, DRUGGABLE GENOME DASATINIB DASATINIB 58895 40210 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GSK690 26837761 58896 40211 BAZ2B 29994 NA DNDI1417548 CHEMBL2094789 58898 40212 SCNN1A 6337 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1398126 AMILORIDE HYDROCHLORIDE 58900 40213 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SJ000293754 CHEMBL486706 58901 40214 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME DEFEROXAMINE DEFEROXAMINE 9112092 58902 40215 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE N/A 19047918,21901340 58904 40216 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-5 58905 40217 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME L-GLUTAMINE GLUTAMINE 14746834 58907 40218 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AG-555 CHEMBL53898 58908 40219 TDGF1 6997 DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR BIIB 015 58909 40220 NCL 4691 NA IPP-204106 58910 40221 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Metoclopramide METOCLOPRAMIDE 58911 40222 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor 178103625 INDISULAM 58912 40223 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-7 58913 40224 BAZ2B 29994 NA GNF-PF-4300 CHEMBL585656 58914 40225 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE AFURESERTIB HYDROCHLORIDE 58919 40226 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME ANABOLIC STEROID 10336050 58920 40227 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (+)-TETRAHYDROBERBERINE CHEMBL476501 58922 40228 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE X-82 X-82 58923 40229 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PENTACHLOROPHENOL PENTACHLOROPHENOL 58925 40230 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Tlouidine sulfonamide derivative 1 58926 40231 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 363894217 VORUCICLIB 58927 40232 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL378544 VINBLASTINE SULFATE 58928 40233 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Midostaurin MIDOSTAURIN 58930 40234 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PROTEIN PHOSPHATASE INHIBITOR 10854062 58931 40235 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200703 CHLORDIAZEPOXIDE HYDROCHLORIDE 58932 40236 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE COL-3 INCYCLINIDE 58933 40237 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME LEPIRUDIN LEPIRUDIN 58934 40238 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GOSSYPOL GOSSYPOL 58935 40239 HDAC11 79885 DRUGGABLE GENOME, ENZYME BUTANOIC ACID BUTANOIC ACID 19053749 58937 40240 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME KD-025 CHEMBL2005186 58939 40241 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-3343 CHEMBL599943 58940 40242 H2AX 3014 NA DOXORUBICIN DOXORUBICIN 15489221 58941 40243 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE SELUMETINIB SELUMETINIB 2549426,22653968,22808163,18719078,21083380,22253748,19078957,25157968,1328859,22733540 58942 40244 BAZ2B 29994 NA OSM-S-31 CHEMBL1588237 58943 40245 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-4945 CHEMBL585628 58944 40246 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 178101308 SERGLIFLOZIN ETABONATE 58945 40247 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE DESIPRAMINE DESIPRAMINE 58947 40248 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DAUNORUBICIN DAUNORUBICIN 10216102 58948 40249 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor 249565636 BMS-777607 58949 40250 SIK1 150094 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565729 58951 40251 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ETONOGESTREL ETONOGESTREL 58953 40252 LPAR6 10161 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MC-1 58956 40253 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE 178101725 58957 40254 DNER 92737 NA CC-90010 58958 40255 KDM4A 9682 DRUGGABLE GENOME, ENZYME 12-METHYL TETRADECANOIC ACID CHEMBL495852 58960 40256 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL1980391 RG-1530 58962 40257 SAE1 10055 ENZYME, DRUGGABLE GENOME LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 58963 40258 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PMID25416646-Compound-Figure5-A 58965 40259 SLC2A2 6514 TRANSPORTER, DRUGGABLE GENOME GLUFOSFAMIDE GLUFOSFAMIDE 58966 40260 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE LIPIDYL PSEUDOPTERANE D LIPIDYL PSEUDOPTERANE D 19061360 58967 40261 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 3,4-DICHLOROISOCOUMARIN CHEMBL24983 58968 40262 PDE3B 5140 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200578 THEOPHYLLINE SODIUM GLYCINATE 58969 40263 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME CYC-116 CYC-116 58974 40264 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME blocker 135652279 58975 40265 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME bevacizumab BEVACIZUMAB 27139155,23149126,26100253,20124951,23953100,20125120,25955730 58978 40266 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AMCINONIDE AMCINONIDE 58983 40267 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE sorafenib SORAFENIB 28362716 58984 40268 POLI 11201 DNA REPAIR NSC-19803 CHEMBL522983 58985 40269 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ALSTERPAULLONE ALSTERPAULLONE 58986 40270 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ARA-C 9252649 58987 40271 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 363894173 58988 40272 TUBA3C 7278 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 58991 40273 MAPT 4137 DRUGGABLE GENOME RO-318220 BISINDOLYLMALEIMIDE IX 58993 40274 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL inhibitor 178102900 58994 40275 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DISULFIRAM DISULFIRAM 58995 40276 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE SJ000196127 CHEMBL605084 58997 40277 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AG-555 CHEMBL53898 58999 40278 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AG-555 CHEMBL53898 59000 40279 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROMAZINE PROMAZINE 59001 40280 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR NYSTATIN NYSTATIN 12941963 59004 40281 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE LIF 16489447 59007 40282 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 249565635 BMS-754807 59008 40283 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 25314129 59009 40284 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 384403681 59010 40285 CAMK1D 57118 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME TCMDC-125758 CHEMBL546797 59011 40286 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR RO-318220 BISINDOLYLMALEIMIDE IX 59012 40287 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A5 59013 40288 U2AF1 7307 CLINICALLY ACTIONABLE N/A 25465125,22389253,22158538 59014 40289 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME ALISERTIB ALISERTIB 59015 40290 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CHOLESTAN-3BETA,5ALPHA,6BETA-TRIOL CHOLESTAN-3BETA,5ALPHA,6BETA-TRIOL 23830695 59016 40291 MAPT 4137 DRUGGABLE GENOME CHLOROTHALONIL CHLOROTHALONIL 59017 40292 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE IDARUBICIN IDARUBICIN 14501384 59018 40293 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE tamsulosin TAMSULOSIN 18695978 59019 40294 CD8A 925 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE Anti-VEGFR2 CD8 cell therapy 59020 40295 EREG 2069 KINASE, GROWTH FACTOR, DRUGGABLE GENOME panitumumab PANITUMUMAB 59021 40296 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME D-DOPA CHEMBL211670 59023 40297 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4-PHENYLPHENOL CHEMBL73380 59026 40298 TSPO 706 DRUGGABLE GENOME SSR-180575 59029 40299 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Pyrimidinyl compound 4 59033 40300 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Antistasin 59034 40301 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE GNF-PF-1702 CHEMBL600313 59037 40302 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 252827463 59038 40303 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX 2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE CHEMBL502774 59039 40304 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME NERAMEXANE NERAMEXANE 59041 40305 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL1201752 IXABEPILONE 59042 40306 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DESMETHOXYYANGONIN DESMETHOXYYANGONIN 59044 40307 MT-RNR1 4549 KINASE streptomycin STREPTOMYCIN 18830133,16875663,9164619,19682603,16631122,21495045,16458854,12031626,16375862,9831149,17637808,22475488,11857751,27397648,9779807,7689389,20111055,9111378,27427311,17698030,11313749,20416460,16168391,24703164,9950117,21504270,11174059,8285309,18790089,15917167,20353758,16955413,16380089,14699607,17999439,14755216,17341440,19376484,15708009,25515069,15555598,11079536,17434445 59048 40308 HTT 3064 DRUGGABLE GENOME CETRIMIDE CETRIMIDE 59050 40309 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME A-315456 CHEMBL362863 59052 40310 SMN1 6606 DRUGGABLE GENOME GENISTEIN GENISTEIN 59053 40311 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE EMD 1214063 26358474,23553846 59054 40312 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GDC-0425 RG-7602 27815358 59055 40313 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER MILTIRONE MILTIRONE 26339922 59056 40314 ALOX15 246 ENZYME, DRUGGABLE GENOME DEPHOSTATIN DEPHOSTATIN 59057 40315 RPSA 3921 NA DAUNORUBICIN DAUNORUBICIN 15161018 59059 40316 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME JCARH125 59060 40317 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PALBOCICLIB PALBOCICLIB 59061 40318 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8598210, Table XV, 4 59062 40319 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650507 59063 40320 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME SJ000089001 CHEMBL591618 59064 40321 APH1B 83464 PROTEASE, DRUGGABLE GENOME modulator CHEMBL190083 TARENFLURBIL 59065 40322 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor 318164849 CDP840 59066 40323 VDAC1 7416 NA VDA-1102 topical ointment 59067 40324 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650930 ROXINDOLE 59068 40325 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME MEGESTROL ACETATE 9806658 59069 40326 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW572401X GW572401X 59072 40327 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DINOSEB DINOSEB 59074 40328 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 404859079 59081 40329 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417260 CHEMBL2094573 59083 40330 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR NG-MONOMETHYL-L-ARGININE 10215909 59084 40331 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CCT-018159 59085 40332 EPB41 2035 TRANSPORTER nicotine NICOTINE 59087 40333 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE THEAFLAVINS 18591783 59088 40334 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL270995 BRIVANIB ALANINATE 59091 40335 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME DAIDZEIN DAIDZEIN 10508216 59092 40336 TMEM97 27346 NA Fused aryl carbocycle derivative 9 59093 40337 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FLOXURIDINE FLOXURIDINE 22931300 59094 40338 MARCKSL1 65108 KINASE TNF-ALPHA 11483670 59095 40339 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1201581 INFLIXIMAB 59096 40340 MAPT 4137 DRUGGABLE GENOME MAHANIMBINE MAHANIMBINE 59097 40341 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SPIRONOLACTONE SPIRONOLACTONE 976190 59098 40342 DTYMK 1841 KINASE D4T STAVUDINE 15134538 59099 40343 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649765 59100 40344 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 59102 40345 NDUFS6 4726 ENZYME inhibitor CHEMBL3545320 ME-344 59103 40346 MBNL1 4154 DRUGGABLE GENOME RAMATROBAN RAMATROBAN 59104 40347 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME EPCAM-targeted CAR-T cells 59106 40348 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TORSEMIDE TORSEMIDE 22931300 59108 40349 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-95397 CHEMBL429095 59110 40350 BAZ2B 29994 NA GNF-PF-3582 CHEMBL606167 59111 40351 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MENTHOFURAN MENTHOFURAN 22931300 59114 40352 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ROXITHROMYCIN ROXITHROMYCIN 16416302 59115 40353 GGH 8836 PROTEASE, ENZYME, DRUGGABLE GENOME methylphenidate METHYLPHENIDATE 29382897 59117 40354 CGA 1081 DRUGGABLE GENOME, HORMONE ACTIVITY CORTICOSTEROIDS 3106008 59118 40355 ITPR1 3708 ION CHANNEL, KINASE, DRUGGABLE GENOME, TRANSPORTER antagonist 135652675 CAFFEINE 59121 40356 ATAD5 79915 NA DIGOXIN DIGOXIN 59122 40357 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 381118818 59124 40358 LAMB3 3914 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 59126 40359 GSTA1 2938 ENZYME, DRUGGABLE GENOME BROMOSULFOPHTHALEIN SULFOBROMOPHTHALEIN SODIUM 22849615 59127 40360 TMEM97 27346 NA PMID30185082-Compound-53 59128 40361 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651161 59129 40362 RAPGEF3 10411 ENZYME 3,8'-BIAPIGENIN CHEMBL515252 59130 40363 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RO4987655 RO-4987655 26438159 59131 40364 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME RETINOID 17001699 59133 40365 TARDBP 23435 TUMOR SUPPRESSOR PHENETHYL PHENYLCARBAMATE PHENETHYL PHENYLCARBAMATE 59135 40366 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE LAUROGUADINE LAUROGUADINE 59136 40367 MPHOSPH8 54737 NA CIPROFIBRATE CIPROFIBRATE 59137 40368 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE GSK-269962A GSK-269962A 59140 40369 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Gefitinib GEFITINIB 24533047,27468240,28089594,22789825,26936917,24410791,17463250,19692680,24165158,25964297,27196752,23980091,17085664,27793840,24353160,25573954,25870145,24736073,22263058,18981003,17349580,26561558,26124204,23344264,20942962,24874286,21422421,25948633,22997455,19147750,22323597,27312529,15737014,26206867,25931286,23542356,27612490 59141 40370 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Calcitriol CALCITRIOL 59142 40371 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ZINC 02849675 CHEMBL605959 59143 40372 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Dasatinib DASATINIB 59144 40373 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR DEFEROXAMINE DEFEROXAMINE 8794898 59145 40374 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR antagonist 178100457 59146 40375 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PAZOPANIB PAZOPANIB 24302556 59150 40376 SMTN 6525 NA TRANSFORMING GROWTH FACTOR 12390831 59151 40377 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL521851 PICTILISIB 59154 40378 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME 3,8'-BIAPIGENIN CHEMBL515252 59155 40379 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE EVEROLIMUS EVEROLIMUS 21358673,27091708 59158 40380 FAAH 2166 ENZYME, DRUGGABLE GENOME PMID26413912-Compound-84 59160 40381 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SOTRASTAURIN SOTRASTAURIN 59161 40382 METTL21A 151194 NA antidepressants 20643483,17548750 59162 40383 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME BERKELEYAMIDE B BERKELEYAMIDE B 18330993 59163 40384 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 387065609 59165 40385 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GENTIAN VIOLET GENTIAN VIOLET 59166 40386 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Aromatic bicyclic compound 5 59168 40387 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER disulfiram DISULFIRAM 59171 40388 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE DASATINIB DASATINIB 59172 40389 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PIRINIXIC ACID PIRINIXIC ACID 59174 40390 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE PD-173074 PD-173074 59175 40391 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650718 59176 40392 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME BETULINIC ACID 9810272 59177 40393 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE N/A 26945349,23894344,23041832,23817809,19755387,26220714,22616558,20560678,23904262,23226625,19915484 59178 40394 SMN2 6607 DRUGGABLE GENOME SELICICLIB SELICICLIB 59179 40395 PDF 64146 DRUGGABLE GENOME Metoprine METOPRINE 59180 40396 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL101253 VATALANIB 59181 40397 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NOBILETIN NOBILETIN 59182 40398 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME NIFEDIPINE NIFEDIPINE 14659970 59184 40399 IL12RB2 3595 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE INCELL-1001+ AD-1001 59185 40400 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER XR-9544 CHEMBL444075 26197160 59186 40401 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME 4-METHYLTHIOAMPHETAMINE 4-METHYLTHIOAMPHETAMINE 19717215 59187 40402 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BUPARLISIB HYDROCHLORIDE 59188 40403 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Pyrazolo[1,5-a]-1,3,5-triazine derivative 1 59189 40404 SDC1 6382 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME HEPARIN HEPARIN 11333985 59190 40405 CRTC2 200186 KINASE N/A 59193 40406 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME R763 59194 40407 MBNL1 4154 DRUGGABLE GENOME BETA-LAPACHONE LAPACHONE 59195 40408 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PF-3893787 PF-03893787 59196 40409 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SULFASALAZINE SULFASALAZINE 22931300 59200 40410 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MITOXANTRONE MITOXANTRONE 59201 40411 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GARCINOLIC ACID GARCINOLIC ACID 59202 40412 MCOLN1 57192 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER activator 354702256 59203 40413 F2RL3 9002 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 329968399 59204 40414 MYO9B 4650 NA CAFFEINE CAFFEINE 8495738 59205 40415 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CARFILZOMIB CARFILZOMIB 59207 40416 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL LORAZEPAM LORAZEPAM 59210 40417 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE BUPRENORPHINE BUPRENORPHINE 59211 40418 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Regorafenib REGORAFENIB 21170960,23629727,25838391,27004155 59213 40419 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR N-(3-OXODODECANOYL)HOMOSERINELACTONE CHEMBL8483 18566250 59215 40420 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL3545000 MK-2201 59216 40421 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CLEMASTINE CLEMASTINE 59217 40422 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 249565839 59218 40423 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-15 59220 40424 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE GLYX-13 RAPASTINEL 59221 40425 LINGO1 84894 DRUGGABLE GENOME inhibitor CHEMBL3544922 OPICINUMAB 59223 40426 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200694 SEVOFLURANE 59224 40427 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE metoprolol METOPROLOL 16027735 59225 40428 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 387065602 59227 40429 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX KINASE INHIBITOR 12624637 59228 40430 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 385612201 59230 40431 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR 2-ENE-VALPROATE CHEMBL117487 17566732 59231 40432 SLC29A4 222962 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 135651305 VERAPAMIL 59232 40433 FKBP5 2289 DRUGGABLE GENOME clomipramine CLOMIPRAMINE 18597649,21449676,20709156,19676097,15565110,23733030,17467808 59234 40434 NPTN 27020 CELL SURFACE, DRUGGABLE GENOME ANTISERUM 9004047 59235 40435 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200692 OLMESARTAN MEDOXOMIL 59236 40436 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME inhibitor 310264741 ENASIDENIB 59237 40437 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE DACTOLISIB DACTOLISIB 59238 40438 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TAMATINIB R-406 59239 40439 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR RAMATROBAN RAMATROBAN 59240 40440 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME TCDD 9924450 59241 40441 METTL21A 151194 NA citalopram CITALOPRAM 20643483,17548750 59243 40442 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER MELPHALAN MELPHALAN 14733945 59245 40443 ABCB5 340273 DRUGGABLE GENOME, ABC TRANSPORTER, TRANSPORTER haloperidol HALOPERIDOL 27023437,25647612 59247 40444 MAP3K10 4294 SERINE THREONINE KINASE, ENZYME, KINASE, DRUGGABLE GENOME inhibitor 249565853 CEP-1347 59249 40445 F5 2153 DRUGGABLE GENOME avatrombopag AVATROMBOPAG 59251 40446 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NORGESTIMATE NORGESTIMATE 59252 40447 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME CHEMBL2108501 LABETUZUMAB 59253 40448 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR MMV000704 CHEMBL582478 59254 40449 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME PMID27998201-Compound-15 59255 40450 CRTC1 23373 CLINICALLY ACTIONABLE INK128 SAPANISERTIB 59256 40451 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NANAOMYCIN NANAOMYCIN 59257 40452 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME ESTAZOLAM ESTAZOLAM 59258 40453 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHYLPREDNISOLONE METHYLPREDNISOLONE 59259 40454 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CGP-60474 CHEMBL300389 59260 40455 GMNN 51053 DRUGGABLE GENOME FOMOCAINE FOMOCAINE 59261 40456 XPC 7508 DNA REPAIR, CLINICALLY ACTIONABLE cisplatin CISPLATIN 19434073,21047201 59262 40457 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR allosteric modulator 404859090 59263 40458 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178103458 VORINOSTAT 59264 40459 MPHOSPH8 54737 NA THIORIDAZINE HYDROCHLORIDE THIORIDAZINE HYDROCHLORIDE 59265 40460 TAT 6898 ENZYME GLUCOCORTICOID 15531725,6127852,6113011 59268 40461 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL1980297 ILORASERTIB 59270 40462 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE RANTES 10559777 59271 40463 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-992 CHEMBL602561 59272 40464 MAP2K3 5606 KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE inhibitor SELUMETINIB SELUMETINIB 59273 40465 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL3137313 AXELOPRAN 59276 40466 CFLAR 8837 DRUG RESISTANCE, DRUGGABLE GENOME, PROTEASE NINTEDANIB NINTEDANIB 59277 40467 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE arteether 59279 40468 TGFBR2 7048 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME inhibitor 223366128 GALUNISERTIB 59280 40469 ATXN2 6311 NA N-AMINOHEXYL-5-CHLORO-1-NAPTHALENESULFONAMIDE HYDROCHLORIDE N-AMINOHEXYL-5-CHLORO-1-NAPTHALENESULFONAMIDE HYDROCHLORIDE 59281 40470 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE BDNF 12486164 59285 40471 XRCC1 7515 CLINICALLY ACTIONABLE TAXANES 17925548 59287 40472 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHABENZTHIAZURON METHABENZTHIAZURON 59288 40473 P4HB 5034 THIOREDOXIN, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE QUERCITRIN QUERCITRIN 59289 40474 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME DOVITINIB DOVITINIB 59290 40475 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SP600125 22438244 59291 40476 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor XL147 PILARALISIB 59292 40477 DPP8 54878 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 363894187 59293 40478 GDF15 9518 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR INDOLE-3-CARBINOL INDOLE-3-CARBINOL 15670751 59294 40479 TXNRD1 7296 DRUGGABLE GENOME Terpyridineplatinum(II) complexe 4 59295 40480 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651101 59296 40481 XDH 7498 DRUGGABLE GENOME, ENZYME Allopurinol ALLOPURINOL 59298 40482 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Ribociclib RIBOCICLIB 59299 40483 HNF1B 6928 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX metformin METFORMIN 59301 40484 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE METHADYL ACETATE 59302 40485 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Tricyclic compound 11 59303 40486 CXCL8 3576 DRUGGABLE GENOME TROGLITAZONE TROGLITAZONE 12364456 59304 40487 HMGCR 3156 ENZYME, DRUGGABLE GENOME Atorvastatin ATORVASTATIN 59308 40488 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE BAY1895344 59310 40489 DOT1L 84444 CLINICALLY ACTIONABLE, DNA REPAIR, METHYL TRANSFERASE, DRUGGABLE GENOME, ENZYME inhibitor 178103949 59311 40490 CP 1356 DRUGGABLE GENOME, ENZYME INTERFERON BETA 2470133 59312 40491 GSTA1 2938 ENZYME, DRUGGABLE GENOME cyclophosphamide CYCLOPHOSPHAMIDE 22188361,29938344,19448608,26222310 59313 40492 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE inhibitor CHEMBL2108702 IMETELSTAT SODIUM 59316 40493 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565901 EPACADOSTAT 59317 40494 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PF-4691502 PF-04691502 59319 40495 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE DS-6051 59320 40496 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE EPIRUBICIN HYDROCHLORIDE EPIRUBICIN HYDROCHLORIDE 59321 40497 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TCMDC-125567 CHEMBL530049 59327 40498 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROMETHAZINE PROMETHAZINE 59332 40499 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME A-77636 HCL CHEMBL1256876 59333 40500 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR TRICHOSTATIN TRICHOSTATIN 20030343,17149860 59334 40501 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 2'-HYDROXYCHALCONE 2'-HYDROXYCHALCONE 59335 40502 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL HEXOBARBITAL HEXOBARBITAL 59337 40503 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PREGNENOLONE SULFATE SODIUM PREGNENOLONE SULFATE SODIUM 59339 40504 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PIRINIXIC ACID PIRINIXIC ACID 59340 40505 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME LGX818 ENCORAFENIB 28363909,27312529,26577700 59342 40506 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor GIVINOSTAT GIVINOSTAT 59343 40507 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SL-0101 CHEMBL240954 25589938 59344 40508 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist CHEMBL38 TRETINOIN 59346 40509 ARSA 410 DRUGGABLE GENOME, ENZYME PICEATANNOL PICEATANNOL 59347 40510 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SAPPANONE A DIMETHYL ETHER SAPPANONE A DIMETHYL ETHER 59348 40511 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME SBI-087 19604259 59350 40512 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CUDC-101 CUDC-101 59352 40513 EPAS1 2034 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX NEOPETROFORMYNE A NEOPETROFORMYNE A 22928967 59353 40514 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 135650039 59355 40515 POLB 5423 DNA REPAIR, DRUGGABLE GENOME DAPHNETIN DAPHNETIN 59356 40516 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR STICTIC ACID STICTIC ACID 59357 40517 HEBP1 50865 DRUGGABLE GENOME 4-(2-cyclohexylethoxy) aniline derivative 4 59358 40518 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9340511, 6 59359 40519 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Isoflavone derivative 8 59360 40520 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE THROMBIN THROMBIN 3023371 59361 40521 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRIPHENYLSTANNYL ACETATE TRIPHENYLSTANNYL ACETATE 59362 40522 PDE4C 5143 DRUGGABLE GENOME, ENZYME DYPHYLLINE DYPHYLLINE 59364 40523 APBA1 320 NA NIFEDIPINE NIFEDIPINE 59365 40524 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Imatinib IMATINIB 28514312 59366 40525 HLA-DQA1 3117 CLINICALLY ACTIONABLE lumiracoxib LUMIRACOXIB 20639878 59371 40526 PEMT 10400 ENZYME CHEMBL2108341 SONTUZUMAB 59372 40527 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TCMDC-138263 CHEMBL535307 59373 40528 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE XL647 TESEVATINIB 18413839,19718025 59374 40529 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LABETALOL LABETALOL 22931300 59377 40530 PTGS1 5742 ENZYME, DRUGGABLE GENOME SULFASALAZINE SULFASALAZINE 59378 40531 PIGF 5281 DRUGGABLE GENOME antibody ZIV-AFLIBERCEPT AFLIBERCEPT 59380 40532 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DANAZOL DANAZOL 59382 40533 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DOXYLAMINE DOXYLAMINE 59384 40534 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Torkinib 21358673 59385 40535 PROS1 5627 DRUGGABLE GENOME ethinyl estradiol / norelgestromin 59386 40536 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER clarithromycin CLARITHROMYCIN 59388 40537 SMN1 6606 DRUGGABLE GENOME CID 695758 CHEMBL260028 59389 40538 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL DEXTROMETHORPHAN DEXTROMETHORPHAN 59390 40539 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME GNF-PF-2301 CHEMBL578061 59392 40540 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME SPIRUCHOSTATIN C SPIRUCHOSTATIN C 21967146 59394 40541 CD38 952 CELL SURFACE, DRUGGABLE GENOME antibody DARATUMUMAB DARATUMUMAB 59395 40542 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE sufentanil SUFENTANIL 22153130,31773688 59397 40543 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE FENTANYL FENTANYL 11772808 59399 40544 GMNN 51053 DRUGGABLE GENOME POMIFERIN POMIFERIN 59402 40545 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102696 59404 40546 SMN1 6606 DRUGGABLE GENOME 2-(2-NITROBENZYLSULFANYL)BENZOXAZOLE CHEMBL112060 59405 40547 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565794 59406 40548 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178101835 59408 40549 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE docetaxel DOCETAXEL 30071039 59409 40550 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE valproic acid 21806385,28763744,15761113 59410 40551 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL3545078 PF-03814735 59412 40552 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME ERYTHROPOIETIN EPOETIN BETA 9104820 59414 40553 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 318164844 59415 40554 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 329968396 CHEMBL493076 59416 40555 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE ANTIINFLAMMATORY DRUGS 12234061 59417 40556 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 315661146 PF-03882845 59418 40557 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Aminopyrimidine derivative 7 59419 40558 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CI-1040 CI-1040 59420 40559 EIF2AK4 440275 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME quetiapine QUETIAPINE 24751813 59421 40560 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL856 PRIMIDONE 59422 40561 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Aminocyclopentenone compound 3 59423 40562 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-29 59424 40563 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201561 PEGINTERFERON ALFA-2B 59425 40564 CTSD 1509 PROTEASE, DRUGGABLE GENOME, ENZYME PMID10498202C1 59426 40565 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE KD-025 CHEMBL2005186 59427 40566 CRP 1401 DRUGGABLE GENOME ISIS 353512 59428 40567 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME sildenafil SILDENAFIL 23007311 59429 40568 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AZTREONAM AZTREONAM 22931300 59432 40569 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY OXYTOCIN OXYTOCIN 12069935 59433 40570 PGF 5228 GROWTH FACTOR, DRUGGABLE GENOME Aflibercept AFLIBERCEPT 59434 40571 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME TACEDINALINE TACEDINALINE 18692397 59435 40572 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135649986 59436 40573 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417156 CHEMBL1504679 59437 40574 EPHX2 2053 DRUGGABLE GENOME, ENZYME inhibitor 348353677 59438 40575 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME 6-Phenylquinazolin-4-amine 59440 40576 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL68055 ACOLBIFENE 59441 40577 USP1 7398 DNA REPAIR, PROTEASE, ENZYME FLUORANTHEN-3-YLAMINE CHEMBL103583 59442 40578 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL406381 KRN-633 59443 40579 ATXN2 6311 NA BETA-LAPACHONE LAPACHONE 59444 40580 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CHEMBL681 ETOMIDATE 59447 40581 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLONAZEPAM CLONAZEPAM 59448 40582 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Fulvestrant FULVESTRANT 59449 40583 TDO2 6999 ENZYME, DRUGGABLE GENOME INSULIN INSULIN 2875868 59450 40584 GMNN 51053 DRUGGABLE GENOME SJ000154295 CHEMBL578502 59451 40585 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME o-desmethyl-tramadol 27082504 59452 40586 RAB9A 9367 ENZYME, DRUGGABLE GENOME PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE CHEMBL114544 59453 40587 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ZINC 03369470 CHEMBL599013 59454 40588 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE Peptide analog 55 59455 40589 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 59458 40590 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-Table1Example8 59461 40591 POLI 11201 DNA REPAIR HOMIDIUM HOMIDIUM 59462 40592 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE Tezacaftor and ivacaftor 59464 40593 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUDROCORTISONE FLUDROCORTISONE 59465 40594 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 135650359 HYDROXYFLUTAMIDE 59466 40595 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE THALIDOMIDE THALIDOMIDE 59467 40596 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 310264738 CERDULATINIB 59468 40597 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME 375973261 59470 40598 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME PYROGALLOL RED PYROGALLOL RED 59471 40599 PDE10A 10846 ENZYME, DRUGGABLE GENOME OMS824 59473 40600 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME risperidone RISPERIDONE 29955115 59474 40601 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 59475 40602 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 310264694 AMG-337 59476 40603 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 59479 40604 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PMX-53 59481 40605 CXCL8 3576 DRUGGABLE GENOME LT-BETA 9029113 59482 40606 MYH14 79784 NA Mavacamten MAVACAMTEN 59483 40607 SLC16A1 6566 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PMA 14525727 59484 40608 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR MOCETINOSTAT MOCETINOSTAT 23829483,26287310 59485 40609 ATAD5 79915 NA SJ000044511 CHEMBL592124 59487 40610 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Valspodar VALSPODAR 59488 40611 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 404859044 59489 40612 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32u 59490 40613 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 cabazitaxel CABAZITAXEL 59491 40614 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HOMIDIUM BROMIDE HOMIDIUM BROMIDE 59493 40615 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL2105667 ORVEPITANT 59494 40616 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL704 MESALAMINE 59495 40617 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CETUXIMAB CETUXIMAB 23020132,22608338,26619011,21483012,22351686,19001320,21156289,20368568,19255327,22048237,19561230,19010912,23549875,25024077,23489023,18541894,24586605,24508103,22773810,23833300,23812671,24576830,19238210,20818844,23612012,23251002,22356324,20857202,22536370,22997239,21163703,15035987,23470635,21663470,24594804,22586120,20413299,22805292,19537845,14679157,22663011,21975775,22038996,22448344,12068308,24163374,19773371,24354346,23325582,24583796,23031422,22735384,21683865,25370471,21639808,22281684,22649091,22241789,24570209,23918947,25989278,22389471,23934108,22180495,23524406,26678033,19018267,24388723,23845441,23614898,25157968,20619739,12460919,24107445,12460918,21594703,20350999,20630094,21426297,19404918,22743296,24396464,22972589,21129611,23406027 59496 40618 POLK 51426 DNA REPAIR, ENZYME TANSHINONE IIA SULFONATE TANSHINONE IIA SULFONATE 59497 40619 GART 2618 ENZYME, DRUGGABLE GENOME PELITREXOL PELITREXOL 59498 40620 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor ALISERTIB ALISERTIB 59499 40621 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CHLOROXINE CHLOROXINE 59501 40622 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER AZITHROMYCIN AZITHROMYCIN 12697643 59503 40623 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL426559 LAROPIPRANT 59504 40624 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102548 ALSTERPAULLONE 59505 40625 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIGOXIN DIGOXIN 22931300 59507 40626 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HYMECROMONE HYMECROMONE 59508 40627 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR 2-CDA CLADRIBINE 12097998 59509 40628 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME agonist CHEMBL979 MEPROBAMATE 59510 40629 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LEFLUNOMIDE LEFLUNOMIDE 59512 40630 MTAP 4507 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE DIFLUOROMETHYLORNITHINE 15534104 59515 40631 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZD5438 26881434 59518 40632 PDE4B 5142 DRUGGABLE GENOME, ENZYME ROLIPRAM ROLIPRAM 59520 40633 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE BUPIVACAINE BUPIVACAINE 15781526 59521 40634 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PHLORETIN PHLORETIN 59523 40635 POLK 51426 DNA REPAIR, ENZYME AG-538 CHEMBL56393 59525 40636 SDC1 6382 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CAR-T cells targeting CD138 59526 40637 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DIPHENIDOL DIPHENIDOL 59528 40638 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER VITAMIN E 16083877,12514119 59529 40639 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor BORTEZOMIB BORTEZOMIB 59530 40640 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor SOPHORETIN QUERCETIN 59531 40641 NECTIN4 81607 DRUGGABLE GENOME antibody AGS-22M6E ENFORTUMAB VEDOTIN 59533 40642 POLK 51426 DNA REPAIR, ENZYME KOPARIN KOPARIN 59534 40643 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178102285 LINIFANIB 59535 40644 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649787 59537 40645 ODC1 4953 DRUGGABLE GENOME, ENZYME inhibitor 178101831 59538 40646 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME L-687384 CHEMBL303336 59539 40647 ALOX15 246 ENZYME, DRUGGABLE GENOME 4-METHOXYDALBERGIONE 4-METHOXYDALBERGIONE 59540 40648 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BAY-11-7085 BAY-11-7085 59541 40649 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DILTIAZEM HYDROCHLORIDE DILTIAZEM HYDROCHLORIDE 59543 40650 KDM4A 9682 DRUGGABLE GENOME, ENZYME XANTHOANGELOL F XANTHOANGELOL F 59544 40651 EPHX2 2053 DRUGGABLE GENOME, ENZYME ALOIN ALOIN 26372074 59549 40652 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BELINOSTAT BELINOSTAT 25937017 59550 40653 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME s-adenosylmethionine ADEMETIONINE 25303295 59551 40654 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FLUPIRTINE FLUPIRTINE 59553 40655 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL2110732 DACOMITINIB 59554 40656 ARSA 410 DRUGGABLE GENOME, ENZYME INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 59557 40657 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL3707446 RIVIPANSEL 59560 40658 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 384403666 59562 40659 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE TAE-684 TAE-684 59563 40660 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CYTOKINES 15354418 59564 40661 HTT 3064 DRUGGABLE GENOME PMID28092474-Compound-32 59565 40662 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PD-0166285 PD-0166285 59566 40663 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME TRANSPLATIN TRANSPLATIN 59567 40664 LY96 23643 DRUGGABLE GENOME antagonist CHEMBL3301672 ERITORAN TETRASODIUM 59569 40665 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Igmesine IGMESINE 59570 40666 MT-RNR1 4549 KINASE amikacin AMIKACIN 18830133,16875663,9164619,19682603,16631122,21495045,16458854,12031626,16375862,9831149,17637808,22475488,11857751,27397648,9779807,7689389,20111055,9111378,27427311,17698030,11313749,20416460,16168391,24703164,9950117,21504270,11174059,8285309,18790089,15917167,20353758,16955413,16380089,14699607,17999439,14755216,17341440,19376484,15708009,25515069,15555598,11079536,17434445 59572 40667 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE OMEPRAZOLE OMEPRAZOLE 16815316 59575 40668 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Tricyclic 5-quinolone derivative 1 59576 40669 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Bevacizumab + Rituximab 59578 40670 SMN2 6607 DRUGGABLE GENOME DNDI1417597 CHEMBL1330352 59580 40671 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME VEMURAFENIB VEMURAFENIB 59582 40672 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BAICALEIN BAICALEIN 21665470 59584 40673 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR 7-azaindole derivative 5 59585 40674 TRPV2 51393 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker 135652746 59586 40675 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Apadoline APADOLINE 59587 40676 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 670282 CHEMBL260213 59588 40677 KCNJ5 3762 TRANSPORTER, ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker 223366037 59590 40678 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER METHYLENEDIOXYMETHAMPHETAMINE MIDOMAFETAMINE 59591 40679 SULT2A1 6822 DRUGGABLE GENOME acetaminophen ACETAMINOPHEN 26049587 59594 40680 TRAF1 7185 NA etanercept ETANERCEPT 23007924 59595 40681 PRMT7 54496 ENZYME, METHYL TRANSFERASE inhibitor 252166606 59596 40682 GBA 2629 DRUGGABLE GENOME, ENZYME ISOFAGOMINE AFEGOSTAT 59597 40683 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MEK INHIBITOR PD0325901 20570890 59598 40684 RACGAP1 29127 NA METHACYCLINE HYDROCHLORIDE METHACYCLINE HYDROCHLORIDE 59599 40685 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE TCMDC-125603 CHEMBL528734 59602 40686 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL FLUDIAZEPAM FLUDIAZEPAM 59603 40687 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-24047 CHEMBL1288013 59604 40688 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE Platinum compounds 19525887 59606 40689 ATAD5 79915 NA SJ000128325 CHEMBL602718 59607 40690 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565731 59609 40691 PTGES 9536 DRUGGABLE GENOME, ENZYME PMID28627961-Compound-31 59611 40692 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-20 59613 40693 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 P-1075 CHEMBL11458 59614 40694 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR MIFEPRISTONE MIFEPRISTONE 17464718 59615 40695 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565692 59616 40696 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE clopidogrel CLOPIDOGREL 21828263,20938371 59617 40697 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE IMMUNOSUPPRESSIVE 14987319 59618 40698 PDE3A 5139 ENZYME, DRUGGABLE GENOME ENOXIMONE ENOXIMONE 59621 40699 BCHE 590 DRUGGABLE GENOME, ENZYME PMID29757691-Compound-10 59623 40700 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR Ocaperidone OCAPERIDONE 59624 40701 HBB 3043 DRUGGABLE GENOME, ENZYME Iron Dextran 59627 40702 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HISTIDINE HISTIDINE 59628 40703 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201629 INSULIN PURIFIED BEEF 59629 40704 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE AMIFOSTINE AMIFOSTINE 9450496 59630 40705 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist CHEMBL1718 NALOXONE HYDROCHLORIDE 59631 40706 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ARACHIDONIC ACID ARACHIDONIC ACID 59633 40707 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Ramucirumab RAMUCIRUMAB 25185099 59634 40708 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER omeprazole OMEPRAZOLE 15976989,29377228 59635 40709 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL blocker 135652746 59636 40710 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR etidronic acid 10692979,12608943,18443790,19020788,15739035,12162507 59638 40711 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME DEXTRAN SULFATE SODIUM 11718223 59639 40712 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME LY-2624587 59642 40713 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Tihourea derivative 1 59644 40714 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-4459 CHEMBL585502 59646 40715 ATAD5 79915 NA CALCIMYCIN CALCIMYCIN 59647 40716 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GW1929 CHEMBL434063 59648 40717 MAPT 4137 DRUGGABLE GENOME HELIOMYCIN HELIOMYCIN 59649 40718 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Omacetaxine 59650 40719 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ETANERCEPT ETANERCEPT 59651 40720 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE AD01 59652 40721 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE vaccine S-3304 S-3304 59655 40722 AKR1C3 8644 ENZYME, DRUGGABLE GENOME N-(benzimidazole/indole) benzoic acid derivative 1 59657 40723 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 328083507 59658 40724 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-E1 59659 40725 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US20138552206 4 59660 40726 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE CLADRIBINE CLADRIBINE 59661 40727 GLS 2744 ENZYME GLUTAMINE GLUTAMINE 9124626,6146632,9392478,11533299,1174515,14722097 59662 40728 TMPRSS11D 9407 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166825 59663 40729 GMNN 51053 DRUGGABLE GENOME GNF-PF-2503 CHEMBL601358 59665 40730 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX FENRETINIDE FENRETINIDE 59666 40731 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BMS-908662 XL-281 59667 40732 GMNN 51053 DRUGGABLE GENOME DIGITOXIN DIGITOXIN 59668 40733 GJA1 2697 ION CHANNEL LABETALOL LABETALOL 16448880 59669 40734 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ACID BLUE 129 ACID BLUE 129 59670 40735 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Minodronate 59672 40736 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE CORTISOL HYDROCORTISONE 11948681 59673 40737 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IIK AESCULIOSIDE IIK 20371180 59675 40738 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 13-EPI-SCLOREOL CHEMBL464176 59676 40739 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 5,7,2'-TRIHYDROXYFLAVONE CHEMBL242385 59678 40740 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME VS-6063 DEFACTINIB HYDROCHLORIDE 59679 40741 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL ALPRAZOLAM ALPRAZOLAM 59681 40742 ATXN2 6311 NA PIMOZIDE PIMOZIDE 59682 40743 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3218576 COPANLISIB 59683 40744 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NSC-125034 CHEMBL239439 59684 40745 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 178101905 MARIMASTAT 59685 40746 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125435 CHEMBL525888 59686 40747 PSMA3 5684 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL2103884 OPROZOMIB 59687 40748 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200804 DICLOFENAC POTASSIUM 59688 40749 CDK18 5129 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR inhibitor CHEMBL3544942 RONICICLIB 59689 40750 MAOA 4128 DRUGGABLE GENOME, ENZYME Ladostigil LADOSTIGIL 59690 40751 EYA2 2139 DNA REPAIR NSC-645827 CHEMBL95704 59693 40752 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME PMID28460551-Compound-3 59694 40753 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1511 ESTRADIOL VALERATE 59695 40754 ALOX15 246 ENZYME, DRUGGABLE GENOME APIOL APIOL 59696 40755 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE Oxazole derivative 1 59697 40756 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PD-404182 CHEMBL595227 59699 40757 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NOREPINEPHRINE NOREPINEPHRINE 59700 40758 UBC 7316 KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US20130237529 35 59701 40759 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TAE-684 TAE-684 59702 40760 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BENZQUINAMIDE BENZQUINAMIDE 59704 40761 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SILODOSIN SILODOSIN 59706 40762 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2408045 SAPITINIB 59707 40763 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TRIFLUOPERAZINE TRIFLUOPERAZINE 59708 40764 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PYM50028 59709 40765 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-29 59710 40766 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Emibetuzumab EMIBETUZUMAB 27803065,25231402 59712 40767 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE BECAPLERMIN BECAPLERMIN 59714 40768 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Tafluposide TAFLUPOSIDE 59715 40769 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME lamotrigine LAMOTRIGINE 19668019 59717 40770 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE GEFITINIB GEFITINIB 59720 40771 TNFRSF18 8784 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME MK-4166 59721 40772 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE SKF-110679 59723 40773 CXCL8 3576 DRUGGABLE GENOME FOSCARNET FOSCARNET 10630964 59724 40774 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY PANTOPRAZOLE PANTOPRAZOLE 7865648 59725 40775 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE INDOMETHACIN INDOMETHACIN 59726 40776 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-102742 CHEMBL1519374 59728 40777 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE AMG-479 GANITUMAB 59729 40778 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME Dihydrothieno [2,3-e]indazole derivative 1 59730 40779 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GSK-269962A GSK-269962A 59731 40780 PPP1CA 5499 KINASE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE DNDI1417601 CHEMBL1503729 59734 40781 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME FPA-008 59735 40782 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FADROZOLE FADROZOLE 14720586 59736 40783 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GIVINOSTAT GIVINOSTAT 59737 40784 TGFB2 7042 GROWTH FACTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME AP12009 59738 40785 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME OLSALAZINE OLSALAZINE 59739 40786 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antagonist CHEMBL1743079 TEPROTUMUMAB 59741 40787 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DNDI1417234 CHEMBL2094549 59743 40788 TXN 7295 DRUGGABLE GENOME, THIOREDOXIN BIOTINYLATED GAMBOGIC ACID BIOTINYLATED GAMBOGIC ACID 22663155 59744 40789 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DOCETAXEL DOCETAXEL 22425996 59746 40790 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME GNF-PF-2442 CHEMBL578420 59749 40791 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyrrolo-pyridine derivative 2 59750 40792 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE etanercept ETANERCEPT 16720636,16909270,23057546,26244882,12847678,18050183,18713756,19365401,22760475,24192118,17343250,22960943,22129793,12190096,18438841 59753 40793 POLI 11201 DNA REPAIR TRANSPLATIN TRANSPLATIN 59754 40794 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RISPERIDONE RISPERIDONE 17337319 59758 40795 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2104986 TEDATIOXETINE 59759 40796 ATAD5 79915 NA ALBENDAZOLE ALBENDAZOLE 59761 40797 ABAT 18 DRUGGABLE GENOME, ENZYME inhibitor 252827498 CHEMBL378577 59764 40798 IFNG 3458 DRUGGABLE GENOME PREDNISONE PREDNISONE 10784002 59765 40799 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CINOLAZEPAM CINOLAZEPAM 59767 40800 ALDH1A1 216 DRUGGABLE GENOME, ENZYME OXITRIPTAN OXITRIPTAN 59770 40801 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING 4-(4-AMINOPHENYL)BUTANOIC ACID CHEMBL1650245 24044874 59774 40802 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME AS101 AMMONIUM TRICHLOROTELLURATE 16889755 59775 40803 KLK8 11202 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 404859023 59776 40804 CPS1 1373 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME l-methionine METHIONINE 24651765 59777 40805 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL139 DICLOFENAC 59778 40806 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE MENTHOL MENTHOL 59780 40807 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 178102082 ADAPALENE 59782 40808 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME LINIFANIB LINIFANIB 59784 40809 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545083 RGB-286638 59785 40810 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME FAT EMULSION 2065036 59787 40811 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-668394 CHEMBL336095 59788 40812 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-124356 CHEMBL22062 59789 40813 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MPI-0479605 21980130 59791 40814 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE DHEA PRASTERONE 18349113 59795 40815 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GO-6976 GO-6976 59796 40816 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 13-CIS-RETINAL CHEMBL1579130 59797 40817 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHENOXYCARB PHENOXYCARB 59798 40818 CBL 867 KINASE, ENZYME, CLINICALLY ACTIONABLE Erlotinib ERLOTINIB 25348515 59800 40819 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME LORATADINE LORATADINE 59802 40820 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Eltrombopag ELTROMBOPAG 59803 40821 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FENTICLOR FENTICLOR 59804 40822 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Imidazo[1,2-b]pyridazine derivative 6 59806 40823 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1614725 TAK-285 59807 40824 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR allosteric modulator 249565625 REFAMETINIB 59808 40825 PAK2 5062 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 310264722 59809 40826 ATAD5 79915 NA DAIDZEIN DAIDZEIN 59810 40827 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 1,2-DIPHENYLDISULFANE CHEMBL462861 59811 40828 PDE3A 5139 ENZYME, DRUGGABLE GENOME Enoximone ENOXIMONE 59813 40829 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CLOBAZAM CLOBAZAM 59815 40830 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR CYCLOHEXIMIDE CYCLOHEXIMIDE 59816 40831 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR Sunitinib SUNITINIB 22105611,26487278 59817 40832 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Platinum compounds 22188361,17409936,27995989,17401013,19203783,20530282,16707601,15213713 59818 40833 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR WITHAFERIN A WITHAFERIN A 26169123 59819 40834 GMNN 51053 DRUGGABLE GENOME METITEPINE METITEPINE 59820 40835 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CETUXIMAB CETUXIMAB 26812186,19603018,25673644,23404247,22586653,22722830,25666295,18946061,28275037,16618717,26371285,20956938,19603024,22246397,18202412,20619739,19223544,20978259,21575616,20570890 59822 40836 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR NAVELBINE NAVELBINE 15934496 59823 40837 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME TCMDC-123789 CHEMBL588859 59825 40838 IMPDH1 3614 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL866 MYCOPHENOLIC ACID 59828 40839 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL649 NADOLOL 59830 40840 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 252166890 CHEMBL1093266 59831 40841 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 hmg coa reductase inhibitors 23436703 59832 40842 ATXN2 6311 NA SJ000193360 CHEMBL607253 59833 40843 PTK6 5753 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, ENZYME ISIS-CRP 59834 40844 EIF2S1 1965 NA STAUROSPORINE STAUROSPORINE 10400313 59836 40845 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL565612 SOTRASTAURIN 59837 40846 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE EFT508 TOMIVOSERTIB 59839 40847 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME IM21 CART 59841 40848 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE modulator CHEMBL190083 TARENFLURBIL 59844 40849 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE IPRIFLAVONE IPRIFLAVONE 59845 40850 PCLAF 9768 TUMOR SUPPRESSOR Indol-3-carbinol 59847 40851 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AM-001 59849 40852 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER haloperidol HALOPERIDOL 59851 40853 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 tipranavir TIPRANAVIR 59852 40854 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-348401 CHEMBL515505 59854 40855 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200586 PRILOCAINE HYDROCHLORIDE 59855 40856 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 336446937 NAPROXCINOD 59856 40857 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SIALYL LEWIS X SIALYL LEWIS X 59857 40858 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 4'-METHOXYFLAVONE 4'-METHOXYFLAVONE 59858 40859 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ISOTHYMONIN ISOTHYMONIN 59859 40860 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENAZOPYRIDINE HYDROCHLORIDE PHENAZOPYRIDINE HYDROCHLORIDE 59860 40861 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME R-1487 R-1487 59861 40862 PSMA3 5684 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 59862 40863 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRAMUSTINE PHOSPHATE ESTRAMUSTINE PHOSPHATE 59863 40864 ALDH1A1 216 DRUGGABLE GENOME, ENZYME MEDROXYPROGESTERONE ACETATE MEDROXYPROGESTERONE ACETATE 59864 40865 HTT 3064 DRUGGABLE GENOME GNF-PF-3716 CHEMBL609606 59865 40866 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545366 VOXTALISIB 59869 40867 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME 681640 CHEMBL379975 59870 40868 GJC1 10052 ION CHANNEL inhibitor 178100972 CARBENOXOLONE 59871 40869 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROPIOMAZINE PROPIOMAZINE 59872 40870 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME elbasvir / grazoprevir 59873 40871 FAAH 2166 ENZYME, DRUGGABLE GENOME quetiapine QUETIAPINE 20631561 59874 40872 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE BENZBROMARONE BENZBROMARONE 59875 40873 HSPB1 3315 DRUGGABLE GENOME ZEARALENONE ZEARALENONE 59876 40874 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIFLUMIZOLE TRIFLUMIZOLE 59878 40875 CA9 768 DRUGGABLE GENOME, ENZYME CHEMBL1743027 GIRENTUXIMAB 59879 40876 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 59880 40877 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER EPIPODOPHYLLOTOXINS 11850258 59881 40878 PAK3 5063 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 310264722 59882 40879 GMNN 51053 DRUGGABLE GENOME DIMETHYL 2-(2-NITROBENZYLIDENE)MALONATE CHEMBL1569494 59884 40880 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL989 FLUOCINOLONE ACETONIDE 59885 40881 ALOX5AP 241 DRUGGABLE GENOME AM-803 FIBOFLAPON 59886 40882 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE S63845 27760111 59887 40883 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 METHYLDOPA METHYLDOPA 22931300 59888 40884 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Idelalisib IDELALISIB 28178345 59889 40885 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME RG-1530 RG-1530 59890 40886 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL1078178 MOMELOTINIB 59891 40887 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE AG-538 CHEMBL56393 59892 40888 RPS6KA6 27330 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME BI-D1870 CHEMBL573107 59893 40889 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR AZD6244, ARRY-142886 59895 40890 TUBB6 84617 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 59897 40891 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PANOBINOSTAT PANOBINOSTAT 24694055 59898 40892 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ALPHA,BETA-DEHYDROCURVULARIN CHEMBL482050 59901 40893 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 59905 40894 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamide derivative 26 59908 40895 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CISPLATIN CISPLATIN 12839662 59909 40896 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3039504 NINTEDANIB ESYLATE 59910 40897 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PF-562271 PF-00562271 59911 40898 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE inhibitor CHEMBL1518 PROPYLTHIOURACIL 59912 40899 TFAP2A 7020 TRANSCRIPTION FACTOR TUMOR NECROSIS FACTOR 11438643 59915 40900 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TEROXIRONE TEROXIRONE 59917 40901 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Lestaurtinib LESTAURTINIB 21926964 59918 40902 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Avastin AVASTIN 21399868 59919 40903 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENHEXAMID FENHEXAMID 59920 40904 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL491473 CEDIRANIB 59924 40905 TH 7054 ENZYME, DRUGGABLE GENOME inhibitor 178101787 METYROSINE 59925 40906 NEK4 6787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PHA-767491 CHEMBL225519 59926 40907 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALACHLOR ALACHLOR 59927 40908 KCNT2 343450 ION CHANNEL, DRUGGABLE GENOME blocker 135652729 59930 40909 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565587 CAPMATINIB 59931 40910 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DICHLOROPHEN DICHLOROPHEN 59933 40911 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TCMDC-124355 CHEMBL531401 59935 40912 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650225 59936 40913 SLC25A29 123096 TRANSPORTER, DRUGGABLE GENOME PROPIONYL-L-CARNITINE 59937 40914 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 310264701 UBLITUXIMAB 59938 40915 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000299520 CHEMBL592305 59939 40916 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102566 59940 40917 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GLAFENINE GLAFENINE 22931300 59942 40918 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR AG-1879 CHEMBL406845 59943 40919 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BYL719 ALPELISIB 27602501,24608574,27312529 59944 40920 PDE10A 10846 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545271 PBF-999 59946 40921 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL52885 ENMD-981693 59948 40922 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor TANDUTINIB TANDUTINIB 59950 40923 MPHOSPH8 54737 NA METHOTREXATE METHOTREXATE 59951 40924 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565808 59953 40925 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME SULFOBROMOPHTHALEIN SULFOBROMOPHTHALEIN 21422191 59955 40926 IDI1 3422 ENZYME inhibitor 135650699 59957 40927 KDM4A 9682 DRUGGABLE GENOME, ENZYME Selenium compound 1 59958 40928 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME ARSENIC TRIOXIDE 16283431 59959 40929 CHRNA5 1138 DRUGGABLE GENOME, ION CHANNEL cocaine COCAINE 32152934 59960 40930 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PI3K-ALPHA INHIBITOR MEN1611 21558396 59961 40931 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL3545332 CEP-2563 59963 40932 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ANTIPSYCHOTIC AGENT 8866916 59964 40933 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651192 59965 40934 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR opioids 25096645 59966 40935 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE DINOPROSTONE DINOPROSTONE 25701254 59967 40936 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Nilotinib NILOTINIB 59969 40937 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID2350207 CHEMBL259615 59970 40938 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME TRACAZOLATE TRACAZOLATE 59973 40939 IRS1 3667 KINASE, CLINICALLY ACTIONABLE epirubicin EPIRUBICIN 59975 40940 MAP3K6 9064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE inhibitor 249565813 59978 40941 IL23A 51561 DRUGGABLE GENOME CNTO-1959 GUSELKUMAB 59979 40942 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR COCAINE COCAINE 59980 40943 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME MEK162 BINIMETINIB 59981 40944 VEGFC 7424 GROWTH FACTOR, TRANSPORTER, DRUGGABLE GENOME inhibitor ENDOSTATIN (84-114)-NH2 (JKC367) 59982 40945 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE E324 E324 59983 40946 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROMAZINE PROMAZINE 59988 40947 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL3545361 ROGARATINIB 59989 40948 HBEGF 1839 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME panitumumab PANITUMUMAB 59990 40949 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR 1-hydroxyl-3,5-bis(4-hydroxylstyryl)benzene derivative 3 59991 40950 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565832 59993 40951 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Fused ring compound 1 59995 40952 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CUDC-101 CUDC-101 59996 40953 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME THIOMERSAL THIMEROSAL 59997 40954 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE TOZASERTIB TOZASERTIB 59998 40955 BRDT 676 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE PMID26924192-Compound-102 60000 40956 SFTPA1 653509 DRUGGABLE GENOME GLUCOCORTICOID 3382698,2843346 60001 40957 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR CAPTOPRIL CAPTOPRIL 9152782 60002 40958 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR OESTRADIOL ESTRADIOL 17210741 60003 40959 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MITOMYCIN C 15218314 60004 40960 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME FENOLDOPAM MESYLATE FENOLDOPAM MESYLATE 60005 40961 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR ATENOLOL ATENOLOL 15049387 60006 40962 CD37 951 DRUGGABLE GENOME TRU-016 OTLERTUZUMAB 60007 40963 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CETUXIMAB CETUXIMAB 24957073 60008 40964 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650825 PIMOZIDE 60009 40965 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL1096380 PLINABULIN 60011 40966 ZNF568 374900 NA opioids 60015 40967 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CAFFEINE CAFFEINE 7864197 60016 40968 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER anthracyclines and related substances 23441093,20938465,16331627,12684679,21900104,18408561 60017 40969 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator 178103410 DANAPAROID 60018 40970 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178103612 MOLIBRESIB 60021 40971 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Ruxolitinib RUXOLITINIB 26475333 60022 40972 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME Saracatinib SARACATINIB 27231123 60023 40973 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IRIGENOL IRIGENOL 60026 40974 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PD-0325901 PD-0325901 26272063,24339963,21325073 60027 40975 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME mexiletine MEXILETINE 60028 40976 SLPI 6590 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR HGF 10970828 60029 40977 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-59 60031 40978 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE ANTIBIOTIC ANTIBIOTIC 12724357 60033 40979 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME CARMUSTINE CARMUSTINE 60035 40980 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Prilocaine PRILOCAINE 60037 40981 TSPO 706 DRUGGABLE GENOME TEMAZEPAM TEMAZEPAM 60038 40982 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Entrectinib ENTRECTINIB 60040 40983 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE REPAGLINIDE REPAGLINIDE 60042 40984 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ALISERTIB ALISERTIB 60045 40985 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3545088 PUQUITINIB 60049 40986 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME 4SCAR19 and 4SCAR20 60051 40987 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE ATORVASTATIN ATORVASTATIN 17130267 60052 40988 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200695 PHENYLPROPANOLAMINE HYDROCHLORIDE 60053 40989 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PYRIPROXYFEN PYRIPROXYFEN 60056 40990 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE celecoxib CELECOXIB 22336956 60057 40991 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GEFITINIB GEFITINIB 60059 40992 ABCC6 368 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER docetaxel DOCETAXEL 20038957 60060 40993 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME AR-42 AR-42 60062 40994 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME FURAMIDINE FURAMIDINE 60064 40995 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CYC-116 CYC-116 60066 40996 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CHLOROTRIANISENE CHLOROTRIANISENE 60067 40997 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-A9 60068 40998 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE inhibitor HESPERADIN HESPERADIN 19035792 60069 40999 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1723 ALFUZOSIN HYDROCHLORIDE 60071 41000 APC 324 CLINICALLY ACTIONABLE FH535 18347139 60075 41001 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PIRENZEPINE HYDROCHLORIDE PIRENZEPINE HYDROCHLORIDE 60077 41002 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 178102570 60079 41003 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE inhibitor 252166829 60080 41004 TNFRSF11B 4982 DRUGGABLE GENOME HORMONES 10469275,10702390 60081 41005 MAOB 4129 DRUGGABLE GENOME, ENZYME TRANYLCYPROMINE TRANYLCYPROMINE 60082 41006 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Pembrolizumab PEMBROLIZUMAB 27225694 60083 41007 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-24 60086 41008 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME CENISERTIB CENISERTIB 60087 41009 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NSC-748118 CHEMBL2063681 22283430 60090 41010 TAC1 6863 DRUGGABLE GENOME IL-3 7691947 60091 41011 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 187051807 SCRIPTAID 60092 41012 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME BOMBESIN ANTAGONIST 1976209 60093 41013 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW682841X GW682841X 60095 41014 C1S 716 ENZYME, PROTEASE, DRUGGABLE GENOME SHP616 60096 41015 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME dolutegravir / abacavir / lamivudine 60098 41016 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 135650003 60099 41017 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Estradiol Valerate 60100 41018 PKMYT1 9088 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565863 60101 41019 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME PMID23981898C11d 60102 41020 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker 135652740 60103 41021 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PSB-1115 CHEMBL8565 60104 41022 PKN1 5585 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565836 60105 41023 GBA 2629 DRUGGABLE GENOME, ENZYME N-NONYLDEOXYNOJIRIMYCIN CHEMBL408500 60106 41024 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 60107 41025 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IIIB AESCULIOSIDE IIIB 20371180 60109 41026 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR FLUDARABINE FLUDARABINE 15059916 60110 41027 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE LY-2090314 LY-2090314 60112 41028 ATAD5 79915 NA BETA-TOXICAROL BETA-TOXICAROL 60114 41029 BAZ2B 29994 NA DNDI1417827 CHEMBL1363249 60115 41030 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RS-17053 CHEMBL88272 60116 41031 HDAC11 79885 DRUGGABLE GENOME, ENZYME BELINOSTAT BELINOSTAT 60120 41032 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY TYROSINE KINASE INHIBITOR 10781369 60121 41033 RGS4 5999 DRUGGABLE GENOME TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 60122 41034 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PMID29671355-Compound-43 60124 41035 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652337 60125 41036 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650730 NORBINALTORPHIMINE 60126 41037 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 340590249 DELGOCITINIB 60127 41038 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE THIOPROPERAZINE MESYLATE THIOPROPERAZINE MESYLATE 60128 41039 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TETRAZOLIUM RED TETRAZOLIUM RED 60131 41040 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1201013 OLSALAZINE SODIUM 60132 41041 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ODT-8 CHEMBL452157 60134 41042 PLK2 10769 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 178102294 BI-2536 60138 41043 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Tivozanib TIVOZANIB 25995436 60140 41044 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE EBSELEN EBSELEN 60142 41045 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CYCLOFENIL CYCLOFENIL 60145 41046 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME DHEA PRASTERONE 16461558 60148 41047 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CENISERTIB CENISERTIB 60149 41048 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Phenylpyridine derivative 1 60151 41049 PTGES 9536 DRUGGABLE GENOME, ENZYME Polycyclic compound 1 60152 41050 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CHLORANIL CHLORANIL 60153 41051 MDM4 4194 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, DRUGGABLE GENOME epirubicin EPIRUBICIN 24958282 60154 41052 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MEFENAMIC ACID MEFENAMIC ACID 22931300 60156 41053 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2103842 VARLITINIB 60159 41054 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE OPIOID 1410529 60161 41055 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME FOLFIRI 25605843 60162 41056 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 178102934 SAXAGLIPTIN 60164 41057 APC 324 CLINICALLY ACTIONABLE Pyrvinium PYRVINIUM 20890287 60165 41058 TUBA1C 84790 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 60166 41059 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AG-538 CHEMBL56393 60167 41060 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR YUANHUADINE YUANHUADINE 21916433 60168 41061 GMNN 51053 DRUGGABLE GENOME EBASTINE EBASTINE 60169 41062 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DEPHOSTATIN DEPHOSTATIN 60170 41063 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AZ8010 23175443,22869148 60171 41064 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ZM-336372 CHEMBL186526 60172 41065 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME etoposide ETOPOSIDE 19364970,19852077,18349289,12181437,17058217,12969965,1651156,18466101,14647407,20562211,19390945,25055799,17728214,12019197,10381366,11037804 60174 41066 SIRT5 23408 ENZYME inhibitor 252827480 60175 41067 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Pelitinib PELITINIB 16710023,16364494 60176 41068 COMT 1312 DRUGGABLE GENOME, ENZYME fentanyl FENTANYL 30281924,30549211 60177 41069 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker CHEMBL284348 DALFAMPRIDINE 60179 41070 PSMD8 5714 NA inhibitor CHEMBL325041 BORTEZOMIB 60181 41071 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor DANUSERTIB DANUSERTIB 60182 41072 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR THIETHYLPERAZINE THIETHYLPERAZINE 60184 41073 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor AUY922 60185 41074 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CIPROFLOXACIN CIPROFLOXACIN 22931300 60186 41075 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Acebutolol ACEBUTOLOL 60187 41076 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME CHEMOPREVENTIVE 10619383,16352317 60189 41077 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE IMGN-388 IMGN-388 60191 41078 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER VESNARINONE VESNARINONE 7750082 60192 41079 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651290 60194 41080 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Bevacizumab BEVACIZUMAB 23940356,26432108 60195 41081 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor BI847325 60199 41082 AQP9 366 ION CHANNEL CISPLATIN CISPLATIN 12396244 60200 41083 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PHA-665752 PHA-665752 26351320 60201 41084 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Panitumumab PANITUMUMAB 28783719,27770002,28514312,27312529,25589621 60202 41085 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE INS117548 60204 41086 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PYRROLNITRIN PYRROLNITRIN 60205 41087 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX KAMEBANIN KAMEBANIN 60206 41088 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Refametinib REFAMETINIB 26582713,27975152,25294897 60210 41089 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Vemurafenib VEMURAFENIB 26343583,21107323,24265153,26267534,27523909,22389471 60211 41090 FURIN 5045 ENZYME, PROTEASE, CELL SURFACE, DRUGGABLE GENOME US9266828, C 60213 41091 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 252827525 60215 41092 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME INSULIN GLARGINE 60216 41093 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 328083457 60217 41094 MAOB 4129 DRUGGABLE GENOME, ENZYME Rasagiline RASAGILINE 60219 41095 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-124064 CHEMBL537045 60222 41096 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650148 N6-CYCLOPENTYLADENOSINE 60225 41097 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650472 60226 41098 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE AMG 479 60227 41099 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103704 BIPERIDEN 60228 41100 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR MAP855 31227518 60229 41101 UGT2B7 7364 DRUGGABLE GENOME (R)-methadone 17178267 60230 41102 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178100961 ASPIRIN 60231 41103 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 223366080 INECALCITOL 60232 41104 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702262 ROGARATINIB 60233 41105 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650144 CYANOPINDOLOL 60235 41106 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BIFENOX BIFENOX 60236 41107 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 60237 41108 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL2105712 AFATINIB DIMALEATE 60238 41109 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651289 60239 41110 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ixabepilone IXABEPILONE 60240 41111 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Talazoparib TALAZOPARIB 60241 41112 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 252827442 SGI-1776 60242 41113 GMNN 51053 DRUGGABLE GENOME DNDI1417941 CHEMBL2095095 60243 41114 NDUFB9 4715 ENZYME inhibitor CHEMBL3545320 ME-344 60244 41115 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY GAMMA-INTERFERON 9687151 60245 41116 POLI 11201 DNA REPAIR NANAOMYCIN NANAOMYCIN 60246 41117 KLRD1 3824 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME infliximab INFLIXIMAB 26453102 60247 41118 ATAD5 79915 NA (E)-2-STYRYLCHROMONE CHEMBL388823 60249 41119 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1633 KETOTIFEN FUMARATE 60250 41120 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545424 AZD-8186 60251 41121 ATAD5 79915 NA DNDI1417083 CHEMBL1564100 60252 41122 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME busulfan BUSULFAN 24165757 60253 41123 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME RESERPINE RESERPINE 60254 41124 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR JNK INHIBITOR VIII CHEMBL210618 60255 41125 SCNN1A 6337 DRUGGABLE GENOME, ION CHANNEL P-552 60256 41126 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200483 PHENMETRAZINE HYDROCHLORIDE 60257 41127 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE oxaliplatin OXALIPLATIN 23314736 60259 41128 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-95397 CHEMBL429095 60260 41129 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DINOPROSTONE DINOPROSTONE 60261 41130 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE WHILE OLIVETOL WHILE OLIVETOL 60262 41131 SLC15A2 6565 TRANSPORTER, DRUGGABLE GENOME sorafenib SORAFENIB 60263 41132 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Human neutral insulin 60265 41133 FKBP5 2289 DRUGGABLE GENOME venlafaxine VENLAFAXINE 18597649,21449676,20709156,19676097,15565110,23733030,17467808 60267 41134 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL activator 135650001 FLINDOKALNER 60270 41135 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Flavonoid derivative 3 60271 41136 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor ENMD-2076 ENMD-2076 60275 41137 GAA 2548 DRUGGABLE GENOME, ENZYME SJ000293754 CHEMBL486706 60276 41138 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650056 CARBACYCLIN 60277 41139 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565726 60279 41140 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Pyrrolidine derivative 13 60280 41141 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME allosteric modulator 385612192 60281 41142 BAZ2B 29994 NA TYRPHOSTIN 23 TYRPHOSTIN 23 60282 41143 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1236962 OMIPALISIB 60283 41144 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565694 CHIR-99021 60284 41145 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME SNS-032 BMS-387032 60285 41146 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-124681 CHEMBL536008 60286 41147 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE RUSALATIDE RUSALATIDE 60288 41148 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME GC-1113 60289 41149 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CLORAZEPATE CLORAZEPIC ACID 60290 41150 TAC1 6863 DRUGGABLE GENOME NIZATIDINE NIZATIDINE 12495560 60291 41151 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103587 MOCETINOSTAT 60292 41152 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ETOXAZOLE ETOXAZOLE 60293 41153 PGF 5228 GROWTH FACTOR, DRUGGABLE GENOME TB-403 TB-403 60294 41154 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 1-BENZYLMALEIMIDE CHEMBL388979 60295 41155 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OXOTREMORINE OXOTREMORINE 60296 41156 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME antibody 315661192 CABIRALIZUMAB 60297 41157 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650682 NALORPHINE 60298 41158 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PIRARUBICIN PIRARUBICIN 60303 41159 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME CONGO RED CONGO RED 60305 41160 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME KOPARIN KOPARIN 60308 41161 ALOX15 246 ENZYME, DRUGGABLE GENOME IRIGINOL HEXAACEATATE IRIGINOL HEXAACEATATE 60309 41162 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BETAMETHASONE BETAMETHASONE 60310 41163 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE Lumacaftor LUMACAFTOR 60314 41164 GAA 2548 DRUGGABLE GENOME, ENZYME VU001171 CHEMBL515763 60316 41165 CAV1 857 TRANSPORTER, KINASE TESTOSTERONE TESTOSTERONE 11389065 60317 41166 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TROGLITAZONE TROGLITAZONE 60319 41167 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE PLX-3397 PEXIDARTINIB 60320 41168 MAPT 4137 DRUGGABLE GENOME HELENALIN HELENALIN 60321 41169 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE AST-487 AST-487 60322 41170 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-4522 CHEMBL585417 60323 41171 KDM4A 9682 DRUGGABLE GENOME, ENZYME ISOQUINOLINE-3-CARBOXYLIC ACID CHEMBL1728638 60324 41172 HLA-DQB1 3119 CLINICALLY ACTIONABLE flupirtine FLUPIRTINE 26959717 60325 41173 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME AG-1879 CHEMBL406845 60326 41174 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135652694 60328 41175 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PIPERIDOLATE PIPERIDOLATE 60330 41176 GMNN 51053 DRUGGABLE GENOME GNF-PF-2947 CHEMBL581677 60331 41177 PSMA4 5685 DRUGGABLE GENOME, PROTEASE BORTEZOMIB BORTEZOMIB 24524217 60332 41178 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME D,L-ARMEPAVINE CHEMBL451722 60333 41179 AOX1 316 DRUGGABLE GENOME XK469 60334 41180 PTGS2 5743 DRUGGABLE GENOME, ENZYME aspirin ASPIRIN 60335 41181 GSTA1 2938 ENZYME, DRUGGABLE GENOME busulfan BUSULFAN 24192117 60336 41182 ACTB 60 TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 12167460 60337 41183 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR DAPHNORIN DAPHNORIN 60338 41184 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DOV 216,303 60339 41185 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SB-220025 SB-220025 60340 41186 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME AG-528 CHEMBL56542 60342 41187 MAPT 4137 DRUGGABLE GENOME METHYLDOPA (RACEMIC) METHYLDOPA (RACEMIC) 60343 41188 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SARCOLYSIN SARCOLYSIN 60344 41189 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME zoledronate ZOLEDRONIC ACID 18594024 60345 41190 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HALCINONIDE HALCINONIDE 60346 41191 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE TRICHLORMETHIAZIDE TRICHLORMETHIAZIDE 60347 41192 KDM4A 9682 DRUGGABLE GENOME, ENZYME N'-(2,4-DIHYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE CHEMBL199592 60350 41193 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CHALCONE CHALCONE 60351 41194 TPP2 7174 ENZYME, PROTEASE inhibitor 252166782 60352 41195 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW679410X GW679410X 60354 41196 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY RETINOL RETINOL 11563543 60356 41197 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME inhibitor 135652074 60357 41198 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 328083469 60359 41199 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Indoline derivative 13 60360 41200 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Oxytocin OXYTOCIN 60362 41201 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1356607 NOREPINEPHRINE BITARTRATE 60363 41202 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GNF-PF-3889 CHEMBL598270 60364 41203 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PAPAVERINE HYDROCHLORIDE PAPAVERINE HYDROCHLORIDE 60366 41204 GART 2618 ENZYME, DRUGGABLE GENOME LY309887 60367 41205 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME ISOSILYBIN A ISOSILYBIN A 23401473 60368 41206 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GW441756X GW441756X 60370 41207 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE HEPARAN SULFATE 8043862 60372 41208 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PLX-3397 PEXIDARTINIB 60374 41209 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME GNF-PF-992 CHEMBL602561 60375 41210 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-35 60376 41211 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL antiepileptics 23859570,22591328,22292851,25155934,21561445 60378 41212 AREG 374 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE PANITUMUMAB PANITUMUMAB 26867820 60379 41213 TUBA4A 7277 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 60383 41214 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE S(+)-ISOPROTERENOL-BITARTRATE CHEMBL1257092 60384 41215 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 178101751 60385 41216 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE E7449 2X-121 26513298 60387 41217 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Piperidinyl triazole derivative 4 60388 41218 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CABOZANTINIB CABOZANTINIB 60389 41219 POLK 51426 DNA REPAIR, ENZYME CROCIN CROCIN 60391 41220 BAZ2B 29994 NA TCMDC-125544 CHEMBL533602 60393 41221 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL688 FENTANYL CITRATE 60394 41222 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Gemcitabine GEMCITABINE 28750271 60397 41223 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor 178101947 RUBOXISTAURIN 60398 41224 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103526 60399 41225 HSPA4 3308 NA AG-858 21898241 60400 41226 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME DS-3078 60401 41227 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Gefitinib GEFITINIB 26936917 60402 41228 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Pembrolizumab PEMBROLIZUMAB 28514312 60404 41229 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE PROPOXYPHENE PROPOXYPHENE 60406 41230 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor BAY80-6946 COPANLISIB 60407 41231 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME AMG520 60408 41232 HTT 3064 DRUGGABLE GENOME 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 60409 41233 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-145669 CHEMBL191611 60411 41234 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME SB-431542 SB-431542 60412 41235 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 53801049 60413 41236 ITPA 3704 ENZYME interferon alfa-2b, recombinant 21503919 60414 41237 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ALPRENOLOL ALPRENOLOL 2903243 60415 41238 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR BMS-833923 BMS-833923 60416 41239 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DNDI1417147 CHEMBL2094484 60417 41240 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME fluoxetine / olanzapine 60419 41241 GAA 2548 DRUGGABLE GENOME, ENZYME CAFFEIC ACID CAFFEIC ACID 60421 41242 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Aripiprazole Lauroxil 60424 41243 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MUC1-TARGETED PEPTIDE GO-203-2C 25245423 60425 41244 MUCL3 135656 NA gemcitabine GEMCITABINE 31616045 60426 41245 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE ABBV-2737 60427 41246 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-32 60428 41247 ATAD5 79915 NA HYDRALAZINE HYDRALAZINE 60430 41248 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER EMD 1214063 26358474 60431 41249 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Dexamethasone palmitate 60433 41250 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID25726713-Compound-49 60434 41251 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR TRIAZOLAM TRIAZOLAM 22137933 60435 41252 TDO2 6999 ENZYME, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 6 60436 41253 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME NSC-139257 CHEMBL1256364 60437 41254 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME TEMAZEPAM TEMAZEPAM 60438 41255 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178103147 60442 41256 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GMI-1271 UPROLESELAN 60443 41257 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME S3I-201 23242808 60444 41258 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME AL3818 ANLOTINIB 60445 41259 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650230 ENADOLINE 60449 41260 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 178102342 FEDRATINIB 60450 41261 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-107 CHEMBL578675 60452 41262 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102411 60453 41263 KCND3 3752 ION CHANNEL, DRUGGABLE GENOME Sodium bicarbonate 60454 41264 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR SANGUINARINE SULFATE SANGUINARINE SULFATE 60455 41265 RAC1 5879 CLINICALLY ACTIONABLE, KINASE, DRUG RESISTANCE DABRAFENIB DABRAFENIB 25056119,24265153 60457 41266 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-48300 CHEMBL1091971 60458 41267 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL27759 ENTINOSTAT 60459 41268 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor SORAFENIB TOSYLATE 60461 41269 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME GDC-0941 PICTILISIB 24251790 60463 41270 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 387065610 60468 41271 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE PMED-1 24819961 60470 41272 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CARBIMAZOLE CARBIMAZOLE 22931300 60471 41273 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME RO5126766 26438159 60472 41274 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE AZD4547 26351320,27595477,27550940,27401245,26936917,27179038,25169980,26294741,22869148 60473 41275 PTPRS 5802 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE, CLINICALLY ACTIONABLE inhibitor 381118819 60474 41276 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AZD9291 OSIMERTINIB 27694386,27102076,24410791,24893891,27959700,25923549,25870145,26286086,25948633,27393507,27252416,25939061,26206867,27216193,28343545,27435396 60476 41277 CDA 978 ENZYME, DRUGGABLE GENOME difluorodeoxyuridine 22838949 60477 41278 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE QUINALIZARIN QUINALIZARIN 60478 41279 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME DONEPEZIL DONEPEZIL 25282266 60479 41280 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DICHLOROPHEN DICHLOROPHEN 60481 41281 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CVBT-141H 60483 41282 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Dexchlorpheniramine Maleate 60484 41283 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-57 60485 41284 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 5-8 60488 41285 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME TAE-684 TAE-684 60489 41286 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Eprosartan EPROSARTAN 60490 41287 GMNN 51053 DRUGGABLE GENOME VINBURNINE VINBURNINE 60493 41288 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1241153 IBUPROFEN SODIUM 60494 41289 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 135652592 60496 41290 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 381118799 60498 41291 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME TNF-ALPHA 18490773 60500 41292 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CONGO RED CONGO RED 60501 41293 POLK 51426 DNA REPAIR, ENZYME 3-METHOXYCATECHOL 3-METHOXYCATECHOL 60502 41294 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME pravastatin PRAVASTATIN 19842935 60503 41295 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody IPILIMUMAB IPILIMUMAB 60504 41296 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE Semapimod SEMAPIMOD 60505 41297 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 340590249 DELGOCITINIB 60506 41298 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL2105728 CRENOLANIB 60507 41299 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 KARANJIN KARANJIN 60508 41300 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PENTAZOCINE PENTAZOCINE 60511 41301 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650855 PROMEGESTONE 60512 41302 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE ARQ 092 60513 41303 GPA33 10223 DRUGGABLE GENOME Radiolabelled-huA33 60514 41304 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR selective beta-2-adrenoreceptor agonists 15282200 60517 41305 ABCC5 10057 DRUGGABLE GENOME, ABC TRANSPORTER, TRANSPORTER leucovorin LEUCOVORIN 26352872 60521 41306 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME tetanus antitoxin 27749688 60522 41307 TSPO 706 DRUGGABLE GENOME Imidazopyridine acetamide analog 5 60523 41308 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE NeuVax 60524 41309 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme7WO2012/098070bottom 60525 41310 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR MITOXANTRONE MITOXANTRONE 60526 41311 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 60528 41312 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MERCURIC CHLORIDE MERCURIC CHLORIDE 60529 41313 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417215 CHEMBL1390650 60530 41314 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME TRIAZOLAM TRIAZOLAM 60531 41315 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE STREPTOZOTOCIN STREPTOZOCIN 10837808 60532 41316 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2109379 NI-0801 60533 41317 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker CHEMBL113461 TEDISAMIL 60535 41318 ENPP3 5169 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AGS-16C3F 60537 41319 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 1,5-ISOQUINOLINEDIOL CHEMBL338314 60538 41320 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CLOZAPINE CLOZAPINE 22931300 60539 41321 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor ROMIDEPSIN ROMIDEPSIN 60541 41322 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME ETHANOL ALCOHOL 16750178 60542 41323 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME flucloxacillin FLOXACILLIN 30664875 60543 41324 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1095 ETHOTOIN 60544 41325 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 187051808 ISCHEMIN 60546 41326 APC 324 CLINICALLY ACTIONABLE NSAID 9934849 60548 41327 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 atazanavir ATAZANAVIR 22394315 60550 41328 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME METHYLERGONOVINE MALEATE METHYLERGONOVINE MALEATE 60551 41329 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE US9156852, 83 60553 41330 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702261 60554 41331 MTRR 4552 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME methotrexate METHOTREXATE 16013960,29743634,15797993,18368069 60555 41332 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ANTIDEPRESSANTS 9574817 60556 41333 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIELDRIN DIELDRIN 60557 41334 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MOMETASONE FUROATE MOMETASONE FUROATE 60558 41335 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NALMEFENE NALMEFENE 60559 41336 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE celecoxib CELECOXIB 18695978 60560 41337 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME thioguanosine monophosphate 26332308 60562 41338 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor MK0752 60565 41339 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Oxindole derivative 2 60566 41340 MAPT 4137 DRUGGABLE GENOME STICTIC ACID STICTIC ACID 60567 41341 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME Drugs For Treatment Of Tuberculosis 22162992 60568 41342 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE SORAFENIB SORAFENIB 60569 41343 GBA 2629 DRUGGABLE GENOME, ENZYME RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 60571 41344 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-254 CHEMBL461579 60572 41345 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR YANGONIN YANGONIN 60574 41346 TLR7 51284 DRUGGABLE GENOME AZD-8848 AZD-8848 60575 41347 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE Y-27632 Y-27632 22257127 60576 41348 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE SP-600125 SP-600125 60577 41349 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE NORDIHYDROGUAIARETIC ACID 15379894 60578 41350 DPEP1 1800 PROTEASE, DRUGGABLE GENOME, ENZYME DEXAMETHASONE DEXAMETHASONE 9806799 60579 41351 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Ixabepilone IXABEPILONE 60580 41352 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE AZD6738 CERALASERTIB 60581 41353 CDH1 999 CLINICALLY ACTIONABLE, DRUGGABLE GENOME PROTEOLYTIC ENZYMES 2211831 60582 41354 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1118 DESVENLAFAXINE 60583 41355 KDM4A 9682 DRUGGABLE GENOME, ENZYME N',N'-DIMETHYLARGININE HCL CHEMBL1255836 60585 41356 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE blocker CHEMBL3545040 AZD7009 60586 41357 MAP3K1 4214 CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME carboplatin CARBOPLATIN 21636554 60590 41358 ATAD5 79915 NA DIMETHYL 2-(2-NITROBENZYLIDENE)MALONATE CHEMBL1569494 60591 41359 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE XL418 XL-418 19644473 60592 41360 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ASTEMIZOLE ASTEMIZOLE 60593 41361 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SB-202190 SB-202190 60594 41362 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE OESTRADIOL ESTRADIOL 9662256 60595 41363 FNTA 2339 ENZYME, DRUGGABLE GENOME GGTI-2418 60596 41364 CDK13 8621 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL445813 AT-7519 60597 41365 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Elapegademase ELAPEGADEMASE 60598 41366 MMP14 4323 PROTEASE, DRUGGABLE GENOME, ENZYME Epigallocatechin gallate 60601 41367 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ATG 9389690 60602 41368 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME BEVASIRANIB BEVASIRANIB 60603 41369 ATAD5 79915 NA N6-METHYLADENOSINE CHEMBL383144 60604 41370 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor 223366206 INFIGRATINIB 60605 41371 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME MYCOPHENOLIC ACID 15571295 60607 41372 GUCY2C 2984 DRUGGABLE GENOME, KINASE Linaclotide LINACLOTIDE 60608 41373 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 385612220 60612 41374 SLC2A2 6514 TRANSPORTER, DRUGGABLE GENOME metformin METFORMIN 60614 41375 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BAY1125976 27699769 60615 41376 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator CHEMBL1201513 HEPARIN CALCIUM 60616 41377 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME Meprobamate MEPROBAMATE 23197040 60617 41378 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor 340590240 60618 41379 PTGS2 5743 DRUGGABLE GENOME, ENZYME Etoricoxib ETORICOXIB 60620 41380 PTGS1 5742 ENZYME, DRUGGABLE GENOME NAPROXEN ETEMESIL 60621 41381 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NANAOMYCIN NANAOMYCIN 60623 41382 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 COUMAPHOS COUMAPHOS 60624 41383 PRKG1 5592 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME GW843682X GW843682X 60625 41384 CYBB 1536 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME, ENZYME inhibitor 363894225 60626 41385 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME Citarinostat CITARINOSTAT 60627 41386 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 mifepristone MIFEPRISTONE 9187528 60628 41387 FES 2242 ENZYME, DRUGGABLE GENOME, KINASE, TYROSINE KINASE LINIFANIB LINIFANIB 60629 41388 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Deguelin DEGUELIN 24978597,20811676 60632 41389 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME Pyridic ketone derivative 1 60633 41390 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Trametinib TRAMETINIB 27222538 60634 41391 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Indacaterol INDACATEROL 60635 41392 CBR3 874 ENZYME, DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, CLINICALLY ACTIONABLE epirubicin EPIRUBICIN 60636 41393 CPN1 1369 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252166875 60640 41394 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE T-DM1 T-DM1 27052654 60641 41395 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME DOVITINIB DOVITINIB 60642 41396 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1512 FLUNISOLIDE 60643 41397 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME CART-10 cells 60644 41398 GLS 2744 ENZYME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 60645 41399 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL520733 SEMAGACESTAT 60646 41400 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PX-866 SONOLISIB 18493606 60648 41401 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE SELICICLIB SELICICLIB 21080703 60649 41402 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR JQ1 25759019 60650 41403 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME CYC-116 CYC-116 60652 41404 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 315661273 ATICAPRANT 60653 41405 ALOX15B 247 DRUGGABLE GENOME, ENZYME CARBONYL CYANIDE P-TRIFLUOROMETHOXYPHENYL HYDRAZONE CHEMBL457504 60655 41406 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ALPHA-ADRENERGIC AGONIST 9601075 60656 41407 PSMB6 5694 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 60658 41408 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MN-201 1.ALPHA.-HYDROXYVITAMIN D5 60659 41409 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135649823 60660 41410 PSMC5 5705 TRANSCRIPTION FACTOR BINDING, PROTEASE inhibitor CHEMBL451887 CARFILZOMIB 60661 41411 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist CHEMBL1265 ADAPALENE 60662 41412 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME BETRIXABAN BETRIXABAN 60665 41413 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE ENMD-2076 ENMD-2076 60666 41414 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR IDARUBICIN IDARUBICIN 60667 41415 GMNN 51053 DRUGGABLE GENOME TCMDC-124377 CHEMBL531269 60668 41416 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650609 MILAMELINE 60669 41417 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 249565910 60670 41418 MAPT 4137 DRUGGABLE GENOME TCMDC-125575 CHEMBL587620 60672 41419 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor PCI-24781 ABEXINOSTAT 60674 41420 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200733 DESFLURANE 60675 41421 KDM4A 9682 DRUGGABLE GENOME, ENZYME SUFENTANIL CITRATE SUFENTANIL CITRATE 60676 41422 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PROPIONYLPROMAZINE HYDROCHLORIDE PROPIONYLPROMAZINE HYDROCHLORIDE 60679 41423 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL284348 DALFAMPRIDINE 60680 41424 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DEGUELIN DEGUELIN 60681 41425 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Antibodie derivative 4 60684 41426 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE PEMBROLIZUMAB PEMBROLIZUMAB 29773717 60686 41427 TOP2B 7155 DRUGGABLE GENOME, ENZYME Tirapazamine TIRAPAZAMINE 60687 41428 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING ARSENIC TRIOXIDE 60688 41429 SLC44A1 23446 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101222 HEMICHOLINIUM-3 60689 41430 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME NSC-95397 CHEMBL429095 60690 41431 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FP-1039 FP-1039 60691 41432 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GW501516 GW501516 20403648,23566516 60694 41433 BAZ2B 29994 NA TANNIC ACID TANNIC ACID 60695 41434 CLCN3 1182 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE, TRANSPORTER DESACETYLBUFOTALIN DESACETYLBUFOTALIN 23799775 60696 41435 NUCB1 4924 DRUGGABLE GENOME antagonist 252166718 60697 41436 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE KETANSERIN TARTRATE KETANSERIN TARTRATE 60698 41437 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PIPERONAL PIPERONAL 60699 41438 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE INSULIN INSULIN 16125526,9287059 60700 41439 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIHYDREXIDINE HYDROCHLORIDE DIHYDREXIDINE HYDROCHLORIDE 60701 41440 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE ATEZOLIZUMAB ATEZOLIZUMAB 26970723,26918451,28472902 60703 41441 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME Cibinetide CIBINETIDE 60709 41442 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SANGUINARINE SULFATE SANGUINARINE SULFATE 60710 41443 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TERBUTALINE SULFATE TERBUTALINE SULFATE 60711 41444 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BENZIODARONE BENZIODARONE 60712 41445 CDKN2D 1032 KINASE DEPSIPEPTIDE ROMIDEPSIN 11753657 60713 41446 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178101563 60714 41447 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL526 PROPOFOL 60715 41448 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ALOSETRON HYDROCHLORIDE ALOSETRON HYDROCHLORIDE 60716 41449 ESRRG 2104 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 310264689 CHEMBL201013 60722 41450 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PRALIDOXIME PRALIDOXIME 22206546,21438612 60725 41451 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 3 60726 41452 KDM4A 9682 DRUGGABLE GENOME, ENZYME AMBUNOL AMBUNOL 60728 41453 TUBB 203068 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 60729 41454 TUBB3 10381 DRUGGABLE GENOME inhibitor 252827511 60733 41455 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MERCAPTOPURINE MERCAPTOPURINE 60735 41456 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME SU5402 15516981 60741 41457 DHFR 1719 DRUGGABLE GENOME, ENZYME Trimethoprim TRIMETHOPRIM 60742 41458 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ACLARUBICIN HYDROCHLORIDE ACLARUBICIN HYDROCHLORIDE 60743 41459 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GR-127935 GR-127935 60744 41460 VAMP2 6844 DRUGGABLE GENOME inhibitor CHEMBL1201569 BOTULINUM TOXIN TYPE B 60745 41461 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME GOSERELIN ACETATE 15338676 60746 41462 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RUBITECAN RUBITECAN 60747 41463 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL IBUTILIDE IBUTILIDE 60748 41464 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor DACOMITINIB DACOMITINIB 60750 41465 NCOA3 8202 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, ENZYME ETOPOSIDE ETOPOSIDE 60751 41466 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 21 60754 41467 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist 178100905 60755 41468 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE TIRATRICOL TIRATRICOL 60756 41469 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR IODINE IODINE 60757 41470 BCHE 590 DRUGGABLE GENOME, ENZYME Oxime derivative 1 60758 41471 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 1225609 CHEMBL444376 60759 41472 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME rucaparib RUCAPARIB 60760 41473 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-19 60761 41474 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3545426 CC-115 60763 41475 ALOX15 246 ENZYME, DRUGGABLE GENOME Tri-substituted benzene derivative 1 60764 41476 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PHYSOSTIGMINE PHYSOSTIGMINE 60765 41477 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ZAPRINAST ZAPRINAST 60766 41478 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SBI-755199 26603897 60767 41479 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME haloperidol HALOPERIDOL 27023437,20031235 60768 41480 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102273 60769 41481 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-645827 CHEMBL95704 60770 41482 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME TRETINOIN TRETINOIN 60771 41483 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HYDROXYUREA HYDROXYUREA 17180388 60772 41484 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist 336446923 ATRACURIUM 60773 41485 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DINACICLIB DINACICLIB 23600925 60774 41486 BAZ2A 11176 ENZYME inhibitor 249565913 60775 41487 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PAZOPANIB PAZOPANIB 60776 41488 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NISOLDIPINE NISOLDIPINE 22931300 60777 41489 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist,allosteric modulator 315661106 60779 41490 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178100990 60781 41491 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR GNF-PF-4864 CHEMBL583558 60782 41492 ATXN2 6311 NA METHIOTHEPIN MESYLATE METHIOTHEPIN MESYLATE 60783 41493 MAPT 4137 DRUGGABLE GENOME NSC-98938 CHEMBL1939691 60785 41494 PRKAG1 5571 ENZYME, KINASE metformin METFORMIN 22722338 60786 41495 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IIIF AESCULIOSIDE IIIF 20371180 60787 41496 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CLOZAPINE CLOZAPINE 60788 41497 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Progesterone PROGESTERONE 60789 41498 GAA 2548 DRUGGABLE GENOME, ENZYME NSC-107022 CHEMBL1601846 60790 41499 ATXN2 6311 NA CLOROTEPINE CLOROTEPINE 60791 41500 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Antiinflammatory agents, non-steroids 10200020 60792 41501 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME KURARINONE KURARINONE 18565755 60793 41502 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FUDOSTEINE FUDOSTEINE 60794 41503 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FINASTERIDE FINASTERIDE 22931300 60796 41504 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL3707266 RIBOCICLIB SUCCINATE 60798 41505 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor ICOTINIB ICOTINIB 60799 41506 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE MANASSANTIN B MANASSANTIN B 15165135 60801 41507 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE TCMDC-124245 CHEMBL587615 23414799 60802 41508 TDO2 6999 ENZYME, DRUGGABLE GENOME inhibitor 315661104 NAVOXIMOD 60804 41509 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-71033 CHEMBL116548 60805 41510 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL428647 PACLITAXEL 60806 41511 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME peginterferon alfa-2b 60808 41512 POLK 51426 DNA REPAIR, ENZYME CADMIUM ACETATE CADMIUM ACETATE 60812 41513 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 249565774 60814 41514 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR RIMEXOLONE RIMEXOLONE 60815 41515 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor ENTINOSTAT ENTINOSTAT 60816 41516 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-2272 CHEMBL601757 60817 41517 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Tricyclic compound 3 60818 41518 LCAT 3931 ENZYME, TRANSPORTER, DRUGGABLE GENOME TESTOSTERONE PROPIONATE 3766045 60819 41519 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CISPLATIN CISPLATIN 11062746 60821 41520 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103584 60823 41521 ATXN2 6311 NA DNDI1417548 CHEMBL2094789 60824 41522 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1421 DASATINIB 60826 41523 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 354702214 60827 41524 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE NB-1011 60828 41525 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME TACROLIMUS TACROLIMUS 17031644 60829 41526 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR A-395 28135237 60831 41527 STX4 6810 CELL SURFACE warfarin WARFARIN 60832 41528 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BITERTANOL BITERTANOL 60833 41529 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE XL820 60835 41530 SLC38A4 55089 TRANSPORTER 178101353 60836 41531 PNP 4860 ENZYME, DRUGGABLE GENOME inhibitor 252166484 FORODESINE 60837 41532 PTGS2 5743 DRUGGABLE GENOME, ENZYME SALSALATE SALSALATE 60838 41533 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651192 60839 41534 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201562 INTERFERON BETA-1A 60840 41535 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 310264739 LIFIRAFENIB 60841 41536 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL BIIB074 VIXOTRIGINE 60843 41537 EIF4E 1977 DRUGGABLE GENOME HYDROXYUREA HYDROXYUREA 10585489 60846 41538 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 60847 41539 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL2110725 VINFLUNINE 60848 41540 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE DOVITINIB DOVITINIB 60853 41541 BMPR2 659 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, CELL SURFACE inhibitor 385612192 60854 41542 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID25656651-Compound-33a 60856 41543 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR IL-1 11429163 60858 41544 MAP2K6 5608 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE, TUMOR SUPPRESSOR inhibitor MEK162 BINIMETINIB 60860 41545 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 (-)-USNIC ACID (-)-USNIC ACID 60861 41546 NDUFAF2 91942 ENZYME inhibitor CHEMBL3545135 NV-128 60862 41547 MAPT 4137 DRUGGABLE GENOME GETIACAULEIN GETIACAULEIN 60866 41548 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME THROMBIN THROMBIN 60868 41549 PTGS2 5743 DRUGGABLE GENOME, ENZYME NABUMETONE NABUMETONE 60873 41550 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME FLURAZEPAM FLURAZEPAM 60874 41551 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BERGAMOTTIN BERGAMOTTIN 60875 41552 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-747264 CHEMBL593110 60877 41553 PGK1 5230 ENZYME, KINASE lamivudine LAMIVUDINE 60880 41554 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178101606 DORSOMORPHIN 60882 41555 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SUPROFEN METHYL ESTER SUPROFEN METHYL ESTER 60883 41556 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649961 60885 41557 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200904 SELEGILINE HYDROCHLORIDE 60886 41558 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 1,3-DIBENZYLTHIOUREA CHEMBL1388908 60888 41559 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ICRF-193 ICRF-193 60889 41560 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102268 60890 41561 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Letrozole LETROZOLE 19786658 60891 41562 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR THIOGUANINE THIOGUANINE 60892 41563 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270010-Compound-Figure24-a 60893 41564 ATAD5 79915 NA FLUNARIZINE FLUNARIZINE 60894 41565 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 E7389 ERIBULIN MESYLATE 18431572 60896 41566 VIM 7431 DRUGGABLE GENOME IL-2 ALDESLEUKIN 7691937 60897 41567 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IL-6 10023678 60898 41568 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE VX-765 BELNACASAN 60901 41569 ORAI1 84876 TRANSCRIPTION FACTOR, ION CHANNEL, TRANSPORTER blocker 375973230 60902 41570 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 5-NITROQUINOLINE CHEMBL164449 60904 41571 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER sevoflurane SEVOFLURANE 60905 41572 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME CENISERTIB CENISERTIB 60907 41573 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565876 60908 41574 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DYDROGESTERONE DYDROGESTERONE 60909 41575 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HOMIDIUM BROMIDE HOMIDIUM BROMIDE 60911 41576 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BETA-BLOCKER 15592325 60913 41577 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor ALVOCIDIB ALVOCIDIB 60914 41578 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GARDENIN B GARDENIN B 60915 41579 PDE10A 10846 ENZYME, DRUGGABLE GENOME inhibitor 340590247 MARDEPODECT 60916 41580 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL12 DIAZEPAM 60917 41581 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME SB-220025 SB-220025 60918 41582 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIPHENYLENEIODONIUM DIPHENYLENEIODONIUM 60919 41583 BRCA2 675 CLINICALLY ACTIONABLE E7449 2X-121 60920 41584 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE 4-(4-ETHOXYPHENOXY)PHENOL CHEMBL455078 18952425 60926 41585 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME DICHLOROACETIC ACID DICHLOROACETIC ACID 25383915 60927 41586 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TCMDC-124544 CHEMBL531322 60928 41587 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102277 60929 41588 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME DOVITINIB DOVITINIB 60930 41589 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2105719 DACOMITINIB 60931 41590 ATAD5 79915 NA 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 60932 41591 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME KAI-1678 KAI-1678 60935 41592 BMP7 655 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR prednisone PREDNISONE 26590194 60937 41593 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE PHENTOLAMINE PHENTOLAMINE 2866100 60938 41594 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE ALENDRONATE ALENDRONIC ACID 60940 41595 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE IL-3 9312020 60942 41596 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1201729 DRONEDARONE HYDROCHLORIDE 60944 41597 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL2105107 INECALCITOL 60945 41598 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE AVELUMAB AVELUMAB 26918451,28472902 60946 41599 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE (20S,21R)-FLUOROCAMPTOTHECIN (20S,21R)-FLUOROCAMPTOTHECIN 24069881 60948 41600 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HALOFANTRINE HYDROCHLORIDE HALOFANTRINE HYDROCHLORIDE 60950 41601 GUCY1A1 2982 ENZYME, DRUGGABLE GENOME activator CHEMBL1311 ISOSORBIDE MONONITRATE 60952 41602 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CEPHALOTHIN CEPHALOTHIN 60953 41603 PDE3A 5139 ENZYME, DRUGGABLE GENOME Cilostazol CILOSTAZOL 60954 41604 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker 135652715 SAXITOXIN 60955 41605 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR DEMETHYLWEDELOLACTONE DEMETHYLWEDELOLACTONE 22926226 60956 41606 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME indinavir INDINAVIR 10353933,7565971,17627617,9630669,17058217,10591539,16809730,16170755,11156391,20562211,20335017,19390945,15297419,17728214,16609363,16118329,9784835,19299905,12181419,20504240,15709193,15007088,16456808,16969497,22050734 60958 41607 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME INCB18424 60959 41608 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651541 EPOPROSTENOL 60960 41609 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Alkynyl-substituted pyrimidinyl-pyrrole derivative 1 60961 41610 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR FASUDIL FASUDIL 60962 41611 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RITONAVIR RITONAVIR 9278209 60965 41612 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 5310801 CHEMBL260451 60968 41613 KDM4A 9682 DRUGGABLE GENOME, ENZYME PROCHLORPERAZINE EDISYLATE PROCHLORPERAZINE EDISYLATE 60969 41614 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist CHEMBL464 ETRETINATE 60971 41615 FAAH 2166 ENZYME, DRUGGABLE GENOME N-alkyl-4-oxazolecar boxamide derivative 1 60972 41616 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME XR-9577 CHEMBL428402 18678495 60973 41617 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650214 DYDROGESTERONE 60975 41618 ITGA2 3673 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist CHEMBL1743086 VATELIZUMAB 60976 41619 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DNQX DNQX 60978 41620 ATAD5 79915 NA COLCHICINE COLCHICINE 60979 41621 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Pimasertib PIMASERTIB 26228206 60982 41622 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE COLCHICINE COLCHICINE 7543498,1363595 60983 41623 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME PALBOCICLIB PALBOCICLIB 60984 41624 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE CEQ-508 21744502 60985 41625 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE ILORASERTIB ILORASERTIB 60986 41626 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 60987 41627 SI 6476 DRUGGABLE GENOME, ENZYME ACARBOSE ACARBOSE 60990 41628 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-57 60991 41629 MYD88 4615 CLINICALLY ACTIONABLE N/A 25055137,22944768,26230596,24903481,26792260 60992 41630 BAZ2B 29994 NA SJ000027778 CHEMBL592588 60993 41631 LCAT 3931 ENZYME, TRANSPORTER, DRUGGABLE GENOME TESTOSTERONE TESTOSTERONE 3383436 60994 41632 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Pyrrolo-pyrrolone derivative 4 60995 41633 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE sulfasalazine SULFASALAZINE 18322994 60999 41634 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 5-(4-PHENYLBUTOXY)PSORALEN CHEMBL1256851 61002 41635 MAPT 4137 DRUGGABLE GENOME SU-4312 CHEMBL328710 61003 41636 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651731 61004 41637 GMNN 51053 DRUGGABLE GENOME CLIOXANIDE CLIOXANIDE 61005 41638 PAH 5053 DRUGGABLE GENOME, ENZYME SAPROPTERIN SAPROPTERIN 61006 41639 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER RIMONABANT RIMONABANT 21511945 61007 41640 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PHA-767491 CHEMBL225519 61008 41641 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME hmg coa reductase inhibitors 61010 41642 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER IMATINIB IMATINIB 15805252 61011 41643 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR KAEMPFEROL KAEMPFEROL 61012 41644 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 252166817 61013 41645 AQP5 362 ION CHANNEL, TRANSPORTER inhibitor 178101032 61015 41646 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LEVOPROPOXYPHENE NAPSYLATE ANHYDROUS LEVOPROPOXYPHENE NAPSYLATE 61017 41647 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CUDC-101 CUDC-101 61018 41648 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TAE226 26090892 61023 41649 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor BAY869766 61024 41650 KDM4A 9682 DRUGGABLE GENOME, ENZYME ALVERINE CITRATE ALVERINE CITRATE 61025 41651 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CAPTAN CAPTAN 61026 41652 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 135652735 61027 41653 ALB 213 TRANSPORTER, DRUGGABLE GENOME Bismuth 61029 41654 ADM 133 DRUGGABLE GENOME, HORMONE ACTIVITY INSULIN INSULIN 12668590 61030 41655 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Alvespimycin ALVESPIMYCIN 26483207 61031 41656 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135651359 ZIPRASIDONE 61032 41657 XPNPEP1 7511 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252827461 61034 41658 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 EDARAVONE EDARAVONE 61037 41659 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME nicotine NICOTINE 26287939,24611668 61038 41660 RPS6KA5 9252 DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE GW843682X GW843682X 61039 41661 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TRIFLOXYSTROBIN TRIFLOXYSTROBIN 61040 41662 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650730 NORBINALTORPHIMINE 61043 41663 RGS4 5999 DRUGGABLE GENOME SALAGEN SALAGEN 61044 41664 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING BELINOSTAT BELINOSTAT 25937017 61048 41665 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Karenitecin KARENITECIN 61049 41666 ABCG1 9619 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME leucovorin LEUCOVORIN 26352872 61050 41667 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PMID27376512-Compound-Figure3CG 61053 41668 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME EUPAFOLIN EUPAFOLIN 61056 41669 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME Omacetaxine 61059 41670 HEBP1 50865 DRUGGABLE GENOME Vinyl sulfone derivative 1 61061 41671 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR BDBM50158791 61064 41672 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650680 NALBUPHINE 61065 41673 TUBB2B 347733 DRUGGABLE GENOME CHEMBL2105643 FOSBRETABULIN TROMETHAMINE 61066 41674 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor CHEMBL1200992 61068 41675 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor PD0325901 PD-0325901 61069 41676 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE FLUPHENAZINE HYDROCHLORIDE FLUPHENAZINE HYDROCHLORIDE 61070 41677 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME DILAZEP DILAZEP 61071 41678 TUBA4A 7277 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 61072 41679 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PROADIFEN HYDROCHLORIDE PROADIFEN HYDROCHLORIDE 61073 41680 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamate derivative 13 61074 41681 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME inhibitor MEK162 BINIMETINIB 61075 41682 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 7-azaindole derivative 8 61076 41683 MT2A 4502 NA PARACETAMOL ACETAMINOPHEN 9570328 61077 41684 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GIVINOSTAT GIVINOSTAT 61078 41685 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE Iomab-B APAMISTAMAB IODINE I-131 61079 41686 GMNN 51053 DRUGGABLE GENOME GNF-PF-3257 CHEMBL601768 61080 41687 MAPT 4137 DRUGGABLE GENOME PARAROSANILINE PARAROSANILINE 61081 41688 CTSA 5476 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 223366205 BOCEPREVIR 61086 41689 RIPK2 8767 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SB-202190 SB-202190 22951114 61087 41690 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME axitinib AXITINIB 26512042 61090 41691 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8669361, 103 61092 41692 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL inhibitor 178101132 61093 41693 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652252 61094 41694 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 178102547 61095 41695 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL2103739 EMEDASTINE DIFUMARATE 61096 41696 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545332 CEP-2563 61097 41697 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR doxorubicin DOXORUBICIN 24141364 61098 41698 SULT1A1 6817 DRUGGABLE GENOME, ENZYME tapentadol TAPENTADOL 61099 41699 USP1 7398 DNA REPAIR, PROTEASE, ENZYME MELITRACEN MELITRACEN 61100 41700 ARSA 410 DRUGGABLE GENOME, ENZYME GNF-PF-5510 CHEMBL578741 61101 41701 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DEVAZEPIDE DEVAZEPIDE 61102 41702 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE inhibitor 178103262 METHIMAZOLE 61103 41703 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Sunitinib SUNITINIB 27149458 61104 41704 KDM4A 9682 DRUGGABLE GENOME, ENZYME PROTOCATECHUALDEHYDE PROTOCATECHUALDEHYDE 61105 41705 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200590 MECLIZINE HYDROCHLORIDE 61107 41706 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE SP-600125 SP-600125 61108 41707 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL blocker 178101137 61109 41708 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650814 ALPROSTADIL 61111 41709 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TAMOXIFEN TAMOXIFEN 61112 41710 GBA 2629 DRUGGABLE GENOME, ENZYME L-755507 L-755507 61115 41711 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE SOMATROPIN RECOMBINANT 61116 41712 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL576982 QUIZARTINIB 61117 41713 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME MELOGLIPTIN 61119 41714 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE AST-487 AST-487 61122 41715 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RG7112 RO-5045337 26459177 61125 41716 COL4A5 1287 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 61127 41717 BAZ2B 29994 NA inhibitor 252166772 61128 41718 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200903 SECOBARBITAL SODIUM 61129 41719 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER CONGO RED CONGO RED 61130 41720 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GEFITINIB GEFITINIB 21258250 61131 41721 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Varlitinib VARLITINIB 61133 41722 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PHA-665752 PHA-665752 26351320 61134 41723 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ERLOTINIB ERLOTINIB 21258250 61135 41724 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SILVER SULFADIAZINE SILVER SULFADIAZINE 61136 41725 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 2 61137 41726 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102571 61138 41727 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE NOREPINEPHRINE NOREPINEPHRINE 2903243 61139 41728 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CCT018159 CHEMBL399530 61140 41729 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME valproic acid 23407051 61141 41730 TUBA1B 10376 DRUGGABLE GENOME CHEMBL2108628 PACLITAXEL POLIGLUMEX 61142 41731 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NCI-10777 CHEMBL189724 61143 41732 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PROROXAN HYDROCHLORIDE PROROXAN HYDROCHLORIDE 61144 41733 CDK16 5127 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL488436 AZD-5438 61145 41734 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALITRETIONINE 61146 41735 TXN 7295 DRUGGABLE GENOME, THIOREDOXIN PX-12 PX-12 61147 41736 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE inhibitor 384403653 61149 41737 MAPT 4137 DRUGGABLE GENOME CYSTEINE METHYL-ESTER HCL CHEMBL1426508 61150 41738 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IIB AESCULIOSIDE IIB 20371180 61151 41739 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody 252166672 TREMELIMUMAB 61153 41740 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE methotrexate METHOTREXATE 29791011 61154 41741 MAPT 4137 DRUGGABLE GENOME ISOVELLERAL ISOVELLERAL 61155 41742 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-22 61156 41743 PSMD2 5708 NA OPROZOMIB OPROZOMIB 61157 41744 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 3196 61158 41745 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor PIMASERTIB PIMASERTIB 61159 41746 ABCB4 5244 TRANSPORTER, DRUGGABLE GENOME, ENZYME, ABC TRANSPORTER imatinib IMATINIB 30237583 61160 41747 TYMSOS 494514 NA asparaginase ASPARAGINASE 61161 41748 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME RG-1530 RG-1530 61164 41749 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ANISOCOUMARIN H ANISOCOUMARIN H 61165 41750 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-L2 61167 41751 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME ALSTERPAULLONE ALSTERPAULLONE 61168 41752 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CYTARABINE CYTARABINE 61169 41753 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker 178101050 KETAMINE 61170 41754 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL598797 CUDC-101 61171 41755 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY TC-99M MIBI 11564916 61173 41756 VKORC1 79001 DRUGGABLE GENOME, ENZYME inhibitor 178103445 PHENPROCOUMON 61175 41757 ALOX15B 247 DRUGGABLE GENOME, ENZYME NSC-48300 CHEMBL1091971 61176 41758 CBX1 10951 NA PERPHENAZINE PERPHENAZINE 61177 41759 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER MEGESTROL ACETATE 9025774 61180 41760 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565834 61181 41761 HBB 3043 DRUGGABLE GENOME, ENZYME Voxelotor VOXELOTOR 61182 41762 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR DOVITINIB DOVITINIB 61184 41763 PSMD8 5714 NA inhibitor CHEMBL2103884 OPROZOMIB 61186 41764 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME vemurafenib VEMURAFENIB 61187 41765 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Aromatic bicyclic compound 6 61189 41766 COL5A2 1290 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 61190 41767 MPHOSPH8 54737 NA DAPH DAPH 61191 41768 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 61192 41769 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ENTRECTINIB ENTRECTINIB 26546295,26565381,28183697 61193 41770 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BELINOSTAT BELINOSTAT 61194 41771 EGLN3 112399 DRUGGABLE GENOME, ENZYME inhibitor 252166666 61195 41772 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE 178101726 61196 41773 TRPV2 51393 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker 135649936 AMILORIDE 61197 41774 PBRM1 55193 CLINICALLY ACTIONABLE IPILIMUMAB IPILIMUMAB 29301960 61198 41775 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX 2-METHOXY-1,4-NAPHTHOQUINONE 2-METHOXY-1,4-NAPHTHOQUINONE 61199 41776 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 252166733 61201 41777 PDE4B 5142 DRUGGABLE GENOME, ENZYME TOFIMILAST TOFIMILAST 61203 41778 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-123920 CHEMBL1606 61204 41779 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 61206 41780 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Nilotinib NILOTINIB 26725216 61209 41781 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LAUROCAPRAM LAUROCAPRAM 61210 41782 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE CILOSTAZOL CILOSTAZOL 61212 41783 NEK7 140609 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME inhibitor 249565885 61213 41784 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SP-600125 SP-600125 61217 41785 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR sorafenib SORAFENIB 20124951 61219 41786 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GOSSYPOL GOSSYPOL 61220 41787 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme9EHT9851 61221 41788 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL592445 GEDATOLISIB 61222 41789 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR TEMOZOLOMIDE TEMOZOLOMIDE 23904111 61223 41790 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR GNF-PF-52 CHEMBL601142 61224 41791 SERPINA1 5265 DRUGGABLE GENOME, PROTEASE INHIBITOR Glassia .ALPHA.1-PROTEINASE INHIBITOR HUMAN 61225 41792 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor LGX818 ENCORAFENIB 61226 41793 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TCMDC-125544 CHEMBL533602 61229 41794 NOS2 4843 DRUGGABLE GENOME, ENZYME SD-6010 61230 41795 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME ILEPCIMIDE ILEPCIMIDE 61231 41796 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER PROBENECID PROBENECID 9182837 61232 41797 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1201173 MEDRYSONE 61234 41798 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL608533 MIDOSTAURIN 61235 41799 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME BMS-582949 BMS-582949 61236 41800 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL944 CHLOROPROCAINE HYDROCHLORIDE 61237 41801 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GW3965 CHEMBL59030 18800767 61238 41802 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR TETRAHYDROCANNABINOL DRONABINOL 15857384 61239 41803 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 1,2-DIPHENYLDISULFANE CHEMBL462861 61241 41804 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL1567 SUNITINIB MALATE 61242 41805 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Dasatinib DASATINIB 26855149 61243 41806 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor VALPROIC ACID DEPAKOTE 61245 41807 ATXN2 6311 NA DNDI1417941 CHEMBL2095095 61247 41808 POLA1 5422 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL803 CYTARABINE 61248 41809 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ALTANSERIN ALTANSERIN 61249 41810 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL1908397 KW-2449 61252 41811 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RILMENIDINE HEMIFUMARATE RILMENIDINE HEMIFUMARATE 61253 41812 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DOVITINIB DOVITINIB 61255 41813 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME ABI-011 61257 41814 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE VACCINE ADJUVANT 11929774 61258 41815 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Palbociclib PALBOCICLIB 26369631 61259 41816 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 8,2'-DIMETHOXYFLAVONE 8,2'-DIMETHOXYFLAVONE 61260 41817 POLI 11201 DNA REPAIR ROTTLERIN ROTTLERIN 61262 41818 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR MEPAZINE ACETATE MEPAZINE ACETATE 61263 41819 PPP1R13L 10848 TRANSCRIPTION FACTOR BINDING Platinum compounds 19203783 61268 41820 EYA2 2139 DNA REPAIR SOLYPERTINE TARTRATE SOLYPERTINE TARTRATE 61269 41821 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR QUERCETIN DIHYDRATE QUERCETIN DIHYDRATE 61270 41822 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME NSC-158389 CHEMBL192626 61271 41823 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME atenolol ATENOLOL 61272 41824 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 363894135 MERESTINIB 61273 41825 RAB9A 9367 ENZYME, DRUGGABLE GENOME TCMDC-124354 CHEMBL546344 61275 41826 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR RG-1530 RG-1530 61276 41827 ALOX15B 247 DRUGGABLE GENOME, ENZYME ETHOPROPAZINE HYDROCHLORIDE ETHOPROPAZINE HYDROCHLORIDE 61277 41828 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200908 HALOBETASOL PROPIONATE 61278 41829 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR T091317 T091317 61279 41830 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME WEDELOLACTONE WEDELOLACTONE 61282 41831 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL389621 HYDROCORTISONE 61285 41832 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 135651754 61288 41833 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR STROPHANTHIDIN STROPHANTHIDIN 61289 41834 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE COLCHICINE COLCHICINE 7666195 61290 41835 KDM4A 9682 DRUGGABLE GENOME, ENZYME LEVODOPA LEVODOPA 61291 41836 NBEA 26960 KINASE metformin METFORMIN 29650774 61293 41837 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE moxifloxacin MOXIFLOXACIN 61294 41838 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE CARBONYL CYANIDE M-CHLOROPHENYLHYDRAZONE 61295 41839 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL oxcarbazepine OXCARBAZEPINE 23859570,21747585,22591328,28753467,25155934,26555147 61296 41840 STING1 340061 CLINICALLY ACTIONABLE, KINASE ADU-S100 ADU-S100 61297 41841 KLC1 3831 NA irinotecan IRINOTECAN 17549067 61298 41842 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TCMDC-123528 CHEMBL529138 61299 41843 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417623 CHEMBL2002849 61300 41844 SLC15A1 6564 DRUGGABLE GENOME, TRANSPORTER 178101217 61301 41845 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 4-Carboxamido-isoindolinone derivative 1 61302 41846 CLK1 1195 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor 249565735 61303 41847 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 363894130 TANZISERTIB 61304 41848 C1S 716 ENZYME, PROTEASE, DRUGGABLE GENOME MBL 10878362 61306 41849 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL451 CHLORDIAZEPOXIDE 61309 41850 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME formoterol FORMOTEROL 61310 41851 GMNN 51053 DRUGGABLE GENOME PD-169316 PD-169316 61311 41852 KDM4A 9682 DRUGGABLE GENOME, ENZYME 5-METHOXYTRYPTAMINE 5-METHOXYTRYPTAMINE 61313 41853 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME LEUCOVORIN LEUCOVORIN 20921465 61315 41854 PTGES3 10728 ENZYME GEDUNIN GEDUNIN 25756299 61316 41855 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PMID28048944-Compound-20 61318 41856 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIPHYLLIN DIPHYLLIN 22119124 61320 41857 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33m 61321 41858 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Ospemifene OSPEMIFENE 61322 41859 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR CETIRIZINE CETIRIZINE 16783450 61324 41860 GMNN 51053 DRUGGABLE GENOME DNDI1417156 CHEMBL1504679 61326 41861 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE 10-METHOXYLRUTAECARPINE CHEMBL85826 61327 41862 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000112483 CHEMBL603024 61328 41863 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR 2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE CHEMBL502774 61329 41864 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL428647 PACLITAXEL 61330 41865 BRCA2 675 CLINICALLY ACTIONABLE olaparib OLAPARIB 61332 41866 SMN1 6606 DRUGGABLE GENOME PHENAMIL PHENAMIL 61335 41867 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Camptothecin CAMPTOTHECIN 24042735,25688157 61336 41868 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR anastrozole ANASTROZOLE 61337 41869 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SALICYLAMIDE SALICYLAMIDE 61338 41870 POLI 11201 DNA REPAIR GNF-PF-67 CHEMBL578512 61339 41871 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ANIRACETAM ANIRACETAM 61340 41872 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER VANOXERINE VANOXERINE 61342 41873 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BAY80-6946 COPANLISIB 61345 41874 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE JNJ-7706621 JNJ-7706621 61347 41875 SLC6A14 11254 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME inhibitor 178101406 61348 41876 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-10 61350 41877 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BENZODIAZEPINE BENZODIAZEPINE 9574817 61351 41878 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE 5-AZACYTIDINE AZACITIDINE 6173384 61352 41879 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE 5-AMINOLAEVULINIC ACID 9868803 61353 41880 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR methoxamine METHOXAMINE 61355 41881 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL1980391 RG-1530 61356 41882 POLK 51426 DNA REPAIR, ENZYME STALLIMYCIN STALLIMYCIN 61357 41883 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-309895 CHEMBL552439 61358 41884 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHLOROQUINE CHLOROQUINE 61359 41885 USP1 7398 DNA REPAIR, PROTEASE, ENZYME NORSTICTIC ACID NORSTICTIC ACID 61362 41886 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor BGJ398 INFIGRATINIB 61363 41887 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor LENVATINIB LENVATINIB 61364 41888 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME epirubicin EPIRUBICIN 27234217 61365 41889 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEFACLOR CEFACLOR 61366 41890 LGALS8 3964 DRUGGABLE GENOME LACTOSE, ANHYDROUS LACTOSE, ANHYDROUS 21524586 61368 41891 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME ILORASERTIB ILORASERTIB 61371 41892 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME BIX-01294 CHEMBL569864 61372 41893 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Prednisone PREDNISONE 61373 41894 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE PMID27410995-Compound-Figure3c 61374 41895 POLK 51426 DNA REPAIR, ENZYME QUERCETIN DIHYDRATE QUERCETIN DIHYDRATE 61375 41896 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME QUERCETIN QUERCETIN 17045724 61377 41897 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE Recombinant human Erbb3 fragment therapeutic tumor vaccine 61379 41898 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-24 61380 41899 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME bepridil BEPRIDIL 16508157 61382 41900 PLAUR 5329 DRUGGABLE GENOME, ENZYME, CELL SURFACE MCP-2 12138365 61383 41901 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 249565855 61384 41902 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 6-14 61385 41903 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME GW459057A GW459057A 16890436 61388 41904 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MIDAZOLAM HYDROCHLORIDE MIDAZOLAM HYDROCHLORIDE 61389 41905 POLA1 5422 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL1750 CLOFARABINE 61392 41906 MT-RNR1 4549 KINASE aminoglycoside antibacterials 18830133,16875663,9164619,19682603,16631122,21495045,16782057,16458854,12031626,17489842,16375862,9831149,1583319,17637808,22475488,11857751,27397648,9779807,7689389,20111055,9111378,27427311,17698030,11313749,20416460,16168391,12496758,24703164,9950117,21504270,11174059,8285309,18790089,15917167,10686428,20353758,21047563,24100002,16955413,16380089,15110318,14699607,17999439,14755216,8910275,16650816,17341440,19371214,25376778,19376484,15708009,22735573,25515069,15555598,16528519,11079536,17434445,18261986 61393 41907 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135650027 61394 41908 CYP7A1 1581 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME atorvastatin ATORVASTATIN 16103896,15262185,26932749,21128988 61397 41909 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist CHEMBL1428 NIMODIPINE 61398 41910 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE D-64131 CHEMBL140220 61401 41911 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE GLUCOCORTICOID 11449367 61403 41912 PSMB7 5695 DRUGGABLE GENOME, PROTEASE inhibitor BORTEZOMIB BORTEZOMIB 61404 41913 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PERPHENAZINE PERPHENAZINE 61405 41914 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178102588 61406 41915 BCHE 590 DRUGGABLE GENOME, ENZYME Mivacurium MIVACURIUM 61408 41916 NOS2 4843 DRUGGABLE GENOME, ENZYME KLH 11359093 61410 41917 TUBB2A 7280 DRUGGABLE GENOME AEZS-112, ZEN-012 61411 41918 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME SALMETEROL XINAFOATE SALMETEROL XINAFOATE 61412 41919 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME N-(pyridin-2-yl)pyridine methylsulfone derivative 1 61413 41920 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 328083470 61414 41921 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BENZOTHIAZYL DISULFIDE BENZOTHIAZYL DISULFIDE 61415 41922 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 223366147 ORANTINIB 61418 41923 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KOPARIN KOPARIN 61419 41924 CXCL8 3576 DRUGGABLE GENOME RIBAVIRIN RIBAVIRIN 61421 41925 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417195 CHEMBL1303948 61422 41926 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DEFLAZACORT DEFLAZACORT 61423 41927 PDE4B 5142 DRUGGABLE GENOME, ENZYME OX914 61424 41928 CES1 1066 DRUGGABLE GENOME, ENZYME capecitabine CAPECITABINE 28139840 61425 41929 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TCMDC-125758 CHEMBL546797 61426 41930 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Gefitinib GEFITINIB 25870145 61427 41931 CXCL8 3576 DRUGGABLE GENOME inhibitor CHEMBL2109616 ABX-IL8 61428 41932 NRXN1 9378 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER duloxetine DULOXETINE 29407288 61431 41933 HFE 3077 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME adalimumab ADALIMUMAB 27115882 61432 41934 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200759 ANAGRELIDE HYDROCHLORIDE 61434 41935 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME AG-808 CHEMBL68534 61436 41936 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1752 DYPHYLLINE 61439 41937 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CUDC-101 CUDC-101 61440 41938 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor CHEMBL1173055 RUCAPARIB 61442 41939 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR antagonist CHEMBL271220 CORT 108297 61443 41940 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME HGF 9454825 61444 41941 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3',4'-DIHYDROXYFLAVONE CHEMBL222556 61446 41942 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NAFOXIDINE NAFOXIDINE 2580656 61447 41943 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650182 DIHYDROERGOTAMINE 61449 41944 ABHD6 57406 PHOSPHOLIPASE, ENZYME ORLISTAT ORLISTAT 26344596 61450 41945 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 135650432 61452 41946 SERPINA6 866 DRUGGABLE GENOME, PROTEASE INHIBITOR BECLOMETHASONE BECLOMETHASONE 61454 41947 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ASCORBYL PALMITATE ASCORBYL PALMITATE 61456 41948 SMN1 6606 DRUGGABLE GENOME DNDI1417548 CHEMBL2094789 61457 41949 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME HALOPERIDOL HALOPERIDOL 12614997 61461 41950 MAPT 4137 DRUGGABLE GENOME CEAROIN CEAROIN 61462 41951 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme7WO2012/098070upper 61463 41952 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135650018 CHEMBL291314 61464 41953 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor VALPROIC ACID DEPAKOTE 61465 41954 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor PF-4691502 PF-04691502 61466 41955 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME VANDETANIB VANDETANIB 61468 41956 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER LB-100 LB-100 25376608 61472 41957 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME KOPARIN KOPARIN 61473 41958 POLI 11201 DNA REPAIR GNF-PF-5510 CHEMBL578741 61474 41959 MAPT 4137 DRUGGABLE GENOME TCMDC-124544 CHEMBL531322 61475 41960 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER QUINOLIN-6-YLAMINE CHEMBL99408 61476 41961 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 61478 41962 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135649686 61480 41963 PTGS1 5742 ENZYME, DRUGGABLE GENOME DICLOFENAC DICLOFENAC 61485 41964 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HELENALIN HELENALIN 61486 41965 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TESAGLITAZAR TESAGLITAZAR 61487 41966 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 3,5-DIPHENYLISOXAZOLE 3,5-DIPHENYLISOXAZOLE 61488 41967 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AZATHIOPRINE AZATHIOPRINE 61494 41968 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565646 PILARALISIB 61495 41969 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE TAE684 20207848 61498 41970 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME tretinoin TRETINOIN 61499 41971 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME AG-1879 CHEMBL406845 61500 41972 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CEPHALEXIN CEPHALEXIN 22166395 61501 41973 C1S 716 ENZYME, PROTEASE, DRUGGABLE GENOME ANTITHROMBIN 61502 41974 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545088 PUQUITINIB 61503 41975 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DEPHOSTATIN DEPHOSTATIN 61504 41976 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Dutasteride + tamsulosin 61505 41977 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor AZD 2281 61507 41978 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2087337 VELUSETRAG 61508 41979 SULT2B1 6820 ENZYME, DRUGGABLE GENOME idarubicin IDARUBICIN 22584460 61509 41980 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ALAZANINE ALAZANINE 61510 41981 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER 10-DEACETOXYPACLITAXEL CHEMBL306786 16271474 61514 41982 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 4'-HYDROXY-FLAVANONE 4'-HYDROXY-FLAVANONE 61516 41983 USP1 7398 DNA REPAIR, PROTEASE, ENZYME EPIRUBICIN HYDROCHLORIDE EPIRUBICIN HYDROCHLORIDE 61517 41984 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE KU-60019 61518 41985 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE OLAPARIB OLAPARIB 18800822 61519 41986 CASP2 835 PROTEASE, DRUGGABLE GENOME, ENZYME N-DECYLBUTYRAMIDE CHEMBL265439 18366176 61520 41987 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE antisense oligonucleotide OBLIMERSEN OBLIMERSEN 61521 41988 MAPT 4137 DRUGGABLE GENOME TCMDC-124518 CHEMBL527584 61526 41989 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Veliparib VELIPARIB 21300883,27638859 61527 41990 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 249565856 61528 41991 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651064 SPIPERONE 61529 41992 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME atorvastatin ATORVASTATIN 61530 41993 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME TINIDAZOLE TINIDAZOLE 14553936 61531 41994 TSPO 706 DRUGGABLE GENOME Imidazo[1,2-b]pyridazine acetamide derivative 1 61532 41995 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 61533 41996 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Carboxamide derivative 5 61534 41997 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METAPHIT METHANESULFONATE METAPHIT METHANESULFONATE 61535 41998 MAPT 4137 DRUGGABLE GENOME EMBELIN EMBELIN 61539 41999 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE ILORASERTIB ILORASERTIB 61541 42000 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR DDI DIDANOSINE 17616550 61543 42001 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PALBOCICLIB PALBOCICLIB 27167191 61544 42002 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE MLN-8054 MLN-8054 61545 42003 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 benzphetamine BENZPHETAMINE 9187528 61546 42004 TEAD1 7003 TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX DEXAMETHASONE DEXAMETHASONE 12207913 61547 42005 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROMAZINE PROMAZINE 61548 42006 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE EKI-285 22046346 61551 42007 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135649889 ACIFRAN 61552 42008 MAPT 4137 DRUGGABLE GENOME SB-408124 CHEMBL1334465 61554 42009 ALPL 249 ENZYME, DRUGGABLE GENOME TERPYRIDINE TERPYRIDINE 61556 42010 KDM4A 9682 DRUGGABLE GENOME, ENZYME ELLAGIC ACID ELLAGIC ACID 61557 42011 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 178102316 CHEMBL1908395 61558 42012 XPNPEP3 63929 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2103847 TOSEDOSTAT 61560 42013 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 385612216 61561 42014 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE ALSTERPAULLONE ALSTERPAULLONE 61562 42015 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR SALT VOLANESORSEN SODIUM 1939057 61563 42016 TUBB2A 7280 DRUGGABLE GENOME CHEMBL492399 VERUBULIN 61566 42017 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TACEDINALINE TACEDINALINE 18692397 61567 42018 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME TAMATINIB R-406 61569 42019 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MDV3100 ENZALUTAMIDE 61570 42020 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MESO-HEXESTROL MESO-HEXESTROL 61571 42021 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 348353674 61572 42022 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TDZD-8 61573 42023 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PALBOCICLIB PALBOCICLIB 61575 42024 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GW642444 VILANTEROL 61578 42025 RRM2 6241 DRUGGABLE GENOME, ENZYME CO-101 GEMCITABINE ELAIDATE 61580 42026 TSPO 706 DRUGGABLE GENOME BAY-85-8102 61582 42027 IFNG 3458 DRUGGABLE GENOME AMITRIPTYLINE AMITRIPTYLINE 10996474 61583 42028 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mizoribine MIZORIBINE 61586 42029 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE AG-014361 CHEMBL65892 61587 42030 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650529 61590 42031 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 310264693 ACALABRUTINIB 61591 42032 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650145 61592 42033 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLORGILINE CLORGILINE 61593 42034 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR CRA-024781 ABEXINOSTAT 61594 42035 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652714 61595 42036 TSPO 706 DRUGGABLE GENOME Benzothiazepine analog 4 61596 42037 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR GNF-PF-67 CHEMBL578512 61597 42038 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL1096380 PLINABULIN 61598 42039 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME P7170 PANULISIB 61599 42040 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3544960 AT-13148 61600 42041 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR FLAVOPIRIDOL ALVOCIDIB 14767524 61601 42042 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CONGO RED CONGO RED 61602 42043 HEBP1 50865 DRUGGABLE GENOME 3-phenyl propanoic derivative 1 61603 42044 COMT 1312 DRUGGABLE GENOME, ENZYME Entacapone+levodopa+carbidopa 61604 42045 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME CHRYSOPHANOL CHRYSOPHANOL 61605 42046 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TAK-285 TAK-285 61606 42047 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649939 AMITRIPTYLINE 61609 42048 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME AZD5153 AZD-5153 61610 42049 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE TRAIL 16153452,16984382 61614 42050 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ALSTERPAULLONE ALSTERPAULLONE 61615 42051 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL inhibitor 374883867 61617 42052 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME TCMDC-123912 CHEMBL106525 61622 42053 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NICLOSAMIDE NICLOSAMIDE 61624 42054 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist EFATUTAZONE EFATUTAZONE 61625 42055 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL LORAZEPAM LORAZEPAM 61626 42056 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME 3-phenyl acrylic acid derivative 1 61627 42057 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 310264693 ACALABRUTINIB 61628 42058 MTR 4548 ENZYME, DRUGGABLE GENOME benazepril BENAZEPRIL 15148588 61629 42059 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME GAMBOGIC ACID GAMBOGIC ACID 61632 42060 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124316 CHEMBL534214 61634 42061 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652528 61637 42062 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-228155 CHEMBL505670 61638 42063 TEP1 7011 NA V934/V935 61639 42064 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR STANOZOLOL STANOZOLOL 61640 42065 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COLCHICINE COLCHICINE 61641 42066 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING CLOFIBRATE CLOFIBRATE 16680159 61642 42067 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CLOBENPROPIT CLOBENPROPIT 61644 42068 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-3 61645 42069 MAP2K5 5607 KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565744 61647 42070 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHRYSOPHANOL CHRYSOPHANOL 61650 42071 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RITONAVIR RITONAVIR 61651 42072 DUSP3 1845 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE MESO-2,3-DIMERCAPTOSUCCINIC ACID CHEMBL28721 61652 42073 FMO3 2328 ENZYME, DRUGGABLE GENOME olanzapine OLANZAPINE 23147717 61654 42074 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Thieno[2,3-c]pyridine derivative 1 61655 42075 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR THIOINOSINE THIOINOSINE 61658 42076 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME NIFLUMIC ACID NIFLUMIC ACID 61661 42077 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor CHEMBL408513 BELINOSTAT 61663 42078 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyrrolo-pyridazine derivative 1 61664 42079 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ROMIDEPSIN ROMIDEPSIN 61665 42080 MPHOSPH8 54737 NA NIFEDIPINE NIFEDIPINE 61666 42081 FCGRT 2217 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antibody 354702273 ROZANOLIXIZUMAB 61668 42082 MAPT 4137 DRUGGABLE GENOME TYRPHOSTIN 51 TYRPHOSTIN 51 61670 42083 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL3545381 PLX-7486 61671 42084 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER N/A 61672 42085 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DI-TERT-BUTYLHYDROQUINONE CHEMBL480626 61674 42086 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE UNC10112764A CHEMBL329040 61675 42087 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME (R,S)-INDATRALINE (R,S)-INDATRALINE 61678 42088 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CARDAMOMIN CARDAMOMIN 25959811 61679 42089 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX ADAPALENE ADAPALENE 61681 42090 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-239272 CHEMBL275798 61683 42091 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ISOTRETINOIN ISOTRETINOIN 61684 42092 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE cyclophosphamide CYCLOPHOSPHAMIDE 61685 42093 TUBA3D 113457 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 61688 42094 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102299 BRIVANIB 61689 42095 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PELUBIPROFEN PELUBIPROFEN 61691 42096 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRICHLOROMONOFLUOROMETHANE TRICHLOROMONOFLUOROMETHANE 61692 42097 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL blocker 135652678 CORREOLIDE 61694 42098 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GF-109203 GF-109203 61695 42099 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CLONAZEPAM CLONAZEPAM 61696 42100 GMNN 51053 DRUGGABLE GENOME WIN-62577 CHEMBL1256845 61697 42101 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL2303638 61700 42102 PTGS2 5743 DRUGGABLE GENOME, ENZYME diclofenac sodium patch 61701 42103 GMNN 51053 DRUGGABLE GENOME SJ000067611 CHEMBL602126 61702 42104 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CADMIUM ACETATE CADMIUM ACETATE 61703 42105 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NONIVAMIDE NONIVAMIDE 61704 42106 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME docetaxel DOCETAXEL 22441531 61706 42107 NF2 4771 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, DRUG RESISTANCE, KINASE CISPLATIN CISPLATIN 25798586 61707 42108 PTGS1 5742 ENZYME, DRUGGABLE GENOME MESALAMINE MESALAMINE 61709 42109 PTPRB 5787 DRUGGABLE GENOME, PROTEIN PHOSPHATASE inhibitor 252827444 61710 42110 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650510 61713 42111 TUBB3 10381 DRUGGABLE GENOME CHEMBL492399 VERUBULIN 61715 42112 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE TOFACITINIB TOFACITINIB 61716 42113 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE ILORASERTIB ILORASERTIB 61717 42114 FABP1 2168 DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 15324484,15532708 61719 42115 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107762 NERISPIRDINE 61720 42116 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER SCUTELLARIN SCUTELLARIN 22822035 61721 42117 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME KO-947 61722 42118 NOS1 4842 DRUGGABLE GENOME, ENZYME PROPOFOL PROPOFOL 16645450 61723 42119 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Sapanisertib SAPANISERTIB 26574479 61724 42120 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Oxazole derivative 1 61726 42121 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Five-membered heteroaromatic compound 1 61728 42122 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME risperidone RISPERIDONE 23859574 61729 42123 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1255840 NEBOGLAMINE 61730 42124 CDK18 5129 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR inhibitor CHEMBL445813 AT-7519 61734 42125 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TELAPRISTONE 61736 42126 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 135651392 CHEMBL169046 61737 42127 KRT10 3858 CELL SURFACE OPIOID 9450624 61738 42128 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME 4-(2-BENZYLPHENOXY)PIPERIDINE CHEMBL1923521 22007643 61739 42129 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE 7-azaindole derivative 6 61740 42130 PDE5A 8654 ENZYME, DRUGGABLE GENOME Rhucin RHUCIN 61741 42131 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE ALMITRINE ALMITRINE 61744 42132 SULT2A1 6822 DRUGGABLE GENOME TGF 3164434 61746 42133 PGM1 5236 ENZYME acetaldehyde ACETALDEHYDE 31002879 61747 42134 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102339 SUNITINIB 61748 42135 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1557 DOPAMINE HYDROCHLORIDE 61750 42136 BARD1 580 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR trastuzumab TRASTUZUMAB 30071039 61752 42137 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor BGJ398 INFIGRATINIB 61753 42138 GLCCI1 113263 NA triamcinolone TRIAMCINOLONE 21991891 61754 42139 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ETOPOSIDE ETOPOSIDE 25466187,20006518,18258442,22867019,25240702,26291037,25003995,26216018,26292628,23360284,23920485,21435753,22867097,16759114,11678653,19386396,24931277,23566520,25922181,25941559,24507920,24775914,23353750,25815139,24012683,19691293,25800514,21644529,22620261,25945730,24334150,23711769,20863598,24095018,26264845,25799376,22364746,23968711,18816045,24326278,19783445 61757 42140 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE IMATINIB IMATINIB 61758 42141 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME IP10 C8 61760 42142 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HYMECROMONE HYMECROMONE 61761 42143 ATXN2 6311 NA HONOKIOL HONOKIOL 61762 42144 KDM4A 9682 DRUGGABLE GENOME, ENZYME THIOMERSAL THIMEROSAL 61763 42145 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL1742994 BRENTUXIMAB VEDOTIN 61765 42146 RBL1 5933 ENZYME, TRANSCRIPTION FACTOR COMPLEX HMBA 9205091 61766 42147 NDUFAF1 51103 NA inhibitor CHEMBL3545320 ME-344 61770 42148 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MIRTAZAPINE MIRTAZAPINE 61771 42149 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME SGN-CD70A 61772 42150 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE GM-CSF REGRAMOSTIM 15107457 61773 42151 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrrole six-membered heteroaryl ring derivative 1 61775 42152 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135651110 61776 42153 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME FISETIN FISETIN 61777 42154 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 135651465 61778 42155 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME Flunarizine FLUNARIZINE 61779 42156 MAPT 4137 DRUGGABLE GENOME OXITRIPTAN OXITRIPTAN 61780 42157 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1201535 PHENYLPROPANOLAMINE POLISTIREX 61782 42158 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178100990 61784 42159 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE AKT INHIBITOR VIII CHEMBL258844 17603540 61785 42160 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 24-OXOCYCLOARTANOL CHEMBL225869 25453801 61788 42161 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE GSK690693 GSK-690693 61789 42162 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BGJ398 INFIGRATINIB 27053219,25294908,22837387,27401245,26270481,23002168,28034880,27870574,25589496 61793 42163 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MESALAMINE MESALAMINE 61794 42164 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER NSC-95397 CHEMBL429095 61795 42165 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME RP5063 61796 42166 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OCTASTATIN VAPREOTIDE ACETATE 8653698 61798 42167 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178100731 61799 42168 POLK 51426 DNA REPAIR, ENZYME RHEIN RHEIN 61802 42169 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Cycloalkyl nitrile pyrazolo pyridone derivative 1 61803 42170 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GEFITINIB GEFITINIB 61804 42171 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Pyridine derivative 21 61805 42172 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME OXIDOPAMINE OXIDOPAMINE 61808 42173 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-5183 CHEMBL577660 61809 42174 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE ILEPCIMIDE ILEPCIMIDE 61810 42175 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE VX-680 TOZASERTIB 61811 42176 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Bis-aminopyrimidine derivative 4 61812 42177 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME BENZALDEHYDE O-4-METHOXYPHENYLCARBAMOYL OXIME CHEMBL599469 61813 42178 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL activator 135652675 CAFFEINE 61815 42179 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NAFTOPIDIL NAFTOPIDIL 61816 42180 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PYRAZOPHOS PYRAZOPHOS 61817 42181 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Desvenlafaxine DESVENLAFAXINE 61819 42182 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 hmg coa reductase inhibitors 61823 42183 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TPKI-24 CHEMBL2392553 61824 42184 SFTPA1 653509 DRUGGABLE GENOME HYDROGEN PEROXIDE 7943250 61825 42185 CXCL8 3576 DRUGGABLE GENOME bevacizumab BEVACIZUMAB 23584701 61826 42186 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650593 61827 42187 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GPX-100 13-DEOXYDOXORUBICIN 61828 42188 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR 2-PYRIDYLCARBOXALDEHYDE P-NITROBENZOYL HYDRAZONE CHEMBL255067 61830 42189 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 61831 42190 CES1 1066 DRUGGABLE GENOME, ENZYME mycophenolic acid 24220207 61832 42191 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE hmg coa reductase inhibitors 61834 42192 HBA2 3040 NA negative modulator CHEMBL18901 EFAPROXIRAL 61835 42193 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor BELINOSTAT BELINOSTAT 61836 42194 SRD5A1 6715 DRUGGABLE GENOME FINASTERIDE FINASTERIDE 61837 42195 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL HALAZEPAM HALAZEPAM 61838 42196 KMO 8564 DRUGGABLE GENOME, ENZYME Benzene sulfonamide derivative 6 61839 42197 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR antagonist,inhibitor 178103613 61841 42198 TNFRSF9 3604 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE Urelumab URELUMAB 61842 42199 RPS6KA6 27330 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME inhibitor 249565819 61843 42200 NDUFA3 4696 ENZYME inhibitor CHEMBL3545135 NV-128 61846 42201 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1201836 OFATUMUMAB 61847 42202 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 223366204 COPANLISIB 61849 42203 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL1738757 REBASTINIB 61850 42204 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE tadalafil TADALAFIL 18695978 61851 42205 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200841 PROCAINE HYDROCHLORIDE 61852 42206 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 L-162313 CHEMBL288174 61854 42207 HTT 3064 DRUGGABLE GENOME SJ000001592 CHEMBL591834 61855 42208 IL1B 3553 KINASE, DRUGGABLE GENOME THYROGLOBULIN THYROGLOBULIN 2788696 61857 42209 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NITROBENZENE NITROBENZENE 61858 42210 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 135651326 61859 42211 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor PIVANEX AN-9 61860 42212 PTGS1 5742 ENZYME, DRUGGABLE GENOME Antiinflammatory agents, non-steroids 20538124 61861 42213 HBB 3043 DRUGGABLE GENOME, ENZYME CID 94381 CHEMBL374632 61862 42214 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR MIFEPRISTONE MIFEPRISTONE 61863 42215 ITGA2 3673 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE clopidogrel CLOPIDOGREL 17157856,16493486,15205592,22940005,16214444 61864 42216 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200323 LABETALOL HYDROCHLORIDE 61865 42217 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE CYPATE CYPATE 22871580 61867 42218 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1628234 DOXEPIN HYDROCHLORIDE 61868 42219 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor SELUMETINIB SELUMETINIB 61870 42220 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR IMMUNOTOXIN 16648577 61871 42221 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME DNDI1417031 CHEMBL1333049 61873 42222 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-2776 CHEMBL578294 61874 42223 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RISPERIDONE RISPERIDONE 61875 42224 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A7 61876 42225 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor 354702260 DEBIO-1347 61879 42226 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4464 CHEMBL600692 61880 42227 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL571948 Y-39983 61881 42228 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3544999 SAMOTOLISIB 61882 42229 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme5 61883 42230 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-172033 CHEMBL238624 61884 42231 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor GSK1070916 GSK-1070916 61887 42232 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER THC DRONABINOL 16439618 61889 42233 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BMS-193885 CHEMBL324554 61890 42234 RIPK2 8767 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102664 61893 42235 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL CHLOROTHIAZIDE CHLOROTHIAZIDE 61894 42236 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651635 61895 42237 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL Diltiazem DILTIAZEM 61896 42238 UBA2 10054 DRUGGABLE GENOME, ENZYME PEVONEDISTAT PEVONEDISTAT 61897 42239 GUCY2C 2984 DRUGGABLE GENOME, KINASE Plecanatide PLECANATIDE 61899 42240 XDH 7498 DRUGGABLE GENOME, ENZYME QUERCETIN QUERCETIN 6099408 61900 42241 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DNDI1417400 CHEMBL1362503 61904 42242 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 385612249 61905 42243 IFNGR1 3459 DRUGGABLE GENOME, CLINICALLY ACTIONABLE INTERFERON GAMMA-1B 61907 42244 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR inhibitor 249565920 61910 42245 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE GW441756X GW441756X 61913 42246 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME XL147 PILARALISIB 25637314,21216929 61914 42247 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BROMOENOL LACTONE BROMOENOL LACTONE 61915 42248 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE MELAGATRAN MELAGATRAN 61916 42249 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BAY80-6946 COPANLISIB 61917 42250 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE antiepileptics 21449672,27816260,22630058,22188362,24624913,25155934,22256867,23697249,24567120,21799461 61922 42251 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SGX523 61923 42252 BAZ2B 29994 NA ECONAZOLE NITRATE ECONAZOLE NITRATE 61925 42253 PTGS2 5743 DRUGGABLE GENOME, ENZYME MEFENAMIC ACID 61927 42254 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL315985 ESLICARBAZEPINE 61930 42255 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamide derivative 1 61931 42256 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE NOX-A12 61933 42257 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4659 CHEMBL584442 61934 42258 FHIT 2272 CLINICALLY ACTIONABLE, ENZYME, TRANSPORTER interferon beta-1a 27001119 61939 42259 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650698 CHEMBL294192 61940 42260 COMT 1312 DRUGGABLE GENOME, ENZYME Ergot alkaloids 25096645 61942 42261 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 E324 E324 61943 42262 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 187051799 DACINOSTAT 61946 42263 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME agonist 348353645 TAPINAROF 61948 42264 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME BORTEZOMIB BORTEZOMIB 20875739 61949 42265 BAZ2B 29994 NA GNF-PF-4283 CHEMBL606166 61951 42266 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE PAZOPANIB PAZOPANIB 61952 42267 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651266 TIOTROPIUM 61953 42268 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417943 CHEMBL1326758 61954 42269 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Bis-aminopyrimidine derivative 2 61955 42270 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-31 61956 42271 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR MELPHALAN MELPHALAN 61958 42272 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Biphenyl derivative 1 61961 42273 CA1 759 DRUGGABLE GENOME, ENZYME ACETAZOLAMIDE ACETAZOLAMIDE 61963 42274 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565636 BMS-777607 61964 42275 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LINOPIRDINE LINOPIRDINE 61965 42276 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 APIOL APIOL 61966 42277 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SANSALVAMIDE A-AMIDE CHEMBL192264 21764310 61967 42278 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ELLAGIC ACID ELLAGIC ACID 61968 42279 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 5 61969 42280 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135649733 61971 42281 F5 2153 DRUGGABLE GENOME Tamoxifen TAMOXIFEN 61972 42282 SMN1 6606 DRUGGABLE GENOME CID 650707 CHEMBL408653 61973 42283 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE MLN-8054 MLN-8054 61975 42284 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME METHOTREXATE METHOTREXATE 22931300 61976 42285 MALAT1 378938 NA Ivabradine IVABRADINE 61977 42286 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Savolitinib SAVOLITINIB 61978 42287 MARCKSL1 65108 KINASE STAUROSPORINE STAUROSPORINE 1730592 61979 42288 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545421 DERAZANTINIB 61980 42289 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Tumor necrosis factor alpha (TNF-alpha) inhibitors 16720636,16909270,23057546,26244882,12847678,18050183,18713756,19365401,22760475,24192118,17343250,22960943,22129793,25311255,12190096,18438841,17673491,15695296 61981 42290 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Metformin METFORMIN 24077915,23877793 61982 42291 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIPARANOL TRIPARANOL 61983 42292 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PF-1228305 61985 42293 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PD-0166285 PD-0166285 61987 42294 HTT 3064 DRUGGABLE GENOME DNDI1417601 CHEMBL1503729 61988 42295 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor MOTESANIB MOTESANIB 61990 42296 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 336446937 NAPROXCINOD 61994 42297 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR DNDI1417523 CHEMBL598663 61995 42298 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DNDI1318925 CHEMBL1390716 61996 42299 POLK 51426 DNA REPAIR, ENZYME 2',3'-DIHYDROXYFLAVONE CHEMBL242171 61997 42300 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME PROTEIN PHOSPHATASE INHIBITOR 11883953 61998 42301 GAA 2548 DRUGGABLE GENOME, ENZYME CHEMBL460785 DUVOGLUSTAT HYDROCHLORIDE 62000 42302 CCR10 2826 DRUGGABLE GENOME, CELL SURFACE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135651681 62002 42303 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL1207366 GW468816 62004 42304 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER desipramine DESIPRAMINE 62005 42305 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE FF-284 26438159 62006 42306 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR DIAPLASININ DIAPLASININ 62007 42307 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-466314A GSK-466314A 62008 42308 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE CAR-T cells targeting EphA2 62009 42309 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NSC-228155 CHEMBL505670 62010 42310 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME VX-702 VX-702 62011 42311 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BROMETHALIN BROMETHALIN 62012 42312 BAZ2B 29994 NA OXOPURPUREINE OXOPURPUREINE 62013 42313 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ETOPOSIDE ETOPOSIDE 23999041 62014 42314 AK4 205 ENZYME, KINASE tenofovir TENOFOVIR 62015 42315 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL571546 KX2-391 62016 42316 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME isatin sulfonamide 34 62017 42317 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 62018 42318 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TICLOPIDINE TICLOPIDINE 22931300 62019 42319 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR QUERCETIN QUERCETIN 62020 42320 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 3,3',4',5-TETRACHLOROSALICYLANILIDE 3,3',4',5-TETRACHLOROSALICYLANILIDE 62021 42321 VKORC1L1 154807 DRUGGABLE GENOME, ENZYME WARFARIN WARFARIN 62022 42322 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AZD7762 AZD-7762 23839309 62023 42323 PTGS2 5743 DRUGGABLE GENOME, ENZYME DIFLUNISAL DIFLUNISAL 62024 42324 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3039518 BATEFENTEROL 62025 42325 HPGDS 27306 ENZYME, DRUGGABLE GENOME HF-0220 62026 42326 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 62027 42327 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE tezacaftor TEZACAFTOR 28930490,29099333,29099344 62028 42328 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ASTEMIZOLE ASTEMIZOLE 62029 42329 TSPO 706 DRUGGABLE GENOME FLUNITRAZEPAM FLUNITRAZEPAM 62030 42330 GMNN 51053 DRUGGABLE GENOME PYRITHIONE ZINC PYRITHIONE ZINC 62031 42331 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME DIBENZ[A,H]ANTHRACENE DIBENZ[A,H]ANTHRACENE 62032 42332 CA9 768 DRUGGABLE GENOME, ENZYME Sulfonamide derivative 12 62033 42333 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME bupropion BUPROPION 21658141 62034 42334 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME 8-AZAGUANINE 8-AZAGUANINE 1207869 62035 42335 MAPT 4137 DRUGGABLE GENOME POMIFERIN POMIFERIN 62037 42336 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME GM6001 62038 42337 ALDH1A1 216 DRUGGABLE GENOME, ENZYME H89 CHEMBL104264 62040 42338 PTPN12 5782 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, KINASE SUNITINIB SUNITINIB 29578538 62041 42339 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR inhibitor LDE225 SONIDEGIB 62043 42340 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE CI-1033 CANERTINIB 62044 42341 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1069 VALSARTAN 62045 42342 BRCA2 675 CLINICALLY ACTIONABLE BGB-290 PAMIPARIB 62046 42343 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL blocker 135652058 62047 42344 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ATROPINE ATROPINE 62049 42345 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DOVITINIB DOVITINIB 62050 42346 KDM4A 9682 DRUGGABLE GENOME, ENZYME 3,4-DIHYDROXYPHENYLACETIC ACID 3,4-DIHYDROXYPHENYLACETIC ACID 62052 42347 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3544966 GSK-1059615 62053 42348 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NALTREXONE NALTREXONE 62057 42349 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE DACTOLISIB DACTOLISIB 62058 42350 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-39 62059 42351 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650388 IMPROMIDINE 62060 42352 PSMD12 5718 NA BORTEZOMIB BORTEZOMIB 24524217 62061 42353 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BAZEDOXIFENE BAZEDOXIFENE 62062 42354 RPS6KA5 9252 DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE US9365572, 5 62063 42355 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Osimertinib OSIMERTINIB 25870145,28416483 62064 42356 PSCA 8000 DRUGGABLE GENOME Anti-PSCA mab 62065 42357 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor CHEMBL488436 AZD-5438 62066 42358 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LEUPROLIDE LEUPROLIDE 22931300 62067 42359 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-arylmethyl-N-phenyl cyclic urea derivative 2 62069 42360 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE methazolamide METHAZOLAMIDE 30242287,20504258,25918017 62070 42361 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR TANSHINONE IIA TANSHINONE IIA 62071 42362 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE BioE-743 62072 42363 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME 2,4-DINITROPHENOL 2,4-DINITROPHENOL 62073 42364 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 atazanavir ATAZANAVIR 22394315 62076 42365 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CCT128930 CHEMBL263664 21191045 62077 42366 GGH 8836 PROTEASE, ENZYME, DRUGGABLE GENOME THIOGUANINE THIOGUANINE 16041371 62079 42367 XPO1 7514 CLINICALLY ACTIONABLE, KINASE GONIOTHALAMIN GONIOTHALAMIN 20381347 62080 42368 TUBB2A 7280 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 62081 42369 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor PF-4691502 PF-04691502 62082 42370 POLB 5423 DNA REPAIR, DRUGGABLE GENOME EUPAFOLIN EUPAFOLIN 62083 42371 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME ROEMERINE ROEMERINE 62084 42372 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565826 62087 42373 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NILUTAMIDE NILUTAMIDE 22931300 62088 42374 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 310264754 OMIPALISIB 62090 42375 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650903 RISPERIDONE 62091 42376 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR CYT006-ANGQB CYT006-ANGQB 62092 42377 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL19 METHAZOLAMIDE 62093 42378 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Ureido-phenyl-substituted triazine derivative 1 62094 42379 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor PX-866 SONOLISIB 62095 42380 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL519504 ALEGLITAZAR 62096 42381 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE N/A 28351930,26785607 62098 42382 FAAH 2166 ENZYME, DRUGGABLE GENOME Aryl urea derivative 5 62099 42383 PLD2 5338 ENZYME, DRUGGABLE GENOME activator 135651544 62100 42384 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TRETINOIN TRETINOIN 62101 42385 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FENOFIBRATE FENOFIBRATE 22931300 62103 42386 PRKG1 5592 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 178101945 62105 42387 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SURAMIN HEXASODIUM SURAMIN HEXASODIUM 62106 42388 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BIOALLETHRIN S-CYCLOPENTENYL ISOMER BIOALLETHRIN S-CYCLOPENTENYL ISOMER 62107 42389 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR ETOPOSIDE ETOPOSIDE 12644023 62108 42390 IMPDH2 3615 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL727 THIOGUANINE 62110 42391 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX antagonist CHEMBL3545173 IRX4310 62112 42392 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME GW843682X GW843682X 62113 42393 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR METHADONE METHADONE 18182069 62114 42394 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Forasartan FORASARTAN 62115 42395 ETV1 2115 DRUG RESISTANCE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRAMETINIB TRAMETINIB 28178529 62116 42396 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CODEINE CODEINE 62119 42397 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR RABEPRAZOLE RABEPRAZOLE 16815316 62120 42398 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE DASATINIB DASATINIB 62121 42399 HDAC11 79885 DRUGGABLE GENOME, ENZYME BML-210 CHEMBL324053 16921367 62122 42400 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Phenylpyrrolidinone derivative 3 62123 42401 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AZACITIDINE AZACITIDINE 62124 42402 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 5,7,2'-TRIHYDROXYFLAVONE CHEMBL242385 62127 42403 AQP1 358 ION CHANNEL, DRUGGABLE GENOME ACETAZOLAMIDE ACETAZOLAMIDE 12147198 62128 42404 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3545207 EVENAMIDE 62129 42405 CDH2 1000 CELL SURFACE, DRUGGABLE GENOME methadone METHADONE 62130 42406 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PWT33597 62131 42407 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102713 62132 42408 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774824-Compound-Figure9Example2up 62134 42409 SSRP1 6749 KINASE, DNA REPAIR CBL0137 62135 42410 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tacrine-caffeic acid hybrid derivative 2 62136 42411 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE AURIN AURIN 62137 42412 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME HEXAMETHYLENE BISACETAMIDE 3856429 62138 42413 TSPO 706 DRUGGABLE GENOME Iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivative 2 62141 42414 TUBB6 84617 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 62145 42415 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651238 TEGASEROD 62146 42416 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417147 CHEMBL2094484 62147 42417 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-2893 CHEMBL312032 62149 42418 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER cyclophosphamide CYCLOPHOSPHAMIDE 19696793 62152 42419 CAMK1D 57118 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 62156 42420 ABCC9 10060 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER Glimepiride GLIMEPIRIDE 62157 42421 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME HOMIDIUM BROMIDE HOMIDIUM BROMIDE 62158 42422 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1659 CHLORPHENIRAMINE MALEATE 62160 42423 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR PMX-60056 DELPARANTAG 22315264 62164 42424 HPSE 10855 ENZYME, DRUGGABLE GENOME PG-545 62165 42425 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Pyrimidine derivative 19 62168 42426 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1716 CYPROHEPTADINE HYDROCHLORIDE 62169 42427 ALOX15 246 ENZYME, DRUGGABLE GENOME FENTICLOR FENTICLOR 62170 42428 P4HB 5034 THIOREDOXIN, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2105662 LOMITAPIDE MESYLATE 62171 42429 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SELEXIPAG SELEXIPAG 62172 42430 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL843 ROSIGLITAZONE MALEATE 62175 42431 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE paclitaxel PACLITAXEL 26033044 62176 42432 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1692 IMIPRAMINE HYDROCHLORIDE 62177 42433 RAPGEF3 10411 ENZYME inhibitor 249565600 62181 42434 MAOB 4129 DRUGGABLE GENOME, ENZYME 8-[(3-TRIFLUOROMETHYL)BENZYLOXY]CAFFEINE CHEMBL602466 20093036 62184 42435 APOE 348 DRUGGABLE GENOME pravastatin PRAVASTATIN 19667110,17289397 62188 42436 PTHLH 5744 HORMONE ACTIVITY, DRUGGABLE GENOME VINBLASTINE VINBLASTINE 9784008 62189 42437 LNPEP 4012 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, TRANSPORTER, PROTEASE inhibitor 252166866 62190 42438 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE V3381 INDANTADOL 62191 42439 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3545284 CERDULATINIB 62192 42440 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE OXALIPLATIN OXALIPLATIN 25072261 62193 42441 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL197672 EMRICASAN 62194 42442 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FENRETINIDE FENRETINIDE 62196 42443 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102657 SELICICLIB 62197 42444 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Veltuzumab subcutaneous 62198 42445 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ASP5878 62199 42446 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CP-55940 CP-55940 62200 42447 APC 324 CLINICALLY ACTIONABLE TASIN-1 27798265 62201 42448 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE MLN0128 SAPANISERTIB 26574479 62203 42449 NCOR2 9612 NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BENZBROMARONE BENZBROMARONE 62204 42450 SMN2 6607 DRUGGABLE GENOME NECROSTATIN NECROSTATIN 62205 42451 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101545 62206 42452 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL2105704 LENVATINIB MESYLATE 62207 42453 MAPT 4137 DRUGGABLE GENOME DNDI1417111 CHEMBL2094456 62210 42454 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 135650039 62213 42455 NDUFB9 4715 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 62214 42456 HAS3 3038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME RETINOIC ACID 10772242 62215 42457 LTA 4049 DRUGGABLE GENOME Anti-LT alpha 62216 42458 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 187051844 OLODATEROL 62217 42459 USP1 7398 DNA REPAIR, PROTEASE, ENZYME BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 62218 42460 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 310264705 PITOLISANT 62219 42461 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Temsirolimus TEMSIROLIMUS 24470557 62223 42462 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME JNJ-40346527 EDICOTINIB 62224 42463 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 252166517 TUCIDINOSTAT 62226 42464 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor CHEMBL3301610 ABEMACICLIB 62227 42465 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 135650917 62230 42466 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUTICASONE PROPIONATE 62231 42467 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FR-901464 CHEMBL494107 17643111 62232 42468 BAZ2B 29994 NA INDIRUBIN SULFATE SU-9516 62234 42469 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUTAMIDE FLUTAMIDE 26000489 62235 42470 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FTORMETAZINE FTORMETAZINE 62236 42471 CHI3L1 1116 CELL SURFACE, DRUGGABLE GENOME ANTI-INFLAMMATORY DRUGS 16035398 62237 42472 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR SB-203580 SB-203580 62238 42473 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 7,8-DIHYDROXYFLAVONE 7,8-DIHYDROXYFLAVONE 62239 42474 GMNN 51053 DRUGGABLE GENOME SARPOGRELATE SARPOGRELATE 62240 42475 GSTM1 2944 DRUGGABLE GENOME, ENZYME ANTICONVULSANT 12499585 62241 42476 BAZ2B 29994 NA CLOTRIMAZOLE CLOTRIMAZOLE 62242 42477 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME KENPAULLONE KENPAULLONE 62246 42478 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL CROMOGLICATE CROMOLYN 62247 42479 HTT 3064 DRUGGABLE GENOME SJ000114740 CHEMBL592068 62248 42480 AKR1B10 57016 DRUGGABLE GENOME, ENZYME URSOLIC ACID URSOLIC ACID 21561086 62249 42481 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME olanzapine OLANZAPINE 23559402 62250 42482 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE AZACYTIDINE AZACITIDINE 10209960 62251 42483 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE SB-415286 CHEMBL322970 62252 42484 HTT 3064 DRUGGABLE GENOME BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE BIS(DIMETHYLAMINETHIOCARBONYL)MONOSULFIDE 62253 42485 BAZ2B 29994 NA SJ000044511 CHEMBL592124 62255 42486 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHYL ABIETATE METHYL ABIETATE 62256 42487 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545002 MP-412 62258 42488 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR URIDINE URIDINE 10712415 62259 42489 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TECTOQUINONE TECTOQUINONE 62261 42490 EGLN3 112399 DRUGGABLE GENOME, ENZYME FG-4592 ROXADUSTAT 62262 42491 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME NS-018 NS-018 62263 42492 ADGRV1 84059 G PROTEIN COUPLED RECEPTOR, TRANSPORTER, CELL SURFACE, KINASE, DRUGGABLE GENOME opioids 62264 42493 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CLENBUTEROL CLENBUTEROL 62266 42494 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 223366074 BRIGATINIB 62269 42495 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CARBACHOL CARBACHOL 62270 42496 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL3544908 AZATADINE MALEATE 62271 42497 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME CATECHOL CATECHOL 62272 42498 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ANISOMYCIN ANISOMYCIN 62275 42499 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 1540545 CHEMBL259784 62276 42500 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE AXITINIB AXITINIB 25686603 62278 42501 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER HDM201 62279 42502 UBE2N 7334 ENZYME, DRUGGABLE GENOME ASN06356088 ASN06356088 62280 42503 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE XL228 XL-228 62281 42504 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR inhibitor 318164851 62286 42505 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33a 62287 42506 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SERTRALINE HYDROCHLORIDE SERTRALINE HYDROCHLORIDE 62288 42507 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MELENGESTROL ACETATE MELENGESTROL ACETATE 62289 42508 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ETHANOL ALCOHOL 15242787,9756045 62290 42509 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME LEVOTHYROXINE LEVOTHYROXINE 62292 42510 GMNN 51053 DRUGGABLE GENOME CHOLECALCIFEROL CHOLECALCIFEROL 62293 42511 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4-PHENOXYPHENOL CHEMBL224318 62294 42512 LY96 23643 DRUGGABLE GENOME agonist 315661222 62295 42513 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PF-05280014 62296 42514 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE oxymetazoline and tetracaine 62298 42515 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME CARFILZOMIB CARFILZOMIB 24524217 62299 42516 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE BOLDINE BOLDINE 62300 42517 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLOFOCTOL CLOFOCTOL 62302 42518 PSMC2 5701 PROTEASE, TRANSCRIPTION FACTOR inhibitor CHEMBL451887 CARFILZOMIB 62303 42519 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME TRAMETINIB TRAMETINIB 24569458 62304 42520 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Ribociclib RIBOCICLIB 62305 42521 EHMT1 79813 ENZYME, DRUGGABLE GENOME inhibitor 178103596 62307 42522 CBLB 868 CLINICALLY ACTIONABLE, ENZYME Fasudil FASUDIL 26177294 62310 42523 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME cyclophosphamide CYCLOPHOSPHAMIDE 62311 42524 RGS4 5999 DRUGGABLE GENOME PROCATEROL PROCATEROL 62314 42525 EYA2 2139 DNA REPAIR NSC-119915 CHEMBL1481974 62315 42526 MMP7 4316 NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166829 62316 42527 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME TACEDINALINE TACEDINALINE 18692397 62320 42528 PTGS1 5742 ENZYME, DRUGGABLE GENOME ibuprofen IBUPROFEN 25502615 62322 42529 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR SORAFENIB SORAFENIB 62325 42530 PDE4B 5142 DRUGGABLE GENOME, ENZYME ROFLUMILAST ROFLUMILAST 62326 42531 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CUCURBITACIN D CUCURBITACIN D 25756299 62327 42532 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CHEMBL681 ETOMIDATE 62328 42533 ITPR2 3709 ION CHANNEL, DRUGGABLE GENOME activator 178101039 62331 42534 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545052 FIMEPINOSTAT 62332 42535 MAPT 4137 DRUGGABLE GENOME R-N-PROPYLNORAPOMORPHINE R-N-PROPYLNORAPOMORPHINE 62333 42536 TFF3 7033 DRUGGABLE GENOME AMINOGLUTETHIMIDE AMINOGLUTETHIMIDE 25900183 62334 42537 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME CEP-32496 CEP-32496 22319199 62335 42538 FAAH2 158584 DRUGGABLE GENOME, ENZYME inhibitor 178101156 URB-597 62337 42539 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102247 ST1535 62340 42540 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL PMID28051882-Compound-XIV 62342 42541 COL18A1 80781 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 62344 42542 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ZK-164015 CHEMBL184074 62345 42543 ATAD5 79915 NA TCMDC-125630 CHEMBL548619 62346 42544 PSMA2 5683 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL2103884 OPROZOMIB 62348 42545 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor SORAFENIB SORAFENIB 62350 42546 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NISOLDIPINE NISOLDIPINE 62351 42547 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME 2-MERCAPTOBENZOTHIAZOLE 2-MERCAPTOBENZOTHIAZOLE 62352 42548 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor BYL719 ALPELISIB 62353 42549 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 varenicline VARENICLINE 25588294 62354 42550 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178100734 62355 42551 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 4-(HEXYLOXY)PHENOL CHEMBL225563 62356 42552 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 4-(4-AMINOPHENYL)BUTANOIC ACID CHEMBL1650245 24044874 62357 42553 ST14 6768 ENZYME, DRUGGABLE GENOME, PROTEASE PROTEASE INHIBITOR 10373425 62359 42554 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 2-(STYRYL)-BENZIMIDAZOLE CHEMBL473721 62360 42555 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 178101239 62362 42556 CA2 760 DRUGGABLE GENOME, ENZYME Dorzolamide DORZOLAMIDE 62363 42557 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHENYLHYDRAZINE PHENYLHYDRAZINE 62364 42558 PRPF31 26121 NA metformin METFORMIN 29650774 62366 42559 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor 178103723 CILOSTAZOL 62368 42560 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor REGORAFENIB REGORAFENIB 62369 42561 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-95397 CHEMBL429095 62370 42562 APC 324 CLINICALLY ACTIONABLE iCRT-5 21393571 62374 42563 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR TAE-684 TAE-684 62375 42564 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL501867 VINCRISTINE SULFATE 62376 42565 PTGS1 5742 ENZYME, DRUGGABLE GENOME Piroxicam PIROXICAM 62377 42566 MAPT 4137 DRUGGABLE GENOME BISANHYDRORUTILANTINONE BISANHYDRORUTILANTINONE 62378 42567 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Diaminopyridine analog 4 62379 42568 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CVX-045 62381 42569 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME INCB039110 ITACITINIB 62382 42570 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL284671 CODEINE SULFATE 62384 42571 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-33 62385 42572 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Hydrocortamate HYDROCORTAMATE 62386 42573 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist ZIBOTENTAN ZIBOTENTAN 62388 42574 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SILIBININ SILIBININ 62390 42575 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL1980297 ILORASERTIB 62391 42576 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1522 ESZOPICLONE 62392 42577 DDC 1644 ENZYME, DRUGGABLE GENOME Vitamin B6 62394 42578 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE prednisone PREDNISONE 27173875 62395 42579 USP1 7398 DNA REPAIR, PROTEASE, ENZYME JUGLONE JUGLONE 62396 42580 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME CAMPTOTHECIN CAMPTOTHECIN 62398 42581 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Gefitinib GEFITINIB 26124204 62400 42582 POLK 51426 DNA REPAIR, ENZYME HOMIDIUM HOMIDIUM 62401 42583 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SB-224289 SB-224289 62403 42584 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MICONAZOLE MICONAZOLE 62404 42585 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102572 62405 42586 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR PD-0325901 PD-0325901 23398453,25766633 62406 42587 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE paclitaxel PACLITAXEL 23963862 62407 42588 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DIPYRIDAMOLE DIPYRIDAMOLE 62408 42589 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 178102550 62411 42590 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Antibodie derivative 11 62412 42591 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor XL-765 VOXTALISIB 62414 42592 GAPDH 2597 DRUGGABLE GENOME, ENZYME GALLIC ACID GALLIC ACID 62415 42593 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ETHYNODIOL DIACETATE 62416 42594 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200787 PHENOXYBENZAMINE HYDROCHLORIDE 62417 42595 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE BENZO[B]FLUORANTHENE BENZO[B]FLUORANTHENE 62418 42596 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE M3814 NEDISERTIB 62420 42597 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL61780 TEZOSENTAN 62423 42598 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AZD4547 27550940,26351323,22837387,27401245,28034880,22869148,26992226,28108151,25589496 62425 42599 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUPREDNISOLONE FLUPREDNISOLONE 62426 42600 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Ragaglitazar RAGAGLITAZAR 62430 42601 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1549 CHEMBL227959 62433 42602 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER levofloxacin LEVOFLOXACIN 62434 42603 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE RG-1530 RG-1530 62436 42604 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AVOSENTAN AVOSENTAN 62440 42605 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-144 62444 42606 MAPT 4137 DRUGGABLE GENOME TRIMETREXATE TRIMETREXATE 62447 42607 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CRYPTOTANSHINONE CRYPTOTANSHINONE 62449 42608 IHH 3549 PROTEASE, DRUGGABLE GENOME TGFBETA1 9112395 62451 42609 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200631 62452 42610 NDUFV1 4723 ENZYME inhibitor CHEMBL3545320 ME-344 62454 42611 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SINENSETIN SINENSETIN 62455 42612 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MLN0128 SAPANISERTIB 26272063,26574479 62457 42613 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178103661 HYDROMORPHONE 62458 42614 GSTA1 2938 ENZYME, DRUGGABLE GENOME cisplatin CISPLATIN 22188361 62459 42615 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650378 ILOPROST 62461 42616 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PICTILISIB PICTILISIB 22802530 62462 42617 SH2B1 25970 KINASE aripiprazole ARIPIPRAZOLE 28694205 62463 42618 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ISOCONAZOLE ISOCONAZOLE 62465 42619 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Platinum compounds 19203783,27498158 62467 42620 TMEM97 27346 NA PMID28051882-Compound-Figure9 62468 42621 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HARPAGOSIDE HARPAGOSIDE 62469 42622 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201546 INSULIN ZINC SUSP PURIFIED BEEF 62470 42623 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Fluorinated compound 1 62472 42624 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME SILIBININ SILIBININ 62474 42625 SMARCA4 6597 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING VINORELBINE VINORELBINE 26671993 62475 42626 CRLF2 64109 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME RUXOLITINIB RUXOLITINIB 22955920 62476 42627 HSPB1 3315 DRUGGABLE GENOME CRIDANIMOD CRIDANIMOD 62479 42628 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME interferon beta-1a 27020477 62480 42629 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL3545224 BURIXAFOR 62482 42630 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TIRATRICOL TIRATRICOL 62483 42631 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Oblimersen OBLIMERSEN 62484 42632 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE IDAZOXAN IDAZOXAN 62485 42633 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER antineoplastic agents 19786980,22188361,18357466,20638924,26696550,19052714 62486 42634 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME T091317 T091317 22579484,18800767,24480357,24268541 62487 42635 EML4 27436 CLINICALLY ACTIONABLE, KINASE X-376 21613408 62488 42636 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR docetaxel DOCETAXEL 62490 42637 BAZ2B 29994 NA PEFLOXACINE MESYLATE PEFLOXACIN MESYLATE 62491 42638 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHAETOCIN CHAETOCIN 62493 42639 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Abemaciclib ABEMACICLIB 62496 42640 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RAD-140 RAD-140 62497 42641 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 178102681 WORTMANNIN 62498 42642 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CARBOPLATIN CARBOPLATIN 62499 42643 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 249565724 62502 42644 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY AMINOGLYCOSIDES 4064470 62503 42645 GMNN 51053 DRUGGABLE GENOME TCMDC-123951 CHEMBL587849 62504 42646 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL227529 ALOGLIPTIN BENZOATE 62505 42647 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR AZA 8635147 62506 42648 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ASPIRIN ASPIRIN 15381054 62508 42649 CTH 1491 ENZYME inhibitor 178101931 62509 42650 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME 3144 28235199 62510 42651 BAZ2B 29994 NA SJ000113372 CHEMBL589912 62511 42652 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME GNF-PF-5151 CHEMBL576208 62512 42653 BAZ2B 29994 NA ACID BLUE 129 ACID BLUE 129 62513 42654 LNPEP 4012 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, TRANSPORTER, PROTEASE inhibitor 252166822 62514 42655 RCE1 9986 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 252166780 62516 42656 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135650216 62517 42657 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102600 62519 42658 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-3889 CHEMBL598270 62521 42659 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AG-34 CHEMBL80155 62525 42660 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL571 KETOPROFEN 62526 42661 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE 3'-NORSPONGIOLACTONE CHEMBL1078000 19601607 62527 42662 ALB 213 TRANSPORTER, DRUGGABLE GENOME NAPROXEN NAPROXEN 10682387 62533 42663 TLR7 51284 DRUGGABLE GENOME IMO-3100 62534 42664 POLK 51426 DNA REPAIR, ENZYME ROSE BENGAL ROSE BENGAL 62535 42665 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 223366014 62538 42666 APC 324 CLINICALLY ACTIONABLE Regorafenib REGORAFENIB 27004155 62541 42667 COP1 64326 CLINICALLY ACTIONABLE, ENZYME Propafenone PROPAFENONE 62542 42668 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRICLOCARBAN TRICLOCARBAN 62543 42669 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DOCETAXEL DOCETAXEL 30807645 62546 42670 SFTPA1 653509 DRUGGABLE GENOME TRICHOSTATIN A 11948134 62547 42671 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1653 PHENIRAMINE MALEATE 62548 42672 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME QUINALPHOS QUINALPHOS 62553 42673 CPB1 1360 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166824 62554 42674 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME 178101232 62555 42675 BAZ2B 29994 NA 2-PICOLINIC ACID 2-PICOLINIC ACID 62556 42676 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor AEE 788 62557 42677 DOT1L 84444 CLINICALLY ACTIONABLE, DNA REPAIR, METHYL TRANSFERASE, DRUGGABLE GENOME, ENZYME inhibitor 178103598 PINOMETOSTAT 62558 42678 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GBR-12935 CHEMBL26320 62560 42679 CHRNA5 1138 DRUGGABLE GENOME, ION CHANNEL antagonist 178100808 62561 42680 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE DOVITINIB DOVITINIB 62562 42681 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ANTICONVULSANT 15044076 62563 42682 NCOA1 8648 ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX tamoxifen TAMOXIFEN 22174377 62564 42683 EREG 2069 KINASE, GROWTH FACTOR, DRUGGABLE GENOME HUMAN CHORIONIC GONADOTROPIN 16543407 62565 42684 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 178103418 ENZALUTAMIDE 62566 42685 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR ETOPOSIDE ETOPOSIDE 9044846 62567 42686 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL MEM 1003 62569 42687 NOS2 4843 DRUGGABLE GENOME, ENZYME MPL-S 62571 42688 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Isoquinoline 1,3-dione derivative 1 62572 42689 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BEZ 235 62573 42690 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 11 62575 42691 ALDH5A1 7915 DRUGGABLE GENOME, ENZYME inhibitor 252827498 CHEMBL378577 62576 42692 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE ROGARATINIB ROGARATINIB 30807645 62577 42693 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417548 CHEMBL2094789 62578 42694 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BEZ235 DACTOLISIB 26270481 62579 42695 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200478 DYCLONINE HYDROCHLORIDE 62586 42696 SLC38A4 55089 TRANSPORTER 178101264 62589 42697 NRP1 8829 DRUGGABLE GENOME ANTI-NRP1 MAB 62592 42698 ATXN2 6311 NA AURIN AURIN 62595 42699 IMPDH2 3615 DRUGGABLE GENOME, ENZYME MYCOPHENOLIC ACID 62597 42700 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE INTERLEUKIN-8 11956101 62599 42701 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OBP-801 OBP-801 62600 42702 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TRIPROLIDINE TRIPROLIDINE 62602 42703 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR FAA 8512819 62603 42704 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-710 CHEMBL596839 62607 42705 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME VITAMIN E 10836612,12057767 62609 42706 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IMETIT IMETIT 62610 42707 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE losartan LOSARTAN 18695978 62611 42708 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-A11 62613 42709 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 135651534 62615 42710 LAP3 51056 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2103847 TOSEDOSTAT 62616 42711 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX ADAPALENE ADAPALENE 62618 42712 CYP51A1 1595 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME FLUCONAZOLE FLUCONAZOLE 12116245 62619 42713 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY AMINOGLUTETHIMIDE AMINOGLUTETHIMIDE 3781413 62620 42714 DDC 1644 ENZYME, DRUGGABLE GENOME ProSavin 62621 42715 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IMIPRAMINE IMIPRAMINE 22931300 62622 42716 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-108783 CHEMBL1489812 62624 42717 PTPRM 5797 DRUGGABLE GENOME, PROTEIN PHOSPHATASE inhibitor 252827513 62625 42718 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR EMETINE DIHYDROCHLORIDE EMETINE HYDROCHLORIDE 62626 42719 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE RAPAMYCIN SIROLIMUS 16027121 62627 42720 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ZINC SULFATE 15715661 62628 42721 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE PENTAZOCINE PENTAZOCINE 62629 42722 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER GW305074X GW305074X 62630 42723 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME O-DEMETHYLATED ADAPALENE O-DEMETHYLATED ADAPALENE 62631 42724 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL3545052 FIMEPINOSTAT 62632 42725 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME SKI-758 CHEMBL219557 62633 42726 POLB 5423 DNA REPAIR, DRUGGABLE GENOME IDARUBICIN IDARUBICIN 62634 42727 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE inhibitor 404859110 62638 42728 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 1-(4-HYDROXYPHENYL)MALEIMIDE CHEMBL565893 62639 42729 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE KN035 ENVAFOLIMAB 62640 42730 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE ESTRONE ESTRONE 12520970,12567859 62641 42731 CYB5R3 1727 DRUGGABLE GENOME, ENZYME rasburicase RASBURICASE 62642 42732 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE RUBITECAN RUBITECAN 62643 42733 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CI-1033 CANERTINIB 62644 42734 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE THIABENDAZOLE THIABENDAZOLE 62645 42735 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-50 62647 42736 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME SOLIFENACIN SOLIFENACIN 62649 42737 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor NMS-1286937 NMS-1286937 62650 42738 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID28048944-Compound-19 62651 42739 PAH 5053 DRUGGABLE GENOME, ENZYME HepaStem 62652 42740 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR neratinib NERATINIB 62653 42741 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HEXACHLOROPHENE HEXACHLOROPHENE 62654 42742 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417213 CHEMBL2094532 62655 42743 DDRGK1 65992 NUCLEAR HORMONE RECEPTOR azathioprine AZATHIOPRINE 21961091 62657 42744 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Iloperidone ILOPERIDONE 62658 42745 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20100022547C81 62660 42746 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DACETUZUMAB DACETUZUMAB 62661 42747 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102684 CLEMASTINE 62662 42748 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-3 62663 42749 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME BELINOSTAT BELINOSTAT 62664 42750 TRPC4 7223 ION CHANNEL, KINASE, DRUGGABLE GENOME, CELL SURFACE blocker,activator 135652740 62665 42751 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651390 62666 42752 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME GM6001 62668 42753 TUBA4A 7277 DRUGGABLE GENOME ABT-751 ABT-751 25468039 62670 42754 MAOB 4129 DRUGGABLE GENOME, ENZYME EVT-302 62671 42755 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TRIDIHEXETHYL TRIDIHEXETHYL 62675 42756 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1090089 PAMAPIMOD 62676 42757 TAC1 6863 DRUGGABLE GENOME OMEPRAZOLE OMEPRAZOLE 15684503,16259735 62677 42758 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor AZD8931 SAPITINIB 62678 42759 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR HOMIDIUM HOMIDIUM 62679 42760 MAPT 4137 DRUGGABLE GENOME L-755507 L-755507 62682 42761 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist 178100976 SELFOTEL 62683 42762 SLC15A1 6564 DRUGGABLE GENOME, TRANSPORTER inhibitor 329968426 62684 42763 E2F1 1869 TRANSCRIPTION FACTOR CISPLATIN CISPLATIN 16849574 62685 42764 PSMD8 5714 NA inhibitor CARFILZOMIB CARFILZOMIB 62686 42765 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME TESTOSTERONE TESTOSTERONE 10630892 62687 42766 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE REBASTINIB REBASTINIB 62691 42767 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE MYOCELL SDF-1 62692 42768 MSH2 4436 CLINICALLY ACTIONABLE, DNA REPAIR DURVALUMAB DURVALUMAB 26674132 62693 42769 CD74 972 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE Milatuzumab MILATUZUMAB 62694 42770 TNFRSF9 3604 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE antibody 315661319 UTOMILUMAB 62697 42771 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RO4987655 RO-4987655 26438159 62698 42772 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tetra-hydro-isoquinoline derivative 3 62699 42773 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PIMONIDAZOLE PIMONIDAZOLE 12829158 62701 42774 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DOCOSATETRA-7Z,10Z,13Z,16Z-ENOYL ETHANOLAMIDE CHEMBL321585 62703 42775 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 VANIPREVIR VANIPREVIR 19841155 62704 42776 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor BIBW 2992 62705 42777 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME IPILIMUMAB IPILIMUMAB 28351930 62706 42778 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL515966 EZLOPITANT 62707 42779 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator CHEMBL1201657 HEPARIN SODIUM 62710 42780 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102285 LINIFANIB 62714 42781 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor SB939 62715 42782 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102244 62716 42783 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME egfr inhibitors 26438111 62717 42784 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR allosteric modulator 310264748 62718 42785 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SIMVASTATIN SIMVASTATIN 62719 42786 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ENOXOLONE ENOXOLONE 22931300 62720 42787 MAPT 4137 DRUGGABLE GENOME CY-208243 CHEMBL313737 62721 42788 SMN1 6606 DRUGGABLE GENOME LEFLUNOMIDE LEFLUNOMIDE 62722 42789 PIP4K2A 5305 ENZYME, KINASE GNF-PF-1678 CHEMBL580340 62723 42790 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE GW843682X GW843682X 62724 42791 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Estrogen ESTROGEN 62726 42792 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER SCUTELLARIN SCUTELLARIN 22822035 62727 42793 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE tacrolimus TACROLIMUS 29318894,28316087 62728 42794 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR INDOLE-3-CARBINOL INDOLE-3-CARBINOL 16322316 62729 42795 TARDBP 23435 TUMOR SUPPRESSOR DNDI1417031 CHEMBL1333049 62731 42796 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 62733 42797 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL27759 ENTINOSTAT 62736 42798 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE trastuzumab emtansine 26920887 62740 42799 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE inhibitor CHEMBL1200686 PIMECROLIMUS 62741 42800 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIMETHYLAMINOETHANOL DIMETHYLAMINOETHANOL 62742 42801 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR peginterferon alfa-2a 62743 42802 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652274 62748 42803 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME NP-01 62749 42804 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 efavirenz EFAVIRENZ 16267764,15622315 62750 42805 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE ANTI-ERBB3 MONOCLONAL ANTIBODY AV-203 25542901 62751 42806 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE 2,3-DIDEOXYADENOSINE 3262616 62752 42807 PTGS2 5743 DRUGGABLE GENOME, ENZYME (Z)-16-NONADECENOIC ACID CHEMBL2171117 22822908 62756 42808 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Tipiracil TIPIRACIL 62757 42809 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL499 TIMOLOL 62758 42810 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 THIRAM THIRAM 62759 42811 KLRD1 3824 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME etanercept ETANERCEPT 26453102 62760 42812 DDC 1644 ENZYME, DRUGGABLE GENOME nicotine NICOTINE 16740595 62761 42813 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME sulfasalazine SULFASALAZINE 25303297 62762 42814 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ETRAVIRINE ETRAVIRINE 21189339 62763 42815 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor 252827519 62764 42816 CASP4 837 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 315661119 62765 42817 ATXN2 6311 NA GNF-PF-1947 CHEMBL585591 62768 42818 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ALPHA-NAPHTHOFLAVONE ALPHA-NAPHTHOFLAVONE 62770 42819 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EQUILIN EQUILIN 62771 42820 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME ALTISSIMACOUMARIN D ALTISSIMACOUMARIN D 22799262 62772 42821 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651239 62774 42822 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL9960 AZD-7624 62775 42823 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135651420 62776 42824 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody CETUXIMAB CETUXIMAB 62777 42825 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL1094 FELBAMATE 62778 42826 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PILOCARPINE PILOCARPINE 62780 42827 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 62781 42828 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE BAY-613606 CHEMBL541400 62782 42829 KDM4A 9682 DRUGGABLE GENOME, ENZYME LUTEOLIN LUTEOLIN 62783 42830 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE AM-101 ESKETAMINE HYDROCHLORIDE 62787 42831 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GARCINONE E GARCINONE E 62789 42832 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure2-Spirooliganone B 62790 42833 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FLOPROPIONE FLOPROPIONE 62791 42834 PTHLH 5744 HORMONE ACTIVITY, DRUGGABLE GENOME DIMETHYL SULFOXIDE 10839458 62794 42835 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-17 62796 42836 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200586 PRILOCAINE HYDROCHLORIDE 62797 42837 MLST8 64223 KINASE inhibitor OSI-027 OSI-027 62799 42838 TUBA3D 113457 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 62801 42839 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME KENPAULLONE KENPAULLONE 62802 42840 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE DOVITINIB DOVITINIB 62803 42841 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME OLAPARIB OLAPARIB 62804 42842 PDE4A 5141 DRUGGABLE GENOME, ENZYME E6005 LOTAMILAST 62805 42843 ADH1C 126 ENZYME, DRUGGABLE GENOME FOMEPIZOLE FOMEPIZOLE 62806 42844 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL940 GABAPENTIN 62808 42845 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 3-METHOXYCATECHOL 3-METHOXYCATECHOL 62809 42846 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DIENOCHLOR DIENOCHLOR 62811 42847 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125614 CHEMBL580609 62812 42848 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650824 PILOCARPINE 62814 42849 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ANILERIDINE ANILERIDINE 62815 42850 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 178102511 CABOZANTINIB 62816 42851 LEPR 3953 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME simvastatin SIMVASTATIN 18854995,14625131 62817 42852 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME ImMucin 62818 42853 BAZ2B 29994 NA CHLORAMBUCIL CHLORAMBUCIL 62819 42854 PSMB6 5694 DRUGGABLE GENOME, PROTEASE, ENZYME CARFILZOMIB CARFILZOMIB 24524217 62820 42855 TARDBP 23435 TUMOR SUPPRESSOR PRASTERONE PRASTERONE 62822 42856 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME PMID27998201-Compound-15 62823 42857 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GO-6976 GO-6976 62824 42858 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL1980297 ILORASERTIB 62826 42859 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL596 FENTANYL 62827 42860 PSMB7 5695 DRUGGABLE GENOME, PROTEASE CARFILZOMIB CARFILZOMIB 24524217 62828 42861 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Cyclohexyl-ethyl-substituted diaza and triaza-tricyclic compound 1 62831 42862 MAPT 4137 DRUGGABLE GENOME SEMAXANIB SEMAXANIB 62832 42863 SCNN1G 6340 ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AMILORIDE AMILORIDE 62833 42864 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME GOSSYPETIN GOSSYPETIN 62835 42865 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102410 62837 42866 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-123730 CHEMBL530280 62838 42867 EPHA1 2041 DRUGGABLE GENOME, KINASE, TYROSINE KINASE inhibitor 249565821 62840 42868 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE GSK683699 62841 42869 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Ponatinib PONATINIB 22238366,23908597,26048680 62844 42870 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GUAIFENESIN GUAIFENESIN 22931300 62845 42871 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ARASERTACONAZOLE ARASERTACONAZOLE 62846 42872 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 3 62848 42873 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 336446951 PF-06840003 62849 42874 CECR2 27443 NA inhibitor 310264732 62850 42875 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist 178100979 CLOMIPHENE 62851 42876 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME INCB24360 62852 42877 GAA 2548 DRUGGABLE GENOME, ENZYME DEOXYNOJIRIMYCIN DUVOGLUSTAT 62853 42878 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME IODOACETAMIDE IODOACETAMIDE 62856 42879 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Venetoclax VENETOCLAX 27520294 62858 42880 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE Methyl 2-amino-4-phenylthiophene-3-carboxylate 62860 42881 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Altiratinib ALTIRATINIB 62861 42882 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ELLIPTECINE ELLIPTECINE 62862 42883 LIPC 3990 ENZYME, PHOSPHOLIPASE, LIPASE, DRUGGABLE GENOME HEPARIN HEPARIN 4082106,3360217 62864 42884 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING HOLACANTHONE HOLACANTHONE 19199792 62867 42885 XPO1 7514 CLINICALLY ACTIONABLE, KINASE Drugs For Treatment Of Tuberculosis 30817003 62869 42886 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 252827426 62871 42887 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR CHR-3996 NANATINOSTAT 62872 42888 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Calcifediol CALCIFEDIOL 62874 42889 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Isoflavone derivative 5 62875 42890 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME ACY-1215 RICOLINOSTAT 26031917 62877 42891 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 2093195 CHEMBL411085 62878 42892 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL ETOMIDATE ETOMIDATE 16884293 62880 42893 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE US9695118, 8 62881 42894 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PYRITHIONE SODIUM PYRITHIONE SODIUM 62882 42895 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PENTAMIDINE ISETHIONATE PENTAMIDINE ISETHIONATE 62883 42896 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrrolo-pyridone derivative 2 62885 42897 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY SAR425899 SAR425899 62888 42898 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL270995 BRIVANIB ALANINATE 62889 42899 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Vortioxetine VORTIOXETINE 62895 42900 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE inhibitor 252827434 62898 42901 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MFGR1877S VOFATAMAB 62900 42902 GLS 2744 ENZYME SENNOSIDE B SENNOSIDE B 62901 42903 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE CLOSANTEL CLOSANTEL 62903 42904 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL1096380 PLINABULIN 62904 42905 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545324 RG-7666 62905 42906 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME RECOMBINANT INTERFERON BETA-1A 11412874 62906 42907 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME OCINAPLON OCINAPLON 62908 42908 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PAZOPANIB PAZOPANIB 25669829 62909 42909 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL1200757 PANCURONIUM BROMIDE 62911 42910 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR POTASSIUM DICHROMATE POTASSIUM DICHROMATE 62914 42911 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SOTRASTAURIN SOTRASTAURIN 62915 42912 NOS2 4843 DRUGGABLE GENOME, ENZYME inhibitor 178101827 PIMAGEDINE 62916 42913 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PRIDINOL METHANESULFONATE PRIDINOL METHANESULFONATE 62917 42914 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ROSIGLITAZONE ROSIGLITAZONE 62918 42915 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME EMBELIN EMBELIN 62920 42916 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 381118814 62921 42917 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 53801088 62922 42918 PSMB3 5691 PROTEASE, DRUGGABLE GENOME CARFILZOMIB CARFILZOMIB 24524217 62924 42919 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-4665 CHEMBL601744 62926 42920 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1743014 ETARACIZUMAB 62929 42921 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Chlorambucil CHLORAMBUCIL 25193512 62930 42922 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Solulin 62932 42923 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545082 RG-7376 62933 42924 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 223365926 BUTORPHANOL 62934 42925 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE CETUXIMAB CETUXIMAB 26046389 62935 42926 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BAY80-6946 COPANLISIB 62936 42927 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME SLV 306 62937 42928 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CETUXIMAB CETUXIMAB 62938 42929 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME DESOXYCORDIFOLINE DESOXYCORDIFOLINE 15568781 62939 42930 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR PROTEIN KINASE INHIBITOR 9133581 62940 42931 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 178101106 62941 42932 HBB 3043 DRUGGABLE GENOME, ENZYME SU-6656 CHEMBL605003 62942 42933 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL1946170 REGORAFENIB 62943 42934 TUBB 203068 DRUGGABLE GENOME 1069C 62944 42935 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ENILURACIL ENILURACIL 62947 42936 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME diclofenac acyl glucuronide 29203276 62948 42937 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table 6-15 62949 42938 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Osimertinib OSIMERTINIB 62953 42939 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME Long-acting erythropoietin conjugate 62954 42940 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE Iboctadekin + rituximab 62955 42941 TUBA3C 7278 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 62956 42942 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GLYCOPYRRONIUM BROMIDE 62957 42943 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE amodiaquine AMODIAQUINE 62958 42944 TARDBP 23435 TUMOR SUPPRESSOR CHRYSIN DIMETHYL ETHER CHRYSIN DIMETHYL ETHER 62960 42945 MAPT 4137 DRUGGABLE GENOME METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 62962 42946 ADH1A 124 DRUGGABLE GENOME acetaldehyde ACETALDEHYDE 31002879 62964 42947 GMNN 51053 DRUGGABLE GENOME TCMDC-125779 CHEMBL531451 62966 42948 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PI-103 PI-103 62968 42949 ATAD5 79915 NA CHLOROXINE CHLOROXINE 62969 42950 NTS 4922 DRUGGABLE GENOME CHLORPROMAZINE CHLORPROMAZINE 1980851 62971 42951 BIRC7 79444 PROTEASE INHIBITOR, TUMOR SUPPRESSOR, DRUG RESISTANCE CISPLATIN CISPLATIN 23188704 62973 42952 ATAD5 79915 NA SEW-03621 CHEMBL1271059 62974 42953 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650421 62975 42954 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME GO-6976 GO-6976 62976 42955 CAMKK2 10645 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE US9623028, Compound 79 62977 42956 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE CA4P 12171907 62979 42957 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 135651427 ADENOSINE DIPHOSPHATE 62981 42958 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Siponimod SIPONIMOD 62982 42959 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 KETOCONAZOLE KETOCONAZOLE 22931300 62985 42960 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME VITAMIN C 17573441 62986 42961 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LINOLEIC ACID LINOLEIC ACID 62987 42962 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE gliclazide GLICLAZIDE 62989 42963 RBP4 5950 DRUGGABLE GENOME A1-10438 62990 42964 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Ceritinib CERITINIB 28520527 62991 42965 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-WO2013082253 31 62993 42966 MAOA 4128 DRUGGABLE GENOME, ENZYME ISOCARBOXAZID ISOCARBOXAZID 62994 42967 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 363894179 62995 42968 NDUFA6 4700 ENZYME inhibitor CHEMBL3545135 NV-128 62997 42969 RGS4 5999 DRUGGABLE GENOME IPA-3 CHEMBL472940 62999 42970 ATAD5 79915 NA IDARUBICIN IDARUBICIN 63000 42971 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CYTOKINES 7540953 63002 42972 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE activator 404859009 63003 42973 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BROMETHALIN BROMETHALIN 63005 42974 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME AZIETOMIDATE AZIETOMIDATE 16884293 63006 42975 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME AZD-1080 AZD-1080 63007 42976 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME 1,6-naphyridine-4-ketone fused heterocyclic derivative 1 63010 42977 TOP2B 7155 DRUGGABLE GENOME, ENZYME BECATECARIN BECATECARIN 63012 42978 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE GLEEVEC IMATINIB 16630177 63013 42979 PDE4A 5141 DRUGGABLE GENOME, ENZYME GSK-356278 GSK-356278 63016 42980 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 249565896 SB-431542 63017 42981 ADRM1 11047 ENZYME inhibitor CHEMBL325041 BORTEZOMIB 63019 42982 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CELECOXIB CELECOXIB 30683736 63023 42983 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125620 CHEMBL530291 63024 42984 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME CLIOQUINOL CLIOQUINOL 63027 42985 SLC2A3 6515 DRUGGABLE GENOME, TRANSPORTER INSULIN INSULIN 12814351 63028 42986 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MOCLOBEMIDE MOCLOBEMIDE 63029 42987 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1200623 ETHYLESTRENOL 63030 42988 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME AZD-1080 AZD-1080 63031 42989 PTGS2 5743 DRUGGABLE GENOME, ENZYME NEPAFENAC NEPAFENAC 63032 42990 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL HU-308 CHEMBL497392 20346682 63033 42991 CA12 771 DRUGGABLE GENOME PHENOL PHENOL 63034 42992 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tetra-hydro-isoquinoline derivative 2 63035 42993 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE RG-1530 RG-1530 63037 42994 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PINDOLOL PINDOLOL 63039 42995 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor CHEMBL3544960 AT-13148 63041 42996 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650779 ASENAPINE 63043 42997 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ACETOCHLOR ACETOCHLOR 63051 42998 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MBX-2044 MBX-2044 63052 42999 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178101156 URB-597 63053 43000 TARDBP 23435 TUMOR SUPPRESSOR TRIADIMENOL TRIADIMENOL 63054 43001 CBX1 10951 NA CANTHARIDIC_ACID CANTHARIDIC_ACID 63055 43002 BUB1 699 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 315661212 63056 43003 SCTR 6344 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100608 63057 43004 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103416 DORZOLAMIDE 63058 43005 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545121 EPITINIB 63059 43006 BIRC7 79444 PROTEASE INHIBITOR, TUMOR SUPPRESSOR, DRUG RESISTANCE PMID25980951-Compound-6 63060 43007 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME CHLORISONDAMINE CHLORISONDAMINE 63061 43008 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE HISTONE DEACETYLASE INHIBITOR 17308065 63062 43009 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CVBT-141B 63063 43010 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME CISPLATIN CISPLATIN 16978399 63064 43011 DGAT1 8694 ENZYME, DRUGGABLE GENOME T863 63066 43012 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SER-101 63067 43013 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME N/A 63068 43014 USP1 7398 DNA REPAIR, PROTEASE, ENZYME REVERSETRIIODOTHYRONINE REVERSETRIIODOTHYRONINE 63069 43015 CCR7 1236 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR agonist 178100551 63070 43016 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME 3-phenyl-5-ureidoisothiazole-4-carboximide and 3-amino-5-phenylisothiazole derivative 1 63071 43017 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME BEZ235 DACTOLISIB 21831957 63072 43018 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652342 63074 43019 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AG-494 CHEMBL56731 63075 43020 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103726 CYCLIZINE 63076 43021 DHFR 1719 DRUGGABLE GENOME, ENZYME ANTIFOLATES 6487372 63077 43022 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE gemcitabine GEMCITABINE 21783417,22285168 63079 43023 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-130813 CHEMBL463783 63081 43024 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE AMB 12755626 63082 43025 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME AFLIBERCEPT AFLIBERCEPT 63085 43026 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor BAY80-6946 COPANLISIB 63086 43027 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000032081 CHEMBL590184 63087 43028 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME ERLOTINIB ERLOTINIB 22180495 63088 43029 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 252827389 63091 43030 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE CANTHIN-6-ONE CANTHIN-6-ONE 63092 43031 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ARACHIDONOYL GABA ARACHIDONOYL GABA 63093 43032 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Sunitinib SUNITINIB 63094 43033 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE CHEMBL256087 MENTHOL 63095 43034 TAC1 6863 DRUGGABLE GENOME ANTIHISTAMINE TERFENADINE 1696438 63096 43035 ALOX15B 247 DRUGGABLE GENOME, ENZYME 2',3'-DIHYDROXYFLAVONE CHEMBL242171 63097 43036 PTPRF 5792 DRUGGABLE GENOME, ENZYME, PROTEIN PHOSPHATASE inhibitor 252827428 63098 43037 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-125034 CHEMBL239439 63099 43038 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME antagonist 178104004 BIRINAPANT 63100 43039 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-15 63101 43040 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650585 METHOCTRAMINE 63103 43041 IFNG 3458 DRUGGABLE GENOME DHPG 2992368 63104 43042 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3545012 DSP-2230 63105 43043 APC 324 CLINICALLY ACTIONABLE G-631 26692561 63107 43044 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CLOXYQUIN CLOXYQUIN 63108 43045 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME BAY1161909 63110 43046 POLB 5423 DNA REPAIR, DRUGGABLE GENOME DEMECLOCYCLINE HYDROCHLORIDE DEMECLOCYCLINE HYDROCHLORIDE 63111 43047 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TAE-684 TAE-684 63112 43048 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER 6-THIOGUANINE THIOGUANINE 14643890 63113 43049 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL3545277 OMS405 63114 43050 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Cyclohexane carboxamide derivative 1 63115 43051 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BI-87E7 CHEMBL523200 63116 43052 GMNN 51053 DRUGGABLE GENOME AMINACRINE HYDROCHLORIDE AMINACRINE HYDROCHLORIDE 63117 43053 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ARA-C 17852453 63118 43054 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE MEHD-7945A DULIGOTUZUMAB 63119 43055 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE thalidomide THALIDOMIDE 26521987 63120 43056 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PROGESTERONE PROGESTERONE 22931300 63122 43057 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Varlitinib VARLITINIB 63123 43058 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-4798 CHEMBL584635 63124 43059 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE MORPHINE MORPHINE 63125 43060 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE (R)-NIPHATENONE A CHEMBL1946013 22148427 63126 43061 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DNQX DNQX 63127 43062 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-724440 CHEMBL515617 63128 43063 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIMETHISOQUIN HYDROCHLORIDE DIMETHISOQUIN HYDROCHLORIDE 63129 43064 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 252827519 63130 43065 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME LY-367385 CHEMBL94631 63131 43066 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME SGN-75 VORSETUZUMAB MAFODOTIN 63133 43067 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZAFIRLUKAST ZAFIRLUKAST 63135 43068 GMNN 51053 DRUGGABLE GENOME GNF-PF-3543 CHEMBL598679 63136 43069 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE activator 381118815 63137 43070 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL3545158 PEXIDARTINIB 63138 43071 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Insulin oral sublingual 63139 43072 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4057 CHEMBL598903 63140 43073 NOTCH2 4853 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE antibody REGN421 63141 43074 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor XL-765 VOXTALISIB 63142 43075 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 385612193 63143 43076 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 404859043 63146 43077 CES1 1066 DRUGGABLE GENOME, ENZYME GR148672X 63147 43078 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Levocabastine LEVOCABASTINE 63148 43079 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NORADRENALINE NOREPINEPHRINE BITARTRATE 63149 43080 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-N3 63150 43081 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE Trametinib TRAMETINIB 22733540 63151 43082 RAB9A 9367 ENZYME, DRUGGABLE GENOME ONONIN ONONIN 63153 43083 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE AEB071 SOTRASTAURIN 22653968,24141786,27507190 63154 43084 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE VATALANIB VATALANIB 63155 43085 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 4SC-202 DOMATINOSTAT 63158 43086 HPRT1 3251 DRUGGABLE GENOME, ENZYME 3TC LAMIVUDINE 17358033 63159 43087 MAPT 4137 DRUGGABLE GENOME ROTTLERIN ROTTLERIN 63160 43088 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE HALOFUGINONE HALOFUGINONE 16769768 63164 43089 SERPING1 710 DRUGGABLE GENOME, PROTEASE INHIBITOR Cinryze CINRYZE 63166 43090 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652271 63167 43091 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME RO-229735 CHEMBL2170369 21751815 63170 43092 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 375973268 63171 43093 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MYCOPHENOLIC ACID MYCOPHENOLIC ACID 63173 43094 LGALS1 3956 KINASE, DRUGGABLE GENOME US8703720, 15 63174 43095 HMGCR 3156 ENZYME, DRUGGABLE GENOME Poly-substituted miazine derivative 1 63176 43096 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME MMF MYCOPHENOLATE MOFETIL 14550820 63178 43097 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DEXAMETHASONE DEXAMETHASONE 22931300 63179 43098 BAZ2B 29994 NA OXYQUINOLINE OXYQUINOLINE 63180 43099 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3622820 ITACITINIB 63181 43100 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE partial agonist CHEMBL3544917 RAPASTINEL 63182 43101 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor PONATINIB PONATINIB 63183 43102 PRKAA2 5563 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME HL010183 CHEMBL2348411 23490148 63184 43103 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MURAGLITAZAR MURAGLITAZAR 63185 43104 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME DESMETHOXYYANGONIN DESMETHOXYYANGONIN 63187 43105 CSNK1G3 1456 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME PHA-767491 CHEMBL225519 63188 43106 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TAMOXIFEN TAMOXIFEN 20659801,16735120,20621492 63189 43107 KMO 8564 DRUGGABLE GENOME, ENZYME Benzene sulfonamide derivative 7 63190 43108 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SKIMMIANINE SKIMMIANINE 63191 43109 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE ABT-702 CHEMBL66089 63192 43110 HMGCR 3156 ENZYME, DRUGGABLE GENOME Lactol derivative 1 63193 43111 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL185 FLUOROURACIL 63194 43112 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME TAMATINIB R-406 63200 43113 CARM1 10498 ENZYME, METHYL TRANSFERASE, DRUGGABLE GENOME inhibitor 315661334 63201 43114 GMNN 51053 DRUGGABLE GENOME 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 63202 43115 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME N/A 24619759,26066800,22955918 63204 43116 MAPT 4137 DRUGGABLE GENOME QUERCETIN QUERCETIN 63205 43117 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL1289494 TIVOZANIB 63206 43118 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GO-6976 GO-6976 63208 43119 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NICOTINE NICOTINE 12851153 63209 43120 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 12-HYDROXY-4,4-BISNOR-4,8,11,13-PODOCARPATETRAEN-3-ONE 12-HYDROXY-4,4-BISNOR-4,8,11,13-PODOCARPATETRAEN-3-ONE 63210 43121 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME 340590272 63211 43122 ANO1 55107 ION CHANNEL blocker 135650269 63212 43123 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-2954 CHEMBL582722 63215 43124 TNFRSF11B 4982 DRUGGABLE GENOME anastrozole ANASTROZOLE 63216 43125 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PYRIDOSTIGMINE PYRIDOSTIGMINE 63218 43126 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 223366124 PACRITINIB 63219 43127 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISOBERGAPTENE ISOBERGAPTENE 63220 43128 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR FLURBIPROFEN FLURBIPROFEN 16531049 63224 43129 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ANASTROZOLE ANASTROZOLE 63225 43130 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME valsartan VALSARTAN 16678545 63227 43131 ATXN2 6311 NA PROPYLPYRAZOLETRIOL PROPYLPYRAZOLETRIOL 63228 43132 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Tricyclic pyrrolopyridine compound 1 63229 43133 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Piboserod PIBOSEROD 63230 43134 POLK 51426 DNA REPAIR, ENZYME DAPHNORIN DAPHNORIN 63231 43135 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR UVB 16598763 63236 43136 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178103086 63237 43137 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ANTI-EGFR MONOCLONAL ANTIBODY 23435830 63238 43138 SMOX 54498 ENZYME, DRUGGABLE GENOME ENZYME INHIBITOR 6885895 63239 43139 BAZ2B 29994 NA DNDI1417254 CHEMBL2094567 63241 43140 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CENISERTIB CENISERTIB 63242 43141 MAPT 4137 DRUGGABLE GENOME 4-HYDROXYESTRADIOL CHEMBL1412489 63243 43142 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 zafirlukast ZAFIRLUKAST 27377818 63244 43143 SLC7A11 23657 TRANSPORTER, DRUGGABLE GENOME, CELL SURFACE inhibitor 135650876 QUISQUALATE 63247 43144 XPO1 7514 CLINICALLY ACTIONABLE, KINASE inhibitor 375973224 SELINEXOR 63248 43145 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Rindopepimut RINDOPEPIMUT 63249 43146 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651407 63251 43147 RAMP2 10266 DRUGGABLE GENOME, CELL SURFACE agonist CHEMBL3833353 PRAMLINTIDE ACETATE 63252 43148 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PHENANTHROLINE PHENANTHROLINE 63253 43149 PSMA7 5688 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL325041 BORTEZOMIB 63254 43150 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME rivastigmine RIVASTIGMINE 18780301 63255 43151 SGSM3 27352 NA RG7304 63256 43152 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 63257 43153 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METIZOLINE METIZOLINE 63258 43154 POLI 11201 DNA REPAIR 3-HYDROXYANTHRANILIC ACID CHEMBL445304 63259 43155 PDE5A 8654 ENZYME, DRUGGABLE GENOME VARDENAFIL VARDENAFIL 63261 43156 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417621 CHEMBL1431017 63262 43157 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME IMD-0354 IMD-0354 63263 43158 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME lovastatin LOVASTATIN 63264 43159 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL142703 VILDAGLIPTIN 63269 43160 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR STAUROSPORINE STAUROSPORINE 63270 43161 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME ETHANOL ALCOHOL 10801782 63272 43162 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4516 CHEMBL586029 63274 43163 CD276 80381 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Enoblituzumab ENOBLITUZUMAB 63276 43164 GLA 2717 ENZYME, DRUGGABLE GENOME PRX-102 PEGUNIGALSIDASE ALFA 63277 43165 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Abicipar pegol 63278 43166 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER L-744,832 16224182 63279 43167 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-4046 CHEMBL600090 63281 43168 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-45382 CHEMBL1214274 63285 43169 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-31 63286 43170 ATXN2 6311 NA DNDI1417185 CHEMBL1549738 63287 43171 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125000 CHEMBL579742 63288 43172 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651266 TIOTROPIUM 63289 43173 HEBP1 50865 DRUGGABLE GENOME OT-551 OT-551 63291 43174 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 4-HYDROPEROXYCYCLOPHOSPHAMIDE PERFOSFAMIDE 9382956 63292 43175 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR antibody SILTUXIMAB SILTUXIMAB 63293 43176 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Romazarit ROMAZARIT 23515070 63294 43177 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-125653 CHEMBL580918 63295 43178 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME blocker 53801024 MICONAZOLE 63296 43179 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Olaparib OLAPARIB 26779812 63298 43180 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178101905 MARIMASTAT 63299 43181 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PHENOLPHTHALEIN PHENOLPHTHALEIN 63300 43182 DOT1L 84444 CLINICALLY ACTIONABLE, DNA REPAIR, METHYL TRANSFERASE, DRUGGABLE GENOME, ENZYME inhibitor 315661281 63303 43183 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE TAPENTADOL TAPENTADOL 63304 43184 TOP2B 7155 DRUGGABLE GENOME, ENZYME L-377202 L-377202 63305 43185 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR inhibitor 381118851 63306 43186 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE ENTRECTINIB ENTRECTINIB 63307 43187 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE A66 26137449,21668414 63309 43188 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 381118813 RUPATADINE 63311 43189 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE agonist 135649916 63312 43190 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 Cobicistat COBICISTAT 63313 43191 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME TOZASERTIB TOZASERTIB 63314 43192 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE NIRAPARIB NIRAPARIB 63315 43193 MPHOSPH8 54737 NA 6,7-ADTN HYDROBROMIDE CHEMBL1255656 63317 43194 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SPIRUCHOSTATIN C SPIRUCHOSTATIN C 21967146 63318 43195 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME blocker 178101108 PROCAINE 63319 43196 SLC28A2 9153 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME boceprevir BOCEPREVIR 25836019 63320 43197 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR URSODEOXYCHOLIC ACID 14747693 63321 43198 PDE11A 50940 DRUGGABLE GENOME, ENZYME inhibitor 178103872 TADALAFIL 63323 43199 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135652706 63324 43200 EPHB2 2048 KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME BVD-523 ULIXERTINIB 63325 43201 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME L-655708 CHEMBL52030 22137933 63326 43202 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-71 63327 43203 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME AZD6482 AZD-6482 26577700 63328 43204 CYP27A1 1593 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CHOLESTYRAMINE CHOLESTYRAMINE 12011083 63329 43205 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE SKI-O-703 63330 43206 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2142592 TALADEGIB 63331 43207 KLK4 9622 PROTEASE, DRUGGABLE GENOME, ENZYME Bortezomib BORTEZOMIB 63332 43208 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FLAVOXATE FLAVOXATE 63333 43209 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102536 63334 43210 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW770249X GW770249X 63335 43211 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE CISPLATIN CISPLATIN 63337 43212 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE LY2835219 ABEMACICLIB 63338 43213 USP1 7398 DNA REPAIR, PROTEASE, ENZYME MK-886 CHEMBL29097 63339 43214 KDM4A 9682 DRUGGABLE GENOME, ENZYME SANGUINARINE SULFATE SANGUINARINE SULFATE 63340 43215 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR TAK-441 TAK-441 24291104 63341 43216 SMN2 6607 DRUGGABLE GENOME GNF-PF-1000 CHEMBL600554 63342 43217 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-35 63343 43218 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL3707330 ROLAPITANT HYDROCHLORIDE 63344 43219 TSPO 706 DRUGGABLE GENOME Quinazoline derivative 2 63345 43220 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PMID27774822-Compound-Figure11Example5 63346 43221 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PMID25726713-Compound-51 63347 43222 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102550 63348 43223 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102445 TREPROSTINIL 63350 43224 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME cabozantinib CABOZANTINIB 27525386 63351 43225 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ATORVASTATIN ATORVASTATIN 17200431 63353 43226 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MENADIONE MENADIONE 63354 43227 CXCL8 3576 DRUGGABLE GENOME BIOSTIM 9304405 63356 43228 PDE8A 5151 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL628 PENTOXIFYLLINE 63357 43229 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650436 63358 43230 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PAZOPANIB PAZOPANIB 23786770 63359 43231 MAPT 4137 DRUGGABLE GENOME 1,2-DIPHENYLDISULFANE CHEMBL462861 63361 43232 RAPGEF3 10411 ENZYME GNF-PF-5061 CHEMBL601385 63362 43233 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651359 ZIPRASIDONE 63363 43234 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE BAS-0338868 CHEMBL378903 63364 43235 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Docetaxel DOCETAXEL 23200175,27876675,26125448,28492898 63365 43236 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CARMUSTINE CARMUSTINE 22931300 63366 43237 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PIMETHIXENE MALEATE PIMETHIXENE MALEATE 63369 43238 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist CHEMBL37676 APC-100 63370 43239 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PHENYLBUTYRYLHYDROXAMIC ACID PHENYLBUTYRYLHYDROXAMIC ACID 21874153 63372 43240 HTT 3064 DRUGGABLE GENOME PROMETHAZINE PROMETHAZINE 63373 43241 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME tenofovir TENOFOVIR 28462920 63375 43242 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE PD-0325901 PD-0325901 27821489 63376 43243 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650335 CHEMBL410478 63377 43244 ARG2 384 ENZYME Difluoromethylornithine 63378 43245 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE BEZ235 DACTOLISIB 23629727,24939055 63379 43246 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME SERTRALINE SERTRALINE 63381 43247 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME fluorouracil FLUOROURACIL 63383 43248 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor ORANTINIB ORANTINIB 63385 43249 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME PMID27539678-Compound-12 63387 43250 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL DIAZEPAM DIAZEPAM 63389 43251 NOD1 10392 CLINICALLY ACTIONABLE, DRUGGABLE GENOME TRACHEAL CYTOTOXIN TRACHEAL CYTOTOXIN 21341753 63390 43252 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TCMDC-123789 CHEMBL588859 63392 43253 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE STILONIUM IODIDE STILONIUM IODIDE 63394 43254 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL1236962 OMIPALISIB 63395 43255 MAPT 4137 DRUGGABLE GENOME MMV006389 CHEMBL586000 63396 43256 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102750 GALANIN 63399 43257 HNRNPC 3183 NA DABIGATRAN DABIGATRAN 22494098 63401 43258 ALOX15 246 ENZYME, DRUGGABLE GENOME AG-808 CHEMBL68534 63403 43259 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-68b 63405 43260 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE 3-(3-STIBONOPHENYL)PROPANOIC ACID CHEMBL2057662 22705189 63406 43261 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-EP20132578214 2 63407 43262 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME MK-8245 MK-8245 21661758 63409 43263 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL FLUDIAZEPAM FLUDIAZEPAM 63411 43264 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MEK162 BINIMETINIB 63412 43265 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL501867 VINCRISTINE SULFATE 63413 43266 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ALPROSTADIL ALPROSTADIL 22931300 63414 43267 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME DIPHENYLENEIODONIUM DIPHENYLENEIODONIUM 63415 43268 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TOPOTECAN HYDROCHLORIDE TOPOTECAN HYDROCHLORIDE 63416 43269 NDUFS6 4726 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 63417 43270 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 63418 43271 GJA1 2697 ION CHANNEL inhibitor 135652731 63419 43272 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE pertuzumab PERTUZUMAB 63421 43273 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME E319 E319 63422 43274 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-Eb 63423 43275 HEBP1 50865 DRUGGABLE GENOME Benzamide derivative 6 63424 43276 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Ponatinib PONATINIB 22238366 63426 43277 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Tiazofurin TIAZOFURIN 63428 43278 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651287 63432 43279 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL1615025 TAK-733 63433 43280 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL antagonist CHEMBL14935 TEZAMPANEL 63434 43281 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE AMG 145 63436 43282 TNNI2 7136 NA TIRAMSETIV 63437 43283 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 4-TRIETHYLGERMYLPHENOL 4-TRIETHYLGERMYLPHENOL 23214428 63438 43284 PGF 5228 GROWTH FACTOR, DRUGGABLE GENOME RO-5323441 TB-403 63441 43285 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 363894217 VORUCICLIB 63443 43286 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME 5,7-DIHYDROXYISOFLAVONE 5,7-DIHYDROXYISOFLAVONE 63445 43287 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME prednisone PREDNISONE 21228734 63446 43288 ABCA4 24 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME STARGEN 63448 43289 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR EPINEPHRINE EPINEPHRINE 63449 43290 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL904 DEXMETHYLPHENIDATE HYDROCHLORIDE 63450 43291 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 178101884 GSK-690693 63451 43292 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-45 63452 43293 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HARMINE HARMINE 63454 43294 CYBA 1535 TRANSPORTER doxorubicin DOXORUBICIN 19448608,28485375,21048526,16330681,25823784 63455 43295 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BMS-754807 BMS-754807 26561558 63456 43296 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR antagonist BIRINAPANT BIRINAPANT 63457 43297 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000294102 CHEMBL607309 63464 43298 PTHLH 5744 HORMONE ACTIVITY, DRUGGABLE GENOME inhibitor CHEMBL2109562 CAL 63465 43299 ATXN2 6311 NA TPCK TPCK 63466 43300 TSPO 706 DRUGGABLE GENOME DISULFIRAM DISULFIRAM 1320691 63468 43301 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME GEFITINIB GEFITINIB 63470 43302 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE PMID29130358-Compound-Figure13(4) 63471 43303 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor DACOMITINIB DACOMITINIB 63472 43304 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CINOLAZEPAM CINOLAZEPAM 63473 43305 TPBG 7162 CELL SURFACE, DRUGGABLE GENOME CV-9201 63474 43306 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CARBETOCIN CARBETOCIN 63475 43307 POLK 51426 DNA REPAIR, ENZYME XCT790 CHEMBL189753 63476 43308 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 63477 43309 ST13 6767 NA corticosteroids 25616159 63479 43310 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR paroxetine PAROXETINE 22965830,21338649,23733030,23619509,19236730,29748862,20016225 63480 43311 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME AT9283 AT-9283 63481 43312 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Triazole derivative 5 63483 43313 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE RO4987655 RO-4987655 26438159 63485 43314 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BCG BCG VACCINE 11359651 63486 43315 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DACTOLISIB DACTOLISIB 63487 43316 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE DASATINIB DASATINIB 63488 43317 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE KARENITECIN KARENITECIN 63489 43318 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME FLUOROURACIL FLUOROURACIL 25924824 63490 43319 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125142 CHEMBL528791 63493 43320 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 63494 43321 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135649719 63495 43322 DEGS1 8560 ENZYME inhibitor 178102663 63496 43323 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER cyclosporine CYCLOSPORINE 23922006,18334915,18444945,24088131,21806386,25536375,17206635,25240575,26107754,18576903,12966368,18717915,20030680,22886152 63498 43324 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME antagonist 223366066 GDC-0152 63499 43325 POLI 11201 DNA REPAIR PURPURIN PURPURIN 63500 43326 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TICLOPIDINE TICLOPIDINE 22931300 63501 43327 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME tipiracil hydrochloride 28992563 63502 43328 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME BIRB-796 DORAMAPIMOD 27154914 63503 43329 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 178102480 63506 43330 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME PMID27998201-Compound-8 63507 43331 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE GAMBOGIC ACID GAMBOGIC ACID 17911251 63508 43332 IDO2 169355 ENZYME 2,3-diamino-benzo[b]thiophene derivative 1 63510 43333 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652640 63512 43334 NOS2 4843 DRUGGABLE GENOME, ENZYME TYROSINE KINASE INHIBITORS 8579596 63513 43335 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774824-Compound-Figure3Example18 63514 43336 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ECHINATIN ECHINATIN 20022509 63515 43337 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME mycophenolic acid 24220207,22572835 63516 43338 RGS4 5999 DRUGGABLE GENOME D-LEUCINE D-LEUCINE 63517 43339 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE 178101778 63518 43340 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NANDROLONE NANDROLONE 63519 43341 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE THIOTEPA THIOTEPA 63520 43342 GMNN 51053 DRUGGABLE GENOME MMV085203 CHEMBL586031 63521 43343 GMNN 51053 DRUGGABLE GENOME CUMINGIANOSIDE A CUMINGIANOSIDE A 63524 43344 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PMID27774822-Compound-Figure7Example63 63525 43345 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LAS38096 CHEMBL375293 63526 43346 POLK 51426 DNA REPAIR, ENZYME FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 63528 43347 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MESTRANOL MESTRANOL 22931300 63530 43348 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OFLOXACIN OFLOXACIN 22931300 63534 43349 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE CHIR-265 RAF-265 63536 43350 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CID 663143 CHEMBL1342336 63539 43351 HTT 3064 DRUGGABLE GENOME PDX-101 63540 43352 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PF-05212384 GEDATOLISIB 23980093,21325073 63542 43353 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE RIMONABANT RIMONABANT 21511945 63543 43354 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652083 63544 43355 HMGCR 3156 ENZYME, DRUGGABLE GENOME ROSUVASTATIN ROSUVASTATIN 63545 43356 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GOSSYPOL GOSSYPOL 63546 43357 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GNF-PF-4283 CHEMBL606166 63548 43358 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE DIGITOXIN DIGITOXIN 63549 43359 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL456237 LXR-623 63550 43360 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CILOSTAZOL CILOSTAZOL 63552 43361 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GEMFIBROZIL GEMFIBROZIL 21889235 63554 43362 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL574737 UCN-01 63555 43363 MT1H 4496 NA 6-AN 11835189 63556 43364 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Sunitinib SUNITINIB 24606768 63557 43365 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-51 63558 43366 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME DEPSIPEPTIDE ROMIDEPSIN 15014036 63562 43367 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Fulvestrant FULVESTRANT 63563 43368 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME GNF-PF-5007 CHEMBL1989853 63565 43369 NDUFC1 4717 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 63566 43370 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NAPROXEN NAPROXEN 22931300 63567 43371 TUBB 203068 DRUGGABLE GENOME Vindesine VINDESINE 63569 43372 ALOX15B 247 DRUGGABLE GENOME, ENZYME RABEPRAZOLE RABEPRAZOLE 63571 43373 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor PWT33597 63572 43374 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR DORAMAPIMOD DORAMAPIMOD 63573 43375 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100298 63574 43376 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME 178101762 ARDENERMIN 63575 43377 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1201583 BEVACIZUMAB 63576 43378 SF3B1 23451 CLINICALLY ACTIONABLE E7107 E7107 27622333 63577 43379 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 4-METHOXYDALBERGIONE 4-METHOXYDALBERGIONE 63579 43380 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor AEE788 AEE-788 63580 43381 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-4364 CHEMBL528647 63581 43382 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Dihydroisoquinoline carboxamide analog 1 63583 43383 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650827 PINDOLOL 63584 43384 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Afatinib AFATINIB 27044931,27694386,27102076,26051236,26354527,26341921,25589492,27083334,25964297,28363995,27207775,28145866,24353160,25559287,25870145,24813888,23816960,17349580,23344264,25077897,26286086,27913578,25948633,22190593,24790411,26206867,23991291,26862733,21617858 63585 43385 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Refametinib REFAMETINIB 19706763 63587 43386 ALPI 248 DRUGGABLE GENOME, ENZYME CEPHALOCHROMIN CEPHALOCHROMIN 63588 43387 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE RUTAECARPINE RUTAECARPINE 63592 43388 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR LY-294002 LY-294002 63593 43389 BAZ2B 29994 NA TENOXICAM TENOXICAM 63597 43390 MAP3K14 9020 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE inhibitor 405560388 63598 43391 PDE8A 5151 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200875 FLAVOXATE HYDROCHLORIDE 63601 43392 HTT 3064 DRUGGABLE GENOME GNF-PF-4829 CHEMBL526034 63603 43393 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 A-70108 CHEMBL86931 63604 43394 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CARVEDILOL CARVEDILOL 63606 43395 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR AP26113 CHEMBL3397300 27780853 63607 43396 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 315661158 EDROPHONIUM 63608 43397 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ZIRAM ZIRAM 63609 43398 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR FKB01MD 63610 43399 TPM3 7170 KINASE, CLINICALLY ACTIONABLE UVB 9270028 63611 43400 MAOB 4129 DRUGGABLE GENOME, ENZYME HALOPERIDOL HALOPERIDOL 7617809 63612 43401 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE 4-CHLORO-BENZOIC ACID 4-CHLORO-BENZOIC ACID 63613 43402 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GLEEVEC IMATINIB 15650049 63615 43403 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE NSC-228155 CHEMBL505670 63616 43404 ALOX5 240 DRUGGABLE GENOME, ENZYME Avastin+/-Tarceva 63618 43405 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE VALRUBICIN VALRUBICIN 63619 43406 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE BGJ398 INFIGRATINIB 25673643 63623 43407 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ANAZOLENE ANAZOLENE 63624 43408 SMN2 6607 DRUGGABLE GENOME CID 739615 CHEMBL260560 63626 43409 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME CHEMBL1699 MEMANTINE HYDROCHLORIDE 63627 43410 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1451 TRIAMCINOLONE 63628 43411 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1743048 OBINUTUZUMAB 63629 43412 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE US8614253, 29-19 63630 43413 MPHOSPH8 54737 NA SB-206553 CHEMBL297784 63631 43414 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TRIOXSALEN TRIOXSALEN 63632 43415 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MELENGESTROL ACETATE MELENGESTROL ACETATE 63633 43416 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SB-204070 CHEMBL68131 63634 43417 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SB-222200 SB-222200 63635 43418 POLI 11201 DNA REPAIR IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 63636 43419 ENG 2022 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRC105 63637 43420 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME 4-HYDROPEROXYCYCLOPHOSPHAMIDE PERFOSFAMIDE 8828830 63638 43421 TGFB2 7042 GROWTH FACTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL1743022 FRESOLIMUMAB 63639 43422 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL3039504 NINTEDANIB ESYLATE 63642 43423 TLR7 51284 DRUGGABLE GENOME antagonist 385612195 63643 43424 DHODH 1723 DRUGGABLE GENOME, ENZYME TERIFLUNOMIDE TERIFLUNOMIDE 63645 43425 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE CEDIRANIB CEDIRANIB 63646 43426 BRCA2 675 CLINICALLY ACTIONABLE GEMCITABINE GEMCITABINE 29338080 63649 43427 MAPT 4137 DRUGGABLE GENOME RG6100 63652 43428 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SILVER SULFADIAZINE SILVER SULFADIAZINE 63654 43429 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE SODIUM BUTYRATE 7905674 63655 43430 PDE4D 5144 DRUGGABLE GENOME, ENZYME Revamilast REVAMILAST 63657 43431 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CHELERYTHRINE CHLORIDE CHELERYTHRINE CHLORIDE 63658 43432 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME QUINACRINE DIHYDROCHLORIDE QUINACRINE DIHYDROCHLORIDE 63659 43433 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE PLATINUM COMPOUND 24240112,21920589 63660 43434 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR VR-147 63661 43435 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LASALOCID A SODIUM LASALOCID A SODIUM 63662 43436 FCER1G 2207 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE aspirin ASPIRIN 18595682,18534082 63663 43437 ATAD5 79915 NA BIOCHANIN BIOCHANIN 63666 43438 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 7,8,3'-TRIHYDROXYFLAVONE CHEMBL225513 63667 43439 ADH1C 126 ENZYME, DRUGGABLE GENOME RETINOIC ACID 11959987 63668 43440 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME acetaminophen / codeine 63672 43441 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201541 INSULIN SUSP PROTAMINE ZINC PURIFIED BEEF 63673 43442 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200464 PROPARACAINE HYDROCHLORIDE 63676 43443 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 178103988 TANAPROGET 63677 43444 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 315661244 ULOCUPLUMAB 63679 43445 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME DHM25 26237138 63680 43446 RACGAP1 29127 NA 6-HYDROXYMELATONIN CHEMBL127421 63681 43447 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Quinoline and quinazoline derivative 5 63684 43448 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE DALTEPARIN DALTEPARIN 12632026 63685 43449 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 63687 43450 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME SSR-128428 63688 43451 DMD 1756 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME MyoDys 63689 43452 GMNN 51053 DRUGGABLE GENOME TCMDC-124315 CHEMBL532363 63690 43453 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TEROXIRONE TEROXIRONE 63691 43454 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650902 RISEDRONIC ACID 63692 43455 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Hertuzumab-vc-MMAE 27509865 63693 43456 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LULICONAZOLE LULICONAZOLE 63694 43457 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR NSC-317605 CHEMBL1312050 63696 43458 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565619 PF-04691502 63697 43459 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-409514 CHEMBL160333 63699 43460 RRM2B 50484 ENZYME, DRUGGABLE GENOME, DNA REPAIR cladribine CLADRIBINE 24024897 63701 43461 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR partial agonist CHEMBL299400 BUTORPHANOL TARTRATE 63702 43462 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102602 63703 43463 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ipilimumab IPILIMUMAB 63704 43464 GHRL 51738 DRUGGABLE GENOME CYT-009-GHRQB 63706 43465 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178102559 NINTEDANIB 63707 43466 SMN2 6607 DRUGGABLE GENOME DNDI1417195 CHEMBL1303948 63708 43467 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE inhibitor ORTERONEL ORTERONEL 63709 43468 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE AMT-011 63712 43469 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ASTX727 63713 43470 BAZ2B 29994 NA NITROXOLINE NITROXOLINE 63714 43471 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL1642 IMATINIB MESYLATE 63717 43472 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FIPEXIDE HYDROCHLORIDE FIPEXIDE HYDROCHLORIDE 63718 43473 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE ERLOTINIB ERLOTINIB 63723 43474 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-43 63724 43475 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000200944 CHEMBL600173 63726 43476 GAPDH 2597 DRUGGABLE GENOME, ENZYME THIRAM THIRAM 63727 43477 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Pyridine derivative 18 63728 43478 FAAH 2166 ENZYME, DRUGGABLE GENOME Benzyl pyrrolyloxoacetamide derivative 1 63729 43479 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME SILYBIN B SILYBIN B 23401473 63730 43480 ALOX15B 247 DRUGGABLE GENOME, ENZYME N-(PHENETHYLCARBAMOTHIOYL)BENZAMIDE CHEMBL1448292 63731 43481 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL14762 SELICICLIB 63732 43482 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME INDOCYANINE GREEN SODIUM INDOCYANINE GREEN 63733 43483 RBP4 5950 DRUGGABLE GENOME inhibitor 252827450 63735 43484 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME PRX-302 TOPSALYSIN 63737 43485 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME RUXOLITINIB RUXOLITINIB 22955920 63740 43486 BMP2K 55589 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565886 63741 43487 BAZ2B 29994 NA NSC-8186 CHEMBL122355 63742 43488 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME RO4987655 RO-4987655 26438159,24947927 63743 43489 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Macrolactam derivative 3 63744 43490 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Taladegib TALADEGIB 25759019 63745 43491 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Erdafitinib ERDAFITINIB 63747 43492 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE BROXYQUINOLINE BROXYQUINOLINE 63749 43493 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL325041 BORTEZOMIB 63750 43494 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE inhibitor 178103400 ACETYLDIGITOXIN 63752 43495 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR cyclophosphamide CYCLOPHOSPHAMIDE 24141364 63753 43496 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE STREPTOZOTOCIN STREPTOZOCIN 10098523,9421368 63756 43497 SMN1 6606 DRUGGABLE GENOME NSC-26699 CHEMBL221721 63759 43498 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 310264680 LIQUIRTIGENIN 63760 43499 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AG-120 IVOSIDENIB 25583779 63761 43500 BAZ2B 29994 NA PYRONIN Y PYRONIN Y 63762 43501 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME LY-2090314 LY-2090314 63764 43502 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NSC-93401 CHEMBL452954 63765 43503 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE WEDELOLACTONE WEDELOLACTONE 63766 43504 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME TANSHINONE IIA TANSHINONE IIA 63769 43505 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AMONAFIDE AMONAFIDE 24054489,23353750,17658777,26211460,20170164 63770 43506 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor GSK1070916 GSK-1070916 63771 43507 PDE8B 8622 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL932 DIPYRIDAMOLE 63772 43508 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ABT-263 NAVITOCLAX 63774 43509 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE TOZASERTIB TOZASERTIB 63775 43510 MPHOSPH8 54737 NA AG-555 CHEMBL53898 63778 43511 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER acenocoumarol ACENOCOUMAROL 24919870 63779 43512 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Aminooxazole carboxamide derivative 1 63781 43513 SH2B1 25970 KINASE quetiapine QUETIAPINE 28694205 63783 43514 NOS1AP 9722 NA amiodarone AMIODARONE 63784 43515 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR GW843682X GW843682X 63786 43516 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME imatinib IMATINIB 63787 43517 SMN1 6606 DRUGGABLE GENOME 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 63788 43518 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE GARLIC GARLIC 17213677 63791 43519 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE ILORASERTIB ILORASERTIB 63793 43520 PTGS2 5743 DRUGGABLE GENOME, ENZYME CG100649 POLMACOXIB 63794 43521 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE MECASERMIN MECASERMIN 63795 43522 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000032154 CHEMBL591876 63797 43523 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor RO 4929097 63801 43524 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE IMATINIB IMATINIB 63802 43525 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ANATIBANT ANATIBANT 63805 43526 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE FLAVONE FLAVONE 63806 43527 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000047240 CHEMBL590706 63809 43528 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 2-HYDROXYESTRADIOL CHEMBL467987 63810 43529 DNER 92737 NA GSK525762 MOLIBRESIB 63811 43530 PDE10A 10846 ENZYME, DRUGGABLE GENOME Triazolo-pyridine derivative 4 63812 43531 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLUMETHASONE PIVALATE FLUMETHASONE PIVALATE 63814 43532 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102575 63815 43533 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME SY-1365 63817 43534 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SEROTONIN SEROTONIN 63819 43535 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AC-480 AC-480 19821562 63820 43536 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SCRIPTAID SCRIPTAID 19966789 63821 43537 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER BIOCHANIN A 12948016 63822 43538 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TRIAMCINOLONE TRIAMCINOLONE 22931300 63826 43539 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NORETHINDRONE NORETHINDRONE 63827 43540 F2RL3 9002 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100885 63828 43541 PTGS2 5743 DRUGGABLE GENOME, ENZYME LUMIRACOXIB LUMIRACOXIB 63829 43542 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Altiratinib ALTIRATINIB 63830 43543 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200543 ANILERIDINE PHOSPHATE 63831 43544 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR CETUXIMAB CETUXIMAB 16651634 63832 43545 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3301607 FILGOTINIB 63833 43546 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Enadoline ENADOLINE 63835 43547 CTPS1 1503 ENZYME Cyclopentenylcytosine 63836 43548 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE EZN-2279 ELAPEGADEMASE 63837 43549 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME lamotrigine LAMOTRIGINE 27610747,29791014,26213157 63838 43550 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Pembrolizumab PEMBROLIZUMAB 26645196 63839 43551 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102574 63840 43552 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER atorvastatin ATORVASTATIN 16103896,21392722,26932749,19802823,19238649,18851956 63841 43553 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME ISIS-2503 63842 43554 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Etoposide ETOPOSIDE 25964101 63843 43555 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 7,3'-DIHYDROXYFLAVONE CHEMBL253786 63844 43556 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE Vandetanib VANDETANIB 27683183 63845 43557 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE EW-A-401 63848 43558 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR docetaxel DOCETAXEL 24193570 63849 43559 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor CHEMBL17 DICHLORPHENAMIDE 63850 43560 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor NERATINIB NERATINIB 63852 43561 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 nevirapine NEVIRAPINE 63853 43562 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 63856 43563 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIMETACRINE DIMETACRINE 63858 43564 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PHENOTHIAZINE PHENOTHIAZINE 63860 43565 BAZ2B 29994 NA ASTERRIC ACID ASTERRIC ACID 63861 43566 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545154 POZIOTINIB 63862 43567 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PMID25416646-Compound-Figure2-J 63864 43568 EEF1A1 1915 TRANSCRIPTION FACTOR PMA 9492285 63865 43569 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651370 63866 43570 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GSK-269962A GSK-269962A 63867 43571 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103656 63869 43572 TDO2 6999 ENZYME, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 8 63870 43573 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BAY80-6946 COPANLISIB 63871 43574 NPTX2 4885 DRUGGABLE GENOME PRM-151 PRM-151 63873 43575 NOS1 4842 DRUGGABLE GENOME, ENZYME NXN-462 63874 43576 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 8 63875 43577 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TAMOXIFEN CITRATE TAMOXIFEN CITRATE 63876 43578 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE enalapril ENALAPRIL 17178264 63878 43579 RGS4 5999 DRUGGABLE GENOME BROMOENOL LACTONE BROMOENOL LACTONE 63879 43580 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor DACTOLISIB DACTOLISIB 63880 43581 TFAP2A 7020 TRANSCRIPTION FACTOR AMPRENAVIR AMPRENAVIR 10996400 63881 43582 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME FLUDIAZEPAM FLUDIAZEPAM 63882 43583 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL24828 VANDETANIB 63883 43584 SV2A 9900 DRUGGABLE GENOME, TRANSPORTER INSULIN INSULIN 16306227 63884 43585 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME RG-1530 RG-1530 63885 43586 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ANGUIDIN ANGUIDIN 63886 43587 CA2 760 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200814 ACETAZOLAMIDE SODIUM 63888 43588 PRSS2 5645 DRUGGABLE GENOME, PROTEASE, ENZYME BORTEZOMIB BORTEZOMIB 20875739 63890 43589 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NS-304 SELEXIPAG 63894 43590 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SDX-101 SDX-101 63895 43591 UCHL3 7347 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166860 63896 43592 PTGS2 5743 DRUGGABLE GENOME, ENZYME KETOROLAC KETOROLAC 63897 43593 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545424 AZD-8186 63898 43594 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ACITRETIN ACITRETIN 63900 43595 ATAD5 79915 NA METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 63901 43596 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME MEDROXYPROGESTERONE MEDROXYPROGESTERONE ACETATE 9436888 63902 43597 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE ALL-TRANS RETINOIC ACID 10837916 63903 43598 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL CARBACHOL CARBACHOL 19419204 63904 43599 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CARBOPLATIN CARBOPLATIN 25672916 63905 43600 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR GUGGULSTERONE GUGGULSTERONE 63907 43601 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL186179 MURAGLITAZAR 63908 43602 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL antagonist 135650889 63909 43603 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 4 63911 43604 GSTM1 2944 DRUGGABLE GENOME, ENZYME azathioprine AZATHIOPRINE 23787247 63913 43605 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-Q1 63914 43606 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BUCLIZINE BUCLIZINE 63916 43607 HEBP1 50865 DRUGGABLE GENOME Pyrazino[2,1-a]isoquinolin derivative 1 63917 43608 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE Obatoclax OBATOCLAX 63918 43609 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TETRABUTYLAMMONIUM BROMIDE TETRABUTYLAMMONIUM BROMIDE 63919 43610 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor AZD 8055 63920 43611 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME R-roscovitine SELICICLIB 63921 43612 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1416985 CHEMBL593211 63922 43613 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIPHENYLSULFANE DIPHENYLSULFANE 63923 43614 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TVB-2640 63924 43615 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 252166579 TACEDINALINE 63926 43616 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL1200666 CALCIPOTRIENE 63927 43617 BAZ2B 29994 NA ERYTHROSINE ERYTHROSINE 63929 43618 NDUFA6 4700 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 63931 43619 MPHOSPH8 54737 NA EPHEDRINE SULFATE EPHEDRINE SULFATE 63932 43620 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE CHEMBL114544 63934 43621 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Chlophedianol CHLOPHEDIANOL 63935 43622 AQP9 366 ION CHANNEL UREA UREA 12594337 63936 43623 PBRM1 55193 CLINICALLY ACTIONABLE TRIAZOLAM TRIAZOLAM 22137933 63937 43624 MAP3K10 4294 SERINE THREONINE KINASE, ENZYME, KINASE, DRUGGABLE GENOME TOZASERTIB TOZASERTIB 63938 43625 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor AZD6244 SELUMETINIB 63939 43626 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor FK-228 ROMIDEPSIN 63942 43627 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TOSUFLOXACIN TOSYLATE TOSUFLOXACIN TOSYLATE 63943 43628 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME rosuvastatin ROSUVASTATIN 27839692 63948 43629 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MITOXANTRONE MITOXANTRONE 63949 43630 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651355 ZAPRINAST 63950 43631 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ACETOCHLOR ACETOCHLOR 63951 43632 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 5-METHOXYISATIN 5-METHOXYISATIN 63952 43633 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Sorafenib SORAFENIB 27213589 63953 43634 METAP1 23173 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166758 63954 43635 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2,3-DIHYDROWITHAFERIN A CHEMBL1934585 26169123 63956 43636 HTT 3064 DRUGGABLE GENOME GNF-PF-2335 CHEMBL601146 63957 43637 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRIBUTYLTIN-OXIDE TRIBUTYLTIN-OXIDE 63958 43638 BAZ2B 29994 NA GR-127935 GR-127935 63959 43639 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Temozolomide TEMOZOLOMIDE 27154916 63964 43640 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CHEMBL220492 TOPIRAMATE 63966 43641 AKR1C3 8644 ENZYME, DRUGGABLE GENOME Indomethacin analog 3 63969 43642 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME SODIUM TETRADECYL SULFATE 63970 43643 RAMP2 10266 DRUGGABLE GENOME, CELL SURFACE PRAMLINTIDE PRAMLINTIDE 63971 43644 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-J3 63972 43645 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HER2 Vaccine 9754653,23585514 63973 43646 TPSB2 64499 DRUGGABLE GENOME, PROTEASE HEPARIN HEPARIN 15265919 63976 43647 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR aspirin ASPIRIN 20824505 63977 43648 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME TAE-684 TAE-684 63981 43649 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME ONT-10 63982 43650 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3545323 PWT-33579 63983 43651 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME MESALAMINE MESALAMINE 63984 43652 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR QUINONE 15652497 63985 43653 PDE8B 8622 DRUGGABLE GENOME, ENZYME inhibitor 178101509 DIPYRIDAMOLE 63986 43654 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ABX-EGF PANITUMUMAB 63987 43655 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178103585 ROMIDEPSIN 63989 43656 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NALED NALED 63991 43657 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROROXAN PROROXAN 63994 43658 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE ALBUMIN ALBUMIN HUMAN 1314659 63997 43659 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HYDROCORTISONE HYDROCORTISONE 63998 43660 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUPRANOLOL BUPRANOLOL 2903243 63999 43661 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DICLOFENAC SODIUM DICLOFENAC SODIUM 64000 43662 PKN1 5585 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor SOPHORETIN QUERCETIN 64001 43663 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME PMID28270010-Compound-Figure5-3 64002 43664 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ROGARATINIB ROGARATINIB 30807645 64003 43665 ABCC6 368 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER SALINE SODIUM CHLORIDE 17151194 64004 43666 ENPP2 5168 ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING NSC-1698 CHEMBL1093490 20349977 64005 43667 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 1-BETA-D-ARABINOFURANOSYLCYTOSINE CYTARABINE 3978635 64007 43668 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SU-6656 CHEMBL605003 64008 43669 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Gemcitabine GEMCITABINE 27196758 64009 43670 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AG-34 CHEMBL80155 64012 43671 PTGS1 5742 ENZYME, DRUGGABLE GENOME FENOPROFEN FENOPROFEN 64013 43672 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME KENPAULLONE KENPAULLONE 64014 43673 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tacrine-indole hybrid derivative 3 64017 43674 PTGS2 5743 DRUGGABLE GENOME, ENZYME LUMIRACOXIB LUMIRACOXIB 64018 43675 HSPA4 3308 NA IFOSFAMIDE IFOSFAMIDE 12530536 64019 43676 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME L-3,4-DEHYDROPROLINE CHEMBL78920 21665470 64020 43677 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE RALOXIFENE RALOXIFENE 16167916 64021 43678 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1521 ZALEPLON 64022 43679 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US10179791, Compound 176 64023 43680 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 252827397 OPROZOMIB 64024 43681 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102572 64027 43682 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE BECAPLERMIN BECAPLERMIN 64028 43683 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME AMG 900 64029 43684 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL3545421 DERAZANTINIB 64033 43685 PSMC1 5700 PROTEASE inhibitor BORTEZOMIB BORTEZOMIB 64035 43686 ITPR1 3708 ION CHANNEL, KINASE, DRUGGABLE GENOME, TRANSPORTER activator 135651446 ADENOSINE TRIPHOSPHATE 64036 43687 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9422240, 1-298 64039 43688 GMNN 51053 DRUGGABLE GENOME DNDI1417006 CHEMBL1415258 64040 43689 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE Curcumin CURCUMIN 64042 43690 CRTC2 200186 KINASE XL765 64044 43691 S100A4 6275 NA DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 64052 43692 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME WIN-552122 WIN-552122 64053 43693 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRICIRIBINE TRICIRIBINE 64055 43694 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor BMS-599626 AC-480 64058 43695 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL1059 PREGABALIN 64060 43696 CFL1 1072 KINASE CLOFIBRATE CLOFIBRATE 16680159 64061 43697 TXK 7294 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 249565825 64063 43698 RPS6KA5 9252 DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 64066 43699 GPR12 2835 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651564 64067 43700 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565841 64071 43701 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME BEVACIZUMAB BEVACIZUMAB 15998951 64073 43702 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE METHADONE METHADONE 64074 43703 PTGES 9536 DRUGGABLE GENOME, ENZYME CURCUMIN PYRAZOLE CURCUMIN PYRAZOLE 24920381 64075 43704 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor PKI-587 GEDATOLISIB 64076 43705 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor SF1126 64078 43706 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Benzamide derivative 10 64079 43707 PRKAA2 5563 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 64081 43708 GMNN 51053 DRUGGABLE GENOME ANTAZOLINE HYDROCHLORIDE ANTAZOLINE HYDROCHLORIDE 64082 43709 PTGS1 5742 ENZYME, DRUGGABLE GENOME ANTIVIRAL 18049160 64084 43710 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-2713 CHEMBL578719 64085 43711 ALDH1A1 216 DRUGGABLE GENOME, ENZYME RALOXIFENE RALOXIFENE 64086 43712 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE MIPOMERSEN MIPOMERSEN 64087 43713 GMNN 51053 DRUGGABLE GENOME DICHLOROPHEN DICHLOROPHEN 64088 43714 GNA11 2767 CLINICALLY ACTIONABLE TAK-733 TAK-733 22515704 64090 43715 MAPT 4137 DRUGGABLE GENOME GNF-PF-130 CHEMBL578890 64092 43716 DNPEP 23549 ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE QGC-001 64093 43717 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME CYC-116 CYC-116 20462263 64094 43718 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor PX-866 SONOLISIB 64095 43719 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HYMECROMONE METHYL ETHER HYMECROMONE METHYL ETHER 64096 43720 IGF2R 3482 ENZYME, DRUGGABLE GENOME, CELL SURFACE PXS-25 64099 43721 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PROPYLTHIOURACIL PROPYLTHIOURACIL 15119959 64101 43722 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PMID26924192-Compound-106 64102 43723 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ribociclib RIBOCICLIB 64104 43724 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103647 64105 43725 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor 404859119 64106 43726 HTT 3064 DRUGGABLE GENOME risperidone RISPERIDONE 64108 43727 KLK4 9622 PROTEASE, DRUGGABLE GENOME, ENZYME Heteroaryl-carboxamide derivative 11 64112 43728 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103119 PRINOMASTAT 64113 43729 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME MAFOSFAMIDE MAFOSFAMIDE 8621235 64114 43730 MBP 4155 CELL SURFACE QUERCETIN QUERCETIN 9482255 64115 43731 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200597 ETIDOCAINE HYDROCHLORIDE 64116 43732 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LOPERAMIDE LOPERAMIDE 64117 43733 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME 252166590 TAFAMIDIS 64119 43734 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME clonidine CLONIDINE 64120 43735 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME 3,4-DICHLOROISOCOUMARIN CHEMBL24983 64121 43736 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SARAFLOXACIN HYDROCHLORIDE SARAFLOXACIN HYDROCHLORIDE 64123 43737 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL696 ETHOSUXIMIDE 64124 43738 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 340590265 64125 43739 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE TELOMESTATIN TELOMESTATIN 17954919 64126 43740 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Sorafenib SORAFENIB 64129 43741 KDM4A 9682 DRUGGABLE GENOME, ENZYME SKF-38393 SKF-38393 64130 43742 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME TAE-684 TAE-684 64131 43743 DTNBP1 84062 KINASE clozapine CLOZAPINE 64132 43744 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE RESVERATROL RESVERATROL 17513867 64133 43745 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 saquinavir SAQUINAVIR 9187528 64134 43746 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8829193, 3 64135 43747 HLA-DQB1 3119 CLINICALLY ACTIONABLE nevirapine NEVIRAPINE 64136 43748 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BEVACIZUMAB BEVACIZUMAB 19571295,19603024,22180495 64138 43749 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME blocker 135651273 64139 43750 STK10 6793 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 64140 43751 GRB14 2888 KINASE INSULIN INSULIN 12242277 64142 43752 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-45382 CHEMBL1214274 64143 43753 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32q 64145 43754 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME inhibitor 249565694 CHIR-99021 64147 43755 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BERGAPTEN BERGAPTEN 64148 43756 NME2 4831 KINASE adefovir dipivoxil 64150 43757 USP1 7398 DNA REPAIR, PROTEASE, ENZYME QUINALIZARIN QUINALIZARIN 64151 43758 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER (R)-VERAPAMIL DEXVERAPAMIL 17646169 64152 43759 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE IL-12 12097373 64154 43760 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME CARVEDILOL CARVEDILOL 18498919 64155 43761 HMOX1 3162 ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE STANNSOPORFIN STANNSOPORFIN 64157 43762 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL220492 TOPIRAMATE 64159 43763 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200563 CERIVASTATIN SODIUM 64161 43764 TARDBP 23435 TUMOR SUPPRESSOR NAPROXEN SODIUM NAPROXEN SODIUM 64163 43765 TUBB 203068 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 64165 43766 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE agonist 178103536 PALIFERMIN 64166 43767 IL1A 3552 CELL SURFACE, DRUGGABLE GENOME MITOMYCIN-C 8195120 64167 43768 ALPL 249 ENZYME, DRUGGABLE GENOME DNDI1417368 CHEMBL2094652 64168 43769 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Diamidothiazole derivative 1 64170 43770 GPR183 1880 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651393 64171 43771 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor SOPHORETIN QUERCETIN 64172 43772 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE SUNITINIB SUNITINIB 64173 43773 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CYC116 64174 43774 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000299520 CHEMBL592305 64175 43775 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-92207 CHEMBL139935 64176 43776 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201023 ORPHENADRINE HYDROCHLORIDE 64177 43777 VKORC1 79001 DRUGGABLE GENOME, ENZYME Phenindione PHENINDIONE 64178 43778 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Phenylpropylamine derivative 1 64180 43779 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor LGX818 ENCORAFENIB 64181 43780 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME GNF-PF-2272 CHEMBL601757 64182 43781 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103924 MACITENTAN 64183 43782 ATXN2 6311 NA SJ000029642 CHEMBL591126 64188 43783 SLCO3A1 28232 TRANSPORTER, DRUGGABLE GENOME 135651569 64189 43784 BAZ2B 29994 NA GNF-PF-5114 CHEMBL601952 64190 43785 SMN2 6607 DRUGGABLE GENOME LOVASTATIN LOVASTATIN 64192 43786 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ENCORAFENIB ENCORAFENIB 25673644 64195 43787 TUBB6 84617 DRUGGABLE GENOME CHEMBL2105643 FOSBRETABULIN TROMETHAMINE 64197 43788 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE CMX-2043 CMX-2043 64198 43789 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE STREPTOZOCIN STREPTOZOCIN 2354749 64199 43790 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TEMEFOS TEMEFOS 64201 43791 PDE4C 5143 DRUGGABLE GENOME, ENZYME IBUDILAST IBUDILAST 64202 43792 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-724440 CHEMBL515617 64203 43793 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE PD-157695 64204 43794 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME TAXANE COMPOUND 24961465 64207 43795 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-56 64208 43796 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ZAFIRLUKAST ZAFIRLUKAST 64209 43797 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME olanzapine OLANZAPINE 23492908 64210 43798 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-677438 CHEMBL118678 64213 43799 GMNN 51053 DRUGGABLE GENOME DOXAZOSIN MESYLATE DOXAZOSIN MESYLATE 64215 43800 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor 178103722 CHLORTHALIDONE 64216 43801 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL215645 RIVASTIGMINE TARTRATE 64217 43802 DIAPH3 81624 KINASE hydrochlorothiazide HYDROCHLOROTHIAZIDE 64218 43803 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL3545143 SR-13668 64220 43804 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 385612233 64223 43805 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AS101 AMMONIUM TRICHLOROTELLURATE 7539780 64225 43806 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178103559 AZIDOPINE 64229 43807 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-1947 CHEMBL585591 64230 43808 POLI 11201 DNA REPAIR ETHACRYNIC ACID ETHACRYNIC ACID 64231 43809 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652143 64233 43810 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 135652636 64234 43811 TSPO 706 DRUGGABLE GENOME ZALEPLON ZALEPLON 64237 43812 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE axitinib AXITINIB 24433361 64239 43813 RACGAP1 29127 NA (-)-EPICATECHIN (-)-EPICATECHIN 64241 43814 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE INK-1117 INK-1117 64246 43815 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE ALSTERPAULLONE ALSTERPAULLONE 64247 43816 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 381744980 ISOSAKUTANETIN 64248 43817 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME GNF-PF-4759 CHEMBL585265 64249 43818 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SKF-89626 CHEMBL284609 64251 43819 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME CABAZITAXEL CABAZITAXEL 25670080 64253 43820 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME DACTOLISIB DACTOLISIB 64254 43821 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AMBRISENTAN AMBRISENTAN 64255 43822 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR CLARITHROMYCIN CLARITHROMYCIN 16815316 64257 43823 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-WO2011127048 34 64258 43824 GJA1 2697 ION CHANNEL inhibitor 178101095 OCTANOL 64259 43825 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ASPIRIN ASPIRIN 22931300 64260 43826 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR TRIIODOTHYRONINE LIOTHYRONINE SODIUM 11250650 64261 43827 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-1947 CHEMBL585591 64262 43828 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR THIOMERSAL THIMEROSAL 64263 43829 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 64264 43830 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME 1,4-DIMETHOXYANTHRAQUINONE 1,4-DIMETHOXYANTHRAQUINONE 64265 43831 GMNN 51053 DRUGGABLE GENOME ETHACRYNIC ACID ETHACRYNIC ACID 64266 43832 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME GOSSYPOL GOSSYPOL 64268 43833 TRIM5 85363 ENZYME, B30_2 SPRY DOMAIN, DRUGGABLE GENOME carboplatin CARBOPLATIN 64270 43834 ATAD5 79915 NA OCTAVERINE OCTAVERINE 64271 43835 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL2012520 LY377604 64272 43836 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1213490 ROMIDEPSIN 64273 43837 CD52 1043 DRUGGABLE GENOME ANDROGENS 10737964 64275 43838 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CHLORQUINALDOL CHLORQUINALDOL 64277 43839 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BITHIONOL BITHIONOL 64278 43840 MAPT 4137 DRUGGABLE GENOME BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 64279 43841 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 64281 43842 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR BMS-387032 BMS-387032 64282 43843 PTPRD 5789 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 381118819 64285 43844 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NICOTINE BITARTRATE NICOTINE BITARTRATE 64286 43845 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AIKO-150 64287 43846 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR JNJ-7706621 JNJ-7706621 64288 43847 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL1200699 DOXYCYCLINE 64289 43848 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 23634759 64290 43849 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL1739 METOCURINE IODIDE 64292 43850 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME ALISERTIB ALISERTIB 64293 43851 AMH 268 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HORMONES 12428210 64294 43852 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME docetaxel DOCETAXEL 25495407 64295 43853 TUBA1B 10376 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 64296 43854 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME ILORASERTIB ILORASERTIB 64298 43855 ATAD5 79915 NA GOSSYPOL GOSSYPOL 64299 43856 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Chlorobenzamide derivative 1 64300 43857 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-3343 CHEMBL599943 64301 43858 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME LOXO-101 LAROTRECTINIB 64302 43859 CA2 760 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL220492 TOPIRAMATE 64303 43860 IL17RA 23765 DRUGGABLE GENOME antagonist CHEMBL1742996 BRODALUMAB 64306 43861 UGT2B7 7364 DRUGGABLE GENOME mycophenolate mofetil 24681964 64308 43862 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist CHEMBL3545239 PF-05019702 64310 43863 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1200833 DIPIVEFRIN HYDROCHLORIDE 64311 43864 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2-ARACHIDONOYLGLYCEROL 2-ARACHIDONOYLGLYCEROL 64312 43865 PSMC3 5702 NA CARFILZOMIB CARFILZOMIB 24524217 64313 43866 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CAMPTOTHECIN CAMPTOTHECIN 15500952 64314 43867 ALDH1A1 216 DRUGGABLE GENOME, ENZYME MERCAPTOPURINE MERCAPTOPURINE 64315 43868 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE IMATINIB IMATINIB 15790786,9438854,21159146,21689725,20088873,24045550,18936790,7530509,15236194,19164557,15201427,15972446,16384925,18024392,15685537,19861435,11276010,21969494,16638875,18986703,21690468,23375402,18980976,22357254,17372901,22504184,24687822,16908931,19175693,16912224,15930355,19812602,23775962,23714533,19671763,25157968,16046538,22932406,17363509,17259998,21642685,16954519,16751810,23582185,22355224,16731599 64316 43869 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CLOMIPRAMINE CLOMIPRAMINE 64319 43870 HSPA4 3308 NA H-103 64320 43871 IDE 3416 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, ENZYME, PROTEASE BIOTIN BIOTIN 64322 43872 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AVELUMAB AVELUMAB 31086949 64323 43873 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 135650237 64324 43874 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DNDI1417309 CHEMBL1341830 64325 43875 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 22044621 64326 43876 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR AZD9496 AZD-9496 64327 43877 PDE4C 5143 DRUGGABLE GENOME, ENZYME US10077269, Example 6 64329 43878 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 385612184 64330 43879 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TCMDC-125580 CHEMBL528807 64333 43880 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER TRIACETIN TRIACETIN 64334 43881 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR REGADENOSON REGADENOSON 64335 43882 MAPKAPK3 7867 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 249565857 64336 43883 SULT1C4 27233 ENZYME thalidomide THALIDOMIDE 20038957 64338 43884 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Encorafenib ENCORAFENIB 27312529 64340 43885 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE INDINAVIR INDINAVIR 11916910 64341 43886 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-668 CHEMBL604528 64342 43887 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NARINGENIN NARINGENIN 64343 43888 DGAT1 8694 ENZYME, DRUGGABLE GENOME Benzamide derivative 19 64344 43889 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1-NITROPYRENE 1-NITROPYRENE 64345 43890 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-Figure3bII 64349 43891 PREP 5550 PROTEASE, ENZYME, DRUGGABLE GENOME ALV-003 LATIGLUTENASE 64351 43892 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CIMETIDINE CIMETIDINE 22931300 64353 43893 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-2588 CHEMBL578636 64354 43894 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-2094 CHEMBL578928 64355 43895 GJB3 2707 TRANSPORTER, ION CHANNEL inhibitor 135652731 64356 43896 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28117607-Compound-7 64357 43897 KDM4A 9682 DRUGGABLE GENOME, ENZYME CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 64360 43898 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME STAUROSPORINE STAUROSPORINE 12401608,12759177 64361 43899 SMYD2 56950 ENZYME, METHYL TRANSFERASE inhibitor 249565919 64362 43900 TAC1 6863 DRUGGABLE GENOME PROTOPORPHYRIN PROTOPORPHYRIN 9677143 64363 43901 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GP-120 9419208 64364 43902 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BROMPERIDOL BROMPERIDOL 64365 43903 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME SP-600125 SP-600125 64369 43904 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE METHOTREXATE METHOTREXATE 2431676 64370 43905 E2F1 1869 TRANSCRIPTION FACTOR HGF 11821989,12064460 64371 43906 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ACETYLSEROTONIN ACETYLSEROTONIN 64372 43907 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CRYPTOLEPINE HYDROCHLORIDE CRYPTOLEPINE HYDROCHLORIDE 23507189 64373 43908 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE 2-PHENYLACETYLAMINOBENZOTHIAZOLE CHEMBL1405979 64375 43909 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 STREPTOZOTOCIN STREPTOZOCIN 8435090 64376 43910 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1318477 CHEMBL428064 64377 43911 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 3-HYDROXYFLAVONOL CHEMBL242172 64378 43912 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BAY80-6946 COPANLISIB 64379 43913 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33c 64381 43914 EPHA7 2045 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 249565821 64382 43915 DDC 1644 ENZYME, DRUGGABLE GENOME AV-201 64383 43916 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Roscovitine derivative 1 64386 43917 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME SF1126 64387 43918 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BUTORPHANOL BUTORPHANOL 22931300 64388 43919 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GNF-PF-3023 CHEMBL535331 64389 43920 HLA-G 3135 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME methotrexate METHOTREXATE 16906016,19088262 64390 43921 KDM4A 9682 DRUGGABLE GENOME, ENZYME THIORIDAZINE HYDROCHLORIDE THIORIDAZINE HYDROCHLORIDE 64391 43922 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650897 64392 43923 ADD1 118 KINASE spironolactone SPIRONOLACTONE 21692745 64393 43924 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AURIN AURIN 64394 43925 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM BROMIDE 64396 43926 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE PAMIDRONATE PAMIDRONIC ACID 64398 43927 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Debio 1347 64399 43928 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL ALLOPREGNANOLONE BREXANOLONE 64401 43929 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PI-88 MUPARFOSTAT 64402 43930 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME activator 363894217 VORUCICLIB 64404 43931 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody IPILIMUMAB IPILIMUMAB 64405 43932 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER mitoxantrone MITOXANTRONE 64408 43933 TGFBR3 7049 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME GM-CSF REGRAMOSTIM 12471017 64409 43934 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102262 64410 43935 UGT1A10 54575 DRUGGABLE GENOME, ENZYME TROGLITAZONE TROGLITAZONE 12433820 64411 43936 LTB4R2 56413 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102782 64413 43937 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ATOMOXETINE ATOMOXETINE 64414 43938 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PF-562271 PF-00562271 64416 43939 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650258 FENTANYL 64417 43940 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178103969 CERITINIB 64419 43941 CDC42BPA 8476 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME DASATINIB DASATINIB 64420 43942 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor VELIPARIB VELIPARIB 64421 43943 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE modulator CHEMBL3545333 MK-0773 64422 43944 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Eptastigmine EPTASTIGMINE 64423 43945 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME URSODEOXYCHOLIC ACID 11033072 64424 43946 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR MERCURIC CHLORIDE MERCURIC CHLORIDE 64425 43947 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LYCOBETAINE LYCOBETAINE 23266176 64426 43948 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE clozapine CLOZAPINE 25751398 64427 43949 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-43 64429 43950 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL384467 DEXAMETHASONE 64430 43951 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME RG7775 64431 43952 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BAY1082439 64432 43953 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CYC-116 CYC-116 64434 43954 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor IMATINIB IMATINIB 64436 43955 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200906 OXYPHENONIUM BROMIDE 64437 43956 ALOX15 246 ENZYME, DRUGGABLE GENOME BITHIONOLATE SODIUM BITHIONOLATE SODIUM 64438 43957 SULT2A1 6822 DRUGGABLE GENOME OXANDROLONE OXANDROLONE 8319371 64440 43958 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-2356 CHEMBL601547 64441 43959 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE STREPTOZOTOCIN STREPTOZOCIN 11978652 64443 43960 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR GI-264879A 64444 43961 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE antibody ONARTUZUMAB ONARTUZUMAB 64445 43962 AKR1C3 8644 ENZYME, DRUGGABLE GENOME NSAID 14996743 64446 43963 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE PF-562271 PF-00562271 64448 43964 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR CC-401 CC-401 64450 43965 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR Ibudilast IBUDILAST 64454 43966 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME pyrimethamine PYRIMETHAMINE 11807801 64455 43967 KLKB1 3818 DRUGGABLE GENOME, PROTEASE, ENZYME antibody 315661179 LANADELUMAB 64456 43968 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METOPROLOL METOPROLOL 64457 43969 UBE2D1 7321 ENZYME, TRANSCRIPTION FACTOR DESFERRIOXAMINE DEFEROXAMINE 9694900 64458 43970 HSF1 3297 TRANSCRIPTION FACTOR, DNA REPAIR HSP70 9499401,9822662 64459 43971 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651583 64462 43972 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201545 INSULIN SUSP ISOPHANE BEEF 64463 43973 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor SODIUM PHENYLBUTYRATE 64464 43974 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME bleomycin BLEOMYCIN 64465 43975 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME simvastatin SIMVASTATIN 24598718 64466 43976 PTGS2 5743 DRUGGABLE GENOME, ENZYME TENOXICAM TENOXICAM 64470 43977 DDC 1644 ENZYME, DRUGGABLE GENOME inhibitor 178101842 BENSERAZIDE 64471 43978 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMPEROZIDE AMPEROZIDE 64472 43979 EYA2 2139 DNA REPAIR FLUPIRTINE FLUPIRTINE 64473 43980 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MEZLOCILLIN MEZLOCILLIN 64475 43981 CDK19 23097 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 178102285 LINIFANIB 64477 43982 ALDH1A1 216 DRUGGABLE GENOME, ENZYME MG-132 MG-132 64478 43983 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 135650190 64481 43984 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GOSSYPOL GOSSYPOL 64482 43985 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME METHACYCLINE HYDROCHLORIDE METHACYCLINE HYDROCHLORIDE 64483 43986 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 223366137 64484 43987 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME PMID26161698-Compound-25 64486 43988 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist CHEMBL1131 ACITRETIN 64487 43989 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME GENISTEIN GENISTEIN 10811979 64488 43990 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody U3-1287 AMG-888 64491 43991 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME I-BET151 27294782 64492 43992 NDUFA7 4701 ENZYME inhibitor CHEMBL3545135 NV-128 64494 43993 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE JT02 64499 43994 PSMD8 5714 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 64502 43995 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NITROBLUE TETRAZOLIUM NITROBLUE TETRAZOLIUM 64504 43996 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR antagonist 135652690 GUGGULSTERONE 64505 43997 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MEDRYSONE MEDRYSONE 64508 43998 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyridine derivative 2 64509 43999 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-38 64510 44000 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 64511 44001 TARDBP 23435 TUMOR SUPPRESSOR SJ000260156 CHEMBL590695 64512 44002 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME CASPASE INHIBITOR 15122333 64513 44003 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LAPACHOL LAPACHOL 64514 44004 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Folic Acid 64516 44005 ENPP2 5168 ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 315661227 64517 44006 BRCA2 675 CLINICALLY ACTIONABLE ABT-767 64519 44007 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE ABCIXIMAB ABCIXIMAB 64520 44008 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200790 METHYPRYLON 64521 44009 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE irbesartan IRBESARTAN 15614026 64522 44010 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME NSC-119889 CHEMBL516616 64526 44011 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE PMID26882240-Compound-6 64530 44012 PSMB9 5698 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 64531 44013 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Ivosidenib IVOSIDENIB 64532 44014 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PARAPLATIN CARBOPLATIN 64533 44015 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME CC-1088 CDC-801 14717786 64534 44016 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor XL999 64535 44017 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME PHA-767491 CHEMBL225519 64536 44018 TUBB2A 7280 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 64537 44019 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME LY3009104 64538 44020 GJB2 2706 ION CHANNEL, TRANSPORTER inhibitor 178100972 CARBENOXOLONE 64540 44021 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 178103566 64542 44022 PTGS2 5743 DRUGGABLE GENOME, ENZYME Flurbiprofen FLURBIPROFEN 64546 44023 KDM2A 22992 DRUGGABLE GENOME, ENZYME inhibitor 178103604 64547 44024 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER venlafaxine VENLAFAXINE 24192121,18215618,21449676,26704739,26757307,22641028,26664259 64548 44025 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL3545173 IRX4310 64550 44026 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX IBRUTINIB IBRUTINIB 64551 44027 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE BHQ-880 BHQ-880 64552 44028 HTT 3064 DRUGGABLE GENOME GNF-PF-5151 CHEMBL576208 64553 44029 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE 6,6-fused nitrogenous heterocyclic compound 2 64554 44030 DNER 92737 NA Mivebresib MIVEBRESIB 64555 44031 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW819230X GW819230X 64556 44032 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE allosteric modulator 315661240 64557 44033 PDK4 5166 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME inhibitor 328083452 64559 44034 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TIDEGLUSIB TIDEGLUSIB 64560 44035 LAMB3 3914 DRUGGABLE GENOME LAMB3-transduced autologous epidermal stem cells 64561 44036 VKORC1 79001 DRUGGABLE GENOME, ENZYME Warfarin WARFARIN 64562 44037 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565795 64565 44038 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Regorafenib REGORAFENIB 23629727 64567 44039 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor SOPHORETIN QUERCETIN 64569 44040 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR INDOMETHACIN INDOMETHACIN 11909699 64570 44041 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE LINIFANIB LINIFANIB 64571 44042 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE IRINOTECAN HYDROCHLORIDE IRINOTECAN HYDROCHLORIDE 64572 44043 TUBB2B 347733 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 64574 44044 GMNN 51053 DRUGGABLE GENOME ZM-39923 HCL CHEMBL538798 64575 44045 TNFRSF1A 7132 CELL SURFACE, DRUGGABLE GENOME etanercept ETANERCEPT 22480748 64576 44046 IL18 3606 DRUGGABLE GENOME HPV-16 E6 16125299 64577 44047 CYB5R2 51700 DRUGGABLE GENOME isosorbide mononitrate 64578 44048 DUSP3 1845 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE GNF-PF-231 CHEMBL601167 64580 44049 ABAT 18 DRUGGABLE GENOME, ENZYME K-828-AB 64582 44050 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL RO-229735 CHEMBL2170369 21751815 64584 44051 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Lusutrombopag LUSUTROMBOPAG 64586 44052 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX PECTOLINARIGENIN PECTOLINARIGENIN 64587 44053 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME FK-070 64588 44054 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ESTRADIOL ESTRADIOL 22931300 64589 44055 GMNN 51053 DRUGGABLE GENOME NSC-636948 CHEMBL1998001 64590 44056 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 19 64592 44057 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 4-(4-CHLOROPHENOXY)ANILINE CHEMBL1521156 64593 44058 RPS6KA5 9252 DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor 249565810 CHEMBL188434 64596 44059 XDH 7498 DRUGGABLE GENOME, ENZYME PAPAVERINE PAPAVERINE 11200484 64597 44060 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 INDOMETHACIN MORPHOLINYLAMIDE INDOMETHACIN MORPHOLINYLAMIDE 64601 44061 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor SOPHORETIN QUERCETIN 64602 44062 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 404859098 SAMIDORPHAN 64603 44063 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545088 PUQUITINIB 64604 44064 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RIMONABANT RIMONABANT 64605 44065 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE SJ000294102 CHEMBL607309 64607 44066 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CYCLOHEXIMIDE CYCLOHEXIMIDE 64609 44067 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Noberastine NOBERASTINE 64610 44068 TUBA3D 113457 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 64611 44069 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME MP0250 MP-0250 64612 44070 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PIRFENIDONE PIRFENIDONE 64614 44071 TYMP 1890 GROWTH FACTOR, DRUGGABLE GENOME Uridine URIDINE 64615 44072 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SALT VOLANESORSEN SODIUM 2557514 64617 44073 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 363894213 64618 44074 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-102030 CHEMBL406834 64620 44075 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PALBOCICLIB PALBOCICLIB 25810375,23569312,27124835,26528855,23898052 64621 44076 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR VX-702 VX-702 64622 44077 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103555 CHLORPHENIRAMINE 64624 44078 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL403989 TG100-801 64626 44079 TUBA3D 113457 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 64627 44080 MCOLN2 255231 ION CHANNEL, DRUGGABLE GENOME activator 178100233 64628 44081 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL15770 SULINDAC 64629 44082 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME DOVITINIB DOVITINIB 64631 44083 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TRACAZOLATE TRACAZOLATE 64632 44084 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME fluorouracil FLUOROURACIL 64633 44085 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565860 64634 44086 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZWITTERGENT 3-12 CHEMBL1235854 64635 44087 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 1,2-DIMETHOXY-ANTHRAQUINONE CHEMBL52884 64636 44088 POLI 11201 DNA REPAIR AMINOQUINOL AMINOQUINOL 64637 44089 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME activator 404859004 64638 44090 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Cyclizine CYCLIZINE 64639 44091 DPP6 1804 DRUGGABLE GENOME, ENZYME, TRANSPORTER, PROTEASE haloperidol HALOPERIDOL 27023437 64641 44092 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BUTACLAMOL HYDROCHLORIDE BUTACLAMOL HYDROCHLORIDE 64643 44093 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Ceritinib CERITINIB 25394791 64644 44094 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Venlafaxine VENLAFAXINE 64646 44095 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 340590231 64647 44096 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR MK-6913 MK-6913 64648 44097 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE TAE-684 TAE-684 64649 44098 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME ENMD-2076 ENMD-2076 64651 44099 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR warfarin WARFARIN 25356900 64652 44100 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565616 SAPANISERTIB 64653 44101 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME interferon alfa-2a, recombinant 64654 44102 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Encorafenib ENCORAFENIB 64655 44103 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Pasireotide PASIREOTIDE 64657 44104 MAOB 4129 DRUGGABLE GENOME, ENZYME Psoralen PSORALEN 64658 44105 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 135651503 64661 44106 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME Odanacatib ODANACATIB 64664 44107 GUCY2C 2984 DRUGGABLE GENOME, KINASE Guanilib 64665 44108 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-22 64666 44109 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DT-200 GLPG0492 64667 44110 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE ELIPRODIL ELIPRODIL 64669 44111 MAOB 4129 DRUGGABLE GENOME, ENZYME 4-Methoxybenzaldehyde ANISALDEHYDE 64671 44112 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLORDANE CHLORDANE 64672 44113 SGK1 6446 SERINE THREONINE KINASE, KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME, DRUG RESISTANCE SGK1-INH 27451907 64674 44114 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME RHEIN RHEIN 64676 44115 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GSK163929 CHEMBL1784521 64678 44116 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651059 CAPESEROD 64679 44117 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SJ000071854 CHEMBL602127 64680 44118 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE PEG-NALOXOL 64684 44119 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE OSI-632 OSI-632 64685 44120 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BUTACAINE BUTACAINE 64686 44121 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR SALERMIDE SALERMIDE 64687 44122 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CONGO RED CONGO RED 64688 44123 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor INCB28060 CAPMATINIB 64689 44124 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200485 SORAFENIB TOSYLATE 64691 44125 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE activator CHEMBL1201420 UROKINASE 64692 44126 TP53AIP1 63970 NA fluorouracil FLUOROURACIL 64693 44127 CSF1 1435 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ANTISERUM 1717026,2546636,8647916,3497819,8889847,3908292,8591991 64696 44128 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ALISERTIB ALISERTIB 64697 44129 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor VORINOSTAT VORINOSTAT 64699 44130 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE 16,16-dimethyl-PGE2 64700 44131 TARDBP 23435 TUMOR SUPPRESSOR LMT-X 64701 44132 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME (-)-PLAKILACTONE C CHEMBL2178586 22934537 64702 44133 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Siplizumab SIPLIZUMAB 64703 44134 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamoyl oxime derivative 1 64706 44135 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 64707 44136 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 64709 44137 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ACID BLUE 129 ACID BLUE 129 64710 44138 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649685 64711 44139 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PHYTOESTROGEN 15331887 64713 44140 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GSK-269962A GSK-269962A 64714 44141 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor NILOTINIB NILOTINIB 64715 44142 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX QUERCETAGETIN QUERCETAGETIN 25190466 64716 44143 HSPB1 3315 DRUGGABLE GENOME CLOXYQUIN CLOXYQUIN 64717 44144 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ISOTRETINOIN ISOTRETINOIN 10621853,10638174 64718 44145 MMP14 4323 PROTEASE, DRUGGABLE GENOME, ENZYME BT-1718 64720 44146 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE GW441756X GW441756X 64721 44147 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME N-Arachidonoyl Dopamine 27760835 64722 44148 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HER2-pulsed DC1 vaccine 27965306 64723 44149 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE SB-203580 SB-203580 64725 44150 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL238804 SELEXIPAG 64726 44151 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BROMOCRIPTINE BROMOCRIPTINE 64727 44152 SULT1A4 445329 ENZYME acetaminophen ACETAMINOPHEN 26049587 64728 44153 CBX1 10951 NA NSC-19063 CHEMBL1310138 64729 44154 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ICI-162846 CHEMBL1593717 64730 44155 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CY-208243 CHEMBL313737 64731 44156 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 328083493 64737 44157 RGS4 5999 DRUGGABLE GENOME ROTTLERIN ROTTLERIN 64741 44158 MTRR 4552 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME vitamin b-complex, plain 22926161 64742 44159 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SANGUINARIUM CHLORIDE SANGUINARIUM CHLORIDE 64744 44160 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE CD40L 17015702 64746 44161 TUBB2A 7280 DRUGGABLE GENOME CHEMBL2304041 SAGOPILONE 64747 44162 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 249565579 APITOLISIB 64748 44163 PBRM1 55193 CLINICALLY ACTIONABLE SUNITINIB SUNITINIB 27751729 64750 44164 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-125034 CHEMBL239439 64751 44165 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL1721885 SU-014813 64753 44166 TUBB 203068 DRUGGABLE GENOME DOLASTATIN-10 DOLASTATIN-10 64756 44167 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ARSANILIC ACID ARSANILIC ACID 64758 44168 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME DIAZEPAM DIAZEPAM 64759 44169 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PUUPEHENONE PUUPEHENONE 22928967 64762 44170 XDH 7498 DRUGGABLE GENOME, ENZYME BENZODIAZEPINE BENZODIAZEPINE 2904285 64763 44171 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE CAROTENE 9101560 64764 44172 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PMID25416646-Compound-Figure5-E 64766 44173 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL2364607 COBIMETINIB FUMARATE 64767 44174 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor BKM120 BUPARLISIB 64768 44175 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor EVEROLIMUS EVEROLIMUS 64769 44176 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL2107771 RALFINAMIDE 64771 44177 FAAH 2166 ENZYME, DRUGGABLE GENOME ANANDAMIDE ANANDAMIDE 21899370 64772 44178 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE EOTAXIN 12489019 64773 44179 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR THEONELLASTEROL B THEONELLASTEROL B 21428459 64774 44180 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2105864 LABRADIMIL 64777 44181 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR esuberaprost ESUBERAPROST 64778 44182 EPHX1 2052 ENZYME, DRUGGABLE GENOME ANTICONVULSANT 10554101 64780 44183 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE DS-1205 64781 44184 KDM4A 9682 DRUGGABLE GENOME, ENZYME SCLEROTIORIN SCLEROTIORIN 64782 44185 TSC2 7249 CLINICALLY ACTIONABLE, KINASE, TUMOR SUPPRESSOR Everolimus EVEROLIMUS 64783 44186 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER R101933 12008197 64784 44187 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER ALSEROXYLON ALSEROXYLON 64785 44188 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIMENHYDRINATE DIMENHYDRINATE 64786 44189 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 178102328 PI-103 64787 44190 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051828 64788 44191 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 2',4'-DIHYDROXY FLAVONE CHEMBL1374610 64789 44192 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1201156 NORTRIPTYLINE HYDROCHLORIDE 64791 44193 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME EVT-201 64792 44194 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME inhibitor AMG 102 RILOTUMUMAB 64793 44195 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TOPOTECAN HYDROCHLORIDE TOPOTECAN HYDROCHLORIDE 64795 44196 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ATENOLOL ATENOLOL 64796 44197 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 64797 44198 GHRL 51738 DRUGGABLE GENOME PSYLLIUM PSYLLIUM SEED HUSKS 17998014 64799 44199 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649808 64800 44200 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MGCD-0103 MOCETINOSTAT 64801 44201 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SB-220025 SB-220025 64803 44202 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME inhibitor 249565597 64804 44203 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Aromatic bicyclic compound 4 64805 44204 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR DIMETHYLADENINE DIMETHYLADENINE 64806 44205 RAB9A 9367 ENZYME, DRUGGABLE GENOME (E)-2-STYRYLCHROMONE CHEMBL388823 64808 44206 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR ACYCLOVIR ACYCLOVIR 16961277 64809 44207 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE PF-562271 PF-00562271 64810 44208 NF2 4771 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, DRUG RESISTANCE, KINASE CARBOPLATIN CARBOPLATIN 25798586 64811 44209 IGFBP1 3484 DRUGGABLE GENOME PMA 8557761 64813 44210 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME (+/-)-VANILLYLMANDELIC ACID CHEMBL1256396 64814 44211 HSPB1 3315 DRUGGABLE GENOME BENZO(K)FLUORANTHENE BENZO(K)FLUORANTHENE 64816 44212 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LAVENDUSTIN C LAVENDUSTIN C 64817 44213 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME DASATINIB DASATINIB 64818 44214 GUCA2A 2980 DRUGGABLE GENOME, ENZYME, HORMONE ACTIVITY ATROPINE ATROPINE 9623669 64819 44215 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor 178103543 ROFLUMILAST 64824 44216 SLC22A3 6581 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER SARCNU SARCNU 11783015,10632359 64825 44217 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SC-19220 CHEMBL112816 64826 44218 AAK1 22848 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME LX9211 64827 44219 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 64828 44220 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 3,3',4'-TRIHYDROXYFLAVONE CHEMBL122701 64829 44221 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CIS-RESVERATROL CIS-RESVERATROL 64830 44222 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE ACACETIN ACACETIN 64831 44223 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME SCRIPTAID SCRIPTAID 19966789 64832 44224 ILK 3611 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 249565796 64833 44225 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103722 CHLORTHALIDONE 64834 44226 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651221 64837 44227 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME CIGLITAZONE CIGLITAZONE 20170185,16643023,23566516 64838 44228 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME OXOTREMORINE METHIODIDE OXOTREMORINE METHIODIDE 64840 44229 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ReACp53 26748848 64841 44230 A2M 2 ENZYME, TRANSPORTER, DRUGGABLE GENOME, PROTEASE INHIBITOR Enzymes 23280790 64842 44231 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LUZINDOLE LUZINDOLE 64845 44232 GMNN 51053 DRUGGABLE GENOME RITANSERIN RITANSERIN 64848 44233 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR OLEOYLETHANOLAMIDE OLEOYLETHANOLAMIDE 26071639,17228882 64850 44234 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27551786-Compound-138 64851 44235 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE Midostaurin MIDOSTAURIN 23131561 64853 44236 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PROTOPORPHYRIN DISODIUM PROTOPORPHYRIN DISODIUM 64854 44237 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SKF-38393 SKF-38393 64855 44238 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Matuzumab MATUZUMAB 64856 44239 ALOX5 240 DRUGGABLE GENOME, ENZYME Darbufelone DARBUFELONE 64857 44240 SLC3A2 6520 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER antibody 252827395 64858 44241 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE ERLOTINIB ERLOTINIB 29802158 64860 44242 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 22 64861 44243 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102712 64867 44244 HTT 3064 DRUGGABLE GENOME IDARUBICIN IDARUBICIN 64868 44245 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SOTRASTAURIN SOTRASTAURIN 64869 44246 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Venetoclax VENETOCLAX 27974663 64870 44247 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor SUNITINIB SUNITINIB 64872 44248 GMNN 51053 DRUGGABLE GENOME 2-(ALPHA-NAPHTHOYL)ETHYLTRIMETHYLAMMONIUM IODIDE CHEMBL1255936 64874 44249 HEBP1 50865 DRUGGABLE GENOME Diterpenoid derivative 2 64876 44250 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE COL-3 INCYCLINIDE 64877 44251 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565842 64878 44252 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR PHA-767491 CHEMBL225519 64879 44253 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CARBARIL CARBARIL 64880 44254 TSPAN5 10098 CELL SURFACE citalopram CITALOPRAM 26903268 64881 44255 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME ANTISERUM 16870138 64884 44256 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774824-Compound-Figure7Example10 64885 44257 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER EFAVIRENZ EFAVIRENZ 21189339,17172311 64886 44258 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-N3 64887 44259 POLK 51426 DNA REPAIR, ENZYME EUPAFOLIN EUPAFOLIN 64889 44260 AREG 374 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE radiotherapy 25026457 64890 44261 IRS2 8660 KINASE, CLINICALLY ACTIONABLE DUAL IGF-1R/INSR INHIBITOR BMS-754807 25527633 64891 44262 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1201341 ECHOTHIOPHATE 64893 44263 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545027 XL-281 64896 44264 TMPRSS2 7113 CLINICALLY ACTIONABLE, PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178101079 NAFAMOSTAT 64897 44265 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME DAPHNETIN DAPHNETIN 64898 44266 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Ergocalciferol ERGOCALCIFEROL 64899 44267 BRDT 676 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE ALPRAZOLAM ALPRAZOLAM 22137933 64900 44268 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE GALLOCATECHIN GALLATE GALLOCATECHIN GALLATE 19839593 64902 44269 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Bicyclic heteroaryl benzamide derivative 4 64903 44270 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME METHYL 2-(4-FLUOROBENZAMIDO)BENZOATE CHEMBL250428 64904 44271 SLC17A9 63910 DRUGGABLE GENOME, TRANSPORTER inhibitor 340590235 64906 44272 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor PI-103 PI-103 64907 44273 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE EPINEPHRINE BITARTRATE EPINEPHRINE BITARTRATE 64909 44274 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER atenolol ATENOLOL 64913 44275 IL23A 51561 DRUGGABLE GENOME MK-3222 TILDRAKIZUMAB 64914 44276 PREP 5550 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 178103179 64918 44277 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 249565715 LEVOBETAXOLOL 64919 44278 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-43 64921 44279 MAPT 4137 DRUGGABLE GENOME TYRPHOSTIN 47 TYRPHOSTIN 47 64922 44280 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651095 SUMATRIPTAN 64923 44281 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME THALIDOMIDE THALIDOMIDE 10823791 64929 44282 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME (+)-CIS-DIOXOLANE IODIDE CHEMBL387632 64930 44283 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL3545427 CM-082 64931 44284 NCOA3 8202 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, ENZYME IRINOTECAN HYDROCHLORIDE HYDRATE IRINOTECAN HYDROCHLORIDE HYDRATE 64932 44285 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DISULFIRAM DISULFIRAM 64933 44286 UGCG 7357 ENZYME, DRUGGABLE GENOME Venglustat VENGLUSTAT 64935 44287 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR laropiprant LAROPIPRANT 26226939 64937 44288 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1200996 MEPHENTERMINE SULFATE 64938 44289 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 simeprevir SIMEPREVIR 64940 44290 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051793 GIVINOSTAT 64942 44291 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Peptidomimetic analog 5 64943 44292 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Navitoclax NAVITOCLAX 25665005,24983357 64945 44293 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METRAZOLINE OXALATE METRAZOLINE OXALATE 64946 44294 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MERSALYL MERSALYL 64949 44295 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 315661305 64951 44296 ABAT 18 DRUGGABLE GENOME, ENZYME CPP-115 CPP-115 64952 44297 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Gefitinib GEFITINIB 64953 44298 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME KX2-391 KX2-391 64954 44299 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GANGALEOIDIN GANGALEOIDIN 64955 44300 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR O-desulfated heparin 64956 44301 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135649896 64957 44302 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER EMODIN EMODIN 64958 44303 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR RHAMNETIN RHAMNETIN 24397781 64960 44304 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178102701 64963 44305 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DEZOCINE DEZOCINE 64964 44306 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR goserelin GOSERELIN 64965 44307 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE VP-16 ETOPOSIDE PHOSPHATE 15496478 64966 44308 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL10041 AFIMOXIFENE 64967 44309 CYP4A11 1579 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME amiloride AMILORIDE 64968 44310 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Tiagabine TIAGABINE 64969 44311 TUBB2A 7280 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 64970 44312 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SELEGILINE SELEGILINE 22931300 64971 44313 APC 324 CLINICALLY ACTIONABLE Sapanisertib SAPANISERTIB 25261369 64974 44314 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Medroxyprogesterone MEDROXYPROGESTERONE ACETATE 64976 44315 DHRS9 10170 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE (+)-ZONAROL CHEMBL461471 19188072 64977 44316 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SBI-0640756 26603897 64978 44317 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER gefitinib GEFITINIB 25554506,27089937 64980 44318 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PD-98059 CHEMBL35482 64981 44319 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650731 NORETHINDRONE 64982 44320 ADAM17 6868 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, NEUTRAL ZINC METALLOPEPTIDASE, TRANSPORTER, ENZYME inhibitor 178103123 CHEMBL489100 64984 44321 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER doxorubicin DOXORUBICIN 16330681 64985 44322 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 QUERCETIN QUERCETIN 64986 44323 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE (2-NITROVINYL)BENZENE (2-NITROVINYL)BENZENE 64988 44324 KLKB1 3818 DRUGGABLE GENOME, PROTEASE, ENZYME Ecallantide ECALLANTIDE 64989 44325 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 340590240 64990 44326 ITPR2 3709 ION CHANNEL, DRUGGABLE GENOME activator 178100946 64992 44327 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 L-732138 L-732138 64993 44328 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PURVALANOLA PURVALANOLA 64994 44329 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE Sulfonamide derivative 15 64996 44330 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL blocker 340590213 64997 44331 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PF-04691502 PF-04691502 65000 44332 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 405067336 65001 44333 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor ARRY380 65004 44334 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER methotrexate METHOTREXATE 25502615,23222202,25348617 65006 44335 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE RO-106-9920 CHEMBL271023 65007 44336 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 252827524 65009 44337 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLUORODIFEN FLUORODIFEN 65012 44338 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DIMETHYLADENINE DIMETHYLADENINE 65014 44339 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MALINAMIDE MALINAMIDE 65016 44340 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1256957 65017 44341 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-2272 CHEMBL601757 65019 44342 POLB 5423 DNA REPAIR, DRUGGABLE GENOME BITHIONOL BITHIONOL 65020 44343 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME ENMD-2076 ENMD-2076 65022 44344 SMN2 6607 DRUGGABLE GENOME THIABENDAZOLE THIABENDAZOLE 65023 44345 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650823 PIBOSEROD 65024 44346 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Debio 1347 65026 44347 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL inhibitor 381118829 65027 44348 RHBDF2 79651 ENZYME morphine MORPHINE 21622719 65029 44349 SLC36A1 206358 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 135651413 SEROTONIN 65032 44350 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AC480 AC-480 21576284 65033 44351 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist 135650370 FULVESTRANT 65034 44352 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME GNF-PF-2301 CHEMBL578061 65035 44353 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME 1,2-NAPHTHOQUINONE 1,2-NAPHTHOQUINONE 65036 44354 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PENTOXIFYLLINE PENTOXIFYLLINE 10363593 65037 44355 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 178102626 65039 44356 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENANTHROLINE PHENANTHROLINE 65040 44357 TUBA1B 10376 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 65041 44358 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OCTAVERINE OCTAVERINE 65044 44359 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR XL844 65045 44360 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3084748 TROSPIUM CHLORIDE 65046 44361 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor GSK2636771 GSK-2636771 65047 44362 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ESMOLOL ESMOLOL 65048 44363 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-13 65050 44364 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME SITAGLIPTIN SITAGLIPTIN 65051 44365 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME APAP ACETAMINOPHEN 16330492 65052 44366 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME HEPARIN HEPARIN 65053 44367 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE GSK933776 GSK933776 20497044 65058 44368 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE BITHIONOL BITHIONOL 65059 44369 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER EFAVIRENZ EFAVIRENZ 21189339 65060 44370 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE nimodipine NIMODIPINE 19205682 65061 44371 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CID 838877 CHEMBL405317 65062 44372 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME pemetrexed PEMETREXED 24732178,19841321,12571805 65063 44373 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE eptifibatide EPTIFIBATIDE 20938371 65064 44374 MAOA 4128 DRUGGABLE GENOME, ENZYME Tacrine-coumarin hybrid derivative 1 65065 44375 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME ANTIBIOTIC ANTIBIOTIC 15773551 65066 44376 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor 348353678 65067 44377 NEDD4 4734 ENZYME warfarin WARFARIN 27488176 65068 44378 SOAT1 6646 DRUGGABLE GENOME EMZETIBE 65070 44379 PSENEN 55851 DRUGGABLE GENOME SEMAGACESTAT SEMAGACESTAT 19443228 65071 44380 ALOX15B 247 DRUGGABLE GENOME, ENZYME TROGLITAZONE TROGLITAZONE 65072 44381 PSME4 23198 DNA REPAIR inhibitor CARFILZOMIB CARFILZOMIB 65073 44382 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE EVT 401 22547202 65074 44383 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR AMIFOSTINE AMIFOSTINE 12005544 65076 44384 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DSM-97 CHEMBL492528 65079 44385 STK16 8576 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME inhibitor 348353651 65082 44386 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor MASITINIB MASITINIB 65085 44387 ADM 133 DRUGGABLE GENOME, HORMONE ACTIVITY TPA ALTEPLASE 10848972 65086 44388 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ACROLEIN ACROLEIN 65087 44389 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 LANSOPRAZOLE SULFIDE LANSOPRAZOLE SULFIDE 65088 44390 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL29741 IRAMPANEL 65090 44391 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Avatrombopag AVATROMBOPAG 65091 44392 ALOX5 240 DRUGGABLE GENOME, ENZYME MESALAMINE MESALAMINE 65092 44393 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR FROVATRIPTAN FROVATRIPTAN 65093 44394 TARDBP 23435 TUMOR SUPPRESSOR PHYLLODULCIN PHYLLODULCIN 65094 44395 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CICLESONIDE CICLESONIDE 65095 44396 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2062265 65096 44397 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CHEMBL3545015 RAD1901 65097 44398 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME N-METHYLHISTAMINE N-METHYLHISTAMINE 65098 44399 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE RECOMBINANT INTERLEUKIN 2569954 65100 44400 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE CEDIRANIB CEDIRANIB 25218906 65101 44401 FAAH 2166 ENZYME, DRUGGABLE GENOME ibuprofen IBUPROFEN 25502615 65102 44402 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR nitrendipine NITRENDIPINE 8952600 65103 44403 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TCMDC-123641 CHEMBL532849 65104 44404 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE PONATINIB PONATINIB 24124571 65106 44405 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME ARQ 087 65108 44406 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 363894208 ILORASERTIB 65109 44407 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME Temsirolimus TEMSIROLIMUS 65111 44408 POLI 11201 DNA REPAIR LINOLENIC ACID LINOLENIC ACID 65112 44409 CCL11 6356 DRUGGABLE GENOME MOMETASONE FUROATE 12877820 65113 44410 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Rucaparib RUCAPARIB 23565244 65114 44411 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-280795 CHEMBL84281 65115 44412 KRT17 3872 NA TCDD 9036934 65117 44413 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-38 65118 44414 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NSC-348401 CHEMBL515505 65119 44415 POLK 51426 DNA REPAIR, ENZYME FISETIN FISETIN 65121 44416 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565733 65122 44417 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR TG-C 65123 44418 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME NU-2058 CHEMBL269881 65124 44419 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BROMPHENIRAMINE BROMPHENIRAMINE 65125 44420 TNFRSF9 3604 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE 178101774 65127 44421 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-43 65128 44422 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ANTISERUM 8314750 65129 44423 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL27759 ENTINOSTAT 65130 44424 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME DOX 11785103 65132 44425 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME DOVITINIB DOVITINIB 65133 44426 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3544999 SAMOTOLISIB 65134 44427 PTGS2 5743 DRUGGABLE GENOME, ENZYME APRICOXIB APRICOXIB 65136 44428 FAAH 2166 ENZYME, DRUGGABLE GENOME Pyrazole derivative 84 65139 44429 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CRIZOTINIB CRIZOTINIB 65140 44430 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME RG-1530 RG-1530 65142 44431 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME regorafenib REGORAFENIB 65143 44432 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME AMINOGLUTETHIMIDE AMINOGLUTETHIMIDE 3427227 65146 44433 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651470 DESMOSTEROL 65148 44434 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME MITOXANTRONE MITOXANTRONE 65149 44435 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1201177 LEVOBUNOLOL HYDROCHLORIDE 65150 44436 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651538 65151 44437 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME EMODIN EMODIN 65153 44438 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1256 ISOFLURANE 65154 44439 CXCL8 3576 DRUGGABLE GENOME DACARBAZINE DACARBAZINE 65155 44440 AXIN2 8313 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Platinum compounds 24980784 65157 44441 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103684 ACEBUTOLOL 65160 44442 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200940 METOCLOPRAMIDE HYDROCHLORIDE 65162 44443 PDCD4 27250 KINASE, DRUGGABLE GENOME PACLITAXEL PACLITAXEL 25928036 65166 44444 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SB-200646 CHEMBL85194 65167 44445 PLA2G7 7941 DRUGGABLE GENOME, ENZYME GSK2647544 65168 44446 HPSE 10855 ENZYME, DRUGGABLE GENOME AMOPYROQUINE AMOPYROQUINE 23415087 65169 44447 CYB5R4 51167 DRUGGABLE GENOME metoclopramide METOCLOPRAMIDE 65170 44448 BAZ2B 29994 NA ALTENUSIN ALTENUSIN 65171 44449 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1017 TELMISARTAN 65172 44450 ADH1C 126 ENZYME, DRUGGABLE GENOME abacavir ABACAVIR 24625462 65173 44451 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME EVEROLIMUS EVEROLIMUS 65174 44452 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR VIOLASTYRENE VIOLASTYRENE 65175 44453 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DAPSONE DAPSONE 22931300 65176 44454 GMNN 51053 DRUGGABLE GENOME SJ000117462 CHEMBL590427 65179 44455 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME FR167653 65180 44456 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME HINOKITIOL HINOKITIOL 65181 44457 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SECAUBRYOLIDE SECAUBRYOLIDE 65182 44458 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE DAB 6712668 65183 44459 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CNS-7056 REMIMAZOLAM 65184 44460 PSMA1 5682 PROTEASE, DRUGGABLE GENOME inhibitor BORTEZOMIB BORTEZOMIB 65186 44461 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME MITOXANTRONE MITOXANTRONE 65187 44462 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-98 65188 44463 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME INCB54707 65190 44464 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME GNF-PF-3996 CHEMBL584458 65192 44465 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 178103586 ENTINOSTAT 65194 44466 DIABLO 56616 NA NM-3 15574755 65195 44467 SOD2 6648 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE methotrexate METHOTREXATE 25330300 65196 44468 PTGS2 5743 DRUGGABLE GENOME, ENZYME RESERPINE RESERPINE 16081063 65197 44469 IRF6 3664 TRANSCRIPTION FACTOR interferon beta-1a 30013178 65198 44470 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER DROLOXIFENE DROLOXIFENE 11721384 65201 44471 SGK1 6446 SERINE THREONINE KINASE, KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 328083509 65203 44472 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PIMOZIDE PIMOZIDE 65205 44473 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME activator 135650896 EZOGABINE 65206 44474 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IVC AESCULIOSIDE IVC 20371180 65207 44475 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR HYDROXYTAMOXIFEN 65208 44476 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SORAFENIB TOSYLATE SORAFENIB TOSYLATE 65209 44477 PLA2G7 7941 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL204021 DARAPLADIB 65210 44478 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-5151 CHEMBL576208 65211 44479 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ICI 182780 17044036 65212 44480 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME GW9662 CHEMBL375270 65213 44481 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMCV 9552048 65214 44482 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME IMMUNOMODULATORS 1517537 65215 44483 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565864 65216 44484 PTGS2 5743 DRUGGABLE GENOME, ENZYME VALDECOXIB VALDECOXIB 20143779 65217 44485 ALB 213 TRANSPORTER, DRUGGABLE GENOME OLMESARTAN MEDOXOMIL OLMESARTAN MEDOXOMIL 22086979 65218 44486 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Imidazoleisoindoles derivative 2 65219 44487 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ALLITRIDIN ALLITRIDIN 65220 44488 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER RS-39604 CHEMBL66114 65221 44489 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE NILOTINIB NILOTINIB 65222 44490 PDE4B 5142 DRUGGABLE GENOME, ENZYME ENPROFYLLINE ENPROFYLLINE 65223 44491 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE MK2206 MK-2206 28178345,26187616,24265152,22025163,21289267 65224 44492 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR activator 178104015 65226 44493 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antidepressants 12815745 65227 44494 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME US9346821, B-42 65228 44495 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TAS-120 FUTIBATINIB 65230 44496 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NITROFURAZONE NITROFURAZONE 65231 44497 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TETRANITROMETHANE TETRANITROMETHANE 65232 44498 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE PT-101 CHEMBL316796 65233 44499 ATXN2 6311 NA GNF-PF-2347 CHEMBL579045 65235 44500 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tetra-hydro-isoquinoline derivative 4 65236 44501 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL clobazam CLOBAZAM 23859570,21747585,28753467,25155934 65238 44502 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME MIBEFRADIL MIBEFRADIL 65239 44503 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIHYDROXANTHOHUMOL DIHYDROXANTHOHUMOL 65240 44504 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565616 SAPANISERTIB 65241 44505 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DICHLORODIPHENYLDICHLOROETHYLENE DICHLORODIPHENYLDICHLOROETHYLENE 65242 44506 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 5-FLUOROURIDINE CHEMBL54918 65243 44507 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NSC-317605 CHEMBL1312050 65244 44508 E2F1 1869 TRANSCRIPTION FACTOR ARQ-171 65246 44509 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE TAE-684 TAE-684 65247 44510 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME LACTACYSTIN LACTACYSTIN 23547757 65248 44511 ARSA 410 DRUGGABLE GENOME, ENZYME MITOXANTRONE MITOXANTRONE 65250 44512 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL970 HALAZEPAM 65251 44513 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME 2-PHENYLPHENOL 2-PHENYLPHENOL 65252 44514 HSPB2 3316 KINASE HERCEPTIN HERCEPTIN 16048908 65253 44515 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 384403673 65254 44516 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NANAOMYCIN NANAOMYCIN 65255 44517 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Regorafenib REGORAFENIB 23629727,25838391 65257 44518 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METHOTREXATE METHOTREXATE 65260 44519 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BINOSPIRONE BINOSPIRONE 65261 44520 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 65262 44521 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME Quizartinib QUIZARTINIB 65263 44522 ABCC9 10060 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER CHEMBL802 MINOXIDIL 65264 44523 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL OXAZEPAM OXAZEPAM 65265 44524 MAPT 4137 DRUGGABLE GENOME PANTOPRAZOLE PANTOPRAZOLE 65269 44525 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2106698 65270 44526 GLS 2744 ENZYME PIRENOXINE PIRENOXINE 65271 44527 HMGCR 3156 ENZYME, DRUGGABLE GENOME HMG-CoA reductase inhibitor 65272 44528 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Viramidine TARIBAVIRIN HYDROCHLORIDE 65273 44529 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR YM-16151-4 65274 44530 GBA 2629 DRUGGABLE GENOME, ENZYME Taliglucerase alfa 65275 44531 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650857 PROPANTHELINE 65281 44532 SIRT3 23410 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 252827436 65283 44533 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BUTANOIC ACID BUTANOIC ACID 19053749 65284 44534 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE pitavastatin PITAVASTATIN 23007012 65286 44535 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100669 65287 44536 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME inhibitor 249565595 LCL-161 65288 44537 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR letrozole LETROZOLE 26536870 65290 44538 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 65291 44539 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME (RS)-ROSCOVITINE (RS)-ROSCOVITINE 65293 44540 CLCN3 1182 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE, TRANSPORTER CINOBUFAGIN CINOBUFAGIN 23799775 65295 44541 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TAMATINIB R-406 65296 44542 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE LIGNAN 12085264 65297 44543 ALOX15 246 ENZYME, DRUGGABLE GENOME PMID26560362-Compound-90 65298 44544 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Axitirome AXITIROME 23667826 65299 44545 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Isoflavone derivative 6 65301 44546 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER itraconazole ITRACONAZOLE 65302 44547 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1200387 AMPHETAMINE ADIPATE 65303 44548 KDM4A 9682 DRUGGABLE GENOME, ENZYME BAS03450373 CHEMBL1576310 65304 44549 GUCY1B1 2983 DRUGGABLE GENOME Cinaciguat CINACIGUAT 65307 44550 NDUFB6 4712 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 65308 44551 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CD19 and CD20 CAR-T Cells 65310 44552 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME SJ000047240 CHEMBL590706 65311 44553 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 363894179 65313 44554 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 387065609 65314 44555 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME IBRITUMOMAB TIUXETAN 65315 44556 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME CYC-116 CYC-116 65317 44557 FAAH 2166 ENZYME, DRUGGABLE GENOME PF-04457845 PF-04457845 21666860 65320 44558 CTSD 1509 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 404859127 65322 44559 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-11 65323 44560 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EFONIDIPINE EFONIDIPINE 65324 44561 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-747266 CHEMBL609570 65326 44562 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR CDP-6038 OLOKIZUMAB 65327 44563 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE AC-100,DENTONIN 65328 44564 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PONATINIB PONATINIB 65329 44565 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AMITHIOZONE AMITHIOZONE 65331 44566 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 6-CHLOROFLAVONE 6-CHLOROFLAVONE 65333 44567 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE vorinostat VORINOSTAT 22693356,9661880 65334 44568 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE RAFAMETINIB 65336 44569 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Naveglitazar NAVEGLITAZAR 65337 44570 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545083 RGB-286638 65339 44571 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-13 65341 44572 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 385612236 ALFLUTINIB 65342 44573 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SCATTER FACTOR 11909963 65343 44574 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID28048944-Compound-4 65345 44575 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AZATHIOPRINE AZATHIOPRINE 22931300 65346 44576 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 223366204 COPANLISIB 65347 44577 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 249565592 GANDOTINIB 65348 44578 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE ERLOTINIB ERLOTINIB 65351 44579 CYB5R3 1727 DRUGGABLE GENOME, ENZYME oxymetazoline and tetracaine 65352 44580 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 65353 44581 HTT 3064 DRUGGABLE GENOME CLIOQUINOL CLIOQUINOL 65356 44582 MPHOSPH8 54737 NA 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 65357 44583 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RO-23-7553 ILX23-7553 65359 44584 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME RO-137410 CHEMBL275311 18951029 65360 44585 NUBPL 80224 NA iloperidone ILOPERIDONE 18521091 65361 44586 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MESO-HEXESTROL MESO-HEXESTROL 65362 44587 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE MEGAKARYOCYTE GROWTH AND DEVELOPMENT FACTOR 9531338 65364 44588 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ITRACONAZOLE ITRACONAZOLE 17923278 65365 44589 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor SODIUM PHENYLBUTYRATE 65367 44590 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SULFINPYRAZONE SULFINPYRAZONE 65368 44591 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME inhibitor 405560329 65369 44592 KDM5C 8242 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 178103606 65370 44593 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME DIMETHYL YELLOW DIMETHYL YELLOW 65371 44594 APC 324 CLINICALLY ACTIONABLE JW55 22440753 65375 44595 HMGCR 3156 ENZYME, DRUGGABLE GENOME TOCOTRIENOL TOCOTRIENOL 65377 44596 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE DABRAFENIB DABRAFENIB 24265155 65378 44597 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FP-045 65380 44598 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL1683544 ERIBULIN MESYLATE 65381 44599 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ESTRADIOL ESTRADIOL 65382 44600 ATAD5 79915 NA TETRABROMOBENZOTRIAZOLE TETRABROMOBENZOTRIAZOLE 65383 44601 BAZ2B 29994 NA PHENANTHROLINE PHENANTHROLINE 65384 44602 KDM4A 9682 DRUGGABLE GENOME, ENZYME CYCLOVALONE CYCLOVALONE 65385 44603 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ZAPA ZAPA 65386 44604 HMGCR 3156 ENZYME, DRUGGABLE GENOME Premarin/Pravachol 65388 44605 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL6 INDOMETHACIN 65389 44606 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME TRIIODOTHYRONINE LIOTHYRONINE SODIUM 7642172 65390 44607 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Estradiol ESTRADIOL 65391 44608 POLL 27343 NA JUGLONE JUGLONE 21903399 65393 44609 MAP2K3 5606 KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE inhibitor PD 0325901 65396 44610 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101500 SERTRALINE 65397 44611 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR modulator CHEMBL267431 ASOPRISNIL 65398 44612 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1200870 TIMOLOL MALEATE 65400 44613 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 3',4'-DIHYDROXYFLAVONE CHEMBL222556 65401 44614 PNPLA3 80339 ENZYME asparaginase ASPARAGINASE 28744905 65402 44615 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ETOPOSIDE ETOPOSIDE 11350408,14977850 65403 44616 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL2107358 OBATOCLAX MESYLATE 65406 44617 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ANTI-EGFR MONOCLONAL ANTIBODY 23729478 65407 44618 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR CUDC-101 CUDC-101 65408 44619 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor 178103171 65409 44620 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL3544971 DEXTROAMPHETAMINE SULFATE 65410 44621 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROMETHAZINE PROMETHAZINE 65411 44622 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KD-3020 65414 44623 CCL2 6347 DRUGGABLE GENOME risperidone RISPERIDONE 24495780 65416 44624 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ETHYNODIOL DIACETATE ETHYNODIOL DIACETATE 65417 44625 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER talinolol TALINOLOL 22725663 65418 44626 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (R)-FELODIPINE (R)-FELODIPINE 65419 44627 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor PELITINIB PELITINIB 65424 44628 BRCA2 675 CLINICALLY ACTIONABLE Veliparib VELIPARIB 26801247,25589624,26842236 65426 44629 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME inhibitor 178103690 AMLEXANOX 65429 44630 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 23622981 65430 44631 PVT1 5820 NA GLIVEC GLIVEC 15251464 65431 44632 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE KENPAULLONE KENPAULLONE 65432 44633 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR U-0126 U-0126 65433 44634 TSPO 706 DRUGGABLE GENOME Quinazoline derivative 6 65434 44635 PADI3 51702 ENZYME, DRUGGABLE GENOME O-CL-AMIDINE CHEMBL1910971 21882827 65435 44636 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US10100051, Compound 2 65436 44637 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL3545049 BAY-1125976 65437 44638 TMEM97 27346 NA PMID28051882-Compound-XI 65441 44639 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME NG2-73 ADIPIPLON 65443 44640 TMSB10 9168 NA PMSG 1989873 65444 44641 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GEMFIBROZIL GEMFIBROZIL 65446 44642 GMNN 51053 DRUGGABLE GENOME SULBENTINE SULBENTINE 65447 44643 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE IMX-110 65448 44644 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 65449 44645 CBX1 10951 NA DIAMIDE DIAMIDE 65450 44646 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME PALBOCICLIB PALBOCICLIB 65452 44647 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME ERYTHROPOIETIN EPOETIN BETA 65453 44648 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BENZBROMARONE BENZBROMARONE 65455 44649 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME fluvastatin FLUVASTATIN 65456 44650 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-123912 CHEMBL106525 65457 44651 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 2-MERCAPTOBENZOTHIAZOLE 2-MERCAPTOBENZOTHIAZOLE 65458 44652 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL563 FLURBIPROFEN 65459 44653 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER taxanes 19203783,12684679 65460 44654 SLC1A5 6510 TRANSPORTER inhibitor 178101228 65461 44655 MUC5AC 4586 DRUGGABLE GENOME GLUCOCORTICOID 11411550 65462 44656 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE AXL1717 65463 44657 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CETRIMIDE CETRIMIDE 65467 44658 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Danusertib DANUSERTIB 26725216 65469 44659 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ENALAPRIL ENALAPRIL 16900775 65470 44660 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PD-0166285 PD-0166285 65471 44661 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565621 MILCICLIB 65473 44662 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DICHLORVOS DICHLORVOS 65474 44663 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME KENPAULLONE KENPAULLONE 65475 44664 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME BMS-387032 BMS-387032 65476 44665 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR AZD7762 AZD-7762 65477 44666 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IVB AESCULIOSIDE IVB 20371180 65479 44667 BAZ2B 29994 NA CEFOXITIN SODIUM CEFOXITIN SODIUM 65480 44668 HSPA4 3308 NA Minnelide 001 65481 44669 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417031 CHEMBL1333049 65482 44670 ALOX15B 247 DRUGGABLE GENOME, ENZYME HINOKITIOL HINOKITIOL 65483 44671 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650581 METERGOLINE 65485 44672 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649666 65488 44673 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME AG-537 CHEMBL67535 65489 44674 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME IL-2 ALDESLEUKIN 1668889,1472476 65490 44675 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR ITRACONAZOLE ITRACONAZOLE 14639950 65492 44676 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME SODIUM SALICYLATE 14634277 65493 44677 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-308 CHEMBL600334 65495 44678 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER phenothiazines with aliphatic side-chain 65496 44679 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BETA-LAPACHONE LAPACHONE 65497 44680 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102585 DOVITINIB 65498 44681 PEMT 10400 ENZYME CHEMBL2109361 PEMTUMOMAB 65500 44682 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ACETAMINOPHEN ACETAMINOPHEN 22931300 65501 44683 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-107022 CHEMBL1601846 65502 44684 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MURAGLITAZAR MURAGLITAZAR 65504 44685 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor PELITINIB PELITINIB 65505 44686 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Quinazoline alkaloid derivative 1 65506 44687 CA2 760 DRUGGABLE GENOME, ENZYME TOPIRAMATE TOPIRAMATE 65507 44688 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BETAMETHASONE VALERATE BETAMETHASONE VALERATE 65508 44689 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE PURVALANOL B PURVALANOL B 65509 44690 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650357 65513 44691 ATAD5 79915 NA MITOXANTRONE MITOXANTRONE 65514 44692 IFNG 3458 DRUGGABLE GENOME URSODEOXYCHOLIC ACID 10784002 65516 44693 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor GDC-0068 IPATASERTIB 65517 44694 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SB-203580 SB-203580 65518 44695 PTGS1 5742 ENZYME, DRUGGABLE GENOME antiinflammatory and antirheumatic products, non-steroids 22336956 65519 44696 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GENTIAN VIOLET GENTIAN VIOLET 65520 44697 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME L-750667 CHEMBL1256738 65521 44698 HSPA4 3308 NA HEPARIN HEPARIN 7548155 65523 44699 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-16736 CHEMBL1728978 65525 44700 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE PROGESTERONE PROGESTERONE 17068109 65526 44701 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DEFERIPRONE DEFERIPRONE 65528 44702 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Dacinostat DACINOSTAT 27443263 65529 44703 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER APR-246 APR-246 65530 44704 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRICIRIBINE TRICIRIBINE 65531 44705 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist CHEMBL806 FLUTAMIDE 65532 44706 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 384403638 65534 44707 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME HALOPERIDOL HALOPERIDOL 11490180 65536 44708 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL24828 VANDETANIB 65538 44709 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL377300 BRIVANIB 65539 44710 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545384 SB-85635 65541 44711 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 lovastatin LOVASTATIN 65545 44712 TUBB3 10381 DRUGGABLE GENOME DOCETAXEL DOCETAXEL 65548 44713 GMNN 51053 DRUGGABLE GENOME ELLIPTECINE ELLIPTECINE 65549 44714 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1650 CORTISONE ACETATE 65550 44715 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 178102328 PI-103 65551 44716 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BITHIONOL BITHIONOL 65552 44717 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME VASOPRESSIN VASOPRESSIN 10679516,11029753 65554 44718 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651308 65555 44719 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 404859096 65558 44720 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Pyrimidine derivative 33 65559 44721 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ONC1-13B 65560 44722 PON1 5444 ENZYME, TRANSPORTER, DRUGGABLE GENOME atorvastatin ATORVASTATIN 18430057,16238680,19904013 65561 44723 TARDBP 23435 TUMOR SUPPRESSOR CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 65562 44724 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Clenbuterol CLENBUTEROL 65563 44725 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BAY1000394 65564 44726 CBR1 873 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 65565 44727 AK4 205 ENZYME, KINASE adefovir dipivoxil 65567 44728 HSPB1 3315 DRUGGABLE GENOME OGX-427 APATORSEN 65568 44729 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE SEMAGACESTAT SEMAGACESTAT 65571 44730 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103484 65572 44731 DROSHA 29102 NA cytarabine CYTARABINE 24614921 65575 44732 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ethanol ALCOHOL 65576 44733 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Fulvestrant FULVESTRANT 65577 44734 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME PHA-767491 CHEMBL225519 65578 44735 PDF 64146 DRUGGABLE GENOME LY333531 65583 44736 TUBA1A 7846 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 65585 44737 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR BUTANOIC ACID BUTANOIC ACID 19053749 65586 44738 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor ICOTINIB ICOTINIB 65587 44739 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR BENZO(K)FLUORANTHENE BENZO(K)FLUORANTHENE 65589 44740 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE BGC-20-1531 19154437 65590 44741 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL70418 CLOBAZAM 65591 44742 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME ME-344 ME-344 65592 44743 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TOLFENAMIC ACID TOLFENAMIC ACID 65593 44744 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Epoxysuccinate derivative 7 65595 44745 RBMS3 27303 NA Bisphosphonates 65598 44746 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 135650118 COLCHICINE 65599 44747 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GW501516 GW501516 65600 44748 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ETHANOL ALCOHOL 8986223 65602 44749 CPS1 1373 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME valproic acid 20456087 65604 44750 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME 3,8'-BIAPIGENIN CHEMBL515252 65605 44751 PPM1D 8493 KINASE, SERINE THREONINE KINASE, ENZYME DOXORUBICIN DOXORUBICIN 25466181 65606 44752 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL1201752 IXABEPILONE 65608 44753 TUBA1B 10376 DRUGGABLE GENOME CHEMBL2103826 DAVUNETIDE 65610 44754 BAZ2B 29994 NA DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 65611 44755 ALOX5 240 DRUGGABLE GENOME, ENZYME 6-PENTYLSALICYLIC ACID CHEMBL502496 24231650 65612 44756 TMPRSS6 164656 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166825 65613 44757 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR CONICASTEROL E CONICASTEROL E 22126372 65616 44758 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER cytarabine CYTARABINE 26842729 65617 44759 NOS1 4842 DRUGGABLE GENOME, ENZYME TRIIODOTHYRONINE LIOTHYRONINE SODIUM 9466951 65618 44760 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE fenofibrate FENOFIBRATE 65619 44761 ALOX15 246 ENZYME, DRUGGABLE GENOME QUINALIZARIN QUINALIZARIN 65621 44762 NOS1AP 9722 NA granisetron GRANISETRON 21663814 65624 44763 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME GW441756X GW441756X 65625 44764 CPS1 1373 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Sodium Phenylbutyrate 65626 44765 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL2109377 PAMREVLUMAB 65627 44766 CBX1 10951 NA GUAIAZULENE GUAIAZULEN 65628 44767 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR REPOTRECTINIB REPOTRECTINIB 30093503 65629 44768 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GO-6976 GO-6976 65630 44769 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME trametinib TRAMETINIB 65631 44770 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OMEPRAZOLE OMEPRAZOLE 9395520 65632 44771 KDM4A 9682 DRUGGABLE GENOME, ENZYME IODOQUINOL IODOQUINOL 65636 44772 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR GATIFLOXACIN GATIFLOXACIN 65637 44773 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GNF-PF-5510 CHEMBL578741 65639 44774 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TRAMADOL TRAMADOL 65640 44775 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor ABT-888 VELIPARIB 65641 44776 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL628 PENTOXIFYLLINE 65642 44777 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-123808 CHEMBL546493 65643 44778 NRP1 8829 DRUGGABLE GENOME antagonist 363894198 65644 44779 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TRAZODONE HYDROCHLORIDE TRAZODONE HYDROCHLORIDE 65645 44780 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL1742994 BRENTUXIMAB VEDOTIN 65646 44781 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR JX-594 PEXASTIMOGENE DEVACIREPVEC 65647 44782 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE DOVITINIB DOVITINIB 65648 44783 GMNN 51053 DRUGGABLE GENOME GNF-PF-4576 CHEMBL527336 65649 44784 RAB9A 9367 ENZYME, DRUGGABLE GENOME ACACETIN ACACETIN 65650 44785 BAZ2B 29994 NA PURPUROGALLIN PURPUROGALLIN 65651 44786 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR BMS-345541 BMS-345541 65652 44787 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME ALPRAZOLAM ALPRAZOLAM 65653 44788 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Steroid derivative 4 65654 44789 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE HEPARIN HEPARIN 9521691,2457642 65657 44790 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PRACINOSTAT PRACINOSTAT 65658 44791 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL646 TRIAZOLAM 65659 44792 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor PAZOPANIB PAZOPANIB 65663 44793 RAB9A 9367 ENZYME, DRUGGABLE GENOME 10-METHOXYLRUTAECARPINE CHEMBL85826 65664 44794 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VINCRISTINE VINCRISTINE 9494516 65665 44795 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-31 65668 44796 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 135651381 65670 44797 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 249565739 AZD-6482 65671 44798 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 7,8-DIHYDROXYFLAVONE 7,8-DIHYDROXYFLAVONE 65672 44799 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PHENANTHROLINE PHENANTHROLINE 65673 44800 IL1B 3553 KINASE, DRUGGABLE GENOME POLYVALENT VACCINE 12909408 65674 44801 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1194 PRILOCAINE 65675 44802 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE Menthol MENTHOL 65678 44803 BSG 682 DRUGGABLE GENOME, TRANSPORTER CHEMBL2109193 GAVILIMOMAB 65679 44804 ALOX15 246 ENZYME, DRUGGABLE GENOME TYRPHOSTIN 47 TYRPHOSTIN 47 65680 44805 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HOMIDIUM BROMIDE HOMIDIUM BROMIDE 65681 44806 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor DOVITINIB DOVITINIB 65682 44807 BRCA2 675 CLINICALLY ACTIONABLE Carboplatin CARBOPLATIN 65685 44808 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PHENOXYBENZAMINE PHENOXYBENZAMINE 65687 44809 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL HALAZEPAM HALAZEPAM 65689 44810 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SYM-004 FUTUXIMAB 65692 44811 NUDT15 55270 ENZYME, CLINICALLY ACTIONABLE MERCAPTOPURINE MERCAPTOPURINE 26878724 65696 44812 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME 3-METHYLCHOLANTHRENE 3-METHYLCHOLANTHRENE 65697 44813 POLB 5423 DNA REPAIR, DRUGGABLE GENOME THIOLACTOMYCIN THIOLACTOMYCIN 65698 44814 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-L1 65701 44815 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178103795 MEPERIDINE 65702 44816 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 374883849 TRIFAROTENE 65703 44817 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE IRESSA IRESSA 16263158 65704 44818 STAG2 10735 CLINICALLY ACTIONABLE, DRUG RESISTANCE VEMURAFENIB VEMURAFENIB 27500726 65705 44819 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody MM-111 MM-111 65706 44820 ACTR2 10097 NA ETOPOSIDE ETOPOSIDE 15900709 65707 44821 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CHLORHEXIDINE CHLORHEXIDINE 65709 44822 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 24456004 65714 44823 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER ANNAMYCIN ANNAMYCIN 9096663 65719 44824 FABP1 2168 DRUGGABLE GENOME CLOFIBRATE CLOFIBRATE 2328261 65721 44825 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME AMG 232 65722 44826 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 336446935 PREXASERTIB 65723 44827 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME ketamine KETAMINE 25702819,17638512,11470993 65724 44828 ALOX15 246 ENZYME, DRUGGABLE GENOME DACTINOMYCIN DACTINOMYCIN 65725 44829 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME ANTISENSE OLIGONUCLEOTIDES 11746820 65726 44830 ATXN2 6311 NA BAY-11-7082 CHEMBL403183 65727 44831 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CINOLAZEPAM CINOLAZEPAM 65728 44832 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL NALTREXONE NALTREXONE 65729 44833 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME perindopril PERINDOPRIL 20712529 65730 44834 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32a 65732 44835 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE CGS-15943 CGS-15943 65733 44836 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME atazanavir / ritonavir 22661571,24516079,17058217,22179231,16170755,23548653,21348813,20504240,21317582,17148966 65734 44837 PTGS1 5742 ENZYME, DRUGGABLE GENOME VB-201 VB-201 65735 44838 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IODOACETAMIDE IODOACETAMIDE 65736 44839 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 65738 44840 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME TF2 65739 44841 ALOX5 240 DRUGGABLE GENOME, ENZYME GLUCOCORTICOID 10668425 65740 44842 KCNA7 3743 ION CHANNEL, DRUGGABLE GENOME blocker 135651249 65741 44843 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME AFUTUZUMAB OBINUTUZUMAB 65743 44844 ALDH1A1 216 DRUGGABLE GENOME, ENZYME THIOPHANATE METHYL THIOPHANATE METHYL 65744 44845 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GNF-PF-4157 CHEMBL584905 65746 44846 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL2040682 CICLESONIDE 65747 44847 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102546 ALOISINE 65750 44848 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLEMIZOLE CLEMIZOLE 65752 44849 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL503 LOVASTATIN 65753 44850 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor BAY869766 65759 44851 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR FLAVONE ACETIC ACID 8512819 65760 44852 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1068 OXCARBAZEPINE 65762 44853 CBX1 10951 NA 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 65763 44854 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 27845419 65765 44855 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TANESPIMYCIN TANESPIMYCIN 25277067,23520985,22480433,21920765,21764310 65768 44856 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BI-87E7 CHEMBL523200 65770 44857 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE G1T28-1 G1T28-1 65771 44858 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IBUDILAST IBUDILAST 65775 44859 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE TRIAMTERENE TRIAMTERENE 65776 44860 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Deuterated 3-cyanoquinoline derivative 1 65777 44861 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SB-222200 SB-222200 65780 44862 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 VALPROIC ACID VALPROIC ACID 22931300 65781 44863 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE DASATINIB DASATINIB 65782 44864 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-27 65784 44865 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME Candoxatril CANDOXATRIL 65785 44866 ADAM17 6868 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, NEUTRAL ZINC METALLOPEPTIDASE, TRANSPORTER, ENZYME INCB7839 65786 44867 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DYCLONINE HYDROCHLORIDE DYCLONINE HYDROCHLORIDE 65789 44868 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PYRIDOSTIGMINE PYRIDOSTIGMINE 22931300 65790 44869 FAAH 2166 ENZYME, DRUGGABLE GENOME PMID26413912-Compound-84 65794 44870 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 404859026 65797 44871 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GO-6976 GO-6976 65798 44872 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME EPZ004777 21741596 65800 44873 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PLUMBAGIN PLUMBAGIN 65801 44874 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BEZ235 DACTOLISIB 26137449 65803 44875 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RHETSININE RHETSININE 65804 44876 ROR1 4919 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CELL SURFACE ROR1R-CAR-T Cell 65806 44877 NOS1 4842 DRUGGABLE GENOME, ENZYME inhibitor 178101806 65807 44878 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE ENMD-2076 ENMD-2076 65808 44879 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE Aminocaproic Acid 65811 44880 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME SJ000120515 CHEMBL592314 65813 44881 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE MECLOFENAMATE SODIUM MECLOFENAMATE SODIUM 65814 44882 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3544931 TAK-659 65815 44883 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHA-793887 PHA-793887 65816 44884 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1201132 NALBUPHINE HYDROCHLORIDE 65818 44885 RGS4 5999 DRUGGABLE GENOME NSC-95397 CHEMBL429095 65820 44886 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor RIBOCICLIB RIBOCICLIB 65821 44887 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 363894207 FLUMATINIB 65822 44888 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SULINDAC SULFOXIDE SULINDAC SULFOXIDE 65824 44889 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545358 4SC-203 65827 44890 MAPT 4137 DRUGGABLE GENOME DNDI1417773 CHEMBL1379900 65829 44891 MAPT 4137 DRUGGABLE GENOME SJ000147784 CHEMBL590186 65830 44892 ATXN2 6311 NA FANCHININ FANCHININ 65831 44893 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 6 65834 44894 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FLUTAMIDE FLUTAMIDE 22931300 65835 44895 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR KINASE INHIBITOR 11881120 65836 44896 POLK 51426 DNA REPAIR, ENZYME TANSHINONE I TANSHINONE I 65837 44897 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ETHOFUMESATE ETHOFUMESATE 65838 44898 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-21 65839 44899 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702259 FUTIBATINIB 65840 44900 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Sulfonamide derivative 9 65842 44901 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-2272 CHEMBL601757 65844 44902 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME KENPAULLONE KENPAULLONE 65848 44903 TARDBP 23435 TUMOR SUPPRESSOR 4'-HYDROXYPHENYL-BENZO[D]THIAZOLE CHEMBL47875 65849 44904 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PHENIRAMINE PHENIRAMINE 65850 44905 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CLOZAPINE CLOZAPINE 65851 44906 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUTAMIDE FLUTAMIDE 65855 44907 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL1908391 MASITINIB 65856 44908 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650333 CHEMBL59030 65857 44909 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ELLAGIC ACID ELLAGIC ACID 65858 44910 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME allosteric modulator 336446946 65859 44911 EZH1 2145 METHYL TRANSFERASE, ENZYME DS-3201 65860 44912 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LY-2456302 ATICAPRANT 65862 44913 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-123916 CHEMBL493863 65866 44914 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE talazoparib TALAZOPARIB 65868 44915 HIPK1 204851 TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 135652717 STAUROSPORINE 65869 44916 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE DIMETHYLCURCUMIN DIMETHYLCURCUMIN 25753330 65870 44917 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166888 65871 44918 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178102274 65872 44919 CXCL8 3576 DRUGGABLE GENOME DINITRO CRESOL DINITRO CRESOL 65873 44920 NQO2 4835 DRUGGABLE GENOME, ENZYME Prolarix 65875 44921 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-228155 CHEMBL505670 65876 44922 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor 249565683 BERZOSERTIB 65877 44923 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE Lumacaftor + ivacaftor 65879 44924 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME QUERCETIN QUERCETIN 65880 44925 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 VANOXERINE VANOXERINE 65881 44926 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MAPROTILINE MAPROTILINE 65882 44927 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SELENIUM 12949386,16632891 65884 44928 GMNN 51053 DRUGGABLE GENOME FLUPHENAZINE HYDROCHLORIDE FLUPHENAZINE HYDROCHLORIDE 65885 44929 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NILUTAMIDE NILUTAMIDE 65886 44930 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417400 CHEMBL1362503 65887 44931 MGAT4A 11320 DRUGGABLE GENOME cetuximab CETUXIMAB 26222057 65888 44932 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652034 65889 44933 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ILOPROST ILOPROST 65890 44934 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125488 METHOTREXATE 65892 44935 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3545169 AZD1305 65894 44936 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME CAR-T Cells targeting MUCI 65896 44937 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SB-415286 CHEMBL322970 65898 44938 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TAMOXIFEN CITRATE TAMOXIFEN CITRATE 65899 44939 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE NITROGEN MUSTARD 16417271 65900 44940 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1642 IMATINIB MESYLATE 65901 44941 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SELECTIVE ESTROGEN RECEPTOR MODULATORS 15755852 65902 44942 MAGEA3 4102 ENZYME, DRUGGABLE GENOME INCOMPLETE FREUND'S ADJUVANT 10546159 65903 44943 CDH1 999 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Capecitabine CAPECITABINE 26487584 65904 44944 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR SALIRASIB SALIRASIB 65905 44945 CYBB 1536 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME, ENZYME CHRYSIN CHRYSIN 23786520 65906 44946 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 252166589 PF-00489791 65908 44947 TNKS2 80351 DRUGGABLE GENOME, ENZYME inhibitor 404859118 65910 44948 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649867 A-119637 65912 44949 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-7 65913 44950 FAAH 2166 ENZYME, DRUGGABLE GENOME Aryl urea derivative 4 65915 44951 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR CYTOKINES 18088439 65916 44952 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 223365978 AEE-788 65918 44953 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Panobinostat PANOBINOSTAT 21464044 65919 44954 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LY-367265 CHEMBL1079460 65920 44955 ALDH1A1 216 DRUGGABLE GENOME, ENZYME APIGENIN APIGENIN 65922 44956 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE JNJ-26483327 JNJ-26483327 65924 44957 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 404859031 65925 44958 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE CHMFL-KIT-031 29340041 65926 44959 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NOREPINEPHRINE NOREPINEPHRINE 65928 44960 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-58 65929 44961 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE BAY1125976 27699769 65930 44962 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL2326966 SF-1126 65931 44963 PSMA7 5688 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL451887 CARFILZOMIB 65934 44964 ALOX5AP 241 DRUGGABLE GENOME inhibitor CHEMBL1922673 FIBOFLAPON SODIUM 65935 44965 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ISOVELLERAL ISOVELLERAL 65936 44966 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PD 0332991 65937 44967 CA2 760 DRUGGABLE GENOME, ENZYME TRICHLORMETHIAZIDE TRICHLORMETHIAZIDE 65938 44968 PDE4B 5142 DRUGGABLE GENOME, ENZYME Oglemilast OGLEMILAST 18660832 65940 44969 TNFRSF11B 4982 DRUGGABLE GENOME RISEDRONATE RISEDRONIC ACID 15777635 65941 44970 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL3545428 CHIAURANIB 65942 44971 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME Motexafin lutetium 65943 44972 THBD 7056 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME warfarin WARFARIN 24602049 65944 44973 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650095 CICLOPROLOL 65945 44974 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL3545154 POZIOTINIB 65946 44975 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1201068 PROPIOMAZINE HYDROCHLORIDE 65947 44976 RORA 6095 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE T091317 T091317 65949 44977 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CARBOPLATIN CARBOPLATIN 16275998 65950 44978 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MESORIDAZINE MESORIDAZINE 65951 44979 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE MLN-8054 MLN-8054 17360485 65952 44980 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME MIDAZOLAM MIDAZOLAM 22137933 65953 44981 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 178103458 VORINOSTAT 65954 44982 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIETHYLSTILBESTROL DIETHYLSTILBESTROL 22931300 65955 44983 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE CYC-116 CYC-116 65956 44984 PLD2 5338 ENZYME, DRUGGABLE GENOME activator 178101987 65957 44985 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LUFENURON LUFENURON 65958 44986 KDM4A 9682 DRUGGABLE GENOME, ENZYME (+/-)-OCTOCLOTHEPIN MALEATE CHEMBL1256660 65959 44987 ALOX15B 247 DRUGGABLE GENOME, ENZYME ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 65960 44988 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650124 CHEMBL159332 65961 44989 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 2 65963 44990 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE U-37883A CHEMBL333121 65965 44991 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PHA-767491 CHEMBL225519 65966 44992 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178101923 ACETAMINOPHEN 65969 44993 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE Famitinib FAMITINIB 65970 44994 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker 135650114 CLOTRIMAZOLE 65972 44995 DCN 1634 DRUGGABLE GENOME HSP70 9292805 65975 44996 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CLOCAPRAMINE CLOCAPRAMINE 65977 44997 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE cyclosporine CYCLOSPORINE 25163792,28624888 65979 44998 TUBB3 10381 DRUGGABLE GENOME CHEMBL2103826 DAVUNETIDE 65980 44999 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME STAUROSPORINE STAUROSPORINE 1444457 65982 45000 TSPYL2 64061 NA RETINOIC ACID 15823505 65983 45001 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME CHIR-99021 CHIR-99021 65985 45002 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103115 FASIDOTRIL 65986 45003 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE PIMASERTIB PIMASERTIB 65987 45004 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE allosteric modulator 310264743 ASCIMINIB 65988 45005 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SALICYLHYDROXAMIC ACID SALICYLHYDROXAMIC ACID 65993 45006 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CHEMBL407 FLUMAZENIL 65994 45007 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ANTICONVULSANTS 14749549 65995 45008 ALOX15 246 ENZYME, DRUGGABLE GENOME E319 E319 65996 45009 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PIRARUBICIN PIRARUBICIN 65998 45010 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166813 66000 45011 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565830 GSK-579289A 66001 45012 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE VITAMIN K 1440518 66002 45013 CA5B 11238 DRUGGABLE GENOME inhibitor CHEMBL18 ETHOXZOLAMIDE 66003 45014 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME dabrafenib DABRAFENIB 66005 45015 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor 178101525 RESERPINE 66006 45016 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE XL820 66007 45017 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PATULIN PATULIN 66009 45018 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SAPPANONE A 7-METHYL ETHER SAPPANONE A 7-METHYL ETHER 66010 45019 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL Selective serotonin reuptake inhibitors 23394390 66011 45020 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Zosuquidar ZOSUQUIDAR 66012 45021 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 318164802 66013 45022 ALOX15 246 ENZYME, DRUGGABLE GENOME 7,8-DIHYDROXYISOFLAVONE CHEMBL241813 17869117 66014 45023 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PSAMMAPLIN A PSAMMAPLIN A 23030799,25884112 66015 45024 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 trimethoprim TRIMETHOPRIM 9187528 66016 45025 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER fluvoxamine FLUVOXAMINE 18215618,26704739,22641028 66017 45026 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 U-50488 METHANE SULFONATE U-50488 METHANE SULFONATE 66018 45027 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL1230609 FORETINIB 66019 45028 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20100022547C82 66021 45029 NOX1 27035 ION CHANNEL, ENZYME, TRANSPORTER, DRUGGABLE GENOME inhibitor 363894227 66022 45030 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME bosutinib BOSUTINIB 66024 45031 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545300 CP-459632 66025 45032 IL23A 51561 DRUGGABLE GENOME Risankizumab RISANKIZUMAB 66026 45033 LGR4 55366 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100588 66029 45034 MPHOSPH8 54737 NA DIHYDREXIDINE HYDROCHLORIDE DIHYDREXIDINE HYDROCHLORIDE 66030 45035 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 310264723 EDICOTINIB 66032 45036 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIPYRIDAMOLE DIPYRIDAMOLE 66033 45037 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 5-NITROACENAPHTHENE CHEMBL423081 66035 45038 PROS1 5627 DRUGGABLE GENOME MENADIONE MENADIONE 66036 45039 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650869 QUETIAPINE 66037 45040 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heteroaryl-carboxamide derivative 2 66038 45041 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ATROPINE ATROPINE 15345469 66039 45042 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE STREPTONIGRIN STREPTONIGRIN 66040 45043 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER isoniazid ISONIAZID 19686464,22162992,29036176 66041 45044 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178103793 66044 45045 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME 178101458 66045 45046 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MITOXANTRONE MITOXANTRONE 66046 45047 AGBL4 84871 PROTEASE, DRUGGABLE GENOME rifampin RIFAMPIN 66047 45048 SMG1 23049 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DNA REPAIR inhibitor 252827484 66048 45049 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE COUMAPHOS COUMAPHOS 66052 45050 MPHOSPH8 54737 NA PAROXETINE HYDROCHLORIDE PAROXETINE HYDROCHLORIDE 66053 45051 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 178102553 66054 45052 ATXN2 6311 NA GNF-PF-3716 CHEMBL609606 66055 45053 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE SP-600125 SP-600125 66056 45054 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR inhibitor 315661348 66059 45055 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL1213490 ROMIDEPSIN 66061 45056 BAZ2B 29994 NA NSC-3323 CHEMBL1270169 66062 45057 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE 3-aminopyridine-2-carboxaldehyde thiosemicarbazone 16493607 66063 45058 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL antagonist 135650806 66064 45059 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL1922094 APITOLISIB 66065 45060 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 3-MORPHOLINOSYDNONIMINE HCL CHEMBL538104 66066 45061 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565851 66067 45062 POU5F1 5460 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE ETHANOL ALCOHOL 16112835 66070 45063 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CHEMOTHERAPY 20619739,23828442 66073 45064 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor PF-03814735 PF-03814735 66074 45065 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolo[2,3-b]pyridine derivative 2 66076 45066 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1256 ISOFLURANE 66077 45067 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE PHENYTOIN PHENYTOIN 10563481 66078 45068 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL48361 DABIGATRAN 66080 45069 DOT1L 84444 CLINICALLY ACTIONABLE, DNA REPAIR, METHYL TRANSFERASE, DRUGGABLE GENOME, ENZYME inhibitor 178103599 66085 45070 ALDH1A1 216 DRUGGABLE GENOME, ENZYME RO-410960 CHEMBL1256291 66089 45071 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650619 66090 45072 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ERLOTINIB ERLOTINIB 19969465,24565969 66091 45073 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GMI-1070 RIVIPANSEL 66092 45074 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrrolo-pyridone derivative 2 66093 45075 GLS 2744 ENZYME PMID30273516-Compound-15 66094 45076 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor PWT33597 66097 45077 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Setipiprant SETIPIPRANT 66098 45078 CES1 1066 DRUGGABLE GENOME, ENZYME Cholic Acid 66100 45079 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Aminopyrimidine derivative 8 66101 45080 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR inhibitor CRIZOTINIB CRIZOTINIB 66102 45081 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR COMBRETASTATIN A4 COMBRETASTATIN A4 22982122 66103 45082 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-2B, RECOMBINANT 66105 45083 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Posaconazole POSACONAZOLE 26823493 66107 45084 PDE8B 8622 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200875 FLAVOXATE HYDROCHLORIDE 66110 45085 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TPCK TPCK 66112 45086 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor BOSUTINIB BOSUTINIB 66113 45087 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CINALUKAST CINALUKAST 66115 45088 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DNDI1318925 CHEMBL1390716 66118 45089 BAZ2B 29994 NA TCMDC-123762 CHEMBL547483 66119 45090 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OXYMETAZOLINE OXYMETAZOLINE 66120 45091 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Naphthyridine and isoquinoline derivative 1 66121 45092 IL23A 51561 DRUGGABLE GENOME CNT0-1959 66123 45093 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PMID29671355-Compound-45a 66124 45094 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NS-398 NS-398 66125 45095 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 8-CYCLOPENTYLTHEOPHYLLINE 8-CYCLOPENTYLTHEOPHYLLINE 66126 45096 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER MCP-1 9748276 66128 45097 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 3,5-DINITROCATECHOL (OR-486) 3,5-DINITROCATECHOL (OR-486) 66129 45098 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ALISOL A-23 ACETATE CHEMBL2059711 24915879 66130 45099 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-9037 CHEMBL1451216 66132 45100 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL3545252 DOCETAXEL 66133 45101 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C19 66136 45102 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE Cholic Acid 66137 45103 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GNF-PF-1878 CHEMBL1500740 66138 45104 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE AXL-1717 AXL-1717 66139 45105 TLR7 51284 DRUGGABLE GENOME DV-1179 66140 45106 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000201788 CHEMBL602923 66142 45107 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE CHLORHEXIDINE CHLORHEXIDINE 66143 45108 DUSP1 1843 PROTEIN PHOSPHATASE, KINASE, DRUGGABLE GENOME VASOPRESSIN VASOPRESSIN 9231829 66145 45109 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME Meso-CART 66147 45110 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1201082 FLUOXETINE HYDROCHLORIDE 66148 45111 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-WO2011127048 32 66149 45112 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Indoline derivative 6 66150 45113 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 381118854 66151 45114 SMN1 6606 DRUGGABLE GENOME GNF-PF-516 CHEMBL602970 66152 45115 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR TOZASERTIB TOZASERTIB 66153 45116 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME BEPRIDIL BEPRIDIL 66154 45117 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE MILATAXEL MILATAXEL 66155 45118 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ISOFENPHOS ISOFENPHOS 66156 45119 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Piperidinyl pyrazole derivative 1 66158 45120 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME carboplatin CARBOPLATIN 25055799 66160 45121 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE AMG0714 66161 45122 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE MT-103 BLINATUMOMAB 66162 45123 MAPT 4137 DRUGGABLE GENOME DNDI1417086 CHEMBL1224755 66164 45124 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENZOFURAN BENZOFURAN 66165 45125 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE CAR-T cells targeting CD117 66166 45126 IMPDH1 3614 ENZYME, DRUGGABLE GENOME inhibitor 178103451 THIOGUANINE 66167 45127 HTT 3064 DRUGGABLE GENOME DAUNORUBICIN DAUNORUBICIN 66168 45128 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX daunorubicin DAUNORUBICIN 66169 45129 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE NBQX NBQX 66170 45130 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PROCHLORPERAZINE PROCHLORPERAZINE 66171 45131 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR CURCUMIN CURCUMIN 15271854 66172 45132 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LGD-4033 VK5211 66173 45133 PDE4B 5142 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1370561 AMINOPHYLLINE 66175 45134 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL494089 GSK-690693 66177 45135 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 E-FLUPENTIXOL E-FLUPENTIXOL 66178 45136 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ANTIANGIOGENIC 11857382 66180 45137 ATXN2 6311 NA THIORIDAZINE THIORIDAZINE 66181 45138 E2F1 1869 TRANSCRIPTION FACTOR PRIMAQUINE PRIMAQUINE 15450938 66182 45139 DHCR24 1718 TUMOR SUPPRESSOR, ENZYME T-226293 66183 45140 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565688 CHEMBL1765740 66184 45141 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TRYPTAMINE TRYPTAMINE 66185 45142 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-348401 CHEMBL515505 66187 45143 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NICARDIPINE NICARDIPINE 66188 45144 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BITHIONOLATE SODIUM BITHIONOLATE SODIUM 66189 45145 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME JNJ-7706621 JNJ-7706621 66190 45146 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME ANTIANGIOGENIC 12954328 66193 45147 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 384403638 66196 45148 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor NINTEDANIB NINTEDANIB 66198 45149 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ARQ 761 66199 45150 TOP2B 7155 DRUGGABLE GENOME, ENZYME Dexrazoxane DEXRAZOXANE 66201 45151 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Irinotecan IRINOTECAN 25714871 66202 45152 IL18 3606 DRUGGABLE GENOME ribavirin RIBAVIRIN 19455410 66203 45153 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PIMOZIDE PIMOZIDE 66204 45154 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE ANETHOLTRITHION ANETHOLTRITHION 20655236 66205 45155 BUB1 699 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565791 66206 45156 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TD-5108 VELUSETRAG 66207 45157 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME NUTLIN-3 NUTLIN-3 21058726,21314128,24268795,19928922 66208 45158 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MONOCILLIN I MONOCILLIN I 16499313 66210 45159 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PQR309 BIMIRALISIB 66212 45160 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 249565926 66213 45161 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178101216 ISRADIPINE 66214 45162 TUBB2A 7280 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 66215 45163 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME TYrosine kinase 2 inhibitor 66217 45164 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DHT ANDROSTANOLONE 10698512 66218 45165 PDK3 5165 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 328083452 66219 45166 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SYROSINGOPINE SYROSINGOPINE 66220 45167 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE EGFR806-specific CAR T cell 66221 45168 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL CROMOGLICATE CROMOLYN 66223 45169 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Synthetic conjugated estrogen 66226 45170 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Alectinib ALECTINIB 28476735 66227 45171 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE TOMUDEX RALTITREXED 10047461 66229 45172 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Lapatinib LAPATINIB 27595477,26432108 66230 45173 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE CENISERTIB CENISERTIB 66231 45174 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor GSK2118436 DABRAFENIB 66232 45175 GPER1 2852 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR Segesterone acetate and ethinyl estradiol vaginal system 66234 45176 ATXN2 6311 NA TRIFLUOPERAZINE TRIFLUOPERAZINE 66235 45177 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE PAPAVERINE PAPAVERINE 16099300 66237 45178 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1356607 NOREPINEPHRINE BITARTRATE 66238 45179 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PAPAVERINE HYDROCHLORIDE PAPAVERINE HYDROCHLORIDE 66240 45180 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker CHEMBL585 TRIAMTERENE 66241 45181 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR CHIDAMIDE CHIDAMIDE 66242 45182 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE 2-CHLOROADENOSINE CHEMBL285819 66244 45183 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652430 66245 45184 ATAD5 79915 NA L-162313 CHEMBL288174 66246 45185 BAZ2B 29994 NA PHTHALYLSULFATHIAZOLE PHTHALYLSULFATHIAZOLE 66247 45186 POLI 11201 DNA REPAIR 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 66248 45187 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 178100438 CIPROFIBRATE 66249 45188 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE IMATINIB IMATINIB 66250 45189 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AMPHOTERICIN B AMPHOTERICIN B 66251 45190 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METITEPINE METITEPINE 18033297 66252 45191 EML4 27436 CLINICALLY ACTIONABLE, KINASE Entrectinib ENTRECTINIB 26939704 66254 45192 GAK 2580 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 178101952 66256 45193 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME NSC-71033 CHEMBL116548 66257 45194 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417599 CHEMBL2094833 66258 45195 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALL-TRANS-RETINOIC ACID 9417874 66259 45196 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3545385 WX-037 66261 45197 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CGS-15943 CGS-15943 66262 45198 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR DEMETHYLENCECALIN DEMETHYLENCECALIN 66263 45199 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-703 CHEMBL609030 66264 45200 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-26699 CHEMBL221721 66265 45201 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-108783 CHEMBL1489812 66268 45202 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652321 66270 45203 PDE8A 5151 DRUGGABLE GENOME, ENZYME inhibitor 348353618 66274 45204 POLK 51426 DNA REPAIR, ENZYME QUINACRINE DIHYDROCHLORIDE QUINACRINE DIHYDROCHLORIDE 66275 45205 ATXN2 6311 NA SJ000059269 CHEMBL590686 66276 45206 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL580 LORAZEPAM 66278 45207 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 310264688 EDAGLITAZONE 66279 45208 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME antibody RILOTUMUMAB RILOTUMUMAB 66280 45209 GAST 2520 DRUGGABLE GENOME, HORMONE ACTIVITY, ENZYME G17DT 66282 45210 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1201745 CHOLINE FENOFIBRATE 66283 45211 PSMA5 5686 PROTEASE, DRUGGABLE GENOME inhibitor BORTEZOMIB BORTEZOMIB 66285 45212 BAZ2B 29994 NA TCMDC-123764 CHEMBL533226 66286 45213 UGT2B7 7364 DRUGGABLE GENOME zidovudine ZIDOVUDINE 22960662 66287 45214 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL1200722 PIPECURONIUM BROMIDE 66288 45215 BAZ2B 29994 NA SJ000018298 CHEMBL591412 66293 45216 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TDR78109 CHEMBL1304363 66294 45217 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PYRONIN Y PYRONIN Y 66295 45218 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2109346 AME-133V 66296 45219 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor PAZOPANIB PAZOPANIB 66297 45220 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GR-103545 CHEMBL277863 66298 45221 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME PILOCARPINE PILOCARPINE 9661997 66299 45222 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME NIACINAMIDE NIACINAMIDE 25884115 66301 45223 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650930 ROXINDOLE 66302 45224 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Dabrafenib DABRAFENIB 27523909,22389471 66303 45225 GMNN 51053 DRUGGABLE GENOME RO-137410 CHEMBL275311 66304 45226 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 26619011,19331127,20542753,19381019,21273588,22869148,25157968 66305 45227 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BEZ235 DACTOLISIB 66306 45228 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-125180 CHEMBL586163 66307 45229 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME Imidazo[4,5-c]pyridine derivative 2 66308 45230 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR PACLITAXEL PACLITAXEL 16778834 66309 45231 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL522892 DOVITINIB 66311 45232 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX HISTONE DEACETYLASE INHIBITOR 12939274 66312 45233 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME TCMDC-123730 CHEMBL530280 66313 45234 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL1200761 CHLOROTRIANISENE 66314 45235 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME TAMATINIB R-406 66317 45236 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 310264761 CONESSINE 66319 45237 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 2-BENZOYL-5-METHOXYBENZOQUINONE 2-BENZOYL-5-METHOXYBENZOQUINONE 66320 45238 AKR1C3 8644 ENZYME, DRUGGABLE GENOME 3-((4-(TRIFLUOROMETHYL)PHENYL)AMINO)BENZOIC ACID CHEMBL1682202 22263837 66321 45239 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 328083522 66322 45240 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME SPLICEOSTATIN-A CHEMBL1221944 17643111 66325 45241 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ILORASERTIB ILORASERTIB 66326 45242 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Lycorine dimer salt derivative 1 66328 45243 KDM4A 9682 DRUGGABLE GENOME, ENZYME GLUTAMIC ACID HYDROCHLORIDE GLUTAMIC ACID HYDROCHLORIDE 66329 45244 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME BEVACIZUMAB BEVACIZUMAB 18182667 66330 45245 ATAD5 79915 NA CID 739615 CHEMBL260560 66332 45246 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 387065585 66334 45247 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE THIOMERSAL THIMEROSAL 66336 45248 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GALETERONE GALETERONE 23713567 66337 45249 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DICYCLOHEXYLCARBODIIMIDE DICYCLOHEXYLCARBODIIMIDE 66342 45250 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE SIMVASTATIN SIMVASTATIN 16321621 66346 45251 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ELEMICIN ELEMICIN 66347 45252 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DROMETRIZOLE DROMETRIZOLE 66349 45253 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE agonist 404859034 66351 45254 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IOBENGUANE IOBENGUANE 66352 45255 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 66353 45256 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL363648 TAK-715 66355 45257 POLK 51426 DNA REPAIR, ENZYME 7,8,2'-TRIHYDROXYFLAVONE CHEMBL244707 66356 45258 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 2-METHOXY-1,4-NAPHTHOQUINONE 2-METHOXY-1,4-NAPHTHOQUINONE 66357 45259 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3544999 SAMOTOLISIB 66358 45260 GM2A 2760 ENZYME BIW-8962 BIW-8962 66359 45261 FES 2242 ENZYME, DRUGGABLE GENOME, KINASE, TYROSINE KINASE SP-600125 SP-600125 66360 45262 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-3543 CHEMBL598679 66361 45263 MBNL1 4154 DRUGGABLE GENOME TCMDC-123591 CHEMBL588234 66363 45264 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3039565 66364 45265 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME 5,6,7-TRIBROMOISATIN CHEMBL376616 17088067 66365 45266 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE DIGOXIN DIGOXIN 66367 45267 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 381118865 66369 45268 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 178101309 REMOGLIFLOZIN 66370 45269 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME TRU-015 TRU-015 66371 45270 IFNG 3458 DRUGGABLE GENOME inhibitor CHEMBL2108459 FONTOLIZUMAB 66372 45271 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME nadolol NADOLOL 24419562 66373 45272 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 354702284 66374 45273 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor PF-4217903 PF-04217903 66375 45274 PSCA 8000 DRUGGABLE GENOME AGS-1C4D4 66376 45275 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME ZM-447439 CHEMBL202721 66378 45276 ERAP1 51752 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 348353642 66379 45277 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME inhibitor 374883876 66382 45278 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE DELAVIRDINE DELAVIRDINE 17172311 66384 45279 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME agonist 178101033 66386 45280 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE AMUVATINIB AMUVATINIB 66387 45281 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHA848125 66389 45282 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER FLUPHENAZINE FLUPHENAZINE 66393 45283 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME CILOSTAZOL CILOSTAZOL 11524048 66394 45284 LTC4S 4056 ENZYME, DRUGGABLE GENOME US20160326143, 38 66395 45285 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SJ000019194 CHEMBL592106 66396 45286 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME XCT790 CHEMBL189753 66398 45287 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FG-4592 ROXADUSTAT 66399 45288 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE SOTRASTAURIN SOTRASTAURIN 66404 45289 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR CH-5132799 PA-799 66405 45290 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 arteether 66410 45291 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE NDGA 10203695 66411 45292 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TRICITRINOL B TRICITRINOL B 21761866 66412 45293 DLL3 10683 NA ROVALPITUZUMAB TESIRINE 27932068 66413 45294 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Icotinib ICOTINIB 24533047,27468240,23372346,2394835,25261231,24438614 66414 45295 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL235191 TACEDINALINE 66416 45296 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 178100305 66417 45297 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 354702236 66419 45298 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 381744923 66420 45299 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER unspecified EGFR antibody 27196767 66421 45300 GSTM1 2944 DRUGGABLE GENOME, ENZYME vinblastine VINBLASTINE 23323945 66422 45301 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 3,4-methylenedioxymethamphetamine 66423 45302 TARDBP 23435 TUMOR SUPPRESSOR FLUORANTHEN-3-YLAMINE CHEMBL103583 66424 45303 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PSAMMAPLIN A PSAMMAPLIN A 22280363,21215647,25884112 66426 45304 IFNG 3458 DRUGGABLE GENOME TRASTUZUMAB TRASTUZUMAB 15297404 66427 45305 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ELLIPTECINE ELLIPTECINE 66428 45306 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR RITUXIMAB RITUXIMAB 11895917 66430 45307 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL agonist 178103535 DEXTROMETHORPHAN 66431 45308 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER SULFINPYRAZONE SULFINPYRAZONE 66433 45309 CBX1 10951 NA AG-537 CHEMBL67535 66434 45310 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR Bevacizumab BEVACIZUMAB 16827904,22931246 66435 45311 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 363894201 TENALISIB 66436 45312 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHOSALONE PHOSALONE 66440 45313 ALOX15 246 ENZYME, DRUGGABLE GENOME NSC-37031 CHEMBL222993 66443 45314 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR exemestane EXEMESTANE 66444 45315 ARF6 382 NA INSULIN INSULIN 11438681 66446 45316 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Autologous Anti-CD 123 CAR TCR/4-1BB-expressing T-lymphocytes 66448 45317 CCN1 3491 DRUGGABLE GENOME INTERLEUKIN-8 18025257 66449 45318 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1200805 DILTIAZEM MALATE 66450 45319 CACNB3 784 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ION CHANNEL SAFINAMIDE SAFINAMIDE 66451 45320 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CANERTINIB CANERTINIB 18408761 66452 45321 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE TNF alpha kinoid 22441388 66453 45322 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE antibody LEXATUMUMAB LEXATUMUMAB 66454 45323 TPBG 7162 CELL SURFACE, DRUGGABLE GENOME TroVax TROVAX 66455 45324 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME LUTEOLIN LUTEOLIN 66456 45325 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE Vorinostat VORINOSTAT 26634271 66459 45326 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL679 EPINEPHRINE 66463 45327 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 178103904 BARASERTIB 66465 45328 ST14 6768 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 252166825 66467 45329 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR GLUTAMINE GLUTAMINE 10377266 66470 45330 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME 5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivative 1 66471 45331 MAOB 4129 DRUGGABLE GENOME, ENZYME Neu-120 66472 45332 TOP2B 7155 DRUGGABLE GENOME, ENZYME Etoposide ETOPOSIDE 66473 45333 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GEOPYXIN A GEOPYXIN A 66474 45334 HTT 3064 DRUGGABLE GENOME MERCURIC CHLORIDE MERCURIC CHLORIDE 66476 45335 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1200947 METIPRANOLOL HYDROCHLORIDE 66477 45336 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PALBOCICLIB PALBOCICLIB 66478 45337 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ARACHIDONIC ACID ARACHIDONIC ACID 66479 45338 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORHEXIDINE CHLORHEXIDINE 66481 45339 MDM4 4194 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, DRUGGABLE GENOME PEMBROLIZUMAB PEMBROLIZUMAB 28351930 66482 45340 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE 404859001 BAMOCAFTOR 66483 45341 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PERTUZUMAB PERTUZUMAB 66484 45342 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME RHGH 10485595 66487 45343 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3353410 OSIMERTINIB 66489 45344 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GO-6976 GO-6976 66490 45345 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 252166899 VERUBECESTAT 66492 45346 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW780159X GW780159X 66493 45347 PTGS2 5743 DRUGGABLE GENOME, ENZYME CSA CYCLOSPORINE 10999939 66494 45348 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW861893X GW861893X 66495 45349 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GNF-PF-1969 CHEMBL601364 66496 45350 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME EGCG EPIGALOCATECHIN GALLATE 16449979 66498 45351 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME LEUCOVORIN LEUCOVORIN 21879757 66500 45352 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RGB-286638 RGB-286638 66502 45353 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW829906X GW829906X 66503 45354 MAPT 4137 DRUGGABLE GENOME ACITRETIN ACITRETIN 66504 45355 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING GIVINOSTAT GIVINOSTAT 66505 45356 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR SELECTIVE ESTROGEN RECEPTOR MODULATORS 15762036 66506 45357 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR NSC-45174 CHEMBL221047 17432842 66508 45358 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651082 66509 45359 LGALS2 3957 NA MITOMYCIN C 17999373 66515 45360 TUBA1B 10376 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 66516 45361 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-18 66517 45362 TOP2B 7155 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2103796 BERUBICIN HYDROCHLORIDE 66520 45363 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000001592 CHEMBL591834 66522 45364 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SB-220025 SB-220025 66523 45365 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-107022 CHEMBL1601846 66525 45366 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545177 AZD-0424 66526 45367 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 66527 45368 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DEXPROPRANOLOL HYDROCHLORIDE DEXPROPRANOLOL HYDROCHLORIDE 66530 45369 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649996 66531 45370 BAZ2B 29994 NA BIFONAZOLE BIFONAZOLE 66532 45371 IL11 3589 DRUGGABLE GENOME, KINASE, GROWTH FACTOR citalopram CITALOPRAM 25916525 66535 45372 CAMK1D 57118 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME RG-1530 RG-1530 66537 45373 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL211471 NEOSTIGMINE METHYLSULFATE 66538 45374 GAPDH 2597 DRUGGABLE GENOME, ENZYME SELENIUM 15653770 66542 45375 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME fluorouracil / salicylic acid 66543 45376 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 178103975 RALTITREXED 66544 45377 GP6 51206 CELL SURFACE, KINASE Revacept 66545 45378 UGT2B15 7366 DRUGGABLE GENOME oxazepam OXAZEPAM 15044558,29737521 66547 45379 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME meclizine MECLIZINE 66548 45380 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 404859105 66550 45381 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 249565638 ALPELISIB 66551 45382 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME GNF-PF-1702 CHEMBL600313 66552 45383 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL603469 LESTAURTINIB 66553 45384 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1200812 METAPROTERENOL SULFATE 66554 45385 TAC1 6863 DRUGGABLE GENOME LORATADINE LORATADINE 1283698,9055977 66555 45386 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE TEMSIROLIMUS TEMSIROLIMUS 19706758 66556 45387 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL1743076 TADOCIZUMAB 66557 45388 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE NSC-749235 CHEMBL2336666 23279865 66559 45389 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME NG2-73 ADIPIPLON 66561 45390 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE amlodipine / atorvastatin / perindopril arginine 66562 45391 ABL2 27 KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME IMATINIB IMATINIB 25207766 66563 45392 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Nivolumab NIVOLUMAB 66564 45393 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME timolol TIMOLOL 7474246,16315032 66565 45394 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MLN1117 SERABELISIB 66566 45395 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270010-Compound-Figure16-b-1 66567 45396 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL49642 INDIBULIN 66568 45397 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33d 66569 45398 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE LINOLENIC ACID LINOLENIC ACID 66570 45399 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE TAE-684 TAE-684 66571 45400 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000170251 CHEMBL603154 66572 45401 ITPR2 3709 ION CHANNEL, DRUGGABLE GENOME activator 135652731 66573 45402 IGFBP1 3484 DRUGGABLE GENOME HORMONES 8619542,8567796 66574 45403 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE erlotinib ERLOTINIB 66575 45404 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (S)-ALAPROCLATE (S)-ALAPROCLATE 66577 45405 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DULOXETINE HYDROCHLORIDE DULOXETINE HYDROCHLORIDE 66578 45406 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE UK-356202 66579 45407 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE TANSHINONE IIA SULFONATE TANSHINONE IIA SULFONATE 66580 45408 IFNG 3458 DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 24776844 66581 45409 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ALITRETINOIN ALITRETINOIN 66582 45410 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL2109047 INTERFERON ALFA-N3 66583 45411 PRKG1 5592 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME LINIFANIB LINIFANIB 66585 45412 FAAH 2166 ENZYME, DRUGGABLE GENOME haloperidol HALOPERIDOL 20631561 66587 45413 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE PD-0166285 PD-0166285 66589 45414 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR docetaxel DOCETAXEL 20038957 66591 45415 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-123764 CHEMBL533226 66592 45416 CFH 3075 DRUGGABLE GENOME ranibizumab RANIBIZUMAB 26439641,23584701,23204795,22840423,22594510,23559864,24070809,26411831,23842101,23337555 66594 45417 PTGES 9536 DRUGGABLE GENOME, ENZYME Benzimidazole derivative 14 66595 45418 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METYRAPONE METYRAPONE 66596 45419 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME URAPIDIL URAPIDIL 66599 45420 TNK1 8711 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 249565737 66601 45421 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME PROTOAPIGENONE PROTOAPIGENONE 66603 45422 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR MUNDULONE ACETATE MUNDULONE ACETATE 66604 45423 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME 1,2-BENZANTHRACENE CHEMBL1873684 66606 45424 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PF-05212384 GEDATOLISIB 24042735,25977343,24823695,17314276,21325073 66609 45425 ALDH1A1 216 DRUGGABLE GENOME, ENZYME MMV085203 CHEMBL586031 66610 45426 CTSV 1515 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 363894149 PETESICATIB 66611 45427 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME S63845 27760111 66612 45428 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PARATHION PARATHION 66613 45429 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-145669 CHEMBL191611 66615 45430 DHFR 1719 DRUGGABLE GENOME, ENZYME VITAMIN B12 3719892 66616 45431 GMNN 51053 DRUGGABLE GENOME ETRETINATE ETRETINATE 66617 45432 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LETROZOLE LETROZOLE 66618 45433 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 363894211 PEXMETINIB 66619 45434 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME fluorouracil FLUOROURACIL 24090479,20125120,25955730 66621 45435 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TRIFLUPERIDOL TRIFLUPERIDOL 66622 45436 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100326 66625 45437 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649687 66626 45438 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DACTOLISIB DACTOLISIB 66627 45439 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-WO2013082253 34 66630 45440 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRIBROMSALAN TRIBROMSALAN 66634 45441 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME CYC-116 CYC-116 66635 45442 PDE10A 10846 ENZYME, DRUGGABLE GENOME Triazolo-pyridine derivative 2 66636 45443 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL ISRADIPINE ISRADIPINE 66638 45444 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 328083481 66639 45445 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor SNS-314 SNS-314 66644 45446 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DNDI1416988 CHEMBL1389794 66647 45447 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL OXAZEPAM OXAZEPAM 66650 45448 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178101947 RUBOXISTAURIN 66651 45449 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER TCMDC-125319 CHEMBL527586 66652 45450 TNFRSF11A 8792 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE acetaminophen ACETAMINOPHEN 26398624 66653 45451 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 178100452 66654 45452 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200870 TIMOLOL MALEATE 66656 45453 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NEBIVOLOL NEBIVOLOL 66658 45454 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR MPA PROGESTERONE 9822358 66660 45455 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE INDOTECAN INDOTECAN 20630766 66661 45456 LPAR5 57121 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100542 ARACHIDONOYL GLYCINE 66662 45457 RGS4 5999 DRUGGABLE GENOME NSC-139257 CHEMBL1256364 66665 45458 CAST 831 PROTEASE INHIBITOR DOX 12650523 66666 45459 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID25991433-Compound-A1 66667 45460 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor ERLOTINIB ERLOTINIB 66668 45461 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 374883884 66669 45462 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER LONAFARNIB LONAFARNIB 14671431 66670 45463 MAOA 4128 DRUGGABLE GENOME, ENZYME GypensapogeninA 66671 45464 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NCI-13239 CHEMBL187216 66672 45465 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 2 66673 45466 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody MM-121 MM-121 66675 45467 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME G207 16391370 66676 45468 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PROGESTERONE PROGESTERONE 22931300 66677 45469 ARSA 410 DRUGGABLE GENOME, ENZYME PHLORETIN PHLORETIN 66678 45470 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-3515 CHEMBL602365 66679 45471 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-141 66680 45472 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CTAP-201 19302594 66681 45473 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHENOLPHTHALEIN PHENOLPHTHALEIN 66682 45474 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIBUCAINE HYDROCHLORIDE DIBUCAINE HYDROCHLORIDE 66684 45475 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565863 66685 45476 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor SARACATINIB SARACATINIB 66687 45477 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR ETOPOSIDE ETOPOSIDE 16002781 66688 45478 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME TAK-442 LETAXABAN 66689 45479 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-125066 CHEMBL533577 66691 45480 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME GLUCAGON GLUCAGON 3130065 66692 45481 ALDH3A1 218 DRUGGABLE GENOME, ENZYME doxorubicin DOXORUBICIN 66693 45482 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ONONETIN ONONETIN 66695 45483 GMNN 51053 DRUGGABLE GENOME TAMOXIFEN CITRATE TAMOXIFEN CITRATE 66697 45484 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200425 PARGYLINE HYDROCHLORIDE 66698 45485 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE antibody LEXATUMUMAB LEXATUMUMAB 66699 45486 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE WYE-125132 20068177 66700 45487 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME THROMBIN THROMBIN 7007650 66701 45488 SIK1 150094 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 340590212 66703 45489 HDAC11 79885 DRUGGABLE GENOME, ENZYME PSAMMAPLIN A PSAMMAPLIN A 25884112 66705 45490 SOS1 6654 KINASE IL-6 9815779 66706 45491 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100613 66707 45492 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME ALTISSIMACOUMARIN F ALTISSIMACOUMARIN F 22799262 66708 45493 TNNI3 7137 DRUGGABLE GENOME NSC-107022 CHEMBL1601846 66709 45494 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL agonist 178100908 66710 45495 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL METHARBITAL METHARBITAL 66711 45496 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Palbociclib PALBOCICLIB 27020857,19874578,25221644 66713 45497 TUBA1B 10376 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 66714 45498 GUCY2C 2984 DRUGGABLE GENOME, KINASE agonist CHEMBL2103867 PLECANATIDE 66716 45499 PDE7A 5150 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL932 DIPYRIDAMOLE 66717 45500 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE TNO155 66718 45501 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650117 CODEINE 66721 45502 RPS6KA5 9252 DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE ILORASERTIB ILORASERTIB 66724 45503 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DNDI1417467 CHEMBL1997335 66726 45504 APC 324 CLINICALLY ACTIONABLE Sirolimus SIROLIMUS 18768809,20080688 66728 45505 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor AZD4547 66729 45506 CPS1 1373 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Carglumic acid 66730 45507 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor XL147 PILARALISIB 66733 45508 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CEVIMELINE CEVIMELINE 66735 45509 KMO 8564 DRUGGABLE GENOME, ENZYME Aryl pyrimidine derivative 7 66736 45510 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME PMID27828716-Compound-16 66737 45511 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE stavudine STAVUDINE 20887379 66738 45512 POLK 51426 DNA REPAIR, ENZYME TCMDC-124266 CHEMBL124006 66739 45513 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL3545348 BKT140 66740 45514 CA1 759 DRUGGABLE GENOME, ENZYME METHAZOLAMIDE METHAZOLAMIDE 66741 45515 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-37 66743 45516 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32v 66744 45517 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AG-126 CHEMBL77387 66746 45518 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 348353671 66749 45519 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-1692 CHEMBL582055 66750 45520 GMNN 51053 DRUGGABLE GENOME TCMDC-124409 CHEMBL587801 66754 45521 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME activator 135652750 66755 45522 SLC15A4 121260 DRUGGABLE GENOME, TRANSPORTER 178101341 66756 45523 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CART-123 cells 66759 45524 SMPD1 6609 ENZYME, DRUGGABLE GENOME inhibitor 404859086 66760 45525 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL ADINAZOLAM ADINAZOLAM 66763 45526 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME H2O2 9624736 66764 45527 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE 178101633 66765 45528 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME NEVIRAPINE NEVIRAPINE 17041008 66766 45529 CX3CL1 6376 CELL SURFACE, DRUGGABLE GENOME COMPLETE FREUND'S ADJUVANT 15993821 66767 45530 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Aminopiperidine derivative 2 66768 45531 CLK1 1195 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor 249565841 66775 45532 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE OSI-632 OSI-632 66776 45533 GMNN 51053 DRUGGABLE GENOME SCOPOLETIN SCOPOLETIN 66777 45534 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR TYROSINE HYDROXYLASE INHIBITOR 11571589 66778 45535 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE EVEROLIMUS EVEROLIMUS 23989949,23582881,27091708 66779 45536 BAZ2B 29994 NA DNDI1416955 CHEMBL1327172 66780 45537 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL blocker 178100875 PICROTOXIN 66781 45538 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NILVADIPINE NILVADIPINE 66782 45539 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyrimidine derivative 9 66785 45540 BRD9 65980 ENZYME inhibitor 252827481 66787 45541 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 66790 45542 POLK 51426 DNA REPAIR, ENZYME GNF-PF-1947 CHEMBL585591 66792 45543 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SP-600125 SP-600125 66793 45544 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ASCJ-9 topical 66794 45545 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor MLN8237 ALISERTIB 66796 45546 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE PMA 15383372 66797 45547 COL18A1 80781 DRUGGABLE GENOME RetinoStat 66798 45548 KLKB1 3818 DRUGGABLE GENOME, PROTEASE, ENZYME Lanadelumab LANADELUMAB 66801 45549 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE celecoxib CELECOXIB 22336956 66802 45550 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CAPTOPRIL CAPTOPRIL 66803 45551 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE cyclosporine CYCLOSPORINE 18444945 66805 45552 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-270156 CHEMBL471226 66806 45553 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ART621 PLACULUMAB 66807 45554 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 223366135 66808 45555 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE OXALIPLATIN OXALIPLATIN 14977850 66811 45556 NQO2 4835 DRUGGABLE GENOME, ENZYME CARICOTAMIDE CARICOTAMIDE 66812 45557 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Linsitinib LINSITINIB 26725216 66813 45558 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL3545243 AS-703988 66814 45559 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649839 66824 45560 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME TG101348 FEDRATINIB 66825 45561 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL1200395 ORPHENADRINE CITRATE 66826 45562 STK38L 23012 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 66827 45563 NOS2 4843 DRUGGABLE GENOME, ENZYME Aminoguanidine PIMAGEDINE 66828 45564 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL2364649 MARGETUXIMAB 66831 45565 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100470 66832 45566 ACVR1B 91 SERINE THREONINE KINASE, CELL SURFACE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 249565800 66833 45567 SMN2 6607 DRUGGABLE GENOME AG-1296 CHEMBL71191 66834 45568 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650975 SABCOMELINE 66836 45569 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME VAPREOTIDE VAPREOTIDE 66840 45570 METAP2 10988 ENZYME, DRUGGABLE GENOME, KINASE, PROTEASE inhibitor 252166655 BELORANIB 66841 45571 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 8 66842 45572 TUBA4A 7277 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 66843 45573 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME antibody 310264725 EMACTUZUMAB 66845 45574 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000029642 CHEMBL591126 66846 45575 PDE4A 5141 DRUGGABLE GENOME, ENZYME DIPYRIDAMOLE DIPYRIDAMOLE 66848 45576 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Prasterone PRASTERONE 66850 45577 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DAPHNORIN DAPHNORIN 66851 45578 PDGFA 5154 GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE Squalamine SQUALAMINE 66853 45579 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL408513 BELINOSTAT 66854 45580 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-2 66857 45581 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME TETRAIDOFLUORESCEIN TETRAIDOFLUORESCEIN 66858 45582 MAPT 4137 DRUGGABLE GENOME GNF-PF-1134 CHEMBL600694 66860 45583 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-372 CHEMBL580155 66861 45584 KLK4 9622 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 404859023 66862 45585 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE allosteric modulator 135650439 IVERMECTIN 66863 45586 FAAH 2166 ENZYME, DRUGGABLE GENOME IW-6118 21764305 66865 45587 DHODH 1723 DRUGGABLE GENOME, ENZYME inhibitor 178103450 TERIFLUNOMIDE 66867 45588 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL101 PHENYLBUTAZONE 66868 45589 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GNF-PF-2301 CHEMBL578061 66869 45590 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSAIDS 9574817 66870 45591 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist 381118908 66873 45592 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME IL-12 15905580 66874 45593 ALOX15B 247 DRUGGABLE GENOME, ENZYME 2-AMINOETHOXYDIPHENYL BORATE CHEMBL169233 66876 45594 CXCL2 2920 DRUGGABLE GENOME DEXTRAN SULFATE SODIUM 18542050 66877 45595 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR MMF MYCOPHENOLATE MOFETIL 16029632,12974756 66878 45596 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 EHNA EHNA 66879 45597 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL3545368 PANOBINOSTAT LACTATE 66881 45598 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 66883 45599 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CHEMOTHERAPEUTIC AGENT 12546364 66884 45600 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor PIVANEX AN-9 66885 45601 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME BORTEZOMIB BORTEZOMIB 66886 45602 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650158 DAMGO 66887 45603 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL3545252 DOCETAXEL 66889 45604 NOX1 27035 ION CHANNEL, ENZYME, TRANSPORTER, DRUGGABLE GENOME inhibitor 363894226 66890 45605 PDE4B 5142 DRUGGABLE GENOME, ENZYME GSK-356278 GSK-356278 66893 45606 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 6 66894 45607 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR HYDROXYTAMOXIFEN 66895 45608 CPT1A 1374 DRUGGABLE GENOME, ENZYME PERHEXILINE PERHEXILINE 66896 45609 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417181 CHEMBL1537417 66897 45610 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Eribulin ERIBULIN 66899 45611 KIF11 3832 DRUGGABLE GENOME ARQ 621 66900 45612 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL1417019 MITOXANTRONE HYDROCHLORIDE 66902 45613 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650629 66905 45614 FLNA 2316 DRUGGABLE GENOME, TRANSPORTER PTI-125 66907 45615 CA1 759 DRUGGABLE GENOME, ENZYME ACETAZOLAMIDE ACETAZOLAMIDE 66909 45616 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor RUCAPARIB RUCAPARIB 66910 45617 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME DABIGATRAN DABIGATRAN 66911 45618 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TEGASEROD MALEATE TEGASEROD MALEATE 66912 45619 HMGCR 3156 ENZYME, DRUGGABLE GENOME Pravastatin derivative 1 66913 45620 POLK 51426 DNA REPAIR, ENZYME ETHACRIDINE LACTATE ETHACRIDINE LACTATE 66914 45621 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL2017974 BUPARLISIB 66915 45622 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE IBRUTINIB IBRUTINIB 28830912 66916 45623 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SYM004 26888827,25962717,24130052,24204198 66918 45624 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DESONIDE DESONIDE 66919 45625 IL11 3589 DRUGGABLE GENOME, KINASE, GROWTH FACTOR VM-501 66920 45626 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME GO-203-2C GO-203-2C 66921 45627 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER capecitabine CAPECITABINE 21142915,22026922 66922 45628 CTSH 1512 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 336446936 66925 45629 GLS 2744 ENZYME BAS 01152706 CHEMBL2002487 66929 45630 GPR37 2861 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist 135652325 66932 45631 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME Sirolimus SIROLIMUS 66934 45632 FANCC 2176 CLINICALLY ACTIONABLE, DNA REPAIR GEMCITABINE GEMCITABINE 16243825 66935 45633 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650382 66937 45634 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL282686 TESAGLITAZAR 66939 45635 SI 6476 DRUGGABLE GENOME, ENZYME STZ STREPTOZOCIN 12940455 66940 45636 MARK4 57787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TOZASERTIB TOZASERTIB 66941 45637 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Indole-based analog 13 66942 45638 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SB-204741 CHEMBL323356 66944 45639 SDS 10993 ENZYME DEXAMETHASONE DEXAMETHASONE 12210718 66946 45640 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme16DMAT 66949 45641 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor 178101417 66950 45642 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY RHIGF-1 8423214 66954 45643 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BIFENAZATE BIFENAZATE 66956 45644 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650367 66958 45645 KCNJ3 3760 EXTERNAL SIDE OF PLASMA MEMBRANE, ION CHANNEL, DRUGGABLE GENOME FLUPIRTINE FLUPIRTINE 66959 45646 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR NORGESTIMATE NORGESTIMATE 66961 45647 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE ARQ 751 26469692 66963 45648 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE (-)-DEMECOLCINE DEMECOLCINE 66964 45649 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME (RS)-ROSCOVITINE (RS)-ROSCOVITINE 66965 45650 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor HESPERADIN HESPERADIN 19035792 66967 45651 TRAP1 10131 DRUGGABLE GENOME inhibitor 315661336 LUMINESPIB 66968 45652 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE DOVITINIB DOVITINIB 66969 45653 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Triptolide TRIPTOLIDE 66970 45654 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME BETAMETHASONE BETAMETHASONE 10495414 66971 45655 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2219422 AFURESERTIB 66972 45656 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME FLURAZEPAM FLURAZEPAM 66973 45657 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BAY1125976 27699769 66976 45658 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ANISINDIONE ANISINDIONE 66977 45659 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RILMENIDINE RILMENIDINE 66979 45660 HTT 3064 DRUGGABLE GENOME GNF-PF-1644 CHEMBL600734 66980 45661 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DOVITINIB DOVITINIB 66981 45662 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-37 66982 45663 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure1-Neonectrolide A 66983 45664 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 348353619 66988 45665 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE FR901228 ROMIDEPSIN 11929951 66989 45666 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR KB3305 66990 45667 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 7-NITROINDAZOLE 7-NITROINDAZOLE 66992 45668 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE MSC2363318A MSC-2363318A 66995 45669 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CLOZAPINE CLOZAPINE 66998 45670 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103655 FLUNISOLIDE 66999 45671 PSMC1 5700 PROTEASE CARFILZOMIB CARFILZOMIB 24524217 67000 45672 LPAR5 57121 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651487 67002 45673 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL403989 TG100-801 67003 45674 GPR87 53836 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650190 67007 45675 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE methacholine METHACHOLINE 23384627 67008 45676 EPHB4 2050 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor XL647 TESEVATINIB 67009 45677 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 9382956 67010 45678 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 404859073 67011 45679 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor SOPHORETIN QUERCETIN 67012 45680 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE LEUCETTAMINE B LEUCETTAMINE B 22998443 67014 45681 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PROGESTERONE PROGESTERONE 22931300 67015 45682 IFNG 3458 DRUGGABLE GENOME INTERFERON ALPHA-2B 10540707,9192993 67016 45683 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CP-339818 CP-339818 67017 45684 MPHOSPH8 54737 NA AG-527 CHEMBL258767 67018 45685 CYB5R3 1727 DRUGGABLE GENOME, ENZYME ropivacaine ROPIVACAINE 67019 45686 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 249565656 67020 45687 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE BLU-285 AVAPRITINIB 67021 45688 TUBA1C 84790 DRUGGABLE GENOME inhibitor CHEMBL2103852 CROLIBULIN 67023 45689 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649790 67027 45690 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE RESVERATROL RESVERATROL 18065527 67028 45691 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME N/A 67030 45692 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 381118805 67031 45693 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SB-242084 SB-242084 67032 45694 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL1096380 PLINABULIN 67033 45695 RAB9A 9367 ENZYME, DRUGGABLE GENOME PIPERINE PIPERINE 67034 45696 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL2035874 EPROTIROME 67035 45697 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL PRAZEPAM PRAZEPAM 67036 45698 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DANAZOL DANAZOL 67037 45699 NOS2 4843 DRUGGABLE GENOME, ENZYME CR-3294 20041326 67042 45700 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY JNJ-64565111 EFINOPEGDUTIDE 67043 45701 BAZ2B 29994 NA GNF-PF-5061 CHEMBL601385 67044 45702 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 178103585 ROMIDEPSIN 67045 45703 MAOB 4129 DRUGGABLE GENOME, ENZYME ANTIDEPRESSANT 6430257 67046 45704 CBX1 10951 NA GNF-PF-1919 CHEMBL576409 67047 45705 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ANTI-VEGF 12554695 67048 45706 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CYSTEINE METHYL-ESTER HCL CHEMBL1426508 67050 45707 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SOFALCONE SOFALCONE 67051 45708 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME HYDROQUINONE HYDROQUINONE 15141365 67054 45709 SIAH1 6477 ENZYME, KINASE OMIGAPIL OMIGAPIL 67057 45710 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL690 PRAVASTATIN SODIUM 67059 45711 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR OXYPHENBUTAZONE OXYPHENBUTAZONE 67060 45712 MGLL 11343 DRUGGABLE GENOME, ENZYME Azetidine-benzoxazin-3(4H)-one derivative 3 67061 45713 VEGFC 7424 GROWTH FACTOR, TRANSPORTER, DRUGGABLE GENOME inhibitor CHEMBL2108313 CONBERCEPT 67062 45714 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE VX-702 VX-702 67063 45715 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR MEGESTROL MEGESTROL 67065 45716 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR VACCINE 16563560 67066 45717 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE PMID27410995-Compound-Figure3k 67068 45718 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME (-)-DICENTRINE CHEMBL478754 67069 45719 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHLORHEXIDINE CHLORHEXIDINE 67070 45720 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Certolizumab CERTOLIZUMAB 67071 45721 ATXN2 6311 NA SERTACONAZOLE NITRATE SERTACONAZOLE NITRATE 67072 45722 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 363894224 HENATINIB 67073 45723 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHENYTOIN PHENYTOIN 22931300 67074 45724 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TCMDC-124224 CHEMBL580421 67077 45725 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE VINORELBINE VINORELBINE 14559807 67078 45726 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 67082 45727 CARM1 10498 ENZYME, METHYL TRANSFERASE, DRUGGABLE GENOME inhibitor 178103609 67083 45728 CA1 759 DRUGGABLE GENOME, ENZYME PHENOL PHENOL 26073005 67084 45729 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ROSMARINIC ACID ROSMARINIC ACID 67085 45730 SCNN1A 6337 DRUGGABLE GENOME, ION CHANNEL TRIAMTERENE TRIAMTERENE 67086 45731 SLC44A4 80736 TRANSPORTER, DRUGGABLE GENOME ASG-5ME ASG-5ME 67087 45732 GAPDH 2597 DRUGGABLE GENOME, ENZYME GNF-PF-2272 CHEMBL601757 67088 45733 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 348353660 67089 45734 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME oxazine 89 67092 45735 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GENISTEIN GENISTEIN 67095 45736 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ERGOCALCIFEROL ERGOCALCIFEROL 67097 45737 KCNG1 3755 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL284348 DALFAMPRIDINE 67098 45738 VKORC1 79001 DRUGGABLE GENOME, ENZYME ACENOCOUMAROL ACENOCOUMAROL 67099 45739 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE Ertumaxomab ERTUMAXOMAB 67100 45740 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ALEGLITAZAR ALEGLITAZAR 67101 45741 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ERUCIC ACID ERUCIC ACID 67102 45742 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE Amediplase AMEDIPLASE 67103 45743 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ROSIGLITAZONE ROSIGLITAZONE 18302760 67104 45744 EIF2AK2 5610 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 178102610 67107 45745 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AMENTOFLAVONE AMENTOFLAVONE 67108 45746 POLI 11201 DNA REPAIR PORFIROMYCIN PORFIROMYCIN 67109 45747 RAC1 5879 CLINICALLY ACTIONABLE, KINASE, DRUG RESISTANCE NSC-23766 CHEMBL257119 19527032 67110 45748 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL598797 CUDC-101 67111 45749 PRKCH 5583 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 249565822 BALANOL 67112 45750 CDA 978 ENZYME, DRUGGABLE GENOME azacitidine AZACITIDINE 25850965 67115 45751 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650726 67116 45752 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TETRACYCLINE TETRACYCLINE 22931300 67117 45753 TSPO 706 DRUGGABLE GENOME Halazepam HALAZEPAM 67118 45754 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME TCMDC-125764 CHEMBL586670 67119 45755 ATAD5 79915 NA SJ000024939 CHEMBL590691 67121 45756 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME BK7 67124 45757 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2108167 VEPALIMOMAB 67125 45758 UGT2B7 7364 DRUGGABLE GENOME ibuprofen IBUPROFEN 25502615 67126 45759 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AT13148 AT-13148 67128 45760 GUCY1A1 2982 ENZYME, DRUGGABLE GENOME activator CHEMBL1200689 NITRIC OXIDE 67129 45761 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE 7,12-DIMETHYL-BENZO[A]ANTHRACENE CHEMBL329673 67130 45762 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102637 67131 45763 DHPS 1725 NA DEOXYSPERGUALIN 11964177 67132 45764 PCSK6 5046 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE inhibitor 252166868 67134 45765 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE fentanyl FENTANYL 22277678,30281924,24365989,27236640,18695978 67135 45766 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1445 FLUOXYMESTERONE 67136 45767 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR SBI-0640756 26603897 67137 45768 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103884 OPROZOMIB 67138 45769 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TW-37 CHEMBL217354 25665005 67139 45770 PROS1 5627 DRUGGABLE GENOME Estradiol ESTRADIOL 67141 45771 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Tetrazole derivative 1 67144 45772 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GNF-PF-4463 CHEMBL584520 67146 45773 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME AZ-4217 67147 45774 SLC40A1 30061 TRANSPORTER, DRUGGABLE GENOME LY2928057 22290531 67148 45775 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME INDAPAMIDE INDAPAMIDE 67149 45776 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ISOCONAZOLE ISOCONAZOLE 67151 45777 NUDT7 283927 ENZYME inhibitor 384403663 67152 45778 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE sirolimus SIROLIMUS 16815317,17941052,26543771,28245187,22094953,26256674,15707415,23974086 67153 45779 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENODANIL BENODANIL 67154 45780 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651573 LIOTHYRONINE SODIUM 67155 45781 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME GNF-PF-159 CHEMBL599924 67156 45782 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRIBUTYLTIN-OXIDE TRIBUTYLTIN-OXIDE 67157 45783 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL1095032 LETAXABAN 67158 45784 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DASATINIB DASATINIB 67159 45785 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor PONATINIB PONATINIB 67161 45786 NPC1L1 29881 DRUGGABLE GENOME, TRANSPORTER EZETIMIBE EZETIMIBE 67162 45787 MAPT 4137 DRUGGABLE GENOME PHENANTHROLINE PHENANTHROLINE 67163 45788 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME LOVASTATIN LOVASTATIN 10543307 67164 45789 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME REV-576 NOMACOPAN 67165 45790 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME SIBUTRAMINE SIBUTRAMINE 67166 45791 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR N-METHYLDOPAMINE HCL CHEMBL1256484 67167 45792 MAPT 4137 DRUGGABLE GENOME EPINEPHRINE BITARTRATE EPINEPHRINE BITARTRATE 67169 45793 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CEVIMELINE CEVIMELINE 67172 45794 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL29919 ELPETRIGINE 67174 45795 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME ICO-25 67175 45796 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GARCINOLIC ACID GARCINOLIC ACID 67176 45797 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL580 LORAZEPAM 67178 45798 TUBA1A 7846 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 67179 45799 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL445813 AT-7519 67180 45800 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL608533 MIDOSTAURIN 67183 45801 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME gemcitabine GEMCITABINE 31616045 67184 45802 TOP2B 7155 DRUGGABLE GENOME, ENZYME AjvW2 67186 45803 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 187051800 BUFEXAMAC 67188 45804 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MK-2461 MK-2461 67189 45805 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TRACAZOLATE TRACAZOLATE 67191 45806 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PX-866 SONOLISIB 67193 45807 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME CARTmeso/19 67194 45808 MAPT 4137 DRUGGABLE GENOME TCMDC-125784 CHEMBL581574 67195 45809 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 405560388 67196 45810 RBP4 5950 DRUGGABLE GENOME US8586571, 6 67197 45811 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME UNC0224 CHEMBL576781 67198 45812 GMNN 51053 DRUGGABLE GENOME DNDI1417420 CHEMBL1546223 67199 45813 GMNN 51053 DRUGGABLE GENOME PROCHLORPERAZINE PROCHLORPERAZINE 67201 45814 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE KENPAULLONE KENPAULLONE 67202 45815 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 artemether ARTEMETHER 18064444,18979093,19926036,19851082,18350255,12920490,12844133 67203 45816 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SJ000244629 CHEMBL592115 67204 45817 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 2-METHOXYPHENAZINE CHEMBL1420181 67205 45818 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135650827 PINDOLOL 67207 45819 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-59 67208 45820 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200935 DARIFENACIN HYDROBROMIDE 67209 45821 NRP2 8828 NA daunorubicin DAUNORUBICIN 18451141 67210 45822 POLA2 23649 NA DACARBAZINE DACARBAZINE 67213 45823 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR D4T STAVUDINE 2538549 67214 45824 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000150791 CHEMBL600572 67215 45825 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TAMOXIFEN TAMOXIFEN 10786679 67216 45826 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000113972 CHEMBL591137 67218 45827 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE GENISTEIN GENISTEIN 11835393 67220 45828 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565579 APITOLISIB 67222 45829 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Exatecan EXATECAN 67223 45830 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX PYRIDINE-2-CARBOTHIOIC ACID PHENYLAMIDE CHEMBL114544 67224 45831 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE HYDROXYCAMPTOTHECIN HYDROXYCAMPTOTHECIN 25481395,22647222,24012683 67228 45832 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 INDINAVIR INDINAVIR 22931300 67231 45833 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME ASN003 67234 45834 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR 5-DEOXY-5-FLUOROURIDINE 12408764 67237 45835 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody 315661210 67238 45836 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1231 OXYBUTYNIN 67239 45837 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Tivozanib TIVOZANIB 26461489 67240 45838 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME ENMD-2076 ENMD-2076 67242 45839 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL521851 PICTILISIB 67243 45840 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MK-1775 ADAVOSERTIB 27601554,27196784,21992793,23520471,21389100,19887545,21799033,28652249,22713237,27998224 67244 45841 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME Inotuzumab Ozogamicin 67245 45842 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-15 67246 45843 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 LABETALOL LABETALOL 22931300 67247 45844 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE EBSELEN EBSELEN 67248 45845 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME FOLFIRI 16636344,17577039,29504153,28502040,17185998,26862009,24815493,20335017,18300238,15297419,18221820,11990381,26857783,19450125,16951398,27160286,16456808,26125934 67250 45846 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR SUBEROHYDROXAMIC ACID SUBEROHYDROXAMIC ACID 16921367 67251 45847 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME inhibitor 178103092 ODANACATIB 67252 45848 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Indoline derivative 17 67253 45849 FAAH 2166 ENZYME, DRUGGABLE GENOME aripiprazole ARIPIPRAZOLE 20631561 67258 45850 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE OLAPARIB OLAPARIB 67259 45851 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Antiandrogens 67261 45852 ERRFI1 54206 CLINICALLY ACTIONABLE ERLOTINIB ERLOTINIB 24550739 67262 45853 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 223366211 CRENOLANIB 67263 45854 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME 2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE CHEMBL412603 67265 45855 TPSAB1 7177 PROTEASE, DRUGGABLE GENOME, ENZYME GM-CSF REGRAMOSTIM 9130550 67266 45856 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Sodium Chloride 67267 45857 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME montelukast MONTELUKAST 19151602,23970434 67269 45858 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME panitumumab PANITUMUMAB 26812186,22537608,26162609,25183481,23071293,22734028,23324806,26371285,27897268,25210463,26438111,20978259,23090619,24727325 67270 45859 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE antibody TRASTUZUMAB TRASTUZUMAB 67271 45860 AKR1C3 8644 ENZYME, DRUGGABLE GENOME BACCHARIN BACCHARIN 22506594 67272 45861 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME NIVOLUMAB NIVOLUMAB 28351930 67273 45862 SFTPA1 653509 DRUGGABLE GENOME RETINOIC ACID 8404646 67274 45863 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor PCI-24781 ABEXINOSTAT 67275 45864 ATAD5 79915 NA CHRYSIN DIMETHYL ETHER CHRYSIN DIMETHYL ETHER 67276 45865 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE UNBS-1450 67277 45866 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-13 67278 45867 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-A5 67279 45868 ALOX15B 247 DRUGGABLE GENOME, ENZYME GNF-PF-2950 CHEMBL602807 67280 45869 TARDBP 23435 TUMOR SUPPRESSOR ESFLURBIPROFEN ESFLURBIPROFEN 67281 45870 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HYPERICIN HYPERICIN 15100173 67283 45871 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL2107762 NERISPIRDINE 67285 45872 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME inhibitor 178102547 67286 45873 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650399 67288 45874 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SULFOBROMOPHTHALEIN SULFOBROMOPHTHALEIN 67289 45875 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME DOVITINIB DOVITINIB 67290 45876 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CEP-1347 CEP-1347 24044867 67291 45877 CYP51A1 1595 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 387065625 67292 45878 EIF2AK2 5610 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 178102648 67293 45879 ATP2A2 488 ENZYME, DRUGGABLE GENOME, TRANSPORTER Gallopamil GALLOPAMIL 67294 45880 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME sorafenib SORAFENIB 27533851 67295 45881 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 249565930 67296 45882 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 67298 45883 GSTM1 2944 DRUGGABLE GENOME, ENZYME clozapine CLOZAPINE 27168101 67300 45884 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-133 67301 45885 GMNN 51053 DRUGGABLE GENOME DIHYDROXANTHOHUMOL DIHYDROXANTHOHUMOL 67302 45886 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 328083461 67303 45887 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL2107341 FISPEMIFENE 67304 45888 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-1549 CHEMBL227959 67306 45889 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651698 67307 45890 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME 681640 CHEMBL379975 67308 45891 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 esomeprazole ESOMEPRAZOLE 67310 45892 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Macitentan MACITENTAN 67311 45893 HKDC1 80201 DRUGGABLE GENOME, KINASE NSC-37642 CHEMBL1707907 67312 45894 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME CYCLOSPORINE CYCLOSPORINE 2337986 67313 45895 IFNG 3458 DRUGGABLE GENOME FONTOLIZUMAB FONTOLIZUMAB 67316 45896 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME BOSUTINIB BOSUTINIB 67317 45897 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor 252827496 67318 45898 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor XL228 XL-228 67319 45899 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BRONOPOL BRONOPOL 67320 45900 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PHN-131 67321 45901 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE PMID27841036-Compound-33 67323 45902 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR JNJ-3534 67324 45903 CRAT 1384 DRUGGABLE GENOME, ENZYME PROPIONYL-L-CARNITINE 67325 45904 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist CHEMBL1274 NILUTAMIDE 67326 45905 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX LIF 15319449 67327 45906 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL482968 ENMD-2076 67328 45907 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-29 67329 45908 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-353263 CHEMBL1383812 67330 45909 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PSD-506 67333 45910 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR METHIMAZOLE METHIMAZOLE 8836317,7991239 67334 45911 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DESIPRAMINE DESIPRAMINE 67335 45912 ATP5F1D 513 TRANSPORTER HALOTHANE HALOTHANE 67336 45913 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor CHEMBL3544942 RONICICLIB 67337 45914 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PHA-767491 CHEMBL225519 67338 45915 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE antibody VITAXIN ETARACIZUMAB 67340 45916 ABCC9 10060 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER CHEMBL2104449 SARAKALIM 67341 45917 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR P-2745 67342 45918 USP1 7398 DNA REPAIR, PROTEASE, ENZYME RO-137410 CHEMBL275311 67344 45919 LGR6 59352 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100588 67345 45920 APH1B 83464 PROTEASE, DRUGGABLE GENOME inhibitor MK0752 67346 45921 ESRRG 2104 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135649800 AFIMOXIFENE 67348 45922 CSK 1445 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE BBI503 67349 45923 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME SNN-0029 67350 45924 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL2108677 PEGINTERFERON BETA-1A 67351 45925 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL117287 PRUCALOPRIDE 67354 45926 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROPOXYPHENE PROPOXYPHENE 67355 45927 HTT 3064 DRUGGABLE GENOME GNF-PF-5134 CHEMBL602969 67356 45928 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-N3 67357 45929 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER BRYOSTATIN-1 67358 45930 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME MEK163 67360 45931 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SCLEROTIORIN SCLEROTIORIN 67361 45932 NAGLU 4669 ENZYME, DRUGGABLE GENOME N-Acetyl-D-glucosamine 67362 45933 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-2383 CHEMBL578915 67363 45934 MT1F 4494 NA CISPLATIN CISPLATIN 12520915 67364 45935 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 340590256 TRILACICLIB 67366 45936 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TAMSULOSIN HYDROCHLORIDE TAMSULOSIN HYDROCHLORIDE 67368 45937 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-137 67370 45938 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3545366 VOXTALISIB 67371 45939 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE IRIGENOL IRIGENOL 67373 45940 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NIFEDIPINE NIFEDIPINE 22931300 67374 45941 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Tamoxifen TAMOXIFEN 67375 45942 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL2062266 DIHYDROCODEINE BITARTRATE 67376 45943 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 252827496 67377 45944 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIBENZ[A,H]ANTHRACENE DIBENZ[A,H]ANTHRACENE 67379 45945 POLI 11201 DNA REPAIR WORTMANNIN WORTMANNIN 67381 45946 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 348353670 TIBOLONE 67382 45947 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TAMATINIB R-406 67383 45948 PRKAB2 5565 KINASE, ENZYME metformin METFORMIN 22722338 67384 45949 TMEM97 27346 NA Isoindoline derivative 2 67385 45950 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650188 67386 45951 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL575448 BMS-754807 67389 45952 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME BEPRIDIL BEPRIDIL 67390 45953 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME LAVENDUSTIN A 12391293 67395 45954 LGR5 8549 G PROTEIN COUPLED RECEPTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 178100587 67396 45955 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KETOCONAZOLE KETOCONAZOLE 67397 45956 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PF-05212384 GEDATOLISIB 16731747,19238632,21325073 67398 45957 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GNF-PF-2301 CHEMBL578061 67402 45958 SCNN1A 6337 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3545352 P-1037 67403 45959 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME TALOTREXIN TALOTREXIN 21879757 67404 45960 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-62 67405 45961 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 67406 45962 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME DOVITINIB DOVITINIB 67409 45963 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-35 67411 45964 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME RO-137410 CHEMBL275311 67413 45965 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 385612212 67415 45966 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METOPROLOL METOPROLOL 67417 45967 AQP1 358 ION CHANNEL, DRUGGABLE GENOME ANDROGENS 12002438 67418 45968 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME lopinavir LOPINAVIR 32022294 67419 45969 CYB5R3 1727 DRUGGABLE GENOME, ENZYME lidocaine / prilocaine 67420 45970 RRM2B 50484 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL1637 GEMCITABINE HYDROCHLORIDE 67423 45971 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 178100940 67424 45972 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE PF-562271 PF-00562271 67426 45973 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE cyclobenzaprine CYCLOBENZAPRINE 18695978 67427 45974 PSMA5 5686 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL325041 BORTEZOMIB 67429 45975 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Tyverb/Tykerb 67430 45976 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SELUMETINIB SELUMETINIB 67431 45977 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DOCONEXENT DOCONEXENT 67432 45978 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RONNEL RONNEL 67433 45979 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PANOBINOSTAT PANOBINOSTAT 67434 45980 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PRASTERONE PRASTERONE 67435 45981 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PYRONIN Y PYRONIN Y 67436 45982 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR NSC-69187 CHEMBL19954 67438 45983 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME 12-O-TETRADECANOYLPHORBOL-13-ACETATE 9242432 67439 45984 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ZIPRASIDONE ZIPRASIDONE 67440 45985 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PIRETANIDE PIRETANIDE 67441 45986 ATP5F1E 514 TRANSPORTER infliximab INFLIXIMAB 26307125 67442 45987 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-704 CHEMBL597449 67443 45988 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TAMOXIFEN CITRATE TAMOXIFEN CITRATE 67444 45989 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102816 67445 45990 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER TARIQUIDAR TARIQUIDAR 67446 45991 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 25003995,22647222,25768699,21783369,23622981,17190463,19530720,25835359 67447 45992 IDO2 169355 ENZYME PMID27172114-Compound-30 67448 45993 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650033 BUPRANOLOL 67450 45994 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Naphthyridine and isoquinoline derivative 1 67452 45995 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649669 67453 45996 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME Gefitinib GEFITINIB 67454 45997 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DARUSENTAN DARUSENTAN 67456 45998 XDH 7498 DRUGGABLE GENOME, ENZYME Fused heterocyclic compound 9 67458 45999 CAMKK2 10645 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE AST-487 AST-487 67459 46000 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CARBIDOPA CARBIDOPA 67460 46001 DDO 8528 DRUGGABLE GENOME MALONIC ACID MALONIC ACID 26322531 67461 46002 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BETHANIDINE BETHANIDINE 67462 46003 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DESOGESTREL DESOGESTREL 67466 46004 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL3545300 CP-459632 67467 46005 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR MILTIRONE MILTIRONE 26339922 67468 46006 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ILORASERTIB ILORASERTIB 67469 46007 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME lusutrombopag LUSUTROMBOPAG 67474 46008 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME THROMBIN THROMBIN 16202257 67476 46009 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200791 OXYMETAZOLINE HYDROCHLORIDE 67477 46010 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CZEN-002 67478 46011 ITGB8 3696 DRUGGABLE GENOME, CELL SURFACE US10035778, Example 12 67480 46012 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650832 PIRENZEPINE 67482 46013 PSME3 10197 NA inhibitor CARFILZOMIB CARFILZOMIB 67483 46014 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME blocker 178100950 AMANTADINE 67484 46015 PDE6D 5147 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL932 DIPYRIDAMOLE 67485 46016 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649744 67486 46017 AKT1S1 84335 KINASE, DRUGGABLE GENOME inhibitor AZD8055 AZD-8055 67488 46018 HSPA4 3308 NA PROTEIN SYNTHESIS INHIBITOR 15827295 67491 46019 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL206834 BAFETINIB 67493 46020 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ETHAVERINE ETHAVERINE 67496 46021 PTGS1 5742 ENZYME, DRUGGABLE GENOME SALSALATE SALSALATE 67498 46022 HLA-DQB1 3119 CLINICALLY ACTIONABLE aspirin ASPIRIN 26366802,15784113,19392989 67500 46023 USP14 9097 ENZYME, CELL SURFACE, PROTEASE inhibitor 328083515 67501 46024 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME RILUZOLE RILUZOLE 67502 46025 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 381118872 67504 46026 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME PMID26161698-Compound-32 67505 46027 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE GDC-0941 PICTILISIB 24322983 67506 46028 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE activator 374883848 67508 46029 TUBB 203068 DRUGGABLE GENOME inhibitor CHEMBL1683544 ERIBULIN MESYLATE 67509 46030 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 cyclophosphamide CYCLOPHOSPHAMIDE 12684728,26894931,18496131 67510 46031 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor 315661265 67512 46032 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-24 67514 46033 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CARFILZOMIB CARFILZOMIB 67516 46034 TIGIT 201633 CELL SURFACE, CLINICALLY ACTIONABLE ASP8374 ASP-8374 67517 46035 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Tricyclic isoxazoloquinazoline derivative 4 67519 46036 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE 5-FU FLUOROURACIL 15206578 67520 46037 ATAD5 79915 NA GNF-PF-67 CHEMBL578512 67521 46038 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE HYDROXYFASUDIL HYDROXYFASUDIL 22257127 67523 46039 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SU-6656 CHEMBL605003 67524 46040 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 67525 46041 ALDH1A1 216 DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 67528 46042 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BAICALEIN BAICALEIN 67531 46043 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL108 CARBAMAZEPINE 67534 46044 MAPT 4137 DRUGGABLE GENOME BITHIONOL BITHIONOL 67536 46045 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201655 INSULIN SUSP ISOPHANE PURIFIED BEEF 67537 46046 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TCMDC-125321 CHEMBL587449 67540 46047 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ATORVASTATIN ATORVASTATIN 11179461 67541 46048 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE VINCRISTINE VINCRISTINE 12874004 67544 46049 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CAULIBUGULONE D CAULIBUGULONE D 67545 46050 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 223366194 67546 46051 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME 20(S)-PROTOPANAXADIOL CHEMBL375563 17261067 67547 46052 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE ENTRECTINIB ENTRECTINIB 67549 46053 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR RS-17053 CHEMBL88272 67550 46054 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-124518 CHEMBL527584 67551 46055 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GW843682X GW843682X 67552 46056 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE etoposide ETOPOSIDE 67553 46057 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME ETAZOLATE ETAZOLATE 67554 46058 MCOLN1 57192 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER activator 178103005 67555 46059 SRSF2 6427 CLINICALLY ACTIONABLE H3B-8800 67556 46060 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE PF-562271 PF-00562271 67558 46061 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ANAZOLENE ANAZOLENE 67561 46062 TSPO 706 DRUGGABLE GENOME Quinazoline derivative 4 67562 46063 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER MORPHINE MORPHINE 18311899 67565 46064 TOP2B 7155 DRUGGABLE GENOME, ENZYME Valrubicin VALRUBICIN 67568 46065 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE MRX-6 67569 46066 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR DIETHYLSTILBESTROL DIETHYLSTILBESTROL 67570 46067 KMO 8564 DRUGGABLE GENOME, ENZYME PMID27172114-Compound-47 67571 46068 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 (S)-ISRADIPINE (S)-ISRADIPINE 67573 46069 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 3,5 DIBROMOTYROSINE DIBROMOTYROSINE 67574 46070 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE ENTINOSTAT ENTINOSTAT 19966789 67575 46071 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AURIN AURIN 67578 46072 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL29741 IRAMPANEL 67579 46073 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TYRPHOSTIN 51 TYRPHOSTIN 51 67582 46074 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ABT-737 ABT 737 21468686 67583 46075 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME PAN-90806 OSI-632 67584 46076 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIMETHYLFORMAMIDE DIMETHYLFORMAMIDE 67585 46077 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ACETAMINOPHEN ACETAMINOPHEN 14644624 67587 46078 NDUFS8 4728 ENZYME inhibitor CHEMBL3545320 ME-344 67588 46079 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 223366077 RGB-286638 67589 46080 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor OSI 027 67591 46081 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PLERIXAFOR PLERIXAFOR 67592 46082 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME SIBUTRAMINE SIBUTRAMINE 67593 46083 SYP 6855 TRANSPORTER MORPHINE MORPHINE 10710628 67595 46084 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME Losmapimod LOSMAPIMOD 67596 46085 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME PEITC 15856023 67597 46086 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROPYLPARABEN PROPYLPARABEN 67599 46087 UBA2 10054 DRUGGABLE GENOME, ENZYME ASTERRIC ACID ASTERRIC ACID 67601 46088 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 67602 46089 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR MK2206 MK-2206 67604 46090 GSTM1 2944 DRUGGABLE GENOME, ENZYME sulfamethoxazole SULFAMETHOXAZOLE 11191886 67607 46091 MAP3K11 4296 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565786 67608 46092 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL296468 BMS-387032 67609 46093 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3545251 SURUFATINIB 67611 46094 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1318477 CHEMBL428064 67614 46095 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME Tricyclic isoxazoloquinazoline derivative 4 67615 46096 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR SULFURIC ACID 1967080 67621 46097 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME ranibizumab RANIBIZUMAB 23570466,22840423,23149126,23559864,23953100,23842101 67622 46098 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL550 PILOCARPINE 67623 46099 UGT1A10 54575 DRUGGABLE GENOME, ENZYME PHENOBARBITAL PHENOBARBITAL 8263600 67625 46100 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME DIMETHYLADENINE DIMETHYLADENINE 67626 46101 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR TAE-684 TAE-684 67627 46102 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135651256 67629 46103 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Flavonoid derivative 4 67630 46104 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME Anti-mesothelin CAR transduced PBL 67631 46105 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL356388 ETAZOLATE 67632 46106 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL BROMAZEPAM BROMAZEPAM 67633 46107 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 fludarabine FLUDARABINE 22584460 67635 46108 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CAMPTOTHECIN CAMPTOTHECIN 7510956 67636 46109 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NITROFURANTOIN NITROFURANTOIN 22931300 67638 46110 HLA-DQB1 3119 CLINICALLY ACTIONABLE lamotrigine LAMOTRIGINE 19668019 67639 46111 SULT1A2 6799 ENZYME, DRUGGABLE GENOME STREPTOZOTOCIN STREPTOZOCIN 7600911 67640 46112 MAPT 4137 DRUGGABLE GENOME FLUPIRTINE MALEATE FLUPIRTINE MALEATE 67642 46113 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-56 67643 46114 SMN2 6607 DRUGGABLE GENOME 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 67644 46115 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GW7074 CHEMBL72365 67645 46116 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CEFIXIME CEFIXIME 67646 46117 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME ATHRAQUINONES A ATHRAQUINONES A 67648 46118 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BAS-8770938 CHEMBL478510 19179076 67649 46119 ATP5F1D 513 TRANSPORTER SEVOFLURANE SEVOFLURANE 67650 46120 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE H2O2 15966013 67651 46121 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE SPIPERONE SPIPERONE 67652 46122 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-2547 CHEMBL601994 67654 46123 RGS4 5999 DRUGGABLE GENOME PALMITOYL-CARNITINE PALMITOYL-CARNITINE 67656 46124 ODC1 4953 DRUGGABLE GENOME, ENZYME EFLORNITHINE EFLORNITHINE 67657 46125 LPAR6 10161 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651509 67658 46126 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3545006 PWT-33587 67659 46127 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 7 67660 46128 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4-AMINOPHENOL 4-AMINOPHENOL 67662 46129 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NOCODAZOLE NOCODAZOLE 67663 46130 SERPINB3 6317 KINASE, PROTEASE INHIBITOR, DRUGGABLE GENOME GONADOTROPINS 8070597 67664 46131 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR PMID26924192-Compound-105 67665 46132 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AS101 AMMONIUM TRICHLOROTELLURATE 9759874 67666 46133 REV3L 5980 DRUGGABLE GENOME, DNA DIRECTED RNA POLYMERASE capecitabine CAPECITABINE 67667 46134 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125567 CHEMBL530049 67670 46135 CD55 1604 DRUGGABLE GENOME, CELL SURFACE INTERLEUKIN-8 14723618 67671 46136 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE ARQ 092 67672 46137 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE mafenide MAFENIDE 4722683 67673 46138 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME CENISERTIB CENISERTIB 67674 46139 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 354702287 67676 46140 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ACACETIN ACACETIN 67677 46141 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME US9024044, 4 67679 46142 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 135652505 67681 46143 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING CUPRIC CHLORIDE CUPRIC CHLORIDE 67682 46144 AQP4 361 ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ACETYLSULFANILAMIDE ACETYLSULFANILAMIDE 18572411 67683 46145 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist 135651899 THYROTROPIN ALFA 67685 46146 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor 384403647 67689 46147 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Azaindazole derivative 2 67690 46148 DNER 92737 NA CPI-0610 67691 46149 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 385612249 67692 46150 GC 2638 DRUGGABLE GENOME Methylene blue 67693 46151 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Sulfisoxazole SULFISOXAZOLE 67694 46152 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE DOXORUBICIN DOXORUBICIN 16905201,12761490 67695 46153 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PT-103 CHEMBL398765 67696 46154 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER rucaparib RUCAPARIB 67697 46155 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 16 67698 46156 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545195 LY-3009120 67699 46157 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE 4-HYDROXY-TAMOXIFEN 11369200 67704 46158 AMD1 262 ENZYME, DRUGGABLE GENOME ORG 34517/34850 67706 46159 MAPT 4137 DRUGGABLE GENOME NIFUROXAZIDE NIFUROXAZIDE 67709 46160 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GALLIC ACID GALLIC ACID 67711 46161 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BROXYQUINOLINE BROXYQUINOLINE 67712 46162 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1742984 AMATUXIMAB 67714 46163 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-138263 CHEMBL535307 67715 46164 MAOB 4129 DRUGGABLE GENOME, ENZYME Selegiline SELEGILINE 67716 46165 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR VALPROIC ACID VALPROIC ACID 18294844,16921367,25304896 67717 46166 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AMBRISENTAN AMBRISENTAN 67718 46167 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME ADINAZOLAM ADINAZOLAM 67719 46168 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME allosteric modulator 385612192 67720 46169 PAPPA 5069 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE TGF 12817760 67723 46170 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 660258 CHEMBL259805 67724 46171 TSC22D3 1831 NA DEXAMETHASONE DEXAMETHASONE 15728202,12707381 67727 46172 FAP 2191 PROTEASE, CELL SURFACE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 363894187 67732 46173 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DIETHYLSTILBESTROL DIPROPIONATE DIETHYLSTILBESTROL DIPROPIONATE 67733 46174 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BERBAMINE BERBAMINE 67738 46175 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR GOSSYPOL GOSSYPOL 67739 46176 SPP1 6696 DRUGGABLE GENOME inhibitor CHEMBL2109530 ASK-8007 67740 46177 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135650180 67741 46178 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TCMDC-123748 CHEMBL530609 67742 46179 FXN 2395 TRANSPORTER, ENZYME CISPLATIN CISPLATIN 12928720 67743 46180 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL454 BUTALBITAL 67744 46181 MAP3K7 6885 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 348353659 67745 46182 PSMD10 5716 TRANSCRIPTION FACTOR BINDING inhibitor CARFILZOMIB CARFILZOMIB 67747 46183 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME inhibitor SIMVASTIN 67748 46184 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 STICTIC ACID STICTIC ACID 67751 46185 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME AG-537 CHEMBL67535 67752 46186 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Isothiazolidine derivative 1 67756 46187 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE FUTUXIMAB/MODOTUXIMAB MIXTURE 26888827 67757 46188 GMNN 51053 DRUGGABLE GENOME DIMERCAPROL DIMERCAPROL 67758 46189 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BUSPIRONE HYDROCHLORIDE BUSPIRONE HYDROCHLORIDE 67759 46190 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TYRPHOSTIN 23 TYRPHOSTIN 23 67760 46191 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME XL888 XL-888 22351686 67761 46192 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor 178101384 67762 46193 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SIRUKUMAB SIRUKUMAB 67763 46194 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE TRICIRIBINE TRICIRIBINE 67765 46195 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR modulator CHEMBL2103846 ULIPRISTAL 67766 46196 ANO1 55107 ION CHANNEL blocker CHEMBL2108184 CROFELEMER 67768 46197 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000117447 CHEMBL592611 67770 46198 PDE3A 5139 ENZYME, DRUGGABLE GENOME MILRINONE MILRINONE 67772 46199 PXN 5829 NA ANTISENSE OLIGONUCLEOTIDES 14576084 67774 46200 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1889140 ROPIVACAINE HYDROCHLORIDE 67776 46201 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DRONEDARONE DRONEDARONE 67777 46202 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 sorafenib SORAFENIB 28362716 67780 46203 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Reparixin REPARIXIN 67781 46204 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE RIFAMPIN RIFAMPIN 6854335 67782 46205 SERPINA1 5265 DRUGGABLE GENOME, PROTEASE INHIBITOR AGTC-0106 67783 46206 APC 324 CLINICALLY ACTIONABLE XAV939 28179481,19759537 67786 46207 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PUTRESCINE DIHYDROCHLORIDE PUTRESCINE DIHYDROCHLORIDE 67788 46208 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VESAMICOL VESAMICOL 67789 46209 RRM2 6241 DRUGGABLE GENOME, ENZYME Gemcitabine GEMCITABINE 67791 46210 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME NONACOG ALFA 67793 46211 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR inhibitor CHEMBL2109585 LY-2382770 67794 46212 CLCN3 1182 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE, TRANSPORTER BUFALIN BUFALIN 23799775 67795 46213 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE LAUROGUADINE LAUROGUADINE 67799 46214 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALL-TRANS RETINOIC ACID 11034076 67800 46215 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DOLASTATIN 12 DOLASTATIN 12 67803 46216 ATXN2 6311 NA NSC-71033 CHEMBL116548 67805 46217 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MEPENZOLATE MEPENZOLATE 67806 46218 SMN2 6607 DRUGGABLE GENOME NSC-26699 CHEMBL221721 67807 46219 DNER 92737 NA PMID26924192-Compound-53 67808 46220 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Heparin Sodium 67809 46221 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME VATALANIB VATALANIB 67811 46222 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PURINE INHIBITORS 10891109,11562960 67813 46223 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME LANSOPRAZOLE LANSOPRAZOLE 67815 46224 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR IL-1 8382509 67816 46225 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME NN-1218 22920797 67817 46226 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 252166785 67818 46227 NDUFA5 4698 ENZYME inhibitor CHEMBL3545135 NV-128 67820 46228 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SOTRASTAURIN SOTRASTAURIN 67821 46229 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 1,4-DIMETHOXYANTHRAQUINONE 1,4-DIMETHOXYANTHRAQUINONE 67822 46230 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL TRIAZOLAM TRIAZOLAM 67824 46231 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL agonist 178103290 67825 46232 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GI-4000 67826 46233 CXCL8 3576 DRUGGABLE GENOME CLARITHROMYCIN CLARITHROMYCIN 12003967 67827 46234 EPHX1 2052 ENZYME, DRUGGABLE GENOME cyclophosphamide CYCLOPHOSPHAMIDE 24533712 67829 46235 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135651419 67830 46236 IFNG 3458 DRUGGABLE GENOME VPM-4-001 67832 46237 BCHE 590 DRUGGABLE GENOME, ENZYME ANESTHETICS 14631501 67834 46238 INSIG2 51141 NA antipsychotics 20877301,18195716,20373477 67835 46239 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CELIPROLOL CELIPROLOL 2903243 67836 46240 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL1287853 FEDRATINIB 67837 46241 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE BAY80-6946 COPANLISIB 67839 46242 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 310264738 CERDULATINIB 67840 46243 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE VERNOLIDE-B CHEMBL2062868 26331426 67842 46244 LGR5 8549 G PROTEIN COUPLED RECEPTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 178100586 67843 46245 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Sirolimus SIROLIMUS 26359452 67844 46246 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME celecoxib CELECOXIB 22336956 67845 46247 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL1079593 VS-5584 67846 46248 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MIFEPRISTONE MIFEPRISTONE 67848 46249 PTGES 9536 DRUGGABLE GENOME, ENZYME Benzimidazole derivative 15 67849 46250 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CHLOROTHALONIL CHLOROTHALONIL 67851 46251 ABCB4 5244 TRANSPORTER, DRUGGABLE GENOME, ENZYME, ABC TRANSPORTER Curcumin CURCUMIN 67853 46252 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 381744979 NARINGENIN 67854 46253 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ETOPOSIDE ETOPOSIDE 14514923,24065105 67856 46254 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR inhibitor 249565597 67858 46255 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor 249565590 CHEMBL1236539 67859 46256 CFLAR 8837 DRUG RESISTANCE, DRUGGABLE GENOME, PROTEASE CABOZANTINIB CABOZANTINIB 67860 46257 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR GAMMA HYDROXYBUTYRIC ACID 67861 46258 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135651527 67862 46259 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIHYDROTACHYSTEROL DIHYDROTACHYSTEROL 67864 46260 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE BISPHOSPHONATES 11984068 67865 46261 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-95397 CHEMBL429095 67867 46262 PSENEN 55851 DRUGGABLE GENOME inhibitor CHEMBL463981 BEGACESTAT 67868 46263 LTB 4050 DRUGGABLE GENOME BAMINERCEPT BAMINERCEPT 67869 46264 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HYPOTAURINE HYPOTAURINE 67870 46265 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CIRAZOLINE CIRAZOLINE 67871 46266 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME RG7304 67872 46267 GCLC 2729 DRUGGABLE GENOME, ENZYME BUTHIONINE SULFOXIMINE 8101766,9610371 67873 46268 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 252166498 TRAMADOL 67874 46269 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 2,7-BIS[3-(PIPERIDINO)PROPIONAMIDO]ANTHRAQUINONE CHEMBL89250 18571928 67875 46270 GMNN 51053 DRUGGABLE GENOME RIMONABANT RIMONABANT 67879 46271 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565638 ALPELISIB 67881 46272 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR inhibitor 315661200 CPI-1205 67882 46273 CXCL8 3576 DRUGGABLE GENOME ALDRIN ALDRIN 67883 46274 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure1-Sarcaboside A 67884 46275 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103116 FASIDOTRILAT 67887 46276 F12 2161 DRUGGABLE GENOME, ENZYME, PROTEASE PENTAMIDINE ISETHIONATE PENTAMIDINE ISETHIONATE 67888 46277 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CID 3237815 CHEMBL410484 67889 46278 ALDH1A1 216 DRUGGABLE GENOME, ENZYME LY-83583 CHEMBL312487 67890 46279 NELFCD 51497 KINASE hydrochlorothiazide HYDROCHLOROTHIAZIDE 67891 46280 TMEM97 27346 NA Benzamide derivative 1 67892 46281 CAMK1D 57118 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME TAE-684 TAE-684 67893 46282 ALPL 249 ENZYME, DRUGGABLE GENOME DNDI1417629 CHEMBL1731432 67894 46283 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor BI847325 67895 46284 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 310264672 67897 46285 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-206553 CHEMBL297784 67898 46286 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL1672054 CASOPITANT 67899 46287 PGA3 643834 PROTEASE, DRUGGABLE GENOME, ENZYME ECABET ECABET 67900 46288 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE lamotrigine LAMOTRIGINE 19668019 67901 46289 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME 2,4-DIAMINOTOLUENE CHEMBL541230 67903 46290 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR GENISTEIN GENISTEIN 7476882 67906 46291 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE GW441756X GW441756X 67907 46292 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor PCI-24781 ABEXINOSTAT 67909 46293 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 67910 46294 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME CAMPTOTHECIN CAMPTOTHECIN 67912 46295 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 315661272 ZYKLOPHIN 67913 46296 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-2812 CHEMBL125044 67914 46297 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Bivalirudin BIVALIRUDIN 67915 46298 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME AMARANTH AMARANTH 67918 46299 ACP1 52 ENZYME, DRUGGABLE GENOME, PROTEIN PHOSPHATASE DNDI1417461 CHEMBL1520282 67919 46300 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR RIZATRIPTAN RIZATRIPTAN 67921 46301 GPR39 2863 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist 223366134 67922 46302 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BENSERAZIDE BENSERAZIDE 67923 46303 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1201115 ESMOLOL HYDROCHLORIDE 67924 46304 POLK 51426 DNA REPAIR, ENZYME TETRAIDOFLUORESCEIN TETRAIDOFLUORESCEIN 67925 46305 SLC9A3 6550 DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE, EXCHANGER RDX-5791 TENAPANOR HYDROCHLORIDE 67928 46306 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR AZD8186 AZD-8186 67929 46307 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR TAK-715 TAK-715 67930 46308 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL481958 AMRUBICIN HYDROCHLORIDE 67932 46309 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BRL-50481 CHEMBL484928 67933 46310 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE SB-218795 CHEMBL9843 67934 46311 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME PC-SPES 14532991 67936 46312 POLK 51426 DNA REPAIR, ENZYME NSC-130813 CHEMBL463783 67937 46313 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TRICHOSTATIN TRICHOSTATIN 67938 46314 PLK3 1263 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME MLN-8054 MLN-8054 67939 46315 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SJ000113972 CHEMBL591137 67942 46316 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE JSM 6427 67944 46317 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE DASATINIB DASATINIB 67945 46318 PDE10A 10846 ENZYME, DRUGGABLE GENOME DIPYRIDAMOLE DIPYRIDAMOLE 67948 46319 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 artemisinin ARTEMISININ 18064444,18979093,19926036,19851082,18350255,12920490,12844133 67950 46320 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME C5A 15313431 67952 46321 TUBB2A 7280 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 67953 46322 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PAROXETINE PAROXETINE 67955 46323 GMNN 51053 DRUGGABLE GENOME FELODIPINE FELODIPINE 67957 46324 COL18A1 80781 DRUGGABLE GENOME CELECOXIB CELECOXIB 12232050 67958 46325 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Epoxysuccinate derivative 5 67960 46326 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE PMSG 2506647,3121412 67962 46327 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIMETHYL GAMBOGATE DIMETHYL GAMBOGATE 67963 46328 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-19803 CHEMBL522983 67964 46329 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SPIRONOLACTONE SPIRONOLACTONE 67965 46330 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE METHYLPREDNISOLONE METHYLPREDNISOLONE 9169090 67968 46331 GART 2618 ENZYME, DRUGGABLE GENOME PEMETREXED PEMETREXED 67969 46332 TAC1 6863 DRUGGABLE GENOME WORTMANNIN WORTMANNIN 9850167 67970 46333 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BISOPROLOL BISOPROLOL 67971 46334 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME NSC-9037 CHEMBL1451216 67972 46335 NT5C3A 51251 ENZYME idarubicin IDARUBICIN 25000516 67973 46336 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CLOZAPINE CLOZAPINE 67974 46337 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL552212 LEXIBULIN 67975 46338 ERAP2 64167 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE inhibitor CHEMBL2103847 TOSEDOSTAT 67977 46339 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GENISTEIN GENISTEIN 7769390 67978 46340 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL2323775 MK-8033 67979 46341 ATXN2 6311 NA EPIRUBICIN HYDROCHLORIDE EPIRUBICIN HYDROCHLORIDE 67981 46342 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-44 67982 46343 GAA 2548 DRUGGABLE GENOME, ENZYME TCMDC-125528 CHEMBL375673 67984 46344 HLA-DQB1 3119 CLINICALLY ACTIONABLE lumiracoxib LUMIRACOXIB 20639878 67985 46345 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR METHYLTESTOSTERONE METHYLTESTOSTERONE 67989 46346 SPP1 6696 DRUGGABLE GENOME 12-O-TETRADECANOYLPHORBOL-13-ACETATE 12009309 67993 46347 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antibody RG7446 ATEZOLIZUMAB 67994 46348 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Topetecan 67995 46349 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME IP10.C8-1 67996 46350 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE REMIFENTANIL REMIFENTANIL 67997 46351 HSPD1 3329 DRUGGABLE GENOME, ENZYME, CELL SURFACE ATORVASTATIN ATORVASTATIN 15678257 67998 46352 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME 1,2,4-triazolo[1,5a]pyridine derivative 2 68000 46353 SLC36A1 206358 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 178101420 68001 46354 CBX1 10951 NA CARISOPRODOL CARISOPRODOL 68002 46355 MARCHF8 220972 ENZYME LEISH-F1 68003 46356 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178101977 68005 46357 GMNN 51053 DRUGGABLE GENOME DASATINIB DASATINIB 68008 46358 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545366 VOXTALISIB 68009 46359 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DILTIAZEM DILTIAZEM 22931300 68010 46360 HSP90B1 7184 DRUGGABLE GENOME inhibitor 315661302 68012 46361 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL PROPOFOL PROPOFOL 68013 46362 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 178102304 TOFACITINIB 68014 46363 FXYD2 486 DRUGGABLE GENOME, TRANSPORTER CYCLOTHIAZIDE CYCLOTHIAZIDE 68017 46364 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8598210, Table XV, 2 68018 46365 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 3',4' DICHLOROBENZAMIL 3',4' DICHLOROBENZAMIL 68019 46366 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TYRPHOSTIN AG-112 CHEMBL76589 68021 46367 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure1-Chukrasone B 68022 46368 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor REGORAFENIB REGORAFENIB 68023 46369 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PRIMAQUINE PHOSPHATE PRIMAQUINE PHOSPHATE 68026 46370 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME allosteric modulator 249565778 TASQUINIMOD 68027 46371 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PLX2853 68028 46372 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 363894133 68030 46373 GUCY2C 2984 DRUGGABLE GENOME, KINASE agonist 178101555 68033 46374 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHYLENE BLUE CHLORIDE HYDRATE METHYLENE BLUE 68034 46375 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MM-111 MM-111 68036 46376 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor VALPROIC ACID DEPAKOTE 68038 46377 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL3545153 DE-104 68039 46378 HMOX1 3162 ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE SORAFENIB SORAFENIB 26309414 68040 46379 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE SDZ-281-240 68041 46380 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651017 68042 46381 CDH1 999 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BI2536 26597303 68043 46382 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUOROSALAN FLUOROSALAN 68044 46383 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TOZASERTIB TOZASERTIB 68045 46384 GAA 2548 DRUGGABLE GENOME, ENZYME TCMDC-125738 CHEMBL527585 68048 46385 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker 135651250 68049 46386 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MILCICLIB MILCICLIB 19603809 68050 46387 HDAC11 79885 DRUGGABLE GENOME, ENZYME TACEDINALINE TACEDINALINE 18692397 68051 46388 ATAD2 29028 NUCLEAR HORMONE RECEPTOR, ENZYME inhibitor 385612205 68052 46389 HDAC11 79885 DRUGGABLE GENOME, ENZYME SCRIPTAID SCRIPTAID 19966789 68053 46390 MDM4 4194 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, DRUGGABLE GENOME ATEZOLIZUMAB ATEZOLIZUMAB 28351930 68054 46391 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1522 ESZOPICLONE 68060 46392 STK33 65975 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 68061 46393 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor ERLOTINIB ERLOTINIB 68064 46394 PPCDC 60490 ENZYME zoledronate ZOLEDRONIC ACID 68066 46395 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL3545073 AMA0076 68067 46396 MARCHF8 220972 ENZYME GSK2592984A 68068 46397 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3286 CHEMBL581880 68069 46398 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000260249 CHEMBL601311 68070 46399 PROS1 5627 DRUGGABLE GENOME estradiol / progesterone 68071 46400 TMEM97 27346 NA Benzamide derivative 11 68073 46401 MAPT 4137 DRUGGABLE GENOME STREPTONIGRIN STREPTONIGRIN 68074 46402 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME AG-555 CHEMBL53898 68077 46403 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE FORMOTEROL FORMOTEROL 68078 46404 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL552212 LEXIBULIN 68079 46405 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-19 68080 46406 BAZ2B 29994 NA PYROGALLOL RED PYROGALLOL RED 68081 46407 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor BAY80-6946 COPANLISIB 68085 46408 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME ENTRECTINIB ENTRECTINIB 68086 46409 CFL1 1072 KINASE MG-132 MG-132 16680159 68087 46410 ALOX15 246 ENZYME, DRUGGABLE GENOME FRAXETIN FRAXETIN 68089 46411 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME SOTRASTAURIN SOTRASTAURIN 68091 46412 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200409 LIDOCAINE HYDROCHLORIDE 68092 46413 ATAD5 79915 NA CID 670282 CHEMBL260213 68093 46414 MPHOSPH8 54737 NA RESERPINE RESERPINE 68095 46415 GMNN 51053 DRUGGABLE GENOME GNF-PF-2335 CHEMBL601146 68098 46416 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TEPOTINIB TEPOTINIB 25736998 68099 46417 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CHRYSENE-1,4-DIONE CHEMBL421215 68101 46418 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Quinoline and quinazoline derivative 6 68102 46419 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER Posiphen R-phenserine 68103 46420 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME GABAPENTIN GABAPENTIN 68104 46421 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME CANNABINOL CANNABINOL 6140904 68105 46422 SMN2 6607 DRUGGABLE GENOME SU-6656 CHEMBL605003 68106 46423 GAA 2548 DRUGGABLE GENOME, ENZYME CARBARIL CARBARIL 68108 46424 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 (R)-PINOCEMBRIN (R)-PINOCEMBRIN 68109 46425 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Flavonoid derivative 8 68111 46426 PRORP 9692 NA zileuton ZILEUTON 25963335 68112 46427 ALOX15 246 ENZYME, DRUGGABLE GENOME PROCARBAZINE PROCARBAZINE 68113 46428 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR 2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE CHEMBL201325 68114 46429 COL2A1 1280 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 68115 46430 POLB 5423 DNA REPAIR, DRUGGABLE GENOME EBSELEN EBSELEN 68116 46431 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME aspirin ASPIRIN 26398624 68118 46432 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE Lexatumumab LEXATUMUMAB 68119 46433 MUCL3 135656 NA carboplatin CARBOPLATIN 31616045 68121 46434 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ARVERAPAMIL 68122 46435 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL3545389 LY2245461 68123 46436 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OXOGLAUCINE OXOGLAUCINE 68127 46437 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE US8614253, 29-1 68128 46438 KDM4A 9682 DRUGGABLE GENOME, ENZYME AZASERINE AZASERINE 68129 46439 APOE 348 DRUGGABLE GENOME IRBESARTAN IRBESARTAN 12827021 68130 46440 RAB9A 9367 ENZYME, DRUGGABLE GENOME 4'-METHOXYFLAVONE 4'-METHOXYFLAVONE 68132 46441 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Chlorpropamide CHLORPROPAMIDE 68133 46442 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE pravastatin PRAVASTATIN 16103896 68136 46443 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME FLURAZEPAM FLURAZEPAM 68137 46444 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR palbociclib PALBOCICLIB 68138 46445 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652056 68139 46446 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CARVEDILOL CARVEDILOL 12835612 68141 46447 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME daunorubicin DAUNORUBICIN 24021215 68142 46448 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE XAV939 28611108 68143 46449 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL2104391 INSULIN DETEMIR 68144 46450 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1-BENZYLMALEIMIDE CHEMBL388979 68146 46451 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 1,2-NAPHTHOQUINONE 1,2-NAPHTHOQUINONE 68147 46452 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 340590279 FOSDAGROCORAT 68149 46453 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BENZO[DE]ISOCHROMEN-1(3H)-ONE CHEMBL1479195 68150 46454 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 404859123 68151 46455 TUBB 203068 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 68152 46456 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 135649950 APOMORPHINE 68155 46457 FST 10468 DRUGGABLE GENOME ANTIBIOTICS 15168744 68157 46458 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME ANTIBIOTIC ANTIBIOTIC 9422737 68158 46459 LRP1 4035 KINASE, DRUGGABLE GENOME ANTISENSE OLIGONUCLEOTIDES 11095961 68159 46460 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME RITANSERIN RITANSERIN 68160 46461 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 329968432 68161 46462 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DABRAFENIB DABRAFENIB 27135738 68162 46463 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TPCK TPCK 68163 46464 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME methotrexate METHOTREXATE 29791011 68168 46465 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 252827463 68169 46466 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OLEANDEROLIDE OLEANDEROLIDE 24326278 68170 46467 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE CENISERTIB CENISERTIB 68171 46468 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR PROTEASOME INHIBITOR 10555040 68172 46469 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme21Left 68174 46470 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650496 68177 46471 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BIIB014 68178 46472 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652624 68179 46473 SETD7 80854 ENZYME, METHYL TRANSFERASE EOSIN EOSIN 18348515 68180 46474 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYCLOPIAZONIC ACID CYCLOPIAZONIC ACID 68182 46475 ICAM3 3385 DRUGGABLE GENOME GM-CSF REGRAMOSTIM 12600815 68183 46476 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650496 68186 46477 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CHOLECALCIFEROL CHOLECALCIFEROL 68188 46478 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME RG-1530 RG-1530 68189 46479 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3360203 PILARALISIB 68194 46480 STMN1 3925 DRUG RESISTANCE PACLITAXEL PACLITAXEL 24587245 68196 46481 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 midazolam MIDAZOLAM 25588320 68197 46482 TRPM7 54822 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ION CHANNEL, ENZYME, TRANSPORTER activator 135652738 68198 46483 PTGS2 5743 DRUGGABLE GENOME, ENZYME Flufenamic Acid 68199 46484 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME vemurafenib VEMURAFENIB 68200 46485 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL1980297 ILORASERTIB 68201 46486 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NAPROXEN NAPROXEN 22931300 68202 46487 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR TAE-684 TAE-684 68203 46488 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE DASATINIB DASATINIB 68204 46489 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME GW8510 CHEMBL1276446 68207 46490 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 68208 46491 CP 1356 DRUGGABLE GENOME, ENZYME DANAZOL DANAZOL 489712 68210 46492 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME ACRIFLAVINE CHLORIDE ACRIFLAVINE 68211 46493 ATAD5 79915 NA TCMDC-124522 CHEMBL526776 68212 46494 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ENTINOSTAT ENTINOSTAT 19966789,20491440 68213 46495 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LANSOPRAZOLE SULFIDE LANSOPRAZOLE SULFIDE 68215 46496 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MGAH22 MARGETUXIMAB 68216 46497 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-59 68219 46498 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1615374 VILAZODONE HYDROCHLORIDE 68220 46499 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DOXEPIN DOXEPIN 68221 46500 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE activator CHEMBL2107885 RETEPLASE 68223 46501 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME TRAMETINIB TRAMETINIB 23020132,29072975,24345920,22798288,25399551,30792255,25452114,29903880,24933606,25265494,22805292,22663011,27283860,22169769,29156677,27048246,24583796,25265492,26314551,28947956,31010895,28891408,29431699 68226 46502 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BENOMYL BENOMYL 68228 46503 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Ponatinib PONATINIB 22328973 68229 46504 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR inhibitor CHEMBL1750 CLOFARABINE 68230 46505 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME ICA-17043 SENICAPOC 68231 46506 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200963 BIMATOPROST 68232 46507 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolo[2,3-d]pyrimidine derivative 4 68234 46508 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE BESTATIN 16800923 68235 46509 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SULFOBROMOPHTHALEIN SULFOBROMOPHTHALEIN 68239 46510 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GFT14 68241 46511 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR TAMARIXETIN TAMARIXETIN 25190466 68244 46512 DGAT1 8694 ENZYME, DRUGGABLE GENOME inhibitor 223366163 68245 46513 HPSE 10855 ENZYME, DRUGGABLE GENOME PI-88 MUPARFOSTAT 68246 46514 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME SILYMARIN SILYBIN A 15290869 68248 46515 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3545411 MF101 68249 46516 FAAH 2166 ENZYME, DRUGGABLE GENOME Azetidine urea derivative 1 68250 46517 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME RGB-286638 RGB-286638 68251 46518 NOS1 4842 DRUGGABLE GENOME, ENZYME GABAPENTIN GABAPENTIN 12817894 68252 46519 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SAR231893 DUPILUMAB 68253 46520 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE RECOMBINANT HUMAN GROWTH HORMONE 68254 46521 S1PR2 9294 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651563 68255 46522 PDE4B 5142 DRUGGABLE GENOME, ENZYME SOTB07 68258 46523 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3137336 UPROSERTIB 68259 46524 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-102742 CHEMBL1519374 68260 46525 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE Drugs used in nicotine dependence 15007373,17224915 68262 46526 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE BRYOSTATIN-1 68263 46527 MAPT 4137 DRUGGABLE GENOME DNDI1417614 CHEMBL1567571 68264 46528 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PF-562271 PF-00562271 68265 46529 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Rigosertib RIGOSERTIB 68266 46530 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor 178103455 TOPIRAMATE 68267 46531 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE LOXO-101 LAROTRECTINIB 68273 46532 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME antibody 354702217 EMICIZUMAB 68274 46533 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BGJ398 INFIGRATINIB 68275 46534 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OUABAIN OUABAIN 68276 46535 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor PI-103 PI-103 68277 46536 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE 178101616 68280 46537 NT5C2 22978 ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MERCAPTOPURINE MERCAPTOPURINE 23377183,23377281 68281 46538 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME methazolamide METHAZOLAMIDE 30242287,25970075,9109770,20504258,25918017 68282 46539 VEGFC 7424 GROWTH FACTOR, TRANSPORTER, DRUGGABLE GENOME LENALIDOMIDE LENALIDOMIDE 68284 46540 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GEFITINIB GEFITINIB 68286 46541 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER LY411575 26855149 68287 46542 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 404859118 68288 46543 BAZ2B 29994 NA AG-538 CHEMBL56393 68291 46544 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALPHA INTERFERON CETUXIMAB 8857944 68292 46545 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IMAZODAN IMAZODAN 68293 46546 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651031 SCOPOLAMINE 68295 46547 COMT 1312 DRUGGABLE GENOME, ENZYME PGX-200097 68296 46548 BAZ2B 29994 NA MEDRONIC ACID MEDRONIC ACID 68297 46549 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR NICOTINE NICOTINE 10198208 68300 46550 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR RG-1530 RG-1530 68301 46551 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR HINOKITIOL HINOKITIOL 68302 46552 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178103951 DINACICLIB 68304 46553 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649797 4-DAMP 68305 46554 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Cabozantinib CABOZANTINIB 68308 46555 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME DT01 26637369 68309 46556 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE RG-1530 RG-1530 68311 46557 MPHOSPH8 54737 NA T-1032 CHEMBL77971 68312 46558 FOXO1 2308 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BET INHIBITOR 28446439 68315 46559 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE CEDIRANIB CEDIRANIB 68316 46560 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME AZD1208 68317 46561 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME NSC-108783 CHEMBL1489812 68318 46562 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR DOCETAXEL DOCETAXEL 24647522 68319 46563 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Cipatinib 68320 46564 ATAD5 79915 NA VINCAMINE VINCAMINE 68322 46565 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL967 TEMAZEPAM 68323 46566 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor 178101942 68324 46567 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1645462 AC-480 68325 46568 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SODIUM AZIDE SODIUM AZIDE 68327 46569 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR modulator CHEMBL3137304 DAGROCORAT 68331 46570 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL2326966 SF-1126 68333 46571 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE blocker CHEMBL1083993 AMIODARONE HYDROCHLORIDE 68334 46572 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE inhibitor CHEMBL1515 METHIMAZOLE 68335 46573 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist CHEMBL2108730 SARILUMAB 68336 46574 LGR6 59352 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100589 68339 46575 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE BAY-613606 CHEMBL541400 68340 46576 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME VANDETANIB VANDETANIB 68341 46577 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BYL719 ALPELISIB 28363909,27312529,26577700 68342 46578 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Gefitinib GEFITINIB 26545934,23220880,17638894 68345 46579 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ROPINIROLE ROPINIROLE 68347 46580 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GW0742 CHEMBL38508 68348 46581 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PMID27336223-Compound-8 68349 46582 MAPT 4137 DRUGGABLE GENOME CGP-53353 CGP-53353 68350 46583 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME SULFASALAZINE SULFASALAZINE 68351 46584 RAPGEF3 10411 ENZYME NSC-228155 CHEMBL505670 68352 46585 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Fluorouracil FLUOROURACIL 26341920 68353 46586 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE DIGITOXIN DIGITOXIN 68355 46587 SERPINF1 5176 DRUGGABLE GENOME, PROTEASE INHIBITOR PEDF gene therapy 68356 46588 TUBB 203068 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 68359 46589 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Pertuzumab PERTUZUMAB 68360 46590 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 328083468 68362 46591 MAOA 4128 DRUGGABLE GENOME, ENZYME ISOCARBOXAZID ISOCARBOXAZID 68363 46592 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR TCMDC-125758 CHEMBL546797 68366 46593 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE CD40L 10520003 68367 46594 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545401 X-82 68369 46595 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME activator 135651521 NADIDE 68371 46596 KDM4A 9682 DRUGGABLE GENOME, ENZYME R(-)-PROPYLNORAPOMORPHINE HCL CHEMBL538542 68372 46597 POLK 51426 DNA REPAIR, ENZYME HYDROXYZINE PAMOATE HYDROXYZINE PAMOATE 68375 46598 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE PERMETHRIN PERMETHRIN 68377 46599 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200694 SEVOFLURANE 68378 46600 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME DASATINIB DASATINIB 68379 46601 DEPTOR 64798 KINASE inhibitor AZD8055 AZD-8055 68381 46602 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE SB-242235 SB-242235 68383 46603 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW301784X GW301784X 68385 46604 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE INOC-005 68386 46605 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FLUMEQUINE FLUMEQUINE 68387 46606 MAPT 4137 DRUGGABLE GENOME NSC-92207 CHEMBL139935 68388 46607 HSPA8 3312 TUMOR SUPPRESSOR NSC-119911 CHEMBL502775 68389 46608 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE 2'H,4H-[2,6'-BICHROMEN]-4-ONE CHEMBL2347759 23600958 68391 46609 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE N/A 26276366,18648004,16384925,25729899,25111512,25193432 68395 46610 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BERBAMINE BERBAMINE 68396 46611 GMNN 51053 DRUGGABLE GENOME DNDI1417181 CHEMBL1537417 68397 46612 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 381118866 68400 46613 BAZ2B 29994 NA GNF-PF-2298 CHEMBL578905 68404 46614 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 codeine CODEINE 9187528 68405 46615 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME MEDI7814 68406 46616 ALOX15 246 ENZYME, DRUGGABLE GENOME SCH-58261 SCH-58261 68407 46617 BAZ2B 29994 NA GNF-PF-3925 CHEMBL584248 68408 46618 F2RL3 9002 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 381744951 68409 46619 DHODH 1723 DRUGGABLE GENOME, ENZYME inhibitor 178103431 LEFLUNOMIDE 68410 46620 KDM4A 9682 DRUGGABLE GENOME, ENZYME DOMOIC ACID DOMOIC ACID 68411 46621 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545324 RG-7666 68412 46622 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CLIOQUINOL CLIOQUINOL 68414 46623 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor 404859123 68417 46624 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33k 68418 46625 CES2 8824 DRUGGABLE GENOME, ENZYME irinotecan IRINOTECAN 68421 46626 HTT 3064 DRUGGABLE GENOME GNF-PF-4057 CHEMBL598903 68423 46627 VKORC1 79001 DRUGGABLE GENOME, ENZYME Warfarin WARFARIN 68424 46628 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PI-3065 24919154 68427 46629 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652102 DESMOPRESSIN 68428 46630 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL421 SULFASALAZINE 68429 46631 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME TAMATINIB R-406 68430 46632 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 68431 46633 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME MITOXANTRONE MITOXANTRONE 68432 46634 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ENDOSULFAN ENDOSULFAN 68434 46635 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL3545402 XL-820 68436 46636 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME PHENOBARBITAL PHENOBARBITAL 9187311 68438 46637 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TCMDC-124522 CHEMBL526776 68439 46638 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 13-CIS-RETINAL CHEMBL1579130 68442 46639 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIBROMSALAN TRIBROMSALAN 68444 46640 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME DEFOROLIMUS RIDAFOROLIMUS 68445 46641 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200521 ALMOTRIPTAN MALATE 68446 46642 RAB9A 9367 ENZYME, DRUGGABLE GENOME 1,2-DIMETHOXY-ANTHRAQUINONE CHEMBL52884 68447 46643 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 warfarin WARFARIN 11353757 68449 46644 SULT2B1 6820 ENZYME, DRUGGABLE GENOME gemtuzumab ozogamicin 22584460 68450 46645 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR OPIATE 7821394 68451 46646 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TENATOPRAZOLE TENATOPRAZOLE 68452 46647 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR NIFEDIPINE NIFEDIPINE 68453 46648 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SOU-001 68454 46649 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHEMBL220492 TOPIRAMATE 68455 46650 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR APG-1387 68457 46651 TYMSOS 494514 NA mercaptopurine MERCAPTOPURINE 68458 46652 UST 10090 NA nortriptyline NORTRIPTYLINE 20360315,25916525 68459 46653 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE OZORALIZUMAB OZORALIZUMAB 68460 46654 FUT3 2525 ENZYME Rebmab-100 68461 46655 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9617250, Example 1 Example 204 of D1 68462 46656 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR ethinyl estradiol / norelgestromin 68463 46657 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE activator CHEMBL1201593 ALTEPLASE 68464 46658 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-40 68468 46659 HMGCR 3156 ENZYME, DRUGGABLE GENOME Hexahydro naphthalene derivative 1 68469 46660 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-63 68471 46661 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME BENZO[B]FLUORANTHENE BENZO[B]FLUORANTHENE 68472 46662 MAPT 4137 DRUGGABLE GENOME HYDROXYZINE PAMOATE HYDROXYZINE PAMOATE 68474 46663 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DIPHENYLPYRALINE DIPHENYLPYRALINE 68475 46664 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DESACETOXYMATRICARIN DESACETOXYMATRICARIN 68476 46665 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ERYTHROSINE ERYTHROSINE 68477 46666 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201177 LEVOBUNOLOL HYDROCHLORIDE 68478 46667 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE pembrolizumab PEMBROLIZUMAB 26086854 68479 46668 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3544966 GSK-1059615 68480 46669 SLC38A3 10991 TRANSPORTER 178101352 68482 46670 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201117 METHOCARBAMOL 68483 46671 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 328083457 68484 46672 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME BORTEZOMIB BORTEZOMIB 68486 46673 GAA 2548 DRUGGABLE GENOME, ENZYME PHENOTHIAZINE PHENOTHIAZINE 68487 46674 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-367089 CHEMBL1543865 68488 46675 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME SP-600125 SP-600125 23634759 68489 46676 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-3464 CHEMBL602213 68490 46677 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TOLAZOLINE TOLAZOLINE 68491 46678 SLC1A2 6506 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE 178101255 68492 46679 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE VS-5584 VS-5584 23270925 68493 46680 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 404859062 BALOVAPTAN 68495 46681 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BEZ235 DACTOLISIB 21966435,26272063,23629727,22543857,27974663,23475782,26270481,28446642,24939055,26627007,19029981,26232337,24927217,26013318,22662154,26137449 68496 46682 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 310264733 FIMEPINOSTAT 68497 46683 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545380 68498 46684 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR EGCG EPIGALOCATECHIN GALLATE 17369354 68500 46685 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CARBAMAZEPINE CARBAMAZEPINE 16981842 68502 46686 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Rucaparib RUCAPARIB 68503 46687 XDH 7498 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200477 ALLOPURINOL SODIUM 68504 46688 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Clomifene CLOMIPHENE 68505 46689 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME DNDI1318477 CHEMBL428064 68506 46690 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL1200699 DOXYCYCLINE 68507 46691 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CARBOPLATIN CARBOPLATIN 11595686 68508 46692 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR GENTIAN VIOLET GENTIAN VIOLET 68510 46693 UBE2N 7334 ENZYME, DRUGGABLE GENOME PERPHENAZINE PERPHENAZINE 68513 46694 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME CISPLATIN CISPLATIN 14871998 68514 46695 POLB 5423 DNA REPAIR, DRUGGABLE GENOME HTS-05057 CHEMBL372629 68517 46696 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME MTOR INHIBITOR 26831717 68521 46697 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR alpelisib ALPELISIB 68524 46698 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME TRIPHENYLSTANNYL ACETATE TRIPHENYLSTANNYL ACETATE 68527 46699 UBE2N 7334 ENZYME, DRUGGABLE GENOME TEGASEROD MALEATE TEGASEROD MALEATE 68528 46700 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LY-2090314 LY-2090314 68529 46701 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME hmg coa reductase inhibitors 17108811,15970799,18650507,24595600,16103896,25673568,17473846,23930675,25446771,24263182,1092254,11477075,26086347,24598718,17620857,21243006,12811365,18794729,12670950,23708174,15226675,26367500,23436703,11134001,21178985,15116054,17177112,21928084,23361102,16678544,24810685,22668755,25630984,28812116,25350695,16014768,17015053 68531 46702 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE cabozantinib CABOZANTINIB 27694386,26432786,25971939,28192597,28396313 68532 46703 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Acolbifene ACOLBIFENE 68534 46704 TUBA1A 7846 DRUGGABLE GENOME ABT-751 ABT-751 25468039 68535 46705 UBC 7316 KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US20130237529 36 68536 46706 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178101897 68537 46707 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GUTHION GUTHION 68538 46708 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124176 CHEMBL588038 68540 46709 IGFBP1 3484 DRUGGABLE GENOME DROLOXIFENE DROLOXIFENE 8645625 68541 46710 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Cabozantinib CABOZANTINIB 27694386 68544 46711 PDE4D 5144 DRUGGABLE GENOME, ENZYME TOFIMILAST TOFIMILAST 68545 46712 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME L-655708 CHEMBL52030 22137933 68546 46713 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIRINIXIC ACID PIRINIXIC ACID 68548 46714 GCLC 2729 DRUGGABLE GENOME, ENZYME L-BUTHIONINE SULFOXIMINE 9660546 68549 46715 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PYRIDOXINE PYRIDOXINE 16277693 68552 46716 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR METHYLENE BLUE CHLORIDE HYDRATE METHYLENE BLUE 68553 46717 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME RECOMBINANT FACTOR IX FC FUSION PROTEIN 68554 46718 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 POLYETHYLENE GLYCOL 10634315 68555 46719 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR olaparib OLAPARIB 68556 46720 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE ZOLEDRONATE ZOLEDRONIC ACID 11984068 68557 46721 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BAY-X-7195 CHEMBL314115 68559 46722 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL PAGOCLONE PAGOCLONE 68563 46723 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-44 68564 46724 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor BARASERTIB BARASERTIB 68565 46725 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BUSULFAN BUSULFAN 22931300 68566 46726 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BENZPHETAMINE BENZPHETAMINE 68567 46727 OGA 10724 ENZYME, DRUGGABLE GENOME STZ STREPTOZOCIN 11336633 68568 46728 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 3-(DIMETHYLAMINO)PHENOL CHEMBL225257 68570 46729 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PMID29671355-Compound-21 68571 46730 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1769 PROPOXYCAINE HYDROCHLORIDE 68574 46731 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CGP-13501 CHEMBL1256746 68578 46732 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME TAK-715 TAK-715 68580 46733 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE LENVATINIB LENVATINIB 68581 46734 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-31 68582 46735 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX VCN-01 26603261 68583 46736 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL514800 APREMILAST 68585 46737 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TRIMEPRAZINE METHYLPROMAZINE 68586 46738 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ARFORMOTEROL ARFORMOTEROL 68587 46739 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ABP 501 68588 46740 ATAD5 79915 NA CAMPTOTHECIN CAMPTOTHECIN 68589 46741 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR OXIDOPAMINE OXIDOPAMINE 68590 46742 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PENTABROMOPHENOL PENTABROMOPHENOL 68592 46743 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE HEXADECYLPHOSPHOCHOLINE MILTEFOSINE 7883777 68593 46744 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PD-98059 CHEMBL35482 10318905 68594 46745 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ENNIATIN B ENNIATIN B 68595 46746 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ERYTHROMYCIN ERYTHROMYCIN 22931300 68596 46747 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE TAMOXIFEN TAMOXIFEN 12469160,12602925 68598 46748 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor XL765 VOXTALISIB 68599 46749 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE ZINC SULFATE 14607573 68600 46750 GMNN 51053 DRUGGABLE GENOME DISULFIRAM DISULFIRAM 68601 46751 IL1B 3553 KINASE, DRUGGABLE GENOME ECHINACEA ECHINACEA, UNSPECIFIED 8951617 68604 46752 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE Trodusquemine TRODUSQUEMINE 68605 46753 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-269962A GSK-269962A 68606 46754 GMNN 51053 DRUGGABLE GENOME CIS(Z)-FLUPENTIXOL DIHYDROCHLORIDE CHEMBL1496351 68607 46755 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL223360 LINIFANIB 68608 46756 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME INDOCYANINE GREEN INDOCYANINE GREEN 68609 46757 ATAD5 79915 NA ABT-702 CHEMBL66089 68612 46758 CA9 768 DRUGGABLE GENOME, ENZYME CHEMBL2108713 IODINE I 124 GIRENTUXIMAB 68613 46759 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR LARGAZOLE LARGAZOLE 21420302,25203782,20491440 68617 46760 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME RG-1530 RG-1530 68618 46761 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100381 68619 46762 XPNPEP2 7512 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166832 68624 46763 CTSO 1519 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL481611 ODANACATIB 68625 46764 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650285 68626 46765 ABAT 18 DRUGGABLE GENOME, ENZYME VALPROIC ACID VALPROIC ACID 11086726 68630 46766 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME METHAPHIT METHAPHIT 68633 46767 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 223366121 ALISERTIB 68636 46768 SMN2 6607 DRUGGABLE GENOME CID 752709 CHEMBL429335 68638 46769 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650284 68641 46770 DGAT1 8694 ENZYME, DRUGGABLE GENOME AZD7687 AZD-7687 68642 46771 NCOA2 10499 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 68643 46772 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor MK0752 68644 46773 NOS1 4842 DRUGGABLE GENOME, ENZYME ROSIGLITAZONE ROSIGLITAZONE 15130775 68649 46774 PDE4B 5142 DRUGGABLE GENOME, ENZYME IBUDILAST IBUDILAST 68650 46775 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor SELUMETINIB SELUMETINIB 68651 46776 VKORC1 79001 DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 68652 46777 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 178103971 IBUDILAST 68653 46778 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL1683544 ERIBULIN MESYLATE 68654 46779 SMN2 6607 DRUGGABLE GENOME 2-(2-NITROBENZYLSULFANYL)BENZOXAZOLE CHEMBL112060 68655 46780 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 187051792 PANOBINOSTAT 68656 46781 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID28048944-Compound-6 68658 46782 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Practolol PRACTOLOL 68659 46783 PSMF1 9491 PROTEASE INHIBITOR inhibitor BORTEZOMIB BORTEZOMIB 68660 46784 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LINIFANIB LINIFANIB 68661 46785 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE cabozantinib CABOZANTINIB 27825638 68663 46786 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME DOXAZOSIN DOXAZOSIN 68666 46787 SMPD1 6609 ENZYME, DRUGGABLE GENOME AMIODARONE HYDROCHLORIDE AMIODARONE HYDROCHLORIDE 68667 46788 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101291 68668 46789 VKORC1 79001 DRUGGABLE GENOME, ENZYME Phenprocoumon PHENPROCOUMON 68669 46790 PTGS2 5743 DRUGGABLE GENOME, ENZYME SULINDAC SULFIDE 15657353 68670 46791 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AMSACRINE AMSACRINE 8823806,8519659,8632768 68671 46792 ATAD5 79915 NA DAIDZIN DAIDZIN 68673 46793 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ASP-3291 68674 46794 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TIBOLONE TIBOLONE 68675 46795 RORB 6096 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, KINASE antagonist 135649918 68676 46796 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-7b 68679 46797 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME CYC-116 CYC-116 68680 46798 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME GW8510 CHEMBL1276446 68681 46799 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000128325 CHEMBL602718 68682 46800 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL3137336 UPROSERTIB 68683 46801 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME 178100664 68684 46802 CBX1 10951 NA AMSACRINE AMSACRINE 68685 46803 ATAD5 79915 NA HARMAN HARMAN 68686 46804 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE warfarin WARFARIN 27581200,26257249,21923605,27740732 68687 46805 CBR1 873 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME daunorubicin DAUNORUBICIN 19204081 68688 46806 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE 3,6-DIMETHOXYFLAVONE 3,6-DIMETHOXYFLAVONE 68689 46807 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE KENPAULLONE KENPAULLONE 68690 46808 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-72a 68691 46809 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 1,7-O-DIACETYLGEOPYXIN A CHEMBL1873045 68692 46810 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL1200629 VECURONIUM BROMIDE 68694 46811 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 249565825 68695 46812 TMEM97 27346 NA PMID30185082-Compound-27 68696 46813 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE PF-562271 PF-00562271 68697 46814 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 valproic acid 16402128,15940289,16952495,19238117,18698229,16891249,9353388,10544257,15660270,11241319,15475735,18212800,20089352,16945988,11725533,19921195,15980104,6437960,19845430,10999944,20155256,16272956,17130279,12042667,21494765,10448083,20596643,12223434,12844137,19604090,15265511,15308589,21521021,16452582,19225447,11779172,12749606,18380793,14981342,17220563,3101178 68698 46815 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Paclitaxel PACLITAXEL 25104330 68699 46816 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME AMLEXANOX AMLEXANOX 68700 46817 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME ON-01135 23841031 68701 46818 IMPDH1 3614 ENZYME, DRUGGABLE GENOME AVN-944 AVN-944 68703 46819 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-20 68704 46820 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1522 ESZOPICLONE 68706 46821 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR STANOLONE STANOLONE 68707 46822 NR2F2 7026 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PYRIDABEN PYRIDABEN 68708 46823 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-WO2011127048 31 68711 46824 BAZ2B 29994 NA CAPSAZEPINE CAPSAZEPINE 68712 46825 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 363894223 68713 46826 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor 363894146 68714 46827 SMN1 6606 DRUGGABLE GENOME IPRIFLAVONE IPRIFLAVONE 68715 46828 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BBI608 68718 46829 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME IMC-CS4 IMC-CS4 68719 46830 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TAMATINIB R-406 68720 46831 IL7R 3575 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CYT 99007 68721 46832 TXNRD1 7296 DRUGGABLE GENOME Triazole gold complexe 1 68722 46833 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME BDBM50173327 68723 46834 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE ALISERTIB ALISERTIB 68724 46835 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR TAK-715 TAK-715 68726 46836 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200841 PROCAINE HYDROCHLORIDE 68727 46837 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CHLORAMBUCIL CHLORAMBUCIL 68728 46838 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR KRESOXIM-METHYL KRESOXIM-METHYL 68729 46839 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME GW441756X GW441756X 68730 46840 KDM4A 9682 DRUGGABLE GENOME, ENZYME BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 68731 46841 TUBB3 10381 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 68732 46842 HTT 3064 DRUGGABLE GENOME HOMIDIUM BROMIDE HOMIDIUM BROMIDE 68735 46843 NR1D1 9572 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME agonist 178101166 68736 46844 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME INTERLEUKIN-11 8641341 68738 46845 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HARMOL HARMOL 68739 46846 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME METHOTREXATE METHOTREXATE 23652803 68740 46847 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME ANDROSTENEDIONE ANDROSTENEDIONE 15590985 68741 46848 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR FANG vaccine 68743 46849 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CENISERTIB CENISERTIB 68744 46850 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR Clazakizumab CLAZAKIZUMAB 68747 46851 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME chlorthalidone CHLORTHALIDONE 68748 46852 GHRL 51738 DRUGGABLE GENOME RHGH 17106185 68749 46853 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY ADENOVIRUS VECTOR 15271884 68750 46854 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE RG-1530 RG-1530 68752 46855 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE EQ-917 68753 46856 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE adalimumab ADALIMUMAB 16720636,16909270,23057546,26244882,12847678,18050183,18713756,19365401,22760475,24192118,17343250,22960943,22129793,12190096,18438841 68754 46857 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ZD9331 14695155 68756 46858 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GINKGO BILOBA 17611934 68757 46859 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEFACLOR CEFACLOR 68758 46860 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Imatinib IMATINIB 68759 46861 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR THIOMERSAL THIMEROSAL 68760 46862 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER NRP104 LISDEXAMFETAMINE DIMESYLATE 68762 46863 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL PRAZEPAM PRAZEPAM 68763 46864 IGFBP1 3484 DRUGGABLE GENOME TRIIODOTHYRONINE LIOTHYRONINE SODIUM 9540232 68764 46865 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME DASATINIB DASATINIB 68765 46866 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3125 CHEMBL534288 68766 46867 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE MASITINIB MASITINIB 68769 46868 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CID 1540545 CHEMBL259784 68770 46869 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Aromatic bicyclic compound 3 68771 46870 IL1B 3553 KINASE, DRUGGABLE GENOME HYDROQUINONE HYDROQUINONE 7589278 68772 46871 ACSS3 79611 NA antidepressants 25916525 68773 46872 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor MUBRITINIB MUBRITINIB 68774 46873 GPR87 53836 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651509 68775 46874 HMGCR 3156 ENZYME, DRUGGABLE GENOME NCX-6560 68776 46875 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLOFIBRATE CLOFIBRATE 22931300 68778 46876 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200578 THEOPHYLLINE SODIUM GLYCINATE 68779 46877 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME BETA-NAPHTHOFLAVONE BETA-NAPHTHOFLAVONE 26222195,14684315 68780 46878 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178102294 BI-2536 68781 46879 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME ILORASERTIB ILORASERTIB 68783 46880 NDUFS2 4720 ENZYME inhibitor CHEMBL3545320 ME-344 68784 46881 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEPHOSTATIN DEPHOSTATIN 68785 46882 PDE4D 5144 DRUGGABLE GENOME, ENZYME HT-0712 HT-0712 68787 46883 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 22047606 68791 46884 ATAD5 79915 NA GNF-PF-1134 CHEMBL600694 68792 46885 BRCA2 675 CLINICALLY ACTIONABLE Vinorelbine VINORELBINE 26801247 68793 46886 PTGES 9536 DRUGGABLE GENOME, ENZYME inhibitor 252827470 68794 46887 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BARDOXOLONE METHYL BARDOXOLONE METHYL 26278028 68795 46888 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4945 CHEMBL585628 68796 46889 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME IRAK1/4 28065413 68797 46890 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-238165 CHEMBL2059074 22524450 68800 46891 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL559 DEXTROTHYROXINE 68801 46892 LAG3 3902 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE antibody 336446922 RELATLIMAB 68802 46893 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR Talminogene laherparepvec 68806 46894 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545368 PANOBINOSTAT LACTATE 68808 46895 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE TANDUTINIB TANDUTINIB 68809 46896 TNFRSF11B 4982 DRUGGABLE GENOME TESTOSTERONE TESTOSTERONE 11932280 68811 46897 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE CHEMBL502774 68812 46898 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-US20120277229 41(1.3) 68813 46899 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME FACTOR VIII 68814 46900 SMN1 6606 DRUGGABLE GENOME DNDI1417260 CHEMBL2094573 68815 46901 GAA 2548 DRUGGABLE GENOME, ENZYME ACARBOSE ACARBOSE 68816 46902 GMNN 51053 DRUGGABLE GENOME TANESPIMYCIN TANESPIMYCIN 68817 46903 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MERCAPTOPURINE HYDRATE MERCAPTOPURINE 68818 46904 FZD7 8324 G PROTEIN COUPLED RECEPTOR, KINASE antagonist CHEMBL2364652 VANTICTUMAB 68819 46905 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME DIHYDROGUAIARETIC ACID DIHYDROGUAIARETIC ACID 25314129 68820 46906 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR HTF 919 68821 46907 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE LACTULOSE LACTULOSE 1418064 68822 46908 ATAD5 79915 NA GNF-PF-3286 CHEMBL581880 68823 46909 EPHA3 2042 ENZYME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 363894214 SITRAVATINIB 68824 46910 BCL2L2 599 CLINICALLY ACTIONABLE, DRUGGABLE GENOME ABT-263 NAVITOCLAX 68825 46911 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DEXAMETHASONE DEXAMETHASONE 29408328 68827 46912 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-353720 CHEMBL1408276 68828 46913 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE BMS-690514 BMS-690514 21531814 68829 46914 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ANTIESTROGEN 15056732 68831 46915 ARID5B 84159 CLINICALLY ACTIONABLE methotrexate METHOTREXATE 24712521 68833 46916 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME 681640 CHEMBL379975 68834 46917 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545361 ROGARATINIB 68837 46918 MAPT 4137 DRUGGABLE GENOME TCMDC-124224 CHEMBL580421 68838 46919 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE XR-5000 68839 46920 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ESTRADIOL ESTRADIOL 68840 46921 CYB5R3 1727 DRUGGABLE GENOME, ENZYME articaine / epinephrine 68841 46922 GMNN 51053 DRUGGABLE GENOME METOCHALCONE METOCHALCONE 68842 46923 ALDH1A1 216 DRUGGABLE GENOME, ENZYME AG-126 CHEMBL77387 68843 46924 CYP24A1 1591 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME inhibitor 252827476 68845 46925 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651430 68846 46926 ABAT 18 DRUGGABLE GENOME, ENZYME VALPROIC ACID 68847 46927 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR SELUMETINIB SELUMETINIB 26324360,19915144,23444215 68849 46928 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE NICOTINE NICOTINE 18784291 68850 46929 HTT 3064 DRUGGABLE GENOME GNF-PF-2357 CHEMBL578257 68855 46930 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SULFAPHENAZOLE SULFAPHENAZOLE 22931300 68856 46931 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME GNF-PF-1919 CHEMBL576409 68857 46932 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR GNF-PF-2812 CHEMBL125044 68858 46933 SPG7 6687 PROTEASE, ENZYME thalidomide THALIDOMIDE 20038957 68859 46934 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 VESNARINONE VESNARINONE 9630823 68860 46935 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CLOCORTOLONE PIVALATE CLOCORTOLONE PIVALATE 68862 46936 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DICUMAROL DICUMAROL 68863 46937 SLC31A1 1317 TRANSPORTER carboplatin CARBOPLATIN 22725681 68865 46938 MAP2K6 5608 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE, TUMOR SUPPRESSOR inhibitor AZD6244 SELUMETINIB 68866 46939 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178103584 68867 46940 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Rapamycin SIROLIMUS 68868 46941 RPL13 6137 NA thalidomide THALIDOMIDE 20038957 68870 46942 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178103764 FLUVOXAMINE 68873 46943 PROS1 5627 DRUGGABLE GENOME lusutrombopag LUSUTROMBOPAG 68877 46944 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-125185 CHEMBL580819 68879 46945 USP1 7398 DNA REPAIR, PROTEASE, ENZYME FLUPENTIXOL FLUPENTIXOL 68880 46946 CLK1 1195 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE LEUCETTAMINE B LEUCETTAMINE B 22998443 68881 46947 MAPT 4137 DRUGGABLE GENOME TCMDC-123916 CHEMBL493863 68882 46948 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MONTELUKAST MONTELUKAST 22931300 68883 46949 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CLORAZEPATE CLORAZEPIC ACID 68884 46950 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RETINOIC ACID 11437362,8639801,8947586 68885 46951 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 178103145 68886 46952 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-1692 CHEMBL582055 68887 46953 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR inhibitor 178101495 GEMCITABINE 68888 46954 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NALBUPHINE NALBUPHINE 68893 46955 ATAD5 79915 NA METHOXYVONE METHOXYVONE 68894 46956 GMNN 51053 DRUGGABLE GENOME IMIQUIMOD IMIQUIMOD 68897 46957 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE allosteric modulator 249565628 MK-2206 68898 46958 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME blocker 178101111 68899 46959 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE ROBUSTIC ACID ROBUSTIC ACID 68900 46960 TARDBP 23435 TUMOR SUPPRESSOR GIPARMEN GIPARMEN 68901 46961 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE Alectinib ALECTINIB 27009859,25749034,25421750 68902 46962 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Ribociclib RIBOCICLIB 27542767,28151717,24795392 68904 46963 TDP2 51567 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME (-)-DICENTRINE CHEMBL478754 68905 46964 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PLATELET-DERIVED GROWTH FACTOR (PDGF) 68907 46965 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ALLOXAN ALLOXAN 68908 46966 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME SOY PROTEIN 12221209 68909 46967 CBX1 10951 NA TRANSTORINE TRANSTORINE 68910 46968 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE THIOGUANINE THIOGUANINE 68911 46969 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrido[3,2-d]pyrimidine derivative 3 68912 46970 TMEM97 27346 NA agonist 178103293 CHEMBL53325 68913 46971 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME TAE-684 TAE-684 68914 46972 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE OSI-632 OSI-632 68915 46973 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TETRAIDOFLUORESCEIN TETRAIDOFLUORESCEIN 68916 46974 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME AME-133v AME-133V 68917 46975 POLK 51426 DNA REPAIR, ENZYME ALPHA,BETA-DEHYDROCURVULARIN CHEMBL482050 68918 46976 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CAPIVASERTIB CAPIVASERTIB 24088382,22294718,28489509 68919 46977 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL49642 INDIBULIN 68920 46978 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 178102432 68921 46979 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE RAPAMYCIN SIROLIMUS 14605212 68922 46980 POLB 5423 DNA REPAIR, DRUGGABLE GENOME N-PHENETHYLCINNAMAMIDE CHEMBL1305393 68923 46981 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135650241 68924 46982 BAZ2B 29994 NA GNF-PF-3464 CHEMBL602213 68926 46983 SMN1 6606 DRUGGABLE GENOME 2-PYRIDYLKETONE BENZOYL HYDRAZONE CHEMBL252151 68927 46984 SRD5A1 6715 DRUGGABLE GENOME DUTASTERIDE DUTASTERIDE 68929 46985 COL5A3 50509 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 68931 46986 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1213490 ROMIDEPSIN 68934 46987 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ERYTHROSINE ERYTHROSINE 68937 46988 SMN2 6607 DRUGGABLE GENOME DNDI1416969 CHEMBL1453126 68940 46989 ATRX 546 ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR VINCRISTINE VINCRISTINE 23904111 68942 46990 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME VEGF GENE THERAPY 68943 46991 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR PLATINUM COMPOUND 15217961 68944 46992 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FLUPIRTINE FLUPIRTINE 68946 46993 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME CPC-212 68947 46994 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE NAPHTHALENE-1,2-DIOL CHEMBL204543 24997687 68948 46995 ALOX15 246 ENZYME, DRUGGABLE GENOME WAY-100135 CHEMBL38288 68949 46996 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652268 68951 46997 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Flavonoid derivative 2 68952 46998 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Valbenazine VALBENAZINE 68955 46999 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME Anti-Mesothelin CAR-T cells 68956 47000 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor 249565590 CHEMBL1236539 68957 47001 SMN2 6607 DRUGGABLE GENOME METHOXYVONE METHOXYVONE 68958 47002 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TOTAL PARENTERAL NUTRITION 14744944 68959 47003 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545245 BAY-1082439 68960 47004 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1200412 NANDROLONE PHENPROPIONATE 68961 47005 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545385 WX-037 68962 47006 SLC1A7 6512 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101349 68963 47007 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SYN004 68964 47008 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-69187 CHEMBL19954 68966 47009 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT 68967 47010 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORFENAPYR CHLORFENAPYR 68968 47011 TUBB4B 10383 DRUGGABLE GENOME 4-(PHENYLCARBAMOYL)BENZYLNITRATE CHEMBL1795737 21664138 68969 47012 GMNN 51053 DRUGGABLE GENOME GNF-PF-1509 CHEMBL576412 68970 47013 POLI 11201 DNA REPAIR 3,8'-BIAPIGENIN CHEMBL515252 68971 47014 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TEBUCONAZOLE TEBUCONAZOLE 68973 47015 ATAD5 79915 NA GNF-PF-4814 CHEMBL585443 68974 47016 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Six-membered heterocyclic benzamide derivative 4 68975 47017 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME inhibitor 249565742 68977 47018 POLI 11201 DNA REPAIR INAMRINONE INAMRINONE 68978 47019 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A10 68979 47020 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652641 68980 47021 PTGS2 5743 DRUGGABLE GENOME, ENZYME FK-3311 68982 47022 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CD20 CAR T cells 68983 47023 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 5,7-DICHLOROKYNURENIC ACID CHEMBL50267 68984 47024 PDE4A 5141 DRUGGABLE GENOME, ENZYME Dyphylline DYPHYLLINE 68986 47025 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR LY2606368 MsOH H2O 68988 47026 RACGAP1 29127 NA TCMDC-123723 CHEMBL525103 68989 47027 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-738482 CHEMBL103098 68992 47028 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMIDATE AMIDATE 68995 47029 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR HISTAMINE HISTAMINE 19053770,20192225 68996 47030 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor APRICOXIB APRICOXIB 68997 47031 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 EBSELEN EBSELEN 68998 47032 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME QUERCETIN QUERCETIN 8759170,7769390 69000 47033 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME ALDICARB ALDICARB 69001 47034 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE GNF-PF-3542 CHEMBL598477 69004 47035 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE ARGATROBAN ARGATROBAN 10611442 69005 47036 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 5,4'-DIHYDROXYFLAVONE CHEMBL484662 69010 47037 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE TCMDC-125575 CHEMBL587620 69011 47038 IFNG 3458 DRUGGABLE GENOME AMIKACIN AMIKACIN 8913387 69012 47039 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GBR-12935 CHEMBL26320 69013 47040 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 310264724 LY-3009120 69014 47041 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 252166636 TAK-954 69016 47042 HDAC11 79885 DRUGGABLE GENOME, ENZYME inhibitor SB939 69017 47043 GAPDH 2597 DRUGGABLE GENOME, ENZYME DEFEROXAMINE DEFEROXAMINE 9486123 69019 47044 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME HALOPERIDOL HALOPERIDOL 12873733 69020 47045 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-20 69021 47046 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME SAFINAMIDE SAFINAMIDE 69022 47047 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ASKP-1240 BLESELUMAB 69023 47048 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE MN-221 BEDORADRINE SULFATE 69025 47049 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 681640 CHEMBL379975 69026 47050 TENT4A 11044 NA gemcitabine GEMCITABINE 22838950 69028 47051 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME METIXENE METHIXENE 69029 47052 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000012773 CHEMBL589715 69030 47053 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BVD-523 ULIXERTINIB 26725216 69031 47054 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PANOBINOSTAT PANOBINOSTAT 69032 47055 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PORFIROMYCIN PORFIROMYCIN 69034 47056 COL4A5 1287 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 69035 47057 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ORLISTAT ORLISTAT 69036 47058 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200538 BETAMETHASONE ACETATE 69038 47059 MAPT 4137 DRUGGABLE GENOME DNDI1417941 CHEMBL2095095 69039 47060 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER POTASSIUM DICHROMATE POTASSIUM DICHROMATE 69043 47061 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR IP-10 11980656 69045 47062 RGS4 5999 DRUGGABLE GENOME QUINACRINE QUINACRINE 69046 47063 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GR-127935 GR-127935 69047 47064 ANO1 55107 ION CHANNEL blocker 178101131 69048 47065 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 69049 47066 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CHEMBL1341 METHOXYFLURANE 69053 47067 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor AZD4547 69054 47068 TGFB3 7043 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR inhibitor CHEMBL1743022 FRESOLIMUMAB 69056 47069 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL3039565 69057 47070 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Pyrrolidine carboxamide derivative 2 69058 47071 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Cisplatin CISPLATIN 23536011 69059 47072 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME PROSTAGLANDIN B1 PROSTAGLANDIN B1 69060 47073 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE CHEMBL2103870 LUMACAFTOR 69061 47074 SMN2 6607 DRUGGABLE GENOME LASSBIO-294 CHEMBL233194 69062 47075 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1068 OXCARBAZEPINE 69063 47076 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-P6 69064 47077 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW775608X GW775608X 69066 47078 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR CYCLOSPORIN A 9933022 69067 47079 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR NORGESTREL NORGESTREL 69068 47080 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651446 ADENOSINE TRIPHOSPHATE 69069 47081 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor SUNITINIB SUNITINIB 69071 47082 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR antagonist 135650370 FULVESTRANT 69073 47083 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DICHLOROPHEN DICHLOROPHEN 69074 47084 POLI 11201 DNA REPAIR TCMDC-123723 CHEMBL525103 69076 47085 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Isothiocyanate derivative 1 69077 47086 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR EMODIN EMODIN 11887862 69078 47087 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Rigosertib RIGOSERTIB 26091808 69079 47088 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE PMID26882240-Compound-3 69080 47089 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor OLAPARIB OLAPARIB 69081 47090 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME GENISTEIN GENISTEIN 17375591 69082 47091 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PENTABROMOPHENOL PENTABROMOPHENOL 69085 47092 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor AT9283 AT-9283 69086 47093 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME carvedilol CARVEDILOL 20643254,16849011 69087 47094 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ROTENONE ROTENONE 16680159 69089 47095 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PF-562271 PF-00562271 69091 47096 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PALMITOYL-DL-CARNITINE CHLORIDE CHEMBL1256761 69092 47097 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-43 69094 47098 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE TAMATINIB R-406 69095 47099 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Afatinib AFATINIB 25870145 69099 47100 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE TPA ALTEPLASE 11679632 69101 47101 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME SODIUM BUTYRATE 2887561 69103 47102 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 Cobicistat/darunavir 69105 47103 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-94 69108 47104 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor PIVANEX AN-9 69109 47105 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR A-443654 A-443654 69110 47106 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PSAMMAPLIN A PSAMMAPLIN A 25884112 69111 47107 THBD 7056 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CURCUMIN CURCUMIN 15733976 69112 47108 ARSA 410 DRUGGABLE GENOME, ENZYME TOSYL-L-LYSINE CHLOROMETHYL KETONE CHEMBL466465 69113 47109 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DESOXYCORTICOSTERONE PIVALATE 69114 47110 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE Vantictumab VANTICTUMAB 22753465 69115 47111 MARK4 57787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 69116 47112 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-60 69119 47113 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650350 HIMBACINE 69121 47114 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-2301 CHEMBL578061 69122 47115 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor GDC-0068 IPATASERTIB 69123 47116 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME NSC-107022 CHEMBL1601846 69124 47117 POLI 11201 DNA REPAIR CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 69127 47118 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor AT13387 ONALESPIB 69128 47119 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER LOPERAMIDE LOPERAMIDE 69129 47120 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Afuresertib AFURESERTIB 24978597 69133 47121 SMN1 6606 DRUGGABLE GENOME 4'-METHOXYFLAVONE 4'-METHOXYFLAVONE 69137 47122 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-33 69138 47123 CCL25 6370 HORMONE ACTIVITY, DRUGGABLE GENOME TNF-ALPHA 15492285 69139 47124 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE GPI-1485 GPI-1485 69141 47125 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE BUPIVACAINE BUPIVACAINE 17294200 69142 47126 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME CYC-116 CYC-116 69143 47127 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME PMID22911925C2 69145 47128 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166829 69146 47129 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR DIETHYLSTILBESTROL DIETHYLSTILBESTROL 69147 47130 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor GSK2636771 GSK-2636771 69148 47131 TARDBP 23435 TUMOR SUPPRESSOR TESTOSTERONE PROPIONATE TESTOSTERONE PROPIONATE 69149 47132 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME clozapine CLOZAPINE 20452607 69150 47133 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-46 69151 47134 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE BMS-708163 AVAGACESTAT 69152 47135 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME TAK-715 TAK-715 69153 47136 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BROMOXYNIL BROMOXYNIL 69154 47137 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Norethindrone NORETHINDRONE 69155 47138 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-124381 CHEMBL579919 69157 47139 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE AMITRIPTYLINE AMITRIPTYLINE 16283318 69158 47140 FGG 2266 DRUGGABLE GENOME, FIBRINOGEN, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE RECOMBINANT FACTOR IX FC FUSION PROTEIN 69159 47141 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME LOMETREXOL LOMETREXOL 21879757 69160 47142 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE HYDROXYUREA HYDROXYUREA 7923130 69161 47143 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME BAY-613606 CHEMBL541400 69162 47144 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 178103556 69163 47145 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 178103821 NEFAZODONE 69164 47146 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME inhibitor 178102546 ALOISINE 69165 47147 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 249565590 CHEMBL1236539 69166 47148 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE HYDROCORTISONE 21-OCTANOATE CHEMBL253989 69167 47149 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TYRPHOSTIN A9 TYRPHOSTIN A9 69168 47150 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL235191 TACEDINALINE 69170 47151 EPHA7 2045 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 249565850 69173 47152 TARDBP 23435 TUMOR SUPPRESSOR DIFENPIRAMIDE DIFENPIRAMIDE 69174 47153 AKR1C3 8644 ENZYME, DRUGGABLE GENOME 3-((4-NITROPHENYL)AMINO)BENZOIC ACID CHEMBL1682200 22263837 69177 47154 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR MOMETASONE MOMETASONE 69179 47155 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 381118856 69180 47156 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ZM-39923 HCL CHEMBL538798 69183 47157 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200802 TALBUTAL 69187 47158 TOP2B 7155 DRUGGABLE GENOME, ENZYME Iboctadekin + Doxil 69189 47159 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3137309 VENETOCLAX 69193 47160 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLUDARABINE FLUDARABINE 69195 47161 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PROPYLPYRAZOLETRIOL PROPYLPYRAZOLETRIOL 69196 47162 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE ACACETIN ACACETIN 21482471 69197 47163 DNER 92737 NA Tetra-hydro-quinoline derivative 2 69198 47164 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR 8-GERANYLOXY PSORALEN CHEMBL1412710 69199 47165 ATXN2 6311 NA DNDI1417614 CHEMBL1567571 69200 47166 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME LAUROGUADINE LAUROGUADINE 69201 47167 FAAH 2166 ENZYME, DRUGGABLE GENOME Boronic acid derivative 3 69203 47168 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Vemurafenib VEMURAFENIB 69206 47169 CPB1 1360 DRUGGABLE GENOME, PROTEASE, ENZYME US8710232, 1 69207 47170 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEPHALOTHIN CEPHALOTHIN 69208 47171 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHENELZINE SULFATE PHENELZINE SULFATE 69209 47172 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE 2-PHENYLQUINOLINE 2-PHENYLQUINOLINE 69210 47173 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Liposomal encapsulated paclitaxel (LEP) 69211 47174 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR CATECHOL CATECHOL 69215 47175 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE TRASTUZUMAB TRASTUZUMAB 25953157 69216 47176 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Ethopropazine ETHOPROPAZINE 69217 47177 TDO2 6999 ENZYME, DRUGGABLE GENOME HORMONES 60273 69219 47178 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CLOMIPRAMINE CLOMIPRAMINE 69220 47179 HTT 3064 DRUGGABLE GENOME LESTAURTINIB LESTAURTINIB 69221 47180 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE NINTEDANIB NINTEDANIB 69223 47181 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125738 CHEMBL527585 69225 47182 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor GDC-0623 RG-7420 69226 47183 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX CHRYSOERIOL CHRYSOERIOL 25190466 69227 47184 ALDH1A1 216 DRUGGABLE GENOME, ENZYME QUERCETIN QUERCETIN 69228 47185 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DILAZEP DILAZEP 69229 47186 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CORTISOL HYDROCORTISONE 16873536 69230 47187 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING AZELASTINE HYDROCHLORIDE AZELASTINE HYDROCHLORIDE 69231 47188 TSPO 706 DRUGGABLE GENOME Flunitrazepam FLUNITRAZEPAM 69232 47189 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE EO9 APAZIQUONE 8509220 69234 47190 CYB5R3 1727 DRUGGABLE GENOME, ENZYME isosorbide dinitrate 69235 47191 HSPB2 3316 KINASE PROPRANOLOL PROPRANOLOL 11368160 69236 47192 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MICONAZOLE NITRATE MICONAZOLE NITRATE 69237 47193 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545074 LEO-15520 69238 47194 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME SNS-032 BMS-387032 69240 47195 FKBP5 2289 DRUGGABLE GENOME Selective serotonin reuptake inhibitors 20709156,15565110 69241 47196 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GW441756X GW441756X 69242 47197 ATAD5 79915 NA S-(2,4-DICHLOROBENZYL)ISOTHIOUREA HYDROBROMIDE CHEMBL1224483 69243 47198 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE CHRYSIN DIMETHYL ETHER CHRYSIN DIMETHYL ETHER 69244 47199 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Indazole derivative 4 69246 47200 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-200646 CHEMBL85194 69247 47201 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor DASATINIB DASATINIB 69249 47202 GHRL 51738 DRUGGABLE GENOME TPN 18197141 69250 47203 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME RETINOIC ACID 15316139 69251 47204 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL3544935 XL-418 69254 47205 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ROBUSTIC ACID ROBUSTIC ACID 69256 47206 GBA 2629 DRUGGABLE GENOME, ENZYME GENTIAN VIOLET GENTIAN VIOLET 69257 47207 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102665 69258 47208 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PMID27774824-Compound-Figure7Example10 69259 47209 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE BI-847325 69260 47210 MAOA 4128 DRUGGABLE GENOME, ENZYME KadcoccitoneA 69265 47211 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE phenytoin PHENYTOIN 26049587 69266 47212 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME flibanserin FLIBANSERIN 69267 47213 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565691 CHEMBL1086377 69268 47214 CBX1 10951 NA GUANIDINONALTRINDOLE GUANIDINONALTRINDOLE 69269 47215 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EMODIN EMODIN 69271 47216 ATAD5 79915 NA GNF-PF-2657 CHEMBL578944 69272 47217 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE LESTAURTINIB LESTAURTINIB 69273 47218 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE MYRICETIN MYRICETIN 69275 47219 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME ACID BLUE 129 ACID BLUE 129 69277 47220 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME ITF2357 GIVINOSTAT 69278 47221 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX LASALOCID A SODIUM LASALOCID A SODIUM 69279 47222 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor 315661116 69280 47223 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE CHEMBL1255944 69281 47224 RBX1 9978 DNA REPAIR, ENZYME inhibitor CHEMBL43452 POMALIDOMIDE 69282 47225 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ATM AVI 69283 47226 SFTPA1 653509 DRUGGABLE GENOME BCG BCG VACCINE 10926544 69284 47227 TUBB 203068 DRUGGABLE GENOME STA-5312 ROSABULIN 69285 47228 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE AEW-541 AEW-541 69287 47229 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BYL719 ALPELISIB 69289 47230 ST14 6768 ENZYME, DRUGGABLE GENOME, PROTEASE US8569313, Inhibitor 15 69293 47231 CXCL8 3576 DRUGGABLE GENOME inhibitor CHEMBL2109617 HUMAX-IL8 69294 47232 MAP3K1 4214 CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME CI-1040 CI-1040 69295 47233 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE GOLIMUMAB GOLIMUMAB 69296 47234 KDM4A 9682 DRUGGABLE GENOME, ENZYME MALEIC ACID MALEIC ACID 69299 47235 TPSAB1 7177 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178101079 NAFAMOSTAT 69300 47236 PTGS1 5742 ENZYME, DRUGGABLE GENOME Meclofenamate Sodium 69302 47237 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 381744915 69304 47238 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 178102655 69305 47239 ALDH1A2 8854 DRUGGABLE GENOME, ENZYME Bisphosphonates 69306 47240 GJB5 2709 ION CHANNEL inhibitor 135650269 69307 47241 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME THIRAM THIRAM 69308 47242 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME LGX818 ENCORAFENIB 27312529 69309 47243 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 310264721 69310 47244 GUCY2C 2984 DRUGGABLE GENOME, KINASE agonist 315661154 PLECANATIDE 69311 47245 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NSC-95397 CHEMBL429095 69314 47246 SMN1 6606 DRUGGABLE GENOME LMI070 BRANAPLAM 69317 47247 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE JNJ-61186372 JNJ-61186372 27216193 69318 47248 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR VER-49009 CHEMBL365617 69319 47249 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR EBSELEN EBSELEN 69320 47250 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CENISERTIB CENISERTIB 69321 47251 NOS1 4842 DRUGGABLE GENOME, ENZYME BSO 10850366 69322 47252 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NITROFEN NITROFEN 69323 47253 ATXN2 6311 NA NSC-695801 CHEMBL461193 69326 47254 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Aminocyclopentenone compound 2 69327 47255 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 328083500 CHEMBL592893 69328 47256 SMN2 6607 DRUGGABLE GENOME GNF-PF-3037 CHEMBL600336 69329 47257 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3545222 AZD8683 69331 47258 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ERGONOVINE ERGONOVINE 69332 47259 PKN1 5585 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE INGENOL MEBUTATE 69333 47260 PTPN13 5783 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE, CLINICALLY ACTIONABLE ANTIESTROGENS 15242314 69334 47261 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER BUTHIONINE SULFOXIMINE 11189941 69335 47262 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TYRPHOSTIN 25 TYRPHOSTIN 25 69336 47263 CDK14 5218 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME inhibitor CHEMBL1230607 PHA-793887 69337 47264 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE PARAROSANILINE PARAROSANILINE 69339 47265 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PROTRIPTYLINE PROTRIPTYLINE 69340 47266 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE NEOMYCIN NEOMYCIN 15024008 69341 47267 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist CHEMBL3545393 XL550 69342 47268 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1823817 CE-224535 69343 47269 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME N-(pyridin-2-yl)pyrimidin-4-amine derivative 1 69344 47270 SLC12A2 6558 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178101541 FUROSEMIDE 69347 47271 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CYTOKINES 17097057 69349 47272 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE GSK2696273 69350 47273 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL3544962 CT-1578 69351 47274 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME GW441756X GW441756X 69352 47275 KDM4A 9682 DRUGGABLE GENOME, ENZYME SENNOSIDE B SENNOSIDE B 69353 47276 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME MIVACURIUM MIVACURIUM 69355 47277 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME UFT 11729480 69356 47278 KDM4A 9682 DRUGGABLE GENOME, ENZYME CHLORPROMAZINE HYDROCHLORIDE CHLORPROMAZINE HYDROCHLORIDE 69357 47279 CLK1 1195 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE NU-2058 CHEMBL269881 69358 47280 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ribociclib RIBOCICLIB 69359 47281 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE RISEDRONIC ACID RISEDRONIC ACID 25630225,26314394 69360 47282 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200597 ETIDOCAINE HYDROCHLORIDE 69361 47283 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME MEMANTINE MEMANTINE 69362 47284 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE CURCUMIN CURCUMIN 25753330 69364 47285 IL1A 3552 CELL SURFACE, DRUGGABLE GENOME MABp1 MABP1 69365 47286 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103829 FAXELADOL 69366 47287 GATA4 2626 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE warfarin WARFARIN 25026456,29298995 69368 47288 ATXN2 6311 NA ALPHA,BETA-DEHYDROCURVULARIN CHEMBL482050 69369 47289 PXN 5829 NA LOVASTATIN LOVASTATIN 11581207 69372 47290 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Dexamethasone DEXAMETHASONE 69373 47291 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME activator 336446901 69375 47292 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Floxuridine FLOXURIDINE 25714871 69377 47293 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER METHYLENE BLUE CHLORIDE HYDRATE METHYLENE BLUE 69379 47294 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Anti-BCMA CAR-T cells 69380 47295 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 328083482 69381 47296 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME CHLORPROMAZINE CHLORPROMAZINE 18834354 69382 47297 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL919 FOSPHENYTOIN SODIUM 69384 47298 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER zidovudine ZIDOVUDINE 23996099 69385 47299 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME DIAZEPAM DIAZEPAM 69386 47300 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL701 BACLOFEN 69388 47301 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE DITHIOLETHIONE DITHIOLETHIONE 20655236 69389 47302 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-2947 CHEMBL581677 69390 47303 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-26 69393 47304 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1201132 NALBUPHINE HYDROCHLORIDE 69394 47305 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL488436 AZD-5438 69395 47306 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3906 CHEMBL599102 69396 47307 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor XL765 VOXTALISIB 69397 47308 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1201607 NATALIZUMAB 69398 47309 DSG1 1828 NA PD-98059 CHEMBL35482 11781826 69399 47310 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL1096380 PLINABULIN 69400 47311 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DICHLORODIPHENYLDICHLOROETHYLENE DICHLORODIPHENYLDICHLOROETHYLENE 69401 47312 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651299 CHEMBL472273 69402 47313 PARP3 10039 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR 3-phenyl isoquinolin-1(2H) derivative 1 69403 47314 ATAD5 79915 NA GNF-PF-5297 CHEMBL602575 69404 47315 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME cisplatin CISPLATIN 24090479 69405 47316 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 135650231 69406 47317 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GDC-0973 COBIMETINIB 69407 47318 PDE4B 5142 DRUGGABLE GENOME, ENZYME RESVERATROL RESVERATROL 69408 47319 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650226 ETHYLKETOCYCLAZOCINE 69409 47320 ATAD5 79915 NA NICARDIPINE NICARDIPINE 69410 47321 ACP1 52 ENZYME, DRUGGABLE GENOME, PROTEIN PHOSPHATASE GNF-PF-992 CHEMBL602561 69412 47322 ATP5F1D 513 TRANSPORTER SEVOFLURANE SEVOFLURANE 69413 47323 SGCA 6442 NA rAAV1.tMCK.human-alpha-sarcoglycan 69414 47324 NPR3 4883 DRUGGABLE GENOME antagonist 178101732 69415 47325 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 252166487 NIRAPARIB 69416 47326 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Pyrimidine derivative 3 69417 47327 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Imidazopyridazine derivative 2 69418 47328 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR MESTRANOL MESTRANOL 69419 47329 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER BIIB054 CINPANEMAB 69422 47330 COMT 1312 DRUGGABLE GENOME, ENZYME sertraline SERTRALINE 69423 47331 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CGP-55845 CHEMBL455185 69425 47332 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYDROCORTISONE SODIUM SUCCINATE HYDROCORTISONE SODIUM SUCCINATE 69426 47333 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1200514 DEMECARIUM BROMIDE 69427 47334 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME AM-101 ESKETAMINE HYDROCHLORIDE 69429 47335 MAPT 4137 DRUGGABLE GENOME CID 4101591 CHEMBL428789 69430 47336 LGR5 8549 G PROTEIN COUPLED RECEPTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 178100589 69431 47337 RFK 55312 KINASE, ENZYME escitalopram ESCITALOPRAM 69433 47338 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102732 69434 47339 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-95397 CHEMBL429095 69435 47340 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CEPHRADINE CEPHRADINE 22166395 69436 47341 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PROPARGITE PROPARGITE 69437 47342 ERAP2 64167 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE SCOPOLETIN SCOPOLETIN 69438 47343 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE BKM120 BUPARLISIB 28416483 69439 47344 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ETHER ETHER 18427905 69440 47345 CBX1 10951 NA MITOXANTRONE MITOXANTRONE 69441 47346 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor AMG900 AMG-900 69444 47347 ERG 2078 DRUGGABLE GENOME, CLINICALLY ACTIONABLE blocker CHEMBL113461 TEDISAMIL 69447 47348 MTTP 4547 DRUGGABLE GENOME Implitapide IMPLITAPIDE 69449 47349 HTT 3064 DRUGGABLE GENOME RESVERATROL RESVERATROL 69450 47350 TGFBR3 7049 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME TG-C 69451 47351 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME PROTRIPTYLINE PROTRIPTYLINE 69453 47352 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 354702290 ELENBECESTAT 69454 47353 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR 3-(2-AZIDOETHYL)THIOPHENE CHEMBL589270 24675380 69456 47354 NOS2 4843 DRUGGABLE GENOME, ENZYME PROPOFOL PROPOFOL 16645450 69458 47355 ALOX15 246 ENZYME, DRUGGABLE GENOME SIBUTRAMINE HYDROCHLORIDE SIBUTRAMINE HYDROCHLORIDE 69460 47356 HSPB1 3315 DRUGGABLE GENOME HYDRASTININE HYDROCHLORIDE HYDRASTININE HYDROCHLORIDE 69463 47357 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE NERATINIB NERATINIB 69464 47358 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 135651381 69466 47359 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL3545092 CR 1447 69467 47360 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 135650300 GENISTEIN 69468 47361 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL408513 BELINOSTAT 69469 47362 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE GW632580X GW632580X 69470 47363 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE modulator CHEMBL3545237 HE3235 69471 47364 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CD40L 12237284,16213477,10520003 69472 47365 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR BETAMETHASONE BETAMETHASONE 69474 47366 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEXAMETHASONE SODIUM PHOSPHATE DEXAMETHASONE SODIUM PHOSPHATE 69476 47367 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8921389, 210 69477 47368 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-34c 69478 47369 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOLONIUM CHLORIDE TOLONIUM CHLORIDE 69479 47370 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CRUFOMATE CRUFOMATE 69480 47371 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor XL-765 VOXTALISIB 69484 47372 ALOX5 240 DRUGGABLE GENOME, ENZYME ACACETIN ACACETIN 24368208 69487 47373 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 384403638 69488 47374 GMNN 51053 DRUGGABLE GENOME GNF-PF-4283 CHEMBL606166 69489 47375 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650684 NALOXONE 69490 47376 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE GNF-PF-5134 CHEMBL602969 69491 47377 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651329 69492 47378 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE fenofibrate FENOFIBRATE 18695978 69493 47379 TAC1 6863 DRUGGABLE GENOME EQUINE GONADOTROPIN 14706561 69497 47380 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME inhibitor 178101837 BATIMASTAT 69498 47381 SAA1 6288 DRUGGABLE GENOME NAPROXEN NAPROXEN 1729367 69499 47382 BACE2 25825 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 223366183 69500 47383 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE PHENFORMIN PHENFORMIN 69501 47384 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE Indole-based analog 2 69502 47385 BAZ2B 29994 NA PENTABROMOPHENOL PENTABROMOPHENOL 69503 47386 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-4057 CHEMBL598903 69504 47387 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PRILOCAINE HYDROCHLORIDE PRILOCAINE HYDROCHLORIDE 69505 47388 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NSC-95397 CHEMBL429095 69506 47389 DDX43 55510 DRUG RESISTANCE SELUMETINIB SELUMETINIB 24899684 69507 47390 ALPL 249 ENZYME, DRUGGABLE GENOME MYRICETIN MYRICETIN 69508 47391 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 375973236 69509 47392 PGF 5228 GROWTH FACTOR, DRUGGABLE GENOME R7334 69511 47393 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE N-{4 69512 47394 PTPRZ1 5803 PROTEIN PHOSPHATASE, DRUGGABLE GENOME VITAMIN D 10809755 69513 47395 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL523299 UMECLIDINIUM BROMIDE 69514 47396 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor CUDC-101 CUDC-101 69515 47397 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE antibody 252166886 MARGETUXIMAB 69516 47398 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ACYCLOVIR ACYCLOVIR 69517 47399 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ILORASERTIB ILORASERTIB 69518 47400 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ESBA105 69519 47401 GRK2 156 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, G PROTEIN COUPLED RECEPTOR, ENZYME BDBM50173306 69520 47402 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Golimumab GOLIMUMAB 69521 47403 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLUFENACET FLUFENACET 69522 47404 POLI 11201 DNA REPAIR GOSSYPOL GOSSYPOL 69523 47405 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL ESTAZOLAM ESTAZOLAM 69524 47406 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Pyrimidopyridazinone derivative 2 69525 47407 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CANRENONE CANRENONE 69528 47408 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor CHEMBL3544961 BI-853520 69529 47409 C3 718 PROTEASE INHIBITOR, DRUGGABLE GENOME, CELL SURFACE COMPSTATIN COMPSTATIN 25494040 69531 47410 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE Tumor necrosis factor alpha (TNF-alpha) inhibitors 20309874,23007924 69532 47411 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33f 69533 47412 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3545096 BGT-226 69534 47413 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE RETINYL ACETATE 16716627 69535 47414 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4085 CHEMBL528181 69536 47415 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER S-166659 CHEMBL252417 69537 47416 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME INCB54828 69538 47417 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE levodopa LEVODOPA 12083967 69540 47418 TSPYL2 64061 NA TGFBETA1 15823505 69542 47419 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-2121 CHEMBL577365 69544 47420 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TRICHOSTATIN TRICHOSTATIN 69547 47421 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Trametinib TRAMETINIB 69548 47422 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TYRPHOSTIN 51 TYRPHOSTIN 51 69550 47423 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135650702 69552 47424 TH 7054 ENZYME, DRUGGABLE GENOME MIBG IOBENGUANE 7576974 69554 47425 CMKLR1 1240 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651892 69556 47426 PSMA5 5686 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL2103884 OPROZOMIB 69558 47427 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TCMDC-124224 CHEMBL580421 69559 47428 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 178103564 69561 47429 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PIPERILATE ETHOBROMIDE PIPERILATE ETHOBROMIDE 69564 47430 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR LARGAZOLE LARGAZOLE 21420302,25203782,20491440 69566 47431 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CNQX DISODIUM CHEMBL1255647 69567 47432 PML 5371 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ARSENIC TRIOXIDE 26537301,11704842 69568 47433 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR FENRETINIDE FENRETINIDE 69569 47434 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TYRPHOSTIN A9 TYRPHOSTIN A9 69570 47435 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Methotrexate METHOTREXATE 69571 47436 POLK 51426 DNA REPAIR, ENZYME ISOTHYMONIN ISOTHYMONIN 69572 47437 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2'-HYDROXYCHALCONE 2'-HYDROXYCHALCONE 69573 47438 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CHLORFENAPYR CHLORFENAPYR 69574 47439 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL1980297 ILORASERTIB 69575 47440 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor 178101910 MILRINONE 69576 47441 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE ZM-447439 CHEMBL202721 69577 47442 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135652066 69578 47443 HEBP1 50865 DRUGGABLE GENOME 4-(2-cyclohexylethoxy) aniline derivative 3 69579 47444 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GW1929 CHEMBL434063 16680159 69580 47445 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 69581 47446 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SALT VOLANESORSEN SODIUM 10775071 69583 47447 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER METHYLPREDNISOLONE METHYLPREDNISOLONE 16684279 69586 47448 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 249565839 69587 47449 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROMETHAZINE HYDROCHLORIDE PROMETHAZINE HYDROCHLORIDE 69588 47450 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650859 69589 47451 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 69590 47452 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DOXAZOSIN DOXAZOSIN 69591 47453 GPR39 2863 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist 223366131 69594 47454 SHMT1 6470 ENZYME irinotecan IRINOTECAN 22044939 69595 47455 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103732 DESLORATADINE 69596 47456 TOR1A 1861 TRANSPORTER haloperidol HALOPERIDOL 27023437 69598 47457 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE QUERCETIN QUERCETIN 9349317 69600 47458 GUCY1B1 2983 DRUGGABLE GENOME activator CHEMBL1311 ISOSORBIDE MONONITRATE 69601 47459 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 N- (9-FLUORENYLMETHOXYCARBONYL)-L-LEUCINE N- (9-FLUORENYLMETHOXYCARBONYL)-L-LEUCINE 69602 47460 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 8 69604 47461 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 363894217 VORUCICLIB 69606 47462 CD38 952 CELL SURFACE, DRUGGABLE GENOME SAR-650984 ISATUXIMAB 69607 47463 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DOCONEXENT DOCONEXENT 69610 47464 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PEMIROLAST PEMIROLAST 69613 47465 BCL2L2 599 CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist 252166530 VENETOCLAX 69614 47466 GPNMB 10457 ENZYME, DRUGGABLE GENOME CHEMBL1743028 GLEMBATUMUMAB VEDOTIN 69615 47467 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor BGJ398 INFIGRATINIB 69618 47468 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME fluorouracil FLUOROURACIL 24018773,24338217,20530282 69620 47469 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 310264783 69621 47470 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME COCLAURINE COCLAURINE 69622 47471 IL23A 51561 DRUGGABLE GENOME inhibitor CHEMBL1201835 USTEKINUMAB 69623 47472 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GSK-269962A GSK-269962A 69625 47473 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-279835 CHEMBL2003658 22524450 69627 47474 MAP3K7 6885 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565869 CEP-11981 69630 47475 ALOX15 246 ENZYME, DRUGGABLE GENOME 1-PHYTEN-3-OL CHEMBL453797 69632 47476 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651533 69633 47477 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR CYC-116 CYC-116 69634 47478 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL ANAVEX 1007 69636 47479 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE allopurinol ALLOPURINOL 27798726 69637 47480 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565836 69639 47481 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE PICOPLATIN PICOPLATIN 15726096 69640 47482 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Trametinib TRAMETINIB 69641 47483 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PYRACLOSTROBIN PYRACLOSTROBIN 69642 47484 MICU1 10367 TRANSPORTER PF-4427429 69643 47485 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME CENISERTIB CENISERTIB 69644 47486 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650050 CANDESARTAN 69646 47487 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME RETINOID 15824860 69647 47488 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor CHEMBL565612 SOTRASTAURIN 69648 47489 PDE5A 8654 ENZYME, DRUGGABLE GENOME Avanafil AVANAFIL 69650 47490 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE PGF2alpha 69652 47491 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor DASATINIB DASATINIB 69653 47492 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 328083493 69654 47493 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MEHD-7945A DULIGOTUZUMAB 69656 47494 GNA11 2767 CLINICALLY ACTIONABLE Everolimus EVEROLIMUS 27507190 69658 47495 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DECITABINE DECITABINE 25968887 69660 47496 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME homoharringtonine OMACETAXINE MEPESUCCINATE 69661 47497 CBX1 10951 NA IPA-3 CHEMBL472940 69662 47498 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GW441756X GW441756X 69664 47499 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR antagonist GDC0917 69667 47500 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 310264772 PYRIDOSTIGMINE 69669 47501 CCND3 896 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME LEE011 RIBOCICLIB 69671 47502 FGG 2266 DRUGGABLE GENOME, FIBRINOGEN, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE tirofiban TIROFIBAN 20938371 69674 47503 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE IMIDOCARB DIPROPIONATE IMIDOCARB DIPROPIONATE 69676 47504 KDM4A 9682 DRUGGABLE GENOME, ENZYME TDR78834 CHEMBL1507526 69678 47505 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME lamivudine LAMIVUDINE 69684 47506 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX FANGCHINOLINE FANGCHINOLINE 69685 47507 MAPT 4137 DRUGGABLE GENOME SJ000147993 CHEMBL601618 69686 47508 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE glibenclamide GLYBURIDE 18004211 69687 47509 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-BROMO-HEXADECANOIC ACID CHEMBL118417 69689 47510 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SAVIRIN SAVIRIN 69691 47511 POLR1G 10849 NA cisplatin CISPLATIN 69692 47512 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2-AMINO-ANTHRAQUINONE CHEMBL84685 69693 47513 DHFR 1719 DRUGGABLE GENOME, ENZYME MDAM 69694 47514 TUBB 203068 DRUGGABLE GENOME ABT-751 ABT-751 69695 47515 MAPT 4137 DRUGGABLE GENOME DNDI1417932 CHEMBL1334191 69696 47516 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME HYCANTHONE HYCANTHONE 69697 47517 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GOSSYPOL GOSSYPOL 69698 47518 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1908391 MASITINIB 69699 47519 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-54 69700 47520 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565861 69701 47521 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME KMI-1795 CHEMBL2047666 69703 47522 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ACID BLUE 129 ACID BLUE 129 69706 47523 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor RDEA119 69707 47524 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PMZ-2123 69708 47525 KDM4A 9682 DRUGGABLE GENOME, ENZYME HYDROXYZINE PAMOATE HYDROXYZINE PAMOATE 69709 47526 TFF1 7031 GROWTH FACTOR, DRUGGABLE GENOME AG-013 69710 47527 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GINGKOLIC ACID GINGKOLIC ACID 69711 47528 PSMA6 5687 PROTEASE, DRUGGABLE GENOME inhibitor BORTEZOMIB BORTEZOMIB 69712 47529 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL20 ACETAZOLAMIDE 69713 47530 TSPO 706 DRUGGABLE GENOME Phenylpurine acetamide analog 2 69715 47531 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-139459 CHEMBL86464 69717 47532 F7 2155 ENZYME, DRUGGABLE GENOME, PROTEASE CB-813 69720 47533 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200952 METHAMPHETAMINE HYDROCHLORIDE 69721 47534 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 249565734 69722 47535 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 losartan LOSARTAN 9187528 69724 47536 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Imidazo[1,2-b]pyridazine derivative 5 69725 47537 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 QUETIAPINE QUETIAPINE 69726 47538 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE PYRIMETHAMINE PYRIMETHAMINE 69728 47539 POLI 11201 DNA REPAIR QUERCETIN DIHYDRATE QUERCETIN DIHYDRATE 69730 47540 MVD 4597 DRUGGABLE GENOME, ENZYME inhibitor 249565676 69732 47541 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME aflibercept AFLIBERCEPT 20124951 69733 47542 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Senktide SENKTIDE 69734 47543 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor SODIUM PHENYLBUTYRATE 69736 47544 PSMD4 5710 NA inhibitor BORTEZOMIB BORTEZOMIB 69738 47545 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE AMPHOTERICIN B AMPHOTERICIN B 69739 47546 BAD 572 KINASE, DRUGGABLE GENOME AT-101 ISOSORBIDE 69741 47547 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Terbutaline TERBUTALINE 69742 47548 PSMA5 5686 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 69743 47549 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135650893 REGLITAZAR 69744 47550 NDUFS6 4726 ENZYME inhibitor CHEMBL3545135 NV-128 69745 47551 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME CARMINE CARMINE 69746 47552 EHMT1 79813 ENZYME, DRUGGABLE GENOME inhibitor 178103594 69747 47553 POLB 5423 DNA REPAIR, DRUGGABLE GENOME PROTOCATECHUIC ACID PROTOCATECHUIC ACID 69748 47554 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 178100863 69749 47555 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-23 69751 47556 MGLL 11343 DRUGGABLE GENOME, ENZYME inhibitor 178101893 69755 47557 SLC33A1 9197 TRANSPORTER US8592431, 181 69757 47558 SLC29A4 222962 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 178101509 DIPYRIDAMOLE 69759 47559 TARDBP 23435 TUMOR SUPPRESSOR TCMDC-125488 METHOTREXATE 69761 47560 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE Riluzole RILUZOLE 69762 47561 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME XANTHOPTERIN XANTHOPTERIN 69763 47562 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Pyrazole and thiophene derivative 2 69765 47563 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CX-5461 27486174 69767 47564 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CHEMBL1200789 TRICLOFOS SODIUM 69769 47565 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL545315 CANERTINIB DIHYDROCHLORIDE 69771 47566 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME PLX7486 69772 47567 COMT 1312 DRUGGABLE GENOME, ENZYME modafinil MODAFINIL 9352569,9631418,11990384,15956988,12605099,12359690,12465073,11840516 69774 47568 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL3707183 QUINIDINE SULFATE 69776 47569 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652099 69777 47570 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Capmatinib CAPMATINIB 69778 47571 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE FOSFONET FOSFONET 69779 47572 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 methoxyflurane METHOXYFLURANE 9187528 69780 47573 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (S)-methadone 17178267 69781 47574 TOP2B 7155 DRUGGABLE GENOME, ENZYME Doxorubicin DOXORUBICIN 69782 47575 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE imatinib IMATINIB 30237583 69784 47576 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME FUROXAN FUROXAN 69786 47577 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME IL-2 ALDESLEUKIN 69790 47578 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE SOTALOL SOTALOL 2903243 69791 47579 ATXN2 6311 NA PROMETHAZINE PROMETHAZINE 69792 47580 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651637 BRADYKININ 69793 47581 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE GLG-801 69794 47582 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Bicyclic heteroaryl benzamide derivative 3 69795 47583 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME THIRAM THIRAM 69796 47584 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DOX 15494689 69797 47585 COL6A1 1291 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 69800 47586 CACNB3 784 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ION CHANNEL VERAPAMIL VERAPAMIL 69801 47587 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE DCC-2618 RIPRETINIB 69802 47588 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE bosutinib BOSUTINIB 69803 47589 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ORSELLINIC ACID ORSELLINIC ACID 69804 47590 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL1421 DASATINIB 69808 47591 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Prasugrel PRASUGREL 69809 47592 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL1614766 RO-4987655 69812 47593 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LABETALOL LABETALOL 69815 47594 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 15 69816 47595 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE HEPARIN HEPARIN 10997602 69818 47596 TFAP2A 7020 TRANSCRIPTION FACTOR TNF-ALPHA 11438643 69820 47597 MCOLN2 255231 ION CHANNEL, DRUGGABLE GENOME activator 178103002 69824 47598 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE fluorouracil FLUOROURACIL 16822847 69825 47599 POLK 51426 DNA REPAIR, ENZYME MITOXANTRONE MITOXANTRONE 69826 47600 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR PILOCARPINE PILOCARPINE 15183516 69830 47601 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL1852688 INFIGRATINIB 69831 47602 PTGS2 5743 DRUGGABLE GENOME, ENZYME DICLOFENAC DICLOFENAC 69832 47603 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR SB-220025 SB-220025 69833 47604 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TIOXOLONE TIOXOLONE 69834 47605 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DECYLUBIQUINONE DECYLUBIQUINONE 69835 47606 CBL 867 KINASE, ENZYME, CLINICALLY ACTIONABLE FLT3-LIGAND 17446348 69836 47607 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PACLITAXEL PACLITAXEL 16753005 69837 47608 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE BDBM50061608 69838 47609 GLS 2744 ENZYME DEXAMETHASONE DEXAMETHASONE 7904483 69839 47610 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor NINTEDANIB NINTEDANIB 69840 47611 BCHE 590 DRUGGABLE GENOME, ENZYME Di-substituted piperidine derivative 1 69842 47612 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE HM61713 OLMUTINIB 69843 47613 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AZD4547 27595477,22869148 69844 47614 FAAH 2166 ENZYME, DRUGGABLE GENOME Azole derivative 4 69845 47615 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PILARALISIB PILARALISIB 23204226 69846 47616 GSTM1 2944 DRUGGABLE GENOME, ENZYME bleomycin BLEOMYCIN 23323945 69847 47617 KDM4A 9682 DRUGGABLE GENOME, ENZYME DIETHYLCARBAMAZINE CITRATE DIETHYLCARBAMAZINE CITRATE 69848 47618 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE NSC-327705 CHEMBL1317986 69849 47619 TUBA1A 7846 DRUGGABLE GENOME inhibitor CHEMBL2103852 CROLIBULIN 69850 47620 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 178101956 69851 47621 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE carboplatin CARBOPLATIN 30071039 69852 47622 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 69855 47623 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 363894236 AZD-0156 69856 47624 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE CEPHRADINE CEPHRADINE 22166395 69857 47625 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME HARMINE HARMINE 22998443 69858 47626 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE DIMETHYL YELLOW DIMETHYL YELLOW 69862 47627 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME ALSTERPAULLONE ALSTERPAULLONE 69863 47628 IL1B 3553 KINASE, DRUGGABLE GENOME AC-201 DIACEREIN 69864 47629 ALOX15 246 ENZYME, DRUGGABLE GENOME 7,8-DIHYDROXYFLAVONE 7,8-DIHYDROXYFLAVONE 69865 47630 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME DAIDZEIN DAIDZEIN 8593857 69867 47631 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE SAN-300 SAN-300 69868 47632 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 363894209 PAMAPIMOD 69869 47633 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX QUINOXALINE QUINOXALINE 69870 47634 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME BK3 69873 47635 XDH 7498 DRUGGABLE GENOME, ENZYME Azole benzene derivative 1 69874 47636 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE PALBOCICLIB PALBOCICLIB 69876 47637 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR AZD6244 SELUMETINIB 69877 47638 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR SB-202190 SB-202190 69878 47639 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME KERACYANIN KERACYANIN 17360708 69879 47640 BAZ2B 29994 NA DOCEBENONE DOCEBENONE 69882 47641 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-4 69883 47642 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 178101633 69884 47643 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL1879463 DACTOLISIB 69885 47644 F11 2160 DRUGGABLE GENOME, PROTEASE, ENZYME SULFATED PENTAGALLOYLGLUCOSIDE SULFATED PENTAGALLOYLGLUCOSIDE 23316863 69886 47645 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-WO2011152671 2 69888 47646 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL1683544 ERIBULIN MESYLATE 69889 47647 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE LIOTHYRONINE SODIUM LIOTHYRONINE SODIUM 69890 47648 DHFR 1719 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200373 69891 47649 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHADONE METHADONE 12756206 69892 47650 NOS2 4843 DRUGGABLE GENOME, ENZYME DMSO DIMETHYL SULFOXIDE 15919216 69893 47651 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME peginterferon alfa-2b 69895 47652 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Fluorouracil FLUOROURACIL 69896 47653 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME INGENOL MEBUTATE 69897 47654 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CEFTRIAXONE CEFTRIAXONE 22931300 69898 47655 CTSA 5476 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 223366215 69900 47656 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE MULTIVITAMINS 17087956 69902 47657 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Carboplatin CARBOPLATIN 25824335,21135055,27998224 69903 47658 ST14 6768 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 252166691 69904 47659 FAAH 2166 ENZYME, DRUGGABLE GENOME cannabinoids NABIXIMOLS 17290447 69906 47660 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL agonist 178103289 69907 47661 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE sorafenib SORAFENIB 20124951 69908 47662 MAPT 4137 DRUGGABLE GENOME SDZ-201106 CHEMBL314639 69911 47663 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652002 ATOSIBAN 69912 47664 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME GABAPENTIN GABAPENTIN 69913 47665 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL HALAZEPAM HALAZEPAM 69915 47666 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR 1-DEOXYRUBRALACTONE CHEMBL260980 18178092 69917 47667 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL MIDAZOLAM MIDAZOLAM 69918 47668 HEBP1 50865 DRUGGABLE GENOME 2-hydroxybenzamide derivative 2 69919 47669 CA1 759 DRUGGABLE GENOME, ENZYME TRICHLORMETHIAZIDE TRICHLORMETHIAZIDE 69921 47670 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME PAROXETINE PAROXETINE 69924 47671 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-124381 CHEMBL579919 69927 47672 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL181954 NAVEGLITAZAR 69929 47673 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL2109458 AMG-108 69930 47674 PSMC6 5706 NA inhibitor CHEMBL325041 BORTEZOMIB 69933 47675 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE inhibitor 223366048 69937 47676 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000029642 CHEMBL591126 69938 47677 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US9409892, 136 69940 47678 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR PHORBOL MYRISTATE ACETATE PHORBOL MYRISTATE ACETATE 24794745 69941 47679 CD248 57124 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE MORAb-004 ONTUXIZUMAB 69945 47680 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650819 PHENYLEPHRINE 69947 47681 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE AXITINIB AXITINIB 69948 47682 MAOB 4129 DRUGGABLE GENOME, ENZYME PARGYLINE PARGYLINE 25542589 69951 47683 FAAH 2166 ENZYME, DRUGGABLE GENOME Ethylaminopyrimidine derivative 1 69952 47684 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 727725 CHEMBL259422 69954 47685 DNER 92737 NA (+)-JQ1 69956 47686 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE H2O2 8699865,8959153 69957 47687 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 135652556 69958 47688 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178102078 SULINDAC 69961 47689 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE Patritumab PATRITUMAB 69962 47690 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE AG-34 CHEMBL80155 69964 47691 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545368 PANOBINOSTAT LACTATE 69965 47692 CYP2R1 120227 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME ribavirin RIBAVIRIN 69966 47693 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE AG-1879 CHEMBL406845 69967 47694 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE GSK-256073 69968 47695 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 381118814 69969 47696 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE MK2206 MK-2206 69972 47697 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CNDO101 69973 47698 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME TCMDC-125543 CHEMBL546170 69974 47699 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545332 CEP-2563 69975 47700 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649899 69976 47701 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME 1,2,4,5-BENZENETETRAAMINE TETRAHYDROCHLORIDE CHEMBL456559 18989950 69978 47702 AKR1B1 231 DRUGGABLE GENOME, ENZYME Befunolol hci 69983 47703 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652302 69985 47704 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE RAPAMYCIN SIROLIMUS 11108720,11108711,11967149 69987 47705 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor SELICICLIB SELICICLIB 69988 47706 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 310264792 69989 47707 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DITHIOLETHIONE DITHIOLETHIONE 69990 47708 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 223366050 SAPITINIB 69991 47709 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER diltiazem DILTIAZEM 69993 47710 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME MITOXANTRONE MITOXANTRONE 14767525,11839668 69994 47711 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102723 69995 47712 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649864 8-OH-DPAT 69996 47713 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ROSMARINIC ACID ROSMARINIC ACID 69997 47714 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MM-302 GANCOTAMAB 69999 47715 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DNDI1417309 CHEMBL1341830 70000 47716 HTT 3064 DRUGGABLE GENOME HBI-8000 TUCIDINOSTAT 70001 47717 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (-)-PROPANOLOL (-)-PROPANOLOL 70002 47718 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME TUMOR NECROSIS FACTOR 1359970 70003 47719 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor GSK2636771 GSK-2636771 70004 47720 PSMB6 5694 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL371405 MARIZOMIB 70005 47721 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME EUPAFOLIN EUPAFOLIN 70006 47722 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR inhibitor 315661326 70007 47723 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE DIDANOSINE DIDANOSINE 9430255 70008 47724 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ECONAZOLE NITRATE ECONAZOLE NITRATE 70010 47725 NTS 4922 DRUGGABLE GENOME ETHANOL ALCOHOL 9023306,1733422,1686369 70011 47726 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE FULVESTRANT FULVESTRANT 24448819 70016 47727 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR AM0010 PEGILODECAKIN 70017 47728 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME BIO-1211 CHEMBL88478 70018 47729 ATXN2 6311 NA PAROXETINE PAROXETINE 70019 47730 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MINOPAFANT HYDROCHLORIDE MINOPAFANT 70020 47731 HLA-DQA1 3117 CLINICALLY ACTIONABLE lapatinib LAPATINIB 24687830,21245432 70021 47732 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SAVOLITINIB SAVOLITINIB 31315834,27694386 70022 47733 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE TAE-684 TAE-684 70023 47734 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PHA-767491 CHEMBL225519 70024 47735 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PAZOPANIB PAZOPANIB 70025 47736 ATAD5 79915 NA SJ000047241 CHEMBL601933 70026 47737 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR GDC-0980 APITOLISIB 26951309 70027 47738 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565748 70028 47739 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE FGFR INHIBITOR AZD4547 27179038 70029 47740 BAZ2B 29994 NA PROSTAGLANDIN A2 PROSTAGLANDIN A2 70030 47741 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ALTENUSIN ALTENUSIN 70031 47742 TYMSOS 494514 NA sulfasalazine SULFASALAZINE 18322994 70032 47743 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL1078983 AZD-2014 70033 47744 UGT2B7 7364 DRUGGABLE GENOME hmg coa reductase inhibitors 70034 47745 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ETHYL EICOSAPENTAENOIC ACID 70035 47746 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR VORINOSTAT VORINOSTAT 19344175,19966789,26211462,23622981,22260166,20491440,21548582,19084294 70036 47747 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Pyrazole derivative 86 70037 47748 NDUFB11 54539 ENZYME inhibitor CHEMBL3545135 NV-128 70038 47749 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE ANTISENSE OLIGONUCLEOTIDES 15829059 70039 47750 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Bis-indolylmaleimide derivative 1 70041 47751 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 375973259 70042 47752 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENOXACOR BENOXACOR 70043 47753 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Macrolactam derivative 2 70044 47754 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE RG-4929 70045 47755 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR heroin DIACETYLMORPHINE 17373729 70047 47756 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CLOROPHENE CLOROPHENE 70049 47757 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 BUSULFAN BUSULFAN 22931300 70050 47758 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102319 LAPATINIB 70051 47759 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE TAMATINIB R-406 70052 47760 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 178102285 LINIFANIB 70053 47761 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FLUAZINAM FLUAZINAM 70054 47762 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor 178103403 BRINZOLAMIDE 70055 47763 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE EVEROLIMUS EVEROLIMUS 70056 47764 ADAM17 6868 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, NEUTRAL ZINC METALLOPEPTIDASE, TRANSPORTER, ENZYME Aderbasib ADERBASIB 70057 47765 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1201180 DICLOFENAC EPOLAMINE 70058 47766 GDF15 9518 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR SULINDAC SULFIDE 15180942 70059 47767 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR DOVITINIB DOVITINIB 70061 47768 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME ILEPATRIL ILEPATRIL 70062 47769 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE MK-571 MK-571 23073734 70063 47770 KIF11 3832 DRUGGABLE GENOME LY2523355 70067 47771 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR H2O2 9722602 70068 47772 LY96 23643 DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 28696418 70069 47773 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE TRAFERMIN TRAFERMIN 70071 47774 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME RO-410960 CHEMBL1256291 70072 47775 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR DAUNORUBICIN DAUNORUBICIN 22260166 70073 47776 LINGO1 84894 DRUGGABLE GENOME BIIB-033 OPICINUMAB 70074 47777 INPP5D 3635 DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE AQX-1125 ROSIPTOR 70075 47778 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL PRAZEPAM PRAZEPAM 70078 47779 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Crizotinib CRIZOTINIB 70081 47780 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DESMOSDUMOTIN C DESMOSDUMOTIN C 70082 47781 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178100246 LUMIRACOXIB 70083 47782 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Regorafenib REGORAFENIB 25905001 70085 47783 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PF-05230905 70088 47784 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE EMD 121974 12154028 70090 47785 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLOCTAFENINE FLOCTAFENINE 70092 47786 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE antibody DULANERMIN DULANERMIN 70093 47787 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Primaquine PRIMAQUINE 70095 47788 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR P-TOLUENESULFONAMIDE P-TOLUENESULFONAMIDE 70096 47789 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NRP290 70098 47790 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Irofulven/Taxotere 70100 47791 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CARMUSTINE CARMUSTINE 22931300 70103 47792 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ARISTOYUNNOLIN A ARISTOYUNNOLIN A 70106 47793 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1201065 THIAMYLAL SODIUM 70107 47794 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR ENZYME INHIBITOR 11928713 70110 47795 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102999 XIMELAGATRAN 70111 47796 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME upadacitinib UPADACITINIB 70112 47797 PTGS2 5743 DRUGGABLE GENOME, ENZYME naproxen NAPROXEN 19602986 70115 47798 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MISONIDAZOLE MISONIDAZOLE 3753520 70117 47799 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1689 TOLAZOLINE HYDROCHLORIDE 70119 47800 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-41 70120 47801 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178103999 VILAZODONE 70122 47802 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor SOPHORETIN QUERCETIN 70126 47803 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL1742986 ATACICEPT 70127 47804 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-32 70128 47805 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORMADINONE ACETATE CHLORMADINONE ACETATE 70129 47806 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DECITABINE DECITABINE 70130 47807 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE ERLOTINIB ERLOTINIB 70131 47808 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PROPYLPYRAZOLETRIOL PROPYLPYRAZOLETRIOL 70133 47809 RTKN2 219790 NA haloperidol HALOPERIDOL 27023437 70135 47810 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ETICLOPRIDE ETICLOPRIDE 70136 47811 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME FENRETINIDE FENRETINIDE 70137 47812 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALPHA-2B 70138 47813 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE RG-1530 RG-1530 70139 47814 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE GIGANTOL GIGANTOL 24844664 70140 47815 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE EPO EPOETIN ALFA 11986208,11971899,12717822 70142 47816 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME FLUOXETINE FLUOXETINE 70144 47817 POLI 11201 DNA REPAIR TCMDC-124266 CHEMBL124006 70145 47818 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 252166729 AZD-8186 70146 47819 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL574737 UCN-01 70147 47820 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Fludrocortisone FLUDROCORTISONE 70149 47821 POLI 11201 DNA REPAIR DL-CATECHIN TRIHYDRATE CHEMBL1172228 70150 47822 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 E324 E324 70151 47823 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Baricitinib BARICITINIB 70152 47824 RHEB 6009 TUMOR SUPPRESSOR, DRUG RESISTANCE, KINASE, CLINICALLY ACTIONABLE SIROLIMUS SIROLIMUS 26255626 70157 47825 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PERAZINE PERAZINE 70158 47826 ANXA5 308 KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER DNR 11986942 70159 47827 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NORTRIPTYLINE NORTRIPTYLINE 70160 47828 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE Bestatin 70161 47829 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-5 70162 47830 SREBF1 6720 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR NEUROTROPHIC FACTOR 12788519 70164 47831 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102248 PRELADENANT 70165 47832 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor PX-866 SONOLISIB 70168 47833 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE COSMOMYCIN C COSMOMYCIN C 22071520 70169 47834 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME RO-0282750 CHEMBL1397270 70170 47835 GC 2638 DRUGGABLE GENOME deferasirox DEFERASIROX 30651574 70171 47836 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Quinine Sulfate 70172 47837 EYA2 2139 DNA REPAIR PURPUROGALLIN PURPUROGALLIN 70174 47838 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME JNJ-42756493 ERDAFITINIB 26324363,25609060,26992226,28341788 70175 47839 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME SCRIPTAID SCRIPTAID 19966789 70176 47840 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL antagonist 329968409 70178 47841 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 387065616 70179 47842 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE GW441756X GW441756X 70184 47843 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CELECOXIB CELECOXIB 70185 47844 GAPDH 2597 DRUGGABLE GENOME, ENZYME OMIGAPIL OMIGAPIL 70187 47845 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 178103589 RICOLINOSTAT 70190 47846 SMN1 6606 DRUGGABLE GENOME HYDRALAZINE HYDRALAZINE 70192 47847 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CALCIUM PANTOTHENATE CALCIUM PANTOTHENATE 70193 47848 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE HOMOTAURINE 70194 47849 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GEFITINIB GEFITINIB 70196 47850 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor CHEMBL3545001 MK-8353 70197 47851 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000117451 CHEMBL592123 70200 47852 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-525334 CHEMBL401570 70202 47853 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME ENTRECTINIB ENTRECTINIB 70203 47854 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE LASALOCID A SODIUM LASALOCID A SODIUM 70205 47855 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-4782 CHEMBL584619 70206 47856 LTC4S 4056 ENZYME, DRUGGABLE GENOME aspirin ASPIRIN 19862937,15100686,16433794 70207 47857 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY ROSIGLITAZONE ROSIGLITAZONE 15640776,16921272 70210 47858 ENG 2022 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRC105 70211 47859 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL514201 TALMAPIMOD 70212 47860 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME ETHINYL ESTRADIOL ETHINYL ESTRADIOL 21030469 70215 47861 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NITAZOXANIDE NITAZOXANIDE 70216 47862 CP 1356 DRUGGABLE GENOME, ENZYME IL-1RA ANAKINRA 7682588 70217 47863 GMNN 51053 DRUGGABLE GENOME MESO-HEXESTROL MESO-HEXESTROL 70219 47864 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME LEVODOPA LEVODOPA 70220 47865 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL741 LAMOTRIGINE 70222 47866 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CITALOPRAM CITALOPRAM 70224 47867 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX N-(3-OXODODECANOYL)HOMOSERINELACTONE CHEMBL8483 18566250 70225 47868 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CISPLATIN CISPLATIN 11595686,14514923 70226 47869 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Piperidine derivative 1 70228 47870 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 249565895 CHEMBL2203843 70229 47871 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR AUS-131 AUS-131 70230 47872 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545180 THELIATINIB 70233 47873 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME antagonist 340590217 70235 47874 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PEGFILGRASTIM PEGFILGRASTIM 70236 47875 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-36 70237 47876 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME US9346821, A-20 70238 47877 VKORC1 79001 DRUGGABLE GENOME, ENZYME phenprocoumon PHENPROCOUMON 22920394,26445138,19225451,18629445,23602689,20833980,18781852,24474498,27581200,27262824,17596133,25519826,20376629,27488176,26984978,18574025,29577257,30983536,25769357,21057703,21148049,26777610,25244877,28689179,25001883,18950464,19270263,24919870,22571356,18698879,18690342,23774101,25521356,21636598,22592842,23299853,29432897,23423913,28033245,16815313,20020283,24224579 70239 47878 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE progesterone PROGESTERONE 18695978 70240 47879 HSPA5 3309 TRANSPORTER, ENZYME, PROTEASE INHIBITOR, CELL SURFACE, DRUGGABLE GENOME IT-139 IT-139 70241 47880 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-14 70242 47881 SIGIRR 59307 NA agonist 178102770 70245 47882 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL2408045 SAPITINIB 70246 47883 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME KHRINONE E KHRINONE E 70247 47884 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Oxazolyl methylthiothiazole derivative 1 70248 47885 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor IMATINIB IMATINIB 70249 47886 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DISULFIRAM DISULFIRAM 70251 47887 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL464 ETRETINATE 70252 47888 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ERB-041 PRINABEREL 70254 47889 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE succimer SUCCIMER 70255 47890 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME GW3965 CHEMBL59030 70256 47891 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR GSK-961081 70257 47892 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE dasatinib DASATINIB 70258 47893 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-7a 70259 47894 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200715 HEXYLCAINE HYDROCHLORIDE 70262 47895 SMN2 6607 DRUGGABLE GENOME PD-98059 CHEMBL35482 70263 47896 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 178100459 FORMOTEROL 70264 47897 MAOB 4129 DRUGGABLE GENOME, ENZYME N-(2-phenylcyclopropyl) amino acid derivative 1 70266 47898 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Dasatinib DASATINIB 27231123 70267 47899 TDO2 6999 ENZYME, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 7 70269 47900 IL1B 3553 KINASE, DRUGGABLE GENOME infliximab INFLIXIMAB 22960943 70270 47901 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME VITAMIN A 14529804 70271 47902 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor CHEMBL1967878 CENISERTIB 70274 47903 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PROTEOLYTIC ENZYMES 8600653 70276 47904 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RADICICOL RADICICOL 16499313 70277 47905 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME R1295 70278 47906 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL blocker 135652686 70279 47907 CHPT1 56994 NA lamivudine LAMIVUDINE 70280 47908 PPP1R13L 10848 TRANSCRIPTION FACTOR BINDING cisplatin CISPLATIN 70281 47909 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 252166784 70282 47910 RAB9A 9367 ENZYME, DRUGGABLE GENOME 2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE CHEMBL201325 70283 47911 F5 2153 DRUGGABLE GENOME tamoxifen TAMOXIFEN 16818854,14512389 70284 47912 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE AEE-788 AEE-788 70286 47913 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CHELERYTHRINE CHLORIDE CHELERYTHRINE CHLORIDE 70287 47914 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER dobutamine DOBUTAMINE 19542315 70288 47915 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL2103851 AMUVATINIB 70289 47916 LAMB1 3912 DRUGGABLE GENOME HEPARAN SULFATE 8873769 70290 47917 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TRIFLUPROMAZINE TRIFLUPROMAZINE 70291 47918 HSPA8 3312 TUMOR SUPPRESSOR CYCLOSPORIN A 1429556 70293 47919 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NANAOMYCIN NANAOMYCIN 70294 47920 TUBB 203068 DRUGGABLE GENOME CHEMBL492399 VERUBULIN 70295 47921 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR XANTHOHUMOL XANTHOHUMOL 22111577 70297 47922 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING TACEDINALINE TACEDINALINE 18692397 70299 47923 SYP 6855 TRANSPORTER 6-HYDROXYDOPAMINE 15765516 70300 47924 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE RO-410960 CHEMBL1256291 70301 47925 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR midazolam MIDAZOLAM 70302 47926 GPR12 2835 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651563 70303 47927 STK4 6789 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 70304 47928 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME RG-1530 RG-1530 70305 47929 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BIFENAZATE BIFENAZATE 70306 47930 PLK2 10769 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565601 ONVANSERTIB 70307 47931 SRPK1 6732 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME RG-1530 RG-1530 70308 47932 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHENYLBUTAZONE PHENYLBUTAZONE 22931300 70309 47933 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-9037 CHEMBL1451216 70310 47934 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1088751 PH-797804 70312 47935 RAB9A 9367 ENZYME, DRUGGABLE GENOME RABEPRAZOLE SODIUM RABEPRAZOLE SODIUM 70313 47936 LY96 23643 DRUGGABLE GENOME inhibitor 315661112 70315 47937 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE TGF 16928297 70316 47938 POLI 11201 DNA REPAIR SJ000001516 CHEMBL592316 70317 47939 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME quinine QUININE 70318 47940 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 135651309 70319 47941 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR NCX-1015 70320 47942 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE everolimus EVEROLIMUS 26458301,24628014 70322 47943 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR EPINEPHRINE EPINEPHRINE 12407113 70324 47944 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103434 METHAZOLAMIDE 70329 47945 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Trimethoprim TRIMETHOPRIM 70330 47946 RACGAP1 29127 NA PARAROSANILINE PARAROSANILINE 70331 47947 ATAD5 79915 NA TRIMETHOBENZAMIDE HYDROCHLORIDE TRIMETHOBENZAMIDE HYDROCHLORIDE 70335 47948 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 381118815 70336 47949 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ANTAZOLINE ANTAZOLINE 70337 47950 POLB 5423 DNA REPAIR, DRUGGABLE GENOME OXYTETRACYCLINE OXYTETRACYCLINE 70338 47951 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL580 LORAZEPAM 70339 47952 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor SB939 70341 47953 THY1 7070 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE FCA 9521021 70342 47954 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME modulator CHEMBL2103836 IMAGABALIN 70343 47955 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE RLX030 SERELAXIN 70344 47956 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ENOXOLONE ENOXOLONE 22931300 70345 47957 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER GREEN TEA POLYPHENOLS 11853888 70346 47958 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MECAMYLAMINE MECAMYLAMINE 22931300 70349 47959 MPHOSPH8 54737 NA SEMAXANIB SEMAXANIB 70350 47960 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME MLN-8054 MLN-8054 70352 47961 AQP1 358 ION CHANNEL, DRUGGABLE GENOME Collagenase COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 70353 47962 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE INCB50465 70354 47963 KDM4A 9682 DRUGGABLE GENOME, ENZYME INDINAVIR SULFATE INDINAVIR SULFATE 70355 47964 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor 178102283 CHEMBL379218 70356 47965 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OCTOCRYLENE OCTOCRYLENE 70358 47966 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR JUGLONE JUGLONE 70359 47967 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ISONIAZID ISONIAZID 22931300 70360 47968 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DNDI1417411 CHEMBL1445650 70364 47969 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200975 CLOCORTOLONE PIVALATE 70365 47970 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PD-169316 PD-169316 70367 47971 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER DOXORUBICIN DOXORUBICIN 26288684 70370 47972 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BORTEZOMIB BORTEZOMIB 70371 47973 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650042 70374 47974 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE GOSSYPOL GOSSYPOL 70375 47975 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102547 70376 47976 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator 178103409 DALTEPARIN 70377 47977 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE THIOGUANOSINE THIOGUANOSINE 70378 47978 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SYMCLOSENE SYMCLOSENE 70380 47979 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27454349-Compound-99 70384 47980 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE THIORIDAZINE HYDROCHLORIDE THIORIDAZINE HYDROCHLORIDE 70385 47981 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 178100567 70386 47982 USP1 7398 DNA REPAIR, PROTEASE, ENZYME SEPIAPTERIN SEPIAPTERIN 70387 47983 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOPOTECAN HYDROCHLORIDE TOPOTECAN HYDROCHLORIDE 70388 47984 IGFBP5 3488 DRUGGABLE GENOME DHT ANDROSTANOLONE 16368782 70389 47985 RIPK2 8767 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 348353647 70390 47986 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DYCLONINE HYDROCHLORIDE DYCLONINE HYDROCHLORIDE 70391 47987 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-710 CHEMBL596839 70392 47988 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR antagonist 223366062 AT-406 70393 47989 DOT1L 84444 CLINICALLY ACTIONABLE, DNA REPAIR, METHYL TRANSFERASE, DRUGGABLE GENOME, ENZYME hydrochlorothiazide HYDROCHLOROTHIAZIDE 22440088 70395 47990 RGS4 5999 DRUGGABLE GENOME risperidone RISPERIDONE 18204343 70396 47991 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Phenothiazine derivatives 70398 47992 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME LEVODOPA LEVODOPA 70401 47993 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR ALISERTIB ALISERTIB 70402 47994 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MAPROTILINE HYDROCHLORIDE MAPROTILINE HYDROCHLORIDE 70403 47995 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CYC-116 CYC-116 70404 47996 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME 178101237 70406 47997 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL384304 RG-547 70407 47998 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME FLAVOXATE FLAVOXATE 70408 47999 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3545383 RG-7167 70410 48000 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE tirofiban TIROFIBAN 20938371 70411 48001 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Demcizumab DEMCIZUMAB 26855149 70414 48002 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME inhibitor 178103142 CHEMBL117225 70415 48003 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103870 SOTALOL 70416 48004 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 70417 48005 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER oxcarbazepine OXCARBAZEPINE 28837897 70418 48006 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AG-126 CHEMBL77387 70420 48007 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-35 70422 48008 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER VERAPAMIL VERAPAMIL 17646169,19725578 70423 48009 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL ethosuximide ETHOSUXIMIDE 23859570,21747585,28753467,25155934 70424 48010 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LGD-2941 LGD-2941 70425 48011 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TOPOTECAN HYDROCHLORIDE TOPOTECAN HYDROCHLORIDE 70426 48012 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652028 70427 48013 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE CORTISOL HYDROCORTISONE 10731548 70429 48014 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 178102666 70431 48015 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR Phenoxodiol 70432 48016 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Dextromethorphan DEXTROMETHORPHAN 70434 48017 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000114741 CHEMBL591370 70435 48018 POLK 51426 DNA REPAIR, ENZYME NSC-60340 CHEMBL1534034 70436 48019 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME quinidine QUINIDINE 70437 48020 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ISOKAEMPFERIDE ISOKAEMPFERIDE 70441 48021 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR fenofibrate FENOFIBRATE 16607077 70442 48022 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor SORAFENIB TOSYLATE 70443 48023 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CHLORANIL CHLORANIL 70444 48024 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE MUNDULONE MUNDULONE 70446 48025 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME inhibitor 135650114 CLOTRIMAZOLE 70447 48026 CALR 811 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME VACCINIA VACCINE 15364449 70448 48027 NBN 4683 CLINICALLY ACTIONABLE, KINASE, TUMOR SUPPRESSOR GPI-15427 25324139 70450 48028 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RETINOIC ACIDS 9262057 70451 48029 POLR2A 5430 NA PSI-7409 CHEMBL486231 20516278 70452 48030 SMN2 6607 DRUGGABLE GENOME BENZENE-1,2-DIAMINE CHEMBL70582 70453 48031 KAT2B 8850 ENZYME, DRUGGABLE GENOME DIETHYL-2-UNDECYLIDENEMALONATE CHEMBL1797707 21292492 70454 48032 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PEGFILGRASTIM PEGFILGRASTIM 70455 48033 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 70456 48034 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650345 HALOPERIDOL 70457 48035 ALDH1A1 216 DRUGGABLE GENOME, ENZYME (E)-DIBENZYLIDENEACETONE CHEMBL17201 70458 48036 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER dipyridamole DIPYRIDAMOLE 70459 48037 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME TAMATINIB R-406 70462 48038 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Intedanib NINTEDANIB 70464 48039 HEXB 3074 ENZYME N-ACETYLGLUCOSAMINE THIAZOLINE CHEMBL257158 20822912 70465 48040 CXCL8 3576 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 9271387 70466 48041 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650091 70467 48042 MPHOSPH8 54737 NA RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 70468 48043 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE RETINOID 15020266 70469 48044 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TEBUFENPYRAD TEBUFENPYRAD 70470 48045 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING DAUNORUBICIN DAUNORUBICIN 22260166 70471 48046 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME R-1487 R-1487 70472 48047 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 249565826 70473 48048 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CABOZANTINIB CABOZANTINIB 70476 48049 BAZ2B 29994 NA 5-NITRO-[1,10]PHENANTHROLINE CHEMBL101815 70479 48050 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor REGORAFENIB REGORAFENIB 70480 48051 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor BELINOSTAT BELINOSTAT 70481 48052 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-67 70483 48053 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OXYBUTYNIN OXYBUTYNIN 70484 48054 HSPA8 3312 TUMOR SUPPRESSOR NSC-119915 CHEMBL1481974 70485 48055 APOE 348 DRUGGABLE GENOME STAUROSPORINE STAUROSPORINE 11948667 70488 48056 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417941 CHEMBL2095095 70492 48057 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME ProstaVac 70493 48058 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CHEMBL220492 TOPIRAMATE 70494 48059 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DEMETHOXYCURCUMIN DEMETHOXYCURCUMIN 23145932 70497 48060 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TRIMETHOPRIM TRIMETHOPRIM 22931300 70498 48061 ADAM17 6868 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, NEUTRAL ZINC METALLOPEPTIDASE, TRANSPORTER, ENZYME inhibitor 348353646 70499 48062 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1088750 ARRY-797 70500 48063 PDE5A 8654 ENZYME, DRUGGABLE GENOME EXISULIND EXISULIND 70501 48064 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME LARGAZOLE LARGAZOLE 21420302,25203782,20491440 70502 48065 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 178102526 70503 48066 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ALT-110 70504 48067 ALOX15 246 ENZYME, DRUGGABLE GENOME TYRPHOSTIN AG-835 CHEMBL261557 70505 48068 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CAL-101 IDELALISIB 70506 48069 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NAN-190 NAN-190 70509 48070 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME CART-BCMA cells 70510 48071 PARP3 10039 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR rucaparib RUCAPARIB 70512 48072 BAZ2B 29994 NA TYRPHOSTIN 51 TYRPHOSTIN 51 70515 48073 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME US9096594, 3 70518 48074 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 340590284 MAPRACORAT 70519 48075 USP1 7398 DNA REPAIR, PROTEASE, ENZYME RO-106-9920 CHEMBL271023 70520 48076 MAOA 4128 DRUGGABLE GENOME, ENZYME V3381 INDANTADOL 70525 48077 AQP8 343 ION CHANNEL ETHINYLESTRADIOL ETHINYL ESTRADIOL 18683753 70526 48078 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME H89 CHEMBL104264 70527 48079 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE ICR62 11235991 70528 48080 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE DIGITOXIGENIN DIGITOXIGENIN 70529 48081 NOTCH3 4854 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME antibody 252166663 TAREXTUMAB 70530 48082 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AR-12286 VEROSUDIL 70531 48083 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor SORAFENIB TOSYLATE 70532 48084 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 2 70534 48085 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SORAFENIB SORAFENIB 70535 48086 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SIMVASTATIN SIMVASTATIN 22931300 70537 48087 POLI 11201 DNA REPAIR DAPHNORIN DAPHNORIN 70538 48088 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651525 70544 48089 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1201477 POLYESTRADIOL PHOSPHATE 70545 48090 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor PONATINIB PONATINIB 70546 48091 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 252166635 VELUSETRAG 70547 48092 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME INFIGRATINIB INFIGRATINIB 27998968,29848605,27870574 70548 48093 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Folic Acid 70549 48094 PAH 5053 DRUGGABLE GENOME, ENZYME PP-1420 70550 48095 PTGS2 5743 DRUGGABLE GENOME, ENZYME diclofenac DICLOFENAC 19602986 70551 48096 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Epitinib EPITINIB 70553 48097 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Sirolimus SIROLIMUS 26144316 70554 48098 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CAPSAZEPINE CAPSAZEPINE 70556 48099 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE cytarabine CYTARABINE 70557 48100 FAAH 2166 ENZYME, DRUGGABLE GENOME Isoxazoline derivative 2 70558 48101 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL587723 AEE-788 70559 48102 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ANECORTAVE ACETATE ANECORTAVE ACETATE 70564 48103 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Ropivacaine ROPIVACAINE 70565 48104 PAPOLA 10914 NA ETOPOSIDE ETOPOSIDE 15503822 70566 48105 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist 381118914 70567 48106 MAPT 4137 DRUGGABLE GENOME SJ000079774 CHEMBL601192 70569 48107 ATP2C1 27032 ENZYME, TRANSPORTER, DRUGGABLE GENOME DESFLURANE DESFLURANE 70571 48108 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CLOZAPINE CLOZAPINE 11490180 70572 48109 SEMA3C 10512 CLINICALLY ACTIONABLE, DRUGGABLE GENOME irinotecan IRINOTECAN 22664479 70574 48110 BCHE 590 DRUGGABLE GENOME, ENZYME PMID29757691-Compound-2a 70575 48111 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CP-724714 CP-724714 70577 48112 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102742 70580 48113 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL646 TRIAZOLAM 70581 48114 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Six-membered heterocyclic benzamide derivative 1 70582 48115 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme5 70583 48116 GAL 51083 DRUGGABLE GENOME ESTRADIOL BENZOATE 14666144 70586 48117 KDM4A 9682 DRUGGABLE GENOME, ENZYME PROTOPORPHYRIN PROTOPORPHYRIN 70587 48118 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME vinorelbine VINORELBINE 22441531 70588 48119 UGT1A9 54600 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE febuxostat FEBUXOSTAT 27798726 70591 48120 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME SJ000201287 CHEMBL590900 70592 48121 BRD9 65980 ENZYME 387065622 70596 48122 RRM2B 50484 ENZYME, DRUGGABLE GENOME, DNA REPAIR LOR-2040 70597 48123 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Imidazoleisoindoles derivative 1 70600 48124 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Cobimetinib COBIMETINIB 70605 48125 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CABOZANTINIB CABOZANTINIB 26673800,25351743,26372962 70606 48126 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FUDR FLOXURIDINE 11115403 70610 48127 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIGITOXIGENIN DIGITOXIGENIN 70611 48128 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME VERAPAMIL VERAPAMIL 7683421 70612 48129 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME phenobarbital PHENOBARBITAL 17638512 70614 48130 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ERGOCRYPTINE ERGOCRYPTINE 70615 48131 MGLL 11343 DRUGGABLE GENOME, ENZYME Pyrazole derivative 82 70616 48132 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CAR-T cells targeting EpCAM 70617 48133 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-33b 70618 48134 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BENZBROMARONE BENZBROMARONE 70619 48135 AOX1 316 DRUGGABLE GENOME Isovanillin ISOVANILLIN 70621 48136 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 3R14S-OCHRATOXIN A 3R14S-OCHRATOXIN A 70622 48137 GMNN 51053 DRUGGABLE GENOME DIPHYLLIN DIPHYLLIN 70623 48138 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE Ergot alkaloids 25096645 70624 48139 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor DACOMITINIB DACOMITINIB 70627 48140 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE SUFENTANIL SUFENTANIL 70629 48141 HDAC11 79885 DRUGGABLE GENOME, ENZYME PMID29671355-Compound-23 70630 48142 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX 10-METHOXYLRUTAECARPINE CHEMBL85826 70633 48143 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE 2,3,4-TRIHYDROXY-4'-ETHOXYBENZOPHENONE 70636 48144 MAOB 4129 DRUGGABLE GENOME, ENZYME 8-[METHYL(4-PHENYLBUTYL)AMINO]CAFFEINE CHEMBL1927684 22055712 70637 48145 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 249565687 70638 48146 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR RO-410960 CHEMBL1256291 70639 48147 MPST 4357 ENZYME, DRUGGABLE GENOME inhibitor 381744892 70640 48148 ABCA1 19 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE simvastatin SIMVASTATIN 20031551 70641 48149 TNFRSF4 7293 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE INCAGN1949 70642 48150 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL448343 LESOGABERAN 70643 48151 EYA2 2139 DNA REPAIR GNF-PF-5007 CHEMBL1989853 70644 48152 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL148674 VARESPLADIB 70646 48153 GBA 2629 DRUGGABLE GENOME, ENZYME GW405833 CHEMBL73711 70647 48154 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 5-METHOXYFLAVONE CHEMBL16685 70650 48155 ITGA3 3675 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE 252827506 70651 48156 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 252166734 70652 48157 FKBP5 2289 DRUGGABLE GENOME mirtazapine MIRTAZAPINE 20709156,15565110 70653 48158 PPA1 5464 ENZYME GUANIDINIUM 8639227 70654 48159 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-67746 CHEMBL333177 70656 48160 TNFRSF9 3604 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE MG7-CART 70658 48161 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-2335 CHEMBL601146 70661 48162 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AMG 337 26432108 70662 48163 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CENISERTIB CENISERTIB 70663 48164 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NALTREXONE NALTREXONE 70665 48165 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270010-Compound-Figure17-3 70666 48166 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE NSC348884 21719597 70667 48167 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZIRAM ZIRAM 70668 48168 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HYDRALAZINE HYDRALAZINE 70669 48169 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000032154 CHEMBL591876 70670 48170 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DITHIOLETHIONE DITHIOLETHIONE 70672 48171 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME VEGF 16400523 70673 48172 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME MASITINIB MASITINIB 70674 48173 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 sulfamethoxazole SULFAMETHOXAZOLE 9187528 70675 48174 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SKF-10047 CHEMBL101510 70676 48175 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME SURAMIN HEXASODIUM SURAMIN HEXASODIUM 70677 48176 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE ISOBAVACHALCONE ISOBAVACHALCONE 24047800 70678 48177 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME HOE-33342 CHEMBL343002 70680 48178 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME ABI-009 70682 48179 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 252166676 70683 48180 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE SEMAGACESTAT SEMAGACESTAT 19443228 70685 48181 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 2-PICOLINIC ACID 2-PICOLINIC ACID 70686 48182 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MEVASTATIN MEVASTATIN 70687 48183 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3756 CHEMBL597035 70688 48184 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME OSI-632 OSI-632 70689 48185 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR activator BEXAROTENE BEXAROTENE 70690 48186 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SB-408124 CHEMBL1334465 70692 48187 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CEFOTAXIME SODIUM CEFOTAXIME SODIUM 70694 48188 CFH 3075 DRUGGABLE GENOME Trumenba 70696 48189 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE vaccine PRINOMASTAT PRINOMASTAT 70697 48190 MAPT 4137 DRUGGABLE GENOME GNF-PF-1947 CHEMBL585591 70698 48191 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME DEOXYCYTIDINE DEOXYCYTIDINE 16276353 70699 48192 USP1 7398 DNA REPAIR, PROTEASE, ENZYME MERCURIC CHLORIDE MERCURIC CHLORIDE 70700 48193 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PURPURIN PURPURIN 70701 48194 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-74859 CHEMBL477936 70702 48195 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING TCMDC-139459 CHEMBL86464 70703 48196 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135650692 70704 48197 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Pyridine derivative 22 70705 48198 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-95397 CHEMBL429095 70707 48199 FAAH 2166 ENZYME, DRUGGABLE GENOME Piperazine carbamic compound 2 70708 48200 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MURAGLITAZAR MURAGLITAZAR 70709 48201 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (S)-PINACIDIL (S)-PINACIDIL 70711 48202 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE lumefantrine LUMEFANTRINE 70713 48203 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME TCMDC-124224 CHEMBL580421 70715 48204 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ERLOTINIB ERLOTINIB 17575239 70716 48205 PDE4D 5144 DRUGGABLE GENOME, ENZYME quetiapine QUETIAPINE 70718 48206 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME lovastatin LOVASTATIN 70719 48207 VCP 7415 TRANSPORTER, ENZYME, DNA REPAIR, DRUGGABLE GENOME CB-5083 CB-5083 26104798 70721 48208 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL2103851 AMUVATINIB 70722 48209 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE EXEMESTANE EXEMESTANE 18256205 70724 48210 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Eribulin ERIBULIN 70729 48211 ABCB11 8647 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE HYDROXYPROGESTERONE CAPROATE HYDROXYPROGESTERONE CAPROATE 23129211 70730 48212 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR PAULLONE PAULLONE 17149860 70731 48213 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR DS-6501B 31399568 70732 48214 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME PMA 9307039 70733 48215 UMPS 7372 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE tegafur TEGAFUR 20647221,16818689 70734 48216 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1200912 PHENTERMINE HYDROCHLORIDE 70735 48217 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor DINACICLIB DINACICLIB 70738 48218 NDUFAF2 91942 ENZYME inhibitor CHEMBL3545320 ME-344 70739 48219 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR MK-6913 MK-6913 70740 48220 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR REBAMIPIDE REBAMIPIDE 17171453 70741 48221 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 249565861 70742 48222 PTGS1 5742 ENZYME, DRUGGABLE GENOME Salicyclic acid 70743 48223 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TESTOSTERONE TESTOSTERONE 16038533 70744 48224 PTGS2 5743 DRUGGABLE GENOME, ENZYME Diflunisal DIFLUNISAL 70746 48225 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000133784 CHEMBL589670 70747 48226 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME 178101761 70748 48227 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 374883884 70749 48228 ATAD5 79915 NA GENISTEIN GENISTEIN 70750 48229 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE DHM25 26237138 70752 48230 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 3-EPI-ISOCUCURBITACIN D CHEMBL2022241 25756299 70753 48231 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 mesoridazine MESORIDAZINE 19923256 70754 48232 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME GLAUCINE METHIODIDE GLAUCINE METHIODIDE 70755 48233 HMGCR 3156 ENZYME, DRUGGABLE GENOME Quinoline derivative 17 70756 48234 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL1687 TUBOCURARINE CHLORIDE 70757 48235 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103820 NEBIVOLOL 70758 48236 PSMA1 5682 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL451887 CARFILZOMIB 70759 48237 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 3',4' DICHLOROBENZAMIL 3',4' DICHLOROBENZAMIL 70760 48238 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PHENMEDIPHAM PHENMEDIPHAM 70761 48239 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CENISERTIB CENISERTIB 70762 48240 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Motesanib MOTESANIB 20633291 70763 48241 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR THYMOSIN BETA-4 70766 48242 GAST 2520 DRUGGABLE GENOME, HORMONE ACTIVITY, ENZYME G17DT 70767 48243 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR SJ000112483 CHEMBL603024 70768 48244 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NITROFURANTOIN NITROFURANTOIN 70771 48245 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor VANDETANIB VANDETANIB 70774 48246 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CORALYNE CORALYNE 70775 48247 CDK17 5128 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR inhibitor CHEMBL445813 AT-7519 70777 48248 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME XK469 12085231 70778 48249 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE RAFOXANIDE RAFOXANIDE 70779 48250 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Amidopyrazole derivative 6 70780 48251 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER VERAPAMIL VERAPAMIL 24607999,22405646,21348461,17964170,22209486,25686592,11754602,22429509,24992153,23683834,18257545,21856049,20363635 70781 48252 PCYT2 5833 ENZYME lamivudine LAMIVUDINE 70783 48253 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR ETHANOL ALCOHOL 16272341 70784 48254 HBB 3043 DRUGGABLE GENOME, ENZYME MERCURIC CHLORIDE MERCURIC CHLORIDE 70785 48255 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Indoline derivative 9 70786 48256 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE JNJ-7706621 JNJ-7706621 70787 48257 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL inhibitor 135652013 70788 48258 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CAFFEIC ACID CAFFEIC ACID 70789 48259 AKR1B1 231 DRUGGABLE GENOME, ENZYME Guanadrel Sulfate 70792 48260 ATXN2 6311 NA CEPHARANTHINE CEPHARANTHINE 70794 48261 TUBA4A 7277 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 70795 48262 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE PMA 10632899 70796 48263 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CONGO RED CONGO RED 70797 48264 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32z 70798 48265 ABL2 27 KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME inhibitor 249565827 70800 48266 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3544966 GSK-1059615 70801 48267 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 darunavir DARUNAVIR 70802 48268 MAP3K10 4294 SERINE THREONINE KINASE, ENZYME, KINASE, DRUGGABLE GENOME TAMATINIB R-406 70803 48269 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME RG-1530 RG-1530 70804 48270 TCF7L2 6934 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR repaglinide REPAGLINIDE 20054294 70805 48271 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR S-(P-AZIDOPHENACYL)GLUTATHIONE CHEMBL1256813 70806 48272 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200875 FLAVOXATE HYDROCHLORIDE 70807 48273 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CLONAZEPAM CLONAZEPAM 70808 48274 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR VITAMIN D 7917316,8961271,11353809,7489414,12649563,9037942 70809 48275 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL1201733 PAZOPANIB HYDROCHLORIDE 70810 48276 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME pazopanib PAZOPANIB 24107802 70813 48277 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649916 70814 48278 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Icatibant ICATIBANT 70815 48279 POLK 51426 DNA REPAIR, ENZYME TCMDC-125465 CHEMBL536151 70816 48280 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME BELINOSTAT BELINOSTAT 70817 48281 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Arsenic trioxide 26823493,21183792 70818 48282 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIPHENIDOL DIPHENIDOL 70819 48283 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Salicylic acid derivative 6 70820 48284 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Saprisartan SAPRISARTAN 70821 48285 NOS1 4842 DRUGGABLE GENOME, ENZYME IDOXIFENE IDOXIFENE 12098595 70823 48286 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 252827418 CHEMBL290376 70824 48287 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PICONOL PICONOL 70825 48288 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651581 TRYPTAMINE 70827 48289 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE ERLOTINIB ERLOTINIB 70829 48290 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VB4-845 OPORTUZUMAB MONATOX 23900680 70831 48291 SERPINA3 12 PROTEASE INHIBITOR, DRUGGABLE GENOME antineoplastic agents 21487324 70832 48292 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR Ilodecakin ILODECAKIN 70833 48293 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TRETINOIN TRETINOIN 22931300 70834 48294 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL744 RILUZOLE 70838 48295 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 7,8,2'-TRIHYDROXYFLAVONE CHEMBL244707 70839 48296 BSG 682 DRUGGABLE GENOME, TRANSPORTER antibody 405560467 70840 48297 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ADXS31-164 20725099 70841 48298 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER POLYPHENOL 11518657 70843 48299 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME PYRONIN Y PYRONIN Y 70844 48300 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL3545145 WX-554 70849 48301 AQP1 358 ION CHANNEL, DRUGGABLE GENOME MRG-201 70850 48302 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR STZ STREPTOZOCIN 16342200 70851 48303 TLR7 51284 DRUGGABLE GENOME ANA773 70852 48304 GLS 2744 ENZYME CURCUMIN CURCUMIN 70853 48305 TMEM97 27346 NA Benzamide derivative 7 70857 48306 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650261 FINGOLIMOD 70858 48307 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor AEE 788 70860 48308 SMN2 6607 DRUGGABLE GENOME PT-103 CHEMBL398765 70861 48309 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ARBACLOFEN ARBACLOFEN 70862 48310 HOMER1 9456 KINASE haloperidol HALOPERIDOL 27023437 70865 48311 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE D4T STAVUDINE 11141242 70866 48312 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME C-1311 C-1311 70867 48313 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-39 70870 48314 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIMPYLATE DIMPYLATE 70871 48315 CDK10 8558 DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR, ENZYME, SERINE THREONINE KINASE ALVOCIDIB ALVOCIDIB 70872 48316 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE SOMATOTROPIN HUMAN GROWTH HORMONE 15760670,2143511 70874 48317 GLS 2744 ENZYME INDOCYANINE GREEN INDOCYANINE GREEN 70879 48318 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651431 70882 48319 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DESIPRAMINE DESIPRAMINE 70883 48320 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545226 ACUMAPIMOD 70884 48321 ME3 10873 ENZYME MALONIC ACID MALONIC ACID 19595601 70885 48322 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ACITRETIN ACITRETIN 70887 48323 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL1079593 VS-5584 70888 48324 KMO 8564 DRUGGABLE GENOME, ENZYME Aryl pyrimidine derivative 4 70889 48325 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE hydromorphone HYDROMORPHONE 18695978 70890 48326 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Gedatolisib GEDATOLISIB 24042735,25688157,21325073 70891 48327 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ZERANOL ZERANOL 70892 48328 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BAS03450373 CHEMBL1576310 70893 48329 MAPT 4137 DRUGGABLE GENOME EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 70894 48330 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR verapamil VERAPAMIL 21562465 70897 48331 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE VM-206 70898 48332 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702259 FUTIBATINIB 70899 48333 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Rosiglitazone + simvastatin 70901 48334 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565646 PILARALISIB 70902 48335 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PHENAMIL METHANESULFONATE PHENAMIL METHANESULFONATE 70903 48336 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR CEFIXIME CEFIXIME 70904 48337 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR METHACYCLINE HYDROCHLORIDE METHACYCLINE HYDROCHLORIDE 70906 48338 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-34 70907 48339 MT-RNR1 4549 KINASE tobramycin TOBRAMYCIN 18830133,16875663,9164619,19682603,16631122,21495045,16458854,12031626,16375862,9831149,17637808,22475488,11857751,27397648,9779807,7689389,20111055,9111378,27427311,17698030,11313749,20416460,16168391,24703164,9950117,21504270,11174059,8285309,18790089,15917167,20353758,16955413,16380089,14699607,17999439,14755216,17341440,19376484,15708009,25515069,15555598,11079536,17434445 70909 48340 ZNF565 147929 NA methylphenidate METHYLPHENIDATE 29382897 70910 48341 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 252827368 PEXIDARTINIB 70912 48342 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE COBALT 60 8547828 70913 48343 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE NVP-AEW541 AEW-541 26577700 70914 48344 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NINTEDANIB NINTEDANIB 70916 48345 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR HISPIDULIN HISPIDULIN 70917 48346 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME EMODIN EMODIN 70919 48347 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME MERCURIC CHLORIDE MERCURIC CHLORIDE 70921 48348 XRCC4 7518 KINASE docetaxel DOCETAXEL 20157331 70923 48349 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR FLAVOPIRIDOL ALVOCIDIB 10887097,15235103,11751522 70924 48350 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TIOPRONIN TIOPRONIN 70925 48351 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR antagonist 223366043 70926 48352 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Imidazo[1,2-b]pyridazine derivative 7 70927 48353 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ETOPOSIDE ETOPOSIDE 70928 48354 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE N-(4-NITROPHENYL)ANTHRANILIC ACID CHEMBL1574420 70929 48355 TNNC1 7134 DRUGGABLE GENOME BEPRIDIL BEPRIDIL 70930 48356 SCARB1 949 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME atorvastatin ATORVASTATIN 20064494 70931 48357 SPARC 6678 CELL SURFACE, DRUGGABLE GENOME NAB-PACLITAXEL 70932 48358 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE LEVOMETHADYL ACETATE 70934 48359 HLA-DPB1 3115 CELL SURFACE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE clozapine CLOZAPINE 11266078 70935 48360 GRK2 156 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 252166647 70936 48361 TARDBP 23435 TUMOR SUPPRESSOR CHENODIOL CHENODIOL 70938 48362 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RO-106-9920 CHEMBL271023 70940 48363 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DAP-81 CHEMBL1242101 70941 48364 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE blocker 178100971 CANNABIDIOL 70942 48365 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME CYANIN CYANIN 70943 48366 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135650441 70944 48367 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL3039588 PASIREOTIDE DIASPARTATE 70945 48368 PTGS1 5742 ENZYME, DRUGGABLE GENOME EPICATECHIN (+)-EPICATECHIN 70946 48369 KLK4 9622 PROTEASE, DRUGGABLE GENOME, ENZYME Cetraxate CETRAXATE 70948 48370 HEBP1 50865 DRUGGABLE GENOME 3-phenyl propanoic derivative 2 70949 48371 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CNI-1493 SEMAPIMOD 70950 48372 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Spiroquinolone derivative 1 70951 48373 FGB 2244 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, FIBRINOGEN, DRUGGABLE GENOME tirofiban TIROFIBAN 20938371 70952 48374 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME LINOLENIC ACID LINOLENIC ACID 70953 48375 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 363894177 70955 48376 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 363894207 FLUMATINIB 70958 48377 PRKG1 5592 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME TAE-684 TAE-684 70959 48378 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178101971 70961 48379 PIPSL 266971 KINASE inhibitor BORTEZOMIB BORTEZOMIB 70962 48380 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE Epigallocatechin gallate 70963 48381 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE partial agonist CHEMBL1134 DECAMETHONIUM BROMIDE 70965 48382 SLC27A1 376497 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 252827459 70966 48383 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SGI-1776 SGI-1776 70967 48384 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE inhibitor CHEMBL1174 EPTIFIBATIDE 70968 48385 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DACTINOMYCIN DACTINOMYCIN 70969 48386 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-28 70971 48387 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME SB-206553 CHEMBL297784 70974 48388 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Isoindoline derivative 3 70975 48389 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GENTAMICIN GENTAMICIN 8779884 70976 48390 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW856804X GW856804X 70977 48391 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PROCATEROL HYDROCHLORIDE PROCATEROL HYDROCHLORIDE 70978 48392 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Galantamine GALANTAMINE 70979 48393 RACGAP1 29127 NA NSC-348401 CHEMBL515505 70980 48394 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BAICALEIN BAICALEIN 70982 48395 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Famitinib FAMITINIB 70984 48396 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100777 SITAXENTAN 70986 48397 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE MK-4827 NIRAPARIB 70987 48398 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME OPB-111077 70988 48399 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-1083 CHEMBL530361 70989 48400 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE ALVOCIDIB ALVOCIDIB 70990 48401 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DS-8201a TRASTUZUMAB DERUXTECAN 27026201 70991 48402 POLK 51426 DNA REPAIR, ENZYME NSC-22225 CHEMBL462314 70992 48403 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CHEMBL2068724 ACAMPROSATE CALCIUM 70993 48404 GMNN 51053 DRUGGABLE GENOME EUPAROTIN ACETATE EUPAROTIN ACETATE 70994 48405 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 53801036 70995 48406 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101282 70996 48407 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PWT33597 70997 48408 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME AMPICILLIN AMPICILLIN 70998 48409 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TILIQUINOL TILIQUINOL 70999 48410 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651738 71000 48411 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE PIPLARTINE PIPLARTINE 71002 48412 BAZ2B 29994 NA BI-87E7 CHEMBL523200 71004 48413 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PKI-179 PKI-179 20797855 71007 48414 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 187051793 GIVINOSTAT 71008 48415 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL289351 FOSBRETABULIN DISODIUM 71010 48416 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TACROLIMUS TACROLIMUS 71011 48417 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TELMISARTAN TELMISARTAN 71013 48418 KDM1B 221656 DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING, ENZYME PMID27019002-Compound-46 71014 48419 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ISOBOLDINE ISOBOLDINE 71015 48420 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME DOVITINIB DOVITINIB 71022 48421 SAE1 10055 ENZYME, DRUGGABLE GENOME LOBARIC ACID LOBARIC ACID 71023 48422 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL598797 CUDC-101 71024 48423 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE E7090 E-7090 18552176,27535969 71025 48424 KEAP1 9817 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING 348353669 71026 48425 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 LINOPIRDINE LINOPIRDINE 71030 48426 ALOX15 246 ENZYME, DRUGGABLE GENOME KOPARIN KOPARIN 71032 48427 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 340590257 71034 48428 AOC3 8639 CELL SURFACE, DRUGGABLE GENOME, ENZYME Hydralazine HYDRALAZINE 71035 48429 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PHENANTHROLINE PHENANTHROLINE 71036 48430 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME TYRPHOSTIN 47 TYRPHOSTIN 47 71038 48431 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Hydroxy amidine derivative 2 71043 48432 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 71044 48433 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE DNDI1417467 CHEMBL1997335 71045 48434 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Dasatinib DASATINIB 26855149,27231123,28280091,27222538,26725216 71046 48435 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LY-2623091 LY2623091 71047 48436 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LYCOPENE LYCOPENE 10806309 71048 48437 RABEP1 9135 CLINICALLY ACTIONABLE, GROWTH FACTOR clozapine CLOZAPINE 28694205 71049 48438 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR N/A 71051 48439 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 6-HYDROXYMELATONIN CHEMBL127421 71052 48440 PABPC1 26986 NA SJ000040829 CHEMBL589711 71057 48441 APOE 348 DRUGGABLE GENOME acenocoumarol ACENOCOUMAROL 29432897 71058 48442 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1611 PHENYTOIN SODIUM 71060 48443 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR BAY 86-5044 71061 48444 PDE10A 10846 ENZYME, DRUGGABLE GENOME RG7203 71063 48445 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME N/A 71064 48446 HTT 3064 DRUGGABLE GENOME RAC-GONIOTHALAMIN CHEMBL1170485 71065 48447 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2104986 TEDATIOXETINE 71067 48448 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR IBUPROFEN IBUPROFEN 15131590 71071 48449 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CID 4101591 CHEMBL428789 71072 48450 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME RG7813 CERGUTUZUMAB AMUNALEUKIN 71074 48451 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING T-5224 71076 48452 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME GEMCITABINE GEMCITABINE 23741071 71077 48453 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1230607 PHA-793887 71078 48454 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME PURPUROGALLIN PURPUROGALLIN 71079 48455 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 363894208 ILORASERTIB 71081 48456 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME SIRTINOL SIRTINOL 23189967 71083 48457 RICTOR 253260 CLINICALLY ACTIONABLE VISTUSERTIB VISTUSERTIB 28028034 71084 48458 MBP 4155 CELL SURFACE PREDNISONE PREDNISONE 10612091 71086 48459 MAPT 4137 DRUGGABLE GENOME CHELERYTHRINE CHELERYTHRINE 71088 48460 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE CHEMBL1255944 71089 48461 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TRIMETHOPRIM TRIMETHOPRIM 22931300 71090 48462 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Ethynodiol Diacetate 71091 48463 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417434 CHEMBL394883 71092 48464 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CLAZOSENTAN CLAZOSENTAN 71093 48465 ARRB2 409 ION CHANNEL, G PROTEIN COUPLED RECEPTOR methamphetamine METHAMPHETAMINE 17233643 71095 48466 PRKG1 5592 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME CENISERTIB CENISERTIB 71096 48467 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME MINAPRINE MINAPRINE 71099 48468 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CAPSAZEPINE CAPSAZEPINE 71101 48469 MAPK7 5598 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 249565737 71103 48470 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Idelalisib IDELALISIB 26137449 71104 48471 ATXN2 6311 NA TEGASEROD MALEATE TEGASEROD MALEATE 71105 48472 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32e 71106 48473 CMKLR1 1240 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 354702257 71107 48474 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 405560328 71108 48475 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774824-Compound-Figure6Example12 71110 48476 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER curcumin CURCUMIN 71111 48477 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ALPHA-METHYL-P-TYROSINE METYROSINE 16390493 71113 48478 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-25 71114 48479 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR CHINESE HERBS 15768879 71115 48480 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 178100441 CHEMBL592652 71116 48481 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ILORASERTIB ILORASERTIB 71118 48482 DDO 8528 DRUGGABLE GENOME 5-AMINONICOTINIC ACID CHEMBL1491941 26322531 71119 48483 RORB 6096 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, KINASE agonist,antagonist 135651435 TRETINOIN 71120 48484 RALA 5898 CELL SURFACE VITAMIN E 16861802 71123 48485 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER temsirolimus TEMSIROLIMUS 28676933 71124 48486 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE CORTICOSTEROIDS 15895680 71125 48487 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor GSK2126458 OMIPALISIB 71126 48488 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE HEMATOXYLIN HEMATOXYLIN 71127 48489 PSMD1 5707 NA BORTEZOMIB BORTEZOMIB 71129 48490 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CHEMBL2109263 ING-1 71130 48491 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PIOGLITAZONE PIOGLITAZONE 71131 48492 CXCL8 3576 DRUGGABLE GENOME TALC TALC 17000556 71133 48493 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ALPHA,BETA-DEHYDROCURVULARIN CHEMBL482050 71134 48494 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178103001 ARGATROBAN 71136 48495 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME sparteine SPARTEINE 8563771,8287064,1844820,8946471,10471060,9241659,15618746,8530011,17001296,9089660,9511177,8655150,18784265,7845481,2211621,17460029 71139 48496 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 178103531 NANDROLONE 71143 48497 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (-)-THYSANONE CHEMBL596082 19783445 71144 48498 ATXN2 6311 NA SAQUINAVIR SAQUINAVIR 71145 48499 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE VX-970 BERZOSERTIB 28148839 71147 48500 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MMV000704 CHEMBL582478 71148 48501 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE GNF-PF-2301 CHEMBL578061 71153 48502 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHALCONE CHALCONE 71155 48503 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 2,7-BIS[2-(DIMETHYLAMINO)ACETAMIDO]ANTHRAQUINONE CHEMBL494283 24094433 71156 48504 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200896 DINOPROST TROMETHAMINE 71157 48505 CD14 929 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME LOVASTATIN LOVASTATIN 7506029 71158 48506 PYGB 5834 DRUGGABLE GENOME, ENZYME PSN357 71159 48507 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER BRECANAVIR BRECANAVIR 17664327 71162 48508 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist 178100901 71163 48509 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE GENTIAN VIOLET GENTIAN VIOLET 71165 48510 TDO2 6999 ENZYME, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 1 71166 48511 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME WEHI-539 27974663 71168 48512 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-216763 SB-216763 71169 48513 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME GNF-PF-1947 CHEMBL585591 71170 48514 PDE3A 5139 ENZYME, DRUGGABLE GENOME SDZ-MKS-492 71171 48515 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE volatile anesthetics 30136624 71172 48516 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Pyrrolo[2,3-d]pyrimidine derivative 10 71173 48517 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PH-797804 PH-797804 71174 48518 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE VANDETANIB VANDETANIB 71175 48519 HSPA8 3312 TUMOR SUPPRESSOR BUPIVACAINE BUPIVACAINE 12791605 71177 48520 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME DOXYCYCLINE DOXYCYCLINE 19258275 71179 48521 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 178102331 71180 48522 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545077 MK-1496 71182 48523 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME OXIDOPAMINE OXIDOPAMINE 71183 48524 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME BORTEZOMIB BORTEZOMIB 71184 48525 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ALISERTIB ALISERTIB 71185 48526 E2F1 1869 TRANSCRIPTION FACTOR NICOTINE NICOTINE 16601104 71186 48527 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE DIPIVEFRIN HYDROCHLORIDE DIPIVEFRIN HYDROCHLORIDE 71187 48528 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE BX-795 BX-795 71188 48529 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PLX7486 71189 48530 PTCH1 5727 CLINICALLY ACTIONABLE, TRANSPORTER Sonidegib SONIDEGIB 71190 48531 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR HOMIDIUM BROMIDE HOMIDIUM BROMIDE 71192 48532 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32j 71193 48533 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PIRENZEPINE PIRENZEPINE 71194 48534 GMNN 51053 DRUGGABLE GENOME VIDARABINE VIDARABINE 71195 48535 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 1,4,5,8-TETRAAMINO-ANTHRAQUINONE CHEMBL87568 71197 48536 ATAD5 79915 NA TCMDC-124573 CHEMBL525826 71198 48537 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-8186 CHEMBL122355 71201 48538 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Alpelisib ALPELISIB 71203 48539 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR L-DOPA LEVODOPA 9458818 71205 48540 ALOX15 246 ENZYME, DRUGGABLE GENOME 3-METHOXYCATECHOL 3-METHOXYCATECHOL 71206 48541 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ARABINOFURANOSYLCYTOSINE 8509220 71207 48542 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 71208 48543 CDC25C 995 KINASE, PROTEIN PHOSPHATASE, DRUGGABLE GENOME WITHAFERIN A WITHAFERIN A 24079846 71210 48544 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ADAPALENE ADAPALENE 71211 48545 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565738 71213 48546 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NALOXONE HYDROCHLORIDE NALOXONE HYDROCHLORIDE 71214 48547 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME Arsenic compounds 16479312 71215 48548 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PANOBINOSTAT PANOBINOSTAT 24694055 71218 48549 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ASCORBIC ACID 18091746 71219 48550 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MANGOSTIN MANGOSTIN 26508549 71221 48551 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE ALISERTIB ALISERTIB 71222 48552 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649762 71223 48553 SMPD1 6609 ENZYME, DRUGGABLE GENOME ETIDRONIC ACID ETIDRONIC ACID 71225 48554 BLVRB 645 ENZYME methylene blue 23913015 71226 48555 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist 135651056 71227 48556 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 71228 48557 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor BGJ398 INFIGRATINIB 71229 48558 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-1030058A GSK-1030058A 71230 48559 F13A1 2162 DRUGGABLE GENOME, ENZYME PMID26560530-Compound-13 71231 48560 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE dicumarol DICUMAROL 71232 48561 TUBA3D 113457 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 71233 48562 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565832 71234 48563 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE MM-151 71235 48564 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OXYQUINOLINE SULFATE OXYQUINOLINE SULFATE 71238 48565 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-37 71239 48566 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200875 FLAVOXATE HYDROCHLORIDE 71240 48567 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GERONTOXANTHONE H GERONTOXANTHONE H 71241 48568 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME Milademetan Tosylate 71243 48569 BAZ2B 29994 NA CRYPTOTANSHINONE CRYPTOTANSHINONE 71244 48570 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 6 71246 48571 TNFRSF9 3604 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1743085 URELUMAB 71247 48572 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Fosfestrol DIETHYLSTILBESTROL DIPHOSPHATE 71248 48573 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE PACLITAXEL PACLITAXEL 23390248 71249 48574 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1201535 PHENYLPROPANOLAMINE POLISTIREX 71252 48575 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200437 QUINIDINE GLUCONATE 71253 48576 PLAT 5327 ENZYME, DRUGGABLE GENOME, PROTEASE, CELL SURFACE inhibitor CHEMBL1046 AMINOCAPROIC ACID 71254 48577 EBP 10682 DRUGGABLE GENOME, ENZYME SR-31747 71255 48578 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE inhibitor 135651334 71256 48579 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652589 71257 48580 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME PHENAZOPYRIDINE HYDROCHLORIDE PHENAZOPYRIDINE HYDROCHLORIDE 71258 48581 NOX4 50507 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 363894229 71261 48582 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 71262 48583 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME inhibitor 178103593 CHEMBL569864 71263 48584 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR ADRIAMYCIN ADRIAMYCIN 7581027 71265 48585 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CPI-1205 CPI-1205 71266 48586 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME agonist 135651597 71269 48587 PSMA2 5683 DRUGGABLE GENOME, PROTEASE inhibitor CARFILZOMIB CARFILZOMIB 71273 48588 TYMSOS 494514 NA irinotecan IRINOTECAN 71275 48589 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE DOVITINIB DOVITINIB 71277 48590 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL1201461 DEXTROMETHORPHAN POLISTIREX 71279 48591 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100707 71280 48592 PAK6 56924 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 310264722 71281 48593 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER chlorpromazine CHLORPROMAZINE 71282 48594 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE GW441756X GW441756X 71283 48595 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 2',4'-DIHYDROXYCHALCONE 2',4'-DIHYDROXYCHALCONE 71284 48596 RGS4 5999 DRUGGABLE GENOME GW7647 GW7647 71285 48597 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PAMICOGREL PAMICOGREL 71286 48598 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME N-METHYL-N-NITROSOUREA 9197527 71287 48599 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist CHEMBL1200801 HISTAMINE PHOSPHATE 71288 48600 PGAP6 58986 NA fentanyl FENTANYL 29207912 71295 48601 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SNS-032 BMS-387032 71296 48602 PCNA 5111 NA PENTOXIFYLLINE PENTOXIFYLLINE 10707869 71297 48603 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Ribociclib RIBOCICLIB 28351928 71298 48604 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL2108508 INTERFERON ALFA-2A 71300 48605 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BCMA-UCART 71301 48606 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL blocker 178100875 PICROTOXIN 71303 48607 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650648 71305 48608 PDE4B 5142 DRUGGABLE GENOME, ENZYME DYPHYLLINE DYPHYLLINE 71307 48609 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MK-8033 MK-8033 71308 48610 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CATECHOL CATECHOL 71310 48611 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Cisplatin CISPLATIN 71312 48612 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PRX-321 PRX-321 71313 48613 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GERONTOXANTHONE I GERONTOXANTHONE I 71315 48614 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8669361, 107 71316 48615 SLC16A1 6566 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 384403683 71319 48616 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ETOPOSIDE ETOPOSIDE 22931300 71320 48617 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor KX2-391 KX2-391 71323 48618 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CYC-116 CYC-116 71324 48619 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL antagonist 135650889 71325 48620 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR MEK164 71326 48621 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING TRICHOSTATIN TRICHOSTATIN 21055848,16921367,19966789,19385600 71327 48622 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME INGENOL MEBUTATE 71328 48623 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME PROTOAPIGENONE PROTOAPIGENONE 71329 48624 TSPYL2 64061 NA SODIUM BUTYRATE 12619135 71331 48625 IL1B 3553 KINASE, DRUGGABLE GENOME Gallium nitrate 71332 48626 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME DISULFIRAM DISULFIRAM 71334 48627 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL2105719 DACOMITINIB 71336 48628 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE INCB028060 71338 48629 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME IL-11 OPRELVEKIN 14734714 71340 48630 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ROEMERINE ROEMERINE 71342 48631 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE disulfiram DISULFIRAM 23335901 71343 48632 CYP27B1 1594 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TRICHOSTATIN A 15860259 71344 48633 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE unspecified EGFR antibody 27196767 71346 48634 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE NOVOBIOCIN NOVOBIOCIN 3528175 71347 48635 DGAT1 8694 ENZYME, DRUGGABLE GENOME Lactam derivative 3 71348 48636 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antibody 315661255 OLARATUMAB 71349 48637 AQP9 366 ION CHANNEL inhibitor 178101102 PHLORETIN 71350 48638 SLC5A3 6526 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSPORTER inhibitor 178101467 PHLORIZIN 71351 48639 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PAPAVERINE PAPAVERINE 71352 48640 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PLUKENETIONE A PLUKENETIONE A 18951805 71354 48641 PSMB9 5698 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CARFILZOMIB CARFILZOMIB 71356 48642 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME bortezomib BORTEZOMIB 21228734 71359 48643 MAPT 4137 DRUGGABLE GENOME ARUNDINE ARUNDINE 71360 48644 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE Autologous T-cell therapy 71362 48645 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME THIOMERSAL THIMEROSAL 71363 48646 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE SNS-314 SNS-314 71366 48647 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING COUMESTROL COUMESTROL 71368 48648 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME CLEMASTINE CLEMASTINE 71369 48649 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651540 71370 48650 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20158969342C84 71371 48651 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME AST-487 AST-487 71372 48652 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ERBSTATIN ERBSTATIN 71373 48653 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER TESMILIFENE TESMILIFENE 71374 48654 ATAD5 79915 NA 4'-METHOXY-AURONE 4'-METHOXY-AURONE 71375 48655 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Sulfonamide derivative 6 71377 48656 BAZ2B 29994 NA THIORIDAZINE HYDROCHLORIDE THIORIDAZINE HYDROCHLORIDE 71378 48657 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR LOMOFUNGIN LOMOFUNGIN 71380 48658 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650457 71381 48659 POLK 51426 DNA REPAIR, ENZYME CEPHALOTHIN CEPHALOTHIN 71382 48660 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ALDRIN ALDRIN 71383 48661 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR NELFINAVIR NELFINAVIR 15388451 71384 48662 FBXW7 55294 DNA REPAIR, CLINICALLY ACTIONABLE Belinostat BELINOSTAT 23274910 71385 48663 SMN2 6607 DRUGGABLE GENOME AG-494 CHEMBL56731 71386 48664 MAOA 4128 DRUGGABLE GENOME, ENZYME NAPHTHOQUINONE NAPHTHOQUINONE 22071524 71387 48665 TUBA3C 7278 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 71388 48666 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Palifermin PALIFERMIN 71391 48667 TNFRSF1B 7133 DRUGGABLE GENOME 178101757 71392 48668 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME RG7828 MOSUNETUZUMAB 71394 48669 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SOTRASTAURIN SOTRASTAURIN 71396 48670 CBL 867 KINASE, ENZYME, CLINICALLY ACTIONABLE TCDD 9918770 71397 48671 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE CALYCOSIN CALYCOSIN 71398 48672 CBX1 10951 NA FPL-64176 CHEMBL93655 71400 48673 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28270010-Compound-Figure5-3 71401 48674 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE alpelisib ALPELISIB 71402 48675 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist CHEMBL1200757 PANCURONIUM BROMIDE 71404 48676 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545264 LY-2874455 71405 48677 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME SLAZINIC ACID SLAZINIC ACID 71407 48678 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 252827411 71408 48679 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GALUTEOLIN GALUTEOLIN 71409 48680 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL2180604 TAK-593 71410 48681 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 310264754 OMIPALISIB 71411 48682 POLI 11201 DNA REPAIR GNF-PF-4418 CHEMBL604321 71412 48683 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MEPINDOLOL MEPINDOLOL 2903243 71413 48684 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER AZT ZIDOVUDINE 15456083 71415 48685 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE MIRTAZAPINE MIRTAZAPINE 16002093 71416 48686 MYO9B 4650 NA NIFEDIPINE NIFEDIPINE 3161480 71417 48687 APOE 348 DRUGGABLE GENOME LUTEIN LUTEIN 11413081 71418 48688 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1752 DYPHYLLINE 71420 48689 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650113 CLOPROSTENOL 71421 48690 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SHP2 INHIBITOR RMC-4630 31776128 71422 48691 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE oxycodone OXYCODONE 18695978,21209234 71424 48692 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ALKS 37 71425 48693 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME UH-301 CHEMBL22778 71426 48694 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178103519 71427 48695 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CEPHALOCHROMIN CEPHALOCHROMIN 71428 48696 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-125556 CHEMBL587092 71430 48697 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Doxil DOXIL 21216929 71431 48698 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME TRIDIHEXETHYL TRIDIHEXETHYL 71434 48699 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PF-562271 PF-00562271 71435 48700 CDK12 51755 KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR, SERINE THREONINE KINASE inhibitor CHEMBL3544942 RONICICLIB 71437 48701 MT-RNR1 4549 KINASE kanamycin KANAMYCIN 18830133,16875663,9164619,19682603,16631122,21495045,16458854,12031626,16375862,9831149,17637808,22475488,11857751,27397648,9779807,7689389,20111055,9111378,27427311,17698030,11313749,20416460,16168391,24703164,9950117,21504270,11174059,8285309,18790089,15917167,20353758,16955413,16380089,14699607,17999439,14755216,17341440,19376484,15708009,25515069,15555598,11079536,17434445 71439 48702 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE cabozantinib CABOZANTINIB 24205792,25836719,27777285 71440 48703 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178102319 LAPATINIB 71443 48704 SMN1 6606 DRUGGABLE GENOME 7-METHOXYISOFLAVONE CHEMBL563919 71444 48705 MAP2K6 5608 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE, TUMOR SUPPRESSOR inhibitor PD 0325901 71445 48706 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR SCRIPTAID SCRIPTAID 19966789 71446 48707 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Palbociclib/ribociclib analog 1 71447 48708 SLC9A3 6550 DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE, EXCHANGER ALBUMIN ALBUMIN HUMAN 11251045,11698229 71448 48709 ATXN2 6311 NA METITEPINE METITEPINE 71451 48710 GUSB 2990 DRUGGABLE GENOME, ENZYME Vestronidase alfa 71453 48711 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NCG-C00094408-01 CHEMBL1256885 71454 48712 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME CHEMBL395091 ESKETAMINE 71455 48713 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 404859134 71457 48714 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102265 71458 48715 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Emibetuzumab EMIBETUZUMAB 71460 48716 MAPT 4137 DRUGGABLE GENOME PHENOTHIAZINE PHENOTHIAZINE 71461 48717 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL501867 VINCRISTINE SULFATE 71462 48718 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MESOTRIONE MESOTRIONE 71463 48719 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Flibanserin FLIBANSERIN 71464 48720 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 6,4'-DIHYDROXYFLAVONE CHEMBL484663 71465 48721 EIF2AK4 440275 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor HESPERADIN HESPERADIN 19035792 71466 48722 IL1B 3553 KINASE, DRUGGABLE GENOME pravastatin PRAVASTATIN 14515062 71468 48723 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DOCOSATETRA-7Z,10Z,13Z,16Z-ENOYL ETHANOLAMIDE CHEMBL321585 71472 48724 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE CALCITRIOL CALCITRIOL 8490200,15598784 71473 48725 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CHRYSIN CHRYSIN 71474 48726 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Fludrocortisone FLUDROCORTISONE 71476 48727 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 363894222 PUQUITINIB 71478 48728 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME GW843682X GW843682X 71480 48729 ARID1A 8289 CLINICALLY ACTIONABLE ATEZOLIZUMAB ATEZOLIZUMAB 29736026 71483 48730 KDM4A 9682 DRUGGABLE GENOME, ENZYME DEPHOSTATIN DEPHOSTATIN 71486 48731 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178101087 71487 48732 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Epidermal growth factor 71488 48733 POLK 51426 DNA REPAIR, ENZYME MONTELUKAST SODIUM MONTELUKAST SODIUM 71489 48734 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE MEDROXYPROGESTERONE MEDROXYPROGESTERONE ACETATE 10764452 71492 48735 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 178103352 IDELALISIB 71496 48736 ABL2 27 KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME inhibitor 363894211 PEXMETINIB 71497 48737 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GLYBURIDE GLYBURIDE 71498 48738 POLI 11201 DNA REPAIR CEFOTIAM HYDROCHLORIDE CEFOTIAM HYDROCHLORIDE 71499 48739 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-11 71500 48740 GALNS 2588 DRUGGABLE GENOME, ENZYME Elosulfase 71501 48741 MALAT1 378938 NA Platinum compounds 26729200 71502 48742 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Camptothecin CAMPTOTHECIN 24042735,25688157 71503 48743 RAB9A 9367 ENZYME, DRUGGABLE GENOME BIOCHANIN BIOCHANIN 71504 48744 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GANGALEOIDIN GANGALEOIDIN 71506 48745 MYO9B 4650 NA DIBUCAINE DIBUCAINE 7631738 71507 48746 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PYRIDABEN PYRIDABEN 71508 48747 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CVBT-141B 71509 48748 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ranolazine RANOLAZINE 71510 48749 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CANDESARTAN CILEXETIL CANDESARTAN CILEXETIL 71512 48750 GMNN 51053 DRUGGABLE GENOME DNDI1417905 CHEMBL1449731 71514 48751 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MLN-8054 MLN-8054 71515 48752 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-62 71516 48753 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR modulator CHEMBL1716091 SDX-101 71517 48754 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CART123 cells 71518 48755 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME AZ628 26351322,27523909 71520 48756 FECH 2235 ENZYME Cholic Acid 71523 48757 POLK 51426 DNA REPAIR, ENZYME NSC-9037 CHEMBL1451216 71525 48758 C3 718 PROTEASE INHIBITOR, DRUGGABLE GENOME, CELL SURFACE POT-4 71526 48759 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Cladribine CLADRIBINE 71527 48760 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE hydroxychloroquine HYDROXYCHLOROQUINE 71528 48761 EEF2 1938 DRUGGABLE GENOME, KINASE CYCLOHEXIMIDE CYCLOHEXIMIDE 20118940 71529 48762 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PF-4691502 PF-04691502 71530 48763 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR INTERFERON GAMMA 9231818 71531 48764 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102108 METHADONE 71533 48765 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Quinoline derivative 14 71534 48766 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Perphenazine PERPHENAZINE 71535 48767 TOP2B 7155 DRUGGABLE GENOME, ENZYME Quinolones 71536 48768 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651802 71537 48769 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PROCATEROL PROCATEROL 71538 48770 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2008079988 71539 48771 COMT 1312 DRUGGABLE GENOME, ENZYME valproic acid 71541 48772 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-3641 CHEMBL599098 71542 48773 MMP7 4316 NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, ENZYME, PROTEASE Marimastat MARIMASTAT 71543 48774 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR DOVITINIB DOVITINIB 71545 48775 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME PROTOPORPHYRIN PROTOPORPHYRIN 71546 48776 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PF-562271 PF-00562271 71547 48777 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SURAMIN SURAMIN 9874182 71548 48778 BUB1 699 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME SCHEMBL16365841 71549 48779 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME METHYLNITROSOUREA 9192819 71550 48780 GMNN 51053 DRUGGABLE GENOME ETHYL NITRITE [SPIRIT] ETHYL NITRITE [SPIRIT] 71552 48781 GLS 2744 ENZYME MESALAMINE MESALAMINE 71554 48782 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Dinoprostone DINOPROSTONE 71555 48783 IL1B 3553 KINASE, DRUGGABLE GENOME ETRETIN ACITRETIN 2954576 71556 48784 MYO9B 4650 NA BCM MANNOMUSTINE 6837263 71557 48785 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BUSULFAN BUSULFAN 15779864 71559 48786 MIF 4282 DRUGGABLE GENOME, CELL SURFACE ISO-1 71560 48787 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CARTEOLOL CARTEOLOL 2903243 71562 48788 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200791 OXYMETAZOLINE HYDROCHLORIDE 71563 48789 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Melogliptin 71564 48790 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME TRIAZENE COMPOUNDS 16412662 71565 48791 ABCA1 19 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Probucol PROBUCOL 71566 48792 NOTCH2 4853 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE Tarextumab TAREXTUMAB 71567 48793 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651030 71570 48794 EPHB4 2050 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 249565821 71574 48795 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL274654 ORANTINIB 71575 48796 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135650063 CERIVASTATIN 71576 48797 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIAMIDE DIAMIDE 71579 48798 VKORC1 79001 DRUGGABLE GENOME, ENZYME warfarin WARFARIN 20072124,21174619,21326313,26445138,14765195,18752379,21635147,24029542,25042728,23602689,16815312,28262345,20833980,17110455,22534826,17124101,17042764,21383771,22528326,29781049,24474498,15358623,25594941,16611310,27581200,27262824,25026456,28382498,21318593,17015052,16141794,18466099,25519826,25312789,19875892,16580898,17989110,16432637,31653973,19135231,16888441,27488176,21900891,19387626,22248286,17189218,22349464,9684798,17456829,16983400,19745563,17391071,26257249,31395958,20203262,21185752,18574025,22854539,29577257,20615525,26219158,17031720,26433837,24728385,22990331,28429387,22616655,23061746,16270629,25769357,18240904,23183958,17510308,21981797,20339978,19874474,18030307,15888487,26223945,19582440,15938684,17049586,20410877,15883587,21148049,17111199,26777610,25244877,28689179,20421126,25001883,16960144,15947090,16821005,17329985,25084205,18950464,11926893,12931134,20833655,29396738,24919870,22075505,19177029,20585834,19794411,22571356,19297219,18698879,16890578,18690342,23774101,22676192,23159229,22010099,27121899,25521356,16847429,22592842,24019055,23208322,14676821,14765194,23104259,23949431,19077919,28049362,16493479,25989350,29054760,29432897,23423913,24330000,21176721,16611750,28033245,20386359,17112295,15865594,17906972,16815313,15930419,16676068,21273734,29298995,22040439,15790782,11127854,22549502,17161452,18234403,21110192,15597574,23279643,23932037,18542936 71581 48799 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1059 PREGABALIN 71583 48800 POLD1 5424 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME inhibitor CHEMBL803 CYTARABINE 71584 48801 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TCMDC-125653 CHEMBL580918 71585 48802 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649811 71587 48803 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL14 CARBACHOL 71588 48804 TRPM6 140803 ION CHANNEL, DRUGGABLE GENOME, ENZYME, TRANSPORTER, KINASE, SERINE THREONINE KINASE blocker 135652731 71591 48805 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NOREPINEPHRINE NOREPINEPHRINE 71595 48806 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALSTERPAULLONE ALSTERPAULLONE 71597 48807 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BUDESONIDE BUDESONIDE 22931300 71600 48808 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545368 PANOBINOSTAT LACTATE 71601 48809 KLF5 688 TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CID 838877 CHEMBL405317 71602 48810 APC 324 CLINICALLY ACTIONABLE G007-LK 28179481,23539443 71603 48811 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL551466 ACLIDINIUM BROMIDE 71605 48812 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR HGS1029 71606 48813 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200545 DIFLORASONE DIACETATE 71607 48814 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE NIRAPARIB NIRAPARIB 71608 48815 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE pindolol PINDOLOL 71609 48816 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BMS-345541 BMS-345541 71610 48817 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 1-AMINOCYCLOPROPANE CARBOXYLIC ACID 1-AMINOCYCLOPROPANE CARBOXYLIC ACID 71613 48818 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE TOLONIUM CHLORIDE TOLONIUM CHLORIDE 71614 48819 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor LINSITINIB LINSITINIB 71616 48820 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[4,3-c]pyridine derivative 1 71617 48821 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor ENZALUTAMIDE ENZALUTAMIDE 71618 48822 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME NICARDIPINE NICARDIPINE 71621 48823 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE vandetanib VANDETANIB 18681783,14990633,16467544,16377102,14990632,18784101,16257339,18003960,23022519,11255078,19339720,18316547,12648464,22594511 71622 48824 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR (S)-ROSCOVITINE (S)-ROSCOVITINE 71623 48825 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ARI-3037MO 71624 48826 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor NELFINAVIR NELFINAVIR 71626 48827 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 363894180 71627 48828 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROROXAN PROROXAN 71628 48829 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL541758 FASITIBANT CHLORIDE 71629 48830 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME RALOXIFENE RALOXIFENE 71630 48831 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BI-847325 27496137,25873592 71631 48832 PSMD3 5709 NA inhibitor CHEMBL325041 BORTEZOMIB 71632 48833 FABP5 2171 NUCLEAR HORMONE RECEPTOR inhibitor 252827455 71633 48834 METAP2 10988 ENZYME, DRUGGABLE GENOME, KINASE, PROTEASE inhibitor 178103100 71634 48835 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME activator 178102130 GABAPENTIN 71635 48836 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TOCILIZUMAB TOCILIZUMAB 71636 48837 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE naltrexone NALTREXONE 32020635,31961981,25715171,22515274,25760804,25410894,31206155,21946895,16960700 71638 48838 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Diethylstilbestrol DIETHYLSTILBESTROL 71639 48839 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME amoxicillin AMOXICILLIN 20800921,10535882,30664875 71641 48840 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1938400 PF-03715455 71642 48841 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ANDROSTENEDIONE ANDROSTENEDIONE 71643 48842 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor AZD6244 SELUMETINIB 71644 48843 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417086 CHEMBL1224755 71646 48844 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME VATALANIB VATALANIB 71647 48845 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 178102669 71648 48846 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE UROKINASE UROKINASE 71649 48847 TSPO 706 DRUGGABLE GENOME Triazolam TRIAZOLAM 71651 48848 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SORAFENIB SORAFENIB 26318998 71652 48849 BMP1 649 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 252166763 71654 48850 ALDH3A2 224 DRUGGABLE GENOME, ENZYME Disulfiram DISULFIRAM 71655 48851 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE MIDOSTAURIN MIDOSTAURIN 71657 48852 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NSC-180246 CHEMBL484640 71659 48853 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIS(2,3-DIBROMOPROPYL)PHOSPHATE TRIS(2,3-DIBROMOPROPYL)PHOSPHATE 71660 48854 MUC16 94025 DRUGGABLE GENOME SODIUM BUTYRATE 1720110,1645702 71661 48855 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CMA-676 GEMTUZUMAB OZOGAMICIN 11986941 71666 48856 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PF-562271 PF-00562271 71668 48857 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NANDROLONE DECANOATE NANDROLONE DECANOATE 71669 48858 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL1201752 IXABEPILONE 71670 48859 APC 324 CLINICALLY ACTIONABLE Erlotinib ERLOTINIB 17909047 71672 48860 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE Elexacaftor ELEXACAFTOR 71674 48861 ATAD5 79915 NA GNF-PF-5007 CHEMBL1989853 71675 48862 RACGAP1 29127 NA GNF-PF-2936 CHEMBL582503 71676 48863 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE cyclophosphamide CYCLOPHOSPHAMIDE 22016816 71677 48864 CA2 760 DRUGGABLE GENOME, ENZYME CG-100649 POLMACOXIB 71678 48865 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 249565801 71680 48866 GSTM1 2944 DRUGGABLE GENOME, ENZYME radiotherapy 71681 48867 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR anastrozole ANASTROZOLE 71682 48868 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GNF-PF-5576 CHEMBL599896 71683 48869 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650818 PHENTOLAMINE 71685 48870 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DESIPRAMINE DESIPRAMINE 71686 48871 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor XL647 TESEVATINIB 71688 48872 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545264 LY-2874455 71689 48873 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (S)-PROMETHAZINE (S)-PROMETHAZINE 71692 48874 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 249565857 71694 48875 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650453 KETANSERIN 71696 48876 GSTO1 9446 ENZYME, DRUGGABLE GENOME inhibitor 405067313 71697 48877 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-5242 CHEMBL600107 71698 48878 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DRONEDARONE DRONEDARONE 71699 48879 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TRIAMCINOLONE TRIAMCINOLONE 22931300 71700 48880 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LOVASTATIN LOVASTATIN 71701 48881 ATF2 1386 TRANSCRIPTION FACTOR H2O2 9773928 71702 48882 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545385 WX-037 71705 48883 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 28 71707 48884 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE etanercept ETANERCEPT 24048425,27044681 71708 48885 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Carboxamide derivative 8 71709 48886 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 sulfadiazine SULFADIAZINE 9187528 71710 48887 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER SODIUM BUTYRATE 11587480 71711 48888 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME G-619 71712 48889 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE TEMOZOLOMIDE TEMOZOLOMIDE 23960094 71713 48890 H2AW 92815 NA GNRH GONADORELIN ACETATE 2544582,1963323 71716 48891 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE GELDANAMYCIN GELDANAMYCIN 12724357 71717 48892 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 IBUPROFEN IBUPROFEN 22931300 71718 48893 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AMI-408 26766589 71719 48894 SLAMF7 57823 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME antibody 252166573 ELOTUZUMAB 71722 48895 E2F1 1869 TRANSCRIPTION FACTOR MTX METHOTREXATE 14654896 71723 48896 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Carbamide derivative 8 71725 48897 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENSULIDE BENSULIDE 71727 48898 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Lorlatinib LORLATINIB 71728 48899 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-1000 CHEMBL600554 71729 48900 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor BMS-690514 BMS-690514 71730 48901 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Dasatinib DASATINIB 23242808,27222538,22649091 71732 48902 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PIPERTRAMINE PIPERTRAMINE 71733 48903 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651285 71734 48904 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BEXAROTENE BEXAROTENE 71735 48905 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ZAMIFENACIN ZAMIFENACIN 71736 48906 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE TYROSINE KINASE INHIBITOR 17539658 71739 48907 PSENEN 55851 DRUGGABLE GENOME IC261 IC261 20350806 71740 48908 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Tricyclic isoxazoloquinazoline derivative 2 71741 48909 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR IL-12 GENE 16525645 71742 48910 POLB 5423 DNA REPAIR, DRUGGABLE GENOME METHOTREXATE METHOTREXATE 71743 48911 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE OSI-632 OSI-632 71744 48912 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR IMATINIB IMATINIB 71745 48913 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PICTILISIB PICTILISIB 71746 48914 MAP2K5 5607 KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor GDC-0973 COBIMETINIB 71750 48915 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103745 DOXAZOSIN 71751 48916 EEF2K 29904 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 252827401 71752 48917 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 71753 48918 ALDH1A1 216 DRUGGABLE GENOME, ENZYME E1501 E1501 71755 48919 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME KC706 71756 48920 POLK 51426 DNA REPAIR, ENZYME CCG-63802 CHEMBL1476646 71757 48921 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PD-0166285 PD-0166285 71759 48922 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIPYRIDAMOLE DIPYRIDAMOLE 71761 48923 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DNDI1417941 CHEMBL2095095 71763 48924 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Six-membered heterocyclic benzamide derivative 2 71764 48925 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antibody VOLOCIXIMAB VOLOCIXIMAB 71765 48926 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-1399 CHEMBL578504 71769 48927 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-4 71770 48928 NOS1 4842 DRUGGABLE GENOME, ENZYME INTERLEUKIN-1 RECEPTOR ANTAGONIST 9206098 71772 48929 MAPT 4137 DRUGGABLE GENOME BETA-LAPACHONE LAPACHONE 71773 48930 STIM2 57620 DRUGGABLE GENOME AMINOGLYCOSIDE ANTIBIOTIC 17905723 71776 48931 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME NITAZOXANIDE NITAZOXANIDE 71777 48932 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2096646 AMINOSALICYLATE SODIUM 71779 48933 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHYL YELLOW METHYL YELLOW 71781 48934 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Brontictuzumab BRONTICTUZUMAB 23774673 71782 48935 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORQUINALDOL CHLORQUINALDOL 71783 48936 AKR1C1 1645 DRUGGABLE GENOME, ENZYME 3,5-DICHLOROSALICYLIC ACID CHEMBL449129 21414777 71784 48937 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER EPOTHILONE D EPOTHILONE D 24992153 71785 48938 COL1A2 1278 DRUGGABLE GENOME COLLAGENASE COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 71786 48939 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME AR-12 AR-12 71787 48940 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CL-976 CL-976 71788 48941 ALOX15 246 ENZYME, DRUGGABLE GENOME APIGENIN APIGENIN 71790 48942 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32j 71791 48943 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 249565710 71792 48944 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME halothane HALOTHANE 25989378,12411786,26951757,8828983,19919814,17710899,7829078,9334205,21965348,11063719,10823104,20681998,25611019,19648156,25256590,12220451,11668625,23736090,14500992,9066328,14641996,18945287,25960145,7889656,11575529,18212565,16284304,8602662,18306019,28326467,11928716,18502356,10352931,12151923,11525881,17122579,16917943,8220422,10700782,16163667,17226826,9389851,16732128,16835904,11448278,29101530,9450902,7547049,23628358,9543323,24361844,26994242,12208234,15448513,16621918,21455645,11553045,12124989,19020143,19191329,27918309,8220423,12059893,10612851,16732084,10793526,27382027,15108991,12709367,12123492,26381711,25268394,28063098,11493496,12434264,12411788,19685112,25735680,8902717,29608462,27663056,7751854,8012359,9520251,15731587,15210166,1510267,10888602,22030266,25466363,17483490,28403410,12237752,1774074,17081152,18564801,10484775,21282829,16244001,7586638,19191333,25086907,7633940,17667581,12883402,19346234,1354642,22415532 71793 48945 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NBQX NBQX 71795 48946 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 IMIPRAMINE IMIPRAMINE 22931300 71796 48947 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR MEGESTROL MEGESTROL 71797 48948 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 fentanyl FENTANYL 24469018 71799 48949 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL ESTAZOLAM ESTAZOLAM 71801 48950 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545089 IMD-0354 71803 48951 RGS4 5999 DRUGGABLE GENOME CAPSAZEPINE CAPSAZEPINE 71805 48952 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist,antagonist 135650608 MIFEPRISTONE 71806 48953 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 135649930 TAMIBAROTENE 71807 48954 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MACITENTAN MACITENTAN 71808 48955 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLORBROMURON CHLORBROMURON 71809 48956 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TIOTIDINE TIOTIDINE 71811 48957 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Venetoclax VENETOCLAX 27974663 71812 48958 ATXN2 6311 NA APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 71813 48959 PSMB6 5694 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor BORTEZOMIB BORTEZOMIB 71815 48960 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CIS-RESVERATROL CIS-RESVERATROL 71820 48961 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DSP-6952 71821 48962 HTT 3064 DRUGGABLE GENOME DNDI1417607 CHEMBL1588679 71822 48963 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-124356 CHEMBL22062 71823 48964 EIF2AK1 27102 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TCMDC-123956 CHEMBL534675 22153346 71824 48965 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIHYDREXIDINE DIHYDREXIDINE 71825 48966 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-43 71827 48967 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GANGLEOIDIN ACETATE GANGLEOIDIN ACETATE 71828 48968 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER INTERFERON ALPHA-2B 16001656 71830 48969 CYP24A1 1591 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME inhibitor 252827509 71831 48970 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1317721 CHEMBL1385558 71833 48971 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME L-733060 CHEMBL27006 71835 48972 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor ALVOCIDIB ALVOCIDIB 71837 48973 ALDH1A1 216 DRUGGABLE GENOME, ENZYME carboplatin CARBOPLATIN 18854779 71838 48974 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL ANAVEX 1-41 71839 48975 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SULISOBENZONE SULISOBENZONE 71842 48976 CCND2 894 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE LEE011 RIBOCICLIB 71843 48977 FAAH 2166 ENZYME, DRUGGABLE GENOME IW-6118 71844 48978 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565798 71846 48979 EPHB2 2048 KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 384403668 71847 48980 RAB9A 9367 ENZYME, DRUGGABLE GENOME SIB-1757 CHEMBL88553 71849 48981 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565844 71851 48982 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL3545026 FAMITINIB 71852 48983 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-4227 CHEMBL585654 71853 48984 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME CHRYSIN CHRYSIN 71855 48985 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GNF-PF-2301 CHEMBL578061 71857 48986 CA2 760 DRUGGABLE GENOME, ENZYME Sulfamylon SULFAMYLON 71859 48987 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE NADOLOL NADOLOL 2903243 71861 48988 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-NITROFLUORENE 2-NITROFLUORENE 71863 48989 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DEHYDROEPIANDROSTERONE ACETATE DEHYDROEPIANDROSTERONE ACETATE 71864 48990 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CHARTREUSIN CHARTREUSIN 71866 48991 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME 7-azaindole derivative 2 71867 48992 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652196 ICATIBANT 71869 48993 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME LANSOPRAZOLE LANSOPRAZOLE 17704577 71871 48994 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-52 CHEMBL601142 71872 48995 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GNF-PF-3537 CHEMBL601110 71873 48996 EGLN2 112398 ENZYME, DRUGGABLE GENOME inhibitor 252827454 71874 48997 HTT 3064 DRUGGABLE GENOME MMV085203 CHEMBL586031 71875 48998 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE CYC-116 CYC-116 71876 48999 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-1919 CHEMBL576409 71877 49000 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor ENMD-2076 ENMD-2076 71878 49001 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PHENTOLAMINE PHENTOLAMINE 71879 49002 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor MEK162 BINIMETINIB 71880 49003 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565814 71881 49004 ATAD5 79915 NA DISULFIRAM DISULFIRAM 71883 49005 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROCHLORPERAZINE PROCHLORPERAZINE 71884 49006 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 252827462 RITONAVIR 71885 49007 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME HEPARAN SULFATE 15797245 71889 49008 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME KENPAULLONE KENPAULLONE 71891 49009 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Metergolin 71892 49010 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 252166791 71893 49011 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GARCINONE E GARCINONE E 71894 49012 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 178103567 71895 49013 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 381118877 TOMIVOSERTIB 71898 49014 NOTCH2 4853 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE OMP-59R5 TAREXTUMAB 71901 49015 ALB 213 TRANSPORTER, DRUGGABLE GENOME Albumin Human 71902 49016 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3545204 QAF805 71906 49017 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ARACHIDONOYL DOPAMINE ARACHIDONOYL DOPAMINE 71908 49018 GPER1 2852 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR agonist 135649800 AFIMOXIFENE 71909 49019 NUDT15 55270 ENZYME, CLINICALLY ACTIONABLE azathioprine AZATHIOPRINE 27530327,26503813,28146264,27558924,30035323,25108385,29923122,27381176,26590936,27193222,30048756,26033531,27416873,26076924,27604507,26735160,27577869,30101994,27095468 71910 49020 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE BASIC FIBROBLAST GROWTH FACTOR 15924676 71911 49021 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME RIGOSERTIB RIGOSERTIB 71912 49022 RPS19 6223 NA DEXAMETHASONE DEXAMETHASONE 15755903 71913 49023 NDUFA11 126328 ENZYME inhibitor CHEMBL3545320 ME-344 71914 49024 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME Novolimus 71915 49025 ATXN2 6311 NA GNF-PF-1919 CHEMBL576409 71916 49026 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE METHYLCURCUMIN METHYLCURCUMIN 25753330 71918 49027 TAC1 6863 DRUGGABLE GENOME DIGOXIN DIGOXIN 1717629 71920 49028 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650728 71922 49029 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SJ000001516 CHEMBL592316 71923 49030 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 7-HYDROXYCHLORPROMAZINE 7-HYDROXYCHLORPROMAZINE 71925 49031 GMNN 51053 DRUGGABLE GENOME TCMDC-125814 CHEMBL533082 71928 49032 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LAPATINIB LAPATINIB 71930 49033 MAPT 4137 DRUGGABLE GENOME GRINIMIBINE GRINIMIBINE 71931 49034 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Aminoarylpyridine derivative 1 71933 49035 PCNA 5111 NA SUNSCREEN 17021352 71934 49036 WWOX 51741 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE TUMOR NECROSIS FACTOR 11058590 71935 49037 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE TOLFENAMIC ACID TOLFENAMIC ACID 71936 49038 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HYDROQUINONE HYDROQUINONE 71937 49039 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE BAY1187982 27543601 71940 49040 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1722209 TOLTERODINE TARTRATE 71941 49041 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE LEVORPHANOL LEVORPHANOL 71942 49042 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CRYPTOTANSHINONE CRYPTOTANSHINONE 71945 49043 GADD45A 1647 DNA REPAIR, TUMOR SUPPRESSOR, KINASE TROGLITAZONE TROGLITAZONE 15064713 71946 49044 DHFR 1719 DRUGGABLE GENOME, ENZYME TRIMETREXATE TRIMETREXATE 71947 49045 ENOSF1 55556 ENZYME ANTIVIRAL 12238529 71949 49046 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLORAZEPATE CLORAZEPIC ACID 71951 49047 H2AW 92815 NA VM-26 TENIPOSIDE 8620504 71952 49048 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR TCMDC-125603 CHEMBL528734 71953 49049 EED 8726 ENZYME, CLINICALLY ACTIONABLE inhibitor 336446911 71954 49050 ICMT 23463 DRUGGABLE GENOME, ENZYME SIMVASTATIN SIMVASTATIN 71955 49051 HMOX1 3162 ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE SUNITINIB SUNITINIB 26309414 71957 49052 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PERHEXILINE MALEATE PERHEXILINE MALEATE 71958 49053 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME OPIOID 10232386 71962 49054 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE EGF816 71964 49055 TBP 6908 TRANSCRIPTION FACTOR RETINOIC ACID 8413615 71966 49056 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR (E)-DIBENZYLIDENEACETONE CHEMBL17201 71968 49057 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme2WO2012/098065bottom 71969 49058 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Phenylpyrrolidinone derivative 2 71973 49059 POLK 51426 DNA REPAIR, ENZYME MK-886 CHEMBL29097 71976 49060 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME OTX-015 BIRABRESIB 71978 49061 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ALISERTIB ALISERTIB 71979 49062 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-68 71980 49063 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME LASSBIO-294 CHEMBL233194 71981 49064 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME APIGENIN APIGENIN 71982 49065 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME MIDAZOLAM MIDAZOLAM 22137933 71985 49066 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME ESCITALOPRAM ESCITALOPRAM 71988 49067 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METHOXAMINE METHOXAMINE 71992 49068 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ETHANOL ALCOHOL 1302037 71994 49069 TOP2B 7155 DRUGGABLE GENOME, ENZYME Fluoroquinolones 71995 49070 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 252166602 NANATINOSTAT 71996 49071 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE OXALIPLATIN OXALIPLATIN 71997 49072 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AG-537 CHEMBL67535 72000 49073 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME DIAZEPAM DIAZEPAM 72002 49074 MAPT 4137 DRUGGABLE GENOME PHENAZINE-2,3-DIAMINE CHEMBL274921 72003 49075 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000201788 CHEMBL602923 72004 49076 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Talotrexin TALOTREXIN 21301589 72006 49077 TNFRSF9 3604 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE Anti-CD137 72007 49078 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR Selective serotonin reuptake inhibitors 24930681 72008 49079 NDUFB2 4708 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 72010 49080 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SAR-407899 SAR-407899 72011 49081 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME EMBELIN EMBELIN 72012 49082 MAPT 4137 DRUGGABLE GENOME KOPARIN KOPARIN 72013 49083 GMNN 51053 DRUGGABLE GENOME MELITRACEN MELITRACEN 72014 49084 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID25726713-Compound-50 72015 49085 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE ISO-IANTHERAN A ISO-IANTHERAN A 17941622 72016 49086 TARDBP 23435 TUMOR SUPPRESSOR TRIADIMEFON TRIADIMEFON 72017 49087 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME GIVINOSTAT GIVINOSTAT 72018 49088 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Daunorubicin DAUNORUBICIN 16243804 72020 49089 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Protokylol Hydrochloride 216448 72021 49090 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE INSULIN INSULIN 8349045,7884509,9918825,8995390,11714021,17616136,8243832,2040701,16423895,17227768,17279354,16754199,10198313,14637133,15083319,11401844,9792680,10778531,17976658,1855475,12054114,1999488,11375332,15365619,10334307,12490950,9048628,9616209,15536229,1324860,8665891,8419118,9176187,7695642,9227455,17400720,8013658,12175706,17462778,9406133,11443199,9437239,17709177,2050674,7585807,12540375,15235327,11079746,10839189,11522683,8636261,8789319,7796936,8412752,15850715,1612011,8675649,15235328,11916910,7750476,10497159,9421368,17959846,16823721,2249650,7575448,17072583,9748297,8391425,15469417,1587399,9175878,9453263,17825496,10542046,9227454,7968595,10871200,12829635,12932196,18322300,7866477,8063042,10080958,16489447,12970362,10834933,15264018,8522056,15258906,18366935,8048627,1858877,8529803,9950801 72022 49091 HEBP1 50865 DRUGGABLE GENOME ABT-RTA-408 72023 49092 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Dasatinib DASATINIB 22328973 72024 49093 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME CYC-116 CYC-116 72026 49094 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 25314129 72028 49095 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX ISORHAMNETIN ISORHAMNETIN 25190466 72031 49096 MAOB 4129 DRUGGABLE GENOME, ENZYME N-(2-phenylcyclopropyl) amino acid derivative 3 72032 49097 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE antagonist 252166790 72035 49098 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 1,3-DIPHENYLTHIOUREA CHEMBL275260 72036 49099 CBX1 10951 NA TCMDC-123762 CHEMBL547483 72037 49100 ATXN2 6311 NA METHIXENE HYDROCHLORIDE METHIXENE HYDROCHLORIDE 72038 49101 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Biricodar BIRICODAR 72039 49102 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE AC-201 DIACEREIN 72041 49103 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR IL-6 7642569 72042 49104 IFNG 3458 DRUGGABLE GENOME THEOPHYLLINE THEOPHYLLINE 11918854 72044 49105 HMBS 3145 ENZYME Givosiran GIVOSIRAN 72045 49106 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE ALPHA-ADRENERGIC ANTAGONIST 10381893 72046 49107 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME ANTICARCINOGENIC 12517412 72047 49108 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE MEDI-543 72048 49109 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME GW843682X GW843682X 72050 49110 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Bosutinib BOSUTINIB 72051 49111 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL219586 GW590735 72052 49112 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER AMPHETAMINE AMPHETAMINE 72054 49113 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 4-AMINOPHENOL 4-AMINOPHENOL 72056 49114 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE PMSG 9071960 72057 49115 ASS1 445 ENZYME, DRUG RESISTANCE sodium phenylbutyrate 72058 49116 ENPP3 5169 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AGS-16M8F 72059 49117 MAPT 4137 DRUGGABLE GENOME FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 72060 49118 GMNN 51053 DRUGGABLE GENOME GLYASPERIN D GLYASPERIN D 72062 49119 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE JNJ-7706621 JNJ-7706621 72063 49120 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE unspecified PD-1 antibody 26833127 72064 49121 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-12 72065 49122 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178103871 SUPROFEN 72067 49123 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME CURCUMIN CURCUMIN 12954328 72069 49124 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE AZD8055 AZD-8055 25436981 72070 49125 ALOX15 246 ENZYME, DRUGGABLE GENOME PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 72072 49126 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR mycophenolate mofetil 18444945 72073 49127 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME TCMDC-124266 CHEMBL124006 72074 49128 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE VANDETANIB VANDETANIB 72075 49129 GAA 2548 DRUGGABLE GENOME, ENZYME SJ000111875 CHEMBL590949 72076 49130 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME MEK INHIBITOR TAK-733 22798288 72077 49131 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Flunisolide FLUNISOLIDE 72078 49132 BAZ2B 29994 NA PHENOTHIAZINE PHENOTHIAZINE 72079 49133 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL antagonist CHEMBL3545042 SELURAMPANEL 72080 49134 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME Temsirolimus TEMSIROLIMUS 72081 49135 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE DEXTRAN SULFATE 2465792 72082 49136 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ZIBOTENTAN ZIBOTENTAN 72083 49137 ATXN2 6311 NA NSC-720622 CHEMBL1287980 72084 49138 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER vemurafenib VEMURAFENIB 23116250 72085 49139 KDM2A 22992 DRUGGABLE GENOME, ENZYME inhibitor 249565909 72088 49140 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ACID BLUE 129 ACID BLUE 129 72089 49141 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor 249565585 UPROSERTIB 72090 49142 CFLAR 8837 DRUG RESISTANCE, DRUGGABLE GENOME, PROTEASE DOVITINIB DOVITINIB 72091 49143 GUCY1A2 2977 ENZYME, DRUGGABLE GENOME activator CHEMBL6622 ISOSORBIDE DINITRATE 72092 49144 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-2718 CHEMBL579143 72095 49145 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CHEMBL681 ETOMIDATE 72097 49146 RYR1 6261 ION CHANNEL, B30_2 SPRY DOMAIN, DRUGGABLE GENOME blocker,activator 178101120 RYANODINE 72098 49147 RIPK2 8767 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 385612168 72102 49148 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ELOCALCITOL ELOCALCITOL 72103 49149 IL18 3606 DRUGGABLE GENOME GSK-1070806 GSK-1070806 21157640 72104 49150 SMN2 6607 DRUGGABLE GENOME 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 72105 49151 TUBA3C 7278 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 21194809,25815147,25369367,25262051,23313639 72106 49152 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CINOLAZEPAM CINOLAZEPAM 72107 49153 ALDH1A1 216 DRUGGABLE GENOME, ENZYME HYDRAZOBENZENE HYDRAZOBENZENE 72108 49154 MIF 4282 DRUGGABLE GENOME, CELL SURFACE PMA 3305746 72109 49155 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE EXEBRYL-1 72112 49156 CSF3 1440 GROWTH FACTOR, DRUGGABLE GENOME LA-EP2006 72113 49157 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME inhibitor 178101349 72115 49158 BAZ2B 29994 NA 2-MERCAPTONICOTINIC ACID 2-MERCAPTONICOTINIC ACID 72116 49159 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PMA 7531948,12225365,7739574 72117 49160 LTA 4049 DRUGGABLE GENOME BAMINERCEPT BAMINERCEPT 72118 49161 PLK2 10769 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE BI2536 72121 49162 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE 2,4-DINITROPHENOL 2,4-DINITROPHENOL 72122 49163 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL1789844 IPILIMUMAB 72123 49164 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ANTIHISTAMINE TERFENADINE 11454724,16842392 72124 49165 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BENZETHONIUM CHLORIDE BENZETHONIUM CHLORIDE 72125 49166 MAGEC2 51438 ENZYME CV-9201 72128 49167 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NEUROPEPTIDE-Y NEUROPEPTIDE-Y 72129 49168 GMNN 51053 DRUGGABLE GENOME GNF-PF-4876 CHEMBL585444 72130 49169 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL107 COLCHICINE 72131 49170 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE L-ASPARAGINASE ASPARAGINASE 15837750 72132 49171 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 385612183 72134 49172 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL CHLORZOXAZONE CHLORZOXAZONE 72135 49173 KDM4A 9682 DRUGGABLE GENOME, ENZYME DEFERIPRONE DEFERIPRONE 72136 49174 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ILOPERIDONE ILOPERIDONE 72137 49175 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL1200567 DOXYCYCLINE HYCLATE 72138 49176 POLI 11201 DNA REPAIR HISPIDIN HISPIDIN 72139 49177 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist,antagonist 135651142 72140 49178 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME DASATINIB DASATINIB 72142 49179 PDE4D 5144 DRUGGABLE GENOME, ENZYME ETAZOLATE ETAZOLATE 72143 49180 MAOA 4128 DRUGGABLE GENOME, ENZYME GypensapogeninB 72144 49181 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR PF-04236921 PF-04236921 72145 49182 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR C-1027 CHEMBL506048 17978180 72146 49183 XRCC1 7515 CLINICALLY ACTIONABLE cyclophosphamide CYCLOPHOSPHAMIDE 19786980,22188361 72147 49184 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650333 CHEMBL59030 72148 49185 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GOSSYPOL GOSSYPOL 16020667 72150 49186 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER valganciclovir VALGANCICLOVIR 27402191 72151 49187 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CABOZANTINIB CABOZANTINIB 72152 49188 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE AMINOCAPROIC ACID 72153 49189 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SJ000029259 CHEMBL592558 72157 49190 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TOZASERTIB TOZASERTIB 72160 49191 HBB 3043 DRUGGABLE GENOME, ENZYME Efaproxyn 72161 49192 CDK11B 984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL1230607 PHA-793887 72162 49193 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650446 72163 49194 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1200599 DIFENOXIN HYDROCHLORIDE 72166 49195 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE MC-1 72168 49196 GMNN 51053 DRUGGABLE GENOME 5-FLUOROURIDINE CHEMBL54918 72169 49197 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE axitinib AXITINIB 25816720 72170 49198 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650475 72171 49199 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 135652670 BILOBALIDE 72172 49200 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CHLORPHENIRAMINE CHLORPHENIRAMINE 72174 49201 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME OSI-632 OSI-632 72176 49202 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SULINDAC SULINDAC 22931300 72177 49203 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME agonist 178104019 PEGINESATIDE 72178 49204 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Amide derivative 2 72179 49205 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TAMATINIB R-406 72181 49206 TARDBP 23435 TUMOR SUPPRESSOR REV-5901 REV-5901 72182 49207 RAPGEF3 10411 ENZYME PURPUROGALLIN PURPUROGALLIN 72184 49208 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 315661265 72185 49209 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US10179791, Compound 171 72187 49210 TUBB2A 7280 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 72188 49211 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE Artemether ARTEMETHER 72192 49212 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Pyrazole and benzimidazole derivative 1 72193 49213 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 6'-IODONONIVAMIDE CHEMBL177809 72195 49214 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-21 72198 49215 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME binimetinib BINIMETINIB 72200 49216 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL605 PROCAINAMIDE HYDROCHLORIDE 72202 49217 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TCMDC-123992 CHEMBL530149 72203 49218 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME PMID27828716-Compound-21 72205 49219 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXANDROLONE OXANDROLONE 72206 49220 MMP14 4323 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 405560328 72207 49221 CMPK1 51727 KINASE, ENZYME cisplatin CISPLATIN 21642870 72209 49222 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CAPTAN CAPTAN 72210 49223 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME FOLIC ACID FOLIC ACID 72212 49224 PSENEN 55851 DRUGGABLE GENOME modulator CHEMBL190083 TARENFLURBIL 72213 49225 SLC36A1 206358 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 178101386 OXITRIPTAN 72214 49226 KDM4A 9682 DRUGGABLE GENOME, ENZYME DEMECLOCYCLINE HYDROCHLORIDE DEMECLOCYCLINE HYDROCHLORIDE 72216 49227 MAPT 4137 DRUGGABLE GENOME AMSACRINE HYDROCHLORIDE AMSACRINE HYDROCHLORIDE 72217 49228 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE VERAPAMIL VERAPAMIL 1511424 72219 49229 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Curcumin analog 1 72221 49230 ACE2 59272 ENZYME, TRANSPORTER, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, CELL SURFACE, PROTEASE 178101824 72222 49231 NOS2 4843 DRUGGABLE GENOME, ENZYME THEOPHYLLINE THEOPHYLLINE 12223230 72223 49232 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR SINENSETIN SINENSETIN 72224 49233 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28270021-Compound-WO2016054807Example1 72225 49234 BAZ2B 29994 NA AG-555 CHEMBL53898 72226 49235 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE 7-azaindole derivative 2 72228 49236 KCNF1 3754 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL284348 DALFAMPRIDINE 72229 49237 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME WITHAFERIN A WITHAFERIN A 20726569 72230 49238 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ARUNDINE ARUNDINE 72232 49239 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME NSC-748118 CHEMBL2063681 22283430 72234 49240 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GNF-PF-2657 CHEMBL578944 72235 49241 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE 178101646 72236 49242 NRIP1 8204 NUCLEAR HORMONE RECEPTOR RETINOIDS 15180561 72237 49243 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 1-[2-(TRIFLUOROMETHYL)PHENYL]IMIDAZOLE CHEMBL277525 72238 49244 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SGC0946 27294782 72239 49245 UBA2 10054 DRUGGABLE GENOME, ENZYME LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 72243 49246 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3545248 DS-7423 72245 49247 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL LIDOCAINE LIDOCAINE 72246 49248 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE BIIB037 23663286 72247 49249 ALOX5 240 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200760 BALSALAZIDE DISODIUM 72249 49250 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-123532 CHEMBL547833 72250 49251 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 381118879 VIDUPIPRANT 72251 49252 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME ONDANSETRON ONDANSETRON 15458770 72253 49253 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor SCH727965 DINACICLIB 72255 49254 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 249565721 72256 49255 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL2104967 FIRATEGRAST 72258 49256 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545235 SIMOTINIB 72259 49257 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HOMIDIUM BROMIDE HOMIDIUM BROMIDE 72260 49258 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL2220486 LUCITANIB 72261 49259 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ASARININ ASARININ 72262 49260 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 72263 49261 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE bis-triazole derivative 10 72264 49262 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ARACHIDONIC ACID ARACHIDONIC ACID 72265 49263 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL1236962 OMIPALISIB 72266 49264 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 178102318 KW-2449 72267 49265 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 375973218 72269 49266 ARSA 410 DRUGGABLE GENOME, ENZYME HGT-1111 72270 49267 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 318164839 PONESIMOD 72272 49268 POR 5447 ENZYME, DRUGGABLE GENOME nicotine NICOTINE 72273 49269 NUDT15 55270 ENZYME, CLINICALLY ACTIONABLE thioguanine THIOGUANINE 27530327 72274 49270 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-124321 CHEMBL526952 72275 49271 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME FRAXETIN FRAXETIN 72276 49272 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE ILORASERTIB ILORASERTIB 72278 49273 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TAMOXIFEN TAMOXIFEN 1315250 72279 49274 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR 315661322 VAMOROLONE 72280 49275 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TOLPERISONE HYDROCHLORIDE TOLPERISONE HYDROCHLORIDE 72282 49276 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DEOXIEPINEPHRINE DEOXIEPINEPHRINE 72283 49277 SGK1 6446 SERINE THREONINE KINASE, KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 328083523 72284 49278 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE SJ000032155 CHEMBL590643 72286 49279 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Encorafenib ENCORAFENIB 72287 49280 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE DOVITINIB DOVITINIB 72288 49281 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR ENTINOSTAT ENTINOSTAT 19966789,20491440 72289 49282 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Golotimod GOLOTIMOD 72290 49283 PTGS2 5743 DRUGGABLE GENOME, ENZYME FENBUFEN FENBUFEN 72291 49284 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-840 CHEMBL601605 72292 49285 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8481586, 40 72293 49286 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SB-334867 CHEMBL291536 72294 49287 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 340590256 TRILACICLIB 72295 49288 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PAZOPANIB PAZOPANIB 72296 49289 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME gefitinib GEFITINIB 31664190 72298 49290 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HE3235 HE3235 72299 49291 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL970 HALAZEPAM 72301 49292 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CI-1040 CI-1040 72303 49293 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 178102337 SORAFENIB 72304 49294 KDM4A 9682 DRUGGABLE GENOME, ENZYME WIN-55212-2 WIN-552122 72306 49295 LCAT 3931 ENZYME, TRANSPORTER, DRUGGABLE GENOME PREDNISOLONE PREDNISOLONE 2314540 72307 49296 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3545238 CS-8080 72308 49297 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME RANIBIZUMAB RANIBIZUMAB 72310 49298 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme24-11H-pyrido[4,3-a]carbazole 72311 49299 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL786 TAMOXIFEN CITRATE 72313 49300 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Ezatiostat EZATIOSTAT 72314 49301 MAPT 4137 DRUGGABLE GENOME MENADIONE MENADIONE 72315 49302 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE FERULIC ACID FERULIC ACID 24076170 72316 49303 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE DEMETHYLWEDELOLACTONE DEMETHYLWEDELOLACTONE 22926226 72317 49304 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ATRANORIN ATRANORIN 72318 49305 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GW441756X GW441756X 72321 49306 POLI 11201 DNA REPAIR CEPHALOTHIN CEPHALOTHIN 72322 49307 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LIPOIC ACID, ALPHA LIPOIC ACID, ALPHA 72324 49308 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL antagonist CHEMBL3707378 CB-189625 72325 49309 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX ALITRETINOIN ALITRETINOIN 72327 49310 ATAD5 79915 NA CID 2056784 CHEMBL261123 72329 49311 TBXAS1 6916 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME NM-702 72330 49312 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ZILEUTON ZILEUTON 22931300 72332 49313 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE (R)-PIA (R)-PIA 72333 49314 GMNN 51053 DRUGGABLE GENOME ISOLIQUIRITIGENIN ISOLIQUIRITIGENIN 72334 49315 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545021 ANLOTINIB 72336 49316 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE TYROSINE KINASE INHIBITORS 15289348 72337 49317 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR PROPYLTHIOURACIL PROPYLTHIOURACIL 11077070 72338 49318 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650718 72340 49319 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor CHEMBL494089 GSK-690693 72342 49320 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME BUTYRYLHYDROXAMIC ACID BUTYRYLHYDROXAMIC ACID 21874153 72344 49321 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103926 UMECLIDINIUM 72345 49322 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME I-CBP112 26552700 72347 49323 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR RELCOVAPTAN RELCOVAPTAN 72348 49324 PLD2 5338 ENZYME, DRUGGABLE GENOME HALOPEMIDE HALOPEMIDE 72349 49325 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GLYCINE GLYCINE 22931300 72351 49326 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DOCEBENONE DOCEBENONE 72353 49327 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME IRIGENOL IRIGENOL 72354 49328 RGS4 5999 DRUGGABLE GENOME TPCK TPCK 72355 49329 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702223 NECROSTATIN 72356 49330 NOS1 4842 DRUGGABLE GENOME, ENZYME inhibitor 315661232 72358 49331 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CAR-T Cells targeting HER2 72360 49332 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PX 104.1 72361 49333 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METHAZOLAMIDE METHAZOLAMIDE 72363 49334 GUCY1B1 2983 DRUGGABLE GENOME Vericigiuat 72365 49335 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL2079587 STANOZOLOL 72367 49336 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 363894217 VORUCICLIB 72370 49337 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR HYDRAMETHYLNON HYDRAMETHYLNON 72371 49338 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (RS)-ROSCOVITINE (RS)-ROSCOVITINE 72372 49339 DAPK1 1612 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME gemcitabine GEMCITABINE 22293537 72373 49340 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ACIFRAN ACIFRAN 25737085 72374 49341 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE LYMPHOKINES 2126274 72376 49342 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BAY-11-7085 BAY-11-7085 72377 49343 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE INTERLEUKIN-1 9185713,7524717 72378 49344 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VER-3323 CHEMBL309760 72380 49345 MED19 219541 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR ethanol ALCOHOL 32451486 72381 49346 PDE10A 10846 ENZYME, DRUGGABLE GENOME 1-aryl-4-methyl-[1,2,4]triazolo[4,3-a]quinoxaline derivative 3 72385 49347 SMN2 6607 DRUGGABLE GENOME IPRIFLAVONE IPRIFLAVONE 72386 49348 TMEM97 27346 NA Bicyclo-heptan-2-amine derivative 2 72387 49349 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MC-3002 72389 49350 DDC 1644 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200748 CARBIDOPA 72390 49351 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE NITRAZEPAM NITRAZEPAM 72391 49352 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-5151 CHEMBL576208 72392 49353 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PMID28048944-Compound-2 72394 49354 ATAD5 79915 NA PIMOZIDE PIMOZIDE 72395 49355 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 310264678 72396 49356 CAMK1 8536 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME ILORASERTIB ILORASERTIB 72398 49357 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE AZD-1152-HQPA AZD-1152-HQPA 72399 49358 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 315661128 APALUTAMIDE 72400 49359 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-47 72401 49360 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME APIGENIN APIGENIN 72402 49361 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3188551 GSK-2636771 72403 49362 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE METHYLDOPA (RACEMIC) METHYLDOPA (RACEMIC) 72404 49363 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 72405 49364 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Bretylium BRETYLIUM 72406 49365 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BRADANICLINE BRADANICLINE 23126648 72407 49366 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL CHEMBL266510 FLINDOKALNER 72408 49367 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 72410 49368 SMN2 6607 DRUGGABLE GENOME 2-(PHENOXYMETHYL)BENZOTHIAZOLE 2-(PHENOXYMETHYL)BENZOTHIAZOLE 72411 49369 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME agonist 178100907 72412 49370 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE TOPIRAMATE TOPIRAMATE 72413 49371 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Ponatinib PONATINIB 72414 49372 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 VERAPAMIL VERAPAMIL 21393461 72415 49373 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME BORTEZOMIB BORTEZOMIB 20875739 72416 49374 MAPT 4137 DRUGGABLE GENOME CHOLECALCIFEROL CHOLECALCIFEROL 72417 49375 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME elagolix ELAGOLIX 72418 49376 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RETINYL ACETATE RETINYL ACETATE 72419 49377 SOAT1 6646 DRUGGABLE GENOME ATORVASTATIN ATORVASTATIN 14644397 72420 49378 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545088 PUQUITINIB 72422 49379 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-18 72423 49380 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME sorafenib SORAFENIB 20124951 72424 49381 KMO 8564 DRUGGABLE GENOME, ENZYME Isoxazoles and isoxazoline derivative 3 72425 49382 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Vincristine VINCRISTINE 72426 49383 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GW9662 CHEMBL375270 72427 49384 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ESCULIN ESCULIN 72428 49385 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CETUXIMAB CETUXIMAB 72429 49386 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME TCMDC-124059 CHEMBL530733 72430 49387 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE GEFITINIB GEFITINIB 21274259 72433 49388 CA1 759 DRUGGABLE GENOME, ENZYME inhibitor 178103413 DICHLORPHENAMIDE 72434 49389 PRCP 5547 ENZYME, DRUGGABLE GENOME, PROTEASE Piperidinyl triazole derivative 1 72436 49390 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist 135650517 72437 49391 PDE4B 5142 DRUGGABLE GENOME, ENZYME MEM-1414 72438 49392 POLI 11201 DNA REPAIR DAPHNETIN DAPHNETIN 72439 49393 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL1200527 ATRACURIUM BESYLATE 72440 49394 FAAH 2166 ENZYME, DRUGGABLE GENOME Tetra-substituted urea derivative 2 72443 49395 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 223366170 NS-018 72444 49396 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 72446 49397 CCN1 3491 DRUGGABLE GENOME HYPOTENSIVE AGENTS 12724323 72448 49398 TNFSF10 8743 DRUGGABLE GENOME TRICHOSTATIN A 16096370 72449 49399 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME AR-42 AR-42 72451 49400 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SULFANITRAN SULFANITRAN 72452 49401 CYP2R1 120227 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME calcidiol CALCIFEDIOL 26661839 72453 49402 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545323 PWT-33579 72454 49403 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ETHER ETHER 16081674 72455 49404 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PENTACHLOROPHENOL PENTACHLOROPHENOL 72457 49405 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME METHYLENE BLUE METHYLENE BLUE 72460 49406 TSPO 706 DRUGGABLE GENOME Benzimidazolone acetamide derivative 1 72461 49407 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PHYSODIC ACID PHYSODIC ACID 72462 49408 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651286 TACALCITOL 72464 49409 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OXATOMIDE OXATOMIDE 72465 49410 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE AG-808 CHEMBL68534 72466 49411 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1479 DANAZOL 72469 49412 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TEBUCONAZOLE TEBUCONAZOLE 72470 49413 SEM1 7979 NA inhibitor CHEMBL325041 BORTEZOMIB 72471 49414 DOCK8 81704 NA gemcitabine GEMCITABINE 31616045 72472 49415 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 310264779 72476 49416 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME FLUDIAZEPAM FLUDIAZEPAM 72477 49417 ALDH5A1 7915 DRUGGABLE GENOME, ENZYME Succinic acid 72479 49418 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL3833368 RUCAPARIB CAMSYLATE 72480 49419 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LANSOPRAZOLE LANSOPRAZOLE 72482 49420 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METOPRINE METOPRINE 72483 49421 NOS1 4842 DRUGGABLE GENOME, ENZYME ENALAPRIL ENALAPRIL 11712645 72486 49422 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE N6-CYCLOPENTYLADENOSINE N6-CYCLOPENTYLADENOSINE 72487 49423 EGLN3 112399 DRUGGABLE GENOME, ENZYME FG-2216 72488 49424 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200437 QUINIDINE GLUCONATE 72491 49425 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651441 72492 49426 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 25427841,16636344,19364970,19852077,17577039,27116457,18349289,17627617,12181437,17058217,17185998,12969965,1651156,18466101,14647407,20562211,19390945,17728214,12019197,18221820,11990381,15179405,10381366,16951398,15007088,11037804 72493 49427 GLS 2744 ENZYME CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 72495 49428 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651260 THIOTHIXENE 72496 49429 AMD1 262 ENZYME, DRUGGABLE GENOME Tromethamine TROMETHAMINE 72497 49430 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 6-METHOXY-HARMALAN CHEMBL338115 72498 49431 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 178102617 72499 49432 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor CHEMBL3137301 SACUBITRIL 72500 49433 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Crizotinib CRIZOTINIB 27595477,27393507,27283993 72501 49434 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-390523 CHEMBL157258 72502 49435 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565686 BX-795 72505 49436 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651435 TRETINOIN 72506 49437 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME mercaptopurine MERCAPTOPURINE 25217962 72507 49438 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NADOLOL NADOLOL 72508 49439 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ALLITRIDIN ALLITRIDIN 72509 49440 ALOX15 246 ENZYME, DRUGGABLE GENOME TACRINE TACRINE 72513 49441 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME CVX-241 21149738 72514 49442 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR GS 6201 GS 6201 72516 49443 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor 178102560 72520 49444 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE allosteric modulator 178100964 72521 49445 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME PD173074 22869148 72523 49446 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIPYRIDYL DIPYRIDYL 72524 49447 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER phenobarbital PHENOBARBITAL 25846690 72525 49448 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 249565648 72526 49449 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PURVALANOLA PURVALANOLA 72528 49450 SLC12A4 6560 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSPORTER BUMETANIDE BUMETANIDE 72529 49451 EPHX2 2053 DRUGGABLE GENOME, ENZYME inhibitor 348353676 72530 49452 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLOROPHACINONE CHLOROPHACINONE 72532 49453 ALOX15B 247 DRUGGABLE GENOME, ENZYME TYRPHOSTIN 23 TYRPHOSTIN 23 72534 49454 CBX1 10951 NA METERGOLINE METERGOLINE 72535 49455 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Regorafenib REGORAFENIB 72536 49456 GADD45A 1647 DNA REPAIR, TUMOR SUPPRESSOR, KINASE GENISTEIN GENISTEIN 15527761 72539 49457 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GENTIAN VIOLET GENTIAN VIOLET 72540 49458 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 374883891 KX2-361 72542 49459 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME XANTHOHUMOL XANTHOHUMOL 22111577 72543 49460 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME MINOCYCLINE MINOCYCLINE 19258275 72544 49461 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200982 BUTABARBITAL SODIUM 72545 49462 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 2,2,3,3,4,4,5,5,6,6,7,7,8,8,8-PENTADECAFLUORO-OCTANOIC ACID CHEMBL172988 72546 49463 CA12 771 DRUGGABLE GENOME inhibitor CHEMBL18 ETHOXZOLAMIDE 72547 49464 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Aminocyclopentenone compound 5 72550 49465 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ESTRADIOL CYPIONATE ESTRADIOL CYPIONATE 72551 49466 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PK1 72552 49467 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME TAXANES 15970709 72555 49468 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PD-0325901 PD-0325901 26272063,22684718,25673820,21516509,26037647,26267534,26582713,27556948,23934108,21325073,20570890 72556 49469 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 249565725 72560 49470 SLCO4A1 28231 DRUGGABLE GENOME, TRANSPORTER 178101458 72563 49471 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HURATOXIN HURATOXIN 24931277 72564 49472 VKORC1 79001 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200772 WARFARIN POTASSIUM 72565 49473 TK1 7083 ENZYME, KINASE, DRUGGABLE GENOME FV-100 VALNIVUDINE HYDROCHLORIDE 72568 49474 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651037 SERTINDOLE 72570 49475 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE CFG920 CFG-920 72571 49476 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR ANTI-INFLAMMATORY DRUGS 14960322 72573 49477 ACKR3 57007 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135651881 72574 49478 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL944 CHLOROPROCAINE HYDROCHLORIDE 72575 49479 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Imatinib IMATINIB 72577 49480 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME FLUORANTHENE FLUORANTHENE 72578 49481 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PICEATANNOL PICEATANNOL 72579 49482 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME FLUOXETINE FLUOXETINE 11487610 72580 49483 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME TAK-715 TAK-715 72583 49484 MAOA 4128 DRUGGABLE GENOME, ENZYME inhibitor 385612213 72584 49485 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL79 LIDOCAINE 72586 49486 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME FLUNARIZINE FLUNARIZINE 72588 49487 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Platinum compounds 25545243,24533712,11160862,21479364,10208650,21946896,18511948 72589 49488 GLS 2744 ENZYME GLUCOCORTICOID 8638663 72591 49489 AKT1S1 84335 KINASE, DRUGGABLE GENOME inhibitor MLN0128 SAPANISERTIB 72592 49490 PTGS1 5742 ENZYME, DRUGGABLE GENOME NCX 4016 72594 49491 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BRAF INHIBITOR 31580757 72596 49492 LAG3 3902 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE IMP-321 72598 49493 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PLUMBAGIN PLUMBAGIN 72599 49494 KDM4A 9682 DRUGGABLE GENOME, ENZYME ZINC 03369470 CHEMBL599013 72600 49495 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY MEDI0382 COTADUTIDE 72601 49496 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 249565803 72602 49497 PRKAB1 5564 ENZYME, KINASE, DRUGGABLE GENOME WORTMANNIN WORTMANNIN 15928020 72603 49498 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1762621 BARDOXOLONE METHYL 72604 49499 BAZ2B 29994 NA STICTIC ACID STICTIC ACID 72605 49500 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CCG-63808 CHEMBL1604848 72606 49501 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME VATALANIB VATALANIB 72608 49502 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TAK-733 TAK-733 26439693 72609 49503 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BRL 35135 72611 49504 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZD5363 CAPIVASERTIB 72612 49505 APH1B 83464 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL520733 SEMAGACESTAT 72613 49506 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102246 VIPADENANT 72614 49507 PDE4A 5141 DRUGGABLE GENOME, ENZYME ROFLUMILAST ROFLUMILAST 72615 49508 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200715 HEXYLCAINE HYDROCHLORIDE 72616 49509 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE Irinotecan IRINOTECAN 22753594 72618 49510 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE TYRPHOSTIN 47 TYRPHOSTIN 47 72619 49511 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor AS703569 CENISERTIB 72621 49512 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR 26739882,27037411 72622 49513 BAZ2B 29994 NA NSC-180246 CHEMBL484640 72623 49514 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME METHYLDOPA METHYLDOPA 72624 49515 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PIMECROLIMUS PIMECROLIMUS 72627 49516 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 328083452 72632 49517 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4459 CHEMBL585502 72633 49518 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ICILLIN ICILLIN 72634 49519 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 72635 49520 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Gefitinib GEFITINIB 26561558 72636 49521 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE mFOLFOX6 27918764 72639 49522 POLK 51426 DNA REPAIR, ENZYME LUTEOLIN LUTEOLIN 72640 49523 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TESTOSTERONE TESTOSTERONE 22931300 72642 49524 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE INDOMETHACIN MORPHOLINYLAMIDE INDOMETHACIN MORPHOLINYLAMIDE 72643 49525 QRFPR 84109 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 381744934 72644 49526 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor AFATINIB AFATINIB 72645 49527 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL19 METHAZOLAMIDE 72646 49528 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME thioguanosine diphosphate 26332308 72647 49529 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-22 72648 49530 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-63 72649 49531 ATXN2 6311 NA GOSSYPOL GOSSYPOL 72650 49532 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 flurbiprofen FLURBIPROFEN 12698304,32423989,25712887 72651 49533 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE carboplatin CARBOPLATIN 21605004,29662106,27995989,20634689,19159907,19307503 72654 49534 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-668394 CHEMBL336095 72655 49535 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR lapatinib LAPATINIB 72656 49536 POLA1 5422 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL1096882 FLUDARABINE PHOSPHATE 72659 49537 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 385612221 72660 49538 TUBA1C 84790 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 72661 49539 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3545345 UR-63325 72662 49540 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 2-AMINOBIPHENYL CHEMBL296021 72663 49541 RGS4 5999 DRUGGABLE GENOME 2-MESATP CHEMBL336208 72666 49542 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 72667 49543 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ERGOCRYPTINE ERGOCRYPTINE 72668 49544 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 178102305 DASATINIB 72669 49545 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 nelfinavir NELFINAVIR 72670 49546 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 381118815 72671 49547 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME esomeprazole ESOMEPRAZOLE 72673 49548 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX SJ000113257 CHEMBL528694 72674 49549 UBE2N 7334 ENZYME, DRUGGABLE GENOME NARINGIN NARINGIN 72675 49550 HEXB 3074 ENZYME CDDP CISPLATIN 2089371 72680 49551 ATXN2 6311 NA XANTHOANGELOL XANTHOANGELOL 72681 49552 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200478 DYCLONINE HYDROCHLORIDE 72682 49553 MAPT 4137 DRUGGABLE GENOME TCMDC-123723 CHEMBL525103 72683 49554 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 363894214 SITRAVATINIB 72684 49555 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME HEPARIN HEPARIN 15935280 72685 49556 HMOX2 3163 ENZYME ANTIOXIDANT 11449996 72686 49557 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-124356 CHEMBL22062 72687 49558 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE AST-487 AST-487 72689 49559 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 72690 49560 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME AMG 420 72691 49561 TSC2 7249 CLINICALLY ACTIONABLE, KINASE, TUMOR SUPPRESSOR MTOR INHIBITOR 26831717 72692 49562 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME inhibitor 375973227 72693 49563 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1950289 TANZISERTIB 72694 49564 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3,3'-DIMETHOXYBENZIDINE CHEMBL398363 72695 49565 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ETHOPROPAZINE HYDROCHLORIDE ETHOPROPAZINE HYDROCHLORIDE 72696 49566 IL1B 3553 KINASE, DRUGGABLE GENOME MELATONIN MELATONIN 8077674 72697 49567 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545088 PUQUITINIB 72700 49568 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-7e 72702 49569 CXCL8 3576 DRUGGABLE GENOME VERAPAMIL VERAPAMIL 2686646 72704 49570 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Diaryl amine derivative 3 72705 49571 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME GSK-269962A GSK-269962A 72706 49572 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE NICLOSAMIDE NICLOSAMIDE 72708 49573 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BUPARLISIB HYDROCHLORIDE 72710 49574 RGS4 5999 DRUGGABLE GENOME MK-212 MK-212 72711 49575 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE FLUOROURACIL FLUOROURACIL 20628391 72713 49576 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE IM23 72714 49577 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor CHEMBL574737 UCN-01 72715 49578 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLORPYRIFOS-METHYL CHLORPYRIFOS-METHYL 72716 49579 ALOX5 240 DRUGGABLE GENOME, ENZYME inhibitor 315661139 PF-4191834 72717 49580 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME RALOXIFENE RALOXIFENE 72718 49581 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Tipifarnib TIPIFARNIB 72719 49582 MAPT 4137 DRUGGABLE GENOME NSC-175743 CHEMBL1609016 72720 49583 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Bevacizumab BEVACIZUMAB 26965451,26432108,25363205 72721 49584 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX LEUPROLIDE ACETATE 14678567 72723 49585 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-44 72724 49586 FAAH 2166 ENZYME, DRUGGABLE GENOME Pyrimidinyl ethylenediamine derivative 1 72725 49587 NOS2 4843 DRUGGABLE GENOME, ENZYME Pimagedine HCl 72728 49588 PTBP1 5725 DRUGGABLE GENOME SJ000044511 CHEMBL592124 72730 49589 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER IL-3 7564516 72731 49590 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BISSALICYL FUMARATE BISSALICYL FUMARATE 72734 49591 CTSH 1512 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 252166814 72736 49592 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651111 72737 49593 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-67 72740 49594 APOE 348 DRUGGABLE GENOME warfarin WARFARIN 21923605,29432897 72741 49595 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Insulin recombinant 72742 49596 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BLZ945 27199435 72746 49597 PLA2G7 7941 DRUGGABLE GENOME, ENZYME inhibitor 178103307 DARAPLADIB 72748 49598 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545083 RGB-286638 72750 49599 DPP9 91039 PROTEASE, ENZYME, DRUGGABLE GENOME Thiomorpholine derivative 1 72751 49600 GLS 2744 ENZYME PMID30273516-Compound-38 72752 49601 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIHYDROXIDINE DIHYDROXIDINE 72755 49602 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-13 72756 49603 CCND2 894 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE PD 0332991 72757 49604 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME HYPERICIN HYPERICIN 72758 49605 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME RETINOIDS 7890733 72759 49606 CA2 760 DRUGGABLE GENOME, ENZYME EPO EPOETIN ALFA 11112384 72760 49607 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE ABIRATERONE ABIRATERONE 72761 49608 ATAD5 79915 NA NSC-139257 CHEMBL1256364 72762 49609 HNRNPH2 3188 NA migalastat MIGALASTAT 72763 49610 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RESVERATROL RESVERATROL 72765 49611 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LIOTHYRONINE LIOTHYRONINE 72767 49612 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2387080 TASELISIB 72768 49613 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 249565855 72769 49614 HMGCR 3156 ENZYME, DRUGGABLE GENOME Sterol derivative 2 72770 49615 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650183 DIHYDROMORPHINE 72771 49616 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 178102296 DORAMAPIMOD 72772 49617 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME BERKELEYDIONE BERKELEYDIONE 17970594 72773 49618 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE FIGITUMUMAB FIGITUMUMAB 72774 49619 SMN1 6606 DRUGGABLE GENOME RETUSIN 7-METHYL ETHER RETUSIN 7-METHYL ETHER 72775 49620 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PHA-680632 PHA-680632 18026198 72776 49621 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIHYDRALAZINE DIHYDRALAZINE 72777 49622 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUDIODARONE BUDIODARONE 72778 49623 KDM4A 9682 DRUGGABLE GENOME, ENZYME N'-(2-HYDROXYBENZYLIDENE)ISONICOTINOHYDRAZIDE SALINAZID 72780 49624 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PERGOLIDE PERGOLIDE 72781 49625 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100477 ATRASENTAN 72784 49626 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 178102341 72785 49627 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 72786 49628 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE IRINOTECAN IRINOTECAN 72787 49629 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME BERBERRUBINE BERBERRUBINE 72789 49630 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Avastin+/-Tarceva 72790 49631 COMT 1312 DRUGGABLE GENOME, ENZYME antipsychotics 12729939,18180754,12815736,16702905,11150892,12372660,11990384,15465976,14610521,9535125,22391769,25048416,15115916,14520117,11525417,15522252 72791 49632 GBA 2629 DRUGGABLE GENOME, ENZYME TCMDC-125278 CHEMBL588327 72792 49633 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CILOSTAMIDE CILOSTAMIDE 72793 49634 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME BIRINAPANT BIRINAPANT 72794 49635 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PINDOLOL PINDOLOL 72796 49636 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SP-600125 SP-600125 72797 49637 SMN2 6607 DRUGGABLE GENOME DNDI1417701 CHEMBL1326164 72798 49638 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME PMID25435179-Compound-WO2012106509Tenovin-6 72800 49639 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ethylmorphine ETHYLMORPHINE 72801 49640 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE RG-1530 RG-1530 72803 49641 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 354702263 72804 49642 MAPT 4137 DRUGGABLE GENOME INAMRINONE INAMRINONE 72805 49643 KDM4A 9682 DRUGGABLE GENOME, ENZYME 2-HYDROXY-NAPHTHALDEHYDE THIOSEMICARBAZONE CHEMBL505209 72807 49644 ITGB6 3694 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE inhibitor CHEMBL2109621 ABITUZUMAB 72808 49645 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ICATIBANT ICATIBANT 72809 49646 CBX1 10951 NA MMV006389 CHEMBL586000 72810 49647 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING NSC-121858 CHEMBL483838 72812 49648 HMGCR 3156 ENZYME, DRUGGABLE GENOME FLUVASTATIN FLUVASTATIN 72813 49649 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DODECYL-TRIMETHYL-AMMONIUM BROMIDE CHEMBL109873 72814 49650 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135651341 (CYCLOHEXYLAMINO)METHYLENEDIPHOSPHONIC ACID 72821 49651 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 252166799 72822 49652 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PROTEASE INHIBITOR 8702992 72824 49653 CXCL8 3576 DRUGGABLE GENOME BIOFLAVONOID 9292787 72825 49654 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE durvalumab DURVALUMAB 72827 49655 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FEPRAZONE FEPRAZONE 72828 49656 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER PSC-833 11189941,9816180 72830 49657 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME NSC-9037 CHEMBL1451216 72833 49658 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102298 BMS-387032 72834 49659 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HINOKITIOL HINOKITIOL 72837 49660 S100A9 6280 DRUGGABLE GENOME, KINASE, ENZYME Paquinimod PAQUINIMOD 72841 49661 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102913 72842 49662 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 328083503 72847 49663 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650187 72849 49664 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE SKF-89626 CHEMBL284609 72850 49665 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-15 72851 49666 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR THIOLACTOMYCIN THIOLACTOMYCIN 72852 49667 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME APIXABAN APIXABAN 72853 49668 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME OCRELIZUMAB OCRELIZUMAB 72855 49669 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AMIODARONE AMIODARONE 72856 49670 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist,antagonist 135651446 ADENOSINE TRIPHOSPHATE 72858 49671 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor XL228 XL-228 72859 49672 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MENTHOFURAN MENTHOFURAN 22931300 72860 49673 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor CHEMBL377559 RETASPIMYCIN HYDROCHLORIDE 72861 49674 KDM4A 9682 DRUGGABLE GENOME, ENZYME SKF-89626 CHEMBL284609 72864 49675 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RO-410960 CHEMBL1256291 72865 49676 TUBB 203068 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 72866 49677 MAP2K5 5607 KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor BAY869766 72867 49678 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR gefitinib GEFITINIB 31664190 72868 49679 NOTCH3 4854 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor MK0752 72869 49680 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE Aluminium 72873 49681 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Androgen restored contraceptive 72874 49682 GMNN 51053 DRUGGABLE GENOME CID 3237815 CHEMBL410484 72875 49683 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME FISETIN FISETIN 72877 49684 IL12RB2 3595 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AS1409 72878 49685 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor 178102320 ENZASTAURIN 72879 49686 NR2F2 7026 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GNF-PF-4659 CHEMBL584442 72880 49687 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL SAFINAMIDE SAFINAMIDE 72882 49688 GAPDH 2597 DRUGGABLE GENOME, ENZYME SODIUM BUTYRATE 9437188 72883 49689 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME QUINPIROLE QUINPIROLE 72884 49690 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702261 72885 49691 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE geldanamycin GELDANAMYCIN 18652519 72886 49692 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR QUINIZARIN QUINIZARIN 72887 49693 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-2657 CHEMBL578944 72891 49694 IL12RB2 3595 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE DENILEUKIN DIFTITOX 72893 49695 GMNN 51053 DRUGGABLE GENOME CRIDANIMOD CRIDANIMOD 72895 49696 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-16 72896 49697 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE SOTRASTAURIN SOTRASTAURIN 72897 49698 KAT2B 8850 ENZYME, DRUGGABLE GENOME DIETHYL-2-TRIDECYLIDENEMALONATE CHEMBL1797709 21292492 72898 49699 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL451 CHLORDIAZEPOXIDE 72899 49700 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565808 72900 49701 UGT2B7 7364 DRUGGABLE GENOME mycophenolic acid 24220207 72901 49702 HEXB 3074 ENZYME THYROXINE THYROXINE 7388056 72902 49703 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DI-TERT-BUTYLHYDROQUINONE CHEMBL480626 72904 49704 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649837 72906 49705 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-4283 CHEMBL606166 72907 49706 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ANANDAMIDE ANANDAMIDE 72908 49707 TSPO 706 DRUGGABLE GENOME Phenylpurine acetamide analog 1 72909 49708 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE APLAVIROC HYDROCHLORIDE APLAVIROC HYDROCHLORIDE 72910 49709 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING BUTYRYLHYDROXAMIC ACID BUTYRYLHYDROXAMIC ACID 21874153 72911 49710 TUBB4B 10383 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 72912 49711 KDM4A 9682 DRUGGABLE GENOME, ENZYME CAPSAZEPINE CAPSAZEPINE 72914 49712 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SJ000072878 CHEMBL601400 72917 49713 LIPC 3990 ENZYME, PHOSPHOLIPASE, LIPASE, DRUGGABLE GENOME simvastatin SIMVASTATIN 16103896 72918 49714 MAPT 4137 DRUGGABLE GENOME R(-)-PROPYLNORAPOMORPHINE HCL CHEMBL538542 72920 49715 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE NERAMEXANE NERAMEXANE 72921 49716 RPS6KA5 9252 DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE LINIFANIB LINIFANIB 72922 49717 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR VCR 12007564 72925 49718 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR OCTYL_GALLATE OCTYL_GALLATE 72927 49719 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TERCONAZOLE TERCONAZOLE 72928 49720 SLC25A5 292 DRUGGABLE GENOME, TRANSPORTER BUTYRATE 10657244 72929 49721 PDE10A 10846 ENZYME, DRUGGABLE GENOME Triazolo-pyridine derivative 5 72930 49722 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 1,5-NAPHTHALENEDIAMINE CHEMBL538965 72931 49723 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME MEMANTINE MEMANTINE 72932 49724 ATP1B1 481 DRUGGABLE GENOME, TRANSPORTER, ENZYME inhibitor CHEMBL1614 DESLANOSIDE 72933 49725 KDM4A 9682 DRUGGABLE GENOME, ENZYME NITROXOLINE NITROXOLINE 72934 49726 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3348923 MLN-2480 72935 49727 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PURPUROGALLIN PURPUROGALLIN 72937 49728 ZEB1 6935 TRANSCRIPTION FACTOR, DRUG RESISTANCE SALINOMYCIN SALINOMYCIN 24013721 72940 49729 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PEITC 12819185 72941 49730 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL antagonist 178102530 72944 49731 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME INTERFERON BETA-1A 12117359 72945 49732 MAPT 4137 DRUGGABLE GENOME RATANIAPHENOL II RATANIAPHENOL II 72947 49733 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIBUTYLDICHLOROSTANNANE DIBUTYLDICHLOROSTANNANE 72948 49734 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE DIGOXIN DIGOXIN 72949 49735 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIPERINE PIPERINE 72950 49736 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 374883892 72951 49737 MAPT 4137 DRUGGABLE GENOME TRIBROMSALAN TRIBROMSALAN 72952 49738 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR TAMATINIB R-406 72953 49739 SLC15A2 6565 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101227 72954 49740 HDAC11 79885 DRUGGABLE GENOME, ENZYME 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 23622981 72955 49741 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200833 DIPIVEFRIN HYDROCHLORIDE 72956 49742 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 223365984 LUCITANIB 72957 49743 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135652664 ALCURONIUM 72958 49744 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TDR77593 CHEMBL1510164 72959 49745 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BGB-283 LIFIRAFENIB 72960 49746 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DISULFIRAM DISULFIRAM 72961 49747 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DITIOCARB SODIUM DITIOCARB SODIUM 72965 49748 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR granisetron GRANISETRON 29177570 72970 49749 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME N/A 72971 49750 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL inhibitor 374883890 72972 49751 CCL3 6348 KINASE, DRUGGABLE GENOME ADJUVANT 17116174 72973 49752 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR SB-203580 SB-203580 25692815 72974 49753 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID27744724-Compound-21 72976 49754 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR digoxin DIGOXIN 22543981 72977 49755 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR modulator CHEMBL3545355 CHF4227 72978 49756 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3-HYDROXY-3',4'-DIMETHOXYFLAVONE 3-HYDROXY-3',4'-DIMETHOXYFLAVONE 72980 49757 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PENTACHLOROPHENOL PENTACHLOROPHENOL 72982 49758 BMP7 655 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR dexamethasone DEXAMETHASONE 26590194 72983 49759 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PICEATANNOL PICEATANNOL 72984 49760 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 328083479 72986 49761 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE INDAPAMIDE INDAPAMIDE 72988 49762 KDM4A 9682 DRUGGABLE GENOME, ENZYME HYDROXYTYROSOL HYDROXYTYROSOL 72990 49763 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME RAFOXANIDE RAFOXANIDE 72991 49764 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE DOVITINIB DOVITINIB 72992 49765 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE Alfa-interferon 72993 49766 COL1A2 1278 DRUGGABLE GENOME TGF-BETA 2 15223827 72994 49767 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor DABRAFENIB MESYLATE 72995 49768 PSMD7 5713 PROTEASE inhibitor CHEMBL325041 BORTEZOMIB 72996 49769 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 178103951 DINACICLIB 72998 49770 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX 6,4'-DIMETHOXYFLAVONE 6,4'-DIMETHOXYFLAVONE 72999 49771 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE CD40L 10725717,10202112 73000 49772 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GNF-PF-1083 CHEMBL530361 73001 49773 CYP2A6 1548 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 pilocarpine PILOCARPINE 11394901,16402128,15940289,16952495,19238117,18698229,16891249,10544257,15660270,20860463,11241319,15475735,18212800,20089352,11725533,19921195,15980104,11237731,19845430,10999944,20155256,16272956,17130279,12042667,15900015,21494765,10448083,20596643,12223434,12844137,19604090,15265511,15308589,21521021,16452582,19225447,11779172,12749606,17178767,18380793,14981342,17220563,17112802 73003 49774 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CRIZOTINIB CRIZOTINIB 24162815 73007 49775 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 315661265 73009 49776 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME clindamycin CLINDAMYCIN 27527109 73010 49777 CSNK1E 1454 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 249565730 CHEMBL2069623 73012 49778 POLI 11201 DNA REPAIR METHYLENE BLUE METHYLENE BLUE 73014 49779 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201630 INSULIN PURIFIED PORK 73017 49780 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ticagrelor TICAGRELOR 25935875 73019 49781 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME lovastatin LOVASTATIN 22281720 73023 49782 PBRM1 55193 CLINICALLY ACTIONABLE DURVALUMAB DURVALUMAB 29301960 73025 49783 USP1 7398 DNA REPAIR, PROTEASE, ENZYME EMODIC ACID EMODIC ACID 73026 49784 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 53801036 73027 49785 NDUFS1 4719 ENZYME inhibitor CHEMBL3545135 NV-128 73030 49786 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103659 73032 49787 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor PLX3603 73033 49788 S100A4 6275 NA GNF-PF-4459 CHEMBL585502 73035 49789 MPHOSPH8 54737 NA CATECHOL CATECHOL 73037 49790 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE IDARUBICIN HYDROCHLORIDE IDARUBICIN HYDROCHLORIDE 73038 49791 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178100978 73041 49792 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178100961 ASPIRIN 73046 49793 GMNN 51053 DRUGGABLE GENOME DIMETHYL SUCCINATE DIMETHYL SUCCINATE 73049 49794 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME QUERCETIN QUERCETIN 73050 49795 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME MARIMASTAT MARIMASTAT 73052 49796 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL activator 135652668 73053 49797 ECE1 1889 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE SLV-334 SLV-334 73054 49798 POLI 11201 DNA REPAIR PHENYLSTIBONIC ACID PHENYLSTIBONIC ACID 73055 49799 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-124266 CHEMBL124006 73056 49800 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL activator 178101135 73058 49801 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME BICALUTAMIDE BICALUTAMIDE 10075669 73059 49802 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SERATRODAST SERATRODAST 73061 49803 TOP2B 7155 DRUGGABLE GENOME, ENZYME XK-469 73062 49804 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE ABT-737 ABT 737 27974663 73064 49805 PURA 5813 NA methylphenidate METHYLPHENIDATE 29382897 73065 49806 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL DIAZEPAM DIAZEPAM 73067 49807 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Imidazo bicyclic iminium derivative 7 73068 49808 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX DNDI1417548 CHEMBL2094789 73069 49809 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR PURPURIN PURPURIN 73070 49810 BMP2 650 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DWP-431 73071 49811 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103638 BECLOMETHASONE DIPROPIONATE 73072 49812 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 374883887 73073 49813 HTT 3064 DRUGGABLE GENOME PMID29671355-Compound-69 73075 49814 ATAD5 79915 NA FIDUXOSIN FIDUXOSIN 73079 49815 ATAD5 79915 NA ENTINOSTAT ENTINOSTAT 73081 49816 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR partial agonist CHEMBL500 PINDOLOL 73082 49817 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME ZOLANTIDINE ZOLANTIDINE 73083 49818 CD44 960 DRUGGABLE GENOME, CELL SURFACE MOMETASONE FUROATE 12877820 73086 49819 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-45382 CHEMBL1214274 73087 49820 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE inhibitor CHEMBL1704 TIROFIBAN HYDROCHLORIDE 73088 49821 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 381118858 73089 49822 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZIRAM ZIRAM 73090 49823 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE CHEMBL1255944 73091 49824 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER BRYOSTATIN BRYOSTATIN 22579485 73092 49825 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TCMDC-123480 CHEMBL588683 73093 49826 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRETINOIN TRETINOIN 73095 49827 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102666 73096 49828 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME SB-216763 SB-216763 73097 49829 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE RO4929097 RG-4733 27556950 73098 49830 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MNU 16344269 73099 49831 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE EPINEPHRINE EPINEPHRINE 15210061 73100 49832 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE busulfan BUSULFAN 73101 49833 RGS2 5997 NA haloperidol HALOPERIDOL 27023437 73102 49834 P4HTM 54681 TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL2338329 ROXADUSTAT 73103 49835 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL3545252 DOCETAXEL 73105 49836 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ACAMPROSATE CALCIUM ACAMPROSATE CALCIUM 73106 49837 TLR7 51284 DRUGGABLE GENOME NKTR-262 73108 49838 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TRASTUZUMAB EMTANSINE 27900589,24793816,31504139,29989854,28526536,24898067,25789838,23382472,21172893,23020162 73109 49839 BAZ2B 29994 NA ZINC 03369470 CHEMBL599013 73111 49840 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Balaglitazone BALAGLITAZONE 73112 49841 USP1 7398 DNA REPAIR, PROTEASE, ENZYME IRL-2500 CHEMBL72410 73114 49842 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CID 887167 CHEMBL260342 73116 49843 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME DIPYRIDAMOLE DIPYRIDAMOLE 73117 49844 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME SB-220025 SB-220025 73118 49845 SMARCA4 6597 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING RETINOIC ACID 9315656 73119 49846 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL ADINAZOLAM ADINAZOLAM 73120 49847 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32k 73121 49848 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR RESVERATROL RESVERATROL 73122 49849 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME METHOTREXATE METHOTREXATE 73123 49850 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME GLUCAGON GLUCAGON 2552996 73125 49851 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Bis-aminopyrimidine derivative 2 73126 49852 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CLOTIAZEPAM CLOTIAZEPAM 73127 49853 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TOZADENANT TOZADENANT 73130 49854 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME DORAMAPIMOD DORAMAPIMOD 73132 49855 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051818 73133 49856 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SYROSINGOPINE SYROSINGOPINE 73136 49857 NOS1 4842 DRUGGABLE GENOME, ENZYME ESTROGEN ANTAGONIST 7515189 73138 49858 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR IDARUBICIN IDARUBICIN 8915668 73139 49859 MAOA 4128 DRUGGABLE GENOME, ENZYME 8-(3-CHLOROBENZYLOXY)CAFFEINE CHEMBL602260 20093036 73140 49860 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL1079593 VS-5584 73141 49861 KDM1B 221656 DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING, ENZYME Tarnylcypromine derivative 2 73142 49862 CHI3L1 1116 CELL SURFACE, DRUGGABLE GENOME CHEMOKINES 15015934 73143 49863 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor NERATINIB NERATINIB 73144 49864 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CENISERTIB CENISERTIB 73145 49865 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor CHEMBL574737 UCN-01 73146 49866 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TANSHINONE IIA TANSHINONE IIA 73148 49867 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL antagonist 135651219 SURAMIN 73150 49868 USP1 7398 DNA REPAIR, PROTEASE, ENZYME S-(P-AZIDOPHENACYL)GLUTATHIONE CHEMBL1256813 73151 49869 F5 2153 DRUGGABLE GENOME DROTRECOGIN ALFA 73153 49870 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER NIMODIPINE NIMODIPINE 14743973 73154 49871 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE inhibitor 249565929 73155 49872 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME SKIMMIANINE SKIMMIANINE 73156 49873 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME QUINACRINE DIHYDROCHLORIDE QUINACRINE DIHYDROCHLORIDE 73157 49874 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102545 73158 49875 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SAR260301 SAR-260301 27196754 73159 49876 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME SP-600125 SP-600125 73160 49877 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW290597X GW290597X 73161 49878 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 4-AMINOPHENOL 4-AMINOPHENOL 73162 49879 UGT2B15 7366 DRUGGABLE GENOME acetaminophen ACETAMINOPHEN 30908574,26049587,16696573 73164 49880 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL1059 PREGABALIN 73165 49881 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME DABRAFENIB DABRAFENIB 23020132,22608338,26619011,21483012,22351686,19001320,21156289,20368568,19255327,22048237,19561230,19010912,23549875,25024077,23489023,18541894,24586605,24508103,22773810,23833300,23812671,24576830,19238210,20818844,23612012,23251002,22356324,20857202,22536370,22997239,21163703,15035987,23470635,21663470,24594804,22586120,20413299,22805292,19537845,14679157,22663011,21975775,22038996,22448344,12068308,24163374,19773371,24354346,23325582,24583796,23031422,22735384,21683865,25370471,21639808,22281684,22649091,22241789,24570209,23918947,25989278,22389471,23934108,22180495,23524406,26678033,19018267,24388723,23845441,23614898,25157968,20619739,12460919,24107445,12460918,21594703,20350999,20630094,21426297,19404918,22743296,24396464,22972589,21129611,23406027,25656898 73167 49882 TOP2B 7155 DRUGGABLE GENOME, ENZYME Annamycin liposomal 73168 49883 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ANTIFOLATES 9256160 73171 49884 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-405662 CHEMBL118378 73174 49885 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CEPHALOCHROMIN CEPHALOCHROMIN 73175 49886 TMEM97 27346 NA N-substituted 9-azabicyclo[3.3.1]nonan-3alpha-yl-phenylcarbamate analog 2 73178 49887 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-59 73179 49888 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME PMID27539678-Compound-10 73180 49889 DNPEP 23549 ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL2103847 TOSEDOSTAT 73181 49890 ALOX5 240 DRUGGABLE GENOME, ENZYME E-6700 73182 49891 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL3137320 TALAZOPARIB 73183 49892 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor PX-866 SONOLISIB 73184 49893 LIPA 3988 ENZYME, DRUGGABLE GENOME SBC-102 SEBELIPASE ALFA 73185 49894 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-28 73186 49895 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR MLN-8054 MLN-8054 73187 49896 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 328083473 CHEMBL1951415 73188 49897 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 178102002 PRIMIDONE 73189 49898 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GALANGIN GALANGIN 73190 49899 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ISOETHARINE ISOETHARINE 73191 49900 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE PMA 10918054 73193 49901 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL1551 URSODIOL 73199 49902 APH1B 83464 PROTEASE, DRUGGABLE GENOME SEMAGACESTAT SEMAGACESTAT 19443228 73200 49903 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NORETHINDRONE NORETHINDRONE 73201 49904 CA2 760 DRUGGABLE GENOME, ENZYME Dichlorphenamide DICHLORPHENAMIDE 73202 49905 UGCG 7357 ENZYME, DRUGGABLE GENOME Genz-682452 VENGLUSTAT 73203 49906 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE TENECTEPLASE TENECTEPLASE 73204 49907 IL1B 3553 KINASE, DRUGGABLE GENOME ABT-981 73205 49908 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ALT-801 ALT-801 73206 49909 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME activator 135651046 73208 49910 MARCKSL1 65108 KINASE HERBIMYCIN A 11483670 73209 49911 HTT 3064 DRUGGABLE GENOME TCMDC-123868 CHEMBL548615 73210 49912 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 178102513 PONATINIB 73211 49913 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200708 BISOPROLOL FUMARATE 73213 49914 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL1742994 BRENTUXIMAB VEDOTIN 73214 49915 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PMID29671355-Compound-25 73215 49916 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ELLAGIC ACID ELLAGIC ACID 73216 49917 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102667 73217 49918 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE SPC4955 73218 49919 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ETHISTERONE ETHISTERONE 73219 49920 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-55 73220 49921 PSMA1 5682 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL371405 MARIZOMIB 73222 49922 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650503 73223 49923 HPSE 10855 ENZYME, DRUGGABLE GENOME Suramin SURAMIN 73224 49924 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1059 PREGABALIN 73225 49925 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE cisplatin CISPLATIN 73226 49926 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GRAVEOLINE GRAVEOLINE 73227 49927 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650458 SILODOSIN 73228 49928 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR NVP-AEW541 AEW-541 28637688 73229 49929 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ENDOXIFEN ENDOXIFEN 73231 49930 TMEM97 27346 NA Aryl azepine derivative 2 73235 49931 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL3545365 ALTIRATINIB 73236 49932 NCF1 653361 ENZYME HYDROGEN PEROXIDE 15840036 73237 49933 DIABLO 56616 NA ANTIOXIDANT 16115949 73238 49934 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 310264693 ACALABRUTINIB 73239 49935 GSTA1 2938 ENZYME, DRUGGABLE GENOME doxorubicin DOXORUBICIN 29938344,24215845,19448608 73241 49936 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CYSTEINE METHYL-ESTER HCL CHEMBL1426508 73242 49937 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565863 73243 49938 TH 7054 ENZYME, DRUGGABLE GENOME opioids 29210332,32232669 73244 49939 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR RALOXIFEN RALOXIFEN 73247 49940 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME BAY1834845 73248 49941 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AZD8931 SAPITINIB 73249 49942 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE IODOQUINOL IODOQUINOL 73250 49943 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BIOMODULATORS 8603452 73253 49944 COL1A2 1278 DRUGGABLE GENOME COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 73254 49945 ALOX15 246 ENZYME, DRUGGABLE GENOME SILVER SULFADIAZINE SILVER SULFADIAZINE 73257 49946 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZELNIDIPINE AZELNIDIPINE 73260 49947 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME SNDX-6352 73261 49948 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 178102341 73262 49949 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 318164795 TOREFORANT 73264 49950 PPIA 5478 DRUGGABLE GENOME, ENZYME CYCLOSPORINE CYCLOSPORINE 19933795 73266 49951 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR QUINOCIDE QUINOCIDE 73268 49952 CD52 1043 DRUGGABLE GENOME ALEMTUZUMAB ALEMTUZUMAB 73270 49953 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Bis-aminopyrimidine derivative 2 73271 49954 KDM4A 9682 DRUGGABLE GENOME, ENZYME A-443654 A-443654 73273 49955 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32q 73277 49956 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417099 CHEMBL1565444 73278 49957 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ALVIMOPAN ALVIMOPAN 73279 49958 CXCL8 3576 DRUGGABLE GENOME OMEPRAZOLE OMEPRAZOLE 17122965 73280 49959 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME PF-562271 PF-00562271 73281 49960 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 22931300 73283 49961 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3792 CHEMBL582983 73285 49962 IL1B 3553 KINASE, DRUGGABLE GENOME Diacerein DIACEREIN 73286 49963 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL12 DIAZEPAM 73287 49964 BMPR1B 658 DRUGGABLE GENOME, CELL SURFACE, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 249565835 73288 49965 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR allosteric modulator 178102293 SELUMETINIB 73289 49966 MTTP 4547 DRUGGABLE GENOME IMPLITAPIDE IMPLITAPIDE 73290 49967 RACGAP1 29127 NA NSC-95397 CHEMBL429095 73291 49968 TRPV2 51393 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker 135651058 73292 49969 GMNN 51053 DRUGGABLE GENOME GNF-PF-1307 CHEMBL585030 73293 49970 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE THRX-198321 73294 49971 FAAH 2166 ENZYME, DRUGGABLE GENOME olanzapine OLANZAPINE 20631561 73297 49972 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME montelukast MONTELUKAST 28940478 73298 49973 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL592445 GEDATOLISIB 73299 49974 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIPROLIDINE HYDROCHLORIDE TRIPROLIDINE HYDROCHLORIDE 73300 49975 CCL5 6352 CELL SURFACE, ENZYME, KINASE, DRUGGABLE GENOME OX40 LIGAND 12161277 73301 49976 PSMC6 5706 NA inhibitor BORTEZOMIB BORTEZOMIB 73302 49977 HMGCR 3156 ENZYME, DRUGGABLE GENOME Poly-substituted azoles statin lactone derivative 1 73304 49978 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125821 CHEMBL547977 73306 49979 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US9682991, 23 73307 49980 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PONATINIB PONATINIB 20512393,14745431,20537386,11861307,15256422,11423618,20963643,22772060,22306673,23676790,11853795,22870928,20697894,21872826,12623848,19466505,12130516,20367437,17114651,18828913,24236021,15381060,23540562,21895409,21489624,23355941,11964322,24456693,18615627,25157968,14559829,21605905,21562040,21505103,19652056,15194504,21762985,12399961 73308 49981 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1409 FLUVOXAMINE MALEATE 73310 49982 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 178101159 IVACAFTOR 73311 49983 HTT 3064 DRUGGABLE GENOME 2-PHENYLAMINO-[1,4]NAPHTHOQUINONE CHEMBL84010 73313 49984 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE XL147 PILARALISIB 24166903,25637314,21216929 73316 49985 MAOB 4129 DRUGGABLE GENOME, ENZYME Tarnylcypromine derivative 3 73321 49986 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CETUXIMAB CETUXIMAB 26619011,19455431,22452896,24934779,23102728,20068085,16707764,17653080,15710947,20479403,25668228,16912157,24893891,15728811,20573926,16258541,19692680,15118125,18227510,24658966,18199554,19922469,20033049,26515464,25923549,21783417,19692684,22753918,16187797,22452895,23945392,15329413,24636847,23816963,24729716,23816960,22285168,19096302,16204070,22270724,24894453,16043828,22215752,21194487,24065731,15118073,20022809,23948351,16115929,18458038,17332364,24623981,19147750,25157968,16011858,21430269,23578570,2302402,15737014,26720284,21670455,21233402,23242437,25923550,22588155,21531810,18303429,19671738,18089823 73322 49987 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650347 73323 49988 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX ALPELISIB ALPELISIB 25002028 73324 49989 HMGCS2 3158 DRUGGABLE GENOME, ENZYME chlorothiazide CHLOROTHIAZIDE 29523524 73329 49990 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 385612240 73331 49991 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 atorvastatin ATORVASTATIN 73333 49992 F5 2153 DRUGGABLE GENOME lusutrombopag LUSUTROMBOPAG 73334 49993 MAPT 4137 DRUGGABLE GENOME 9,10-PHENANTHRENEQUINONE 9,10-PHENANTHRENEQUINONE 73337 49994 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PREGNENOLONE PREGNENOLONE 73338 49995 GMNN 51053 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 73339 49996 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor IMATINIB MESYLATE 73340 49997 TUBB6 84617 DRUGGABLE GENOME NSC-753582 CHEMBL2036124 22543234 73342 49998 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PA-824 PRETOMANID 73344 49999 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ETHYL 2,4,6-TRIHYDROXYBENZOATE CHEMBL2204435 22579484 73345 50000 SRD5A1 6715 DRUGGABLE GENOME inhibitor CHEMBL1200969 DUTASTERIDE 73346 50001 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE KU-55933 KU-55933 25870146 73348 50002 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE cetuximab CETUXIMAB 22117530,16788380,18349392 73350 50003 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor RUXOLITINIB RUXOLITINIB 73351 50004 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Cyanomethyl pypazole carboxamide derivative 1 73352 50005 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE TOPIRAMATE TOPIRAMATE 73353 50006 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE RADICICOL RADICICOL 10349833 73356 50007 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR RALOXIFENE RALOXIFENE 73357 50008 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME VORINOSTAT VORINOSTAT 21696956,24766560,19344175,24304348,21080647,19966789,26211462,23622981,22260166,20491440,21548582,23672185,26331334,19084294 73358 50009 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR EGCG EPIGALOCATECHIN GALLATE 9000119,15637567 73359 50010 LANCL2 55915 NA 384403644 73361 50011 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ISOTHYMONIN ISOTHYMONIN 73363 50012 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL29741 IRAMPANEL 73365 50013 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX VP-16 ETOPOSIDE PHOSPHATE 12046067 73366 50014 PDE10A 10846 ENZYME, DRUGGABLE GENOME 1,2,4-triazole [4,3-a]quinoxaline derivative 2 73367 50015 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Lapatinib LAPATINIB 73368 50016 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178103317 73370 50017 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME CART-BCMA 73372 50018 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Topotecan TOPOTECAN 26438783 73373 50019 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DACOMITINIB DACOMITINIB 73374 50020 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME celecoxib CELECOXIB 22336956 73377 50021 SLC2A1 6513 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE 17 BETA-ESTRADIOL 9227446 73381 50022 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME RESERPINE RESERPINE 16081063 73382 50023 XRCC4 7518 KINASE radiotherapy 28796378 73383 50024 PARD3B 117583 NA fluorouracil FLUOROURACIL 22310351 73387 50025 CA12 771 DRUGGABLE GENOME Sulfamylon SULFAMYLON 73389 50026 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor INCB018424 RUXOLITINIB 73390 50027 BCHE 590 DRUGGABLE GENOME, ENZYME Decyle nelycorine dibromo salt derivative 1 73391 50028 POLK 51426 DNA REPAIR, ENZYME ORTHO-PHTHALALDEHYDE ORTHO-PHTHALALDEHYDE 73392 50029 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-26 73393 50030 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL VERAPAMIL VERAPAMIL 73396 50031 GUCY2C 2984 DRUGGABLE GENOME, KINASE agonist 178101643 73397 50032 NOS1AP 9722 NA dolasetron DOLASETRON 21663814 73398 50033 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100686 73400 50034 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NILUTAMIDE NILUTAMIDE 22931300 73401 50035 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL3707402 PF-06372865 73402 50036 RGS4 5999 DRUGGABLE GENOME XCT790 CHEMBL189753 73403 50037 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE FORETINIB FORETINIB 23213094 73404 50038 INPPL1 3636 KINASE, ENZYME, DRUGGABLE GENOME ANTISENSE OLIGONUCLEOTIDES 10958682 73406 50039 ITPR3 3710 ION CHANNEL, DRUGGABLE GENOME activator 178101039 73408 50040 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1201047 ANILERIDINE HYDROCHLORIDE 73413 50041 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Amidopyrazole derivative 3 73414 50042 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR TANESPIMYCIN TANESPIMYCIN 73415 50043 HEBP1 50865 DRUGGABLE GENOME Diterpenoid derivative 1 73416 50044 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME NF-KB DECOY 73417 50045 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE PF-4708671 73419 50046 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE vardenafil VARDENAFIL 21934637 73420 50047 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SORAFENIB SORAFENIB 24569458 73421 50048 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR MER-102 73422 50049 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 363894219 BALAMAPIMOD 73423 50050 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-9037 CHEMBL1451216 73425 50051 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ALTENUSIN ALTENUSIN 73426 50052 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1201003 ELETRIPTAN HYDROBROMIDE 73427 50053 MAPT 4137 DRUGGABLE GENOME DNDI1318925 CHEMBL1390716 73428 50054 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL272980 MOCETINOSTAT 73429 50055 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DEOXIEPINEPHRINE DEOXIEPINEPHRINE 73430 50056 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE TAE-684 TAE-684 22335897 73432 50057 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE AZD-5122 73433 50058 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BMS-754807 BMS-754807 26725216 73434 50059 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME SB-202190 SB-202190 22951114 73435 50060 DHODH 1723 DRUGGABLE GENOME, ENZYME VIDOFLUDIMUS VIDOFLUDIMUS 73436 50061 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL598797 CUDC-101 73437 50062 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PASIREOTIDE PASIREOTIDE 73438 50063 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SB-203580 SB-203580 73439 50064 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME DOVITINIB DOVITINIB 73440 50065 TUBB6 84617 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 73441 50066 TUBB2B 347733 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 73442 50067 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SHP099 27362227 73443 50068 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME VITAMIN E 9750015,16166287 73444 50069 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ONO-7579 73445 50070 HDAC11 79885 DRUGGABLE GENOME, ENZYME PMID29671355-Compound-25 73447 50071 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER melphalan MELPHALAN 73448 50072 TARDBP 23435 TUMOR SUPPRESSOR EQUILIN EQUILIN 73449 50073 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DACTINOMYCIN DACTINOMYCIN 73450 50074 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HYDROQUINONE HYDROQUINONE 15833037 73452 50075 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1696 DESIPRAMINE HYDROCHLORIDE 73453 50076 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE QUARFLOXIN QUARFLOXIN 28211448 73454 50077 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 8 73455 50078 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565601 ONVANSERTIB 73456 50079 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ICRF-193 ICRF-193 73458 50080 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME EVANS BLUE EVANS BLUE 73459 50081 GMNN 51053 DRUGGABLE GENOME TRIFLUPROMAZINE HYDROCHLORIDE TRIFLUPROMAZINE HYDROCHLORIDE 73460 50082 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Selumetinib SELUMETINIB 26438159 73461 50083 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE OLAPARIB OLAPARIB 31157963,23346317,30345884,25366685,19553641,28792849,25218906,28578601,21862407,30797618,31538027,24882434 73463 50084 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE JNJ-7706621 JNJ-7706621 73464 50085 BUB1 699 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME SCHEMBL16322760 73467 50086 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME SORAFENIB SORAFENIB 73469 50087 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CR-845 iv infusion 19430912 73473 50088 POLK 51426 DNA REPAIR, ENZYME CEFOTETAN CEFOTETAN 73475 50089 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DEXTROMETHORPHAN DEXTROMETHORPHAN 12151071 73476 50090 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BAS-8770949 CHEMBL476025 19179076 73477 50091 ABCG1 9619 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME irinotecan IRINOTECAN 26352872 73478 50092 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL3545298 AZD-6918 73481 50093 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TARENFLURBIL TARENFLURBIL 73482 50094 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR HEPARIN HEPARIN 73484 50095 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135649714 73485 50096 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME MNU 10391687 73487 50097 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR HEXACHLOROPHENE HEXACHLOROPHENE 73488 50098 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE Almitrine ALMITRINE 73490 50099 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TRACAZOLATE TRACAZOLATE 73493 50100 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Anti-CD123 CAR-T cells 73494 50101 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1723343 ZOLPIDEM TARTRATE 73495 50102 OGDH 4967 NA valproic acid 23407051 73496 50103 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR 1-PHYTEN-3-OL CHEMBL453797 73500 50104 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX MORUSINOL MORUSINOL 24901948 73501 50105 KIF11 3832 DRUGGABLE GENOME MK-0731 CHEMBL481931 73502 50106 ALOX5 240 DRUGGABLE GENOME, ENZYME UCB-35440 73503 50107 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ILORASERTIB ILORASERTIB 73504 50108 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME SP-600125 SP-600125 73505 50109 MAOB 4129 DRUGGABLE GENOME, ENZYME MOFEGILINE MOFEGILINE 19053775 73507 50110 PSMD1 5707 NA CARFILZOMIB CARFILZOMIB 24524217 73508 50111 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME N-methylmethanesulfonamide derivative 1 73509 50112 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BECLOMETHASONE DIPROPIONATE BECLOMETHASONE DIPROPIONATE 73511 50113 TNNT2 7139 DRUGGABLE GENOME NSC-107022 CHEMBL1601846 73512 50114 CP 1356 DRUGGABLE GENOME, ENZYME TETRANDRINE 10682587 73513 50115 SLC40A1 30061 TRANSPORTER, DRUGGABLE GENOME antibody 252166626 73514 50116 PTPRD 5789 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Antihypertensives 73515 50117 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ARSENIC TRIOXIDE 15587394,16950207 73518 50118 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER LOVASTATIN LOVASTATIN 15616150,10213372 73519 50119 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650621 MOLINDONE 73520 50120 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 2-(METHYLSULFONAMIDO)BENZOIC ACID CHEMBL491550 73521 50121 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME JQ1 20871596 73523 50122 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME ADXS-PSA 73524 50123 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CHLORPROPAMIDE CHLORPROPAMIDE 73526 50124 SETD4 54093 METHYL TRANSFERASE doxorubicin DOXORUBICIN 19204081 73528 50125 FAAH 2166 ENZYME, DRUGGABLE GENOME Boronic acid derivative 1 73529 50126 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR RHIL-11 7694867 73530 50127 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Aminocaproic Acid 73533 50128 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 178103458 VORINOSTAT 73535 50129 FBXW7 55294 DNA REPAIR, CLINICALLY ACTIONABLE MRK-003 17646409 73536 50130 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 336446906 73537 50131 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME MLN-8054 MLN-8054 73540 50132 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE ELLIPTECINE ELLIPTECINE 73541 50133 TUBA1B 10376 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 73543 50134 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME INCB039110 ITACITINIB 73544 50135 PEBP1 5037 KINASE, PROTEASE INHIBITOR DHT ANDROSTANOLONE 12417618 73545 50136 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR FESOTERODINE FESOTERODINE 73546 50137 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PMID25416646-Compound-Figure2-K 73548 50138 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135651137 73549 50139 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE HEXAHYDROCURCUMIN HEXAHYDROCURCUMIN 19112019 73550 50140 ALOX15B 247 DRUGGABLE GENOME, ENZYME CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 73551 50141 MTR 4548 ENZYME, DRUGGABLE GENOME cisplatin CISPLATIN 21605004,29662106,19159907 73552 50142 HSPB2 3316 KINASE VCR 16525997 73553 50143 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor 178102628 73554 50144 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BERBERINE CHLORIDE BERBERINE CHLORIDE 73555 50145 HTT 3064 DRUGGABLE GENOME INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 73556 50146 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER fluoxetine FLUOXETINE 24192121,18215618,24663076 73557 50147 XDH 7498 DRUGGABLE GENOME, ENZYME Fused heterocyclic compound 11 73558 50148 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER CEFOPERAZONE CEFOPERAZONE 22166395 73560 50149 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME RO-137410 CHEMBL275311 73562 50150 GJB2 2706 ION CHANNEL, TRANSPORTER inhibitor 178101095 OCTANOL 73563 50151 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178103826 OXAPROZIN 73567 50152 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHENYLARSINE OXIDE PHENYLARSINE OXIDE 73568 50153 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DOCEBENONE DOCEBENONE 73569 50154 TUBA1B 10376 DRUGGABLE GENOME ABT-751 ABT-751 25468039 73570 50155 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER METHYLBENZETHONIUM CHLORIDE METHYLBENZETHONIUM CHLORIDE 73571 50156 BAP1 8314 PROTEASE, TUMOR SUPPRESSOR, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE TRICHOSTATIN A 22038994 73572 50157 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor 404859105 73573 50158 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200903 SECOBARBITAL SODIUM 73575 50159 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR SL-327 CHEMBL261237 73576 50160 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Toremifene TOREMIFENE 73577 50161 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-223133 CHEMBL1888586 73578 50162 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE GSK-269962A GSK-269962A 73580 50163 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2107771 RALFINAMIDE 73583 50164 GJB2 2706 ION CHANNEL, TRANSPORTER inhibitor 135650269 73585 50165 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE CENISERTIB CENISERTIB 73586 50166 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BUPIRIMATE BUPIRIMATE 73587 50167 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Nilotinib NILOTINIB 18794084 73588 50168 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101339 73589 50169 CD44 960 DRUGGABLE GENOME, CELL SURFACE A-6 73592 50170 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 381118896 73594 50171 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 73595 50172 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL1079593 VS-5584 73596 50173 SUGCT 79783 ENZYME hormonal contraceptives for systemic use 28750087 73599 50174 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID27744724-Compound-18 73600 50175 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DESLANOSIDE DESLANOSIDE 73604 50176 CES1 1066 DRUGGABLE GENOME, ENZYME HL-004 73605 50177 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GNF-PF-1678 CHEMBL580340 73607 50178 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor 374883851 73609 50179 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME OSI-027 OSI-027 73611 50180 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR 16282176 73612 50181 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME LY-294002 LY-294002 73613 50182 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME R763 73615 50183 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CETUXIMAB CETUXIMAB 28275037,20619739 73616 50184 ANGPT1 284 KINASE, DRUGGABLE GENOME, FIBRINOGEN AMG 780 73618 50185 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR Doxorubicin DOXORUBICIN 25605023 73619 50186 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE Ixazomib IXAZOMIB 26634271 73620 50187 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 73622 50188 PTGS2 5743 DRUGGABLE GENOME, ENZYME NAPROXCINOD NAPROXCINOD 73624 50189 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CISPLATIN CISPLATIN 73625 50190 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE AMG 337 73626 50191 HSPA4 3308 NA KINASE INHIBITOR 2010034 73628 50192 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 315661180 ZOTIRACICLIB 73630 50193 EYA2 2139 DNA REPAIR CARMINE CARMINE 73631 50194 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME 123-Iodine-labeled MFE-23 10677374 73632 50195 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AFIMOXIFENE AFIMOXIFENE 20179196 73635 50196 ATXN2 6311 NA ENCLOMIPHENE ENCLOMIPHENE 73638 50197 BCL2L2 599 CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID27744724-Compound-18 73639 50198 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 381118806 ACALISIB 73640 50199 MAPT 4137 DRUGGABLE GENOME APOMORPHINE APOMORPHINE 73643 50200 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CI-1040 CI-1040 73644 50201 NR1D2 9975 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 310264681 SR9011 73646 50202 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE DOVITINIB DOVITINIB 73647 50203 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 249565870 73649 50204 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME JNJ-7706621 JNJ-7706621 73650 50205 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DINITROPHENYLENE DINITROPHENYLENE 73651 50206 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE OLAPARIB OLAPARIB 28490518 73652 50207 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER (R)-INDOPROFEN (R)-INDOPROFEN 73653 50208 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 249565812 73659 50209 GHRL 51738 DRUGGABLE GENOME TNF-ALPHA 17187875 73660 50210 KDM4A 9682 DRUGGABLE GENOME, ENZYME ROXARSONE ROXARSONE 73662 50211 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LOVASTATIN LOVASTATIN 22931300 73663 50212 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME Romiplostim ROMIPLOSTIM 22970246 73664 50213 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 178100691 73665 50214 MAOB 4129 DRUGGABLE GENOME, ENZYME SELEGILINE SELEGILINE 73666 50215 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102423 D-TRYPTOPHAN 73667 50216 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651393 73668 50217 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL378544 VINBLASTINE SULFATE 73672 50218 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CARMINIC ACID CARMINIC ACID 73673 50219 TMEM97 27346 NA Isoindoline derivative 4 73674 50220 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SERTACONAZOLE NITRATE SERTACONAZOLE NITRATE 73676 50221 PDE4A 5141 DRUGGABLE GENOME, ENZYME Oxtriphylline OXTRIPHYLLINE 73677 50222 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR NELFINAVIR MESYLATE NELFINAVIR MESYLATE 73678 50223 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME everolimus EVEROLIMUS 25893859 73679 50224 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135650658 73681 50225 RACGAP1 29127 NA CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM BROMIDE 73683 50226 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE VINCRISTINE VINCRISTINE 2804079 73684 50227 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 363894235 73685 50228 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Inecalcitol oral 73687 50229 KDM4A 9682 DRUGGABLE GENOME, ENZYME ASTERRIC ACID ASTERRIC ACID 73688 50230 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Ibuprofen IBUPROFEN 73689 50231 IL13RA1 3597 EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE, DRUGGABLE GENOME AER001,AEROVANT 73690 50232 ACO1 48 ENZYME ANTIOXIDANT 10037708 73691 50233 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME ADINAZOLAM ADINAZOLAM 73692 50234 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 2056784 CHEMBL261123 73693 50235 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor SORAFENIB TOSYLATE 73694 50236 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME inhibitor 318164817 73695 50237 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME TAMATINIB R-406 73696 50238 TMEM97 27346 NA Fused aryl carbocycle derivative 2 73697 50239 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102728 CHEMBL506495 73699 50240 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 meloxicam MELOXICAM 24322170,9493314,24615047 73700 50241 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME MELAGATRAN MELAGATRAN 73702 50242 H2AX 3014 NA N-ACETYLCYSTEINE ACETYLCYSTEINE 15489221 73704 50243 POLA1 5422 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL1637 GEMCITABINE HYDROCHLORIDE 73705 50244 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651451 73706 50245 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CARBAMAZEPINE CARBAMAZEPINE 22931300 73707 50246 MAPT 4137 DRUGGABLE GENOME NIGULDIPINE NIGULDIPINE 73708 50247 KDM4A 9682 DRUGGABLE GENOME, ENZYME MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 73710 50248 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Alkyl sulfone derivative 1 73712 50249 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ENU 7695496 73713 50250 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL29741 IRAMPANEL 73715 50251 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE NSC-172614 CHEMBL1317506 73717 50252 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Sapanisertib SAPANISERTIB 25261369 73719 50253 GMNN 51053 DRUGGABLE GENOME ZOMEPIRAC SODIUM ZOMEPIRAC SODIUM 73720 50254 PPIG 9360 DRUGGABLE GENOME MELARSOPROL MELARSOPROL 73721 50255 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3545052 FIMEPINOSTAT 73722 50256 NCL 4691 NA ACT-GRO-777 25057429 73723 50257 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565640 KX2-391 73724 50258 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Niraparib NIRAPARIB 73725 50259 IDH2 3418 CLINICALLY ACTIONABLE, ENZYME Enasidenib ENASIDENIB 73726 50260 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME MORIN MORIN 73727 50261 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 178103585 ROMIDEPSIN 73728 50262 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 4 73729 50263 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ARSENIC TRIOXIDE 17121903 73730 50264 GRK2 156 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, G PROTEIN COUPLED RECEPTOR, ENZYME US9493490, D 73731 50265 RBP4 5950 DRUGGABLE GENOME ROSIGLITAZONE ROSIGLITAZONE 16034410 73734 50266 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE OLTIPRAZ OLTIPRAZ 20655236 73735 50267 DYRK2 8445 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 249565851 73736 50268 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652220 73737 50269 MAPT 4137 DRUGGABLE GENOME 3,4-DIMETHOXYDALBERGIONE 3,4-DIMETHOXYDALBERGIONE 73739 50270 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SIMVASTATIN SIMVASTATIN 22931300 73740 50271 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER 2',4'-DIHYDROXYCHALCONE 2',4'-DIHYDROXYCHALCONE 22112540 73742 50272 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651223 T091317 73744 50273 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL SANDARACOPIMARIC ACID SANDARACOPIMARIC ACID 21793559 73745 50274 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor VALPROIC ACID DEPAKOTE 73746 50275 CAMK2B 816 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CYC-116 CYC-116 73749 50276 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL1200542 DESOXYCORTICOSTERONE ACETATE 73750 50277 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CUDC-101 CUDC-101 73753 50278 TOB1 10140 NA STEROID HORMONE 15664454 73754 50279 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR GSK-269962A GSK-269962A 73755 50280 CDK17 5128 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR inhibitor CHEMBL3544942 RONICICLIB 73756 50281 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Irinotecan IRINOTECAN 23209031,25185971 73757 50282 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649942 73759 50283 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIAMTERENE TRIAMTERENE 73760 50284 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE tafenoquine TAFENOQUINE 73761 50285 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 2-AMINOANTHRACENE 2-AMINOANTHRACENE 73763 50286 MAPT 4137 DRUGGABLE GENOME NSC-95397 CHEMBL429095 73764 50287 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE SORAFENIB SORAFENIB 73765 50288 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR GSK461364 GSK-461364 25156567 73766 50289 KRT18 3875 DRUGGABLE GENOME RIBAVIRIN RIBAVIRIN 17713161 73767 50290 POLI 11201 DNA REPAIR AMARANTH AMARANTH 73770 50291 GRK3 157 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565822 BALANOL 73771 50292 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AG-808 CHEMBL68534 73773 50293 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL SECOBARBITAL SECOBARBITAL 73774 50294 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME TAK-715 TAK-715 73775 50295 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME CPT-11 IRINOTECAN HYDROCHLORIDE 12032863 73777 50296 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 22154664 73778 50297 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TAS-115 TAS-115 24140932 73779 50298 POLB 5423 DNA REPAIR, DRUGGABLE GENOME EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 73780 50299 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BITHIONOL BITHIONOL 73782 50300 POLK 51426 DNA REPAIR, ENZYME WEDELOLACTONE WEDELOLACTONE 73783 50301 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME inhibitor 340590229 RO-5045337 73784 50302 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE cyclophosphamide CYCLOPHOSPHAMIDE 27173875 73785 50303 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CGP-13501 CHEMBL1256746 73788 50304 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BUPIRIMATE BUPIRIMATE 73789 50305 CD55 1604 DRUGGABLE GENOME, CELL SURFACE ONYVAX-105 (105AD7) 73790 50306 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL70418 CLOBAZAM 73793 50307 GRK5 2869 G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME SOTRASTAURIN SOTRASTAURIN 73794 50308 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE ANTIMALARIALS 10639753 73797 50309 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME agonist 178100891 73798 50310 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor SB939 73799 50311 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME METHANTHELINE METHANTHELINE 73800 50312 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE erlotinib ERLOTINIB 18652519,18681783,14990633,16467544,16377102,14990632,18784101,17020982,21921847,16912157,19589612,18309947,16258541,16257339,21783417,19692684,17085664,18003960,19381876,15217965,22285168,22982650,16043828,22215752,26490356,23022519,11255078,17285735,18349398,19339720,18316547,22760226,12648464,21233402,18992959,21969500,22594511 73803 50313 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE HINOKININ HINOKININ 24112084 73804 50314 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR METHOXYCHLOR METHOXYCHLOR 73805 50315 LAMA2 3908 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 73806 50316 MAPT 4137 DRUGGABLE GENOME PITTSBURGH COMPOUND B PITTSBURGH COMPOUND B 73808 50317 NECTIN4 81607 DRUGGABLE GENOME enfortumab vedotin 73809 50318 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR allosteric modulator 328083529 MIRANSERTIB 73812 50319 SMARCA4 6597 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING RIBOCICLIB RIBOCICLIB 30718512 73814 50320 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Peptidomimetic analog 4 73815 50321 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CADMIUM DICHLORIDE CADMIUM DICHLORIDE 73816 50322 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL2110725 VINFLUNINE 73819 50323 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL2218893 BEDORADRINE SULFATE 73820 50324 BAZ2B 29994 NA NSC-50690 CHEMBL1388703 73821 50325 ARNT 405 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PROTEASOME INHIBITOR 10409767 73822 50326 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE SPIRONOLACTONE SPIRONOLACTONE 16837769 73825 50327 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200984 AMLODIPINE MALEATE 73827 50328 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 385612197 73830 50329 BRCA2 675 CLINICALLY ACTIONABLE QUARFLOXIN QUARFLOXIN 28211448 73831 50330 LAMA1 284217 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 73832 50331 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL3545065 VEROSUDIL 73834 50332 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME INTERLEUKINS 16252257 73835 50333 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565599 73838 50334 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL447955 SERLOPITANT 73839 50335 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135650219 VINBURNINE 73840 50336 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BDBM50177012 73841 50337 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200403 BUCLIZINE HYDROCHLORIDE 73843 50338 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 73848 50339 TUBB 203068 DRUGGABLE GENOME inhibitor 178103430 IXABEPILONE 73851 50340 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-MTC-424 73854 50341 HLA-G 3135 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME capecitabine CAPECITABINE 73856 50342 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR SCH-900776 SCH-900776 73858 50343 PTGS1 5742 ENZYME, DRUGGABLE GENOME IMRECOXIB IMRECOXIB 73859 50344 SMN2 6607 DRUGGABLE GENOME 2-(2'-METHOXYPHENYL)-1H-INDOLE 2-(2'-METHOXYPHENYL)-1H-INDOLE 73860 50345 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME LORATADINE LORATADINE 73863 50346 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR SANSALVAMIDE A-AMIDE CHEMBL192264 21764310 73865 50347 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE (-)-DEMECOLCINE DEMECOLCINE 73868 50348 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AG-1296 CHEMBL71191 73869 50349 TSHZ2 128553 TRANSCRIPTION FACTOR allopurinol ALLOPURINOL 29193002 73870 50350 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL646 TRIAZOLAM 73872 50351 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor BGJ398 INFIGRATINIB 73873 50352 MPHOSPH8 54737 NA AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 73874 50353 ALDH1A1 216 DRUGGABLE GENOME, ENZYME IRIGENOL IRIGENOL 73877 50354 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME 2-CHLORO-ADENOSINETRIPHOSPHATE CHEMBL1368696 73878 50355 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR KRM-189 CHEMBL449063 19081248 73879 50356 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 363894206 ALLITINIB 73881 50357 MYD88 4615 CLINICALLY ACTIONABLE eFT508 TOMIVOSERTIB 73882 50358 PTP4A3 11156 DRUGGABLE GENOME, PROTEIN PHOSPHATASE EMODIN EMODIN 22137788 73884 50359 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GNF-PF-2301 CHEMBL578061 73885 50360 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE 681640 CHEMBL379975 73887 50361 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200395 ORPHENADRINE CITRATE 73888 50362 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 73889 50363 MAOB 4129 DRUGGABLE GENOME, ENZYME SAFINAMIDE MESYLATE 73893 50364 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME VX-702 VX-702 73894 50365 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649958 73896 50366 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE IMATINIB IMATINIB 22114577,15201427,21953054,16143141,21690468,17372901,16624552,25239608,18421059,18955451,23775962,19671763,17699867,14645423,21642685,16954519,16434489 73897 50367 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME NERVIANO NERVIANO 20621725 73898 50368 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 404859155 73900 50369 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CHEMBL220492 TOPIRAMATE 73901 50370 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME AG-494 CHEMBL56731 73902 50371 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650453 KETANSERIN 73903 50372 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SIMOCYCLINONE D8 SIMOCYCLINONE D8 22867097 73905 50373 SLC33A1 9197 TRANSPORTER US8592431, 185 73906 50374 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER everolimus EVEROLIMUS 73907 50375 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CHEMOTHERAPY 24740294,23515910 73909 50376 HMOX1 3162 ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE ASPIRIN ASPIRIN 12927812 73913 50377 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-25 73914 50378 PI4KB 5298 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102681 WORTMANNIN 73915 50379 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER METOCHALCONE METOCHALCONE 22112540 73916 50380 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 73917 50381 FNTB 2342 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL298734 LONAFARNIB 73919 50382 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CICLOPIROX OLAMINE CICLOPIROX OLAMINE 73920 50383 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE NIRAPARIB NIRAPARIB 73921 50384 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FLOXURIDINE FLOXURIDINE 22931300 73922 50385 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME Dusigitumab DUSIGITUMAB 73923 50386 TUBA1A 7846 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 73925 50387 MTTP 4547 DRUGGABLE GENOME KD020 73926 50388 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME celecoxib CELECOXIB 22336956 73927 50389 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR allosteric modulator 178102544 73929 50390 PCSK1 5122 DRUGGABLE GENOME, PROTEASE, ENZYME CALCITONIN CALCITONIN 14566018 73930 50391 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE NEVIRAPINE NEVIRAPINE 17172311 73931 50392 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 405067336 73932 50393 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PRASTERONE PRASTERONE 73933 50394 ITGB5 3693 CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL429876 CILENGITIDE 73936 50395 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SB-202190 SB-202190 22951114 73938 50396 TLR7 51284 DRUGGABLE GENOME HYDROXYCHLOROQUINE HYDROXYCHLOROQUINE 73942 50397 FFAR2 2867 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 381118817 73944 50398 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME SLAZINIC ACID SLAZINIC ACID 73945 50399 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL3120215 OSI-027 73947 50400 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE BARASERTIB BARASERTIB 73948 50401 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-53 73949 50402 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROMAZINE PROMAZINE 73951 50403 GLS 2744 ENZYME IODOPHTHALEIN IODOPHTHALEIN 73952 50404 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME DASATINIB DASATINIB 73954 50405 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ADAPALENE ADAPALENE 73955 50406 TARDBP 23435 TUMOR SUPPRESSOR DNDI1417599 CHEMBL2094833 73956 50407 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C6 73957 50408 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651371 73958 50409 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME DOVITINIB DOVITINIB 73959 50410 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PMID27774824-Compound-Figure9Example2up 73960 50411 FAAH 2166 ENZYME, DRUGGABLE GENOME Enol carbamate derivative 1 73961 50412 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Isoflavone derivative 3 73962 50413 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME INDOPROFEN INDOPROFEN 73963 50414 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE PD-0166285 PD-0166285 73964 50415 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE oxaliplatin OXALIPLATIN 24980946 73966 50416 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565630 VOLASERTIB 73967 50417 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE SEMAGACESTAT SEMAGACESTAT 19443228 73969 50418 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME TAE-684 TAE-684 73971 50419 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE tegafur TEGAFUR 22486600 73972 50420 CHRNA5 1138 DRUGGABLE GENOME, ION CHANNEL cotinine COTININE 73973 50421 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL ISRADIPINE ISRADIPINE 73974 50422 PPM1A 5494 ENZYME, KINASE, TUMOR SUPPRESSOR VP-102 73975 50423 POLK 51426 DNA REPAIR, ENZYME FAGARONINE FAGARONINE 73976 50424 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER CEPHRADINE CEPHRADINE 22166395 73977 50425 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Nilotinib NILOTINIB 28514312 73979 50426 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ABT-700 TELISOTUZUMAB 73981 50427 SLC1A7 6512 TRANSPORTER, DRUGGABLE GENOME 178101410 73984 50428 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178103494 IBRUTINIB 73985 50429 SLC1A2 6506 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE inhibitor 178101292 DIHYDROKAINATE 73987 50430 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEFDINIR CEFDINIR 73988 50431 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE RetinoStat 73989 50432 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ESTRADIOL ESTRADIOL 73990 50433 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER trabectedin TRABECTEDIN 24024892 73992 50434 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR Estrogen ESTROGEN 73993 50435 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE tacrolimus TACROLIMUS 25587129 73995 50436 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME antagonist 336446956 73996 50437 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CH-5015765 CHEMBL1834096 21875802 73997 50438 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME WITHAFERIN A WITHAFERIN A 24079846 73998 50439 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE allosteric modulator 178102684 CLEMASTINE 74000 50440 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CISPLATIN CISPLATIN 27922681 74002 50441 SMN2 6607 DRUGGABLE GENOME CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 74005 50442 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL70418 CLOBAZAM 74006 50443 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL2096631 CLORAZEPATE DIPOTASSIUM 74007 50444 HTT 3064 DRUGGABLE GENOME NSC-228155 CHEMBL505670 74008 50445 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR APIGENIN APIGENIN 74009 50446 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CHIDAMIDE CHIDAMIDE 74010 50447 GMNN 51053 DRUGGABLE GENOME SJ000120081 CHEMBL606532 74011 50448 PDE5A 8654 ENZYME, DRUGGABLE GENOME PF-489791 74013 50449 BAZ2B 29994 NA GNF-PF-4786 CHEMBL602363 74015 50450 NUDT15 55270 ENZYME, CLINICALLY ACTIONABLE THIOGUANINE THIOGUANINE 26878724 74016 50451 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MITOMYCIN MITOMYCIN 22931300 74020 50452 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME zoledronate ZOLEDRONIC ACID 74021 50453 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MEBEVERINE HYDROCHLORIDE MEBEVERINE HYDROCHLORIDE 74022 50454 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C3 74023 50455 HKDC1 80201 DRUGGABLE GENOME, KINASE SENNOSIDE B SENNOSIDE B 74024 50456 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651331 XANOMELINE 74025 50457 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9181182, 40 74027 50458 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE BERKELEYAMIDE B BERKELEYAMIDE B 18330993 74028 50459 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR phenylephrine PHENYLEPHRINE 74029 50460 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR WORTMANNIN WORTMANNIN 74030 50461 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Azaindazole derivative 3 74031 50462 ALOX5 240 DRUGGABLE GENOME, ENZYME BALSALAZIDE BALSALAZIDE 74033 50463 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CATECHOL CATECHOL 74035 50464 PSMD1 5707 NA MLN-9708 IXAZOMIB CITRATE 74036 50465 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE RG-1530 RG-1530 74038 50466 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE abiraterone ABIRATERONE 25157341 74040 50467 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ARTEMISININ ARTEMISININ 74041 50468 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ANTI-CANCER AGENTS 15300809 74042 50469 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME NSC-107022 CHEMBL1601846 74044 50470 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme25-3 74045 50471 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-71033 CHEMBL116548 74046 50472 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME APRAMIDE A APRAMIDE A 10978206 74047 50473 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRICLOSAN TRICLOSAN 74050 50474 KDM4A 9682 DRUGGABLE GENOME, ENZYME BAS-8770949 CHEMBL476025 74052 50475 HSPA4 3308 NA GDNF 9618697 74053 50476 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 5,7-DIHYDROXY-4-METHYLCOUMARIN 5,7-DIHYDROXY-4-METHYLCOUMARIN 74054 50477 SRI 6717 NA VINCRISTINE VINCRISTINE 1975203 74055 50478 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE CID 3237815 CHEMBL410484 74056 50479 ATAD5 79915 NA TREQUINSIN TREQUINSIN 74058 50480 TRIM5 85363 ENZYME, B30_2 SPRY DOMAIN, DRUGGABLE GENOME paclitaxel PACLITAXEL 74059 50481 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE SAR245409 VOXTALISIB 24634413 74060 50482 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GNF-PF-4612 CHEMBL601550 74061 50483 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME Opioid anesthetics 30136624 74062 50484 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Indoline derivative 16 74064 50485 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PURPURIN PURPURIN 74066 50486 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE MITOXANTRONE MITOXANTRONE 12878861 74067 50487 HTT 3064 DRUGGABLE GENOME Ampicidin analog 2 74068 50488 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Insulin, porcine 74069 50489 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE cytarabine CYTARABINE 15564883 74070 50490 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE SODIUM 2-PHENOXYBENZOATE CHEMBL2172378 22889313 74072 50491 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR Regorafenib REGORAFENIB 21170960 74073 50492 RGS4 5999 DRUGGABLE GENOME RS-67506 CHEMBL83899 74077 50493 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CLOXYQUIN CLOXYQUIN 74078 50494 HMGCR 3156 ENZYME, DRUGGABLE GENOME PMID27537201-Compound-Figure17 74079 50495 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME blocker 135652735 74080 50496 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME agonist CHEMBL2108572 BALUGRASTIM 74081 50497 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ZOLPIDEM ZOLPIDEM 74085 50498 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR BISMUTH SUBSALICYLATE BISMUTH SUBSALICYLATE 74086 50499 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MK-2206 MK-2206 74087 50500 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME (-)-LEPTOCLINIDAMINE B CHEMBL2208197 23189988 74088 50501 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ACTH CORTICOTROPIN 8698834 74089 50502 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor TELATINIB TELATINIB 74091 50503 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME SJ000040549 CHEMBL589421 74094 50504 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE VORINOSTAT VORINOSTAT 74097 50505 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 384403651 74098 50506 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NSC-91340 CHEMBL1376091 74099 50507 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL30219 METHOHEXITAL SODIUM 74100 50508 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652306 74101 50509 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200947 METIPRANOLOL HYDROCHLORIDE 74102 50510 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE RX-3117 FLUOROCYCLOPENTENYLCYTOSINE 74103 50511 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME OLOMOUCINE OLOMOUCINE 74104 50512 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME MK-4827 NIRAPARIB 74108 50513 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PH-011685 CHEMBL126804 74109 50514 PDE4B 5142 DRUGGABLE GENOME, ENZYME CHF 6001 74110 50515 MAPT 4137 DRUGGABLE GENOME CHELERYTHRINE CHLORIDE CHELERYTHRINE CHLORIDE 74112 50516 GUCY1B1 2983 DRUGGABLE GENOME activator CHEMBL730 NITROGLYCERIN 74113 50517 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 404859078 74115 50518 GAS6 2621 DRUG RESISTANCE, DRUGGABLE GENOME, KINASE WARFARIN WARFARIN 16014032 74116 50519 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYAZOFAMID CYAZOFAMID 74117 50520 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 252166737 74118 50521 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200602 74120 50522 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL1489 AZACITIDINE 74121 50523 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR ANTISENSE OLIGONUCLEOTIDES 9108414 74122 50524 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME DOVITINIB DOVITINIB 74123 50525 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000200944 CHEMBL600173 74124 50526 PTGS2 5743 DRUGGABLE GENOME, ENZYME NABUMETONE NABUMETONE 74125 50527 PIP4K2A 5305 ENZYME, KINASE FLUPIRTINE MALEATE FLUPIRTINE MALEATE 74129 50528 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL1201558 INTERFERON ALFA-2B 74130 50529 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Carboxamide derivative 4 74131 50530 EPHB4 2050 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 249565627 TESEVATINIB 74132 50531 USP1 7398 DNA REPAIR, PROTEASE, ENZYME AMINOQUINURIDE AMINOQUINURIDE 74133 50532 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX RO-137410 CHEMBL275311 18951029 74134 50533 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GR-127935 GR-127935 74135 50534 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-19803 CHEMBL522983 74137 50535 KDM4A 9682 DRUGGABLE GENOME, ENZYME METHYLDOPA METHYLDOPA 74138 50536 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYC-116 CYC-116 74140 50537 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME QUAZEPAM QUAZEPAM 74141 50538 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME PHA-767491 CHEMBL225519 74144 50539 IL18 3606 DRUGGABLE GENOME DEXTRAN SULFATE SODIUM 16235535 74145 50540 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PROGESTERONE PROGESTERONE 8603579 74146 50541 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE sodium nitrite 74147 50542 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE DORAMAPIMOD DORAMAPIMOD 74149 50543 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650278 FLUSPIRILENE 74150 50544 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME AC-55649 CHEMBL425027 74151 50545 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ANDROSTENEDIONE ANDROSTENEDIONE 74152 50546 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 53801040 NICOTINE 74155 50547 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 328083526 CITARINOSTAT 74156 50548 NDUFB1 4707 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 74157 50549 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 223366152 74158 50550 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER E-FLUPENTIXOL E-FLUPENTIXOL 74160 50551 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CHEMBL2108667 YTTRIUM Y 90 IBRITUMOMAB TIUXETAN 74161 50552 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE XL647 TESEVATINIB 74163 50553 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE ETHAMSYLATE ETHAMSYLATE 74165 50554 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE XL647 TESEVATINIB 74167 50555 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Tamoxifen TAMOXIFEN 74168 50556 GSTT1 2952 DRUGGABLE GENOME clozapine CLOZAPINE 27168101 74169 50557 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME CYC-116 CYC-116 74171 50558 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antibody 381744918 VOLOCIXIMAB 74173 50559 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100739 74174 50560 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR NITROFURANTOIN NITROFURANTOIN 74176 50561 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE VINCRISTINE VINCRISTINE 74177 50562 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME DIACEREIN DIACEREIN 74178 50563 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3545207 EVENAMIDE 74181 50564 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR PEITC 14635187 74184 50565 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BITHIONOL BITHIONOL 74185 50566 VEGFB 7423 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR aflibercept AFLIBERCEPT 20124951 74189 50567 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR infliximab INFLIXIMAB 24253594 74190 50568 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR GELDANAMYCIN GELDANAMYCIN 25756299,25277067,24428777,24984936,18408713,18020309,21273068,21861487,23859777,25105924 74191 50569 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DINITRO CRESOL DINITRO CRESOL 74192 50570 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE CEFOXITIN CEFOXITIN 22166395 74194 50571 SIK1 150094 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 178102305 DASATINIB 74196 50572 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TAMATINIB R-406 74198 50573 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FELBAMATE FELBAMATE 22931300 74199 50574 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE adalimumab ADALIMUMAB 24048425,27044681 74200 50575 ACAT1 38 ENZYME SULFASALAZINE SULFASALAZINE 74201 50576 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-2243 CHEMBL600908 74202 50577 PTGS1 5742 ENZYME, DRUGGABLE GENOME CURCUMIN CURCUMIN 24920381 74203 50578 HTT 3064 DRUGGABLE GENOME NSC-102742 CHEMBL1519374 74205 50579 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor GELFITINIB 74207 50580 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist CHEMBL1023 BEXAROTENE 74208 50581 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME KERACYANIN KERACYANIN 17360708 74209 50582 HMGCR 3156 ENZYME, DRUGGABLE GENOME Quinoline derivative 1 74210 50583 CA12 771 DRUGGABLE GENOME inhibitor CHEMBL17 DICHLORPHENAMIDE 74211 50584 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME HDM2 INHIBITOR MK-8242 28240971 74214 50585 MAPT 4137 DRUGGABLE GENOME GW441756X GW441756X 74215 50586 MAPT 4137 DRUGGABLE GENOME SAPPANONE A DIMETHYL ETHER SAPPANONE A DIMETHYL ETHER 74216 50587 PSMD4 5710 NA CARFILZOMIB CARFILZOMIB 24524217 74217 50588 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 310264739 LIFIRAFENIB 74218 50589 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Deguelin DEGUELIN 24978597,20811676 74220 50590 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CYC-116 CYC-116 74221 50591 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor AV951 74222 50592 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE BETA-NAPHTHOFLAVONE BETA-NAPHTHOFLAVONE 74223 50593 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME inhibitor 387065575 74228 50594 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2010077680 803 74229 50595 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE SORAFENIB SORAFENIB 74230 50596 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME lovastatin LOVASTATIN 74231 50597 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME KO-947 74232 50598 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE FMDC TEZACITABINE 10961690 74233 50599 TTN 7273 DRUGGABLE GENOME, TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, ENZYME PROTEASE INHIBITORS 9648223 74234 50600 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME DNDI1417467 CHEMBL1997335 74235 50601 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL995 LOSARTAN POTASSIUM 74236 50602 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL2110725 VINFLUNINE 74237 50603 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antagonist CHEMBL1743024 GANITUMAB 74238 50604 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME TD-1473 74239 50605 GPR12 2835 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NEOCYCLOCITRINOL C NEOCYCLOCITRINOL C 18656987 74240 50606 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL2110732 DACOMITINIB 74243 50607 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Sym013 74244 50608 ATAD5 79915 NA NSC-102045 CHEMBL483633 74245 50609 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE IMATINIB IMATINIB 74247 50610 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE 178101360 74248 50611 CAST 831 PROTEASE INHIBITOR THROMBIN THROMBIN 8358337 74249 50612 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PANOBINOSTAT PANOBINOSTAT 24694055 74251 50613 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME 2-METHOXY-1,4-NAPHTHOQUINONE 2-METHOXY-1,4-NAPHTHOQUINONE 74252 50614 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GSK3052230 FP-1039 23536011 74255 50615 ALDH1A1 216 DRUGGABLE GENOME, ENZYME N-(PHENETHYLCARBAMOTHIOYL)BENZAMIDE CHEMBL1448292 74256 50616 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102541 74257 50617 MAGEA3 4102 ENZYME, DRUGGABLE GENOME DNA VACCINE 15750833 74259 50618 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MT110 SOLITOMAB 74261 50619 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135652728 74266 50620 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 315661186 BRIMAPITIDE 74267 50621 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE RG-1530 RG-1530 74269 50622 MAPT 4137 DRUGGABLE GENOME INDIRUBIN SULFATE SU-9516 74273 50623 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR PROPAZINE PROPAZINE 74274 50624 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NOR-BINALTORPHIMINE DIHYDROCHLORIDE CHEMBL2374078 74276 50625 ADAM10 102 ENZYME, CELL SURFACE, TRANSPORTER, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE MARIMASTAT MARIMASTAT 26192023 74277 50626 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ALX-5407 CHEMBL180966 74278 50627 VKORC1 79001 DRUGGABLE GENOME, ENZYME PHENPROCOUMON PHENPROCOUMON 74280 50628 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ZINC 03369470 CHEMBL599013 74281 50629 MAP3K1 4214 CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 27670765 74282 50630 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL2109475 PG-102 74283 50631 SAE1 10055 ENZYME, DRUGGABLE GENOME ASTERRIC ACID ASTERRIC ACID 74284 50632 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME 5-FU FLUOROURACIL 15067352 74286 50633 NDUFB3 4709 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 74287 50634 SMN1 6606 DRUGGABLE GENOME CID 887167 CHEMBL260342 74289 50635 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE GSK1070916A 74290 50636 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR imidapril IMIDAPRIL 12522467 74291 50637 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SE-(METHYL)SELENOCYSTEINE HCL CHEMBL1256174 74294 50638 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CLOFLUCARBAN CLOFLUCARBAN 74295 50639 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE Abiraterone acetate 74297 50640 CPT1A 1374 DRUGGABLE GENOME, ENZYME PROPIONYL-L-CARNITINE 74299 50641 NOS1 4842 DRUGGABLE GENOME, ENZYME PRAVASTATIN PRAVASTATIN 15126084 74300 50642 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1416969 CHEMBL1453126 74303 50643 EPOR 2057 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME Epoetin alfa 74304 50644 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME CORTICOSTEROIDS 2144977 74306 50645 CA12 771 DRUGGABLE GENOME topiramate TOPIRAMATE 21278619 74308 50646 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX FIDUXOSIN HYDROCHLORIDE FIDUXOSIN HYDROCHLORIDE 74309 50647 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-21 74310 50648 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE TAMATINIB R-406 74311 50649 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE LUZINDOLE LUZINDOLE 74313 50650 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CENISERTIB CENISERTIB 74314 50651 XPA 7507 CLINICALLY ACTIONABLE, DNA REPAIR IMMUNOSUPPRESSIVE 11313422 74315 50652 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME SAHA VORINOSTAT 16951239 74319 50653 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GW282974X GW282974X 74320 50654 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ERGOCORNINE ERGOCORNINE 74321 50655 ALOX15B 247 DRUGGABLE GENOME, ENZYME LUTEOLIN LUTEOLIN 74322 50656 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-21 74323 50657 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FIIN-01 20338520 74324 50658 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CHLORPROMAZINE CHLORPROMAZINE 22931300 74325 50659 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIBROMOACETIC ACID DIBROMOACETIC ACID 74326 50660 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774822-Compound-Figure10Example1 74328 50661 SERPINA6 866 DRUGGABLE GENOME, PROTEASE INHIBITOR ALCLOMETASONE ALCLOMETASONE 74330 50662 NR4A3 8013 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, TRANSPORTER, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE ANTISENSE OLIGONUCLEOTIDES 14962944 74332 50663 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME TAMATINIB R-406 74333 50664 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651113 74336 50665 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME ALPRAZOLAM ALPRAZOLAM 74337 50666 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL DEXTROMETHORPHAN DEXTROMETHORPHAN 74338 50667 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 2 74339 50668 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Risperidone RISPERIDONE 74340 50669 NRP1 8829 DRUGGABLE GENOME Pegaptanib PEGAPTANIB SODIUM 74343 50670 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 404859045 74344 50671 RGS2 5997 NA antipsychotics 18347610 74345 50672 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR PD0332991 PALBOCICLIB 25156567 74346 50673 MAPT 4137 DRUGGABLE GENOME CARNOSIC ACID CARNOSIC ACID 74347 50674 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER imatinib IMATINIB 23127916 74348 50675 GMNN 51053 DRUGGABLE GENOME SJ000012773 CHEMBL589715 74349 50676 NOS1 4842 DRUGGABLE GENOME, ENZYME ATORVASTATIN ATORVASTATIN 15639473 74354 50677 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-44 74355 50678 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL107 COLCHICINE 74356 50679 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CURCUMIN CURCUMIN 18076140 74357 50680 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PANTOPRAZOLE PANTOPRAZOLE 74358 50681 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 385612248 74360 50682 SPP1 6696 DRUGGABLE GENOME GENTAMICIN GENTAMICIN 11274264 74361 50683 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL971 PENTOBARBITAL SODIUM 74362 50684 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME FENOLDOPAM BROMIDE FENOLDOPAM BROMIDE 74363 50685 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PF-05212384 GEDATOLISIB 24042735,23012248,12068308,17314276,21325073 74364 50686 PTGS2 5743 DRUGGABLE GENOME, ENZYME CARPROFEN CARPROFEN 74365 50687 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME fasudil FASUDIL 22541434 74366 50688 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE DABRAFENIB DABRAFENIB 23171796 74367 50689 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME L-3,4-DIHYDROXYPHENYLALANINE METHYL ESTER HCL CHEMBL1255756 74368 50690 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE glibenclamide GLYBURIDE 21147013,20701405,15126005,8562390 74370 50691 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 74371 50692 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Dexamethasone DEXAMETHASONE 28151717 74374 50693 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE ESTRADIOL BENZOATE ESTRADIOL BENZOATE 74375 50694 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 340590231 74376 50695 GMNN 51053 DRUGGABLE GENOME CHLORACYZINE CHLORACYZINE 74377 50696 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR rituximab RITUXIMAB 26384320 74379 50697 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIGOXIN DIGOXIN 22931300 74380 50698 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AG-34 CHEMBL80155 74382 50699 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 9 74383 50700 PTGS2 5743 DRUGGABLE GENOME, ENZYME DICLOFENAC DICLOFENAC 74385 50701 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL2103741 LEVOTHYROXINE SODIUM 74386 50702 TBC1D1 23216 NA olanzapine OLANZAPINE 23364847 74387 50703 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME PRAZEPAM PRAZEPAM 74390 50704 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE KU-0060648 CHEMBL1086377 23761041 74393 50705 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor GSK2636771 GSK-2636771 74395 50706 HMOX1 3162 ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE VITAMIN D 15225803 74397 50707 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUORODIFEN FLUORODIFEN 74399 50708 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL180101 ESREBOXETINE 74400 50709 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE XL880 FORETINIB 74401 50710 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-4 74402 50711 PSMA3 5684 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL371405 MARIZOMIB 74403 50712 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BYL719 ALPELISIB 27602501,27126994,26627007,24608574,26013318,27604488,28119489 74404 50713 DGAT1 8694 ENZYME, DRUGGABLE GENOME Pyridine-carboximide derivative 2 74406 50714 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE GEFITINIB GEFITINIB 74407 50715 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178101056 74408 50716 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE AST-487 AST-487 74410 50717 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SP-600125 SP-600125 74412 50718 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE THYROTROPIN THYROTROPIN 3125035,3726540 74414 50719 SLC6A11 6538 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GSK683699 74415 50720 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE inhibitor CHEMBL1908360 EVEROLIMUS 74416 50721 PRKCH 5583 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor SOPHORETIN QUERCETIN 74418 50722 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CYTOPROTECTIVE AGENT 18254247 74419 50723 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE MG98 74422 50724 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR VISMODEGIB VISMODEGIB 19726788,25759020,22550175,22679179 74423 50725 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME PMID28270010-Compound-Figure24-a 74425 50726 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 178103584 74426 50727 COL4A6 1288 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 74429 50728 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME SJ000044511 CHEMBL592124 74431 50729 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32p 74432 50730 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 74435 50731 POLI 11201 DNA REPAIR PICEATANNOL PICEATANNOL 74437 50732 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL3545402 XL-820 74438 50733 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 178102431 74440 50734 CD38 952 CELL SURFACE, DRUGGABLE GENOME CD38 and BCMA CAR-T Cells 74441 50735 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 7RH 26855149 74442 50736 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 5-FU FLUOROURACIL 8888499 74445 50737 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CORYNANTHEINE CORYNANTHEINE 74446 50738 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AG-555 CHEMBL53898 74447 50739 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Carboxamide derivative 11 74448 50740 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 404859074 74449 50741 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PMID25416646-Compound-Figure5-H 74450 50742 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE CLOFOCTOL CLOFOCTOL 74451 50743 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL2107731 AXOMADOL 74452 50744 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE SCRIPTAID SCRIPTAID 19966789 74455 50745 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649965 74456 50746 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR FULVESTRANT FULVESTRANT 19845386 74458 50747 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 14767525 74459 50748 RAB9A 9367 ENZYME, DRUGGABLE GENOME N-(3,4-DIMETHOXYPHENYL)PICOLINAMIDE CHEMBL572346 74460 50749 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PF-03893787 PF-03893787 21920751 74461 50750 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OCTADECYLAMINE OCTADECYLAMINE 74462 50751 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MINOCYCLINE MINOCYCLINE 22931300 74463 50752 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL ERUCIN ERUCIN 26263397 74465 50753 PDE5A 8654 ENZYME, DRUGGABLE GENOME DIPYRIDAMOLE DIPYRIDAMOLE 74466 50754 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DICHLOFENTHION DICHLOFENTHION 74467 50755 GATA2 2624 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX bortezomib BORTEZOMIB 22541434 74468 50756 FAAH 2166 ENZYME, DRUGGABLE GENOME PMID29053063-Compound-15 74471 50757 SLC15A3 51296 TRANSPORTER, DRUGGABLE GENOME 178101341 74474 50758 ASS1 445 ENZYME, DRUG RESISTANCE sodium benzoate / sodium phenylacetate 74476 50759 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103953 CHEMBL56331 74479 50760 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 LEUPROLIDE LEUPROLIDE 22931300 74481 50761 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME risperidone RISPERIDONE 23859574,20031235 74486 50762 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Anti-BCMA CART Cells 74487 50763 NOS1 4842 DRUGGABLE GENOME, ENZYME ISOTHIOUREA 74489 50764 RARRES1 5918 NA TRETINOIN TRETINOIN 74491 50765 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DIHYDROCAPSAICIN DIHYDROCAPSAICIN 74492 50766 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR AG-538 CHEMBL56393 74493 50767 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor DACOMITINIB DACOMITINIB 74494 50768 GCKR 2646 ENZYME ethanol ALCOHOL 32451486 74495 50769 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME promethazine PROMETHAZINE 17986163 74496 50770 SLC2A3 6515 DRUGGABLE GENOME, TRANSPORTER GLUFOSFAMIDE GLUFOSFAMIDE 74497 50771 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR cisplatin CISPLATIN 19786980,22188361,18347182,21902499,25069034,21057378,29662106,19362955,23962907,19203783,27498158,21262916,22026922,22329723 74498 50772 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DEPHOSTATIN DEPHOSTATIN 74501 50773 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor NINTEDANIB NINTEDANIB 74502 50774 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GW642444 VILANTEROL 74505 50775 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE VATALANIB VATALANIB 74507 50776 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Docetaxel DOCETAXEL 26202948 74508 50777 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME WX-554 WX-554 74509 50778 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SU-4312 CHEMBL328710 74511 50779 CTSV 1515 ENZYME, DRUGGABLE GENOME, PROTEASE PMID27998201-Compound-12 74512 50780 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME ONONIN ONONIN 74514 50781 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE antithrombotic agents 74515 50782 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR TACEDINALINE TACEDINALINE 18692397 74517 50783 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE ILORASERTIB ILORASERTIB 74518 50784 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DIACYLGLYCEROL KINASE INHIBITOR II DIACYLGLYCEROL KINASE INHIBITOR II 74519 50785 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE 7-HYDROXYFLAVONE 7-HYDROXYFLAVONE 74521 50786 UGT1A10 54575 DRUGGABLE GENOME, ENZYME MYCOPHENOLIC ACID 15039300,10688250 74523 50787 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 381744956 74524 50788 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HYDROXYFLUTAMIDE HYDROXYFLUTAMIDE 18571420,26295173 74525 50789 CXCL8 3576 DRUGGABLE GENOME CYTOKINES 11285034 74528 50790 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Glitazone GLITAZONE 74529 50791 RCE1 9986 ENZYME, PROTEASE, DRUGGABLE GENOME ACRIDIN-1-YLAMINE CHEMBL146525 74530 50792 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BIIB-021 BIIB021 74532 50793 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor BMS-536924 CHEMBL401930 74533 50794 UGT2B7 7364 DRUGGABLE GENOME carbamazepine CARBAMAZEPINE 21738081 74535 50795 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME ABT-639 ABT-639 74538 50796 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME NILUTAMIDE NILUTAMIDE 9186345 74539 50797 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651242 TELMISARTAN 74542 50798 IL4R 3566 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Dupilumab DUPILUMAB 74543 50799 METAP2 10988 ENZYME, DRUGGABLE GENOME, KINASE, PROTEASE M8891 74544 50800 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME XL228 XL-228 74546 50801 PRKAA2 5563 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSPORTER, ENZYME SAPONARIN SAPONARIN 26471090 74548 50802 S100A12 6283 DRUGGABLE GENOME, KINASE MK-1602 UBROGEPANT 74549 50803 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE SIMVASTATIN SIMVASTATIN 74551 50804 ITGB8 3696 DRUGGABLE GENOME, CELL SURFACE US10035778, Example 1 74553 50805 PSMB4 5692 DRUGGABLE GENOME, PROTEASE inhibitor CARFILZOMIB CARFILZOMIB 74556 50806 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Cyclic sulfonamide derivative 1 74557 50807 SLC29A2 3177 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE 6-MERCAPTOPURINE MERCAPTOPURINE 17088032 74558 50808 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL235191 TACEDINALINE 74560 50809 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME GENTAMICIN GENTAMICIN 8861105 74561 50810 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE NEW AGENTS 9026436 74562 50811 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652219 74563 50812 NR4A1 3164 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX CYCLOSPORIN A 7831306 74564 50813 FAAH 2166 ENZYME, DRUGGABLE GENOME 6-OHDA 12716433 74565 50814 PPIA 5478 DRUGGABLE GENOME, ENZYME modulator CHEMBL160 CYCLOSPORINE 74566 50815 KIF11 3832 DRUGGABLE GENOME NSC-12352 CHEMBL392369 19167222 74567 50816 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Tri-substituted urea derivative 1 74568 50817 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125000 CHEMBL579742 74569 50818 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL1230607 PHA-793887 74570 50819 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 nateglinide NATEGLINIDE 74571 50820 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor XL228 XL-228 74572 50821 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4097 CHEMBL597246 74573 50822 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 178103352 IDELALISIB 74575 50823 MAP2K6 5608 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE, TUMOR SUPPRESSOR VX-745 NEFLAMAPIMOD 74576 50824 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Propiomazine PROPIOMAZINE 74577 50825 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RETINAL RETINAL 74578 50826 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ALUM 12672065 74579 50827 POLK 51426 DNA REPAIR, ENZYME CEFSULODIN SODIUM CEFSULODIN SODIUM 74581 50828 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-K2 74583 50829 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MICONAZOLE NITRATE MICONAZOLE NITRATE 74585 50830 ARNT 405 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR EPICATECHIN GALLATE EPICATECHIN GALLATE 15620252 74586 50831 RACGAP1 29127 NA 3,3'-DIMETHOXYBENZIDINE CHEMBL398363 74588 50832 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL2165191 AZD-6482 74589 50833 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR antagonist CHEMBL3545357 JTE-151 74590 50834 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE PMID26882240-Compound-4 74591 50835 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565927 74594 50836 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Glimepiride GLIMEPIRIDE 74597 50837 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2012819831110 74598 50838 USP1 7398 DNA REPAIR, PROTEASE, ENZYME GNF-PF-2272 CHEMBL601757 74601 50839 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IODOPHENPROPIT IODOPHENPROPIT 74602 50840 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL744 RILUZOLE 74603 50841 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-16 74605 50842 ATAD5 79915 NA NU-6027 CHEMBL303958 74606 50843 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ADJUVANT 15048719 74607 50844 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 223366139 74608 50845 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL blocker 135652732 74610 50846 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Nebivolol NEBIVOLOL 74611 50847 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME SYR-472 TRELAGLIPTIN 74612 50848 ROR1 4919 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CELL SURFACE ROR1 CAR-specific Autologous T-Lymphocytes 74613 50849 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ONONETIN ONONETIN 74615 50850 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME poziotinib POZIOTINIB 21306821 74616 50851 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME RANITIDINE RANITIDINE 74618 50852 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER sunitinib SUNITINIB 25778465,27564227,24874929,26244574,24013576 74619 50853 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2105712 AFATINIB DIMALEATE 74620 50854 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Yttrium (90Y) clivatuzumab tetraxetan 74624 50855 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME acetaminophen ACETAMINOPHEN 26398624 74626 50856 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME inhibitor CHEMBL1969664 AZD-1080 74627 50857 GBA 2629 DRUGGABLE GENOME, ENZYME 2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE 2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE 74628 50858 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR YEZOQUINOLIDE YEZOQUINOLIDE 21142112 74629 50859 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME IRL-2500 CHEMBL72410 74631 50860 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME ARSENIC TRIOXIDE 74632 50861 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 252166526 ESUBERAPROST 74634 50862 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME VX-970 BERZOSERTIB 28363999 74636 50863 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545236 BPI-9016 74637 50864 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL BROMAZEPAM BROMAZEPAM 74639 50865 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR PROGESTIN PROGESTERONE 74640 50866 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME clozapine CLOZAPINE 26876050 74641 50867 PDE1A 5136 ENZYME, DRUGGABLE GENOME activator 135652052 74644 50868 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME EDELFOSINE EDELFOSINE 16540473 74645 50869 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE VANDETANIB VANDETANIB 74648 50870 ACVR1B 91 SERINE THREONINE KINASE, CELL SURFACE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE US9682983, 33 74650 50871 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-209931 CHEMBL472656 74651 50872 MUC2 4583 DRUGGABLE GENOME DEXTRAN SULFATE SODIUM 16831596 74652 50873 PTGS1 5742 ENZYME, DRUGGABLE GENOME ACETAMINOPHEN ACETAMINOPHEN 74653 50874 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE SCH-900271 SCH-900271 74656 50875 IL18 3606 DRUGGABLE GENOME interferons 19455410 74657 50876 GMNN 51053 DRUGGABLE GENOME COLCHICINE COLCHICINE 74658 50877 SMN2 6607 DRUGGABLE GENOME TCMDC-124585 CHEMBL587856 74660 50878 MAPT 4137 DRUGGABLE GENOME NSC-377852 CHEMBL1466186 74663 50879 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE VANDETANIB VANDETANIB 74664 50880 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE HERBIMYCIN A 11245436 74665 50881 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE ABT-348 ILORASERTIB 74667 50882 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR TRIIODOTHYRONINE LIOTHYRONINE SODIUM 8288635 74668 50883 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-arylmethyl-N-phenyl cyclic urea derivative 1 74672 50884 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME IRINOTECAN HYDROCHLORIDE IRINOTECAN HYDROCHLORIDE 74673 50885 TFPI2 7980 PROTEASE INHIBITOR, DRUGGABLE GENOME PROTEASE INHIBITORS 3276312 74675 50886 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING ATOMOXETINE HYDROCHLORIDE ATOMOXETINE HYDROCHLORIDE 74677 50887 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR DAPH DAPH 74679 50888 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE lansoprazole LANSOPRAZOLE 18695978 74680 50889 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR ALVOCIDIB ALVOCIDIB 74681 50890 MAPT 4137 DRUGGABLE GENOME SANGUINARIUM SANGUINARIUM 74683 50891 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL ALPRAZOLAM ALPRAZOLAM 74684 50892 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135650189 74685 50893 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 381744939 74686 50894 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE SCH-23390 SCH-23390 74687 50895 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE LINIFANIB LINIFANIB 74688 50896 FAAH 2166 ENZYME, DRUGGABLE GENOME Isoxazoline derivative 1 74689 50897 XRCC1 7515 CLINICALLY ACTIONABLE VINORELBINE VINORELBINE 19157633 74690 50898 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME BELINOSTAT BELINOSTAT 25937017 74691 50899 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL452 CLONAZEPAM 74692 50900 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE FIBRIN SEALANT 16925334 74693 50901 RABEP1 9135 CLINICALLY ACTIONABLE, GROWTH FACTOR aripiprazole ARIPIPRAZOLE 28694205 74694 50902 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CISPLATIN CISPLATIN 8205547 74697 50903 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-14 74699 50904 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME BENZENE-1,2-DIAMINE CHEMBL70582 74700 50905 CD9 928 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE HERBIMYCIN A 7592610 74701 50906 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME AST-487 AST-487 74702 50907 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME ENTRECTINIB ENTRECTINIB 74703 50908 CBX1 10951 NA LY-294002 LY-294002 74705 50909 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME AZACYTIDINE AZACITIDINE 12543079 74706 50910 NOS2 4843 DRUGGABLE GENOME, ENZYME CONJUGATED ESTROGENS 10997912 74708 50911 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE POLYPHENOL 12238566 74709 50912 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR antagonist BIRINAPANT BIRINAPANT 74711 50913 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-75270 CHEMBL1333982 22524450 74712 50914 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME PREGABALIN PREGABALIN 74713 50915 MAPT 4137 DRUGGABLE GENOME PROTOAPIGENONE PROTOAPIGENONE 74714 50916 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE ALBUTROPIN 74715 50917 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Hydrocortisone HYDROCORTISONE 74716 50918 IFI27 3429 NUCLEAR HORMONE RECEPTOR VITAMIN D 15086558 74720 50919 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 4-Carboxamido-isoindolinone derivative 4 74721 50920 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR timolol TIMOLOL 16315032 74722 50921 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR AILANTHINONE AILANTHINONE 19199792 74723 50922 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BISACODYL BISACODYL 74727 50923 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME N/A 74728 50924 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR SCOPOLETIN SCOPOLETIN 74729 50925 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE RIBOFLAVIN RIBOFLAVIN 74730 50926 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME FASUDIL FASUDIL 74731 50927 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE RG-1530 RG-1530 74733 50928 POLI 11201 DNA REPAIR QUERCETIN QUERCETIN 74734 50929 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor GDC-0941 PICTILISIB 74736 50930 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE RETINOID 17024972 74737 50931 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR QUINESTROL QUINESTROL 74738 50932 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE IDELALISIB IDELALISIB 26466009 74739 50933 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BYL719 ALPELISIB 74740 50934 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-H1 74742 50935 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR AMPHETAMINE AMPHETAMINE 74743 50936 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4798 CHEMBL584635 74744 50937 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE NSC-663284 CHEMBL337173 74745 50938 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor PELITINIB PELITINIB 74748 50939 PDE4A 5141 DRUGGABLE GENOME, ENZYME RPL-554 74750 50940 SMN2 6607 DRUGGABLE GENOME 5,7-DIMETHOXYISOFLAVONE 5,7-DIMETHOXYISOFLAVONE 74752 50941 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL2107832 PIMASERTIB 74753 50942 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME COBALT 8131214 74754 50943 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE inhibitor 385612210 74755 50944 ULK3 25989 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 74756 50945 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102322 TANDUTINIB 74757 50946 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BI2536 26573800 74758 50947 KDM4A 9682 DRUGGABLE GENOME, ENZYME AG-538 CHEMBL56393 74761 50948 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 tacrolimus TACROLIMUS 28316087 74763 50949 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PECTOLINARIGENIN PECTOLINARIGENIN 74764 50950 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME OMEPRAZOLE OMEPRAZOLE 22931300 74765 50951 CISH 1154 NA EPO EPOETIN ALFA 12396724 74767 50952 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor XL820 74771 50953 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL501867 VINCRISTINE SULFATE 74772 50954 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX FLUSPIRILENE FLUSPIRILENE 74774 50955 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 249565826 74777 50956 NF1 4763 CLINICALLY ACTIONABLE, DRUG RESISTANCE SELUMETINIB SELUMETINIB 28029918,31151904 74778 50957 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650410 IPRATROPIUM 74779 50958 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor 178103416 DORZOLAMIDE 74780 50959 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME PMID28594589-Compound-TABLE3C2 74781 50960 MLLT3 4300 CLINICALLY ACTIONABLE cisplatin CISPLATIN 27150640 74782 50961 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER 3,4-DIHYDROXYXANTHONE 3,4-DIHYDROXYXANTHONE 74783 50962 PDE3A 5139 ENZYME, DRUGGABLE GENOME Enoximone ENOXIMONE 74785 50963 ALOX15 246 ENZYME, DRUGGABLE GENOME GERALDOL GERALDOL 74787 50964 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME 6-O-BENZYLGUANINE 6-O-BENZYLGUANINE 22932317,18973327 74788 50965 TUBB2A 7280 DRUGGABLE GENOME PACLITAXEL PACLITAXEL 23631389,25369367,25768699,24457094,22595423,23313639,17887662,23387901,19758808,23725535,24953821 74789 50966 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER MICONAZOLE MICONAZOLE 15969931 74790 50967 NOX4 50507 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 363894225 74791 50968 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 328083480 74795 50969 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR US10040779, Example 4 74796 50970 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TENOVIN-1 CHEMBL1436543 74801 50971 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PYRIDOSTIGMINE PYRIDOSTIGMINE 22931300 74803 50972 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2109295 ASCRINVACUMAB 74804 50973 CBX1 10951 NA SQ-22536 CHEMBL64239 74806 50974 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor AZD4547 74807 50975 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NELFINAVIR MESYLATE NELFINAVIR MESYLATE 74809 50976 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME MK-6302 74810 50977 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565874 74812 50978 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL PRIMIDONE PRIMIDONE 74813 50979 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME DOVITINIB DOVITINIB 74814 50980 MAOB 4129 DRUGGABLE GENOME, ENZYME Secondary and tertiary (hetero)arylamide derivative 1 74815 50981 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE CURCUMIN PYRAZOLE CURCUMIN PYRAZOLE 19128977 74817 50982 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor DINACICLIB DINACICLIB 74819 50983 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PF-562271 PF-00562271 74826 50984 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor GSK2636771 GSK-2636771 74827 50985 ATAD5 79915 NA ACRIDIN-1-YLAMINE CHEMBL146525 74829 50986 GMNN 51053 DRUGGABLE GENOME TCMDC-123884 CHEMBL580955 74831 50987 FAAH 2166 ENZYME, DRUGGABLE GENOME Piperazine carbamic compound 1 74832 50988 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CYC-116 CYC-116 74833 50989 MAPT 4137 DRUGGABLE GENOME DICHLOROPHEN DICHLOROPHEN 74836 50990 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME GNF-PF-3542 CHEMBL598477 74838 50991 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME SB-202190 SB-202190 74839 50992 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR DEFIBROTIDE DEFIBROTIDE 11441984 74840 50993 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ORG-25935 ORG-25935 74841 50994 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX PMID27336223-Compound-14 74842 50995 BCHE 590 DRUGGABLE GENOME, ENZYME PMID29757691-Compound-8c 74843 50996 PTGS1 5742 ENZYME, DRUGGABLE GENOME Bromfenac BROMFENAC 74844 50997 TGFBR2 7048 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME inhibitor 249565800 74845 50998 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 363894208 ILORASERTIB 74846 50999 FGA 2243 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, FIBRINOGEN ALTEPLASE ALTEPLASE 74848 51000 SMAD2 4087 KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX AMIFOSTINE AMIFOSTINE 12410567 74849 51001 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CYTOKINES 14611111 74850 51002 TSG101 7251 TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME NSC-106547 CHEMBL223575 74851 51003 FAAH2 158584 DRUGGABLE GENOME, ENZYME inhibitor 178101892 74852 51004 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME nefazodone NEFAZODONE 74855 51005 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL1234354 PF-04691502 74856 51006 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME BUTACLAMOL BUTACLAMOL 74858 51007 KDM5B 10765 ENZYME inhibitor 381118851 74859 51008 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 WHILE OLIVETOL WHILE OLIVETOL 74861 51009 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-48 74862 51010 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Ondansetron ONDANSETRON 74863 51011 CBX1 10951 NA N6-PHENYLADENOSINE N6-PHENYLADENOSINE 74864 51012 TBC1D1 23216 NA clozapine CLOZAPINE 23364847 74865 51013 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor GDC-0941 PICTILISIB 74867 51014 MAPT 4137 DRUGGABLE GENOME TCMDC-124032 CHEMBL536375 74871 51015 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Dexamethasone DEXAMETHASONE 28151717 74872 51016 TXNRD1 7296 DRUGGABLE GENOME Bis-sulfonamide derivative 2 74873 51017 ADD1 118 KINASE diuretics 17189961,11926892 74874 51018 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Palbociclib PALBOCICLIB 74876 51019 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-123927 CHEMBL531268 74877 51020 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ISOLIQUIRITIGENIN ISOLIQUIRITIGENIN 74878 51021 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME activator 135652731 74880 51022 SLC39A6 25800 TRANSPORTER, ENZYME, DRUGGABLE GENOME, CELL SURFACE SGN LIV1A 74882 51023 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME DNDI1417523 CHEMBL598663 74884 51024 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER inhibitor 178101472 74885 51025 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE GW441756X GW441756X 74887 51026 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BCT303 74888 51027 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME GNF-PF-3037 CHEMBL600336 74889 51028 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR ENALAPRIL ENALAPRIL 16772709 74890 51029 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CHRYSOPHANOL CHRYSOPHANOL 74891 51030 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE Trametinib TRAMETINIB 26343583 74892 51031 LRP1B 53353 CLINICALLY ACTIONABLE, DRUG RESISTANCE DOXORUBICIN DOXORUBICIN 22896685 74893 51032 IL15RA 3601 DRUGGABLE GENOME, CELL SURFACE ALT-803 ALT-803 74895 51033 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Romiplostim ROMIPLOSTIM 74896 51034 IMPDH1 3614 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1643 RIBAVIRIN 74898 51035 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135652699 74902 51036 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR inhibitor 252827436 74903 51037 ATXN2 6311 NA FLUOXETINE FLUOXETINE 74905 51038 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 249565852 74906 51039 CBX1 10951 NA PYRIDOSTIGMINE PYRIDOSTIGMINE 74907 51040 KDM4A 9682 DRUGGABLE GENOME, ENZYME CARBIDOPA CARBIDOPA 74909 51041 GLS 2744 ENZYME ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 74910 51042 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RIBOCICLIB RIBOCICLIB 25810375,29408328 74911 51043 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651540 74912 51044 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE Interferon beta-1b 74913 51045 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545322 PANULISIB 74915 51046 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650164 74916 51047 TUBB6 84617 DRUGGABLE GENOME CHEMBL2103826 DAVUNETIDE 74918 51048 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Alkylating Agents 21430602 74919 51049 TUBB3 10381 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 74920 51050 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3545171 PF-05089771 74922 51051 COL4A3 1285 KINASE, DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 74923 51052 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Cetuximab CETUXIMAB 74925 51053 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR daunorubicin DAUNORUBICIN 24141364 74926 51054 GLS 2744 ENZYME CEFOXITIN SODIUM CEFOXITIN SODIUM 74928 51055 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor AZD8330 74931 51056 UGT1A7 54577 DRUGGABLE GENOME, ENZYME risperidone RISPERIDONE 74932 51057 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178103571 74935 51058 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME fluphenazine FLUPHENAZINE 74936 51059 CYP2C18 1562 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME inhibitor 252827490 74937 51060 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MECAMYLAMINE MECAMYLAMINE 22931300 74940 51061 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR NPS-1034 24165158 74941 51062 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1255654 TETRACAINE HYDROCHLORIDE 74942 51063 TOP2B 7155 DRUGGABLE GENOME, ENZYME MLN-576 74943 51064 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-353720 CHEMBL1408276 74944 51065 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-24 74945 51066 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE MDX-1100 ELDELUMAB 74947 51067 ATAD5 79915 NA TCMDC-124307 CHEMBL546865 74950 51068 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME TACRINE TACRINE 25282266 74951 51069 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR MISOPROSTOL MISOPROSTOL 74952 51070 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-6 74953 51071 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 7,8,3'-TRIHYDROXYFLAVONE CHEMBL225513 74955 51072 BAZ2B 29994 NA GNF-PF-3641 CHEMBL599098 74957 51073 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME 2-HYDROXYPHENAZINE 5,10-DIOXIDE CHEMBL179611 74959 51074 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650829 PIOGLITAZONE 74962 51075 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 135650595 METRIBOLONE 74963 51076 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GRAMICIDIN S GRAMICIDIN S 74964 51077 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL564829 MILCICLIB 74965 51078 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME RETINYL ACETATE RETINYL ACETATE 74968 51079 FES 2242 ENZYME, DRUGGABLE GENOME, KINASE, TYROSINE KINASE DASATINIB DASATINIB 74969 51080 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 249565589 BAFETINIB 74970 51081 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME dolutegravir DOLUTEGRAVIR 24329186 74971 51082 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RIFAMPICIN RIFAMPIN 22931300 74972 51083 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor PX-866 SONOLISIB 74973 51084 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CHLOROXINE CHLOROXINE 74976 51085 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Fluoxetine FLUOXETINE 74977 51086 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME AMPHETAMINE AMPHETAMINE 2874568 74978 51087 DNER 92737 NA Isoxazole-based bicyclic compound 7 74979 51088 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Streptokinase STREPTOKINASE 74981 51089 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor GDC-0980 APITOLISIB 74983 51090 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR METHOXYARACHIDONOYL FLUOROPHOSPHONATE METHOXYARACHIDONOYL FLUOROPHOSPHONATE 74984 51091 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ENTRECTINIB ENTRECTINIB 74988 51092 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ANASTROZOLE ANASTROZOLE 74989 51093 PSMA4 5685 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL325041 BORTEZOMIB 74990 51094 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE unspecified IGF-1R antibody 26577700 74991 51095 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor TEMSIROLIMUS TEMSIROLIMUS 74993 51096 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR activator CHEMBL1201448 ARDEPARIN SODIUM 74994 51097 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 178103352 IDELALISIB 74997 51098 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL30219 METHOHEXITAL SODIUM 74998 51099 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 384403651 74999 51100 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor ENMD-2076 ENMD-2076 75000 51101 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CATECHOL CATECHOL 75002 51102 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor CHEMBL598797 CUDC-101 75003 51103 TOP2B 7155 DRUGGABLE GENOME, ENZYME 13-DEOXYADRIAMYCIN HYDROCHLORIDE 75004 51104 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME AURANOFIN AURANOFIN 75005 51105 COL3A1 1281 DRUGGABLE GENOME COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 75006 51106 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME activator 375973254 75008 51107 CBX1 10951 NA AMIODARONE AMIODARONE 75012 51108 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME INCOMPLETE FREUND'S ADJUVANT 11768621 75016 51109 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-125784 CHEMBL581574 75018 51110 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DNDI1417086 CHEMBL1224755 75020 51111 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE MORONIC ACID MORONIC ACID 21453996 75021 51112 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Aryl methoxyacrylate derivative 1 75022 51113 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE ENMD-2076 ENMD-2076 75023 51114 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME topotecan TOPOTECAN 27052877 75025 51115 XDH 7498 DRUGGABLE GENOME, ENZYME Azaindole derivative 7 75027 51116 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME US9024044, 1 75030 51117 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR ACTIVIN 12606325 75031 51118 GALK1 2584 ENZYME, DRUGGABLE GENOME, KINASE SURAMIN HEXASODIUM SURAMIN HEXASODIUM 75032 51119 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL1950289 TANZISERTIB 75037 51120 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-8 75038 51121 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIAZIRINE DIAZIRINE 20006518 75039 51122 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EVEROLIMUS EVEROLIMUS 75040 51123 TPP2 7174 ENZYME, PROTEASE inhibitor 252166783 75042 51124 FGF19 9965 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR FGFR4 INHIBITOR H3B-6527 29247039 75043 51125 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1034 DICLOFENAC SODIUM 75044 51126 TK1 7083 ENZYME, KINASE, DRUGGABLE GENOME Penciclovir PENCICLOVIR 75045 51127 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor 178101944 ROLIPRAM 75046 51128 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE TYROSINE KINASE INHIBITOR 15498512 75047 51129 RABEP1 9135 CLINICALLY ACTIONABLE, GROWTH FACTOR quetiapine QUETIAPINE 28694205 75048 51130 CYP2J2 1573 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 amiodarone AMIODARONE 19923256 75051 51131 TNFSF14 8740 DRUGGABLE GENOME BAMINERCEPT BAMINERCEPT 75053 51132 PDE4D 5144 DRUGGABLE GENOME, ENZYME AVE-8112 24343458 75054 51133 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BATILOL BATILOL 75055 51134 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2103840 DINACICLIB 75056 51135 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME ALRN-6924 75058 51136 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CVT-6883 GS 6201 75061 51137 TXNRD1 7296 DRUGGABLE GENOME Golden phosphorous acetyletic compound 1 75063 51138 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135649858 DAIDZEIN 75065 51139 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor GSK461364 GSK-461364 75069 51140 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SP-600125 SP-600125 75070 51141 LGR6 59352 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102182 75071 51142 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR 4-TERT-BUTYLCATECHOL CHEMBL220845 75072 51143 TUBA4A 7277 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 75073 51144 SCNN1G 6340 ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE GS-9411 75075 51145 POLK 51426 DNA REPAIR, ENZYME LAVENDUSTIN B LAVENDUSTIN B 75076 51146 SMN1 6606 DRUGGABLE GENOME 2-(2'-METHOXYPHENYL)-1H-INDOLE 2-(2'-METHOXYPHENYL)-1H-INDOLE 75078 51147 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR ALPHA-TOCOPHEROL VITAMIN E 9608545 75079 51148 USP1 7398 DNA REPAIR, PROTEASE, ENZYME 2,4-DIHYDROXYBENZOPHENONE 2,4-DIHYDROXYBENZOPHENONE 75082 51149 DPP9 91039 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 252166751 75083 51150 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME LACTACYSTIN LACTACYSTIN 23547757 75084 51151 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2017974 BUPARLISIB 75085 51152 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE antibody CONATUMUMAB CONATUMUMAB 75086 51153 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME CENISERTIB CENISERTIB 75087 51154 COL1A1 1277 CLINICALLY ACTIONABLE, DRUGGABLE GENOME COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 75088 51155 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-220025 SB-220025 75089 51156 TARDBP 23435 TUMOR SUPPRESSOR DNDI1417181 CHEMBL1537417 75091 51157 BCL2L11 10018 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR corticosteroids 29282361 75093 51158 TARDBP 23435 TUMOR SUPPRESSOR ONONETIN ONONETIN 75094 51159 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ZD1839 GEFITINIB 15155841 75095 51160 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-4786 CHEMBL602363 75097 51161 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PMID30124346-Compound-LDT8 75098 51162 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CID 663143 CHEMBL1342336 75099 51163 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE DOVITINIB DOVITINIB 24448819 75100 51164 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME N/A 75101 51165 DHFR 1719 DRUGGABLE GENOME, ENZYME TOMUDEX RALTITREXED 9816025 75103 51166 BDKRB2 624 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BRADYKININ BRADYKININ 75105 51167 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ZM-39923 HCL CHEMBL538798 75108 51168 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE MOD-4023 SOMATROGON 75109 51169 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE GDC-0980 APITOLISIB 75110 51170 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor ENTINOSTAT ENTINOSTAT 75113 51171 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32y 75114 51172 CSF1 1435 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PEXIDARTINIB PEXIDARTINIB 26222558 75116 51173 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649712 75118 51174 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZD5363 CAPIVASERTIB 75119 51175 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (S,S)-(+)-FENOTEROL CHEMBL389390 75120 51176 GART 2618 ENZYME, DRUGGABLE GENOME AG2034 75121 51177 POLI 11201 DNA REPAIR PURPUROGALLIN PURPUROGALLIN 75122 51178 CFAP44 55779 PROTEASE hmg coa reductase inhibitors 25602530 75123 51179 ALOX15 246 ENZYME, DRUGGABLE GENOME IODOACETAMIDE IODOACETAMIDE 75124 51180 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 315661265 75125 51181 ARG2 384 ENZYME inhibitor 178101800 75127 51182 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-124518 CHEMBL527584 75129 51183 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor RDEA119 75130 51184 LGR4 55366 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100586 75131 51185 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C9 75132 51186 ALOX15 246 ENZYME, DRUGGABLE GENOME THYROXINE THYROXINE 75134 51187 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE PMID25726713-Compound-47 75135 51188 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME capecitabine CAPECITABINE 24338217,20530282 75137 51189 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PHENANTHROLINE PHENANTHROLINE 75138 51190 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DASATINIB DASATINIB 75142 51191 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME L-751250 75143 51192 VCP 7415 TRANSPORTER, ENZYME, DNA REPAIR, DRUGGABLE GENOME HEXACHLOROPHENE HEXACHLOROPHENE 75145 51193 DCLK1 9201 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 75147 51194 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BIMATOPROST BIMATOPROST 75148 51195 MUC16 94025 DRUGGABLE GENOME JCAR020 75149 51196 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE DASATINIB DASATINIB 75150 51197 ATAD5 79915 NA GR-127935 GR-127935 75151 51198 TUBA1A 7846 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 75152 51199 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE L-DOPA LEVODOPA 11134247 75154 51200 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-12 75155 51201 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL377559 RETASPIMYCIN HYDROCHLORIDE 75156 51202 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor PAZOPANIB PAZOPANIB 75158 51203 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ZK-164015 CHEMBL184074 75159 51204 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 381118873 75160 51205 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BECLOMETHASONE BECLOMETHASONE 75165 51206 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CALCITRIOL CALCITRIOL 75166 51207 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE IMATINIB IMATINIB 75168 51208 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 14 75169 51209 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1194 PRILOCAINE 75170 51210 ATXN2 6311 NA PERHEXILINE MALEATE PERHEXILINE MALEATE 75171 51211 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102573 75173 51212 SMN1 6606 DRUGGABLE GENOME INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 75174 51213 PSMC6 5706 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 75175 51214 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME IRETOL IRETOL 75176 51215 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME HEPARIN HEPARIN 75177 51216 LTC4S 4056 ENZYME, DRUGGABLE GENOME US20160326143, 50 75178 51217 BAZ2B 29994 NA NSC-11437 CHEMBL1814509 75179 51218 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CEDIRANIB CEDIRANIB 75181 51219 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 75182 51220 TUBB3 10381 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 75184 51221 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE antithymocyte globulin 24322002 75185 51222 PSMA8 143471 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL325041 BORTEZOMIB 75186 51223 EPHB2 2048 KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 381118815 75187 51224 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME CARFILZOMIB CARFILZOMIB 24524217,23547757 75188 51225 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 75189 51226 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHRYSOPHANOL CHRYSOPHANOL 75190 51227 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE LINIFANIB LINIFANIB 75192 51228 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ROMIDEPSIN ROMIDEPSIN 75193 51229 COL2A1 1280 DRUGGABLE GENOME COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 75194 51230 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000193360 CHEMBL607253 75198 51231 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME DOXEPIN DOXEPIN 75199 51232 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DEQUALINIUM DEQUALINIUM 75202 51233 MAPT 4137 DRUGGABLE GENOME DNDI1417080 CHEMBL1498652 75204 51234 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME THUNBERGINOL B THUNBERGINOL B 75205 51235 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor GDC-0973 COBIMETINIB 75206 51236 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-3925 CHEMBL584248 75208 51237 POLI 11201 DNA REPAIR TYRPHOSTIN 25 TYRPHOSTIN 25 75209 51238 CBX1 10951 NA CYSTAMINE CYSTAMINE 75210 51239 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE Vx-001 75213 51240 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME KENPAULLONE KENPAULLONE 75214 51241 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME HYDRALAZINE HYDRALAZINE 75215 51242 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE OESTRADIOL ESTRADIOL 17068109 75216 51243 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TCMDC-124336 CHEMBL527271 75219 51244 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1201081 METHYLPREDNISOLONE SODIUM SUCCINATE 75220 51245 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 363894221 CENISERTIB 75222 51246 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200395 ORPHENADRINE CITRATE 75223 51247 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33j 75225 51248 POLI 11201 DNA REPAIR DITHIAZANINE DITHIAZANINE 75228 51249 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 METHOTREXATE METHOTREXATE 22931300 75229 51250 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE PI-88 MUPARFOSTAT 75231 51251 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649668 75232 51252 STAR 6770 NA BDNF 15485793 75233 51253 MXI1 4601 TRANSCRIPTION FACTOR TGFBETA1 11420421 75234 51254 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ANCITABINE HYDROCHLORIDE ANCITABINE HYDROCHLORIDE 75235 51255 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor IMATINIB IMATINIB 75236 51256 TGFBR2 7048 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME HESPERETIN HESPERETIN 23153811 75237 51257 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Bavencio avelumab 75239 51258 ALOX15 246 ENZYME, DRUGGABLE GENOME RS-17053 CHEMBL88272 75241 51259 RCE1 9986 ENZYME, PROTEASE, DRUGGABLE GENOME GNF-PF-763 CHEMBL1576338 75242 51260 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102568 75243 51261 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR antagonist 135649927 75244 51262 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 223366137 75245 51263 PPIA 5478 DRUGGABLE GENOME, ENZYME IMMUNOSUPPRESSIVE 7680683 75246 51264 DNER 92737 NA Isoxazole-based bicyclic compound 3 75247 51265 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AMSACRINE HYDROCHLORIDE AMSACRINE HYDROCHLORIDE 75249 51266 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME INSULIN INSULIN 9329777 75251 51267 GMNN 51053 DRUGGABLE GENOME 5-HYDROXYINDOLE CHEMBL404923 75254 51268 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Hydrazide derivative 4 75255 51269 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL488436 AZD-5438 75257 51270 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE BUTEIN BUTEIN 8982701 75258 51271 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 363894183 75259 51272 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Conjugated estrogens b 75260 51273 GFRA3 2676 EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE, DRUGGABLE GENOME Neublastin 75261 51274 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1401 CHEMBL313938 75263 51275 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker 135651305 VERAPAMIL 75264 51276 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DIALLYLDISULFIDE DIALLYLDISULFIDE 75265 51277 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR BELINOSTAT BELINOSTAT 25937017 75267 51278 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DACTOLISIB DACTOLISIB 22392911 75271 51279 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 EUGENYL BENZOAT EUGENYL BENZOAT 75273 51280 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME GP-120 9878821 75274 51281 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DINITRAMINE DINITRAMINE 75275 51282 PPP1R1B 84152 KINASE ITI-007 LUMATEPERONE 75278 51283 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-22 75279 51284 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor CHEMBL1980391 RG-1530 75281 51285 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE LY3164530 LY-3164530 75283 51286 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650423 75284 51287 LIMK2 3985 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565798 75286 51288 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR LITHIUM LITHIUM 16300803 75287 51289 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR tamoxifen TAMOXIFEN 24185512,24185510,17713466 75288 51290 TAT 6898 ENZYME BENZNIDAZOLE BENZNIDAZOLE 17678649 75291 51291 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE CYC-116 CYC-116 75292 51292 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Vismodegib VISMODEGIB 75293 51293 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Figure2-Artoxanthochromane 75294 51294 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXADIAZON OXADIAZON 75295 51295 TMSB10 9168 NA MELATONIN MELATONIN 12188030 75299 51296 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-1731 CHEMBL581251 75301 51297 KDM4A 9682 DRUGGABLE GENOME, ENZYME 4-({[2-(BENZYLOXY)PHENYL]METHYL}AMINO)PHENOL CHEMBL1465049 75302 51298 AMH 268 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ETHINYL ESTRADIOL 4049280 75303 51299 CD7 924 DRUGGABLE GENOME Anti-CD7 CAR-T cells 75304 51300 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL568 OXAZEPAM 75305 51301 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MLS003106905 75306 51302 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 405560388 75307 51303 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 178102525 75308 51304 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GUANIDINONALTRINDOLE GUANIDINONALTRINDOLE 75309 51305 PSMA2 5683 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL371405 MARIZOMIB 75310 51306 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HALOTHANE HALOTHANE 75311 51307 ALDH1A1 216 DRUGGABLE GENOME, ENZYME LAWSONE LAWSONE 75312 51308 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ESTRADIOL ESTRADIOL 75313 51309 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME BGB-283 LIFIRAFENIB 26208524 75314 51310 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROMAZINE HYDROCHLORIDE PROMAZINE HYDROCHLORIDE 75315 51311 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist 178100807 75316 51312 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALPHA-PHELLANDRENE ALPHA-PHELLANDRENE 75317 51313 TUBB6 84617 DRUGGABLE GENOME NSC-751382 CHEMBL1935538 22435708 75318 51314 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE PROTEIN KINASE C INHIBITOR 7684044 75319 51315 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135649755 75320 51316 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Romiplostim ROMIPLOSTIM 75321 51317 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ATROPINE ATROPINE 75322 51318 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MEGESTROL MEGESTROL 75324 51319 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 384403641 RG-1530 75328 51320 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200865 LOTEPREDNOL ETABONATE 75329 51321 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME 20(S)-GINSENOSIDE RG3 CHEMBL398412 24968750 75330 51322 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BROMOCRIPTINE MESYLATE BROMOCRIPTINE MESYLATE 75331 51323 CA2 760 DRUGGABLE GENOME, ENZYME inhibitor 385612194 75332 51324 BAZ2B 29994 NA GNF-PF-372 CHEMBL580155 75333 51325 S100B 6285 DRUGGABLE GENOME, KINASE STZ STREPTOZOCIN 14583344 75334 51326 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME MEDICATION 12614997 75335 51327 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor ORANTINIB ORANTINIB 75337 51328 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Dibenzo [c,f]-[2,7]naphthyridine derivative 1 75340 51329 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER ENZASTAURIN ENZASTAURIN 75341 51330 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE RIMONABANT RIMONABANT 21511945 75342 51331 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME mycophenolate mofetil 21142914,21878834 75343 51332 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 178101088 75345 51333 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 328083473 CHEMBL1951415 75347 51334 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor CHEMBL3544964 RAVOXERTINIB 75348 51335 GSTM1 2944 DRUGGABLE GENOME, ENZYME ANTITUBERCULOSIS 11595069 75349 51336 PGA5 5222 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166834 75350 51337 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL52885 ENMD-981693 75351 51338 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL1091644 LINSITINIB 75352 51339 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CCT241161 25500121,23431193 75354 51340 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Selexipag SELEXIPAG 75355 51341 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER daunorubicin DAUNORUBICIN 25558979,20938465,25567217,16331627 75356 51342 DLL3 10683 NA Rova-T ROVALPITUZUMAB TESIRINE 75357 51343 SLCO1A2 6579 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101449 NARINGIN 75358 51344 NUDT15 55270 ENZYME, CLINICALLY ACTIONABLE Azathioprine AZATHIOPRINE 75359 51345 EPHB6 2051 DRUGGABLE GENOME, KINASE, TYROSINE KINASE inhibitor CHEMBL24828 VANDETANIB 75361 51346 PAK2 5062 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 310264718 PF-03758309 75364 51347 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor GANETESPIB GANETESPIB 75365 51348 PAK3 5063 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 310264718 PF-03758309 75368 51349 ALOX15 246 ENZYME, DRUGGABLE GENOME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 75369 51350 TUBA1C 84790 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 75371 51351 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ERGONOVINE ERGONOVINE 75373 51352 HEXB 3074 ENZYME CORTISONE CORTISONE 7388056 75375 51353 TAC1 6863 DRUGGABLE GENOME BACLOFEN BACLOFEN 2467977 75378 51354 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BELINOSTAT BELINOSTAT 25937017 75379 51355 EPHA3 2042 ENZYME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL24828 VANDETANIB 75381 51356 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 354702258 DERAZANTINIB 75382 51357 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE AC480 AC-480 75383 51358 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DYCLONINE HYDROCHLORIDE DYCLONINE HYDROCHLORIDE 75384 51359 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME THERAPEUTIC GLUCOCORTICOID 21390130 75386 51360 MPHOSPH8 54737 NA ZM-39923 HCL CHEMBL538798 75387 51361 TRH 7200 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 6774314 75389 51362 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SBI-0640756 20531415,26603897 75390 51363 POLK 51426 DNA REPAIR, ENZYME AMENTOFLAVONE AMENTOFLAVONE 75391 51364 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE SULFINPYRAZONE SULFINPYRAZONE 75392 51365 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME SAFINAMIDE SAFINAMIDE 75394 51366 DPP7 29952 PROTEASE, ENZYME, DRUGGABLE GENOME BDBM50434164 75396 51367 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR YM-598 NEBENTAN 75398 51368 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME PMID27539678-Compound-9 75400 51369 SPTLC2 9517 ENZYME inhibitor 178103276 MYRIOCIN 75401 51370 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651848 OXYTOCIN 75402 51371 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL2364574 DOXYCYCLINE CALCIUM 75403 51372 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652109 75404 51373 KMO 8564 DRUGGABLE GENOME, ENZYME Aryl pyrimidine derivative 5 75405 51374 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL17350 TRAXOPRODIL 75406 51375 NDUFS4 4724 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 75407 51376 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 75409 51377 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL428647 PACLITAXEL 75411 51378 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545263 LGX-806 75413 51379 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME activator 375973254 75415 51380 NQO2 4835 DRUGGABLE GENOME, ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 29938344,21946896 75416 51381 POLI 11201 DNA REPAIR CLOZAPINE CLOZAPINE 75417 51382 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 135650234 EPHEDRINE 75418 51383 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR KETOCONAZOLE KETOCONAZOLE 75419 51384 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE TOZASERTIB TOZASERTIB 75421 51385 CD52 1043 DRUGGABLE GENOME GZ402668 75422 51386 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BICALUTAMIDE BICALUTAMIDE 12517791,26000489,29211833 75423 51387 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE MK2206 MK-2206 26187616,26627007,26084990,21289267,22932669 75424 51388 KCNJ5 3762 TRANSPORTER, ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME activator 135651544 75426 51389 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 4 75427 51390 HSPA4 3308 NA DEFEROXAMINE DEFEROXAMINE 11579132 75428 51391 SLC19A2 10560 TRANSPORTER 178101346 75429 51392 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Ipatasertib IPATASERTIB 24141624 75430 51393 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-117023 CHEMBL2059274 22524450 75432 51394 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR K-252A K-252A 16797499 75433 51395 EYA2 2139 DNA REPAIR NSC-107022 CHEMBL1601846 75435 51396 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CLARITHROMYCIN CLARITHROMYCIN 22931300 75436 51397 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Erlotinib ERLOTINIB 75438 51398 ATAD5 79915 NA N-PHENETHYLCINNAMAMIDE CHEMBL1305393 75440 51399 PDE4A 5141 DRUGGABLE GENOME, ENZYME MEM-1414 75441 51400 HSPB2 3316 KINASE RESVERATROL RESVERATROL 17125593,16759640 75442 51401 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565843 75444 51402 PON1 5444 ENZYME, TRANSPORTER, DRUGGABLE GENOME QUERCETIN QUERCETIN 23623675 75448 51403 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME PREDNICARBATE PREDNICARBATE 75454 51404 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PANITUMUMAB PANITUMUMAB 19223544 75455 51405 LOXL2 4017 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 252166622 SIMTUZUMAB 75457 51406 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DINALINE DINALINE 75458 51407 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE KRIBB11 75459 51408 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 223366166 LOSMAPIMOD 75461 51409 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 249565841 75465 51410 MAPT 4137 DRUGGABLE GENOME GNF-PF-4227 CHEMBL585654 75467 51411 MCOLN2 255231 ION CHANNEL, DRUGGABLE GENOME activator 381744982 75469 51412 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME ASTERRIC ACID ASTERRIC ACID 75472 51413 ALOX15 246 ENZYME, DRUGGABLE GENOME AG-555 CHEMBL53898 75477 51414 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 252166674 75480 51415 FAAH 2166 ENZYME, DRUGGABLE GENOME Tetra-hydro-naphthalene derivative 1 75481 51416 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE SIROLIMUS SIROLIMUS 75482 51417 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CHF 4227 75484 51418 MMP7 4316 NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, ENZYME, PROTEASE Prinomastat PRINOMASTAT 75486 51419 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE Temsirolimus TEMSIROLIMUS 27016228 75489 51420 PLAUR 5329 DRUGGABLE GENOME, ENZYME, CELL SURFACE DIPHTHERIA TOXIN 11959893 75490 51421 TOP2B 7155 DRUGGABLE GENOME, ENZYME Rosoxacin ROSOXACIN 75491 51422 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DROFENINE HYDROCHLORIDE DROFENINE HYDROCHLORIDE 75492 51423 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME tetrabenazine TETRABENAZINE 23280482 75493 51424 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME PHA-739358 DANUSERTIB 75495 51425 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ASC-J9 75497 51426 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE ALISERTIB ALISERTIB 75498 51427 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist CHEMBL1131 ACITRETIN 75499 51428 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME TAE-684 TAE-684 75501 51429 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME inhibitor 178103582 PLUMBAGIN 75502 51430 ALDH1A1 216 DRUGGABLE GENOME, ENZYME HARMINE HARMINE 75503 51431 SIRT5 23408 ENZYME NSC-74859 CHEMBL477936 75504 51432 PRDX5 25824 ENZYME Diterpene triepoxide derivative 1 75505 51433 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME Dihydrothieno [2,3-e]indazole derivative 3 75507 51434 DGAT1 8694 ENZYME, DRUGGABLE GENOME Azole derivative 6 75508 51435 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME TOZASERTIB TOZASERTIB 75509 51436 FUT2 2524 DRUGGABLE GENOME, ENZYME ethanol ALCOHOL 32451486 75510 51437 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CANDESARTAN CILEXETIL CANDESARTAN CILEXETIL 75511 51438 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME inhibitor 178100439 GEMFIBROZIL 75512 51439 PGA5 5222 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL2367706 SUCRALFATE 75513 51440 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME TAE-684 TAE-684 75514 51441 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR KETOCONAZOLE KETOCONAZOLE 75515 51442 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 249565576 ENMD-2076 75517 51443 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BUTYL 2-AMINOBENZOATE BUTYL 2-AMINOBENZOATE 75518 51444 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201149 NALTREXONE HYDROCHLORIDE 75519 51445 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 249565720 75521 51446 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200420 MIDAZOLAM HYDROCHLORIDE 75523 51447 SLC1A1 6505 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME 178101410 75524 51448 UBE2N 7334 ENZYME, DRUGGABLE GENOME FLUPHENAZINE HYDROCHLORIDE FLUPHENAZINE HYDROCHLORIDE 75525 51449 BAZ2B 29994 NA GNF-PF-3350 CHEMBL600747 75527 51450 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IODOFORM IODOFORM 75531 51451 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 18 75533 51452 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-36 75534 51453 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-180246 CHEMBL484640 75535 51454 GMNN 51053 DRUGGABLE GENOME ISOVELLERAL ISOVELLERAL 75536 51455 ATAD5 79915 NA IDAZOXAN IDAZOXAN 75538 51456 ALDH1A1 216 DRUGGABLE GENOME, ENZYME RO-194603 RO-194603 75539 51457 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME COUMARIN COUMARIN 22931300 75541 51458 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ETHAMSYLATE ETHAMSYLATE 75542 51459 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ALTENUSIN ALTENUSIN 75543 51460 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE GAMBOGIC AMIDE GAMBOGIC AMIDE 17911251 75545 51461 TUBB6 84617 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 75546 51462 MUC16 94025 DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 10629663 75547 51463 L1CAM 3897 CELL SURFACE, DRUGGABLE GENOME, KINASE JCAR023 75549 51464 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FOLPET FOLPET 75550 51465 F7 2155 ENZYME, DRUGGABLE GENOME, PROTEASE Activated recombinant FVII-albumin fusion protein 75551 51466 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CEFOPERAZONE CEFOPERAZONE 22931300 75552 51467 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME DACARBAZINE DACARBAZINE 14512787 75555 51468 MAPT 4137 DRUGGABLE GENOME GNF-PF-3756 CHEMBL597035 75556 51469 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME CELECOXIB CELECOXIB 12000750 75557 51470 CCND3 896 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PD 0332991 75558 51471 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 75559 51472 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE Muromonab MUROMONAB-CD3 75560 51473 TSPO 706 DRUGGABLE GENOME Benzothiazepine analog 8 75561 51474 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Olodaterol OLODATEROL 75562 51475 GSTT1 2952 DRUGGABLE GENOME xenobiotics 9285043,9851677,11317340 75563 51476 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 363894207 FLUMATINIB 75566 51477 GRB2 2885 NA TCDD 9918770 75567 51478 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CE-224535 CE-224535 75568 51479 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR AZD0284 75569 51480 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BIPHENYL-4-AMINE BIPHENYL-4-AMINE 75570 51481 KDM4A 9682 DRUGGABLE GENOME, ENZYME S(+)-ISOPROTERENOL-BITARTRATE CHEMBL1257092 75571 51482 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME paclitaxel PACLITAXEL 27075627 75573 51483 CXCL8 3576 DRUGGABLE GENOME NAPROXEN NAPROXEN 11852880 75574 51484 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TDR84367 CHEMBL1485420 75576 51485 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME GNF-PF-5151 CHEMBL576208 75577 51486 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor 223366136 75578 51487 CCN2 1490 DRUGGABLE GENOME, GROWTH FACTOR SPIRONOLACTONE SPIRONOLACTONE 17602195 75579 51488 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PYRILAMINE PYRILAMINE 22931300 75580 51489 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178100903 75581 51490 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 7-METHOXYISOFLAVONE CHEMBL563919 75582 51491 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME CRA-024781 ABEXINOSTAT 75583 51492 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE TETRANDRINE 8250973 75584 51493 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME antibody ZIV-AFLIBERCEPT AFLIBERCEPT 75585 51494 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME platinum PLATINUM 19434073,22188361,29662106,22026922,21449681 75587 51495 BAZ2B 29994 NA MMV085203 CHEMBL586031 75588 51496 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AFATINIB AFATINIB 75589 51497 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DEXPROPRANOLOL DEXPROPRANOLOL 75591 51498 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 252827503 CGS-27023A 75592 51499 BAZ2B 29994 NA SULFURETIN SULFURETIN 75593 51500 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 329968433 75594 51501 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor DACTOLISIB DACTOLISIB 75597 51502 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME blocker 178101137 75598 51503 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LINOLENIC ACID LINOLENIC ACID 75599 51504 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER inhibitor 249565822 BALANOL 75604 51505 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE VIROSOME-BASED BREAST CANCER VACCINE 75605 51506 STING1 340061 CLINICALLY ACTIONABLE, KINASE MK-1454 75606 51507 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200586 PRILOCAINE HYDROCHLORIDE 75608 51508 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME MESO-2,3-DIMERCAPTOSUCCINIC ACID CHEMBL28721 75610 51509 TUBB4B 10383 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 75612 51510 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545322 PANULISIB 75614 51511 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SVT-40776 TARAFENACIN 75615 51512 PAH 5053 DRUGGABLE GENOME, ENZYME Sapropterin hydrochloride 75616 51513 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PD-0166285 PD-0166285 75619 51514 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NOT DISCLOSED 75620 51515 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DIMERCAPROL DIMERCAPROL 75621 51516 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Palbociclib PALBOCICLIB 27012813,22711607,27020857,26649278,27488531,20354191 75622 51517 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL3545165 AFACIFENACIN 75628 51518 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 hormonal contraceptives for systemic use 28750087 75629 51519 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Tonapofylline TONAPOFYLLINE 75630 51520 ANO1 55107 ION CHANNEL blocker 178101087 75631 51521 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME LIFITEGRAST LIFITEGRAST 75632 51522 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME CENISERTIB CENISERTIB 75634 51523 RACGAP1 29127 NA NSC-155693 CHEMBL68096 75635 51524 MMP7 4316 NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor CHEMBL2364574 DOXYCYCLINE CALCIUM 75637 51525 MGAT4A 11320 DRUGGABLE GENOME oxaliplatin OXALIPLATIN 26222057 75638 51526 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-49 75639 51527 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-308 CHEMBL600334 75641 51528 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OT-730 75642 51529 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ACRIFLAVINE CHLORIDE ACRIFLAVINE 75645 51530 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME 2-ENE-VALPROATE CHEMBL117487 17566732 75646 51531 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 252166732 75648 51532 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 8-GERANYLOXY PSORALEN CHEMBL1412710 75651 51533 IL1R1 3554 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ANAKINRA ANAKINRA 75652 51534 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME TRIAMCINOLONE TRIAMCINOLONE 75653 51535 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL inhibitor 178102896 75654 51536 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE FLUOROURACIL FLUOROURACIL 18704422,26693073 75657 51537 MAPT 4137 DRUGGABLE GENOME NSC-111847 CHEMBL1984884 75658 51538 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME DNA fusion vaccine 75659 51539 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL BUTABARBITAL BUTABARBITAL 75662 51540 PTGS2 5743 DRUGGABLE GENOME, ENZYME ACETAMINOPHEN ACETAMINOPHEN 75663 51541 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL2103852 CROLIBULIN 75664 51542 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR ALISOL A-23 ACETATE CHEMBL2059711 24915879 75665 51543 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor 354702261 75670 51544 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545431 HMN-214 75671 51545 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GANETESPIB GANETESPIB 75673 51546 POLI 11201 DNA REPAIR 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 75675 51547 BMP7 655 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR cytarabine CYTARABINE 26590194 75679 51548 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178102354 75680 51549 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CYCLOSPORINE CYCLOSPORINE 22931300 75681 51550 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-640584 CHEMBL476968 21074425 75683 51551 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE MP470 75684 51552 NOS2 4843 DRUGGABLE GENOME, ENZYME DNCB 17373747 75685 51553 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL atorvastatin ATORVASTATIN 27839692,25753936 75687 51554 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-62 75688 51555 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178103586 ENTINOSTAT 75689 51556 TUBB2A 7280 DRUGGABLE GENOME inhibitor CHEMBL501867 VINCRISTINE SULFATE 75690 51557 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 363894134 75691 51558 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Dabrafenib DABRAFENIB 25370473,24265153,22389471,27312529,24463458,24265154 75694 51559 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHYL ALCOHOL METHYL ALCOHOL 75699 51560 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 405560388 75701 51561 GATA4 2626 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE NSC-140905 CHEMBL1684097 21310620 75702 51562 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Adenosine triphosphate 75704 51563 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR PMID27410995-Compound-Figure3j 75705 51564 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 75706 51565 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE EVT-401 EVT401 75710 51566 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR TCMDC-124266 CHEMBL124006 75712 51567 IL1RN 3557 DRUGGABLE GENOME Tumor necrosis factor alpha (TNF-alpha) inhibitors 24776844 75713 51568 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL1421 DASATINIB 75715 51569 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL1079175 MK-2206 75717 51570 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PD98509 22662154 75718 51571 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AMIODARONE HYDROCHLORIDE AMIODARONE HYDROCHLORIDE 75719 51572 NDUFV2 4729 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 75723 51573 KLK4 9622 PROTEASE, DRUGGABLE GENOME, ENZYME Benzyl amine derivative 2 75724 51574 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL2364638 UBROGEPANT 75725 51575 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FENTHION FENTHION 75726 51576 POLD1 5424 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME HYMENOIC ACID HYMENOIC ACID 18364258 75727 51577 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 5 75728 51578 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE ENMD-2076 ENMD-2076 75729 51579 GMNN 51053 DRUGGABLE GENOME DIBUCAINE HYDROCHLORIDE DIBUCAINE HYDROCHLORIDE 75731 51580 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME blocker CHEMBL1697 DILTIAZEM HYDROCHLORIDE 75732 51581 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CARNOSIC ACID CARNOSIC ACID 75733 51582 POLK 51426 DNA REPAIR, ENZYME CARMINIC ACID CARMINIC ACID 75734 51583 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL289351 FOSBRETABULIN DISODIUM 75738 51584 PTGES 9536 DRUGGABLE GENOME, ENZYME Benzimidazole derivative 11 75741 51585 PSMB6 5694 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL2103884 OPROZOMIB 75742 51586 PIK3C2B 5287 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor SOPHORETIN QUERCETIN 75743 51587 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ALEFACEPT ALEFACEPT 75744 51588 CBX1 10951 NA ELLIPTECINE ELLIPTECINE 75745 51589 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME R667 75746 51590 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL partial agonist CHEMBL2103791 ADIPIPLON 75750 51591 RABEP1 9135 CLINICALLY ACTIONABLE, GROWTH FACTOR paliperidone PALIPERIDONE 28694205 75751 51592 CPS1 1373 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME antiepileptics 20456087 75754 51593 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ramucirumab RAMUCIRUMAB 75755 51594 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649785 75758 51595 ALPL 249 ENZYME, DRUGGABLE GENOME TCMDC-123713 CHEMBL586135 75760 51596 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NEOSTIGMINE BROMIDE NEOSTIGMINE BROMIDE 22931300 75762 51597 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME (S)-(+)-Dimethindene maleate 75763 51598 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME mianserin MIANSERIN 14652703,1527229,8062494,9408809 75764 51599 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-13 75769 51600 COMT 1312 DRUGGABLE GENOME, ENZYME levodopa LEVODOPA 75770 51601 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME ISOKAEMPFERIDE ISOKAEMPFERIDE 75771 51602 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER CEFTRIAXONE CEFTRIAXONE 22166395 75772 51603 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor MASITINIB MASITINIB 75773 51604 IRS1 3667 KINASE, CLINICALLY ACTIONABLE cyclophosphamide CYCLOPHOSPHAMIDE 75775 51605 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME HORMONES 8593784 75779 51606 KDM5C 8242 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE SUNITINIB SUNITINIB 27751729 75781 51607 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TYRPHOSTIN 47 TYRPHOSTIN 47 75782 51608 SMYD2 56950 ENZYME, METHYL TRANSFERASE inhibitor 310264734 75783 51609 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Suronacrine maleate 75784 51610 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR ARRY-162 BINIMETINIB 75785 51611 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 7-OXOCALLITRISIC ACID, METHYL ESTER 7-OXOCALLITRISIC ACID, METHYL ESTER 75786 51612 BCHE 590 DRUGGABLE GENOME, ENZYME oxymetazoline and tetracaine 75787 51613 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE mepivacaine MEPIVACAINE 75788 51614 FSCN1 6624 NA NP-G2-044 NP-G2-044 75789 51615 GAPDH 2597 DRUGGABLE GENOME, ENZYME PROTEIN SYNTHESIS INHIBITOR 9437188 75790 51616 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 erythromycin ERYTHROMYCIN 9187528,23327575 75791 51617 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME Estradiol ESTRADIOL 75793 51618 ATXN2 6311 NA IDARUBICIN IDARUBICIN 75795 51619 TUBA3C 7278 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 75796 51620 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 7,8,2'-TRIHYDROXYFLAVONE CHEMBL244707 75797 51621 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Flavonoid derivative 6 75798 51622 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZO(K)FLUORANTHENE BENZO(K)FLUORANTHENE 75799 51623 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NSC-663284 CHEMBL337173 75800 51624 KDM4A 9682 DRUGGABLE GENOME, ENZYME CB7969312 CHEMBL599255 75801 51625 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-3029 CHEMBL601554 75802 51626 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME ENMD-2076 ENMD-2076 75803 51627 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE METHYLCURCUMIN METHYLCURCUMIN 25753330 75804 51628 MAOA 4128 DRUGGABLE GENOME, ENZYME TRANYLCYPROMINE TRANYLCYPROMINE 75805 51629 ACP1 52 ENZYME, DRUGGABLE GENOME, PROTEIN PHOSPHATASE FIDUXOSIN HYDROCHLORIDE FIDUXOSIN HYDROCHLORIDE 75806 51630 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE DURVALUMAB DURVALUMAB 31086949 75809 51631 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-2383 CHEMBL578915 75810 51632 SOAT1 6646 DRUGGABLE GENOME URSODEOXYCHOLIC ACID 7949265 75811 51633 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME EPINASTINE EPINASTINE 75812 51634 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PRN1371 75814 51635 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 252827493 75815 51636 GPA33 10223 DRUGGABLE GENOME KRN-330 KRN-330 75816 51637 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor CHEMBL52885 ENMD-981693 75818 51638 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 9-AMINOCAMPTOTHECIN 9-AMINOCAMPTOTHECIN 75820 51639 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545196 PD-0166285 75821 51640 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BENZO(K)FLUORANTHENE BENZO(K)FLUORANTHENE 75825 51641 S100A2 6273 NA ANTISERUM 9463588 75826 51642 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIFLUPREDNATE DIFLUPREDNATE 75827 51643 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 354702234 75828 51644 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 erdafitinib ERDAFITINIB 75829 51645 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TEBUFENOZIDE TEBUFENOZIDE 75830 51646 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IPCONAZOLE IPCONAZOLE 75833 51647 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL656 OXYCODONE 75836 51648 TSPO 706 DRUGGABLE GENOME Indole-based analog 9 75837 51649 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CATECHOL CATECHOL 75838 51650 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TAMOXIFEN CITRATE TAMOXIFEN CITRATE 75841 51651 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME MLN-8237 ALISERTIB 75842 51652 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE HYCANTHONE HYCANTHONE 75844 51653 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME FK 506 14550820 75847 51654 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DNDI1417132 CHEMBL1492017 75848 51655 EIF2AK4 440275 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME haloperidol HALOPERIDOL 27023437,24751813 75850 51656 BAZ2B 29994 NA 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 75851 51657 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Tramiprosate TRAMIPROSATE 75852 51658 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor SAR260301 SAR-260301 75853 51659 ATP1A2 477 ENZYME, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME inhibitor CHEMBL1751 DIGOXIN 75854 51660 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ARACHIDONOYL GABA ARACHIDONOYL GABA 75857 51661 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME INTERFERON BETA 9075665 75858 51662 CBX1 10951 NA TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 75859 51663 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-16 75860 51664 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME allosteric modulator 178102297 BMS-345541 75862 51665 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103497 75863 51666 CBX1 10951 NA CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 75865 51667 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200773 TOCAINIDE HYDROCHLORIDE 75866 51668 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 315661205 75868 51669 TUBB 203068 DRUGGABLE GENOME Vincristine VINCRISTINE 75869 51670 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CYCLOSPORINE CYCLOSPORINE 1972761 75873 51671 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PF-05212384 GEDATOLISIB 75874 51672 NEK11 79858 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565802 75876 51673 BAZ2B 29994 NA DEFERIPRONE DEFERIPRONE 75878 51674 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE LAPATINIB LAPATINIB 17192538,16091755,22257673,27108243,26296355,25398453,24868024,26811533,23122784,22046346,19228746,23220880,22493419,27697991,26243863,20124187 75879 51675 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME PINAFIDE PINAFIDE 75880 51676 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME COBALT 15878362 75881 51677 NLK 51701 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565802 75882 51678 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody MEHD7945 A 75884 51679 TNNC1 7134 DRUGGABLE GENOME PYROGALLOL RED PYROGALLOL RED 75885 51680 POLB 5423 DNA REPAIR, DRUGGABLE GENOME HYCANTHONE HYCANTHONE 75888 51681 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651020 75890 51682 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VER-49009 CHEMBL365617 75893 51683 GBA 2629 DRUGGABLE GENOME, ENZYME 404859144 75894 51684 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651400 DP001 75895 51685 RPS6KA2 6196 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565718 CHEMBL573107 75896 51686 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Everolimus EVEROLIMUS 23629727,20664174,20664172,26725216,22662154 75897 51687 GAA 2548 DRUGGABLE GENOME, ENZYME NSC-638080 CHEMBL136344 75898 51688 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX BIX-01294 CHEMBL569864 75900 51689 QRFPR 84109 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178100650 75901 51690 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antibody RAMUCIRUMAB RAMUCIRUMAB 75902 51691 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TORMENTIC ACID METHYL ESTER TORMENTIC ACID METHYL ESTER 20100662 75904 51692 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME VAN-10-4-eluting stent 75906 51693 CASP14 23581 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL197672 EMRICASAN 75909 51694 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME inhibitor REOLYSIN PELAREOREP 75910 51695 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME INDIRUBIN SULFATE SU-9516 75911 51696 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 354702275 75912 51697 TARDBP 23435 TUMOR SUPPRESSOR DNDI1417254 CHEMBL2094567 75913 51698 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CENISERTIB CENISERTIB 75914 51699 HSPA4 3308 NA SODIUM SALICYLATE 16184763 75915 51700 GAS6 2621 DRUG RESISTANCE, DRUGGABLE GENOME, KINASE DOCETAXEL DOCETAXEL 27153245 75916 51701 GSTM1 2944 DRUGGABLE GENOME, ENZYME dacarbazine DACARBAZINE 23323945 75917 51702 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HEXYLRESORCINOL HEXYLRESORCINOL 75918 51703 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 249565775 75921 51704 DNER 92737 NA BMS-986158 BMS-986158 75922 51705 FAAH 2166 ENZYME, DRUGGABLE GENOME Pyrazole derivative 82 75923 51706 BRCA2 675 CLINICALLY ACTIONABLE VELIPARIB VELIPARIB 75924 51707 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 249565800 75925 51708 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON BETA-1A 75926 51709 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Quinine Sulfate 75927 51710 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AMBUNOL AMBUNOL 75929 51711 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545152 PEGCANTRATINIB 75934 51712 ADH1A 124 DRUGGABLE GENOME inhibitor CHEMBL1308 FOMEPIZOLE 75937 51713 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR FULVESTRANT FULVESTRANT 24185510 75940 51714 GMNN 51053 DRUGGABLE GENOME TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 75941 51715 POLB 5423 DNA REPAIR, DRUGGABLE GENOME RHEIN RHEIN 75942 51716 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME IMATINIB IMATINIB 24186003 75943 51717 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME PAROXETINE PAROXETINE 75945 51718 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545251 SURUFATINIB 75946 51719 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor 249565581 AFURESERTIB 75947 51720 RAB9A 9367 ENZYME, DRUGGABLE GENOME TCMDC-124327 CHEMBL581929 75948 51721 DDC 1644 ENZYME, DRUGGABLE GENOME inhibitor 178101851 CARBIDOPA 75950 51722 BMP2 650 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BUTYL 4-ACETAMIDOBENZOATE CHEMBL1321401 22041064 75951 51723 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Anagliptin ANAGLIPTIN 19246581 75953 51724 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME celecoxib CELECOXIB 22336956 75954 51725 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-(phenylpyrazolyl)benzamide derivative 1 75955 51726 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-710 CHEMBL596839 75956 51727 USP1 7398 DNA REPAIR, PROTEASE, ENZYME QUINACRINE QUINACRINE 75957 51728 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR MT203 NAMILUMAB 75958 51729 SERPINH1 871 PROTEASE INHIBITOR, DRUGGABLE GENOME 11D10 8567753 75959 51730 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME COLFORSIN COLFORSIN 19966789 75961 51731 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NORTRIPTYLINE HYDROCHLORIDE NORTRIPTYLINE HYDROCHLORIDE 75962 51732 APOE 348 DRUGGABLE GENOME HUMAN CHORIONIC GONADOTROPIN 1709885 75963 51733 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor MEKINIST MEKINIST 75964 51734 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Leucovorin LEUCOVORIN 26432108 75965 51735 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PD-0166285 PD-0166285 75967 51736 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME NIMODIPINE NIMODIPINE 8301097 75968 51737 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist CHEMBL3545114 KD3010 75969 51738 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 LORATADINE LORATADINE 75970 51739 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SBI-0640726 26603897 75971 51740 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE GSK-269962A GSK-269962A 75972 51741 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 381118905 75977 51742 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR inhibitor CRIZOTINIB CRIZOTINIB 75978 51743 ATXN2 6311 NA NICLOSAMIDE NICLOSAMIDE 75979 51744 C3 718 PROTEASE INHIBITOR, DRUGGABLE GENOME, CELL SURFACE APL-2 PEGCETACOPLAN 75980 51745 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME Tricyclic compound 8 75981 51746 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3218576 COPANLISIB 75983 51747 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME ANDROGRAPHOLIDE ANDROGRAPHOLIDE 25615020 75984 51748 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ISOTRETINOIN ISOTRETINOIN 75985 51749 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 COUMARIN COUMARIN 22931300 75986 51750 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ALFUZOSIN ALFUZOSIN 75987 51751 RFK 55312 KINASE, ENZYME citalopram CITALOPRAM 75990 51752 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CARBIDOPA CARBIDOPA 75992 51753 ATF2 1386 TRANSCRIPTION FACTOR ALPHA-DIFLUOROMETHYLORNITHINE 17804813 75994 51754 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Promethazine PROMETHAZINE 75995 51755 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER EMBELIN EMBELIN 75997 51756 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TINORIDINE TINORIDINE 76002 51757 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ERGOCALCIFEROL ERGOCALCIFEROL 76003 51758 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE CBP-501 CBP-501 76004 51759 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME blocker 135649695 76005 51760 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE N6-PHENYLADENOSINE N6-PHENYLADENOSINE 76007 51761 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor 252166525 TALAZOPARIB 76008 51762 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GW7647 GW7647 76009 51763 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL1614701 SELUMETINIB 76011 51764 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR ALL TRANS-RETINOIC ACID 11720243 76012 51765 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME protriptyline PROTRIPTYLINE 76014 51766 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 310264756 NS-398 76017 51767 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER LGX818 ENCORAFENIB 76018 51768 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BUTACHLOR BUTACHLOR 76019 51769 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LOVASTATIN LOVASTATIN 9553123 76020 51770 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL235191 TACEDINALINE 76021 51771 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME valproic acid 21806385 76022 51772 STAG3 10734 DRUG RESISTANCE VEMURAFENIB VEMURAFENIB 27500726 76026 51773 CP 1356 DRUGGABLE GENOME, ENZYME CARDIOPROTECTIVE AGENT 8285144 76027 51774 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Imatinib IMATINIB 21224473 76028 51775 RPTOR 57521 CLINICALLY ACTIONABLE, KINASE inhibitor OSI-027 OSI-027 76030 51776 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME LINSITINIB LINSITINIB 25670080 76032 51777 GMNN 51053 DRUGGABLE GENOME DECITABINE DECITABINE 76036 51778 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Sulfasalazine SULFASALAZINE 76037 51779 HSD11B2 3291 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CORTISOL HYDROCORTISONE 12788832,15134813 76038 51780 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BIFONAZOLE BIFONAZOLE 76039 51781 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AG-808 CHEMBL68534 76040 51782 BMP7 655 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR vincristine VINCRISTINE 26590194 76041 51783 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 7,12-DIMETHYL-BENZO[A]ANTHRACENE CHEMBL329673 76042 51784 FAAH 2166 ENZYME, DRUGGABLE GENOME Aryl urea derivative 3 76043 51785 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE PKI-594 76044 51786 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TCMDC-123916 CHEMBL493863 76045 51787 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE Pyridine derivative 18 76046 51788 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR E232 E232 76047 51789 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649988 BETHANECHOL 76048 51790 MAPT 4137 DRUGGABLE GENOME 1,2-NAPHTHOQUINONE 1,2-NAPHTHOQUINONE 76050 51791 E2F1 1869 TRANSCRIPTION FACTOR VITAMIN C 16640900,16944783 76051 51792 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE CEFMETAZOLE CEFMETAZOLE 22166395 76053 51793 ALOX5 240 DRUGGABLE GENOME, ENZYME ANACARDIC ACID 24231650 76055 51794 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SANGUINARIUM SANGUINARIUM 76056 51795 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heteroaryl-carboxamide derivative 3 76057 51796 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Methacholine Chloride 76058 51797 PRMT1 3276 ENZYME, METHYL TRANSFERASE EOSIN EOSIN 18348515 76059 51798 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-124544 CHEMBL531322 76060 51799 PSMF1 9491 PROTEASE INHIBITOR inhibitor CARFILZOMIB CARFILZOMIB 76061 51800 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL inhibitor 135651166 76063 51801 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR EPROSARTAN EPROSARTAN 76064 51802 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE antibody CONATUMUMAB CONATUMUMAB 76066 51803 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-105827 CHEMBL171699 76067 51804 XDH 7498 DRUGGABLE GENOME, ENZYME PMID27841045-Compound-135 76068 51805 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 178101871 FASUDIL 76070 51806 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME IL-1 1908322 76072 51807 SMN2 6607 DRUGGABLE GENOME PIPERINE PIPERINE 76073 51808 MARCHF8 220972 ENZYME HB-AS02V 76074 51809 TK1 7083 ENZYME, KINASE, DRUGGABLE GENOME DEOXYCYTIDINE DEOXYCYTIDINE 76075 51810 KLRD1 3824 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME glucocorticoids 26453102 76076 51811 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE homoharringtonine OMACETAXINE MEPESUCCINATE 76078 51812 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PONATINIB PONATINIB 22238366 76079 51813 PSENEN 55851 DRUGGABLE GENOME BMS-708163 AVAGACESTAT 76082 51814 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE inhibitor OPB 51602 76083 51815 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE BUNITROLOL BUNITROLOL 2903243 76084 51816 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ETIDRONIC ACID ETIDRONIC ACID 22931300 76085 51817 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 315661270 76086 51818 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME BMS 936564 76087 51819 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PHA-767491 CHEMBL225519 76088 51820 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 252166792 76089 51821 MAPT 4137 DRUGGABLE GENOME HARMALOL HARMALOL 76090 51822 PDE4A 5141 DRUGGABLE GENOME, ENZYME MEM 1414 76092 51823 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PACLITAXEL PACLITAXEL 76094 51824 GHRL 51738 DRUGGABLE GENOME IL-1RA ANAKINRA 16959954 76095 51825 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 223365887 LOFEPRAMINE 76096 51826 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR SUMATRIPTAN SUMATRIPTAN 76097 51827 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME peginterferon alfa-2a 21572301 76098 51828 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Nadolol NADOLOL 76100 51829 GMNN 51053 DRUGGABLE GENOME FLUORANTHEN-3-YLAMINE CHEMBL103583 76101 51830 TSPO 706 DRUGGABLE GENOME ALPRAZOLAM ALPRAZOLAM 76102 51831 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RO-137410 CHEMBL275311 76103 51832 TXNRD1 7296 DRUGGABLE GENOME Acyl oxymethyl acrylamide ester derivative 2 76106 51833 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650194 DIPRENORPHINE 76107 51834 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-16 76109 51835 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Darusentan DARUSENTAN 76110 51836 SLC29A4 222962 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 135650872 QUINIDINE 76112 51837 MBP 4155 CELL SURFACE INSULIN INSULIN 8948451 76113 51838 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 381118857 76115 51839 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALISERTIB ALISERTIB 76116 51840 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE BARASERTIB BARASERTIB 20684549 76117 51841 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor GSK461364 GSK-461364 76118 51842 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Peginterferon beta 76119 51843 CDH17 1015 TRANSPORTER, CELL SURFACE HGF/SF 10438566 76120 51844 CA1 759 DRUGGABLE GENOME, ENZYME CATECHOL CATECHOL 26073005 76127 51845 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME NORDEFRIN NORDEFRIN 76128 51846 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BRYOSTATIN-1 14980523 76129 51847 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 cytarabine CYTARABINE 22584460 76132 51848 MAP3K9 4293 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565817 76133 51849 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LOVASTATIN LOVASTATIN 18302447,17655375 76134 51850 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME RUFLOXACIN RUFLOXACIN 76135 51851 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHENODIOL CHENODIOL 76136 51852 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417614 CHEMBL1567571 76137 51853 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TYRPHOSTIN 23 TYRPHOSTIN 23 76138 51854 HTT 3064 DRUGGABLE GENOME FLUORESCEIN FLUORESCEIN 76139 51855 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE XL820 76141 51856 GMNN 51053 DRUGGABLE GENOME BITHIONOLOXIDE BITHIONOLOXIDE 76142 51857 CXCL8 3576 DRUGGABLE GENOME QUESTIOMYCIN B QUESTIOMYCIN B 76143 51858 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BITHIONOL BITHIONOL 76144 51859 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Metformin METFORMIN 23986086 76145 51860 STK17A 9263 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME CYC-116 CYC-116 76146 51861 METAP2 10988 ENZYME, DRUGGABLE GENOME, KINASE, PROTEASE SDX-7320 76147 51862 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651784 RELAXIN 76148 51863 GMNN 51053 DRUGGABLE GENOME DNDI1417400 CHEMBL1362503 76149 51864 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR 5-FU FLUOROURACIL 9268987 76151 51865 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Anti-CD3 and anti-Her2/neu bispecific antibody-armed activated T cells 76153 51866 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE 315661316 76154 51867 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201634 INSULIN ZINC SUSP PURIFIED BEEF/PORK 76155 51868 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CLOFAZIMINE CLOFAZIMINE 76156 51869 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME CYC-116 CYC-116 76157 51870 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MACROCARPAL B MACROCARPAL B 22934600 76158 51871 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1201065 THIAMYLAL SODIUM 76159 51872 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KW-2478 KW-2478 76160 51873 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE IMATINIB IMATINIB 76161 51874 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL384304 RG-547 76164 51875 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Vemurafenib VEMURAFENIB 24265153,26137449 76167 51876 ATAD5 79915 NA DNDI1417941 CHEMBL2095095 76168 51877 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor AMUVATINIB AMUVATINIB 76169 51878 PHEX 5251 ENZYME, PROTEASE, DRUGGABLE GENOME RECOMBINANT HUMAN GROWTH HORMONE 9323282 76170 51879 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR NORGESTIMATE NORGESTIMATE 76172 51880 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 249565775 76173 51881 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TEGAFUR TEGAFUR 23988873 76174 51882 TSPO 706 DRUGGABLE GENOME TEMAZEPAM TEMAZEPAM 76178 51883 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650687 NALTREXONE 76179 51884 ATAD5 79915 NA DIPHENYLENEIODONIUM DIPHENYLENEIODONIUM 76183 51885 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1654 CHEMBL602776 76185 51886 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 223366050 SAPITINIB 76186 51887 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE TPCK TPCK 76187 51888 GAD1 2571 DRUGGABLE GENOME, ENZYME methadone METHADONE 31866536 76188 51889 TUBA1B 10376 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 76189 51890 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651432 ALDOSTERONE 76193 51891 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 D-64131 CHEMBL140220 76194 51892 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-MTC-434 76195 51893 ALDH1A1 216 DRUGGABLE GENOME, ENZYME AG-370 CHEMBL59150 76196 51894 CD58 965 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE interferon beta-1b 76199 51895 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE MYRICETIN MYRICETIN 22212721 76200 51896 PMEL 6490 DRUGGABLE GENOME IMCgp100 TEBENTAFUSP 23263452 76203 51897 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE MANNITOL MANNITOL 3142269 76204 51898 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Cevimeline CEVIMELINE 76205 51899 BAZ2B 29994 NA TERPYRIDINE TERPYRIDINE 76206 51900 SLC4A8 9498 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ethanol ALCOHOL 32451486 76208 51901 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Maleimides derivative 2 76211 51902 ALOX15B 247 DRUGGABLE GENOME, ENZYME QUERCETIN QUERCETIN 76212 51903 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME VITEXIN VITEXIN 76213 51904 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYCLOBENZAPRINE HYDROCHLORIDE CYCLOBENZAPRINE HYDROCHLORIDE 76217 51905 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE TAK-715 TAK-715 76218 51906 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME binimetinib BINIMETINIB 76221 51907 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR SILIBININ SILIBININ 21273068 76222 51908 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR anastrozole ANASTROZOLE 76225 51909 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CETUXIMAB CETUXIMAB 25520391 76226 51910 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE metformin METFORMIN 22722338 76227 51911 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LYCOBETAINE LYCOBETAINE 23266176 76228 51912 SULT2B1 6820 ENZYME, DRUGGABLE GENOME anthracyclines and related substances 23441093,21900104 76230 51913 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Imatinib IMATINIB 22328973,15928335,21224473,22718859,28514312,16357008,24132921,14645423,22323597,22745105 76231 51914 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE PEMBROLIZUMAB PEMBROLIZUMAB 30742119 76232 51915 GMNN 51053 DRUGGABLE GENOME TESMILIFENE TESMILIFENE 76233 51916 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR BAX-499 ARC-19499 76234 51917 ALOX5 240 DRUGGABLE GENOME, ENZYME inhibitor 178101859 76235 51918 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CISPLATIN CISPLATIN 23764753 76236 51919 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE ILORASERTIB ILORASERTIB 76237 51920 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 6,4'-DIMETHOXYFLAVONE 6,4'-DIMETHOXYFLAVONE 76240 51921 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BAY80-6946 COPANLISIB 76242 51922 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME 9-NITRO-ANTHRACENE CHEMBL166112 76243 51923 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME ENTRECTINIB ENTRECTINIB 76244 51924 PTGS1 5742 ENZYME, DRUGGABLE GENOME Flufenamic Acid 76246 51925 TSPO 706 DRUGGABLE GENOME PMID27599163-Compound-77 76247 51926 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 223366211 CRENOLANIB 76248 51927 HSPD1 3329 DRUGGABLE GENOME, ENZYME, CELL SURFACE DiaPep-277 DIAPEP-277 76250 51928 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR ANDROGENS 18635743 76252 51929 PIEZO1 9780 ION CHANNEL, TRANSPORTER activator 354702289 76253 51930 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLOZAPINE CLOZAPINE 17504220 76257 51931 MGAT4A 11320 DRUGGABLE GENOME capecitabine CAPECITABINE 26222057 76260 51932 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE QUINESTROL QUINESTROL 76261 51933 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE PENTOSTATIN PENTOSTATIN 76262 51934 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE leucovorin LEUCOVORIN 23314736 76263 51935 ANO1 55107 ION CHANNEL inhibitor 187051756 CROFELEMER 76264 51936 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102325 PAZOPANIB 76266 51937 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER INOSITOL INOSITOL 16733561 76270 51938 ITGB8 3696 DRUGGABLE GENOME, CELL SURFACE inhibitor 385612210 76273 51939 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyrrolo-pyrimidine derivative 9 76274 51940 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AM-404 CHEMBL39878 76275 51941 BCHE 590 DRUGGABLE GENOME, ENZYME PMID29757691-Compound-7 76276 51942 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 L-655240 CHEMBL362223 76278 51943 GAA 2548 DRUGGABLE GENOME, ENZYME EUPAFOLIN EUPAFOLIN 76279 51944 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE KINASE INHIBITOR 16880527 76281 51945 POLI 11201 DNA REPAIR SB-415286 CHEMBL322970 76283 51946 GSTT1 2952 DRUGGABLE GENOME thalidomide THALIDOMIDE 21435719 76285 51947 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LINTITRIPT LINTITRIPT 76286 51948 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER saquinavir SAQUINAVIR 76288 51949 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME N-(pyridin-2-yl)pyridine methylsulfone derivative 1 76289 51950 GMNN 51053 DRUGGABLE GENOME DNDI1417072 CHEMBL1310701 76290 51951 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR INDIUM CHLORIDE INDIUM CHLORIDE 76291 51952 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME AG-1288 CHEMBL166486 76292 51953 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Regorafenib REGORAFENIB 76293 51954 APC 324 CLINICALLY ACTIONABLE StAx-35 23071338 76296 51955 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor CHEMBL3545199 RG-7741 76298 51956 PDE4D 5144 DRUGGABLE GENOME, ENZYME SOTB07 76299 51957 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 4,4'-DIMETHOXYDALBERGIONE 4,4'-DIMETHOXYDALBERGIONE 76300 51958 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Indoline derivative 11 76301 51959 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CYC-116 CYC-116 76302 51960 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PYROGALLOL PYROGALLOL 76303 51961 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1201575 EFALIZUMAB 76306 51962 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME 681640 CHEMBL379975 76307 51963 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-124278 CHEMBL534423 76308 51964 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME DASATINIB DASATINIB 76309 51965 LOX 4015 ENZYME, DRUGGABLE GENOME inhibitor 385612245 76310 51966 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SJ000039423 CHEMBL589207 76311 51967 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LUPEOL LUPEOL 11754608 76312 51968 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE sorafenib SORAFENIB 23237922 76313 51969 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Niraparib NIRAPARIB 27717299,23810788 76314 51970 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR BN-GU-005-DHP 76315 51971 GMNN 51053 DRUGGABLE GENOME DNDI1383301 CHEMBL1509103 76317 51972 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME inhibitor 404859125 76319 51973 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE PMID25656651-Compound-21a 76322 51974 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000120449 CHEMBL609027 76324 51975 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 VESNARINONE VESNARINONE 9630823 76325 51976 CBX1 10951 NA AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 76326 51977 COMT 1312 DRUGGABLE GENOME, ENZYME etoposide catechol 76330 51978 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Curcumin analog 2 76335 51979 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200654 BENOXINATE HYDROCHLORIDE 76336 51980 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE SURAMIN SURAMIN 15833899 76337 51981 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME NIMUSTINE HYDROCHLORIDE 9537648 76338 51982 RAB9A 9367 ENZYME, DRUGGABLE GENOME HTS-05057 CHEMBL372629 76339 51983 DHFR 1719 DRUGGABLE GENOME, ENZYME TALOTREXIN TALOTREXIN 76340 51984 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200337 METOPROLOL SUCCINATE 76341 51985 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE PF-562271 PF-00562271 76344 51986 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-2272 CHEMBL601757 76345 51987 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE CHAULMOSULFONE CHAULMOSULFONE 76346 51988 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CHEMBL1743052 OPORTUZUMAB MONATOX 76347 51989 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR ACE INHIBITOR 14615289 76348 51990 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-123808 CHEMBL546493 76349 51991 RHBDF2 79651 ENZYME oxycodone OXYCODONE 21622719 76351 51992 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE TNF-ALPHA ADENOVECTOR 76352 51993 AQP4 361 ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME LAMOTRIGINE LAMOTRIGINE 18572411 76353 51994 CBX1 10951 NA FENOLDOPAM FENOLDOPAM 76354 51995 KDM4A 9682 DRUGGABLE GENOME, ENZYME BROXURIDINE BROXURIDINE 76356 51996 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 10 76360 51997 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE peginterferon alfa-2a 28703131 76361 51998 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME DOCETAXEL DOCETAXEL 76362 51999 POLI 11201 DNA REPAIR ISOTHYMONIN ISOTHYMONIN 76363 52000 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE VANDETANIB VANDETANIB 76364 52001 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHANANDAMIDE METHANANDAMIDE 76365 52002 UBA2 10054 DRUGGABLE GENOME, ENZYME 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 76366 52003 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CIMIRACEMATE A CIMIRACEMATE A 19835377 76367 52004 NPEPL1 79716 PROTEASE, ENZYME inhibitor CHEMBL2103847 TOSEDOSTAT 76369 52005 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME DIMETHYLSPINGOSINE DIMETHYLSPINGOSINE 19469544 76370 52006 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR T3D-959 DB959 76371 52007 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DIPHENIDOL DIPHENIDOL 76372 52008 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE HYPERBARIC OXYGEN 16001273,11236678 76374 52009 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR doxycycline DOXYCYCLINE 24185512 76375 52010 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 1096708-71-2 76376 52011 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-1211 CHEMBL600968 76381 52012 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 315661119 76382 52013 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR TROGLITAZONE TROGLITAZONE 15498850 76384 52014 HLA-DRA 3122 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE flucloxacillin FLOXACILLIN 30664875 76385 52015 RNF8 9025 KINASE, ENZYME trastuzumab TRASTUZUMAB 30071039 76386 52016 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME 4-(thiazol-5-yl)-pyrimidine derivative 1 76387 52017 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE CELECOXIB CELECOXIB 16917206 76389 52018 ESRRG 2104 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 135651472 DIETHYLSTILBESTROL 76390 52019 ACSS2 55902 ENZYME, TRANSCRIPTION FACTOR cisplatin CISPLATIN 21636554 76391 52020 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME eliglustat ELIGLUSTAT 20864621 76392 52021 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-123781 CHEMBL581194 76393 52022 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CL-976 CL-976 76394 52023 PIP 5304 DRUGGABLE GENOME TAMOXIFEN TAMOXIFEN 1930624 76396 52024 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C24 76397 52025 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 LAMOTRIGINE LAMOTRIGINE 22931300 76398 52026 MKNK1 8569 SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, ENZYME inhibitor 381118877 TOMIVOSERTIB 76399 52027 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME IODOACETAMIDE IODOACETAMIDE 76404 52028 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SJ000071821 CHEMBL589924 76405 52029 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME trifluridine TRIFLURIDINE 28992563 76407 52030 CTSL 1514 PROTEASE, DRUGGABLE GENOME, ENZYME PMID27998201-Compound-7 76408 52031 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR antagonist LCL161 LCL-161 76409 52032 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL580 LORAZEPAM 76410 52033 DIABLO 56616 NA HYDROGEN PEROXIDE 16085184,14987999 76411 52034 BAZ2B 29994 NA DEMECLOCYCLINE HYDROCHLORIDE DEMECLOCYCLINE HYDROCHLORIDE 76413 52035 LIMK2 3985 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 384403681 76414 52036 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FERROUS SULFATE FERROUS SULFATE 22931300 76415 52037 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 76416 52038 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1201486 QUINIDINE POLYGALACTURONATE 76417 52039 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE MARAVIROC MARAVIROC 76418 52040 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE BLU-285 AVAPRITINIB 76419 52041 PTGS2 5743 DRUGGABLE GENOME, ENZYME ASPIRIN ASPIRIN 17522398 76420 52042 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXIGLUTATIONE OXIGLUTATIONE 76422 52043 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SEROTONIN HYDROCHLORIDE SEROTONIN HYDROCHLORIDE 76423 52044 MAPT 4137 DRUGGABLE GENOME TDR77593 CHEMBL1510164 76424 52045 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Heterocyclic derivative 26 76425 52046 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SERMS 14553828 76426 52047 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE MECYSTEINE HYDROCHLORIDE MECYSTEINE HYDROCHLORIDE 76427 52048 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME EBSELEN EBSELEN 76428 52049 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR NSC-753574 CHEMBL2088730 22982122 76429 52050 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201167 CARVEDILOL PHOSPHATE 76430 52051 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 94381 CHEMBL374632 76431 52052 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME HINOKITIOL HINOKITIOL 76432 52053 PTGES 9536 DRUGGABLE GENOME, ENZYME MK-886 CHEMBL29097 19884011,24697244,25686392 76434 52054 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE OPB-51602 76438 52055 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Fulvestrant FULVESTRANT 76440 52056 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Dovitinib DOVITINIB 22238366,23658459,23443805,23908597,26036639 76441 52057 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 649849 CHEMBL405914 76443 52058 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ampicillin AMPICILLIN 9609616 76444 52059 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TCMDC-123869 CHEMBL546597 76445 52060 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1201891 DEFLAZACORT 76446 52061 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200774 FLUPREDNISOLONE 76447 52062 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIMETHENAMID DIMETHENAMID 76448 52063 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CUDC-907 FIMEPINOSTAT 22693356,19165201,19490892,20570890 76450 52064 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CABOZANTINIB CABOZANTINIB 76451 52065 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE EPICATECHIN GALLATE EPICATECHIN GALLATE 19839593 76452 52066 POLK 51426 DNA REPAIR, ENZYME MYRICETIN MYRICETIN 76453 52067 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE mFOLFOX6 27918764 76454 52068 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME 681640 CHEMBL379975 76455 52069 GMNN 51053 DRUGGABLE GENOME DNDI1417599 CHEMBL2094833 76456 52070 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE RECOMBINANT C5A 1683814 76457 52071 GAL 51083 DRUGGABLE GENOME antidepressants 76458 52072 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417260 CHEMBL2094573 76459 52073 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-39 76461 52074 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE CLOTRIMAZOLE CLOTRIMAZOLE 76462 52075 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME URSOLIC ACID URSOLIC ACID 19534471 76464 52076 CALR 811 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME RETINOID 9013706 76465 52077 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR UVB 16114492 76466 52078 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER RUBOXISTAURIN RUBOXISTAURIN 76471 52079 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME LUPRON LEUPROLIDE ACETATE 9433928 76476 52080 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor XL888 XL-888 76479 52081 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CARTEOLOL CARTEOLOL 76480 52082 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3039504 NINTEDANIB ESYLATE 76481 52083 PRPS1 5631 DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, ENZYME MERCAPTOPURINE MERCAPTOPURINE 25962120 76484 52084 NAT1 9 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200765 SIBUTRAMINE HYDROCHLORIDE 76485 52085 USP1 7398 DNA REPAIR, PROTEASE, ENZYME L-732138 L-732138 76486 52086 MAPT 4137 DRUGGABLE GENOME BILIRUBIN BILIRUBIN 76487 52087 SMN1 6606 DRUGGABLE GENOME 3',4'-DIHYDROXYFLAVONE CHEMBL222556 76489 52088 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor PANOBINOSTAT PANOBINOSTAT 76490 52089 CDH17 1015 TRANSPORTER, CELL SURFACE CISPLATIN CISPLATIN 10381631 76491 52090 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178103840 PHENELZINE 76492 52091 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 76493 52092 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody 178103465 PANITUMUMAB 76494 52093 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor 178102559 NINTEDANIB 76495 52094 DNER 92737 NA PMID26924192-Compound-50 76497 52095 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1201023 ORPHENADRINE HYDROCHLORIDE 76498 52096 TUBB4B 10383 DRUGGABLE GENOME Vinblastine VINBLASTINE 76499 52097 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR NIMODIPINE NIMODIPINE 23688559 76501 52098 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR PMID29671355-Compound-8 76502 52099 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL antagonist 135649822 76503 52100 KMO 8564 DRUGGABLE GENOME, ENZYME Isoxazoles and isoxazoline derivative 4 76504 52101 TSPO 706 DRUGGABLE GENOME FLUNITRAZEPAM FLUNITRAZEPAM 76505 52102 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Rituxan Immunology 76507 52103 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE gemcitabine GEMCITABINE 12477049,25162786,20665488,22705007,23230131 76508 52104 TUBB 203068 DRUGGABLE GENOME CHEMBL2304041 SAGOPILONE 76509 52105 POLI 11201 DNA REPAIR NSC-19063 CHEMBL1310138 76511 52106 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME inhibitor 178101459 76513 52107 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ETHACRYNIC ACID 10900222 76514 52108 TP53AIP1 63970 NA cyclophosphamide CYCLOPHOSPHAMIDE 76515 52109 CYB5R4 51167 DRUGGABLE GENOME isosorbide dinitrate 76516 52110 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE MMP INHIBITOR 15030579 76518 52111 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYCANTHONE HYCANTHONE 76519 52112 ESYT2 57488 NA methylphenidate METHYLPHENIDATE 29382897 76520 52113 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE Tivozanib TIVOZANIB 76521 52114 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE AZD-6765 LANICEMINE 76523 52115 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME ATORVASTATIN ATORVASTATIN 17192770 76524 52116 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CRIDANIMOD CRIDANIMOD 76525 52117 OGG1 4968 ENZYME inhibitor 381118894 76526 52118 ARG1 383 ENZYME selective beta-2-adrenoreceptor agonists 76527 52119 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ZOXAZOLAMINE ZOXAZOLAMINE 22931300 76528 52120 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102288 MOTESANIB 76530 52121 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ICI-118551 ICI-118551 2903243 76531 52122 TACSTD2 4070 NA N/A 76532 52123 PDE1A 5136 ENZYME, DRUGGABLE GENOME inhibitor 315661236 CRISABOROLE 76533 52124 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR RETINOL RETINOL 76536 52125 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FLAVOKAWAIN B FLAVOKAWAIN B 76537 52126 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME Diaryl amine derivative 3 76538 52127 HEXA 3073 DRUGGABLE GENOME, ENZYME PYRIMETHAMINE PYRIMETHAMINE 25984755,17237499 76539 52128 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135652667 ATROPINE 76540 52129 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 178103384 OFATUMUMAB 76541 52130 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Capecitabine CAPECITABINE 26920887 76542 52131 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL27759 ENTINOSTAT 76544 52132 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE SULFAMIDE SULFAMIDE 76545 52133 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NOVOBIOCIN NOVOBIOCIN 21129982,23859777 76547 52134 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME CPI-613 76548 52135 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME valbenazine VALBENAZINE 76549 52136 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE MOTESANIB MOTESANIB 76550 52137 SLC1A2 6506 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE inhibitor 178101349 76551 52138 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL agonist 178101004 DYSIHERBAINE 76552 52139 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE RITODRINE RITODRINE 76554 52140 NEK4 6787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SP-600125 SP-600125 76555 52141 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE MANOALIDE MANOALIDE 76559 52142 NDUFB7 4713 ENZYME inhibitor CHEMBL3545135 NV-128 76560 52143 TPM3 7170 KINASE, CLINICALLY ACTIONABLE 6-THIOGUANINE THIOGUANINE 7687657 76563 52144 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TRV027 76564 52145 MAOB 4129 DRUGGABLE GENOME, ENZYME PHENELZINE PHENELZINE 76565 52146 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME CEP-11981 CEP-11981 22148921 76566 52147 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Irinotecan IRINOTECAN 28783719,25714871 76567 52148 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE BERKELEYACETAL B BERKELEYACETAL B 17970594 76570 52149 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Carboplatin CARBOPLATIN 28514312 76571 52150 RTN4 57142 DRUGGABLE GENOME ANTISENSE OLIGONUCLEOTIDES 14574981 76572 52151 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE HOMOHARRINGTONINE OMACETAXINE MEPESUCCINATE 12744738 76573 52152 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME DEHYDROXYMETHYLEPOXYQUINOMICIN DEHYDROXYMETHYLEPOXYQUINOMICIN 18729348 76574 52153 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE GSK2849330 76576 52154 HMGCR 3156 ENZYME, DRUGGABLE GENOME PMID27537201-Compound-Figure15a 76577 52155 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-29 76578 52156 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME IRIGINOL HEXAACEATATE IRIGINOL HEXAACEATATE 76579 52157 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LIDOFLAZINE LIDOFLAZINE 76582 52158 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 4-(thiazol-5-yl)-pyrimidine derivative 2 76583 52159 BCL2L2 599 CLINICALLY ACTIONABLE, DRUGGABLE GENOME NAVITOCLAX, ABT-263 76584 52160 INPPL1 3636 KINASE, ENZYME, DRUGGABLE GENOME inhibitor 252827535 76585 52161 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 76586 52162 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR RX-0201 ARCHEXIN 76587 52163 PDE4B 5142 DRUGGABLE GENOME, ENZYME MK-0873 MK-0873 76588 52164 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Mutant ras vaccine 76590 52165 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Salicylic acid derivative 7 76591 52166 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102725 76592 52167 GMNN 51053 DRUGGABLE GENOME GNF-PF-1577 CHEMBL600315 76593 52168 CBX1 10951 NA CISPLATIN CISPLATIN 76594 52169 ATAD5 79915 NA ENOXIMONE ENOXIMONE 76595 52170 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR PROCARBAZINE PROCARBAZINE 10640980 76596 52171 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Asparaginase ASPARAGINASE 28151717 76598 52172 SIK3 23387 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565729 76599 52173 TUBB 203068 DRUGGABLE GENOME ABT-751 ABT-751 25468039 76600 52174 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR SB-203580 SB-203580 76601 52175 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRILOSTANE TRILOSTANE 76603 52176 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYLEPHEDRINE METHYLEPHEDRINE 76604 52177 PDE5A 8654 ENZYME, DRUGGABLE GENOME TADALAFIL TADALAFIL 76605 52178 DCN 1634 DRUGGABLE GENOME ASCORBIC ACID 7944410 76607 52179 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE activator CHEMBL3707226 DEFIBROTIDE SODIUM 76608 52180 LSS 4047 ENZYME, DRUGGABLE GENOME inhibitor 178103322 76610 52181 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PMID27551786-Compound-I 76611 52182 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME DNDI1417467 CHEMBL1997335 76612 52183 ATAD5 79915 NA LASSBIO-294 CHEMBL233194 76613 52184 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LY-518674 LY-518674 76614 52185 MAPT 4137 DRUGGABLE GENOME BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 76615 52186 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL1173055 RUCAPARIB 76619 52187 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 354702207 76622 52188 ALDH1A1 216 DRUGGABLE GENOME, ENZYME MMV396705 CHEMBL1594640 76623 52189 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TCMDC-125322 CHEMBL580324 76625 52190 TNFRSF11A 8792 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE aspirin ASPIRIN 26398624 76627 52191 IMPDH2 3615 DRUGGABLE GENOME, ENZYME inhibitor 178103437 76628 52192 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-125142 CHEMBL528791 76629 52193 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TAMOXIFEN TAMOXIFEN 24185510 76630 52194 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHOLESTEROL CHOLESTEROL 76631 52195 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 249565693 76632 52196 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AG-527 CHEMBL258767 76633 52197 POLK 51426 DNA REPAIR, ENZYME ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 76636 52198 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tacrine-caffeic acid hybrid derivative 1 76637 52199 OTOS 150677 DRUGGABLE GENOME cisplatin CISPLATIN 25410892,31666714 76639 52200 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR antagonist CHEMBL1276308 MIFEPRISTONE 76642 52201 KDM4A 9682 DRUGGABLE GENOME, ENZYME TCMDC-125221 CHEMBL546649 76643 52202 COMT 1312 DRUGGABLE GENOME, ENZYME benztropine BENZTROPINE 76645 52203 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201642 INSULIN ZINC SUSP PROMPT BEEF 76647 52204 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ZW25 76648 52205 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE E7449 2X-121 76649 52206 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE BEVACIZUMAB BEVACIZUMAB 26921265 76650 52207 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR PMID25980951-Compound-43 76651 52208 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOLONIUM CHLORIDE TOLONIUM CHLORIDE 76652 52209 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BAY80-6946 COPANLISIB 76653 52210 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME lovastatin LOVASTATIN 16103896,26020121,15616150,10601278 76654 52211 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR (E),(E)-2,4-DECACIENAL CHEMBL443949 76656 52212 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 381118857 76661 52213 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME CYC-116 CYC-116 76662 52214 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME BEZ235 DACTOLISIB 24251790 76664 52215 ALDH1A1 216 DRUGGABLE GENOME, ENZYME LUTEOLIN LUTEOLIN 76665 52216 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TRASTUZUMAB TRASTUZUMAB 76667 52217 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME ALPRAZOLAM ALPRAZOLAM 76668 52218 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor 178102667 76670 52219 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME EV-077-3201-2TBS 76671 52220 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 363894132 76672 52221 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 178101973 76673 52222 IL1B 3553 KINASE, DRUGGABLE GENOME CANAKINUMAB CANAKINUMAB 76676 52223 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE SPC-2996 76677 52224 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE SB-265610 76679 52225 CD44 960 DRUGGABLE GENOME, CELL SURFACE BIWA 4 76680 52226 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME JQ1 26552700 76682 52227 APOE 348 DRUGGABLE GENOME TROGLITAZONE TROGLITAZONE 15057551 76683 52228 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROPICONAZOLE PROPICONAZOLE 76684 52229 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 (S)-FELODIPINE (S)-FELODIPINE 76685 52230 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX MULBERROFURAN H MULBERROFURAN H 24901948 76686 52231 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 385612204 76687 52232 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Incadronate 76689 52233 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651783 76690 52234 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PF-562271 PF-00562271 76691 52235 MAPT 4137 DRUGGABLE GENOME CEFACLOR CEFACLOR 76692 52236 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Tafenoquine TAFENOQUINE 76693 52237 PSMC4 5704 NA BORTEZOMIB BORTEZOMIB 24524217 76694 52238 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE XL765 76695 52239 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Radiotherapy 26358474 76696 52240 MAPKAP1 79109 KINASE inhibitor MLN0128 SAPANISERTIB 76697 52241 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ETIDRONIC ACID ETIDRONIC ACID 22931300 76699 52242 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PROBENECID PROBENECID 9182837 76700 52243 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BUMETANIDE BUMETANIDE 76702 52244 GLS 2744 ENZYME GNF-PF-2755 CHEMBL600738 76703 52245 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL217092 SARACATINIB 76704 52246 PLD1 5337 ENZYME, DRUGGABLE GENOME inhibitor 252827440 76705 52247 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME BEVACIZUMAB BEVACIZUMAB 76706 52248 BCORL1 63035 CLINICALLY ACTIONABLE N/A 26879601 76707 52249 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE US8889696, 39 76709 52250 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 223365915 OCRELIZUMAB 76710 52251 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE LEE011 RIBOCICLIB 76711 52252 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE ILORASERTIB ILORASERTIB 76712 52253 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme9EHT3356 76713 52254 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL190 THEOPHYLLINE 76714 52255 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Anti-CD123-CAR-transduced T cells 76717 52256 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CLOPIDOGREL CLOPIDOGREL 76719 52257 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774822-Compound-Figure1Example20 76720 52258 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CEFOTAXIME SODIUM CEFOTAXIME SODIUM 76721 52259 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW831091X GW831091X 76722 52260 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DENATONIUM BENZOATE DENATONIUM BENZOATE 76723 52261 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-1678 CHEMBL580340 76724 52262 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135651044 76726 52263 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 363894210 PANULISIB 76727 52264 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME AS-605240 CHEMBL568150 76728 52265 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor MGCD265 GLESATINIB 76729 52266 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Everolimus EVEROLIMUS 26951309,23629727,27797976,20664174,20664172,27893038,21358673,22662154 76730 52267 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102284 MASITINIB 76732 52268 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME RITUXIMAB RITUXIMAB 76734 52269 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 385612189 76735 52270 HTT 3064 DRUGGABLE GENOME FLUSPIRILENE FLUSPIRILENE 76736 52271 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME N/A 76737 52272 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Tretinoin TRETINOIN 76738 52273 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME SJ000040829 CHEMBL589711 76739 52274 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor TOZASERTIB TOZASERTIB 19035792,23808327 76740 52275 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Flurbiprofen FLURBIPROFEN 76741 52276 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME DIPYRITHIONE DIPYRITHIONE 76743 52277 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME RABEPRAZOLE SODIUM RABEPRAZOLE SODIUM 76744 52278 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ARACHIDONOYL GLYCINE ARACHIDONOYL GLYCINE 76747 52279 MPHOSPH8 54737 NA DOCEBENONE DOCEBENONE 76748 52280 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE OK-432 1371977 76750 52281 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX PALBOCICLIB PALBOCICLIB 29236940,20473330,20354191 76751 52282 CCL18 6362 DRUGGABLE GENOME LD78 9233607 76752 52283 MAPT 4137 DRUGGABLE GENOME MECYSTEINE HYDROCHLORIDE MECYSTEINE HYDROCHLORIDE 76755 52284 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-1184 CHEMBL600347 76757 52285 BCHE 590 DRUGGABLE GENOME, ENZYME GALANTAMINE GALANTAMINE 23540646 76758 52286 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME GNF-PF-3148 CHEMBL81782 76759 52287 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 INDINAVIR INDINAVIR 22931300 76760 52288 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200604 TROPICAMIDE 76761 52289 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PD-160170 CHEMBL422942 76763 52290 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 223366033 76764 52291 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CHLORPHENIRAMINE CHLORPHENIRAMINE 76765 52292 ARG1 383 ENZYME inhibitor 252827464 76766 52293 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE VX-661 TEZACAFTOR 76767 52294 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL571 KETOPROFEN 76769 52295 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CYCLOSPORINE CYCLOSPORINE 9777701 76771 52296 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME LFB-R603 LFB-R603 76772 52297 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL15770 SULINDAC 76773 52298 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TKM-PLK1 76775 52299 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE sunitinib SUNITINIB 22015057,24013576 76777 52300 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-69187 CHEMBL19954 76778 52301 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME POTASSIUM DICHROMATE POTASSIUM DICHROMATE 76779 52302 XDH 7498 DRUGGABLE GENOME, ENZYME Fused heterocyclic compound 2 76780 52303 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Ergotidine 76782 52304 DNER 92737 NA PMID26924192-Compound-57 76783 52305 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE NINTEDANIB NINTEDANIB 76786 52306 GATA4 2626 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE NSC-126866 CHEMBL1684099 21310620 76787 52307 CXCL8 3576 DRUGGABLE GENOME COLCHICINE COLCHICINE 76789 52308 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR inhibitor CHEMBL2107872 DELCASERTIB 76790 52309 POLI 11201 DNA REPAIR TALAROFLAVONE TALAROFLAVONE 18178092 76792 52310 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR STIROFOS STIROFOS 76795 52311 CRBN 51185 ENZYME, DRUG RESISTANCE 387065604 AVADOMIDE 76797 52312 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME SOTRASTAURIN SOTRASTAURIN 76798 52313 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE inhibitor 381744994 LEROCICLIB 76799 52314 ALDH1A1 216 DRUGGABLE GENOME, ENZYME U-73122 CHEMBL1256678 76800 52315 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650470 76801 52316 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 249565723 PF-00477736 76803 52317 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL3545087 GSK159802 76806 52318 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Bisoprolol BISOPROLOL 76807 52319 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PROPRANOLOL PROPRANOLOL 22931300 76809 52320 GGCX 2677 DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 76810 52321 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 315661193 ARRY-382 76811 52322 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651743 76812 52323 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32l 76814 52324 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ETHACRIDINE LACTATE ETHACRIDINE LACTATE 76815 52325 SULT1E1 6783 ENZYME, DRUGGABLE GENOME acetaminophen ACETAMINOPHEN 23462933,26049587 76816 52326 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME ticlopidine TICLOPIDINE 17638512 76819 52327 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ALL-TRANS-RETINOIC ACID 11939262 76820 52328 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ERLOTINIB ERLOTINIB 76822 52329 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR SCLEROTIORIN SCLEROTIORIN 76825 52330 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Encorafenib ENCORAFENIB 27312529 76826 52331 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE ASP3026 ASP-3026 27009859,25749034,25421750 76829 52332 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL blocker,inhibitor 178100956 76832 52333 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BENZBROMARONE BENZBROMARONE 76834 52334 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE Miltefosine MILTEFOSINE 76835 52335 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3559672 RAUWOLFIA SERPENTINA 76837 52336 RACGAP1 29127 NA DAIDZEIN DAIDZEIN 76838 52337 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CLONAZEPAM CLONAZEPAM 76839 52338 NR6A1 2649 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ANTISERUM 15273870,12606326 76840 52339 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SHIKONIN SHIKONIN 76841 52340 TUBB2A 7280 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 76842 52341 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1201754 RUFINAMIDE 76843 52342 ARID1A 8289 CLINICALLY ACTIONABLE PEMBROLIZUMAB PEMBROLIZUMAB 29736026 76844 52343 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650849 PRAZOSIN 76846 52344 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-22 76849 52345 TMEM97 27346 NA Benzamide derivative 4 76850 52346 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102605 CHEMBL406375 76852 52347 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NSC-107022 CHEMBL1601846 76853 52348 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE 681640 CHEMBL379975 76854 52349 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178103083 LEPIRUDIN 76855 52350 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE celecoxib CELECOXIB 23778325 76856 52351 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CHEMBL1341 METHOXYFLURANE 76857 52352 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE PF-06438179 76858 52353 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING ISOLIQUIRITIGENIN ISOLIQUIRITIGENIN 21866899 76859 52354 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SPIRONOLACTONE SPIRONOLACTONE 76860 52355 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Indazole amide derivative 1 76861 52356 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BAICALEIN BAICALEIN 76862 52357 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROGABIDE PROGABIDE 76863 52358 GMNN 51053 DRUGGABLE GENOME TCMDC-125539 CHEMBL533388 76864 52359 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR US9714230, 12 76866 52360 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Pyrrolo[2,3-d]pyrimidine derivative 9 76867 52361 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 348353651 76868 52362 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER KINETIN RIBOSIDE KINETIN RIBOSIDE 76869 52363 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000147784 CHEMBL590186 76870 52364 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200803 SOLIFENACIN SUCCINATE 76872 52365 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE H-Gly-PMe-Glu-OH 76873 52366 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE ARQ092 26469692 76875 52367 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME VAPITADINE VAPITADINE 76876 52368 MAOA 4128 DRUGGABLE GENOME, ENZYME PHENELZINE PHENELZINE 76877 52369 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102579 76878 52370 KDM1A 23028 DRUGGABLE GENOME, ENZYME, CELL SURFACE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING PARNATE PARNATE 21382717 76879 52371 KDM1A 23028 DRUGGABLE GENOME, ENZYME, CELL SURFACE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING NAMOLINE NAMOLINE 24007511 76882 52372 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME inhibitor 135651043 SIBUTRAMINE 76883 52373 DGAT1 8694 ENZYME, DRUGGABLE GENOME inhibitor 223366159 76885 52374 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME Sorafenib SORAFENIB 21517818 76888 52375 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR 3,8'-BIAPIGENIN CHEMBL515252 76889 52376 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor GDC-0973 COBIMETINIB 76893 52377 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR INTERFERON ALPHA-2B 10522033 76894 52378 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Enoxaparin ENOXAPARIN 16686945 76895 52379 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE CID 663143 CHEMBL1342336 76896 52380 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor XL147 PILARALISIB 76897 52381 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME TRIFLUOPERAZINE TRIFLUOPERAZINE 76900 52382 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME HEREGULIN 10376522 76901 52383 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OXYPHENCYCLIMINE OXYPHENCYCLIMINE 76902 52384 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Penbutolol PENBUTOLOL 76903 52385 COL6A2 1292 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 76904 52386 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor MASITINIB MASITINIB 76905 52387 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000160630 CHEMBL591404 76906 52388 HTT 3064 DRUGGABLE GENOME HELIOMYCIN HELIOMYCIN 76908 52389 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SGT-53 76909 52390 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL THIOPENTAL THIOPENTAL 76910 52391 PDE3A 5139 ENZYME, DRUGGABLE GENOME AMRINONE INAMRINONE 76911 52392 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 5310655 CHEMBL408563 76914 52393 PSMB10 5699 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL371405 MARIZOMIB 76915 52394 ABCA5 23461 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME LIM-0705 QUERCETIN-3'-O-PHOSPHATE 76917 52395 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (-)-ROLIPRAM (-)-ROLIPRAM 76918 52396 KDM4A 9682 DRUGGABLE GENOME, ENZYME 1-(4-HYDROXYPHENYL)MALEIMIDE CHEMBL565893 76920 52397 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING HEXACHLOROPHENE HEXACHLOROPHENE 76921 52398 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL574737 UCN-01 76925 52399 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER DAUNORUBICIN DAUNORUBICIN 10655559 76927 52400 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrazolo[1,5-a]pyrimidine derivative 25 76928 52401 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 252827368 PEXIDARTINIB 76930 52402 RIPOR2 9750 NA rifampin RIFAMPIN 30720667 76931 52403 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MK-1308 76932 52404 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME SPIRONOLACTONE SPIRONOLACTONE 76933 52405 PLCG2 5336 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE, PHOSPHOLIPASE IBRUTINIB IBRUTINIB 24869598 76934 52406 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 3,5-DINITROCATECHOL (OR-486) 3,5-DINITROCATECHOL (OR-486) 76937 52407 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME PIRFENIDONE PIRFENIDONE 76940 52408 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR OLANZAPINE OLANZAPINE 76942 52409 GMNN 51053 DRUGGABLE GENOME DNDI1417309 CHEMBL1341830 76943 52410 NDUFA11 126328 ENZYME inhibitor CHEMBL3545135 NV-128 76944 52411 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NARATRIPTAN NARATRIPTAN 76945 52412 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME ABT-494 UPADACITINIB 76946 52413 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR IONIS-GCCRRX 76947 52414 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MK-1775 ADAVOSERTIB 28652249,24791855,27998224 76949 52415 TNFSF10 8743 DRUGGABLE GENOME SODIUM BUTYRATE 16096370 76950 52416 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME ETIDRONATE DISODIUM 3923787 76951 52417 CRBN 51185 ENZYME, DRUG RESISTANCE LENALIDOMIDE LENALIDOMIDE 23480694 76952 52418 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 2-(3,4-METHYLENEDIOXYPHENYL)BENZOTHIAZOLE CHEMBL201325 76953 52419 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 76955 52420 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE BAY 80-6946 76956 52421 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME HEXAMETHYLENE BISACETAMIDE 2211839 76958 52422 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GUGGULSTERONE GUGGULSTERONE 76959 52423 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE NVP-BEZ235 DACTOLISIB 76960 52424 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178103476 76962 52425 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE activator 135651442 76963 52426 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME cerivastatin CERIVASTATIN 15365880,11844864 76964 52427 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME MDX-1203 76966 52428 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE DNDI1417467 CHEMBL1997335 76969 52429 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102425 76970 52430 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL3545026 FAMITINIB 76971 52431 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME Erythropoietin-transfected autologous cell therapy 76972 52432 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR ZALCITABINE ZALCITABINE 76974 52433 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Pimasertib PIMASERTIB 23629727 76976 52434 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 10 76977 52435 DHODH 1723 DRUGGABLE GENOME, ENZYME inhibitor 363894154 VIDOFLUDIMUS 76978 52436 NEK4 6787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ILORASERTIB ILORASERTIB 76980 52437 SMN1 6606 DRUGGABLE GENOME TRICHOSTATIN TRICHOSTATIN 76981 52438 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL1201129 DECITABINE 76983 52439 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME HDM201 76985 52440 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER simvastatin SIMVASTATIN 19802823,16321621,19891551 76987 52441 MAPT 4137 DRUGGABLE GENOME HOMIDIUM HOMIDIUM 76988 52442 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CHLORANIL CHLORANIL 76989 52443 UGCG 7357 ENZYME, DRUGGABLE GENOME MIGLUSTAT MIGLUSTAT 76990 52444 GSTT1 2952 DRUGGABLE GENOME CISPLATINUM CISPLATIN 12851839 76991 52445 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE BEPRIDIL BEPRIDIL 76995 52446 IFNG 3458 DRUGGABLE GENOME AMG 811 76997 52447 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ICI-164384 CHEMBL1222035 20659801 76998 52448 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME BETRIXABAN BETRIXABAN 76999 52449 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE fluorouracil FLUOROURACIL 25545243,24533712,11160862,21479364,10208650,21946896,18511948 77001 52450 POLK 51426 DNA REPAIR, ENZYME MANUMYCIN A MANUMYCIN A 77002 52451 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL1742994 BRENTUXIMAB VEDOTIN 77003 52452 MAPKAP1 79109 KINASE inhibitor AZD8055 AZD-8055 77004 52453 KDM4A 9682 DRUGGABLE GENOME, ENZYME PHENELZINE SULFATE PHENELZINE SULFATE 77005 52454 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR inhibitor 315661286 ULIXERTINIB 77006 52455 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Ruxolitinib RUXOLITINIB 77008 52456 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NECROSTATIN NECROSTATIN 77009 52457 ACACA 31 ENZYME, DRUGGABLE GENOME inhibitor 178101963 77010 52458 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE ALLOXAN ALLOXAN 77011 52459 CBLB 868 CLINICALLY ACTIONABLE, ENZYME Fluorouracil FLUOROURACIL 24351824 77012 52460 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 77014 52461 HSPA4 3308 NA CELECOXIB CELECOXIB 16646082 77015 52462 MBP 4155 CELL SURFACE ATX-MS-1467 77016 52463 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME paclitaxel PACLITAXEL 21151855 77017 52464 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Salbutamol ALBUTEROL 77018 52465 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE interferons 21159314 77019 52466 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor DASATINIB DASATINIB 77022 52467 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AMOROLFINE AMOROLFINE 77023 52468 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PROADIFEN PROADIFEN 77024 52469 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME QUESTIOMYCIN B QUESTIOMYCIN B 77025 52470 NDUFB4 4710 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 77026 52471 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR TOZASERTIB TOZASERTIB 77027 52472 RBX1 9978 DNA REPAIR, ENZYME inhibitor CHEMBL848 LENALIDOMIDE 77030 52473 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1096 AMLEXANOX 77031 52474 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SOTALOL SOTALOL 77032 52475 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE agonist 178100369 77033 52476 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR 7-azaindole derivative 3 77038 52477 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor 178104000 MOCLOBEMIDE 77039 52478 PDE4A 5141 DRUGGABLE GENOME, ENZYME DG071 77041 52479 TUBB 203068 DRUGGABLE GENOME Batabulin BATABULIN 77042 52480 PTGES 9536 DRUGGABLE GENOME, ENZYME PMID28627961-Compound-41 77043 52481 STAT1 6772 DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR, KINASE CISPLATIN CISPLATIN 15726096 77044 52482 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-36 77045 52483 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DOCETAXEL DOCETAXEL 30452336,22149875,25693012 77046 52484 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME METHYSERGIDE MALEATE 77048 52485 SLPI 6590 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR TNF-ALPHA 12668158,17114478 77049 52486 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR US9073931, E1 77050 52487 UQCR10 29796 NA FAMOXADONE FAMOXADONE 10843216 77051 52488 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor BMS-599626 AC-480 77052 52489 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE BEPRIDIL BEPRIDIL 77054 52490 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135650665 77056 52491 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor DS-3078A DS-3078A 77057 52492 HTT 3064 DRUGGABLE GENOME SHAPE 77058 52493 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR TAE-684 TAE-684 77059 52494 POLK 51426 DNA REPAIR, ENZYME FLAVANONE FLAVANONE 77061 52495 CA2 760 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL18 ETHOXZOLAMIDE 77062 52496 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE NINTEDANIB NINTEDANIB 77063 52497 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor DASATINIB DASATINIB 77064 52498 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TAMARIXETIN TAMARIXETIN 25190466 77066 52499 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme14BINDY 77067 52500 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL ISONIPECOTIC ACID ISONIPECOTIC ACID 25038482 77069 52501 ATXN2 6311 NA STREPTONIGRIN STREPTONIGRIN 77071 52502 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-353720 CHEMBL1408276 77072 52503 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor 252166602 NANATINOSTAT 77074 52504 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Curcumin CURCUMIN 77076 52505 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR TAMOXIFEN TAMOXIFEN 77078 52506 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 METHOXSALEN METHOXSALEN 77079 52507 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 926663 CHEMBL265686 77080 52508 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 2-ENE-VALPROATE CHEMBL117487 17566732 77081 52509 PDE4B 5142 DRUGGABLE GENOME, ENZYME GPD-1116 77082 52510 COMT 1312 DRUGGABLE GENOME, ENZYME inhibitor 310264766 OPICAPONE 77086 52511 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Sorafenib SORAFENIB 20538618,23629727,16880785,23792568,22394203,24885690,27388325 77089 52512 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DESMOPRESSIN DESMOPRESSIN 24874785 77091 52513 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-WO2013082253 33 77092 52514 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE 1,3-BIS(3-NITROPHENYL)UREA CHEMBL1443422 77093 52515 PSMA3 5684 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL325041 BORTEZOMIB 77097 52516 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BENZOTHIAZYL DISULFIDE BENZOTHIAZYL DISULFIDE 77098 52517 CBR3 874 ENZYME, DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, CLINICALLY ACTIONABLE doxorubicin DOXORUBICIN 20007405,21048526,18551042 77099 52518 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME CORTISONE CORTISONE 3503494 77100 52519 MAPT 4137 DRUGGABLE GENOME SULFURETIN SULFURETIN 77102 52520 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor ONARTUZUMAB ONARTUZUMAB 77103 52521 MAOB 4129 DRUGGABLE GENOME, ENZYME Flavanone FLAVANONE 77104 52522 PRMT5 10419 ENZYME, METHYL TRANSFERASE GSK3326595 77105 52523 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-27 77108 52524 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE SP-600125 SP-600125 77109 52525 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-28 77110 52526 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor PF-00562271 PF-00562271 77112 52527 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Cariprazine CARIPRAZINE 77113 52528 ATAD5 79915 NA GNF-PF-4012 CHEMBL584269 77114 52529 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZEARALENONE ZEARALENONE 77116 52530 POLK 51426 DNA REPAIR, ENZYME GARCINONE E GARCINONE E 77119 52531 PDE4A 5141 DRUGGABLE GENOME, ENZYME OX-914 HT-0712 77120 52532 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR ALD518 CLAZAKIZUMAB 77121 52533 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE HYDROQUINONE HYDROQUINONE 10393963 77122 52534 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DILAZEP DILAZEP 77123 52535 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 252166577 PRACINOSTAT 77124 52536 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL3301595 DASOTRALINE 77125 52537 SMN1 6606 DRUGGABLE GENOME DNDI1416988 CHEMBL1389794 77126 52538 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pacritinib PACRITINIB 77128 52539 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Bicyclic heteroaryl benzamide derivative 5 77129 52540 TSPO 706 DRUGGABLE GENOME Quinazoline derivative 7 77131 52541 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist 53801069 PROCATEROL 77132 52542 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TCMDC-124518 CHEMBL527584 77133 52543 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 310264733 FIMEPINOSTAT 77135 52544 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENACYL CHLORIDE PHENACYL CHLORIDE 77136 52545 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MICHLER'S KETONE MICHLER'S KETONE 77137 52546 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BIMATOPROST BIMATOPROST 77138 52547 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE NI-101 24353405 77139 52548 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor PALBOCICLIB PALBOCICLIB 77141 52549 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 178103458 VORINOSTAT 77142 52550 MAOB 4129 DRUGGABLE GENOME, ENZYME Schiff base compound 1 77144 52551 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650514 77145 52552 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE vitamin b-complex, plain 22926161 77146 52553 RAB5A 5868 NA HGF 16423831 77147 52554 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME fenofibrate FENOFIBRATE 77148 52555 NOS1 4842 DRUGGABLE GENOME, ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 77149 52556 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-125606 CHEMBL536166 77151 52557 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME ESTRAMUSTINE ESTRAMUSTINE 11391599 77152 52558 ALDH1A1 216 DRUGGABLE GENOME, ENZYME P-HYDROXYCINNAMALDEHYDE P-HYDROXYCINNAMALDEHYDE 77154 52559 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME nevirapine NEVIRAPINE 77157 52560 ERAP1 51752 PROTEASE, ENZYME, DRUGGABLE GENOME SCOPOLETIN SCOPOLETIN 77158 52561 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Aphanin 27333990 77159 52562 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-2950 CHEMBL602807 77160 52563 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME ALVOCIDIB ALVOCIDIB 18469809,23301767 77164 52564 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLOBAZAM CLOBAZAM 77167 52565 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2017974 BUPARLISIB 77168 52566 KDM4A 9682 DRUGGABLE GENOME, ENZYME SERTACONAZOLE NITRATE SERTACONAZOLE NITRATE 77169 52567 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME R-1487 R-1487 77170 52568 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MEGESTROL ACETATE 77171 52569 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor BYL719 ALPELISIB 77172 52570 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ENCLOMIPHENE CITRATE ENCLOMIPHENE CITRATE 77173 52571 SLC29A4 222962 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 135650171 DESIPRAMINE 77177 52572 GAL 51083 DRUGGABLE GENOME benzodiazepine derivatives 77178 52573 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME VX-11e 25370473,27974663 77179 52574 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Dihydropyrido phthalazinone derivative 1 77180 52575 ATXN1L 342371 DRUG RESISTANCE DABRAFENIB DABRAFENIB 28178529 77181 52576 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE ALSTERPAULLONE ALSTERPAULLONE 77183 52577 PDE3A 5139 ENZYME, DRUGGABLE GENOME ENOXIMONE ENOXIMONE 77184 52578 MAP3K2 10746 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565786 77185 52579 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ETONOGESTREL ETONOGESTREL 77186 52580 CP 1356 DRUGGABLE GENOME, ENZYME BSO 8619904 77188 52581 POLK 51426 DNA REPAIR, ENZYME ALAZANINE ALAZANINE 77190 52582 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 348353625 77191 52583 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME NAPHTHOQUINONE NAPHTHOQUINONE 77192 52584 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME BAS-0338868 CHEMBL378903 77194 52585 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MITONAFIDE MITONAFIDE 77195 52586 PSMC4 5704 NA inhibitor CHEMBL451887 CARFILZOMIB 77196 52587 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GO-6976 GO-6976 77197 52588 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METHOXAMINE METHOXAMINE 77198 52589 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME GW441756X GW441756X 77201 52590 TSPO 706 DRUGGABLE GENOME PYRAZOLE PYRAZOLE 15544788 77203 52591 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE SPC5001 77204 52592 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SULFAQUINOXALINE SULFAQUINOXALINE 77205 52593 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Pegmusirudin PEGMUSIRUDIN 77206 52594 PTPN4 5775 PROTEIN PHOSPHATASE, DRUGGABLE GENOME ALENDRONATE ALENDRONIC ACID 77207 52595 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE BENZO[E]PYRENE BENZO[E]PYRENE 77209 52596 BRCA2 675 CLINICALLY ACTIONABLE TEMOZOLOMIDE TEMOZOLOMIDE 32043779 77210 52597 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 178104006 BUDESONIDE 77211 52598 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor VEMURAFENIB VEMURAFENIB 77212 52599 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME DOCETAXEL DOCETAXEL 25670080 77214 52600 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-INT767 77215 52601 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME FLT3 LIGAND 8916965 77216 52602 SCNN1G 6340 ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE TRIAMTERENE TRIAMTERENE 77217 52603 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE BAY-613606 CHEMBL541400 77218 52604 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME HYCANTHONE HYCANTHONE 9609323 77219 52605 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 WARFARIN WARFARIN 15050794 77220 52606 PSMA1 5682 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 77221 52607 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1318477 CHEMBL428064 77222 52608 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GW2016 12467226 77223 52609 KDM4A 9682 DRUGGABLE GENOME, ENZYME PHENANTHROLINE PHENANTHROLINE 77224 52610 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AMOXICILLIN AMOXICILLIN 77225 52611 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL181954 NAVEGLITAZAR 77227 52612 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TCMDC-123951 CHEMBL587849 77229 52613 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3301606 SOLCITINIB 77230 52614 ALOX15 246 ENZYME, DRUGGABLE GENOME TRICETIN TRICETIN 77232 52615 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Olaparib OLAPARIB 77234 52616 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1522 ESZOPICLONE 77238 52617 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 328083470 77240 52618 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE MOFEBUTAZONE MOFEBUTAZONE 77241 52619 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BKM120 BUPARLISIB 77242 52620 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME GW441756X GW441756X 77243 52621 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL856 PRIMIDONE 77244 52622 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2014129431Example8-1 77245 52623 PSMD1 5707 NA inhibitor CHEMBL451887 CARFILZOMIB 77246 52624 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE E5555 ATOPAXAR 77248 52625 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIMETHYL-OCTADECYL-AMMONIUM CHLORIDE TRIMETHYL-OCTADECYL-AMMONIUM CHLORIDE 77249 52626 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL agonist 178101048 77250 52627 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME activator CHEMBL266510 FLINDOKALNER 77251 52628 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 INAMRINONE INAMRINONE 77254 52629 ALDH1A1 216 DRUGGABLE GENOME, ENZYME WAY-100135 CHEMBL38288 77255 52630 POLD1 5424 DNA DIRECTED RNA POLYMERASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME inhibitor CHEMBL1096882 FLUDARABINE PHOSPHATE 77257 52631 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PF-04691502 PF-04691502 21750219 77258 52632 MAP3K10 4294 SERINE THREONINE KINASE, ENZYME, KINASE, DRUGGABLE GENOME inhibitor CHEMBL290352 CEP-1347 77259 52633 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DNDI1417995 CHEMBL1439833 77260 52634 TSPO 706 DRUGGABLE GENOME Imidazopyridine acetamide analog 3 77261 52635 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-4300 CHEMBL585656 77262 52636 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PERBROMOBENZENE PERBROMOBENZENE 77263 52637 ALOX5 240 DRUGGABLE GENOME, ENZYME 6BIO 6BIO 24697244 77266 52638 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIPHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER DIPHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER 77268 52639 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor BYL719 ALPELISIB 77270 52640 TUBB2A 7280 DRUGGABLE GENOME CYCLOSTREPTIN CYCLOSTREPTIN 17206139 77273 52641 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHYLPARABEN METHYLPARABEN 77274 52642 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE SB-204741 CHEMBL323356 77275 52643 BCHE 590 DRUGGABLE GENOME, ENZYME inhibitor 178103214 BAMBUTEROL 77276 52644 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BROMOCRIPTINE BROMOCRIPTINE 77277 52645 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE antagonist CHEMBL3039531 DANIRIXIN 77278 52646 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME SRT-2183 CHEMBL403308 18046409 77279 52647 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BTCP CHEMBL279556 77281 52648 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEPHALOTHIN CEPHALOTHIN 77282 52649 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME PSN602 77283 52650 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 77286 52651 THOP1 7064 DRUGGABLE GENOME, PROTEASE Nemonoxacin NEMONOXACIN 77287 52652 PDE4A 5141 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL628 PENTOXIFYLLINE 77288 52653 ERRFI1 54206 CLINICALLY ACTIONABLE EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR 23935914 77290 52654 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antibody MEDI-575 TOVETUMAB 77291 52655 CHKA 1119 ENZYME, KINASE DEXAMETHASONE DEXAMETHASONE 10077342 77292 52656 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DACARBAZINE DACARBAZINE 22931300 77293 52657 MPHOSPH8 54737 NA INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 77295 52658 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000154295 CHEMBL578502 77298 52659 PSMD3 5709 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 77301 52660 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Niraparib NIRAPARIB 28148839 77302 52661 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME NITROXOLINE NITROXOLINE 77303 52662 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME SJ000044417 CHEMBL609438 77304 52663 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Trametinib TRAMETINIB 27338794 77305 52664 MAPT 4137 DRUGGABLE GENOME SJ000044511 CHEMBL592124 77307 52665 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor MASITINIB MASITINIB 77308 52666 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-1339 CHEMBL600353 77309 52667 SPECC1L 23384 NA methotrexate METHOTREXATE 18539621 77310 52668 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME PMID26924192-Compound-105 77313 52669 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE US9040714, 7 77314 52670 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR inhibitor 249565595 LCL-161 77315 52671 GLRA2 2742 DRUGGABLE GENOME, ION CHANNEL HU-210 DEXANABINOL 20346682 77316 52672 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DICLAZURIL DICLAZURIL 77317 52673 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AST-487 AST-487 77319 52674 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 328083506 77320 52675 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051811 77321 52676 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3184679 AZD-4547 77322 52677 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BITHIONOL BITHIONOL 77323 52678 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 L-741626 CHEMBL445102 77324 52679 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BCMA CART 77326 52680 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CUCURBITACIN B CUCURBITACIN B 17190463 77330 52681 ATXN2 6311 NA PAROXETINE HYDROCHLORIDE PAROXETINE HYDROCHLORIDE 77335 52682 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL2105759 BARICITINIB 77336 52683 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL celecoxib CELECOXIB 22336956 77337 52684 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL448 PENTOBARBITAL 77338 52685 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME MYRICETIN MYRICETIN 77339 52686 HTT 3064 DRUGGABLE GENOME MIBEFRADIL DIHYDROCHLORIDE MIBEFRADIL DIHYDROCHLORIDE 77340 52687 PDE7A 5150 ENZYME, DRUGGABLE GENOME inhibitor 315661236 CRISABOROLE 77343 52688 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 135650002 77344 52689 PROCR 10544 DRUGGABLE GENOME, CELL SURFACE GED-APC 77345 52690 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ACID BLUE 129 ACID BLUE 129 77346 52691 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE ERLOTINIB ERLOTINIB 77348 52692 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE TRAMETINIB TRAMETINIB 25952648 77349 52693 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME DOVITINIB DOVITINIB 77351 52694 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME TRIAMCINOLONE TRIAMCINOLONE 12123742 77352 52695 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1095292 BRETYLIUM TOSYLATE 77353 52696 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME cisplatin CISPLATIN 19434073,22188361,29662106,22026922,21449681 77354 52697 NDUFA4L2 56901 NA inhibitor CHEMBL3545320 ME-344 77355 52698 POLB 5423 DNA REPAIR, DRUGGABLE GENOME HYDROXYSTILBAMIDINE ISETHIONATE HYDROXYSTILBAMIDINE ISETHIONATE 77359 52699 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME PMID26560530-Compound-12 77360 52700 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME MILNACIPRAN MILNACIPRAN 77361 52701 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME GSK-269962A GSK-269962A 77362 52702 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PRECLINICAL 22238366,21367659,18552176,23002168,25157968 77363 52703 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME URSOLIC ACID URSOLIC ACID 19534471 77365 52704 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL lamotrigine LAMOTRIGINE 23859570,21747585,28753467,25155934 77366 52705 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DESOGESTREL DESOGESTREL 77367 52706 POLK 51426 DNA REPAIR, ENZYME INDOCYANINE GREEN SODIUM INDOCYANINE GREEN 77368 52707 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OXYMETHOLONE OXYMETHOLONE 77369 52708 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE CRYPTOTANSHINONE CRYPTOTANSHINONE 23957426 77370 52709 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE inhibitor 252827447 CHRYSIN 77371 52710 ALOX5 240 DRUGGABLE GENOME, ENZYME METHOTREXATE METHOTREXATE 8151588 77372 52711 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL2364607 COBIMETINIB FUMARATE 77374 52712 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ABIRATERONE ABIRATERONE 25184630 77376 52713 HDAC11 79885 DRUGGABLE GENOME, ENZYME BUTYRYLHYDROXAMIC ACID BUTYRYLHYDROXAMIC ACID 21874153 77377 52714 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-92207 CHEMBL139935 77378 52715 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR E319 E319 77379 52716 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3545196 PD-0166285 77380 52717 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-402538 CHEMBL121556 77381 52718 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE EGFR CART 77382 52719 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TANSHINONE IIA TANSHINONE IIA 77384 52720 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ARQ-197 TIVANTINIB 77386 52721 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102317 CHEMBL1908396 77387 52722 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL METHYLPHENOBARBITAL MEPHOBARBITAL 77388 52723 IL1B 3553 KINASE, DRUGGABLE GENOME antipsychotics 25560300 77389 52724 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ROCILETINIB ROCILETINIB 24065731,28202511,25923550 77390 52725 MAP3K5 4217 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, ENZYME inhibitor 315661125 SELONSERTIB 77391 52726 HTT 3064 DRUGGABLE GENOME Valproate 77392 52727 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DICLOFENAC SODIUM DICLOFENAC SODIUM 77395 52728 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102667 77396 52729 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE carboplatin CARBOPLATIN 31616045 77397 52730 SMN1 6606 DRUGGABLE GENOME HYDRALAZINE HYDROCHLORIDE HYDRALAZINE HYDROCHLORIDE 77398 52731 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BISOPROLOL BISOPROLOL 77401 52732 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PLX4720 PLX-4720 23533272,31937621,23845441 77402 52733 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER METHOTREXATE METHOTREXATE 12036927 77403 52734 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor CHEMBL3545378 MK-6592 77404 52735 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32s 77405 52736 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER doxorubicin DOXORUBICIN 19696793 77406 52737 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ponatinib PONATINIB 77407 52738 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR ESTRADIOL ESTRADIOL 77408 52739 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE sulfanilamide SULFANILAMIDE 10793824 77409 52740 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME ASTERRIC ACID ASTERRIC ACID 77410 52741 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR BISINDOLYLMALEIMIDE IX BISINDOLYLMALEIMIDE IX 20030343,17149860 77412 52742 ITGA1 3672 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE SAN-300 SAN-300 77417 52743 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE SUNITINIB SUNITINIB 77418 52744 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME S-(4-CHLOROBENZYL)ISOTHIOUREA HCL CHEMBL1224312 20688518 77419 52745 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AC-480 AC-480 19821562 77420 52746 TXNRD2 10587 DRUGGABLE GENOME ARSENIC TRIOXIDE ARSENIC TRIOXIDE 17640917 77421 52747 PSMB10 5699 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL451887 CARFILZOMIB 77426 52748 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER A-77636 CHEMBL291143 77427 52749 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL14762 SELICICLIB 77429 52750 TSPO 706 DRUGGABLE GENOME Quinoline carboxamide derivative 5 77430 52751 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TVB-2640 24900571 77435 52752 TSPAN5 10098 CELL SURFACE escitalopram ESCITALOPRAM 26903268 77437 52753 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MSC2156119 77438 52754 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME tacrolimus TACROLIMUS 77439 52755 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ALPHA-TERTHIENYL ALPHA-TERTHIENYL 77440 52756 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NIFEDIPINE NIFEDIPINE 77441 52757 ATXN2 6311 NA OLEOYL DOPAMINE OLEOYL DOPAMINE 77442 52758 IGFBP1 3484 DRUGGABLE GENOME PROTEIN SYNTHESIS INHIBITOR 7688368 77443 52759 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME ALTISSIMACOUMARIN E ALTISSIMACOUMARIN E 22799262 77444 52760 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR LY-294002 LY-294002 77445 52761 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor PANOBINOSTAT PANOBINOSTAT 77446 52762 PLA2G10 8399 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME VARESPLADIB VARESPLADIB 77447 52763 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHENOLONE ENANTHATE METHENOLONE ENANTHATE 77448 52764 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME LUTEOLIN LUTEOLIN 77450 52765 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417099 CHEMBL1565444 77453 52766 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 178100439 GEMFIBROZIL 77454 52767 POLK 51426 DNA REPAIR, ENZYME OXIDOPAMINE OXIDOPAMINE 77455 52768 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE DIMETHYLADENINE DIMETHYLADENINE 77458 52769 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR CAPTAN CAPTAN 77459 52770 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2010077680 811 77462 52771 CX3CL1 6376 CELL SURFACE, DRUGGABLE GENOME ATEZOLIZUMAB ATEZOLIZUMAB 25428504 77463 52772 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE cyclophosphamide CYCLOPHOSPHAMIDE 26521987 77465 52773 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Entinostat ENTINOSTAT 77467 52774 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME AZELASTINE AZELASTINE 21381763 77468 52775 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051805 QUISINOSTAT 77469 52776 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW801372X GW801372X 77471 52777 IMPDH1 3614 ENZYME, DRUGGABLE GENOME inhibitor 178103437 77472 52778 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DNDI1417346 CHEMBL1490332 77474 52779 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor NIRAPARIB NIRAPARIB 77476 52780 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 252166751 77477 52781 MPHOSPH8 54737 NA QUERCETIN QUERCETIN 77479 52782 PMEL 6490 DRUGGABLE GENOME Gp100:209-217(210M) peptide vaccine 77480 52783 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 2-ACETYLPYRIDINE N4(ETHYL)THIOSEMICARBAZONE CHEMBL507986 21391686 77482 52784 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178103585 ROMIDEPSIN 77484 52785 MPHOSPH8 54737 NA TYRPHOSTIN A9 TYRPHOSTIN A9 77485 52786 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ALITRETIONINE 77486 52787 GABBR2 9568 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL701 BACLOFEN 77487 52788 DLG5 9231 KINASE fluorouracil FLUOROURACIL 77490 52789 NPR3 4883 DRUGGABLE GENOME 178101546 77491 52790 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-9 77493 52791 CXCL8 3576 DRUGGABLE GENOME PAMIDRONATE PAMIDRONIC ACID 12006522 77495 52792 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR 3R14S-OCHRATOXIN A 3R14S-OCHRATOXIN A 77496 52793 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE eribulin ERIBULIN 77497 52794 ATXN2 6311 NA CARMINIC ACID CARMINIC ACID 77499 52795 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 7,8-DIHYDROXYFLAVONE 7,8-DIHYDROXYFLAVONE 77501 52796 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL2138601 REFAMETINIB 77502 52797 PLK2 10769 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE WORTMANNIN WORTMANNIN 17135248 77503 52798 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR METHYL PARATHIONE METHYL PARATHIONE 77506 52799 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32c 77507 52800 ADK 132 DRUGGABLE GENOME, ENZYME, KINASE inhibitor 178101822 77508 52801 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR SORBINIL SORBINIL 24819954 77513 52802 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417165 CHEMBL1406948 77514 52803 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OXYCARBOXIN OXYCARBOXIN 77515 52804 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME agonist 135651881 77517 52805 SMN2 6607 DRUGGABLE GENOME CID 650707 CHEMBL408653 77518 52806 TUBB4B 10383 DRUGGABLE GENOME inhibitor CHEMBL428647 PACLITAXEL 77519 52807 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BITHIONOL BITHIONOL 77520 52808 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 77521 52809 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Oxaliplatin OXALIPLATIN 28784859,26432108,24300914 77524 52810 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DEQUALINIUM CHLORIDE DEQUALINIUM CHLORIDE 77525 52811 TSPO 706 DRUGGABLE GENOME Indole-based analog 5 77526 52812 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME BROMAZEPAM BROMAZEPAM 77528 52813 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME antagonist 252166531 NAVITOCLAX 77529 52814 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1162 NORETHINDRONE 77530 52815 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor GDC-0973 COBIMETINIB 77532 52816 SMN2 6607 DRUGGABLE GENOME 2-METHOXYPHENAZINE CHEMBL1420181 77533 52817 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DEXAMETHASONE DEXAMETHASONE 77534 52818 NOS1 4842 DRUGGABLE GENOME, ENZYME NXN-188 77535 52819 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 13 77537 52820 ATP5F1D 513 TRANSPORTER ENFLURANE ENFLURANE 77538 52821 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME FOLIC ACID FOLIC ACID 25234128 77539 52822 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL SECOBARBITAL SECOBARBITAL 77540 52823 EMP2 2013 CELL SURFACE HORMONES 18400107 77541 52824 POLI 11201 DNA REPAIR DIOTYROSINE DIOTYROSINE 77542 52825 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Liothyronine LIOTHYRONINE 77543 52826 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor BAY1000394 77544 52827 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 4 77545 52828 MPHOSPH8 54737 NA TREQUINSIN HYDROCHLORIDE TREQUINSIN HYDROCHLORIDE 77546 52829 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR FLUOCINOLONE ACETONIDE 77547 52830 TRPC4 7223 ION CHANNEL, KINASE, DRUGGABLE GENOME, CELL SURFACE blocker 178101072 77548 52831 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE benzodiazepine derivatives 77550 52832 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 178100873 77551 52833 POLK 51426 DNA REPAIR, ENZYME LAVENDUSTIN C LAVENDUSTIN C 77553 52834 TUBA1C 84790 DRUGGABLE GENOME ZAMPANOLIDE ZAMPANOLIDE 19877653 77555 52835 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE CEFTRIAXONE CEFTRIAXONE 22166395 77557 52836 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME LEUCOVORIN LEUCOVORIN 31871216 77558 52837 TUBA3D 113457 DRUGGABLE GENOME CURCUMIN CURCUMIN 23830698 77559 52838 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Imidazo[4,5-c]pyridine derivative 2 77561 52839 CDC42BPA 8476 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME PHA-767491 CHEMBL225519 77563 52840 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ETHACRYNIC ACID ETHACRYNIC ACID 77564 52841 TSPO 706 DRUGGABLE GENOME CHLORMEZANONE CHLORMEZANONE 77565 52842 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650055 CARBACHOL 77566 52843 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME 3,4,5,6-TETRACHLORO-[1,2]BENZOQUINONE CHEMBL364729 77568 52844 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-228155 CHEMBL505670 77569 52845 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME Flunarizine FLUNARIZINE 77570 52846 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist CHEMBL1201101 TESTOSTERONE CYPIONATE 77571 52847 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL3545025 INSM-18 77572 52848 TNFAIP1 7126 NA IL-2 ALDESLEUKIN 9357823 77573 52849 ALOX15 246 ENZYME, DRUGGABLE GENOME 3,3',5,5'-TETRABROMOBISPHENOL A CHEMBL184450 77575 52850 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Taselisib TASELISIB 77576 52851 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PI-88/Taxotere 77577 52852 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FLUTAMIDE FLUTAMIDE 77579 52853 FKBP1A 2280 DRUGGABLE GENOME, ENZYME, KINASE GPI-1485 GPI-1485 77580 52854 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DIGITOXIN DIGITOXIN 77581 52855 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TUBERCIDIN TUBERCIDIN 77583 52856 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR BAY-613606 CHEMBL541400 77584 52857 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 77585 52858 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME carboplatin CARBOPLATIN 16875718 77587 52859 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102477 77588 52860 GMNN 51053 DRUGGABLE GENOME GNF-PF-4418 CHEMBL604321 77589 52861 EMP1 2012 NA GEFITINIB GEFITINIB 16087880 77590 52862 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ATORVASTATIN ATORVASTATIN 11882317,12119202,9598838,15864114,10357840,12562847,10537160,15353498,12145148 77591 52863 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DNDI1417719 CHEMBL1420370 77593 52864 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PD-0325901 PD-0325901 23398453 77594 52865 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE NERVE GROWTH FACTOR 11166474,10617652,15209791 77595 52866 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME Lexipafant LEXIPAFANT 77597 52867 ALOX15 246 ENZYME, DRUGGABLE GENOME DEOXYVASICINONE DEOXYVASICINONE 77598 52868 TUBB2A 7280 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 23708010,23916255 77600 52869 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE ZEARALENONE ZEARALENONE 77601 52870 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THIORIDAZINE THIORIDAZINE 77604 52871 LIPF 8513 ENZYME, DRUGGABLE GENOME ORLISTAT ORLISTAT 77605 52872 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-1919 CHEMBL576409 77607 52873 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR SURAMIN HEXASODIUM SURAMIN HEXASODIUM 77608 52874 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR BRIGATINIB BRIGATINIB 26372962 77609 52875 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE 178101219 77611 52876 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE WX-UK1 77612 52877 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SJ000082806 CHEMBL494668 77613 52878 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR ENTINOSTAT ENTINOSTAT 19966789,20491440,22321215 77614 52879 CBX1 10951 NA RITANSERIN RITANSERIN 77616 52880 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE OXETHAZAINE OXETHAZAINE 77617 52881 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL ESTAZOLAM ESTAZOLAM 77619 52882 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE TPN 12005453 77620 52883 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650781 77622 52884 PDE10A 10846 ENZYME, DRUGGABLE GENOME TAK-063 BALIPODECT 25815469 77623 52885 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Sotalol SOTALOL 77624 52886 PAH 5053 DRUGGABLE GENOME, ENZYME TETRAHYDROBIOPTERIN SAPROPTERIN 77625 52887 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 252827421 77626 52888 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME Nadroparin calcium 77627 52889 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR WORTMANNIN WORTMANNIN 77628 52890 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR antagonist 252166890 CHEMBL1093266 77629 52891 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME modulator CHEMBL3545047 BMS-852927 77630 52892 NOS1 4842 DRUGGABLE GENOME, ENZYME CHEMOPREVENTIVE 12082549 77631 52893 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GS-6637 77633 52894 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LOMOFUNGIN LOMOFUNGIN 77634 52895 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL139 DICLOFENAC 77636 52896 NR2C1 7181 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME RETINOIC ACID 9071982 77638 52897 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Hydrazide derivative 3 77640 52898 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR AVE0897 77641 52899 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME PMID27539678-Compound-6 77642 52900 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TRIAMCINOLONE TRIAMCINOLONE 22931300 77643 52901 CXCL8 3576 DRUGGABLE GENOME HYDROQUINONE HYDROQUINONE 17118622 77644 52902 CD58 965 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE interferon beta-1a 77645 52903 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Pertuzumab PERTUZUMAB 77648 52904 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PAXILLINE PAXILLINE 77649 52905 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor XL228 XL-228 77650 52906 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR antagonist 135650786 77652 52907 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR HYDROCODONE HYDROCODONE 77655 52908 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DANTHRON DANTHRON 77657 52909 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME IFN 12232043 77658 52910 USP1 7398 DNA REPAIR, PROTEASE, ENZYME MMV085203 CHEMBL586031 77659 52911 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PONATINIB PONATINIB 26703895 77660 52912 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AGN-208397 77662 52913 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER mifepristone MIFEPRISTONE 77666 52914 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-19803 CHEMBL522983 77667 52915 HMGCR 3156 ENZYME, DRUGGABLE GENOME ATORVASTATIN ATORVASTATIN 77668 52916 KCNMA1 3778 DRUGGABLE GENOME, ION CHANNEL blocker 135652466 77669 52917 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE BPR1J373 27512117 77670 52918 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102270 77671 52919 SULT1A3 6818 DRUGGABLE GENOME, ENZYME tapentadol TAPENTADOL 77673 52920 ATXN2 6311 NA (S)-FLUOXETINE CHEMBL1169388 77674 52921 CD3D 915 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE OTELIXIZUMAB OTELIXIZUMAB 77675 52922 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL3545394 DRF-10945 77676 52923 CD38 952 CELL SURFACE, DRUGGABLE GENOME antibody 404859056 77677 52924 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CARBOPLATIN CARBOPLATIN 77678 52925 GUCY1A2 2977 ENZYME, DRUGGABLE GENOME activator CHEMBL730 NITROGLYCERIN 77679 52926 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME (R)-NITRENDIPINE (R)-NITRENDIPINE 77680 52927 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME elacridar ELACRIDAR 77681 52928 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 6-METHOXY-HARMALAN CHEMBL338115 77682 52929 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME Ancrod ANCROD 77683 52930 XDH 7498 DRUGGABLE GENOME, ENZYME ERYTHROMYCIN ERYTHROMYCIN 14730107 77684 52931 BAZ2B 29994 NA SALICYLALDEHYDE THIOSEMICARBAZONE SALICYLALDEHYDE THIOSEMICARBAZONE 77685 52932 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist CHEMBL1657 TAZAROTENE 77688 52933 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME activator 178101112 77689 52934 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR atenolol ATENOLOL 21562465 77691 52935 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000173328 CHEMBL591613 77692 52936 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BRL-52656 CHEMBL433508 77693 52937 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME 6,4'-DIHYDROXYFLAVONE CHEMBL484663 77694 52938 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TPKI-24 CHEMBL2392553 77695 52939 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL2107818 ALDOXORUBICIN 77696 52940 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PIMARIC ACID PIMARIC ACID 77697 52941 ITGA5 3678 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE CILENGITIDE CILENGITIDE 77698 52942 PTGS2 5743 DRUGGABLE GENOME, ENZYME URSOLIC ACID URSOLIC ACID 9784154 77701 52943 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME DNDI1417467 CHEMBL1997335 77702 52944 GMNN 51053 DRUGGABLE GENOME GNF-PF-2893 CHEMBL312032 77703 52945 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PACLITAXEL PACLITAXEL 22139083 77704 52946 MPHOSPH8 54737 NA MIFEPRISTONE MIFEPRISTONE 77706 52947 SGK2 10110 ION CHANNEL, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME FASUDIL FASUDIL 77707 52948 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHLORANIL CHLORANIL 77708 52949 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ALISERTIB ALISERTIB 77709 52950 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR FORASARTAN FORASARTAN 77710 52951 MPHOSPH8 54737 NA AG-538 CHEMBL56393 77711 52952 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE IL-5 2090920 77712 52953 ALOX15 246 ENZYME, DRUGGABLE GENOME THIOMERSAL THIMEROSAL 77713 52954 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051807 SCRIPTAID 77714 52955 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL2103840 DINACICLIB 77715 52956 POLB 5423 DNA REPAIR, DRUGGABLE GENOME STICTIC ACID STICTIC ACID 77718 52957 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 4-Carboxamido-isoindolinone derivative 5 77720 52958 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME VEL-0230 CHEMBL1085282 77721 52959 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL GDC0310 77722 52960 GPER1 2852 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR agonist 135651233 TAMOXIFEN 77723 52961 HPSE 10855 ENZYME, DRUGGABLE GENOME METERGOLINE METERGOLINE 23415087 77725 52962 TMEM97 27346 NA Piperidine derivative 6 77726 52963 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME BIM23A760 77728 52964 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL967 TEMAZEPAM 77729 52965 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LINSIDOMINE LINSIDOMINE 77730 52966 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE TCMDC-123480 CHEMBL588683 77733 52967 ACP5 54 ENZYME, DRUGGABLE GENOME M-CSF CILMOSTIM 12390325 77734 52968 ATAD5 79915 NA SIB-1757 CHEMBL88553 77737 52969 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor EVEROLIMUS EVEROLIMUS 77739 52970 PSMD1 5707 NA inhibitor BORTEZOMIB BORTEZOMIB 77741 52971 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TEDATIOXETINE TEDATIOXETINE 77742 52972 PTGS1 5742 ENZYME, DRUGGABLE GENOME Mesalazine MESALAMINE 77744 52973 CA9 768 DRUGGABLE GENOME, ENZYME PMID30074415-Compound-12 77748 52974 ALOX15 246 ENZYME, DRUGGABLE GENOME HOMIDIUM BROMIDE HOMIDIUM BROMIDE 77749 52975 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE VEGF 15687494 77751 52976 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 249565861 77752 52977 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE 681640 CHEMBL379975 77753 52978 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OLANZAPINE OLANZAPINE 77754 52979 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1574 PHENTERMINE 77755 52980 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE LOBAPLATIN LOBAPLATIN 11116285 77756 52981 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE antibody PF-04605412 PF-04605412 77757 52982 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE MILTEFOSINE MILTEFOSINE 16752184 77759 52983 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PHENANTHROLINE PHENANTHROLINE 77762 52984 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CR-665 77764 52985 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AMOXAPINE AMOXAPINE 77766 52986 HPSE 10855 ENZYME, DRUGGABLE GENOME HEPARAN SULFATE 17121850,2998789 77767 52987 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Cetuximab CETUXIMAB 27149458,27102076,27216155,26341921,24063894,27251290,26843189,27207775,24813888,22270724,25948633,27312529,24141978 77769 52988 SELE 6401 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CY-1503 77770 52989 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME SORAFENIB SORAFENIB 77771 52990 EPHA7 2045 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, TYROSINE KINASE inhibitor CHEMBL24828 VANDETANIB 77772 52991 NRP1 8829 DRUGGABLE GENOME PALIFERMIN PALIFERMIN 77773 52992 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE GNF-PF-860 CHEMBL593254 77775 52993 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CEPHALOTHIN SODIUM CEPHALOTHIN SODIUM 77776 52994 XDH 7498 DRUGGABLE GENOME, ENZYME FEBUXOSTAT FEBUXOSTAT 77777 52995 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR ARABINOFURANOSYLCYTOSINE 16505115 77778 52996 MPST 4357 ENZYME, DRUGGABLE GENOME THYROXINE THYROXINE 10709617 77781 52997 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR P-276 77782 52998 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE EUPATORIN EUPATORIN 77783 52999 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Paracetamol, combinations excl. Psycholeptics (Vicks MediNait Sirup) 77785 53000 E2F1 1869 TRANSCRIPTION FACTOR PACLITAXEL PACLITAXEL 16849574 77787 53001 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME ZSTK474 24251790 77788 53002 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR GW441756X GW441756X 77789 53003 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-30 77790 53004 NOS1 4842 DRUGGABLE GENOME, ENZYME AZITHROMYCIN AZITHROMYCIN 14730107 77791 53005 TUBB6 84617 DRUGGABLE GENOME MAYTANSINE MAYTANSINE 563462 77794 53006 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ONO-9054 SEPETAPROST 77795 53007 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 187051830 77796 53008 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME NSC-139257 CHEMBL1256364 77797 53009 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME FLUORANTHEN-3-YLAMINE CHEMBL103583 77798 53010 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178103660 HYDROCODONE 77802 53011 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ARRY-380 TUCATINIB 77803 53012 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME ERBSTATIN ERBSTATIN 77804 53013 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32x 77806 53014 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME IMATINIB IMATINIB 77808 53015 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TAMOXIFEN TAMOXIFEN 22931300 77809 53016 CES2 8824 DRUGGABLE GENOME, ENZYME mycophenolate mofetil 24220207 77810 53017 SP1 6667 TRANSCRIPTION FACTOR metformin METFORMIN 24853734,29352482 77811 53018 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE Diflorasone DIFLORASONE 77812 53019 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-21 77814 53020 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051805 QUISINOSTAT 77817 53021 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DAIDZIN DAIDZIN 77818 53022 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR ALVESPIMYCIN ALVESPIMYCIN 77820 53023 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102258 77821 53024 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME LY2784544 GANDOTINIB 77823 53025 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL411907 SONOLISIB 77826 53026 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650194 DIPRENORPHINE 77827 53027 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 77829 53028 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR ADRIAMYCIN ADRIAMYCIN 11751478 77832 53029 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-71a 77833 53030 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PRACTOLOL PRACTOLOL 77834 53031 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ANTHRAQUINONE ANTHRAQUINONE 16357514 77835 53032 KCNJ3 3760 EXTERNAL SIDE OF PLASMA MEMBRANE, ION CHANNEL, DRUGGABLE GENOME blocker 135652729 77836 53033 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME BW-723C86 CHEMBL1255834 77837 53034 MLLT3 4300 CLINICALLY ACTIONABLE montelukast MONTELUKAST 26083242 77840 53035 PRDX4 10549 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME docetaxel DOCETAXEL 20157331 77841 53036 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME TEMAZEPAM TEMAZEPAM 77844 53037 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 3,4-DICHLOROISOCOUMARIN CHEMBL24983 77845 53038 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417447 CHEMBL1307453 77846 53039 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR STANOLONE STANOLONE 77847 53040 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HYDROCORTISONE 21-OCTANOATE CHEMBL253989 77848 53041 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ZERANOL ZERANOL 77849 53042 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE ISOETHARINE MESYLATE ISOETHARINE MESYLATE 77850 53043 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CENISERTIB CENISERTIB 77852 53044 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 5-(4-PHENYLBUTOXY)PSORALEN CHEMBL1256851 77853 53045 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE RDP58 77854 53046 SPP1 6696 DRUGGABLE GENOME PROTEIN PHOSPHATASE INHIBITOR 11818502 77856 53047 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 178102516 VEMURAFENIB 77857 53048 ALOX15 246 ENZYME, DRUGGABLE GENOME DL-TRYPTOPHAN DL-TRYPTOPHAN 77858 53049 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME CTS-21166 77859 53050 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR inhibitor 178103408 CLOFARABINE 77860 53051 PIP4K2A 5305 ENZYME, KINASE TDR77225 CHEMBL1353528 77861 53052 DCN 1634 DRUGGABLE GENOME RAPAMYCIN SIROLIMUS 17200203 77862 53053 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME CHLORPYRAMIN HYDROCHLORIDE CHLORPYRAMIN HYDROCHLORIDE 19610651 77863 53054 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE LEVOSALBUTAMOL LEVOSALBUTAMOL 77864 53055 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102339 SUNITINIB 77865 53056 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR SP-600125 SP-600125 77867 53057 POLK 51426 DNA REPAIR, ENZYME CEFOTIAM HYDROCHLORIDE CEFOTIAM HYDROCHLORIDE 77868 53058 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 16 77871 53059 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antibody MPDL3280A ATEZOLIZUMAB 77872 53060 NAT1 9 ENZYME, DRUGGABLE GENOME ACETYLSALICYLIC ACID 10547619 77873 53061 PARP3 10039 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR KU-0058948 CHEMBL380648 19354255 77874 53062 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME AC-264613 CHEMBL494502 18720984 77875 53063 SMN2 6607 DRUGGABLE GENOME CID 4101591 CHEMBL428789 77876 53064 MAPT 4137 DRUGGABLE GENOME TCMDC-123904 CHEMBL586061 77877 53065 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME HYPERICIN HYPERICIN 77878 53066 BAZ2B 29994 NA PROTOCATECHUALDEHYDE PROTOCATECHUALDEHYDE 77881 53067 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE QUERCETIN QUERCETIN 17045724 77884 53068 MAOA 4128 DRUGGABLE GENOME, ENZYME Desoxypeganine 77885 53069 GAA 2548 DRUGGABLE GENOME, ENZYME (-)-EPICATECHIN (-)-EPICATECHIN 77888 53070 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Cyclofenil CYCLOFENIL 77889 53071 MUC2 4583 DRUGGABLE GENOME CHEMOPREVENTIVE AGENT 15754327 77890 53072 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000032151 CHEMBL592600 77891 53073 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE alemtuzumab ALEMTUZUMAB 27173875 77895 53074 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102755 77899 53075 KLRD1 3824 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME certolizumab pegol 26453102 77900 53076 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME oxaliplatin OXALIPLATIN 19434073,22188361,29662106,18267032,20385995,22026922,20078613,21449681 77902 53077 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor KX2-391 KX2-391 77903 53078 SLC47A1 55244 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 135650099 CIMETIDINE 77904 53079 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE agonist CHEMBL2108508 INTERFERON ALFA-2A 77905 53080 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL494089 GSK-690693 77906 53081 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-242718 CHEMBL275724 77908 53082 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE GAMMA-FAGARINE GAMMA-FAGARINE 77911 53083 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE RADIATION THERAPY 28476872 77912 53084 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME P-276 77913 53085 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME VX-745 NEFLAMAPIMOD 17659871 77914 53086 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ETHINYL ESTRADIOL ETHINYL ESTRADIOL 77915 53087 KCNF1 3754 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL113461 TEDISAMIL 77916 53088 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor VEMURAFENIB VEMURAFENIB 77917 53089 POLI 11201 DNA REPAIR GW305074X GW305074X 77918 53090 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102338 SU-014813 77919 53091 ADCY1 107 DRUGGABLE GENOME, ENZYME lithium LITHIUM 29121268 77920 53092 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 (R)-FLECAINIDE (R)-FLECAINIDE 77921 53093 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR Antiinflammatory agents, non-steroids 28750137 77922 53094 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor VORINOSTAT VORINOSTAT 77924 53095 TSPO 706 DRUGGABLE GENOME Tricyclic indole compound 6 77925 53096 ALOX15 246 ENZYME, DRUGGABLE GENOME GW7074 CHEMBL72365 77926 53097 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Veliparib VELIPARIB 77927 53098 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY ACEBUTOLOL ACEBUTOLOL 2878948 77929 53099 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME PMID27828716-Compound-20 77930 53100 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE CELECOXIB CELECOXIB 16172791 77931 53101 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING (-)-CAMPHOR (-)-CAMPHOR 77932 53102 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor 223366206 INFIGRATINIB 77933 53103 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME OSI-632 OSI-632 77935 53104 SYT1 6857 KINASE, TRANSPORTER cocaine COCAINE 31059723 77936 53105 FN1 2335 DRUGGABLE GENOME AS1409 77937 53106 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200845 HALCINONIDE 77938 53107 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VORINOSTAT VORINOSTAT 24694055,19344175,19966789,26211462,23622981,22260166,18381238,20491440,21548582,23672185,19084294 77939 53108 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-119913 CHEMBL471004 22524450 77940 53109 VKORC1 79001 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL16694 PHENPROCOUMON 77941 53110 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-28 77942 53111 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE CEFOPERAZONE CEFOPERAZONE 22166395 77943 53112 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE EXEMESTANE EXEMESTANE 77944 53113 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ENDOXIFEN ENDOXIFEN 24805199 77945 53114 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CERTOLIZUMAB PEGOL 77946 53115 CA1 759 DRUGGABLE GENOME, ENZYME PARABEN PARABEN 77947 53116 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32g 77948 53117 SMN1 6606 DRUGGABLE GENOME GNF-PF-3037 CHEMBL600336 77949 53118 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417221 CHEMBL1459280 77951 53119 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 249565916 77954 53120 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 252166807 77956 53121 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME METHYSERGIDE MALEATE 77959 53122 MAPK13 5603 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME N-(3-OXODODECANOYL)HOMOSERINELACTONE CHEMBL8483 18566250 77961 53123 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist CHEMBL107430 NRX195183 77962 53124 PDE3A 5139 ENZYME, DRUGGABLE GENOME NM-702 77963 53125 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BETAINE HYDROCHLORIDE BETAINE HYDROCHLORIDE 77964 53126 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-21 77965 53127 GMNN 51053 DRUGGABLE GENOME TCMDC-123457 CHEMBL285157 77966 53128 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PYRAZINOIC ACID PYRAZINOIC ACID 77967 53129 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE TAE-684 TAE-684 77969 53130 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME FINASTERIDE FINASTERIDE 7835306 77970 53131 SMN2 6607 DRUGGABLE GENOME LEFLUNOMIDE LEFLUNOMIDE 77971 53132 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE antibody VOLOCIXIMAB VOLOCIXIMAB 77972 53133 RAB9A 9367 ENZYME, DRUGGABLE GENOME 3,5-DIPHENYLISOXAZOLE 3,5-DIPHENYLISOXAZOLE 77976 53134 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SARCOLYSIN SARCOLYSIN 77977 53135 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE CENISERTIB CENISERTIB 77978 53136 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 310264718 PF-03758309 77979 53137 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ESTAZOLAM ESTAZOLAM 77981 53138 TYMSOS 494514 NA etoposide ETOPOSIDE 77982 53139 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PACLITAXEL PACLITAXEL 16020661 77984 53140 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RO5126766 26438159 77985 53141 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME KAEMPFEROL KAEMPFEROL 25190466 77986 53142 SMN2 6607 DRUGGABLE GENOME DAIDZEIN DAIDZEIN 77987 53143 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER vindesine VINDESINE 25637052 77988 53144 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE Everolimus EVEROLIMUS 21189378,27615706 77989 53145 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER OLVANIL OLVANIL 77990 53146 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 252166703 77992 53147 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE ELND005 SCYLLITOL 77993 53148 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200703 CHLORDIAZEPOXIDE HYDROCHLORIDE 77996 53149 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME DORAMAPIMOD DORAMAPIMOD 18602262 77997 53150 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ASENAPINE ASENAPINE 77998 53151 CYBB 1536 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME, ENZYME LUTEOLIN LUTEOLIN 23786520 77999 53152 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR SILMITASERTIB SILMITASERTIB 22832316 78000 53153 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL BUTETHAL BUTETHAL 78002 53154 ICAM3 3385 DRUGGABLE GENOME METHOTREXATE METHOTREXATE 16215763 78003 53155 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME VALPROIC ACID 78005 53156 GPT 2875 ENZYME TACROLIMUS TACROLIMUS 9825815 78006 53157 HMGCR 3156 ENZYME, DRUGGABLE GENOME ATORVASTATIN ATORVASTATIN 78007 53158 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE (S)APOMORPHINE (S)APOMORPHINE 78009 53159 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MEDI4276 MEDI-4276 78011 53160 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Oxindole derivative 3 78012 53161 KDM5B 10765 ENZYME inhibitor 178103606 78013 53162 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652566 78015 53163 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650245 ETONITAZENE 78018 53164 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME PHYSODIC ACID PHYSODIC ACID 78019 53165 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-2657 CHEMBL578944 78021 53166 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Selective serotonin reuptake inhibitors 26871771 78022 53167 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CEFDITORIN PIVOXIL CEFDITORIN PIVOXIL 78023 53168 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME aspirin ASPIRIN 78024 53169 TYMP 1890 GROWTH FACTOR, DRUGGABLE GENOME 5-DEOXY-5-FLUOROURIDINE 11956613 78025 53170 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE GENISTEIN GENISTEIN 8424658 78026 53171 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651284 TROPISETRON 78028 53172 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME CLOSANTEL CLOSANTEL 78030 53173 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE QUESTIOMYCIN B QUESTIOMYCIN B 78031 53174 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME Phenoxodiol 78032 53175 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME RESVERATROL RESVERATROL 17270149,15837718,14729643 78034 53176 BCHE 590 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 4 78035 53177 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LAPATINIB LAPATINIB 22511346 78036 53178 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE XL418 XL-418 78037 53179 EYA2 2139 DNA REPAIR NSC-119889 CHEMBL516616 78040 53180 ATAD5 79915 NA GNF-PF-910 CHEMBL585408 78041 53181 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor AXITINIB AXITINIB 78044 53182 GHRL 51738 DRUGGABLE GENOME ETANERCEPT ETANERCEPT 18400355 78045 53183 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor XL281 XL-281 78046 53184 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME HAEMATOXYLIN HAEMATOXYLIN 78047 53185 AHCY 191 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 178101808 CHEMBL202701 78048 53186 RGS4 5999 DRUGGABLE GENOME inhibitor 249565713 78049 53187 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME SELUMETINIB SELUMETINIB 26544513 78051 53188 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CYC-116 CYC-116 78052 53189 KIF11 3832 DRUGGABLE GENOME ALN-VSP 78055 53190 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL3545285 XL-999 78057 53191 CRTC1 23373 CLINICALLY ACTIONABLE NVP-BEZ235 DACTOLISIB 78058 53192 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Taxol/Paraplatin/Herceptin 78059 53193 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE INCB13739 78060 53194 NCOA3 8202 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, ENZYME DNDI1417478 CHEMBL1972216 78061 53195 PSMD13 5719 NA BORTEZOMIB BORTEZOMIB 24524217 78062 53196 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL2103849 UDENAFIL 78064 53197 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 4',7-DIMETHOXY-5-HYDROXYGENISTEIN 78067 53198 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LOFEPRAMINE LOFEPRAMINE 78069 53199 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE BAS 01152706 CHEMBL2002487 78070 53200 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING 1,3-DIPHENYLTHIOUREA CHEMBL275260 78071 53201 ORAI1 84876 TRANSCRIPTION FACTOR, ION CHANNEL, TRANSPORTER blocker 375973229 78072 53202 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME N-(cyanomethyl)-4-(2-(phenylamino)pyrimidin-4-yl)benzamide derivative 1 78073 53203 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME HEXACHLOROPHENE HEXACHLOROPHENE 78074 53204 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR WORTMANNIN WORTMANNIN 78075 53205 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PIMASERTIB PIMASERTIB 78076 53206 ALB 213 TRANSPORTER, DRUGGABLE GENOME Ebselen EBSELEN 78077 53207 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL462018 TRICIRIBINE PHOSPHATE 78079 53208 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CLOXYQUIN CLOXYQUIN 78082 53209 PON1 5444 ENZYME, TRANSPORTER, DRUGGABLE GENOME fluorouracil FLUOROURACIL 78083 53210 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NITROXOLINE NITROXOLINE 78084 53211 TUBB2A 7280 DRUGGABLE GENOME MKC-1 ENMD-981693 78085 53212 ALOX15 246 ENZYME, DRUGGABLE GENOME BRL-50481 CHEMBL484928 78087 53213 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE Pyrimidopyridazinone derivative 2 78090 53214 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 249565883 CHEMBL1956070 78091 53215 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME XL888 XL-888 22351686 78092 53216 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE TAE-684 TAE-684 78094 53217 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME TRIAZOLAM TRIAZOLAM 78095 53218 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178103494 IBRUTINIB 78096 53219 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Ado-Trastuzumab Emtansine 78097 53220 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME OXALIPLATIN OXALIPLATIN 17127229 78098 53221 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE DASATINIB DASATINIB 78099 53222 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SELUMETINIB SELUMETINIB 78100 53223 DNER 92737 NA BI 894999 78102 53224 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GERALDOL GERALDOL 78103 53225 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565910 78106 53226 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME PYROGALLOL RED PYROGALLOL RED 78107 53227 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE Acetyldigitoxin ACETYLDIGITOXIN 78108 53228 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor OSIMERTINIB OSIMERTINIB 78109 53229 CDC42BPA 8476 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME KENPAULLONE KENPAULLONE 78111 53230 PTGES 9536 DRUGGABLE GENOME, ENZYME Benzamide derivative 16 78113 53231 ADAMTS4 9507 ENZYME, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE inhibitor 252166754 78114 53232 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME partial agonist CHEMBL3544917 RAPASTINEL 78116 53233 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-43 78118 53234 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE LANATOSIDE C LANATOSIDE C 78119 53235 PSMC4 5704 NA inhibitor CHEMBL325041 BORTEZOMIB 78120 53236 SLC47A2 146802 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 135650099 CIMETIDINE 78121 53237 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051792 PANOBINOSTAT 78122 53238 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor ALVOCIDIB ALVOCIDIB 78123 53239 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme2WO2012/098065bottom 78124 53240 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 178100453 78125 53241 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-43 78126 53242 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME DASATINIB DASATINIB 78127 53243 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME arformoterol ARFORMOTEROL 78128 53244 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE MOTESANIB MOTESANIB 78130 53245 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor PKI-587 GEDATOLISIB 78132 53246 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME VE-822 BERZOSERTIB 78133 53247 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME NISOLDIPINE NISOLDIPINE 78134 53248 TSPO 706 DRUGGABLE GENOME ZOPICLONE ZOPICLONE 78135 53249 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1095 ETHOTOIN 78136 53250 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AZOSEMIDE AZOSEMIDE 78140 53251 KDM1A 23028 DRUGGABLE GENOME, ENZYME, CELL SURFACE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING inhibitor 315661201 78141 53252 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor CHEMBL283120 AXL-1717 78142 53253 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 223366179 78143 53254 ADH1A 124 DRUGGABLE GENOME Fomepizole FOMEPIZOLE 78144 53255 CFL1 1072 KINASE CINNARIZINE CINNARIZINE 16680159 78146 53256 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ARQ092 26469692 78147 53257 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 310264733 FIMEPINOSTAT 78148 53258 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME modulator CHEMBL1059 PREGABALIN 78149 53259 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GNF-PF-1859 CHEMBL1520837 78150 53260 AKR1B10 57016 DRUGGABLE GENOME, ENZYME ENOXOLONE ENOXOLONE 21561086 78151 53261 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor SNS-314 SNS-314 78152 53262 GPNMB 10457 ENZYME, DRUGGABLE GENOME MONOMETHYL-AURISTATIN E ADC CONJUGATE 78154 53263 CA4 762 DRUGGABLE GENOME, ENZYME, TRANSPORTER, CELL SURFACE inhibitor CHEMBL20 ACETAZOLAMIDE 78156 53264 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE BISDEMETHOXYCURCUMIN BISDEMETHOXYCURCUMIN 19112019 78162 53265 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 78163 53266 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME KRP-104 BISEGLIPTIN 78165 53267 MGLL 11343 DRUGGABLE GENOME, ENZYME Azetidinyl-piperazine derivative 1 78168 53268 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 178103311 PRINABEREL 78169 53269 COL3A1 1281 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 78170 53270 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Phenylpropylamine derivative 5 78171 53271 IMPDH1 3614 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1200955 MYCOPHENOLATE MOFETIL HYDROCHLORIDE 78174 53272 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL129857 AS-602868 78175 53273 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME 2S,1'S,2'S)-2-(CARBOXYCYCLOPROPYL)GLYCINE CHEMBL280563 78176 53274 CFD 1675 ENZYME, DRUGGABLE GENOME, PROTEASE ACH-4471 78177 53275 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TROGLITAZONE TROGLITAZONE 22931300 78178 53276 PDE4D 5144 DRUGGABLE GENOME, ENZYME Papaverine PAPAVERINE 78179 53277 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL428690 ALVOCIDIB 78181 53278 TUBB 203068 DRUGGABLE GENOME Mebendazole MEBENDAZOLE 78182 53279 BARD1 580 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR docetaxel DOCETAXEL 30071039 78183 53280 ARG2 384 ENZYME inhibitor 315661102 78185 53281 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE RITODRINE RITODRINE 78188 53282 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL PHENACEMIDE PHENACEMIDE 78189 53283 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE AllerB 78192 53284 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-55 78193 53285 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 telithromycin TELITHROMYCIN 78194 53286 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CEFOTETAN CEFOTETAN 78197 53287 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TPCK TPCK 78202 53288 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME STREPTOMYCIN STREPTOMYCIN 78203 53289 HEBP1 50865 DRUGGABLE GENOME Benzo[d]oxazole derivative 3 78204 53290 TUBA4A 7277 DRUGGABLE GENOME inhibitor CHEMBL107 COLCHICINE 78205 53291 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE CDA 10606241 78206 53292 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME CeaVac 78207 53293 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-ETHYLANTHRAQUINONE CHEMBL42355 78208 53294 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HARMINE HARMINE 78210 53295 ERCC3 2071 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME Platinum compounds 25069034 78211 53296 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1789842 INDACATEROL MALEATE 78212 53297 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 METHOCARBAMOL METHOCARBAMOL 22931300 78213 53298 CAT 847 ENZYME, DRUGGABLE GENOME anthracyclines and related substances 19863340 78214 53299 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SU-11274 CHEMBL261641 17595299,23403296 78215 53300 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 178103586 ENTINOSTAT 78217 53301 CCR6 1235 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, G PROTEIN COUPLED RECEPTOR agonist 178100546 78218 53302 GAPDH 2597 DRUGGABLE GENOME, ENZYME OESTRADIOL ESTRADIOL 9883985 78219 53303 MAPK7 5598 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 328083482 78220 53304 PTGIR 5739 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 223365888 SELEXIPAG 78221 53305 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL2103882 TIVANTINIB 78222 53306 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor NIRAPARIB NIRAPARIB 78223 53307 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 7,12-DIMETHYL-BENZO[A]ANTHRACENE CHEMBL329673 78225 53308 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 135652717 STAUROSPORINE 78226 53309 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CD123CAR-41BB-CD3zeta-EGFRt-expressing T cells 78227 53310 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Phenylpyrrolidinone derivative 4 78229 53311 CHD1 1105 NA EPIRUBICIN EPIRUBICIN 78231 53312 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TYRPHOSTIN 1 TYRPHOSTIN 1 78233 53313 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME ESCITALOPRAM ESCITALOPRAM 78235 53314 MAGEA3 4102 ENZYME, DRUGGABLE GENOME Polynoma-1 78236 53315 RIPOR2 9750 NA Drugs For Treatment Of Tuberculosis 30720667 78237 53316 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor MASITINIB MASITINIB 78238 53317 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE Zadaxin/lamivudine 78239 53318 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR GSK-269962A GSK-269962A 78242 53319 MAPT 4137 DRUGGABLE GENOME LINOLENIC ACID LINOLENIC ACID 78244 53320 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 1-[2-(TRIFLUOROMETHYL)PHENYL]IMIDAZOLE CHEMBL277525 78245 53321 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR MCP-1 16452499 78246 53322 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL428690 ALVOCIDIB 78249 53323 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135652672 BRUCINE 78250 53324 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 135649975 TICAGRELOR 78251 53325 ADH1B 125 DRUGGABLE GENOME, ENZYME abacavir ABACAVIR 24625462 78252 53326 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 318164841 NETARSUDIL 78253 53327 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor TRAMETINIB TRAMETINIB 78254 53328 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL969 PRAZEPAM 78255 53329 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE inhibitor 223366174 AZD-1236 78256 53330 ZSCAN25 221785 NA tacrolimus TACROLIMUS 29318894,29454235 78258 53331 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ANTIFUNGALS 11751127 78259 53332 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PMID28048944-Compound-5 78260 53333 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME HOMIDIUM BROMIDE HOMIDIUM BROMIDE 78261 53334 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME NEU-2000 78262 53335 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL970 HALAZEPAM 78264 53336 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME BENZBROMARONE BENZBROMARONE 78265 53337 USP1 7398 DNA REPAIR, PROTEASE, ENZYME XCT790 CHEMBL189753 78266 53338 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DOCEBENONE DOCEBENONE 78267 53339 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102711 78270 53340 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR BAY-613606 CHEMBL541400 78271 53341 HTT 3064 DRUGGABLE GENOME DACTINOMYCIN DACTINOMYCIN 78272 53342 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GW7647 GW7647 78273 53343 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE PROTEIN KINASE INHIBITOR 9579573 78276 53344 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE repaglinide REPAGLINIDE 22414228 78278 53345 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME GEMCITABINE GEMCITABINE 17079475 78279 53346 GMNN 51053 DRUGGABLE GENOME PHENAZINE-1-CARBOXYLIC ACID PHENAZINE-1-CARBOXYLIC ACID 78281 53347 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 252827527 78282 53348 POLI 11201 DNA REPAIR FOSFONET FOSFONET 78283 53349 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR MORAb-022 GIMSILUMAB 78285 53350 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor SOPHORETIN QUERCETIN 78287 53351 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417263 CHEMBL1431115 78288 53352 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE XL765 78293 53353 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 252166739 78295 53354 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 antiepileptics 78298 53355 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000040837 CHEMBL590672 78304 53356 ALDH1A1 216 DRUGGABLE GENOME, ENZYME RETINAL RETINAL 78306 53357 CHRNA5 1138 DRUGGABLE GENOME, ION CHANNEL antagonist 178100796 78307 53358 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME doxorubicin DOXORUBICIN 11351295 78308 53359 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 8392465 78309 53360 DCBLD1 285761 NA irinotecan IRINOTECAN 23478653 78310 53361 TUBA3C 7278 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 78311 53362 CSNK2A2 1459 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME, TRANSCRIPTION FACTOR US8791257, 38 78314 53363 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor 178103109 TRAMETINIB 78315 53364 RPS6KA5 9252 DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE DOVITINIB DOVITINIB 78316 53365 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR IRBESARTAN IRBESARTAN 78319 53366 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 381118844 78320 53367 BAZ2B 29994 NA DNDI1417485 CHEMBL1346468 78321 53368 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE DS-1205b 78322 53369 USP1 7398 DNA REPAIR, PROTEASE, ENZYME BENZBROMARONE BENZBROMARONE 78324 53370 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist CHEMBL1131 ACITRETIN 78325 53371 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE BMS-754807 BMS-754807 26561558 78328 53372 FAAH 2166 ENZYME, DRUGGABLE GENOME Spirocyclic diamine urea derivative 1 78329 53373 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CINNARIZINE CINNARIZINE 16680159 78330 53374 ATXN2 6311 NA ENCLOMIPHENE CITRATE ENCLOMIPHENE CITRATE 78331 53375 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BVT.115959 BVT.115959 78332 53376 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650228 78333 53377 CXCL8 3576 DRUGGABLE GENOME MDX-018 78334 53378 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1256 ISOFLURANE 78335 53379 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE TAE-684 TAE-684 78336 53380 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID27724045-Compound-17 78340 53381 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Aminocyclopentenone compound 4 78341 53382 CDK11B 984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL488436 AZD-5438 78342 53383 UGT1A6 54578 ENZYME, DRUGGABLE GENOME anthracyclines and related substances 23441093,21900104 78344 53384 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER 7,8,3'-TRIHYDROXYFLAVONE CHEMBL225513 78345 53385 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE NIROGACESTAT NIROGACESTAT 26407235 78347 53386 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BIOALLETHRIN S-CYCLOPENTENYL ISOMER BIOALLETHRIN S-CYCLOPENTENYL ISOMER 78348 53387 MAPT 4137 DRUGGABLE GENOME RABEPRAZOLE RABEPRAZOLE 78349 53388 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME PROPOFOL PROPOFOL 78350 53389 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE Codrituzumab CODRITUZUMAB 78351 53390 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NCG-C00094421-01 CHEMBL553503 78354 53391 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL346631 CEP-7055 78356 53392 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME CHELERYTHRINE CHELERYTHRINE 78357 53393 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 249565871 78358 53394 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor PANOBINOSTAT PANOBINOSTAT 78359 53395 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650179 78362 53396 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1743047 NECITUMUMAB 78363 53397 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 178102333 78364 53398 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Carebastine CAREBASTINE 78365 53399 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE LY3012212 78367 53400 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE GENISTEIN GENISTEIN 9712063 78368 53401 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE Triciribine prodrug 78370 53402 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ESTRADIOL ESTRADIOL 22931300 78371 53403 GLS 2744 ENZYME RHEIN RHEIN 78372 53404 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor TOZASERTIB TOZASERTIB 19035792 78374 53405 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE BEZ235 DACTOLISIB 24939055 78375 53406 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE NERATINIB NERATINIB 28679771,24009064,29523624,26874901,29146401,20142587,25287822,23220880,26243863 78376 53407 PRKAB1 5564 ENZYME, KINASE, DRUGGABLE GENOME METFORMIN METFORMIN 78377 53408 FZD7 8324 G PROTEIN COUPLED RECEPTOR, KINASE antibody 381118907 VANTICTUMAB 78378 53409 MAP3K9 4293 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565750 PRT-2607 78379 53410 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE KAEMPFEROL KAEMPFEROL 78380 53411 USP1 7398 DNA REPAIR, PROTEASE, ENZYME HOMIDIUM BROMIDE HOMIDIUM BROMIDE 78381 53412 HCK 3055 TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME US9108950, 1 78382 53413 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME GI-6207 78386 53414 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME MACROLIDES 18212111 78387 53415 CDK13 8621 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL1230607 PHA-793887 78388 53416 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-US20120277229 44(1.4) 78389 53417 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178101639 GEFITINIB 78390 53418 SLC15A3 51296 TRANSPORTER, DRUGGABLE GENOME 178101385 78391 53419 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME rucaparib RUCAPARIB 78393 53420 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650688 NALTRIBEN 78394 53421 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME 2,5-DINITRO-PHENOL CHEMBL107513 78395 53422 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL ISRADIPINE ISRADIPINE 78401 53423 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 VALERIAN VALERIAN 15900287 78403 53424 HDC 3067 DRUGGABLE GENOME, ENZYME ALPHA-FMH 78404 53425 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER inhibitor 384403652 78405 53426 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ARQ 087 78407 53427 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Epoxysuccinate derivative 10 78410 53428 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor JNJ38877605 78411 53429 USP1 7398 DNA REPAIR, PROTEASE, ENZYME DNDI1417080 CHEMBL1498652 78412 53430 KDM4A 9682 DRUGGABLE GENOME, ENZYME 6,7-ADTN HYDROBROMIDE CHEMBL1255656 78416 53431 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE Retroviral vector-transduced autologous T cells to express anti-GPC3 CARs 78417 53432 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-23 78418 53433 XDH 7498 DRUGGABLE GENOME, ENZYME Febuxostat FEBUXOSTAT 78419 53434 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME EVT100 78420 53435 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE STAUROSPORINE STAUROSPORINE 8068015 78426 53436 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME PHATHALIMIDE PHATHALIMIDE 18295491 78428 53437 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GNF-PF-2301 CHEMBL578061 78429 53438 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-123747 CHEMBL530698 78430 53439 FOS 2353 TRANSCRIPTION FACTOR, DRUGGABLE GENOME BROMOCRIPTINE BROMOCRIPTINE 11680511 78431 53440 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME APOMORPHINE APOMORPHINE 78434 53441 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER FUROXAN FUROXAN 78435 53442 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME COLCHICINE COLCHICINE 78436 53443 EIF3A 8661 NA carboplatin CARBOPLATIN 23127338 78438 53444 HTT 3064 DRUGGABLE GENOME CXD-101 CXD-101 78439 53445 CACNA1C 775 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200805 DILTIAZEM MALATE 78440 53446 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR agonist CHEMBL454138 TUROFEXORATE ISOPROPYL 78441 53447 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL1090771 AVAGACESTAT 78442 53448 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL3545176 DB959 78443 53449 CSK 1445 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE inhibitor HESPERADIN HESPERADIN 19035792 78444 53450 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201115 ESMOLOL HYDROCHLORIDE 78446 53451 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FENOFIBRIC ACID FENOFIBRIC ACID 23566516 78447 53452 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 363894223 78448 53453 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ZM-447439 CHEMBL202721 78449 53454 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1533 DESOGESTREL 78451 53455 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE inhibitor MK0752 78458 53456 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME HOMIDIUM BROMIDE HOMIDIUM BROMIDE 78459 53457 POLB 5423 DNA REPAIR, DRUGGABLE GENOME TCMDC-123532 CHEMBL547833 78460 53458 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER losartan LOSARTAN 27338075 78461 53459 VCAN 1462 DRUGGABLE GENOME CSA CYCLOSPORINE 14974815 78462 53460 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE LAPATINIB LAPATINIB 25587029 78464 53461 FZD1 8321 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, KINASE antagonist CHEMBL2364652 VANTICTUMAB 78466 53462 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR 4-HPR FENRETINIDE 8993839 78467 53463 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000296655 CHEMBL589734 78469 53464 PSMB2 5690 DRUGGABLE GENOME, PROTEASE, ENZYME CLASTO-LACTACYSTIN BETA-LACTONE CHEMBL490829 18801655 78472 53465 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE AT13148 AT-13148 22781553 78473 53466 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE BMS-708163 AVAGACESTAT 78474 53467 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist 310264667 78475 53468 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX ANGUSTIBALIN ANGUSTIBALIN 78477 53469 ATAD5 79915 NA ZEARALENONE ZEARALENONE 78478 53470 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Masitinib MASITINIB 78479 53471 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE RX-0201 ARCHEXIN 78480 53472 SLC6A1 6529 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE TIAGABINE TIAGABINE 78481 53473 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME (RS)-ROSCOVITINE (RS)-ROSCOVITINE 78483 53474 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 135651276 TRIAMCINOLONE 78486 53475 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER clozapine CLOZAPINE 27168101,19593168,22722500 78487 53476 PROM1 8842 CELL SURFACE, DRUGGABLE GENOME Anti-CD133-CAR vector-transduced T cells 78488 53477 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME LINOLENIC ACID LINOLENIC ACID 78489 53478 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 78490 53479 TOP2B 7155 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2107313 BECATECARIN 78492 53480 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1095 ETHOTOIN 78493 53481 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL3545366 VOXTALISIB 78494 53482 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE SELENIUM 9884517 78495 53483 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME COLLAGENASE COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 78497 53484 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NALOXONE NALOXONE 78498 53485 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor CHEMBL1230607 PHA-793887 78499 53486 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PIRITREXIM ISETHIONATE PIRITREXIM ISETHIONATE 78500 53487 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heteroaryl-carboxamide derivative 4 78501 53488 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE HALICLONADIAMINE HALICLONADIAMINE 22928967 78502 53489 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 249565749 78503 53490 GUCY1A2 2977 ENZYME, DRUGGABLE GENOME NAPROXCINOD NAPROXCINOD 78504 53491 IL1B 3553 KINASE, DRUGGABLE GENOME inhibitor CHEMBL1201834 CANAKINUMAB 78507 53492 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1910936 MK3207 78508 53493 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CLOFOCTOL CLOFOCTOL 78509 53494 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 348353622 78511 53495 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE sunitinib SUNITINIB 19248971 78512 53496 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2103749 BIVALIRUDIN 78513 53497 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR NSC-632536 CHEMBL1367933 78514 53498 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR BUTYLATED HYDROXYTOLUENE 11228746 78515 53499 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE LOBARIC ACID LOBARIC ACID 19362837 78516 53500 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL carbamazepine CARBAMAZEPINE 23859570,21747585,22591328,19289736,22292851,28753467,22188362,26314341,25155934,26555147,21561445 78517 53501 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME RG7221 26692321 78518 53502 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL1079742 ERLOTINIB HYDROCHLORIDE 78519 53503 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALFATRADIOL ALFATRADIOL 78520 53504 HBB 3043 DRUGGABLE GENOME, ENZYME Iron 78521 53505 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME FRENTIZOLE FRENTIZOLE 78522 53506 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME EBASTINE EBASTINE 78524 53507 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME METHABENZTHIAZURON METHABENZTHIAZURON 78525 53508 IDE 3416 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, ENZYME, PROTEASE inhibitor 252166797 78526 53509 MTTP 4547 DRUGGABLE GENOME inhibitor CHEMBL2105662 LOMITAPIDE MESYLATE 78529 53510 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME EMODIN EMODIN 78530 53511 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200903 SECOBARBITAL SODIUM 78531 53512 ZBTB22 9278 NA aspirin ASPIRIN 78532 53513 MAOB 4129 DRUGGABLE GENOME, ENZYME 2-Methoxyphenol GUAIACOL HYDROCHLORIDE 78533 53514 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DROSPIRENONE DROSPIRENONE 78535 53515 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE SCH-527123 NAVARIXIN 78537 53516 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CEFAMANDOLE SODIUM CEFAMANDOLE SODIUM 78541 53517 CA9 768 DRUGGABLE GENOME, ENZYME BAY 79-4620 78542 53518 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME Ublituximab + umbralisib 78544 53519 KCNJ3 3760 EXTERNAL SIDE OF PLASMA MEMBRANE, ION CHANNEL, DRUGGABLE GENOME THYROTROPIN THYROTROPIN 10075694 78548 53520 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ticlopidine TICLOPIDINE 17339877 78550 53521 SERPIND1 3053 DRUGGABLE GENOME, PROTEASE INHIBITOR SULODEXIDE SULODEXIDE 78551 53522 MAOB 4129 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 4 78552 53523 NOS1 4842 DRUGGABLE GENOME, ENZYME CIMETIDINE CIMETIDINE 7543704 78555 53524 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE allosteric modulator 310264748 78557 53525 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PINAFIDE PINAFIDE 78558 53526 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102555 JNJ-7706621 78559 53527 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE PMID29130358-Compound-Figure17(13) 78560 53528 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIHYDROTANSHINONE I DIHYDROTANSHINONE I 78561 53529 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000290256 CHEMBL590666 78566 53530 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME GNF-PF-5510 CHEMBL578741 78568 53531 TLR7 51284 DRUGGABLE GENOME imiquimod IMIQUIMOD 26556041 78569 53532 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME DIHYDREXIDINE DIHYDREXIDINE 78570 53533 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR THIRAM THIRAM 78572 53534 TUBB2A 7280 DRUGGABLE GENOME VINORELBINE VINORELBINE 78575 53535 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME FELBAMATE FELBAMATE 78576 53536 HSPA4 3308 NA PHOTOFRIN PHOTOFRIN 8625311 78578 53537 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RAMATROBAN RAMATROBAN 78581 53538 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE INCB54828 78582 53539 TMEM97 27346 NA Bicyclo-heptan-2-amine derivative 3 78583 53540 KDM4A 9682 DRUGGABLE GENOME, ENZYME ISOORIENTIN ISOORIENTIN 78586 53541 MAPT 4137 DRUGGABLE GENOME GW7074 CHEMBL72365 78589 53542 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor BYL719 ALPELISIB 78591 53543 PSMD13 5719 NA CARFILZOMIB CARFILZOMIB 24524217 78594 53544 GDA 9615 ENZYME THIOGUANINE THIOGUANINE 7384171 78596 53545 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor FORETINIB FORETINIB 78597 53546 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME MISONIDAZOLE MISONIDAZOLE 3759562 78598 53547 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 7,8-DIHYDROXYFLAVONE 7,8-DIHYDROXYFLAVONE 78599 53548 POLB 5423 DNA REPAIR, DRUGGABLE GENOME METHYLDOPA METHYLDOPA 78602 53549 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545085 XL-228 78605 53550 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE lovastatin LOVASTATIN 78606 53551 NOD1 10392 CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 310264668 78608 53552 IMPDH1 3614 ENZYME, DRUGGABLE GENOME PMID28074661-Compound-US20120264760C82 78610 53553 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE VERAPAMIL VERAPAMIL 3436366 78611 53554 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME partial agonist CHEMBL3544917 RAPASTINEL 78612 53555 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME DNDI1417614 CHEMBL1567571 78613 53556 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME R-1487 R-1487 78616 53557 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US10179791, Compound 296 78617 53558 POLK 51426 DNA REPAIR, ENZYME HISPIDIN HISPIDIN 78619 53559 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor CHEMBL565612 SOTRASTAURIN 78620 53560 RTN4 57142 DRUGGABLE GENOME antibody 249565934 OZANEZUMAB 78623 53561 UNC119 9094 KINASE 374883853 78625 53562 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PYROGALLOL RED PYROGALLOL RED 78626 53563 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BITHIONOL BITHIONOL 78629 53564 DCK 1633 DRUGGABLE GENOME, ENZYME, KINASE CLADRIBINE CLADRIBINE 18570408 78630 53565 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 sertindole SERTINDOLE 9187528 78632 53566 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE SAPONARIN SAPONARIN 26471090 78635 53567 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TERPYRIDINE TERPYRIDINE 78642 53568 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE agonist CHEMBL1743008 DROZITUMAB 78643 53569 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE BERKELEYACETAL A BERKELEYACETAL A 17970594 78644 53570 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME UNGEREMINE UNGEREMINE 22014547 78645 53571 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3184679 AZD-4547 78646 53572 PTGES 9536 DRUGGABLE GENOME, ENZYME Carboxylic acid derivative 1 78648 53573 TAOK3 51347 DNA REPAIR, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565898 78649 53574 PTGS2 5743 DRUGGABLE GENOME, ENZYME RALOXIFENE RALOXIFENE 15243281 78650 53575 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651412 78651 53576 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME DUTOGLIPTIN DUTOGLIPTIN 78653 53577 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 glipizide GLIPIZIDE 24442125,10208645 78655 53578 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545159 R-333 78657 53579 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME LINIFANIB LINIFANIB 78659 53580 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TCMDC-125575 CHEMBL587620 78661 53581 ADAM17 6868 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, NEUTRAL ZINC METALLOPEPTIDASE, TRANSPORTER, ENZYME CB7969312 CHEMBL599255 78663 53582 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 252166900 TIROTUNDIN 78664 53583 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME CYC116 78667 53584 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NALBUPHINE NALBUPHINE 22931300 78668 53585 CSNK1D 1453 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 178102563 78669 53586 PORCN 64840 ENZYME, DRUGGABLE GENOME, TRANSPORTER ETC-1922159 ETC-159 78671 53587 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME THIETHYLPERAZINE MALATE THIETHYLPERAZINE MALATE 78672 53588 SULT1A1 6817 DRUGGABLE GENOME, ENZYME estrogens ESTRONE SODIUM SULFATE 11062153,11906176,12034366,9068609 78673 53589 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR DDTC 1381236 78675 53590 SMN2 6607 DRUGGABLE GENOME CID 3238892 CHEMBL261118 78676 53591 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL695 TRIMETHADIONE 78677 53592 TNFRSF10A 8797 DRUGGABLE GENOME, CELL SURFACE agonist 310264670 CHEMBL1790415 78678 53593 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME GNF-PF-4068 CHEMBL584668 78680 53594 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME nutlin-3 NUTLIN-3 14704432 78681 53595 ANKS1B 56899 NA methamphetamine METHAMPHETAMINE 31462767 78682 53596 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR METHOTREXATE METHOTREXATE 78683 53597 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE SUNITINIB SUNITINIB 78685 53598 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GFT-505 ELAFIBRANOR 78686 53599 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-640559 CHEMBL1287866 21074425 78688 53600 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CAMPTOTHECIN CAMPTOTHECIN 16258022 78695 53601 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIAZOXIDE DIAZOXIDE 78696 53602 MAPT 4137 DRUGGABLE GENOME ROSMARINIC ACID ROSMARINIC ACID 78697 53603 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE NILOTINIB NILOTINIB 26191369 78698 53604 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE GNF-PF-3023 CHEMBL535331 78700 53605 PRKX 5613 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE PF-562271 PF-00562271 78702 53606 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME HMG-COA REDUCTASE INHIBITOR 16624629 78704 53607 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME DOVITINIB DOVITINIB 78706 53608 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DIFFRACTAIC ACID DIFFRACTAIC ACID 78707 53609 SMN2 6607 DRUGGABLE GENOME CID 867101 CHEMBL406557 78708 53610 SLC22A11 55867 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER zidovudine ZIDOVUDINE 22960662 78710 53611 NEDD4L 23327 ENZYME hydrochlorothiazide HYDROCHLOROTHIAZIDE 18591455,21052022,19635985 78711 53612 OGG1 4968 ENZYME SELENIUM 16759981 78715 53613 MAPT 4137 DRUGGABLE GENOME ISOBOLDINE ISOBOLDINE 78716 53614 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 310264696 AZD-8835 78717 53615 RAB9A 9367 ENZYME, DRUGGABLE GENOME PD-98059 CHEMBL35482 78718 53616 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1201167 CARVEDILOL PHOSPHATE 78719 53617 SMG1 23049 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DNA REPAIR Bisquaternary salt 78720 53618 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING VORINOSTAT VORINOSTAT 19344175,19966789,26211462,23622981,22260166,20491440,21548582,19084294 78722 53619 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR RADANAMYCIN RADANAMYCIN 16464590 78724 53620 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 187051758 INDACATEROL 78725 53621 RRM2B 50484 ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor CHEMBL2105467 TEZACITABINE 78726 53622 ALOX15B 247 DRUGGABLE GENOME, ENZYME TYRPHOSTIN 47 TYRPHOSTIN 47 78727 53623 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER olanzapine OLANZAPINE 18086475,29443543,17038883 78729 53624 RAC1 5879 CLINICALLY ACTIONABLE, KINASE, DRUG RESISTANCE ZU-4194738 CHEMBL554475 19527032 78730 53625 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME FOTEMUSTINE FOTEMUSTINE 11279615 78731 53626 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist 178100809 78732 53627 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE cannabinoids NABIXIMOLS 11840318,31246565 78734 53628 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL ISOPROPYL ISOTHIOCYANATE ISOPROPYL ISOTHIOCYANATE 26263397 78735 53629 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AURIN AURIN 78736 53630 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor CHEMBL2219421 RECILISIB 78738 53631 DHFR 1719 DRUGGABLE GENOME, ENZYME Aminosalicylic Acid 78739 53632 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE CYC-116 CYC-116 78742 53633 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CHLORPROMAZINE CHLORPROMAZINE 78743 53634 CXCL8 3576 DRUGGABLE GENOME CETUXIMAB CETUXIMAB 15908664 78744 53635 ARSA 410 DRUGGABLE GENOME, ENZYME TRANILAST TRANILAST 78746 53636 ATP1A2 477 ENZYME, TRANSPORTER, ION CHANNEL, DRUGGABLE GENOME inhibitor CHEMBL1614 DESLANOSIDE 78747 53637 MAPT 4137 DRUGGABLE GENOME SB-200646 CHEMBL85194 78748 53638 APC 324 CLINICALLY ACTIONABLE 5-AZA-2'-DEOXYCYTIDINE 17065059,12097272 78749 53639 MT2A 4502 NA ETHANOL ALCOHOL 1733046 78750 53640 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME TAMATINIB R-406 78751 53641 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR inhibitor 252827366 GILTERITINIB 78752 53642 CYP24A1 1591 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME telaprevir TELAPREVIR 26158282 78754 53643 UGT1A10 54575 DRUGGABLE GENOME, ENZYME DICLOFENAC DICLOFENAC 8511777 78755 53644 KDM4A 9682 DRUGGABLE GENOME, ENZYME L-750667 CHEMBL1256738 78756 53645 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PRACINOSTAT PRACINOSTAT 78759 53646 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Dasatinib DASATINIB 26758680 78761 53647 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3545043 ASAPIPRANT 78762 53648 IL1B 3553 KINASE, DRUGGABLE GENOME MAFOSFAMIDE MAFOSFAMIDE 3497116 78763 53649 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL3545300 CP-459632 78764 53650 VEGFB 7423 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR Aflibercept AFLIBERCEPT 78765 53651 ABHD6 57406 PHOSPHOLIPASE, ENZYME Piperazine carbamic compound 1 78767 53652 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Amphetamine AMPHETAMINE 78769 53653 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor PIVANEX AN-9 78771 53654 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME IMATINIB IMATINIB 16254145 78774 53655 UBA2 10054 DRUGGABLE GENOME, ENZYME BENSERAZIDE HYDROCHLORIDE BENSERAZIDE HYDROCHLORIDE 78776 53656 MAPT 4137 DRUGGABLE GENOME BAS 01152706 CHEMBL2002487 78778 53657 DPYS 1807 ENZYME atenolol ATENOLOL 78779 53658 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW827106X GW827106X 78780 53659 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1200485 SORAFENIB TOSYLATE 78781 53660 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR US9359293, TA 78783 53661 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER partial agonist CHEMBL1134 DECAMETHONIUM BROMIDE 78784 53662 CACNB4 785 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL2103836 IMAGABALIN 78785 53663 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME VITAMIN K 10930097 78786 53664 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor AZD 1152 78787 53665 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135650268 FLUDROCORTISONE 78788 53666 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE EPINEPHRINE BITARTRATE EPINEPHRINE BITARTRATE 78791 53667 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR CENISERTIB CENISERTIB 78794 53668 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME KW-2449 KW-2449 78796 53669 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE MGAH22 MARGETUXIMAB 28119295 78797 53670 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE 178101218 78798 53671 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TRIACETYLRESVERATROL TRIACETYLRESVERATROL 78800 53672 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE KAINIC ACID KAINIC ACID 78801 53673 XDH 7498 DRUGGABLE GENOME, ENZYME didanosine DIDANOSINE 23315321 78802 53674 POLK 51426 DNA REPAIR, ENZYME MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 78804 53675 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor 354702259 FUTIBATINIB 78805 53676 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Exemestane EXEMESTANE 78806 53677 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID25991433-Compound-J5 78807 53678 MAPT 4137 DRUGGABLE GENOME (E)-DIBENZYLIDENEACETONE CHEMBL17201 78808 53679 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565687 78809 53680 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650021 78810 53681 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL2068839 RISLENEMDAZ 78812 53682 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME CAR-BCMA T cell 78814 53683 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Naveglitazar NAVEGLITAZAR 78815 53684 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2011137219 36(3-5) 78817 53685 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor 363894211 PEXMETINIB 78818 53686 SMN1 6606 DRUGGABLE GENOME TCMDC-124585 CHEMBL587856 78819 53687 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME inhibitor CHEMBL2109355 DUSIGITUMAB 78821 53688 BAZ2B 29994 NA MMV000704 CHEMBL582478 78822 53689 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME COAGULATION FACTOR IX 78823 53690 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE LAUROGUADINE LAUROGUADINE 78825 53691 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME PROTOPORPHYRIN DISODIUM PROTOPORPHYRIN DISODIUM 78828 53692 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651794 78830 53693 LAG3 3902 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE IMP-701 78831 53694 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Nintedanib NINTEDANIB 22238366 78832 53695 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Irinotecan IRINOTECAN 25567130,24042735,23209031,16707468,25714871,26341920,21325073,24798549,25322874 78833 53696 KEAP1 9817 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING 375973258 78834 53697 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR MESALAMINE MESALAMINE 78835 53698 POLI 11201 DNA REPAIR CHLOROTHALONIL CHLOROTHALONIL 78836 53699 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL VOACANGINE VOACANGINE 24484240 78837 53700 CXCL12 6387 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, KINASE MyoCell SDF-1 78838 53701 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE TCMDC-124416 CHEMBL530664 78839 53702 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE NG-MONOMETHYL-L-ARGININE 1846547 78840 53703 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE agonist 315661330 78841 53704 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DES DIETHYLSTILBESTROL 14647453 78843 53705 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL2396661 ALPELISIB 78844 53706 KCNH6 81033 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 78847 53707 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Goserelin GOSERELIN 78848 53708 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 354702284 78849 53709 MARCHF8 220972 ENZYME Fluvirin A(H1N1) 78850 53710 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ILORASERTIB ILORASERTIB 78852 53711 NT5C3A 51251 ENZYME gemcitabine GEMCITABINE 22838949 78853 53712 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE IMMUNOLOGICAL ADJUVANT 9161882 78855 53713 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME CID 5310801 CHEMBL260451 78856 53714 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL220492 TOPIRAMATE 78859 53715 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME DTPA PENTETIC ACID 9343371 78861 53716 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID29671355-Compound-36 78862 53717 GSTA1 2938 ENZYME, DRUGGABLE GENOME ETHACRYNIC ACID 11092982 78864 53718 CBX1 10951 NA KETOCONAZOLE KETOCONAZOLE 78866 53719 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Anti-BCMA CAR T cells 78868 53720 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR DEBIO 0932 78869 53721 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR Vemurafenib VEMURAFENIB 24265153,21383288,22389471,24448821,27312529 78870 53722 UBA2 10054 DRUGGABLE GENOME, ENZYME GINGKOLIC ACID GINGKOLIC ACID 23920437 78875 53723 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE Ribociclib RIBOCICLIB 28151717 78877 53724 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GDC-0941 PICTILISIB 24265153,22693356,27020857,23136191,9661880,26058079,26577700,19276360,24322983,28119489,26733612 78878 53725 CCL11 6356 DRUGGABLE GENOME TYROSINE KINASE INHIBITOR 10527858 78880 53726 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE PERTUZUMAB PERTUZUMAB 26206558,25216528 78881 53727 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALCLOMETASONE DIPROPIONATE ALCLOMETASONE DIPROPIONATE 78884 53728 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR 6-HYDROXYFLAVONOL CHEMBL210411 19592245 78885 53729 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME CC-223 CC-223 78888 53730 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR SKF-38393 SKF-38393 78889 53731 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR VX-11e 25370473 78890 53732 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME MK-5108 MK-5108 78893 53733 ERAP1 51752 PROTEASE, ENZYME, DRUGGABLE GENOME ESCULETIN ESCULETIN 78894 53734 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL450 METHARBITAL 78896 53735 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649973 78898 53736 ALOX15B 247 DRUGGABLE GENOME, ENZYME EBSELEN EBSELEN 78899 53737 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Eplerenone EPLERENONE 78900 53738 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649786 78901 53739 FHIT 2272 CLINICALLY ACTIONABLE, ENZYME, TRANSPORTER Fructose FRUCTOSE 78902 53740 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2096646 AMINOSALICYLATE SODIUM 78903 53741 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GARLIC GARLIC 11962257 78905 53742 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Bidentate ligands of Markush derivative 1 78907 53743 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CALPEPTIN CALPEPTIN 78908 53744 NLRP1 22861 PROTEASE DITHIAZANINE IODIDE DITHIAZANINE IODIDE 78911 53745 EPHA6 285220 DRUGGABLE GENOME, KINASE, TYROSINE KINASE inhibitor CHEMBL24828 VANDETANIB 78912 53746 PSMD12 5718 NA inhibitor CHEMBL451887 CARFILZOMIB 78913 53747 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR 8-FLUOROTRYPTANTHRIN CHEMBL1098875 78915 53748 RHOA 387 KINASE, CLINICALLY ACTIONABLE simvastatin SIMVASTATIN 23166513 78916 53749 U2AF1 7307 CLINICALLY ACTIONABLE H3B-8800 78919 53750 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL2177390 IPATASERTIB 78920 53751 BAZ2B 29994 NA HARMAN-3-CARBOXYLIC ACID HARMAN-3-CARBOXYLIC ACID 78922 53752 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR IL-3 8604024,8219192 78924 53753 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME inhibitor 348353657 CEP-37440 78925 53754 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME METHADONE METHADONE 8149590 78927 53755 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200733 DESFLURANE 78929 53756 HBB 3043 DRUGGABLE GENOME, ENZYME PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 78931 53757 ALOX15 246 ENZYME, DRUGGABLE GENOME Indolizine derivative 1 78932 53758 SLC47A2 146802 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 178101231 78933 53759 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MASITINIB MASITINIB 78936 53760 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROCYCLIDINE PROCYCLIDINE 78937 53761 GMNN 51053 DRUGGABLE GENOME ALEXIDINE DIHYDROCHLORIDE ALEXIDINE DIHYDROCHLORIDE 78938 53762 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PLX7904 27523909 78939 53763 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BENZOPHENONE-THIOSEMICARBAZONE BENZOPHENONE-THIOSEMICARBAZONE 78941 53764 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE AMPKINONE AMPKINONE 20873794 78942 53765 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE peginterferon alfa-2a 78943 53766 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 94381 CHEMBL374632 78944 53767 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE UNII-DRL23N424R 78945 53768 DIABLO 56616 NA CLADRIBINE CLADRIBINE 12948851 78946 53769 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 78947 53770 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME ADRIAMYCIN ADRIAMYCIN 16871999 78949 53771 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DECYLUBIQUINONE DECYLUBIQUINONE 78950 53772 GRM6 2916 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650629 78951 53773 PSENEN 55851 DRUGGABLE GENOME inhibitor MK0752 78952 53774 FURIN 5045 ENZYME, PROTEASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 252166858 78953 53775 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR SOTRASTAURIN SOTRASTAURIN 78954 53776 ATP1B1 481 DRUGGABLE GENOME, TRANSPORTER, ENZYME inhibitor CHEMBL254219 DIGITOXIN 78955 53777 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TOLTERODINE TOLTERODINE 78956 53778 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME VITAMIN B2 VITAMIN B2 78958 53779 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1200877 FLUMETHASONE PIVALATE 78962 53780 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE antibody ONARTUZUMAB ONARTUZUMAB 78965 53781 GLS 2744 ENZYME PMID30273516-Compound-12 78966 53782 HSD17B2 3294 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME inhibitor 385612198 78967 53783 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR HELENALIN HELENALIN 78969 53784 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE LY2780301 78972 53785 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYPROTERONE CYPROTERONE 78973 53786 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE lopinavir LOPINAVIR 78974 53787 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Diamidothiazole derivative 1 78976 53788 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME tropisetron TROPISETRON 12728290,12065557 78977 53789 PDE4A 5141 DRUGGABLE GENOME, ENZYME DYPHYLLINE DYPHYLLINE 78978 53790 VEGFC 7424 GROWTH FACTOR, TRANSPORTER, DRUGGABLE GENOME SUNITINIB SUNITINIB 21787417 78979 53791 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE GEFITINIB GEFITINIB 78980 53792 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NSC-119915 CHEMBL1481974 78981 53793 PDE3A 5139 ENZYME, DRUGGABLE GENOME Inamrinone Lactate 78982 53794 H2AW 92815 NA CISPLATIN CISPLATIN 11008128 78984 53795 NDUFV3 4731 ENZYME inhibitor CHEMBL3545320 ME-344 78985 53796 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 4'-METHOXYFLAVONE 4'-METHOXYFLAVONE 78986 53797 GATA4 2626 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE RIBAVIRIN MONOPHOSPHATE RIBAVIRIN MONOPHOSPHATE 21310620 78987 53798 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650361 78988 53799 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CAD-106 78989 53800 POLK 51426 DNA REPAIR, ENZYME TCMDC-123723 CHEMBL525103 78990 53801 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL1200395 ORPHENADRINE CITRATE 78991 53802 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DEXAMETHASONE DEXAMETHASONE 15817834 78992 53803 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135651116 78993 53804 ALOX15B 247 DRUGGABLE GENOME, ENZYME CONGO RED CONGO RED 78995 53805 ATP2A2 488 ENZYME, DRUGGABLE GENOME, TRANSPORTER Mydicar 78996 53806 MAPT 4137 DRUGGABLE GENOME DIHYDROGAMBOGIC ACID DIHYDROGAMBOGIC ACID 78997 53807 CRBN 51185 ENZYME, DRUG RESISTANCE POMALIDOMIDE POMALIDOMIDE 23480694 78998 53808 TLR7 51284 DRUGGABLE GENOME Imiquimod IMIQUIMOD 79000 53809 CBX1 10951 NA GW405833 CHEMBL73711 79001 53810 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE BUTORPHANOL BUTORPHANOL 79002 53811 SOCS6 9306 NA INSULIN INSULIN 18356406 79003 53812 CTSG 1511 DRUGGABLE GENOME, PROTEASE, ENZYME, CELL SURFACE TNF-ALPHA 7499869 79004 53813 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME US8481733, 106 79005 53814 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE P7170 PANULISIB 25700704 79006 53815 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SEL-24 79007 53816 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HYCANTHONE HYCANTHONE 22931300 79008 53817 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Carboprost Tromethamine 79009 53818 TNKS 8658 DRUGGABLE GENOME, ENZYME inhibitor 404859119 79010 53819 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 381118865 79015 53820 BAP1 8314 PROTEASE, TUMOR SUPPRESSOR, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE OLAPARIB OLAPARIB 28389374,22683710 79017 53821 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 249565845 79018 53822 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-124354 CHEMBL546344 79020 53823 ABI1 10006 CLINICALLY ACTIONABLE, KINASE ponatinib PONATINIB 79021 53824 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL3039504 NINTEDANIB ESYLATE 79022 53825 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME DINACICLIB DINACICLIB 27378523 79023 53826 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417080 CHEMBL1498652 79024 53827 APC 324 CLINICALLY ACTIONABLE ICG-001 15314234 79025 53828 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE STI571 IMATINIB MESYLATE 79026 53829 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE UE-2343 79027 53830 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TRIAMTERENE TRIAMTERENE 79028 53831 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME inhibitor CHEMBL362558 LY-2090314 79029 53832 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CLOPIDOGREL CLOPIDOGREL 79030 53833 GMNN 51053 DRUGGABLE GENOME AG-490 CHEMBL56543 79031 53834 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE Certolizumab pegol 79032 53835 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CT 327 79034 53836 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME A66 26137449 79035 53837 UGCG 7357 ENZYME, DRUGGABLE GENOME inhibitor 178101543 MIGLUSTAT 79036 53838 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL526 PROPOFOL 79037 53839 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200760 BALSALAZIDE DISODIUM 79041 53840 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-2812 CHEMBL125044 79042 53841 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DOXORUBICIN DOXORUBICIN 22931300 79043 53842 BAZ2B 29994 NA DNDI1417941 CHEMBL2095095 79044 53843 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE Marimastat MARIMASTAT 79045 53844 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 187051797 APICIDIN 79048 53845 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PREDNISOLONE PREDNISOLONE 17329922 79049 53846 MAPT 4137 DRUGGABLE GENOME GNF-2 CHEMBL483847 79050 53847 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PRACINOSTAT PRACINOSTAT 79051 53848 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-46 79053 53849 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor MASITINIB MASITINIB 79054 53850 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Indoline derivative 1 79055 53851 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIOTYROSINE DIOTYROSINE 79056 53852 TUBB6 84617 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 79058 53853 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE EPICATECHIN GALLATE EPICATECHIN GALLATE 15620252 79061 53854 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME RESMINOSTAT RESMINOSTAT 79063 53855 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Dasatinib DASATINIB 27231123,19098899,27154914,27222538 79064 53856 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME EPINASTINE EPINASTINE 79065 53857 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 178102569 79067 53858 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME CISPLATIN CISPLATIN 15790433 79068 53859 USP1 7398 DNA REPAIR, PROTEASE, ENZYME 2-BENZOYL-5-METHOXYBENZOQUINONE 2-BENZOYL-5-METHOXYBENZOQUINONE 79069 53860 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME NBQX NBQX 79070 53861 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME celecoxib CELECOXIB 22336956 79071 53862 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650107 NAMODENOSON 79072 53863 POLK 51426 DNA REPAIR, ENZYME ERUCIC ACID ERUCIC ACID 79073 53864 SF3B1 23451 CLINICALLY ACTIONABLE H3B-8800 79075 53865 ATAD2B 54454 ENZYME inhibitor 385612205 79076 53866 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME HYCANTHONE HYCANTHONE 79077 53867 RRM2B 50484 ENZYME, DRUGGABLE GENOME, DNA REPAIR cytarabine CYTARABINE 24024897 79078 53868 CBX1 10951 NA AG-527 CHEMBL258767 79079 53869 PCSK1 5122 DRUGGABLE GENOME, PROTEASE, ENZYME PHOSPHODIESTERASE INHIBITOR 8822509 79080 53870 AKR1C3 8644 ENZYME, DRUGGABLE GENOME N-(indolylcarbonyl)-piperidine derivative 1 79082 53871 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE FAS1 79083 53872 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-neostenine 79084 53873 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL522892 DOVITINIB 79088 53874 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR raloxifene RALOXIFENE 27546373 79089 53875 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DROMETRIZOLE DROMETRIZOLE 79090 53876 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650518 79091 53877 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 405067319 79095 53878 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3545403 BMS-833923 79097 53879 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor ENTINOSTAT ENTINOSTAT 79098 53880 PLA2G7 7941 DRUGGABLE GENOME, ENZYME Bicyclic pyrimidine derivative 2 79099 53881 GMNN 51053 DRUGGABLE GENOME 2'-HYDROXYCHALCONE 2'-HYDROXYCHALCONE 79101 53882 DKC1 1736 CLINICALLY ACTIONABLE V934/V935 79103 53883 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME SHO-SAIKO-TO 10716612 79105 53884 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Anti-hCD70 CAR transduced PBL 79108 53885 NTS 4922 DRUGGABLE GENOME AZASERINE AZASERINE 1993548 79110 53886 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HER2p63-71 peptide vaccine 79111 53887 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SCH772984 26725216 79112 53888 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE PHA-767491 CHEMBL225519 79113 53889 NPTN 27020 CELL SURFACE, DRUGGABLE GENOME GP100 8779689 79114 53890 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PHENYTOIN PHENYTOIN 22931300 79115 53891 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL1201421 PEGAPTANIB SODIUM 79117 53892 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650462 79118 53893 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME blocker 135652744 79119 53894 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE Entrectinib ENTRECTINIB 26939704 79120 53895 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 223366207 BUPARLISIB 79123 53896 TPO 7173 ENZYME, DRUGGABLE GENOME, CELL SURFACE METHIMAZOLE METHIMAZOLE 79124 53897 MPHOSPH8 54737 NA GW7074 CHEMBL72365 79125 53898 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME fesoterodine FESOTERODINE 79126 53899 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME GNF-PF-5061 CHEMBL601385 79128 53900 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE THYMIDINE MONOPHOSPHATE THYMIDINE MONOPHOSPHATE 6434741 79129 53901 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PSAMMAPLIN A PSAMMAPLIN A 25884112 79130 53902 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PROMAZINE PROMAZINE 79131 53903 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE CAMPTOTHECIN CAMPTOTHECIN 22386982 79133 53904 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME HORMONES 1978836 79135 53905 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ALISERTIB ALISERTIB 79136 53906 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102343 VANDETANIB 79138 53907 CYP7B1 9420 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SAQUINAVIR SAQUINAVIR 12461038 79139 53908 BAZ2B 29994 NA BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 79140 53909 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 79141 53910 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ETAZOLATE ETAZOLATE 79144 53911 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE inhibitor 178103412 DESLANOSIDE 79147 53912 ABCC6 368 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER CHONDROITIN SULFATE 12600949 79148 53913 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE EUCALYPTIN A EUCALYPTIN A 22934600 79149 53914 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-45 79150 53915 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 5,7-DIHYDROXYISOFLAVONE 5,7-DIHYDROXYISOFLAVONE 79151 53916 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL1236962 OMIPALISIB 79152 53917 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME R-roscovitine SELICICLIB 79155 53918 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME 3,8'-BIAPIGENIN CHEMBL515252 79156 53919 TAC1 6863 DRUGGABLE GENOME ETHER ETHER 2421032 79157 53920 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME GALACTITOL GALACTITOL 11098845 79158 53921 COL4A4 1286 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 79159 53922 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL LORAZEPAM LORAZEPAM 79160 53923 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE BITHIONOL BITHIONOL 79162 53924 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 223366072 ALECTINIB 79163 53925 MAP2K6 5608 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TYROSINE KINASE, TUMOR SUPPRESSOR WX-554 WX-554 79165 53926 HTT 3064 DRUGGABLE GENOME MECHLORETHAMINE HYDROCHLORIDE MECHLORETHAMINE HYDROCHLORIDE 79166 53927 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178103791 LORATADINE 79167 53928 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL DIAZEPAM DIAZEPAM 79168 53929 CA12 771 DRUGGABLE GENOME ETHOXZOLAMIDE ETHOXZOLAMIDE 23159038 79169 53930 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FURAFYLLINE FURAFYLLINE 79170 53931 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178102294 BI-2536 79171 53932 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER vaccine EP-2101 79172 53933 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor SUNITINIB SUNITINIB 79173 53934 CIC 23152 CLINICALLY ACTIONABLE, DRUG RESISTANCE VEMURAFENIB VEMURAFENIB 28178529 79177 53935 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CLADRIBINE CLADRIBINE 79179 53936 BAZ2B 29994 NA GNF-PF-5134 CHEMBL602969 79180 53937 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME PD-98059 CHEMBL35482 12883735 79182 53938 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER sertraline SERTRALINE 24192121,18215618,26704739,22641028 79183 53939 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 rucaparib RUCAPARIB 79186 53940 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME PHENYLBUTYRYLHYDROXAMIC ACID PHENYLBUTYRYLHYDROXAMIC ACID 21874153 79187 53941 ATAD5 79915 NA TCMDC-125602 CHEMBL580183 79188 53942 MYD88 4615 CLINICALLY ACTIONABLE fentanyl FENTANYL 79190 53943 PTGS2 5743 DRUGGABLE GENOME, ENZYME RWJ-67657 RWJ-67657 79191 53944 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4612 CHEMBL601550 79192 53945 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR VITAMIN C 16944783 79193 53946 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DOXORUBICIN DOXORUBICIN 12438277 79194 53947 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME LEO 124249 79195 53948 GADD45A 1647 DNA REPAIR, TUMOR SUPPRESSOR, KINASE NB1011 12477050 79197 53949 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CEFONICID CEFONICID 79198 53950 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-21 79201 53951 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545248 DS-7423 79203 53952 GGT1 2678 CELL SURFACE, ENZYME, PROTEASE, DRUGGABLE GENOME PHENYTOIN PHENYTOIN 12402220,1346382 79204 53953 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antagonist FULVESTRANT FULVESTRANT 79205 53954 LNPEP 4012 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, TRANSPORTER, PROTEASE US10023583, Example 5 79206 53955 CREB1 1385 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR antidepressants 23537502,20643483,17548750 79208 53956 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL1200996 MEPHENTERMINE SULFATE 79209 53957 RGS4 5999 DRUGGABLE GENOME AG-538 CHEMBL56393 79212 53958 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE TOZASERTIB TOZASERTIB 79214 53959 MMP1 4312 DRUGGABLE GENOME, PROTEASE, ENZYME RAPAMYCIN SIROLIMUS 16914544 79215 53960 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 5-NITROQUINOLINE CHEMBL164449 79216 53961 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME EC20 79217 53962 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650349 HEXOCYCLIUM 79220 53963 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 178103994 DACOMITINIB 79221 53964 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME MERCURIC CHLORIDE MERCURIC CHLORIDE 79222 53965 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME ESTAZOLAM ESTAZOLAM 22137933 79223 53966 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME inhibitor 381118840 79225 53967 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE VELIPARIB VELIPARIB 79227 53968 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Copanlisib COPANLISIB 79228 53969 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME BAICALEIN BAICALEIN 79230 53970 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR VRT11E 24265153 79232 53971 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME ENTRECTINIB ENTRECTINIB 79233 53972 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL1789843 BELIMUMAB 79234 53973 MGLL 11343 DRUGGABLE GENOME, ENZYME Piperazine carbamic compound 3 79235 53974 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Thiadiazolidindione derivative 3 79237 53975 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE BMS-345541 BMS-345541 79238 53976 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR CUCURBITACIN D CUCURBITACIN D 25756299 79239 53977 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-5061 CHEMBL601385 79240 53978 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-5 79241 53979 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME BUTYRATE 12896903 79243 53980 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ILORASERTIB ILORASERTIB 79244 53981 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PF-06840003 PF-06840003 79246 53982 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE inhibitor CHEMBL3301622 GILTERITINIB 79249 53983 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR MESTRANOL MESTRANOL 3023023 79250 53984 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL359744 DOXORUBICIN HYDROCHLORIDE 79252 53985 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME TENOVIN-6 CHEMBL595354 22304848 79254 53986 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor ABT-888 VELIPARIB 79255 53987 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ALPRAZOLAM ALPRAZOLAM 79256 53988 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME PROMETHAZINE PROMETHAZINE 79258 53989 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE PD-0166285 PD-0166285 79259 53990 COMT 1312 DRUGGABLE GENOME, ENZYME heroin DIACETYLMORPHINE 79261 53991 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ARASERTACONAZOLE ARASERTACONAZOLE 79262 53992 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-704 CHEMBL597449 79263 53993 CDH1 999 CLINICALLY ACTIONABLE, DRUGGABLE GENOME ANTISERUM 3880756 79265 53994 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE cetuximab CETUXIMAB 23296156,27897268,17704420,28719596,30318772 79268 53995 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR TENOVIN-6 CHEMBL595354 22304848 79272 53996 ALOX5 240 DRUGGABLE GENOME, ENZYME TENIDAP TENIDAP 79273 53997 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR DNDI1417063 CHEMBL2094422 79274 53998 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 249565590 CHEMBL1236539 79276 53999 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR SULFENTRAZONE SULFENTRAZONE 79277 54000 RRM2 6241 DRUGGABLE GENOME, ENZYME NKP-46 79278 54001 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME inhibitor 249565939 79280 54002 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME TAS-119 TAS-119 79281 54003 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME GNF-PF-1260 CHEMBL584849 79282 54004 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CYCLOPHOSPHAMIDE CYCLOPHOSPHAMIDE 1682037 79284 54005 HMGCS1 3157 DRUGGABLE GENOME, ENZYME inhibitor 135651558 79285 54006 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CLONAZEPAM CLONAZEPAM 79286 54007 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE N-(4-CHLOROBENZOYL)EVODIAMINE CHEMBL1277315 20942490 79289 54008 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PMID28766366-Compound-Scheme9EHT6840 79291 54009 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CHEMBL2108354 UBLITUXIMAB 79295 54010 MARCHF8 220972 ENZYME Quattvaxem 79298 54011 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE DASATINIB DASATINIB 79300 54012 APOE 348 DRUGGABLE GENOME ANTIDEPRESSANT 14512205 79303 54013 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor 310264675 CUDC-101 79304 54014 PTGS1 5742 ENZYME, DRUGGABLE GENOME SUPROFEN SUPROFEN 79305 54015 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME Pyrido[1,2-a]indole-1.-carboxylic acid analog 6 79306 54016 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 404859011 79307 54017 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor VOLASERTIB VOLASERTIB 79309 54018 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor CHEMBL1678 DONEPEZIL HYDROCHLORIDE 79310 54019 EML4 27436 CLINICALLY ACTIONABLE, KINASE ASP3026 ASP-3026 27009859,25228534 79311 54020 NOS1 4842 DRUGGABLE GENOME, ENZYME NIMESULIDE NIMESULIDE 10741939 79312 54021 AIP 9049 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR TCDD 10986286 79315 54022 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYSTAMINE DIHYDROCHLORIDE CYSTAMINE DIHYDROCHLORIDE 79316 54023 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650988 79318 54024 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178101497 KETOPROFEN 79319 54025 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE AZD-1775 ADAVOSERTIB 79320 54026 MAPT 4137 DRUGGABLE GENOME IRIGENOL IRIGENOL 79321 54027 NPR3 4883 DRUGGABLE GENOME agonist 315661152 PL-3994 79322 54028 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SURAMIN SURAMIN 79325 54029 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US9670220, 77 79326 54030 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR agonist 348353672 79327 54031 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME anastrozole ANASTROZOLE 79328 54032 GGCX 2677 DRUGGABLE GENOME, ENZYME acenocoumarol ACENOCOUMAROL 25042728,25519826,24927344,29432897 79332 54033 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME EMETINE EMETINE 79333 54034 AKR1B1 231 DRUGGABLE GENOME, ENZYME inhibitor 178103976 TOLRESTAT 79336 54035 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE SB-203580 SB-203580 79339 54036 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Cethrin 79340 54037 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor DOVITINIB DOVITINIB 79341 54038 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Benzene sulfonamide derivative 8 79342 54039 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor PD0325901 PD-0325901 79344 54040 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 cisplatin CISPLATIN 22188361 79345 54041 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565859 PF-03715455 79347 54042 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor AT9283 AT-9283 79348 54043 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE 2-(4-ISOPROPYLPHENYL)BENZOTHIAZOLE CHEMBL1351908 79350 54044 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME CISPLATIN CISPLATIN 79352 54045 CD27 939 PROTEASE INHIBITOR, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Varlilumab VARLILUMAB 79353 54046 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1068 OXCARBAZEPINE 79354 54047 PIK3R4 30849 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor DACTOLISIB DACTOLISIB 79355 54048 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4803 CHEMBL585240 79356 54049 GJC1 10052 ION CHANNEL inhibitor 135652731 79358 54050 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME THIABENDAZOLE THIABENDAZOLE 79359 54051 UBE2I 7329 TRANSCRIPTION FACTOR BINDING, ENZYME irinotecan IRINOTECAN 19859084 79360 54052 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3707183 QUINIDINE SULFATE 79364 54053 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE MELPHALAN MELPHALAN 7923130 79365 54054 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME PF-562271 PF-00562271 79367 54055 HMGCR 3156 ENZYME, DRUGGABLE GENOME Cerivastatin CERIVASTATIN 79369 54056 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor AT9283 AT-9283 79371 54057 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-2906 CHEMBL579957 79373 54058 CSNK1E 1454 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, DNA REPAIR SB-202190 SB-202190 22951114 79374 54059 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR antagonist HGS 1029 79375 54060 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ETIPREDNOL DICLOACETATE 79376 54061 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE MEK INHIBITOR CI-1040 24504448 79379 54062 RRM1 6240 DRUGGABLE GENOME, ENZYME, DNA REPAIR FLUDARABINE FLUDARABINE 79380 54063 RAMP2 10266 DRUGGABLE GENOME, CELL SURFACE PRAMLINTIDE PRAMLINTIDE 79382 54064 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 404859079 79384 54065 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SU-6656 CHEMBL605003 79385 54066 PROS1 5627 DRUGGABLE GENOME warfarin WARFARIN 79386 54067 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE lapatinib LAPATINIB 25199759 79387 54068 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IODOMELATONIN IODOMELATONIN 79388 54069 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 7,12-DIMETHYL-BENZO[A]ANTHRACENE CHEMBL329673 79389 54070 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIDECAN-1-OL TRIDECAN-1-OL 79391 54071 PDE5A 8654 ENZYME, DRUGGABLE GENOME PENTOXIFYLLINE PENTOXIFYLLINE 79392 54072 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME TG-0054 BURIXAFOR 79393 54073 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME SIPLIZUMAB SIPLIZUMAB 79395 54074 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE THIOSEMICARBAZIDE THIOSEMICARBAZIDE 79397 54075 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NIGULDIPINE NIGULDIPINE 79401 54076 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE PACLITAXEL PACLITAXEL 22139083 79403 54077 ATXN2 6311 NA CANTHARIDIC_ACID CANTHARIDIC_ACID 79405 54078 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Ramucirumab RAMUCIRUMAB 25877855 79406 54079 COL11A2 1302 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 79407 54080 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TOMELUKAST TOMELUKAST 79409 54081 TXN 7295 DRUGGABLE GENOME, THIOREDOXIN PX-12 PX-12 79410 54082 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor 315661336 LUMINESPIB 79411 54083 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CID2350207 CHEMBL259615 79412 54084 SLC4A1 6521 ENZYME, TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME atenolol ATENOLOL 79413 54085 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR Ardeparin 79415 54086 KDM4A 9682 DRUGGABLE GENOME, ENZYME Hydroxamate analog 1 79417 54087 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR DORAMAPIMOD DORAMAPIMOD 79418 54088 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NIFEDIPINE NIFEDIPINE 22931300 79419 54089 CRBN 51185 ENZYME, DRUG RESISTANCE inhibitor CHEMBL848 LENALIDOMIDE 79420 54090 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SAPANISERTIB SAPANISERTIB 79422 54091 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE MK-2461 MK-2461 79423 54092 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR BENZALKONIUM CHLORIDE BENZALKONIUM CHLORIDE 79424 54093 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 178102328 PI-103 79426 54094 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Selumetinib SELUMETINIB 24939055,25870145,27287717,28416483,27312529 79427 54095 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR NSC-123414 CHEMBL16751 79429 54096 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178101318 79431 54097 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME UREA UREA 3223934 79432 54098 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 381118873 79433 54099 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SJ000143975 CHEMBL196585 79437 54100 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178101982 79439 54101 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE AT13148 AT-13148 22781553 79440 54102 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME DOXYLAMINE DOXYLAMINE 79441 54103 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ASTERRIC ACID ASTERRIC ACID 79442 54104 FAAH 2166 ENZYME, DRUGGABLE GENOME Carbamate derivative 17 79443 54105 ATP1A1 476 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER, ENZYME, CLINICALLY ACTIONABLE OUABAIN OUABAIN 79444 54106 GBA 2629 DRUGGABLE GENOME, ENZYME (S)-FLUOXETINE CHEMBL1169388 79445 54107 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CENISERTIB CENISERTIB 79447 54108 STAG2 10735 CLINICALLY ACTIONABLE, DRUG RESISTANCE Vemurafenib VEMURAFENIB 27500726 79448 54109 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GLUTARAL GLUTARAL 79449 54110 GCH1 2643 ENZYME Guanine GUANINE 79450 54111 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR DS-3201 79451 54112 THRA 7067 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LEVOTHYROXINE LEVOTHYROXINE 79452 54113 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME EVEROLIMUS EVEROLIMUS 79453 54114 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Irinotecan IRINOTECAN 24042735,16707468,25714871,21325073 79455 54115 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TRICHOSTATIN TRICHOSTATIN 21055848,16921367,18054239,19966789,22280363,19385600 79456 54116 HSPA4 3308 NA FLUTICASONE PROPIONATE 9645591 79457 54117 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER INDOMETHACIN INDOMETHACIN 20455578 79458 54118 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 178102289 AST-487 79459 54119 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 135650177 DICLOFENAC 79460 54120 FAAH 2166 ENZYME, DRUGGABLE GENOME Pyrazole derivative 80 79462 54121 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor BAFETINIB BAFETINIB 79463 54122 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME CPC-250 79464 54123 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE AN-1792 79465 54124 SMN2 6607 DRUGGABLE GENOME FRENTIZOLE FRENTIZOLE 79466 54125 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Imatinib IMATINIB 79468 54126 MAT2A 4144 ENZYME AG-270 79470 54127 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME CYCLOSPORINE CYCLOSPORINE 22101135 79471 54128 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL1200794 OXYMORPHONE HYDROCHLORIDE 79472 54129 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650277 FLUPROSTENOL 79473 54130 PPOX 5498 DRUGGABLE GENOME, ENZYME givosiran GIVOSIRAN 79474 54131 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME TCMDC-123916 CHEMBL493863 79475 54132 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Dabrafenib DABRAFENIB 79478 54133 TLR7 51284 DRUGGABLE GENOME RESIQUIMOD RESIQUIMOD 24383475 79479 54134 MAPT 4137 DRUGGABLE GENOME SB-415286 CHEMBL322970 79480 54135 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DEXTROMETHORPHAN DEXTROMETHORPHAN 12151071 79481 54136 TLR7 51284 DRUGGABLE GENOME CPG 52364 79483 54137 MUC16 94025 DRUGGABLE GENOME BUSERELIN ACETATE 1533376 79484 54138 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GNF-PF-3257 CHEMBL601768 79488 54139 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR SJ000293754 CHEMBL486706 79489 54140 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE RESVERATROL RESVERATROL 79492 54141 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME VITAMIN A 15736054 79493 54142 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR OXIDOPAMINE OXIDOPAMINE 79495 54143 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE Imatinib IMATINIB 28514312 79496 54144 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME LY-2090314 LY-2090314 79497 54145 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NADOLOL NADOLOL 79498 54146 HSP90B1 7184 DRUGGABLE GENOME HS-110 VIAGENPUMATUCEL-L 79499 54147 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Tegaserod TEGASEROD 79500 54148 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL3039504 NINTEDANIB ESYLATE 79501 54149 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX Palovarotene PALOVAROTENE 79502 54150 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR N-(4-CARBOXYMETHENE)PHENYLPYRROLE CHEMBL258756 79503 54151 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE NSC-636948 CHEMBL1998001 79505 54152 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL285674 ESTAZOLAM 79506 54153 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE VORINOSTAT VORINOSTAT 19966789 79508 54154 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 385612234 79509 54155 PPP1R1B 84152 KINASE FLUOXETINE FLUOXETINE 17125745 79510 54156 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR THIAMINE CHLORIDE THIAMINE 79511 54157 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME FPA-008 79512 54158 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 79514 54159 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200569 CAFFEINE, CITRATED 79515 54160 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ESTRAMUSTINE ESTRAMUSTINE 79517 54161 GPR35 2859 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ZAPRINAST ZAPRINAST 22572579 79518 54162 FKBP5 2289 DRUGGABLE GENOME lithium LITHIUM 18597649,21449676,20709156,19676097,15565110,23733030,17467808 79520 54163 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SP-600125 SP-600125 79522 54164 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME GLABRONE GLABRONE 20022509 79524 54165 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Atiprimod ATIPRIMOD 79525 54166 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL1421 DASATINIB 79526 54167 DNER 92737 NA Quinazolinone derivative 5 79527 54168 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 385612226 79528 54169 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CGM097 CGM-097 27659046 79529 54170 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME CCNU LOMUSTINE 9393761 79530 54171 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE PLASMIN FIBRINOLYSIN, HUMAN 79531 54172 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE AMG900 AMG-900 79533 54173 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME WZ4002 25870145 79535 54174 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME blocker 135652747 79536 54175 PSMD9 5715 NA inhibitor CARFILZOMIB CARFILZOMIB 79537 54176 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE SUNITINIB SUNITINIB 79538 54177 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING PHENYLBUTYRYLHYDROXAMIC ACID PHENYLBUTYRYLHYDROXAMIC ACID 21874153 79539 54178 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565639 GOLVATINIB 79540 54179 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 404859098 SAMIDORPHAN 79544 54180 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL451887 CARFILZOMIB 79547 54181 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OMEPRAZOLE OMEPRAZOLE 22931300 79549 54182 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME 4-amino-3,5-di-substituted-thiazole derivative 1 79550 54183 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE OP449 26563471 79556 54184 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME BENZO[D]ISOTHIAZOL-3-ONE CHEMBL297304 79557 54185 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NICLOSAMIDE NICLOSAMIDE 79558 54186 PSMA4 5685 DRUGGABLE GENOME, PROTEASE cotinine COTININE 79560 54187 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Reovirus 79561 54188 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Isoflavone derivative 6 79562 54189 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LEVODOPA LEVODOPA 79563 54190 MPHOSPH8 54737 NA PERPHENAZINE PERPHENAZINE 79566 54191 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE SNS-314 SNS-314 79567 54192 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651487 79569 54193 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Lobeglitazone LOBEGLITAZONE 79570 54194 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME SF1126 25425962 79571 54195 FCER1G 2207 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE BENZYLPENICILLOYL POLYLYSINE 79572 54196 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650970 79573 54197 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 385612197 79574 54198 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135652085 79575 54199 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME bacampicillin BACAMPICILLIN 9609616 79577 54200 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME FURAMIDINE FURAMIDINE 79578 54201 MAPT 4137 DRUGGABLE GENOME 2,3-DIHYDROXY-4-METHOXY-4'-ETHOXYBENZOPHENONE 2,3-DIHYDROXY-4-METHOXY-4'-ETHOXYBENZOPHENONE 79581 54202 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME BEXAROTENE BEXAROTENE 79582 54203 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME THIRAM THIRAM 79583 54204 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE OTSGC-A24 79585 54205 SIRT5 23408 ENZYME SURAMIN SURAMIN 25818461,23195732 79586 54206 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Panitumumab PANITUMUMAB 26243863 79587 54207 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE CEDIRANIB CEDIRANIB 79589 54208 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING MECHLORETHAMINE HYDROCHLORIDE MECHLORETHAMINE HYDROCHLORIDE 79590 54209 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 363894211 PEXMETINIB 79591 54210 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME LARGAZOLE LARGAZOLE 21420302,25203782,20491440 79592 54211 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR Platinum compounds 19786980,22188361,18347182,21902499,25069034,21057378,29662106,19362955,23962907,19203783,27498158,21262916,28796378,22026922,22329723 79593 54212 FGG 2266 DRUGGABLE GENOME, FIBRINOGEN, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE abciximab ABCIXIMAB 20938371 79594 54213 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR TICARCILLIN TICARCILLIN 7875147 79595 54214 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE SOMATROPIN SOMATROPIN 79597 54215 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CID 1245272 CHEMBL408850 79599 54216 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PHA-767491 CHEMBL225519 18469809 79601 54217 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME AMIODARONE AMIODARONE 79603 54218 SPR 6697 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME antagonist CHEMBL206253 NETUPITANT 79604 54219 DES 1674 NA THROMBIN THROMBIN 3040412 79605 54220 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PHENAMIL METHANESULFONATE PHENAMIL METHANESULFONATE 79606 54221 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 252827451 SAR-260301 79607 54222 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SML-10-70-1 24259466 79608 54223 MPHOSPH8 54737 NA GBR-12909 VANOXERINE 79609 54224 MEN1 4221 CLINICALLY ACTIONABLE, DNA REPAIR NITROBLUE TETRAZOLIUM NITROBLUE TETRAZOLIUM 79611 54225 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR PIOGLITAZONE PIOGLITAZONE 17407709 79612 54226 MAPT 4137 DRUGGABLE GENOME CISPLATIN CISPLATIN 79613 54227 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL513 CARMUSTINE 79614 54228 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 252166901 79615 54229 NPR3 4883 DRUGGABLE GENOME NESIRITIDE NESIRITIDE 79618 54230 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650290 79619 54231 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 3-HYDROXYCOUMARIN 3-HYDROXYCOUMARIN 79621 54232 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME BUTANOIC ACID BUTANOIC ACID 19053749 79622 54233 BAZ2B 29994 NA LOMOFUNGIN LOMOFUNGIN 79625 54234 PDE3A 5139 ENZYME, DRUGGABLE GENOME Milrinone MILRINONE 79626 54235 HDAC11 79885 DRUGGABLE GENOME, ENZYME VALPROIC ACID VALPROIC ACID 18294844,16921367,25304896 79628 54236 GHRL 51738 DRUGGABLE GENOME EPINEPHRINE EPINEPHRINE 16527847 79629 54237 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME SGN-70 79630 54238 MPHOSPH8 54737 NA S-(P-AZIDOPHENACYL)GLUTATHIONE CHEMBL1256813 79631 54239 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DNDI1417719 CHEMBL1420370 79632 54240 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL395429 OXYTOCIN 79633 54241 PRLR 5618 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, KINASE Endostatin ENDOSTATIN 79634 54242 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RETINAL RETINAL 79635 54243 F2RL1 2150 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE, ENZYME agonist 178100605 79636 54244 ALDH1A1 216 DRUGGABLE GENOME, ENZYME GNF-PF-2298 CHEMBL578905 79637 54245 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR GW0742 CHEMBL38508 79638 54246 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE TST10088 79639 54247 RGS4 5999 DRUGGABLE GENOME SANGUINARIUM SANGUINARIUM 79640 54248 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-C1 79642 54249 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE PACLITAXEL PACLITAXEL 12684687 79643 54250 COMT 1312 DRUGGABLE GENOME, ENZYME venlafaxine VENLAFAXINE 22417933,28627776,23706899 79646 54251 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL109648 CLAZOSENTAN 79650 54252 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER rocuronium ROCURONIUM 25279974 79652 54253 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 178102622 KENPAULLONE 79653 54254 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE inhibitor 252827422 79655 54255 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIPERONYL BUTOXIDE PIPERONYL BUTOXIDE 79660 54256 TARDBP 23435 TUMOR SUPPRESSOR ENILCONAZOLE ENILCONAZOLE 79661 54257 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME MK-3102 OMARIGLIPTIN 79663 54258 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BORTEZOMIB BORTEZOMIB 79665 54259 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME MEK162 BINIMETINIB 79667 54260 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ALMOTRIPTAN ALMOTRIPTAN 79672 54261 HTT 3064 DRUGGABLE GENOME GNF-PF-1947 CHEMBL585591 79673 54262 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4279 CHEMBL601320 79680 54263 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SB-203580 SB-203580 79683 54264 COMT 1312 DRUGGABLE GENOME, ENZYME bupropion BUPROPION 16876132 79685 54265 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor AS703569 CENISERTIB 79686 54266 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME SNS-032 BMS-387032 79688 54267 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ALITRETINOIN ALITRETINOIN 79689 54268 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2364605 CEBRANOPADOL 79690 54269 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL3330650 RG-7420 79691 54270 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201539 INSULIN PORK 79692 54271 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-32 79693 54272 TXNRD1 7296 DRUGGABLE GENOME Golden phosphorous acetyletic compound 3 79694 54273 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX BROMOPYROGALLOL RED BROMOPYROGALLOL RED 16759101 79695 54274 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING TRIFLUPROMAZINE HYDROCHLORIDE TRIFLUPROMAZINE HYDROCHLORIDE 79699 54275 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME FOLFIRI 28404754,25877855,25605843 79702 54276 SULT2B1 6820 ENZYME, DRUGGABLE GENOME fludarabine FLUDARABINE 22584460 79703 54277 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Carbamide derivative 14 79705 54278 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Aminopiperidine derivative 1 79706 54279 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 381118858 79708 54280 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME OXALIPLATIN OXALIPLATIN 19571295,19603024 79709 54281 MAOB 4129 DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 22071524 79712 54282 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE tianeptine TIANEPTINE 79713 54283 PRKACB 5567 ENZYME, KINASE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL494089 GSK-690693 79715 54284 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME WORTMANNIN WORTMANNIN 79716 54285 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR VEGF 15930297 79717 54286 AGT 183 ENZYME, DRUGGABLE GENOME, PROTEASE INHIBITOR, G PROTEIN COUPLED RECEPTOR, HORMONE ACTIVITY, GROWTH FACTOR ENALAPRIL ENALAPRIL 11928713 79718 54287 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178103661 HYDROMORPHONE 79720 54288 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NSC-81747 CHEMBL1371696 79721 54289 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ivosidenib IVOSIDENIB 79722 54290 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DIBUTYLDICHLOROSTANNANE DIBUTYLDICHLOROSTANNANE 79723 54291 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DNR 11368357 79725 54292 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME HELENALIN HELENALIN 79726 54293 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL552212 LEXIBULIN 79727 54294 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME 7-ETHYL-10-HYDROXY-CAMPTOTHECIN 7-ETHYL-10-HYDROXYCAMPTOTHECIN 23622981 79733 54295 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TDR77585 CHEMBL1333386 79734 54296 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Cyclic sulfonamide derivative 4 79735 54297 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GLAUCINE METHIODIDE GLAUCINE METHIODIDE 79738 54298 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Estropipate ESTROPIPATE 79740 54299 ANKS1B 56899 NA heroin DIACETYLMORPHINE 31462767 79741 54300 GBA 2629 DRUGGABLE GENOME, ENZYME AMBROXOL AMBROXOL 22762530 79742 54301 MAPT 4137 DRUGGABLE GENOME TRICETIN TRICETIN 79743 54302 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 TCMDC-124336 CHEMBL527271 79748 54303 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME bevacizumab BEVACIZUMAB 27139155 79749 54304 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BROMOENOL LACTONE BROMOENOL LACTONE 79750 54305 CBX1 10951 NA 4-HYDROXYESTRADIOL CHEMBL1412489 79751 54306 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PANOBINOSTAT PANOBINOSTAT 79752 54307 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Sorafenib SORAFENIB 23629727 79753 54308 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 384403666 79756 54309 BAZ2B 29994 NA SJ000032149 CHEMBL600778 79757 54310 HBB 3043 DRUGGABLE GENOME, ENZYME PHENAZOPYRIDINE HYDROCHLORIDE PHENAZOPYRIDINE HYDROCHLORIDE 79758 54311 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 OLVANIL OLVANIL 79761 54312 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE erythromycin ERYTHROMYCIN 79762 54313 SMN1 6606 DRUGGABLE GENOME 2-(4-NITROBENZYLSULFANYL)BENZOXAZOLE CHEMBL412603 79763 54314 MAPT 4137 DRUGGABLE GENOME METHYLENE BLUE METHYLENE BLUE 79764 54315 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Vemurafenib VEMURAFENIB 79766 54316 DUT 1854 ENZYME, DRUGGABLE GENOME TAS-114 79768 54317 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME FRAXIDIN METHYL ETHER FRAXIDIN METHYL ETHER 79769 54318 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 79770 54319 POLK 51426 DNA REPAIR, ENZYME AMINOQUINURIDE AMINOQUINURIDE 79772 54320 CMPK1 51727 KINASE, ENZYME gemcitabine GEMCITABINE 21642870,22838949,22838950,24361227 79773 54321 SLC28A1 9154 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE IL-6 15464233 79774 54322 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR P-CYANOCHALCONE CHEMBL445153 79775 54323 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE Ceritinib CERITINIB 27009859,25749034,25421750 79776 54324 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL2368861 BUPRENORPHINE HYDROCHLORIDE 79777 54325 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SB-202190 SB-202190 22951114 79778 54326 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200967 BROMODIPHENHYDRAMINE HYDROCHLORIDE 79779 54327 GLS 2744 ENZYME DICLOXACILLIN DICLOXACILLIN 79782 54328 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME PHENOXODIOL 79784 54329 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER doxorubicin DOXORUBICIN 29938344,22016816,25637052,18377430,25582575,18408561 79785 54330 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-123904 CHEMBL586061 79787 54331 GLS 2744 ENZYME inhibitor 315661138 TELAGLENASTAT 79789 54332 CALR 811 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME N/A 26697989,25873496,26071474,26449662 79790 54333 GLS 2744 ENZYME TETROQUINONE TETROQUINONE 79791 54334 ATAD5 79915 NA CINOBUFAGIN CINOBUFAGIN 79792 54335 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE 681640 CHEMBL379975 79793 54336 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME FLUOCINONIDE FLUOCINONIDE 79794 54337 ATAD5 79915 NA TCMDC-123781 CHEMBL581194 79795 54338 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-1549 CHEMBL227959 79796 54339 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ALX-0651 20864805 79797 54340 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE MSC2363318A MSC-2363318A 27186432 79798 54341 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL2107313 BECATECARIN 79800 54342 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE AXITINIB AXITINIB 79801 54343 ALPL 249 ENZYME, DRUGGABLE GENOME GNF-PF-3148 CHEMBL81782 79802 54344 ITPR1 3708 ION CHANNEL, KINASE, DRUGGABLE GENOME, TRANSPORTER Nitroprusside NITROPRUSSIDE 79803 54345 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565859 PF-03715455 79805 54346 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Nintedanib NINTEDANIB 22238366 79807 54347 MAPT 4137 DRUGGABLE GENOME AGROCLAVINE AGROCLAVINE 79808 54348 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ATROPINE METHYL BROMIDE ATROPINE METHYLBROMIDE 79809 54349 CDK12 51755 KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR, SERINE THREONINE KINASE inhibitor CHEMBL488436 AZD-5438 79810 54350 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DACTHAL DACTHAL 79811 54351 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR JNJ-7706621 JNJ-7706621 79812 54352 ZNF134 7693 NA methylphenidate METHYLPHENIDATE 29382897 79813 54353 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CYSTEINE METHYL-ESTER HCL CHEMBL1426508 79815 54354 STK38 11329 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565889 79816 54355 TNFRSF1B 7133 DRUGGABLE GENOME STAVUDINE STAVUDINE 9430255 79817 54356 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor VELIPARIB VELIPARIB 79818 54357 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PSAMMAPLIN A PSAMMAPLIN A 16643023 79819 54358 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME MIP-1 ALPHA 9176534 79821 54359 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR HINOKITIOL HINOKITIOL 79822 54360 GLS 2744 ENZYME EMODIC ACID EMODIC ACID 79823 54361 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 223366170 NS-018 79824 54362 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE MEDI4736 DURVALUMAB 79825 54363 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME trichloroethylene TRICHLOROETHYLENE 79828 54364 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-4967 CHEMBL585827 79829 54365 FN1 2335 DRUGGABLE GENOME L19-TNF-alpha 79830 54366 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISRADIPINE ISRADIPINE 79832 54367 PKM 5315 ENZYME, KINASE, DRUGGABLE GENOME ERBSTATIN ERBSTATIN 79833 54368 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Roscovitine derivative 1 79834 54369 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL861 MEPHENYTOIN 79836 54370 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-23 79839 54371 RACGAP1 29127 NA TCMDC-123916 CHEMBL493863 79840 54372 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PIMETHIXENE MALEATE PIMETHIXENE MALEATE 79842 54373 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR CENISERTIB CENISERTIB 79846 54374 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DIGITOXIGENIN DIGITOXIGENIN 79848 54375 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME VALRUBICIN VALRUBICIN 79850 54376 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Fenoterol FENOTEROL 79852 54377 ALB 213 TRANSPORTER, DRUGGABLE GENOME N-TRIFLUOROACETYLHOMOCYSTEINE THIOLACTONE CHEMBL1945287 21632244 79853 54378 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-49 79854 54379 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE 178101727 79855 54380 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR PENICILLAMINE PENICILLAMINE 11526215 79856 54381 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR DONEPEZIL DONEPEZIL 17990049 79857 54382 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor CHEMBL1213490 ROMIDEPSIN 79858 54383 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME N-METHYLANTHRANILIC ACID N-METHYLANTHRANILIC ACID 79859 54384 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE GW843682X GW843682X 79860 54385 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649828 79861 54386 NPM1 4869 CLINICALLY ACTIONABLE, DNA REPAIR, DRUGGABLE GENOME, DRUG RESISTANCE AP26113 CHEMBL3397300 27009859,25749034,25421750,27780853 79862 54387 ETV6 2120 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE Altiratinib ALTIRATINIB 79865 54388 PSMD1 5707 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 79866 54389 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor PKI-587 GEDATOLISIB 79868 54390 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL3545207 EVENAMIDE 79869 54391 MMP13 4322 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 252166836 79870 54392 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 374883876 79871 54393 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME antipsychotics 20031235 79872 54394 TUBA3D 113457 DRUGGABLE GENOME inhibitor CHEMBL1742994 BRENTUXIMAB VEDOTIN 79875 54395 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE PMID25726713-Compound-51 79876 54396 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE THALIDOMIDE THALIDOMIDE 11838958 79877 54397 GLS 2744 ENZYME PMID30273516-Compound-22a 79878 54398 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PMID27774824-Compound-Figure6Example6 79879 54399 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR PROGESTERONE PROGESTERONE 19883083 79880 54400 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 135650147 79881 54401 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist 178100976 SELFOTEL 79882 54402 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME lamivudine / abacavir 79883 54403 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 135652594 79884 54404 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PF-00734200 GOSOGLIPTIN 79885 54405 GSTA1 2938 ENZYME, DRUGGABLE GENOME PHENOBARBITAL PHENOBARBITAL 16608922 79887 54406 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 79888 54407 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME 4-(4-AMINOPHENYL)BUTANOIC ACID CHEMBL1650245 24044874 79889 54408 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Pyrazole derivative 63 79890 54409 CES1 1066 DRUGGABLE GENOME, ENZYME methylphenidate METHYLPHENIDATE 19733552 79891 54410 ATXN2 6311 NA ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 79892 54411 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ACRIFLAVINE CHLORIDE ACRIFLAVINE 79894 54412 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME AMG 211 79895 54413 ALOX15 246 ENZYME, DRUGGABLE GENOME 5,7-DIHYDROXYISOFLAVONE 5,7-DIHYDROXYISOFLAVONE 79897 54414 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR TAS-116 TAS-116 79898 54415 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL3544935 XL-418 79899 54416 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CEPHALOTHIN SODIUM CEPHALOTHIN SODIUM 79900 54417 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ERGOTAMINE ERGOTAMINE 79902 54418 SLITRK6 84189 CELL SURFACE ASG-15ME 79904 54419 GFRA1 2674 KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE ANTISENSE OLIGONUCLEOTIDES 11079571 79905 54420 PSMA2 5683 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL325041 BORTEZOMIB 79907 54421 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ABT-263 NAVITOCLAX 27659046 79908 54422 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR JQEZ5 27312177 79909 54423 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 178101303 CANAGLIFLOZIN 79910 54424 PTGS1 5742 ENZYME, DRUGGABLE GENOME MECLOFENAMIC ACID 79911 54425 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME PENTAMIDINE ISETHIONATE PENTAMIDINE ISETHIONATE 79913 54426 PKN2 5586 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE inhibitor 249565864 79915 54427 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR etanercept ETANERCEPT 24253594 79917 54428 UGT2B7 7364 DRUGGABLE GENOME valproic acid 21806385,17687269,27406852,23099353,29243113 79918 54429 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor 178103007 BORTEZOMIB 79919 54430 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-5510 CHEMBL578741 79920 54431 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651293 79921 54432 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL inhibitor 178102359 79922 54433 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME 22(S)-HYDROXYCHOLESTEROL CHEMBL1243244 24480357,24268541 79923 54434 APOE 348 DRUGGABLE GENOME CN-105 79924 54435 IL1RN 3557 DRUGGABLE GENOME MTX METHOTREXATE 8877917 79926 54436 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135652580 79929 54437 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME CATECHOL CATECHOL 79930 54438 PI4K2B 55300 ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, KINASE inhibitor 135651426 ADENOSINE 79932 54439 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TEMSIROLIMUS TEMSIROLIMUS 79933 54440 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Sunitinib SUNITINIB 79934 54441 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545005 PLX-8394 79935 54442 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Pyrimidinyl compound 3 79937 54443 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TAK-632 27523909 79938 54444 TUBB6 84617 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 16539377,21664138,23916255 79939 54445 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR UROKINASE-TYPE PLASMINOGEN ACTIVATOR 11865026 79941 54446 PTGES 9536 DRUGGABLE GENOME, ENZYME Phthalazinone derivative 1 79942 54447 PRKG1 5592 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME PHA-767491 CHEMBL225519 79943 54448 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 79946 54449 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME CHEMBL2364609 ESKETAMINE HYDROCHLORIDE 79947 54450 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE CETUXIMAB CETUXIMAB 17704420 79948 54451 HSPB1 3315 DRUGGABLE GENOME NOCODAZOLE NOCODAZOLE 22435708 79949 54452 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 zonisamide ZONISAMIDE 9187528 79950 54453 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 354702292 79951 54454 CXCL2 2920 DRUGGABLE GENOME TPA ALTEPLASE 18199827 79954 54455 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ZM-241385 ZM-241385 79956 54456 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178100984 79957 54457 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL24828 VANDETANIB 79958 54458 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR INDOPROFEN INDOPROFEN 79959 54459 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHEMOPREVENTIVE 15901726,16513647 79961 54460 RAB9A 9367 ENZYME, DRUGGABLE GENOME NSC-50690 CHEMBL1388703 79965 54461 PTGS2 5743 DRUGGABLE GENOME, ENZYME celecoxib CELECOXIB 22336956,19602986 79969 54462 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Geminally-substituted cyanoethylpypazolo pyridone derivative 1 79970 54463 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 310264699 SAMOTOLISIB 79971 54464 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Triazole derivative 1 79972 54465 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Larotrectinib LAROTRECTINIB 79974 54466 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NICLOSAMIDE NICLOSAMIDE 79975 54467 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER irinotecan IRINOTECAN 23478653 79978 54468 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SAPPANONE A TRIMETHYL ETHER SAPPANONE A TRIMETHYL ETHER 79979 54469 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE RU-56187 CHEMBL1099140 20381361 79981 54470 ATAD5 79915 NA 2-METHOXY-1,4-NAPHTHOQUINONE 2-METHOXY-1,4-NAPHTHOQUINONE 79982 54471 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE MM-141 ISTIRATUMAB 79983 54472 ALPL 249 ENZYME, DRUGGABLE GENOME (-)-EPICATECHIN (-)-EPICATECHIN 79984 54473 CYSLTR2 57105 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100420 79985 54474 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 315661265 79987 54475 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PROTOPORPHYRIN PROTOPORPHYRIN 79988 54476 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-1852 CHEMBL533293 79989 54477 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Antibodie derivative 8 79990 54478 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE C-1311 C-1311 79991 54479 TNNC1 7134 DRUGGABLE GENOME NSC-107022 CHEMBL1601846 79992 54480 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR TRIFLUOPERAZINE TRIFLUOPERAZINE 1690578 79994 54481 GMNN 51053 DRUGGABLE GENOME LANATOSIDE C LANATOSIDE C 79995 54482 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME Dipeptide analog 3 79996 54483 CLK1 1195 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE TG003 79998 54484 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Rucaparib RUCAPARIB 79999 54485 HTT 3064 DRUGGABLE GENOME GNF-PF-1509 CHEMBL576412 80000 54486 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING SANGIVAMYCIN SANGIVAMYCIN 17371872 80001 54487 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TRICLOFENOL TRICLOFENOL 80002 54488 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER GINKGO BILOBA 15577230 80003 54489 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PROCYMIDONE PROCYMIDONE 80004 54490 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CUDC-101 CUDC-101 25107918 80005 54491 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 80006 54492 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-699479 CHEMBL1701915 80007 54493 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE BMS-754807 BMS-754807 19778024 80008 54494 GMNN 51053 DRUGGABLE GENOME GNF-PF-3582 CHEMBL606167 80009 54495 ATAD5 79915 NA TCMDC-123641 CHEMBL532849 80011 54496 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME FARGLITAZAR FARGLITAZAR 80012 54497 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NOT DISCLOSED 80013 54498 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor DACTOLISIB DACTOLISIB 80014 54499 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 rifampin RIFAMPIN 24839948 80015 54500 COL4A6 1288 DRUGGABLE GENOME CHEMBL2108709 COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 80017 54501 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ENU 12963544 80018 54502 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Peptide analog 46 80020 54503 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR PREXASERTIB PREXASERTIB 28490518 80021 54504 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE PD 0332991 80023 54505 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME SB-204741 CHEMBL323356 80024 54506 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ER2 27040853 80026 54507 GMNN 51053 DRUGGABLE GENOME LOMERIZINE LOMERIZINE 80027 54508 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROSULTIAMINE PROSULTIAMINE 80028 54509 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 80029 54510 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ZM-39923 HCL CHEMBL538798 80030 54511 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CHLOROTHALONIL CHLOROTHALONIL 80031 54512 VNN1 8876 ENZYME inhibitor 381118911 80032 54513 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 178102910 80033 54514 HYOU1 10525 DRUGGABLE GENOME DABIGATRAN DABIGATRAN 22494098 80034 54515 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Temsirolimus TEMSIROLIMUS 21216929,26725216,27016228 80036 54516 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Epinephrine EPINEPHRINE 80037 54517 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR GNF-PF-1919 CHEMBL576409 80038 54518 HLA-DPB1 3115 CELL SURFACE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE aspirin ASPIRIN 15007363,15784113,19392989,9179433 80039 54519 HRH4 59340 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1915540 PF-03893787 80040 54520 GABBR1 2550 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR LESOGABERAN LESOGABERAN 80041 54521 CTSD 1509 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178103155 80042 54522 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SULINDAC SULINDAC 22931300 80044 54523 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ERYTHROMYCIN ERYTHROMYCIN 21393461 80045 54524 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 178103847 PIROXICAM 80046 54525 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME RESVERATROL RESVERATROL 80051 54526 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME PENTABROMOPHENOL PENTABROMOPHENOL 80053 54527 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TESTOSTERONE TESTOSTERONE 80056 54528 DUSP1 1843 PROTEIN PHOSPHATASE, KINASE, DRUGGABLE GENOME ANTISENSE OLIGONUCLEOTIDES 11988488 80057 54529 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL1614701 SELUMETINIB 80059 54530 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Pyrrole six-membered heteroaryl ring derivative 1 80060 54531 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CHEMBL1743000 CITATUZUMAB BOGATOX 80061 54532 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL565 CLOFIBRATE 80063 54533 TNK1 8711 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 363894223 80065 54534 IL11 3589 DRUGGABLE GENOME, KINASE, GROWTH FACTOR DOXORUBICIN DOXORUBICIN 9363868 80066 54535 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLOROACETIC ACID CHLOROACETIC ACID 80068 54536 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Ixabepilone IXABEPILONE 80070 54537 FFAR4 338557 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650341 GW9508 80071 54538 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME 5-BENZYLOXYTRYPTAMINE 5-BENZYLOXYTRYPTAMINE 80072 54539 P4HB 5034 THIOREDOXIN, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE NSC-19803 CHEMBL522983 80074 54540 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3039502 DUVELISIB 80077 54541 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE HYCANTHONE HYCANTHONE 80078 54542 GPC3 2719 DRUGGABLE GENOME, CELL SURFACE, CLINICALLY ACTIONABLE antibody 252166616 CODRITUZUMAB 80082 54543 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Efungumab EFUNGUMAB 80083 54544 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE 2'H,4H-[2,5'-BICHROMEN]-4-ONE 2'H,4H-[2,5'-BICHROMEN]-4-ONE 23600958 80084 54545 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME AMPICILLIN TRIHYDRATE AMPICILLIN TRIHYDRATE 80085 54546 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 2,7-BIS[3-(PYRROLIDINO)PROPIONAMIDO]ANTHRAQUINONE CHEMBL144757 18571928 80086 54547 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GNF-PF-4097 CHEMBL597246 80087 54548 ATXN2 6311 NA LOBARIC ACID LOBARIC ACID 80088 54549 IL23A 51561 DRUGGABLE GENOME inhibitor CHEMBL2364648 GUSELKUMAB 80089 54550 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Sorafenib SORAFENIB 23629727,26743856,23224737,26307133,25294897,27480147,25363205 80090 54551 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR BORTEZOMIB BORTEZOMIB 16357160 80091 54552 XPO1 7514 CLINICALLY ACTIONABLE, KINASE OSTHOLE OSTHOLE 20493693 80092 54553 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME antagonist CHEMBL3707355 AZD8108 80093 54554 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE BMS-986020 BMS-986020 80094 54555 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor 354702249 DIFAMILAST 80097 54556 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Clomipramine CLOMIPRAMINE 80098 54557 WNK1 65125 SERINE THREONINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE, DRUGGABLE GENOME, ENZYME hydrochlorothiazide HYDROCHLOROTHIAZIDE 18591455 80103 54558 HLA-B 3106 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME zidovudine / lamivudine / abacavir 80106 54559 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME OXYTETRACYCLINE OXYTETRACYCLINE 80108 54560 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PMID25656651-Compound-21b 80109 54561 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL CHEMBL1257 ENFLURANE 80110 54562 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 404859099 OXYCODEGOL 80111 54563 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE ETRAVIRINE ETRAVIRINE 21189339 80112 54564 SIRT3 23410 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME NIACINAMIDE NIACINAMIDE 22835719 80113 54565 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME AM-101 ESKETAMINE HYDROCHLORIDE 80115 54566 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME LISSOCLINIDINE B LISSOCLINIDINE B 18977148 80116 54567 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DOVITINIB DOVITINIB 80117 54568 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE PMID25726713-Compound-50 80118 54569 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NALBUPHINE NALBUPHINE 22931300 80120 54570 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AUY922 25870087 80121 54571 POLI 11201 DNA REPAIR METHOTREXATE METHOTREXATE 80122 54572 IL1B 3553 KINASE, DRUGGABLE GENOME Glucosamine GLUCOSAMINE 80123 54573 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-12 80124 54574 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME COAGULATION FACTOR IX 80125 54575 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650232 ENPROSTIL 80126 54576 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 310264733 FIMEPINOSTAT 80129 54577 DNMT3A 1788 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL1489 AZACITIDINE 80132 54578 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME CA19-9 10773785 80133 54579 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE inhibitor 178101905 MARIMASTAT 80134 54580 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME BITHIONOLATE SODIUM BITHIONOLATE SODIUM 80136 54581 MAPT 4137 DRUGGABLE GENOME CHLORANIL CHLORANIL 80138 54582 TLR7 51284 DRUGGABLE GENOME PF-4878691 CPG-52852 80139 54583 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HOE-33342 CHEMBL343002 80140 54584 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Tamoxifen TAMOXIFEN 80143 54585 POLI 11201 DNA REPAIR GNF-PF-1852 CHEMBL533293 80144 54586 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-37031 CHEMBL222993 80145 54587 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR DEXTRAN SULFATE SODIUM 17365404 80147 54588 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Metformin METFORMIN 28375706 80148 54589 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ISOVELLERAL ISOVELLERAL 80149 54590 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PEMIGATINIB PEMIGATINIB 32203698 80150 54591 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME AG-538 CHEMBL56393 80151 54592 ABCC5 10057 DRUGGABLE GENOME, ABC TRANSPORTER, TRANSPORTER glibenclamide GLYBURIDE 27403931 80152 54593 CBX1 10951 NA BAY-11-7085 BAY-11-7085 80154 54594 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME agonist CHEMBL1201567 FILGRASTIM 80155 54595 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DACTINOMYCIN DACTINOMYCIN 22931300 80156 54596 POLI 11201 DNA REPAIR ISOKAEMPFERIDE ISOKAEMPFERIDE 80157 54597 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PACLITAXEL PACLITAXEL 24065105 80158 54598 CD74 972 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE antibody MILATUZUMAB MILATUZUMAB 80159 54599 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PW12 22391131 80161 54600 FIP1L1 81608 CLINICALLY ACTIONABLE, KINASE imatinib IMATINIB 24433361 80162 54601 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER LOPINAVIR LOPINAVIR 17664327 80168 54602 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR ZEARALENONE ZEARALENONE 80169 54603 F13A1 2162 DRUGGABLE GENOME, ENZYME aspirin ASPIRIN 12515735 80171 54604 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER MK-8242 28240971 80172 54605 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 2-BROMO-HEXADECANOIC ACID CHEMBL118417 80173 54606 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor CHEMBL462018 TRICIRIBINE PHOSPHATE 80175 54607 CA12 771 DRUGGABLE GENOME TRIFLUOROMETHANESULFONAMIDE TRIFLUOROMETHANESULFONAMIDE 23159038 80176 54608 PDE4A 5141 DRUGGABLE GENOME, ENZYME AWD-12-281 80177 54609 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-3501 CHEMBL581910 80178 54610 NCAM1 4684 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CD56-specific gene-engineered T cells 80179 54611 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME atenolol ATENOLOL 15188945 80180 54612 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ISOBUTYLMETHYLXANTHINE ISOBUTYLMETHYLXANTHINE 80181 54613 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651060 80182 54614 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1229517 VEMURAFENIB 80185 54615 SLC28A2 9153 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, DRUGGABLE GENOME THYMIDINE THYMIDINE 11602688 80187 54616 HTT 3064 DRUGGABLE GENOME SJ000154295 CHEMBL578502 80188 54617 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME agonist 178100991 (D)-SERINE 80189 54618 ANGPT2 285 KINASE, FIBRINOGEN, DRUGGABLE GENOME antibody CVX-060 80190 54619 CTNNB1 1499 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, DRUG RESISTANCE Recombinant human endostatin 80191 54620 POLK 51426 DNA REPAIR, ENZYME NSC-348401 CHEMBL515505 80192 54621 GLS 2744 ENZYME CARBENICILLIN INDANYL CARBENICILLIN INDANYL 80193 54622 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1387 NORETHYNODREL 80194 54623 UGT1A6 54578 ENZYME, DRUGGABLE GENOME deferiprone DEFERIPRONE 24036429 80195 54624 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME tositumomab TOSITUMOMAB 80197 54625 ALPI 248 DRUGGABLE GENOME, ENZYME DIHYDRODAPHNODORIN B DIHYDRODAPHNODORIN B 80198 54626 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR HEXACHLOROPHENE HEXACHLOROPHENE 80200 54627 MUC16 94025 DRUGGABLE GENOME Abagovomab ABAGOVOMAB 80201 54628 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DICHLORISONE ACETATE DICHLORISONE ACETATE 80202 54629 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-5217 CHEMBL601970 80203 54630 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist 53801005 80204 54631 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR 6EP 80206 54632 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE TPA ALTEPLASE 8615653 80208 54633 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-31 80210 54634 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CIANIDANOL CIANIDANOL 80211 54635 BRCA2 675 CLINICALLY ACTIONABLE AZD6738 CERALASERTIB 28062704 80212 54636 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Procysteine PROCYSTEINE 80213 54637 POLI 11201 DNA REPAIR SJ000082806 CHEMBL494668 80214 54638 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE EPHEDRINE SULFATE EPHEDRINE SULFATE 80215 54639 NOS2 4843 DRUGGABLE GENOME, ENZYME isoniazid ISONIAZID 22341855 80216 54640 KDM4A 9682 DRUGGABLE GENOME, ENZYME AG-555 CHEMBL53898 80218 54641 TNNT1 7138 NA TIRAMSETIV 80219 54642 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565894 80220 54643 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651539 DINOPROSTONE 80221 54644 CDC42BPA 8476 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565877 80223 54645 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PROPACHLOR PROPACHLOR 80224 54646 BHLHE40 8553 NA RETINOIC ACID 10737769 80226 54647 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR AMCINONIDE AMCINONIDE 80228 54648 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL608533 MIDOSTAURIN 80229 54649 MAPT 4137 DRUGGABLE GENOME TANSHINONE I TANSHINONE I 80230 54650 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Hydoxyamidine derivative 1 80231 54651 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PSORALEN PSORALEN 80232 54652 PSMB4 5692 DRUGGABLE GENOME, PROTEASE BORTEZOMIB BORTEZOMIB 24524217 80234 54653 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR inhibitor 178103605 80235 54654 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CERITINIB CERITINIB 26372962 80236 54655 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE agonist 135651702 80237 54656 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE 17-ALLYL-AMINOGELDANAMYCIN 16267832 80238 54657 ATXN2 6311 NA BAY-11-7085 BAY-11-7085 80240 54658 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE DACTOLISIB DACTOLISIB 19010894,23619167,19029981 80241 54659 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-228155 CHEMBL505670 80242 54660 TF 7018 CELL SURFACE, DRUGGABLE GENOME CALAA-01 80243 54661 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE ENZALUTAMIDE ENZALUTAMIDE 25544636 80244 54662 IFNG 3458 DRUGGABLE GENOME GLUCOCORTICOID 7543821 80246 54663 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHRYSENE-1,4-DIONE CHEMBL421215 80247 54664 MTTP 4547 DRUGGABLE GENOME SLX-4090 SLX-4090 80248 54665 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ACTINOMYCIN D 15883285 80249 54666 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000147784 CHEMBL590186 80250 54667 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME HUPERZINE-A 80251 54668 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HARMAN HARMAN 80253 54669 HDAC11 79885 DRUGGABLE GENOME, ENZYME PHENYLBUTYRYLHYDROXAMIC ACID PHENYLBUTYRYLHYDROXAMIC ACID 21874153 80254 54670 CA1 759 DRUGGABLE GENOME, ENZYME CHLOROTHIAZIDE CHLOROTHIAZIDE 80256 54671 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PI-88 MUPARFOSTAT 80257 54672 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE CC-223 CC-223 26177599 80258 54673 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 12 80259 54674 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR HEXACHLOROPHENE HEXACHLOROPHENE 80261 54675 KDM4A 9682 DRUGGABLE GENOME, ENZYME BENZOXAZOLINONE BENZOXAZOLINONE 80264 54676 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR INSULIN INSULIN 1698537 80267 54677 RGS4 5999 DRUGGABLE GENOME S-(P-AZIDOPHENACYL)GLUTATHIONE CHEMBL1256813 80270 54678 MPHOSPH8 54737 NA CGP-74514A CHEMBL1256911 80271 54679 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME GLPG0634 80272 54680 MAOA 4128 DRUGGABLE GENOME, ENZYME CX157 80273 54681 RAB9A 9367 ENZYME, DRUGGABLE GENOME RUTAECARPINE RUTAECARPINE 80274 54682 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 2,4-DIHYDROXYBENZOPHENONE 2,4-DIHYDROXYBENZOPHENONE 80275 54683 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE METHYL 7-DESHYDROXYPYROGALLIN-4-CARBOXYLATE 80277 54684 CALCRL 10203 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME AMG 334 80279 54685 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR DIMETHYLADENINE DIMETHYLADENINE 80280 54686 CBX1 10951 NA CYSTAMINE HYDROCHLORIDE CYSTAMINE HYDROCHLORIDE 80281 54687 IL18 3606 DRUGGABLE GENOME ANTIVIRAL 12559970 80285 54688 SMN1 6606 DRUGGABLE GENOME 2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE 2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE 80286 54689 ATXN2 6311 NA GNF-PF-4510 CHEMBL586024 80287 54690 SMN2 6607 DRUGGABLE GENOME BROXURIDINE BROXURIDINE 80288 54691 LNPEP 4012 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, TRANSPORTER, PROTEASE US10023583, Example 24 80289 54692 RRM2 6241 DRUGGABLE GENOME, ENZYME inhibitor 178103408 CLOFARABINE 80290 54693 RBP4 5950 DRUGGABLE GENOME US9434727, 153 80291 54694 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR DENSPM 12902979 80292 54695 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME modulator CHEMBL146506 MOFAROTENE 80294 54696 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME 8-MOP METHOXSALEN 3319774 80295 54697 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RAC-GONIOTHALAMIN CHEMBL1170485 80297 54698 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME INTERLEUKIN 2 80298 54699 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR TAMATINIB R-406 80299 54700 DGAT1 8694 ENZYME, DRUGGABLE GENOME Pyrazine carboxamide derivative 1 80300 54701 HSPB2 3316 KINASE VP-16 ETOPOSIDE PHOSPHATE 15911090 80301 54702 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR AZACITIDINE AZACITIDINE 80302 54703 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE TOPOTECAN TOPOTECAN 80303 54704 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 17 80304 54705 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor 178103458 VORINOSTAT 80305 54706 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NAPROXEN NAPROXEN 14691574 80306 54707 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE antagonist 135650770 80307 54708 HEBP1 50865 DRUGGABLE GENOME 4-(2-cyclohexylethoxy) aniline derivative 1 80308 54709 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CALMIDAZOLIUM CHLORIDE CALMIDAZOLIUM CHLORIDE 80309 54710 GMNN 51053 DRUGGABLE GENOME TCMDC-123641 CHEMBL532849 80310 54711 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ADJUVANT 17179731,15446556,14519634 80313 54712 CTLA4 1493 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME melphalan MELPHALAN 21228734 80315 54713 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CD123/CLL1 CAR-T Cells 80316 54714 CASP8 841 DRUGGABLE GENOME, PROTEASE, ENZYME, CLINICALLY ACTIONABLE 20(S)-PROTOPANAXADIOL CHEMBL375563 17261067 80317 54715 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102568 80318 54716 XDH 7498 DRUGGABLE GENOME, ENZYME Fused heterocyclic compound 1 80319 54717 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ACETALDEHYDE ACETALDEHYDE 80320 54718 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME PAZOPANIB PAZOPANIB 80321 54719 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME cyclosporine CYCLOSPORINE 80322 54720 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE 5-azolone derivative 1 80323 54721 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL3707355 AZD8108 80324 54722 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME inhibitor VELIPARIB VELIPARIB 80325 54723 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Antibodie derivative 3 80326 54724 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BCMA CAR T cells 80327 54725 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-3889 CHEMBL598270 80329 54726 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE antibody MM121 80330 54727 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GNF-PF-3276 CHEMBL582081 80331 54728 CDA 978 ENZYME, DRUGGABLE GENOME ARA-C 8791999,12008078 80333 54729 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR KB002 80336 54730 C5 727 PROTEASE INHIBITOR, DRUGGABLE GENOME, ENZYME ECULIZUMAB ECULIZUMAB 80337 54731 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE AV-203 AV-203 80338 54732 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PMA 11035812 80340 54733 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor CHEMBL1922094 APITOLISIB 80341 54734 MAPT 4137 DRUGGABLE GENOME OXYTETRACYCLINE OXYTETRACYCLINE 80343 54735 MAPT 4137 DRUGGABLE GENOME MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 80344 54736 KIF11 3832 DRUGGABLE GENOME DIMETHYLENASTRON DIMETHYLENASTRON 20138511 80345 54737 CHRNB1 1140 DRUGGABLE GENOME, ION CHANNEL, TRANSPORTER antagonist CHEMBL1200648 ROCURONIUM BROMIDE 80346 54738 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER IODOQUINOL IODOQUINOL 80347 54739 UCP2 7351 TRANSPORTER, DRUGGABLE GENOME CL-316,243 80349 54740 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Imatinib IMATINIB 80351 54741 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR OMEPRAZOLE OMEPRAZOLE 80352 54742 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NSC-95397 CHEMBL429095 80353 54743 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL1201733 PAZOPANIB HYDROCHLORIDE 80355 54744 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FENTICLOR FENTICLOR 80356 54745 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650527 80358 54746 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE agonist 135651474 ANDROSTANOLONE 80361 54747 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME DOXORUBICIN DOXORUBICIN 80362 54748 EGLN2 112398 ENZYME, DRUGGABLE GENOME AKB-6548 VADADUSTAT 80363 54749 PDE5A 8654 ENZYME, DRUGGABLE GENOME Vardenafil VARDENAFIL 80364 54750 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL2107387 VORTIOXETINE HYDROBROMIDE 80367 54751 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR RETINAL RETINAL 80368 54752 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Obatoclax OBATOCLAX 80369 54753 KCNC3 3748 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107762 NERISPIRDINE 80371 54754 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SJ000128325 CHEMBL602718 80372 54755 UGT1A10 54575 DRUGGABLE GENOME, ENZYME valproic acid 21806385,28763744,15761113 80373 54756 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME CENISERTIB CENISERTIB 80374 54757 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX QUERCETIN QUERCETIN 25190466 80375 54758 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DEQUALINIUM CHLORIDE DEQUALINIUM CHLORIDE 80376 54759 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE NSC-105827 CHEMBL171699 80379 54760 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE TAK-733 TAK-733 22515704 80381 54761 NNMT 4837 DRUGGABLE GENOME ARI-3037MO 80387 54762 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE MITOXANTRONE MITOXANTRONE 12684687 80388 54763 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR TRITON X TRITON X 80391 54764 PPOX 5498 DRUGGABLE GENOME, ENZYME Givosiran GIVOSIRAN 80392 54765 RGS4 5999 DRUGGABLE GENOME 5-HYDROXYINDOLACETIC ACID CHEMBL395915 80393 54766 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051813 80397 54767 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR 2-METHOXYESTRADIOL 2-METHOXYESTRADIOL 9647742 80398 54768 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor SUNITINIB SUNITINIB 80399 54769 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 249565645 MK-2461 80400 54770 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BUTANAL BUTANAL 80401 54771 ALPL 249 ENZYME, DRUGGABLE GENOME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 80402 54772 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE MGCD265 GLESATINIB 80403 54773 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C7 80406 54774 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR agonist CHEMBL705 ALITRETINOIN 80407 54775 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545248 DS-7423 80408 54776 CBX1 10951 NA HOMOVANILLIC ACID HOMOVANILLIC ACID 80409 54777 PRKD1 5587 DRUGGABLE GENOME, KINASE, ENZYME, TRANSCRIPTION FACTOR, SERINE THREONINE KINASE inhibitor CHEMBL3545332 CEP-2563 80410 54778 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE DNDI1417607 CHEMBL1588679 80411 54779 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SB-203580 SB-203580 80412 54780 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor AXITINIB AXITINIB 80414 54781 BMP2 650 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ISOPROPYL 4-AMINOBENZOATE CHEMBL1467165 22041064 80415 54782 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME inhibitor 187051792 PANOBINOSTAT 80416 54783 ATG4B 23192 ENZYME, DRUGGABLE GENOME, PROTEASE GNF-PF-159 CHEMBL599924 80417 54784 F3 2152 DRUGGABLE GENOME, CELL SURFACE simvastatin SIMVASTATIN 19027114 80418 54785 PIK3R2 5296 CLINICALLY ACTIONABLE, KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME, DRUG RESISTANCE inhibitor BYL719 ALPELISIB 80419 54786 MAP3K8 1326 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178102629 80420 54787 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXYMETHOLONE OXYMETHOLONE 80422 54788 ABAT 18 DRUGGABLE GENOME, ENZYME Vigabatrin VIGABATRIN 80423 54789 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME LY-517717 CHEMBL1271162 80424 54790 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8536181, C35 80425 54791 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE CARBOPLATIN CARBOPLATIN 25847936 80426 54792 TSPO 706 DRUGGABLE GENOME PMID27599163-Compound-78 80427 54793 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417006 CHEMBL1415258 80429 54794 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Androgen restored contraceptive 80430 54795 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME TOZASERTIB TOZASERTIB 80432 54796 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200420 MIDAZOLAM HYDROCHLORIDE 80433 54797 NDUFB8 4714 ENZYME inhibitor CHEMBL3545135 NV-128 80434 54798 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CHLORANIL CHLORANIL 80435 54799 CBX1 10951 NA AG-490 CHEMBL56543 80436 54800 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-25 80437 54801 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody DALOTUZUMAB DALOTUZUMAB 80440 54802 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME N-(arylamino)sulfonamide derivative 1 80442 54803 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 405560388 80443 54804 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Nitrogen mustard derivative 1 80444 54805 ADH1B 125 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1308 FOMEPIZOLE 80446 54806 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CI-1040 CI-1040 23948973 80449 54807 VHL 7428 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TRANSCRIPTION FACTOR Olaparib OLAPARIB 28346230 80450 54808 SMARCB1 6598 CLINICALLY ACTIONABLE Fenretinide FENRETINIDE 23764045 80452 54809 ALDH1A2 8854 DRUGGABLE GENOME, ENZYME RETINOIC ACID 11306068,15652703,14623241 80453 54810 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 315661124 ERDAFITINIB 80454 54811 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TAK-632 28416483 80455 54812 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Propranolol PROPRANOLOL 80456 54813 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL586701 ZSTK-474 80457 54814 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Mteron-F1 80458 54815 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Hydroxychloroquine HYDROXYCHLOROQUINE 80460 54816 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650893 REGLITAZAR 80462 54817 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR OESTRADIOL ESTRADIOL 12553866 80463 54818 HTT 3064 DRUGGABLE GENOME antagonist CHEMBL1631540 GSK163090 80464 54819 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DEXTROTHYROXINE DEXTROTHYROXINE 80466 54820 PSMD13 5719 NA inhibitor CHEMBL2103884 OPROZOMIB 80467 54821 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 IRBESARTAN IRBESARTAN 80469 54822 HMGCR 3156 ENZYME, DRUGGABLE GENOME lovastatin LOVASTATIN 17563401,18815589,18332269,16103896,18261733,15199031 80475 54823 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist CHEMBL3545175 PF-03882845 80477 54824 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ZM-449829 CHEMBL154580 80478 54825 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NIMESULIDE NIMESULIDE 22931300 80480 54826 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE TAMOXIFEN TAMOXIFEN 18283314 80481 54827 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650606 MIANSERIN 80482 54828 GMNN 51053 DRUGGABLE GENOME SJ000029642 CHEMBL591126 80483 54829 AKR1B1 231 DRUGGABLE GENOME, ENZYME Dabelotine DABELOTINE 80484 54830 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NICOTINE NICOTINE 15231866 80485 54831 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE AZD-6765 LANICEMINE 80488 54832 POU5F1 5460 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE allopurinol ALLOPURINOL 21801394 80489 54833 PSMB8 5696 ENZYME, PROTEASE, DRUGGABLE GENOME CARFILZOMIB CARFILZOMIB 24524217 80490 54834 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DYCLONINE DYCLONINE 80493 54835 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CC-223 CC-223 24978597,25855786,26177599 80495 54836 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE DASATINIB DASATINIB 80496 54837 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Tricyclic heterocycle derivative 2 80498 54838 PRKCH 5583 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor CHEMBL574737 UCN-01 80499 54839 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CAT 1004 80501 54840 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 fosamprenavir FOSAMPRENAVIR 80502 54841 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Clomiphene Citrate 80503 54842 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 3-oxo-2,3-dihydro-1H-indazole-4-carboxamide derivative 2 80505 54843 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME INCB054828 PEMIGATINIB 80506 54844 PTGS2 5743 DRUGGABLE GENOME, ENZYME DIFLUNISAL DIFLUNISAL 80507 54845 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Mepyramine maleate 80508 54846 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME DNDI1417165 CHEMBL1406948 80510 54847 RAB9A 9367 ENZYME, DRUGGABLE GENOME CID 1540951 CHEMBL259421 80512 54848 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 381118865 80515 54849 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GW441756X GW441756X 80516 54850 SQLE 6713 DRUGGABLE GENOME, ENZYME Naftifine NAFTIFINE 80521 54851 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BPX-101 80524 54852 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME PMID28870136-Compound-39 80526 54853 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CHLORHEXIDINE HYDROCHLORIDE CHLORHEXIDINE HYDROCHLORIDE 80530 54854 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IPA-3 CHEMBL472940 80531 54855 TGFBR3 7049 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME TGF-BETA 2 1744125 80532 54856 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000121255 CHEMBL590422 80533 54857 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL38 TRETINOIN 80534 54858 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME DACTOLISIB DACTOLISIB 23410005 80535 54859 CD14 929 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME IC14 IC14 80536 54860 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE Lamotrigine LAMOTRIGINE 80537 54861 CD84 8832 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE etanercept ETANERCEPT 27564082 80538 54862 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ALDESLEUKIN ALDESLEUKIN 80539 54863 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME CVBT-141H 80541 54864 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE inhibitor 252166806 80542 54865 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR TANESPIMYCIN TANESPIMYCIN 25277067,23520985,22480433,25105924,17603540,21764310 80543 54866 HNF4A 3172 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR efavirenz EFAVIRENZ 26774523 80545 54867 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor 178101964 TRANYLCYPROMINE 80546 54868 MPHOSPH8 54737 NA SB-202190 SB-202190 80547 54869 TGFB3 7043 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR Avotermin AVOTERMIN 80548 54870 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME PICTILISIB PICTILISIB 80549 54871 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PIROXICAM PIROXICAM 22931300 80550 54872 RORA 6095 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE US9598431, 3 80551 54873 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFA-N3 80552 54874 CACNB2 783 DRUGGABLE GENOME, ION CHANNEL AMLODIPINE AMLODIPINE 80553 54875 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR Quinoxaline derivative 1 80554 54876 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 178102284 MASITINIB 80555 54877 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 329968373 80557 54878 TUBA4A 7277 DRUGGABLE GENOME 10,11-DIHYDROEPOTHILONE D CHEMBL453818 12141877 80558 54879 DPYD 1806 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME FLUOROURACIL FLUOROURACIL 23988873,31871216 80559 54880 ALDH1A1 216 DRUGGABLE GENOME, ENZYME EMBELIN EMBELIN 80560 54881 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE ALENDRONATE ALENDRONIC ACID 80561 54882 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100688 80563 54883 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL180022 NERATINIB 80564 54884 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR entrectinib ENTRECTINIB 80565 54885 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME ENTRECTINIB ENTRECTINIB 80566 54886 HMGB1 3146 DRUGGABLE GENOME, CELL SURFACE, TRANSCRIPTION FACTOR CHELATORS 9398056 80569 54887 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME COUMESTROL COUMESTROL 80570 54888 MAD1L1 8379 NA carboplatin CARBOPLATIN 23407047 80572 54889 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CETUXIMAB CETUXIMAB 80573 54890 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DNDI1417149 CHEMBL1622802 80576 54891 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-123748 CHEMBL530609 80577 54892 DHFR 1719 DRUGGABLE GENOME, ENZYME inhibitor 178103446 PRALATREXATE 80581 54893 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER BORTEZOMIB BORTEZOMIB 28679691 80582 54894 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR MYRISTIC ACID MYRISTIC ACID 80583 54895 CASP4 837 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252166835 80584 54896 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME SJ000120515 CHEMBL592314 80586 54897 POLI 11201 DNA REPAIR ELLAGIC ACID ELLAGIC ACID 80587 54898 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1201833 GOLIMUMAB 80588 54899 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE SB-220025 SB-220025 80589 54900 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ASTEMIZOLE ASTEMIZOLE 80591 54901 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-18 80593 54902 CACNB4 785 DRUGGABLE GENOME, ION CHANNEL celecoxib CELECOXIB 22336956 80595 54903 CTSF 8722 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 405067337 80596 54904 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME blocker 135650590 80603 54905 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ticlopidine TICLOPIDINE 17339877 80604 54906 SMARCA4 6597 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING CISPLATIN CISPLATIN 26671993 80605 54907 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Buparlisib BUPARLISIB 80606 54908 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NALTREXONE NALTREXONE 80607 54909 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antipsychotics 80609 54910 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR conjugated estrogens 9860300 80610 54911 SLCO2A1 6578 TRANSPORTER, DRUGGABLE GENOME 135651569 80611 54912 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ANTHRACYCLINES 11850258 80612 54913 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DANAZOL DANAZOL 22931300 80613 54914 GC 2638 DRUGGABLE GENOME Isosorbide Mononitrate 80614 54915 GAA 2548 DRUGGABLE GENOME, ENZYME TERAZOSIN HYDROCHLORIDE HYDRATE TERAZOSIN HYDROCHLORIDE HYDRATE 80615 54916 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135650095 CICLOPROLOL 80616 54917 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE Dasatinib DASATINIB 80618 54918 PLA2G4A 5321 ENZYME, DRUGGABLE GENOME ZPL521 80619 54919 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CADMIUM DICHLORIDE CADMIUM DICHLORIDE 80620 54920 KAT2B 8850 ENZYME, DRUGGABLE GENOME inhibitor 178103582 PLUMBAGIN 80622 54921 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME VORINOSTAT VORINOSTAT 80623 54922 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ESBA-105 80624 54923 NFIB 4781 CLINICALLY ACTIONABLE methylphenidate METHYLPHENIDATE 29382897 80625 54924 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DAUNORUBICIN DAUNORUBICIN 80626 54925 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE CAMPTOTHECIN CAMPTOTHECIN 80628 54926 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE NEVIRAPINE NEVIRAPINE 17172311 80630 54927 DGAT1 8694 ENZYME, DRUGGABLE GENOME PMID25470667-Compound-AZD3988 80631 54928 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Vemurafenib VEMURAFENIB 26343583,28783719,22798288,23489023,21107323,24035431,24265153,23733758,26352686,25665005,25706985,27760111,25939769,26343582,21383288,26267534,24265152,25265494,26732095,25515853,27297867,27500726,22448344,26287849,27523909,27048246,28514312,28649441,27196754,21639808,22281684,22389471,24283590,26582644,26918217,24448821,27312529,26137449,27048951,26603897,23365119,25589621,26460303,24523613,26984758 80634 54929 CRKL 1399 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE DASATINIB DASATINIB 22591714 80635 54930 TF 7018 CELL SURFACE, DRUGGABLE GENOME PF-06763809 80636 54931 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SJ000001516 CHEMBL592316 80638 54932 CXCL2 2920 DRUGGABLE GENOME BETA-GLUCAN 12419803 80639 54933 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME PMID25980951-Compound-41 80640 54934 XDH 7498 DRUGGABLE GENOME, ENZYME febuxostat FEBUXOSTAT 27798726,24915143 80641 54935 IL15 3600 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, CELL SURFACE, KINASE inhibitor CHEMBL2109467 AMG-714 80642 54936 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DEXTROMETHORPHAN DEXTROMETHORPHAN 21422192 80643 54937 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME OXAZEPAM OXAZEPAM 80645 54938 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR CHRYSOERIOL CHRYSOERIOL 25190466 80646 54939 GMNN 51053 DRUGGABLE GENOME SB-202190 SB-202190 80648 54940 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER ATORVASTATIN ATORVASTATIN 15616150 80649 54941 MAOA 4128 DRUGGABLE GENOME, ENZYME MyriberineA 80651 54942 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME agonist CHEMBL312443 GABOXADOL 80653 54943 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PENTACHLOROPHENOL PENTACHLOROPHENOL 80654 54944 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor CHEMBL512351 BETRIXABAN 80655 54945 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR BML-210 CHEMBL324053 16921367 80656 54946 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE GENISTEIN GENISTEIN 80658 54947 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Benzimidazole and imidazopyridine derivative 1 80660 54948 TUBA3D 113457 DRUGGABLE GENOME COMBRETASTATIN A4 COMBRETASTATIN A4 23631389,16913727,22543234,25584687,24669888,17765552,25192811 80661 54949 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Triazole derivative 2 80662 54950 P2RY1 5028 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, CELL SURFACE antagonist 135651183 80663 54951 MAOB 4129 DRUGGABLE GENOME, ENZYME Tacrine-coumarin hybrid derivative 1 80664 54952 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME IFN 12868960 80666 54953 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME TETROQUINONE TETROQUINONE 80667 54954 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650227 ELETRIPTAN 80670 54955 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER LX-4211 SOTAGLIFLOZIN 80671 54956 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Bosutinib BOSUTINIB 27196758 80672 54957 PSMA4 5685 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL371405 MARIZOMIB 80676 54958 TXK 7294 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 310264693 ACALABRUTINIB 80678 54959 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE CANERTINIB CANERTINIB 23930994 80680 54960 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 80682 54961 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GW7074 CHEMBL72365 80683 54962 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 328083484 80684 54963 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE OXYMETHOLONE OXYMETHOLONE 3238652 80687 54964 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE C-MET INHIBITOR 25952648 80688 54965 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ESTRADIOL VALERATE ESTRADIOL VALERATE 80689 54966 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME NITROBENZYLMERCAPTOPURINE RIBONUCLEOSIDE NITROBENZYLMERCAPTOPURINE RIBONUCLEOSIDE 19574048 80690 54967 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR HYDROCHLOROTHIAZIDE HYDROCHLOROTHIAZIDE 11836266 80691 54968 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 328083493 80695 54969 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME NSC-753576 CHEMBL2088731 22982122 80696 54970 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GERONTOXANTHONE H GERONTOXANTHONE H 80697 54971 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX GENISTEIN GENISTEIN 15963949 80699 54972 ALPI 248 DRUGGABLE GENOME, ENZYME 5,7,3',5'-TETRAHYDROXYFLAVANONE CHEMBL307893 80700 54973 TK1 7083 ENZYME, KINASE, DRUGGABLE GENOME Rilapladib RILAPLADIB 80703 54974 PTGER4 5734 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, KINASE agonist 135651374 80704 54975 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CITICOLINE SODIUM CITICOLINE SODIUM 80705 54976 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Erlotinib ERLOTINIB 27900369 80707 54977 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heteroaryl-carboxamide derivative 1 80708 54978 SMARCB1 6598 CLINICALLY ACTIONABLE Palbociclib PALBOCICLIB 21871868 80710 54979 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HBI-8000 TUCIDINOSTAT 80711 54980 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PROROXAN HYDROCHLORIDE PROROXAN HYDROCHLORIDE 80713 54981 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DICHLOROISOPROTERENOL DICHLOROISOPROTERENOL 2903243 80714 54982 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist CHEMBL284671 CODEINE SULFATE 80715 54983 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME BrevaRex 80716 54984 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME SAR408701 SAR-408701 80720 54985 SRGN 5552 DRUGGABLE GENOME, ENZYME HEPARIN HEPARIN 8613703 80721 54986 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051822 80724 54987 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR HYDROXYPROGESTERONE HYDROXYPROGESTERONE 80725 54988 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 178102317 CHEMBL1908396 80726 54989 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545096 BGT-226 80727 54990 TUBA4A 7277 DRUGGABLE GENOME CHEMBL2108628 PACLITAXEL POLIGLUMEX 80728 54991 DGAT1 8694 ENZYME, DRUGGABLE GENOME inhibitor 223366158 AZD-7687 80729 54992 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor LAPATINIB LAPATINIB 80730 54993 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL ADINAZOLAM ADINAZOLAM 80731 54994 UGT2B7 7364 DRUGGABLE GENOME diclofenac acyl glucuronide 29203276 80732 54995 HLA-E 3133 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE etanercept ETANERCEPT 80733 54996 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME inhibitor 223366190 80736 54997 GMNN 51053 DRUGGABLE GENOME TOREMIFENE CITRATE TOREMIFENE CITRATE 80737 54998 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE inhibitor 249565807 80738 54999 GMNN 51053 DRUGGABLE GENOME DYCLONINE HYDROCHLORIDE DYCLONINE HYDROCHLORIDE 80740 55000 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR FENOFIBRATE FENOFIBRATE 80741 55001 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL454 BUTALBITAL 80742 55002 TXNRD1 7296 DRUGGABLE GENOME ARSENIC TRIOXIDE 80745 55003 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3545006 PWT-33587 80746 55004 BAZ2B 29994 NA CLIOQUINOL CLIOQUINOL 80750 55005 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR BRYOSTATIN BRYOSTATIN 80751 55006 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 340590256 TRILACICLIB 80752 55007 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ARRY-797 ARRY-797 80753 55008 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE ZINC 00035263 CHEMBL2059068 22524450 80754 55009 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-234945 CHEMBL260311 80755 55010 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER TEMOZOLOMIDE TEMOZOLOMIDE 24248532 80756 55011 CACNA2D3 55799 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL2103836 IMAGABALIN 80757 55012 ALOX5AP 241 DRUGGABLE GENOME IL-3 11246129 80758 55013 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL2219421 RECILISIB 80759 55014 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR BMS-582949 BMS-582949 80761 55015 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IODOQUINOL IODOQUINOL 80762 55016 E2F1 1869 TRANSCRIPTION FACTOR HORMONES 8918469 80763 55017 PTGES 9536 DRUGGABLE GENOME, ENZYME Benzimidazole derivative 17 80764 55018 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ARS-1620 29373830,31776128 80765 55019 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME AZD-1080 AZD-1080 80767 55020 CD70 970 CLINICALLY ACTIONABLE, DRUGGABLE GENOME BMS-936561 80768 55021 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist CHEMBL409 BICALUTAMIDE 80769 55022 BCL2A1 597 DRUGGABLE GENOME US8937193-compound-7 80770 55023 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Benzanilide compound 1 80772 55024 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR BELINOSTAT BELINOSTAT 80773 55025 CBX1 10951 NA DNDI1417055 CHEMBL1486366 80774 55026 TGM2 7052 PROTEASE, DRUGGABLE GENOME, ENZYME VASCULAR ENDOTHELIAL GROWTH FACTOR 16914140 80776 55027 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE GNF-PF-1654 CHEMBL602776 80778 55028 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor POZIOTINIB POZIOTINIB 80780 55029 PTGES 9536 DRUGGABLE GENOME, ENZYME PMID28627961-Compound-44 80781 55030 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 223366168 SPEBRUTINIB 80782 55031 HTT 3064 DRUGGABLE GENOME SJ000294102 CHEMBL607309 80784 55032 MMP14 4323 PROTEASE, DRUGGABLE GENOME, ENZYME PYROGALLOL RED PYROGALLOL RED 80786 55033 ATAD5 79915 NA GNF-PF-1094 CHEMBL415914 80787 55034 CALM1 801 ION CHANNEL, KINASE, ENZYME, DRUGGABLE GENOME BEPRIDIL BEPRIDIL 80789 55035 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 FIPEXIDE FIPEXIDE 80790 55036 RGS4 5999 DRUGGABLE GENOME DEPHOSTATIN DEPHOSTATIN 80791 55037 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Ixabepilone IXABEPILONE 80792 55038 ALB 213 TRANSPORTER, DRUGGABLE GENOME EPICATECHIN GALLATE EPICATECHIN GALLATE 20598557 80793 55039 STAG2 10735 CLINICALLY ACTIONABLE, DRUG RESISTANCE Rucaparib RUCAPARIB 21852505,24356817 80794 55040 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR EPIRUBICIN HYDROCHLORIDE EPIRUBICIN HYDROCHLORIDE 80796 55041 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545052 FIMEPINOSTAT 80798 55042 GJA1 2697 ION CHANNEL ATENOLOL ATENOLOL 16448880 80800 55043 SRSF2 6427 CLINICALLY ACTIONABLE N/A 26508027,26769228 80801 55044 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist CHEMBL1201165 QUINESTROL 80802 55045 CD8A 925 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE LIPO-4 80803 55046 SMN2 6607 DRUGGABLE GENOME TRICHOSTATIN TRICHOSTATIN 80804 55047 ATXN2 6311 NA GNF-PF-2383 CHEMBL578915 80805 55048 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME GNF-PF-3770 CHEMBL597874 80807 55049 UGT1A7 54577 DRUGGABLE GENOME, ENZYME valproic acid 21806385,28763744,15761113 80812 55050 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor AS703569 CENISERTIB 80815 55051 HDAC11 79885 DRUGGABLE GENOME, ENZYME LARGAZOLE LARGAZOLE 21420302,25203782,20491440 80822 55052 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8669361, 102 80824 55053 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565750 PRT-2607 80825 55054 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TIMOLOL TIMOLOL 80826 55055 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor SF1126 80827 55056 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor CHEMBL235191 TACEDINALINE 80828 55057 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ZM-447439 CHEMBL202721 80829 55058 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GUANIDINYL-NALTRINDOLE DI-TRIFLUOROACETATE CHEMBL1255944 80833 55059 PSMA5 5686 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL371405 MARIZOMIB 80834 55060 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme7WO2012/098070bottom 80835 55061 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER FANCHININ FANCHININ 80836 55062 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER topotecan TOPOTECAN 80837 55063 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 135651483 ESTRIOL 80838 55064 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 80840 55065 ALB 213 TRANSPORTER, DRUGGABLE GENOME RU-101 14507766 80841 55066 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME AT-406 AT-406 25520882 80842 55067 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE THONZONIUM BROMIDE THONZONIUM BROMIDE 80844 55068 APOE 348 DRUGGABLE GENOME AEM-28 80845 55069 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE PAZOPANIB PAZOPANIB 80846 55070 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135651027 80847 55071 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AZELASTINE HYDROCHLORIDE AZELASTINE HYDROCHLORIDE 80848 55072 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 223365984 LUCITANIB 80853 55073 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 flibanserin FLIBANSERIN 80854 55074 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE cobimetinib COBIMETINIB 22084396 80856 55075 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE NSC-102742 CHEMBL1519374 80857 55076 PRKAA1 5562 KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, TRANSPORTER, SERINE THREONINE KINASE SOTRASTAURIN SOTRASTAURIN 80858 55077 PDE4B 5142 DRUGGABLE GENOME, ENZYME LIRIMILAST LIRIMILAST 80860 55078 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Dydrogesterone DYDROGESTERONE 80865 55079 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME inhibitor 381744901 80866 55080 POU5F1 5460 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE carbamazepine CARBAMAZEPINE 80868 55081 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME 178101388 80870 55082 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME Gallopamil GALLOPAMIL 80871 55083 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-3416 CHEMBL579550 80872 55084 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR WORTMANNIN WORTMANNIN 12391262 80873 55085 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME PURPURIN PURPURIN 80874 55086 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2014078408Example1 80875 55087 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME IDARUBICIN IDARUBICIN 80876 55088 TUBB2A 7280 DRUGGABLE GENOME VINBLASTINE VINBLASTINE 80877 55089 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE LAPATINIB LAPATINIB 80879 55090 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DNDI1417777 CHEMBL1412002 80881 55091 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE METHYLPREDNISOLONE METHYLPREDNISOLONE 16141680,16684279 80884 55092 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR AMPICILLIN SODIUM AMPICILLIN SODIUM 80885 55093 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING BITHIONOLOXIDE BITHIONOLOXIDE 80886 55094 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PROGESTERONE PROGESTERONE 80890 55095 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR TAE-684 TAE-684 80891 55096 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY ETHANOL ALCOHOL 8289752 80892 55097 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE Palbociclib PALBOCICLIB 27020857 80893 55098 KLKB1 3818 DRUGGABLE GENOME, PROTEASE, ENZYME BCX4161 80895 55099 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUPRENORPHINE BUPRENORPHINE 80897 55100 TUBA3C 7278 DRUGGABLE GENOME VORINOSTAT VORINOSTAT 20491440 80898 55101 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME LARGAZOLE LARGAZOLE 21420302,25203782,20491440 80900 55102 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor CHEMBL1201439 BASILIXIMAB 80901 55103 PSMD14 10213 PROTEASE, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL325041 BORTEZOMIB 80902 55104 RGS4 5999 DRUGGABLE GENOME LINSIDOMINE LINSIDOMINE 80904 55105 MVK 4598 KINASE, ENZYME inhibitor 135651495 80906 55106 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CHLOROXURON CHLOROXURON 80907 55107 PSMA7 5688 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL2103884 OPROZOMIB 80909 55108 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GLPG0492 GLPG0492 80910 55109 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL valproic acid 23859570,21747585,28753467,25155934 80912 55110 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000113972 CHEMBL591137 80915 55111 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE VELIPARIB VELIPARIB 80918 55112 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE CURCUMIN CURCUMIN 12446602 80919 55113 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME clozapine CLOZAPINE 22565219 80920 55114 MAOB 4129 DRUGGABLE GENOME, ENZYME FERULIC ACID 80921 55115 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME CHEMBL1341 METHOXYFLURANE 80922 55116 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor MGCD265 GLESATINIB 80927 55117 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE antagonist CHEMBL1207366 GW468816 80929 55118 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE NADOLOL NADOLOL 80931 55119 CCL11 6356 DRUGGABLE GENOME Bertilimumab BERTILIMUMAB 80933 55120 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Anti-PD-L1 CSR T cells 80934 55121 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE ribavirin RIBAVIRIN 28703131 80935 55122 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heteroaryl-carboxamide derivative 5 80937 55123 BAZ2B 29994 NA EPINEPHRINE BITARTRATE EPINEPHRINE BITARTRATE 80938 55124 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 249565775 80939 55125 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME CID 4101591 CHEMBL428789 80940 55126 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3545054 INCB-40093 80941 55127 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CLORGYLINE HYDROCHLORIDE CLORGYLINE HYDROCHLORIDE 80942 55128 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR BROMOXYNIL BROMOXYNIL 80943 55129 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 178103311 PRINABEREL 80944 55130 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE PF-05212384 GEDATOLISIB 17314276,21325073 80946 55131 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 363894210 PANULISIB 80947 55132 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME Pyridine derivative 21 80948 55133 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Metformin METFORMIN 26921394,26951660 80951 55134 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE CPT-11 IRINOTECAN HYDROCHLORIDE 15809721 80952 55135 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME PMID27774824-Compound-Figure3Example18 80953 55136 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor BMS-690514 BMS-690514 80954 55137 KLK2 3817 PROTEASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Avoralstat AVORALSTAT 80955 55138 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BUCLADESINE BUCLADESINE 80956 55139 MUC1 4582 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME YTTRIUM (90Y) CLIVATUZUMAB TETRAXETAN 80957 55140 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PKI-587 GEDATOLISIB 80959 55141 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CHLORPROMAZINE CHLORPROMAZINE 16810505 80960 55142 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 FLUTAMIDE FLUTAMIDE 22931300 80961 55143 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Potassium Chloride 80962 55144 ALOX15 246 ENZYME, DRUGGABLE GENOME ARACHIDONIC ACID ARACHIDONIC ACID 80963 55145 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 249565802 80964 55146 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-32 80965 55147 ALB 213 TRANSPORTER, DRUGGABLE GENOME FLUCONAZOLE FLUCONAZOLE 25301772 80966 55148 TARDBP 23435 TUMOR SUPPRESSOR FAGARONINE FAGARONINE 80967 55149 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CEFIXIME CEFIXIME 80968 55150 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME tolterodine TOLTERODINE 21352267,20530222,10190648,9630826,10583026,28087463 80969 55151 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TYRPHOSTIN AG-1478 TYRPHOSTIN AG-1478 80970 55152 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Etonogestrel ETONOGESTREL 80972 55153 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 249565900 80973 55154 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 178103162 80975 55155 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE daunorubicin DAUNORUBICIN 8648264 80977 55156 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CLONAZEPAM CLONAZEPAM 80978 55157 CBX1 10951 NA CAMBINOL CAMBINOL 80979 55158 PBRM1 55193 CLINICALLY ACTIONABLE PEMBROLIZUMAB PEMBROLIZUMAB 29301960 80980 55159 BAZ2B 29994 NA SJ000201681 CHEMBL602135 80981 55160 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Vismodegib VISMODEGIB 26676867,19726788,25759020,26823493,25759019 80982 55161 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OXYPHENCYCLIMINE OXYPHENCYCLIMINE 80983 55162 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME CENISERTIB CENISERTIB 80987 55163 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE XL765 80988 55164 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING SUBEROHYDROXAMIC ACID SUBEROHYDROXAMIC ACID 16921367 80991 55165 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CHEMBL1200789 TRICLOFOS SODIUM 80992 55166 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR exemestane EXEMESTANE 26536870 80993 55167 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ANTHRAQUINONE ANTHRAQUINONE 80995 55168 USP14 9097 ENZYME, CELL SURFACE, PROTEASE Tricyclic heterocycle derivative 4 80996 55169 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME OSI-027 OSI-027 80997 55170 PROC 5624 PROTEASE, DRUGGABLE GENOME, ENZYME phenprocoumon PHENPROCOUMON 80999 55171 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME VEMURAFENIB VEMURAFENIB 25462267 81001 55172 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-7 81004 55173 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME activator 135651473 81005 55174 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR AZD-8330 AZD-8330 81007 55175 PSMD7 5713 PROTEASE inhibitor CHEMBL2103884 OPROZOMIB 81012 55176 TMPRSS15 5651 PROTEASE, DRUGGABLE GENOME, ENZYME US9024044, 2 81014 55177 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE ANTITHYMOCYTE GLOBULIN 81015 55178 GAA 2548 DRUGGABLE GENOME, ENZYME MIGALASTAT MIGALASTAT 81018 55179 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME XL147 PILARALISIB 25637314 81019 55180 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL1200472 QUAZEPAM 81020 55181 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Salicylic acid derivative 2 81021 55182 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX PMID27336223-Compound-9 81022 55183 PARP2 10038 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, HISTONE MODIFICATION, DNA REPAIR, ENZYME Tetra-cyclic pyridophthalazinone derivative 1 81023 55184 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME CIGLITAZONE CIGLITAZONE 81024 55185 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 135650177 DICLOFENAC 81025 55186 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL3182621 AZD-8330 81026 55187 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Levonorgestrel LEVONORGESTREL 81028 55188 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE IRBESARTAN IRBESARTAN 18162196 81029 55189 RACGAP1 29127 NA PROCHLORPERAZINE EDISYLATE PROCHLORPERAZINE EDISYLATE 81030 55190 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 340590255 ROVAZOLAC 81034 55191 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL598797 CUDC-101 81037 55192 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME RUXOLITINIB RUXOLITINIB 23634996,23656643 81038 55193 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME NIACIN RECEPTOR AGONIST 81039 55194 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TETRABROMOBENZOTRIAZOLE TETRABROMOBENZOTRIAZOLE 81040 55195 MAPT 4137 DRUGGABLE GENOME TCMDC-123869 CHEMBL546597 81041 55196 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER JNJ-1661010 CHEMBL460273 81042 55197 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR INDIRUBIN SULFATE SU-9516 81043 55198 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NIFEDIPINE NIFEDIPINE 81044 55199 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 310264719 81045 55200 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651409 81046 55201 GMNN 51053 DRUGGABLE GENOME PAXILLINE PAXILLINE 81048 55202 UGT1A6 54578 ENZYME, DRUGGABLE GENOME valproic acid 21806385,28763744,23099353,15761113 81051 55203 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR KD-025 CHEMBL2005186 81053 55204 PDE5A 8654 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL779 TADALAFIL 81054 55205 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE CEDIRANIB CEDIRANIB 81057 55206 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME CHLORPYRIFOS-METHYL CHLORPYRIFOS-METHYL 81058 55207 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TAE-684 TAE-684 81059 55208 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME PRX302 TOPSALYSIN 81060 55209 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3545179 AZD-7451 81062 55210 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR DIHYDROTANSHINONE I DIHYDROTANSHINONE I 26339922 81063 55211 POLK 51426 DNA REPAIR, ENZYME GALLIC ACID GALLIC ACID 81065 55212 POLK 51426 DNA REPAIR, ENZYME 3,3',4'-TRIHYDROXYFLAVONE CHEMBL122701 81066 55213 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1201013 OLSALAZINE SODIUM 81067 55214 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ACETAMIDE ACETAMIDE 81068 55215 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NAPROXEN NAPROXEN 22931300 81070 55216 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE HEXACHLOROPHENE HEXACHLOROPHENE 81072 55217 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME AZD-1775 ADAVOSERTIB 81073 55218 CDX2 1045 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TPN 10712262 81075 55219 MPHOSPH8 54737 NA TYRPHOSTIN 25 TYRPHOSTIN 25 81077 55220 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Epoxysuccinate derivative 8 81080 55221 ACSS2 55902 ENZYME, TRANSCRIPTION FACTOR carboplatin CARBOPLATIN 21636554 81081 55222 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME NINTEDANIB NINTEDANIB 81082 55223 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor XL228 XL-228 81085 55224 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE RINDOPEPIMUT RINDOPEPIMUT 81088 55225 NOX4 50507 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME GKT-137831 22806357 81089 55226 DHFR 1719 DRUGGABLE GENOME, ENZYME TRIMETREXATE TRIMETREXATE 81090 55227 ALPL 249 ENZYME, DRUGGABLE GENOME ISOQUERCETIN ISOQUERCETIN 81093 55228 RAB9A 9367 ENZYME, DRUGGABLE GENOME AG1295 AG1295 81094 55229 USP1 7398 DNA REPAIR, PROTEASE, ENZYME TETRABROMOBENZOTRIAZOLE TETRABROMOBENZOTRIAZOLE 81095 55230 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 3-METHOXYFLAVONOL CHEMBL272005 81099 55231 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CLOPIDOGREL CLOPIDOGREL 81100 55232 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE GDC-0199 VENETOCLAX 81101 55233 HKDC1 80201 DRUGGABLE GENOME, KINASE DNDI1417722 CHEMBL1503190 81102 55234 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178100445 81103 55235 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME LARGAZOLE LARGAZOLE 21420302,25203782,20491440 81105 55236 HDAC5 10014 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 187051807 SCRIPTAID 81106 55237 EP300 2033 CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME inhibitor 178103580 GARCINOL 81108 55238 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME Pyrazole N-1 aryl and heteroaryl derivative 1 81109 55239 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Tramadol TRAMADOL 81111 55240 RAPGEF3 10411 ENZYME 4'-EPICHAETOVIRIDIN A CHEMBL1306556 81116 55241 ATAD5 79915 NA DILAZEP DILAZEP 81117 55242 HEBP1 50865 DRUGGABLE GENOME PMID28454500-Compound-96 81118 55243 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME XANTHOHUMOL XANTHOHUMOL 22111577 81121 55244 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CHEMBL939 GEFITINIB 81122 55245 AKR1C3 8644 ENZYME, DRUGGABLE GENOME N-(pyridinepyrroylylcarbonyl)-piperidine derivative 1 81124 55246 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE lapatinib LAPATINIB 81125 55247 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-2812 CHEMBL125044 81126 55248 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME MANGOSTIN MANGOSTIN 81128 55249 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-123634 CHEMBL530499 81129 55250 HSPB1 3315 DRUGGABLE GENOME BUFOTENINE BUFOTENINE 81131 55251 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BISACODYL BISACODYL 81134 55252 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3544942 RONICICLIB 81135 55253 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HOMIDIUM BROMIDE HOMIDIUM BROMIDE 81136 55254 KDM4A 9682 DRUGGABLE GENOME, ENZYME CATECHOL CATECHOL 81137 55255 TUBB6 84617 DRUGGABLE GENOME inhibitor CHEMBL428647 PACLITAXEL 81138 55256 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL494089 GSK-690693 81139 55257 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR CHOLECALCIFEROL CHOLECALCIFEROL 81140 55258 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE BDBM50061601 81142 55259 USP1 7398 DNA REPAIR, PROTEASE, ENZYME BITHIONOLATE SODIUM BITHIONOLATE SODIUM 81143 55260 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545368 PANOBINOSTAT LACTATE 81146 55261 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE 5-BENZYLOXYTRYPTAMINE 5-BENZYLOXYTRYPTAMINE 20965726 81147 55262 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE agonist 178101669 MECASERMIN 81151 55263 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565852 81152 55264 DHODH 1723 DRUGGABLE GENOME, ENZYME inhibitor 178103978 BREQUINAR 81154 55265 WEE1 7465 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME MK-1775 ADAVOSERTIB 81155 55266 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8592455, 3 81156 55267 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR LY2157299 81159 55268 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Clozapine CLOZAPINE 81160 55269 LIFR 3977 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE Emfilermin EMFILERMIN 15089810 81161 55270 POLB 5423 DNA REPAIR, DRUGGABLE GENOME GNF-PF-2357 CHEMBL578257 81165 55271 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME LYMPHOKINES 8007461 81167 55272 CXCL8 3576 DRUGGABLE GENOME FENRETINIDE FENRETINIDE 16979119 81168 55273 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR modulator CHEMBL146506 MOFAROTENE 81169 55274 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CERTOLIZUMAB PEGOL 81170 55275 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 249565689 81171 55276 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR OXYCODONE OXYCODONE 81172 55277 CDK12 51755 KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, TUMOR SUPPRESSOR, SERINE THREONINE KINASE inhibitor CHEMBL1230607 PHA-793887 81173 55278 FADD 8772 NA FAS LIGAND 11384965 81174 55279 ADH1C 126 ENZYME, DRUGGABLE GENOME ethanol ALCOHOL 14693654,32451486 81175 55280 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AMPHOTERICIN B AMPHOTERICIN B 22931300 81176 55281 ALDH5A1 7915 DRUGGABLE GENOME, ENZYME Chlormerodrin CHLORMERODRIN 81177 55282 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Quinazolinedione derivative 1 81178 55283 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 8-CYCLOPENTYLTHEOPHYLLINE 8-CYCLOPENTYLTHEOPHYLLINE 81179 55284 PTGDS 5730 ENZYME, TRANSPORTER, DRUGGABLE GENOME inhibitor 381744942 81180 55285 ARRB2 409 ION CHANNEL, G PROTEIN COUPLED RECEPTOR buprenorphine BUPRENORPHINE 30549211 81181 55286 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME fluorouracil FLUOROURACIL 81182 55287 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 avatrombopag AVATROMBOPAG 81183 55288 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DIMETHYL SULFOXIDE 16896803 81184 55289 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX gefitinib GEFITINIB 31664190 81185 55290 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Crizotinib CRIZOTINIB 27338794,25232318,26432108 81187 55291 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MERCURIC CHLORIDE MERCURIC CHLORIDE 81188 55292 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BQ-123 BQ-123 81189 55293 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE CETUXIMAB CETUXIMAB 25520391 81192 55294 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 252827496 81194 55295 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE DEXTRAN SULFATE 7920442 81199 55296 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME UCB-35440 81200 55297 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL1230607 PHA-793887 81201 55298 RELA 5970 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, TRANSCRIPTION FACTOR COMPLEX FRENTIZOLE FRENTIZOLE 81202 55299 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL1201752 IXABEPILONE 81203 55300 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-4 81204 55301 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NSC-668394 CHEMBL336095 81205 55302 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE IL-11 OPRELVEKIN 8641341 81206 55303 DPP8 54878 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 363894186 TALABOSTAT 81207 55304 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TCMDC-123641 CHEMBL532849 81208 55305 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 19 81209 55306 GMNN 51053 DRUGGABLE GENOME FLAZALONE FLAZALONE 81210 55307 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 NEOSTIGMINE BROMIDE NEOSTIGMINE BROMIDE 22931300 81211 55308 SLC6A19 340024 DRUGGABLE GENOME, TRANSPORTER inhibitor 381744938 CINROMIDE 81214 55309 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME pravastatin PRAVASTATIN 81215 55310 GSTT1 2952 DRUGGABLE GENOME carboplatin CARBOPLATIN 81216 55311 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR FENOFIBRATE FENOFIBRATE 15543343 81217 55312 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PROPYL GALLATE PROPYL GALLATE 81218 55313 PSMD11 5717 KINASE inhibitor CHEMBL2103884 OPROZOMIB 81219 55314 PLAUR 5329 DRUGGABLE GENOME, ENZYME, CELL SURFACE Ruxolitinib RUXOLITINIB 81220 55315 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME Pyrimidinyl compound 2 81221 55316 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE SIROLIMUS SIROLIMUS 24934779,25157968,18089823 81222 55317 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (S)-ALAPROCLATE (S)-ALAPROCLATE 81224 55318 MGLL 11343 DRUGGABLE GENOME, ENZYME PMID29053063-Compound-7d 81225 55319 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE MITOTANE MITOTANE 81227 55320 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR agonist 135651505 81228 55321 ERBB4 2066 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GGF-2 81229 55322 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME AMG-181 ABRILUMAB 81230 55323 TUBA1C 84790 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 81231 55324 DNER 92737 NA PMID26924192-Compound-51 81233 55325 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PAZOPANI 81234 55326 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE Phthalazine derivative 3 81237 55327 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Warfarin WARFARIN 81238 55328 MAPT 4137 DRUGGABLE GENOME (S)APOMORPHINE (S)APOMORPHINE 81239 55329 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL186179 MURAGLITAZAR 81240 55330 TOP2B 7155 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545337 C-1311 81241 55331 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor NINTEDANIB NINTEDANIB 81242 55332 PTPRB 5787 DRUGGABLE GENOME, PROTEIN PHOSPHATASE SUNITINIB SUNITINIB 24633157 81243 55333 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE antagonist 252166838 GALETERONE 81244 55334 MAOA 4128 DRUGGABLE GENOME, ENZYME PIPERINE PIPERINE 81246 55335 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING FENOFIBRATE FENOFIBRATE 16680159 81247 55336 TYMS 7298 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE 5-FLUOROURACIL FLUOROURACIL 81248 55337 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 223366211 CRENOLANIB 81251 55338 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PYRONIN Y PYRONIN Y 81252 55339 MPHOSPH8 54737 NA CEPHAPIRIN SODIUM CEPHAPIRIN SODIUM 81255 55340 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor DASATINIB DASATINIB 81256 55341 HSPG2 3339 KINASE, DRUGGABLE GENOME PALIFERMIN PALIFERMIN 81258 55342 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME pegaptanib PEGAPTANIB SODIUM 23953100 81260 55343 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SPICLOMAZINE SPICLOMAZINE 81262 55344 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL2220486 LUCITANIB 81264 55345 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME AZD-1080 AZD-1080 81265 55346 POLK 51426 DNA REPAIR, ENZYME TYRPHOSTIN 23 TYRPHOSTIN 23 81266 55347 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE inhibitor 178103159 81267 55348 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL568 OXAZEPAM 81269 55349 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Denagliptin DENAGLIPTIN 81270 55350 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME Quinolinyl pyrazinyl urea derivative 2 81272 55351 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Hepapoietin 81273 55352 GMNN 51053 DRUGGABLE GENOME AMCINONIDE AMCINONIDE 81275 55353 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Trastuzumab TRASTUZUMAB 17936563,21676217,24470511,26469692,28167203,23940356,26245675,21558396 81276 55354 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 COUMARIN COUMARIN 22931300 81278 55355 BAZ2B 29994 NA GNF-PF-3148 CHEMBL81782 81281 55356 MAP3K11 4296 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME CEP-1347 CEP-1347 24044867 81282 55357 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 178102338 SU-014813 81283 55358 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Methylsulfonylbenzamide derivative 2 81284 55359 TRPM8 79054 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE PF-05105679 PF-05105679 81287 55360 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ESTRONE ESTRONE 81289 55361 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL PENTOBARBITAL PENTOBARBITAL 81291 55362 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 223365932 PRALIDOXIME 81292 55363 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE antibody LY2875358 81293 55364 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Pembrolizumab PEMBROLIZUMAB 81298 55365 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BICALUTAMIDE BICALUTAMIDE 81299 55366 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 381118867 81301 55367 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-4242 CHEMBL584514 81302 55368 MAGEA3 4102 ENZYME, DRUGGABLE GENOME IDM-2101 81303 55369 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME aspirin ASPIRIN 81304 55370 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE ALISERTIB ALISERTIB 81305 55371 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME HEPARIN HEPARIN 11243881 81308 55372 CSNK1E 1454 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, DNA REPAIR inhibitor 178102608 IC261 81310 55373 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Mycophenolic acid/nucleotide derivative 7 81312 55374 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Trapidil TRAPIDIL 81314 55375 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER VX-970 BERZOSERTIB 81316 55376 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker 178102357 81318 55377 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-21 81319 55378 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME imatinib IMATINIB 30237583 81320 55379 FGB 2244 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, FIBRINOGEN, DRUGGABLE GENOME METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 81321 55380 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650783 81323 55381 POLK 51426 DNA REPAIR, ENZYME 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 3,4-DIDESMETHYL-5-DESHYDROXY-3'-ETHOXYSCLEROIN 81324 55382 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565623 GEDATOLISIB 81325 55383 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 5 81326 55384 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE PHA-793887 PHA-793887 81327 55385 CPB2 1361 DRUGGABLE GENOME, ENZYME, PROTEASE C5A 14525995 81329 55386 POLK 51426 DNA REPAIR, ENZYME N-(4-CARBOXYPHENYL)RHODANINE CHEMBL450802 81331 55387 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PILOCARPINE PILOCARPINE 10101239 81332 55388 KDM4A 9682 DRUGGABLE GENOME, ENZYME FENOLDOPAM MESYLATE FENOLDOPAM MESYLATE 81333 55389 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NIFEDIPINE NIFEDIPINE 81334 55390 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE ANESTHETICS 16428543 81335 55391 ALDH1A1 216 DRUGGABLE GENOME, ENZYME OXYBENZONE OXYBENZONE 81336 55392 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME MMV006513 CHEMBL585622 81338 55393 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME ARA 290 81339 55394 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 310264675 CUDC-101 81341 55395 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE CD123-specific gene-engineered T cells 81343 55396 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR CIGLITAZONE CIGLITAZONE 23566516 81344 55397 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL LORAZEPAM LORAZEPAM 81345 55398 PFKFB3 5209 ENZYME, KINASE PFK-158 81346 55399 GBA 2629 DRUGGABLE GENOME, ENZYME PHLORETIN PHLORETIN 81347 55400 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ESR0114 81348 55401 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE GV1001 TERTOMOTIDE 81349 55402 TUBB3 10381 DRUGGABLE GENOME ABT-751 ABT-751 25468039 81350 55403 F10 2159 DRUGGABLE GENOME, PROTEASE, ENZYME MANGIFERIN HEPTASULFATE MANGIFERIN HEPTASULFATE 21732671 81353 55404 IL18 3606 DRUGGABLE GENOME CORTICOSTEROIDS 12689659 81354 55405 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE BETA-NAPHTHOFLAVONE BETA-NAPHTHOFLAVONE 23600958 81355 55406 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME ROMIDEPSIN ROMIDEPSIN 26331334 81356 55407 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE inhibitor CHEMBL1206245 BRICICLIB 81359 55408 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE TANDUTINIB TANDUTINIB 81361 55409 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651557 81362 55410 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PALIFERMIN PALIFERMIN 81363 55411 ATIC 471 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE methotrexate METHOTREXATE 27885916,18322994,27217051,26799664,25084201,27676277,29520081,16947783,20847201,15457444 81364 55412 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TOLAZAMIDE TOLAZAMIDE 81365 55413 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE antibody DROZITUMAB DROZITUMAB 81367 55414 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE RACEPINEPHRINE HYDROCHLORIDE RACEPINEPHRINE HYDROCHLORIDE 81368 55415 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor BEZ235 DACTOLISIB 81369 55416 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE Crenolanib CRENOLANIB 24132921,22745105 81370 55417 BAZ2B 29994 NA TDR78109 CHEMBL1304363 81371 55418 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL QUAZEPAM QUAZEPAM 81373 55419 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GANGALEOIDIN GANGALEOIDIN 81374 55420 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CILOSTAZOL CILOSTAZOL 22931300 81375 55421 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor AMG208 81376 55422 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Conjugated estrogens a 81377 55423 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE Florbetapir F-18 81378 55424 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME AG-1288 CHEMBL166486 81379 55425 TNIK 23043 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE inhibitor 249565872 81381 55426 PSMD4 5710 NA BORTEZOMIB BORTEZOMIB 24524217 81382 55427 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ERGOLOID MESYLATE 81384 55428 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE LYNGBYABELLIN A LYNGBYABELLIN A 81385 55429 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SK-7041 CHEMBL152133 81386 55430 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE CENISERTIB CENISERTIB 81388 55431 DGAT2 84649 ENZYME PF-06427878 81389 55432 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 340590266 GDC-0077 81392 55433 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 nevirapine NEVIRAPINE 81394 55434 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135649886 81395 55435 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor CHEMBL2095208 COBICISTAT 81396 55436 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME Phenylalanine derivative 1 81397 55437 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3360203 PILARALISIB 81398 55438 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE LINIFANIB LINIFANIB 81399 55439 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE CEPHALOCHROMIN CEPHALOCHROMIN 81400 55440 ATXN2 6311 NA TCMDC-124166 CHEMBL528712 81401 55441 IFNG 3458 DRUGGABLE GENOME RECOMBINANT INTERLEUKIN-1-BETA 8383325 81406 55442 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE TRICHOSTATIN A 12198113 81407 55443 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ETHANOL ALCOHOL 18759561 81408 55444 HTT 3064 DRUGGABLE GENOME Rocilinostat 81409 55445 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE SAR260301 SAR-260301 27196754,24387221 81411 55446 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thieno[3,2-c]pyridine-7-carboxamide derivative 2 81412 55447 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor 348353650 81413 55448 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE PHOSPHODIESTERASE INHIBITOR 3021458 81414 55449 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE ARQ092 81415 55450 GANAB 23193 DRUGGABLE GENOME, ENZYME MIGLUSTAT MIGLUSTAT 21292481 81416 55451 ADAM17 6868 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, NEUTRAL ZINC METALLOPEPTIDASE, TRANSPORTER, ENZYME inhibitor 178103096 APRATASTAT 81417 55452 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107762 NERISPIRDINE 81418 55453 THSD7B 80731 NA ethanol ALCOHOL 32451486 81419 55454 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-3418 CHEMBL582099 81420 55455 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR PMID25980951-Compound-41 81422 55456 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME CENISERTIB CENISERTIB 81423 55457 HTT 3064 DRUGGABLE GENOME PROFLAVINE PROFLAVINE 81425 55458 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565636 BMS-777607 81426 55459 CDKN3 1033 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, TUMOR SUPPRESSOR, ENZYME, KINASE inhibitor CHEMBL1230607 PHA-793887 81427 55460 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SIMVASTATIN SIMVASTATIN 18302447 81429 55461 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PETROSIOL A PETROSIOL A 23415061 81430 55462 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 3-METHOXYFLAVONOL CHEMBL272005 81432 55463 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Erlotinib ERLOTINIB 81434 55464 RORA 6095 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE MELATONIN MELATONIN 8702678,12595746 81435 55465 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYLENE BLUE CHLORIDE HYDRATE METHYLENE BLUE 81436 55466 KDM4C 23081 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME SJ000154295 CHEMBL578502 81438 55467 RGS5 8490 NA fluorouracil FLUOROURACIL 25069475 81439 55468 GMNN 51053 DRUGGABLE GENOME DEMECOLCINE DEMECOLCINE 81444 55469 C1R 715 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 178101079 NAFAMOSTAT 81445 55470 NGB 58157 NA SODIUM SALICYLATE 16094504 81446 55471 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME THIRAM THIRAM 81447 55472 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor VALPROIC ACID DEPAKOTE 81452 55473 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 EFAVIRENZ EFAVIRENZ 16176117 81453 55474 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Aminotriazolopyridine derivative 1 81454 55475 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER EGCG EPIGALOCATECHIN GALLATE 14511674 81455 55476 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE modulator CHEMBL467888 LGD-2941 81458 55477 CTSB 1508 DRUGGABLE GENOME, PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, ENZYME PMID27998201-Compound-2 81459 55478 BAZ2B 29994 NA NSC-71097 CHEMBL1939687 81460 55479 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 336446945 81463 55480 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27744724-Compound-18 81464 55481 SCNN1G 6340 ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE blocker CHEMBL585 TRIAMTERENE 81465 55482 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL Menthol MENTHOL 81466 55483 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SP-600125 SP-600125 81467 55484 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TYRPHOSTIN 47 TYRPHOSTIN 47 81468 55485 POLK 51426 DNA REPAIR, ENZYME NSC-74859 CHEMBL477936 81470 55486 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR 17-AAG TANESPIMYCIN 12738674 81471 55487 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY OCTREOTIDE OCTREOTIDE 14530610 81472 55488 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE QUERCETIN QUERCETIN 81473 55489 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 384403648 AVAPRITINIB 81474 55490 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR inhibitor TANESPIMYCIN TANESPIMYCIN 81475 55491 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200467 HYDROXYZINE PAMOATE 81476 55492 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor CHEMBL3545401 X-82 81477 55493 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE RUCAPARIB RUCAPARIB 81480 55494 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME PF-562271 PF-00562271 81481 55495 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 81482 55496 ESRRA 2101 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Corticosteroid 81484 55497 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME OCTREOTIDE OCTREOTIDE 12721506,18198230 81485 55498 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DISULFIRAM DISULFIRAM 81486 55499 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565905 81487 55500 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FLUPHENAZINE FLUPHENAZINE 81488 55501 DDR1 780 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor 178102324 NILOTINIB 81489 55502 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PMID28270021-Compound-WO2010077680 201 81490 55503 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW827105X GW827105X 81492 55504 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR ESTRADIOL ESTRADIOL 81493 55505 KDM4A 9682 DRUGGABLE GENOME, ENZYME METRAZOLINE OXALATE METRAZOLINE OXALATE 81494 55506 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR OXYQUINOLINE OXYQUINOLINE 81495 55507 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME AD 337 81498 55508 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE ARSENIC TRIOXIDE 81499 55509 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME RITONAVIR RITONAVIR 14977870 81500 55510 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER dexamethasone DEXAMETHASONE 29177954,18408561 81502 55511 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SJ000044511 CHEMBL592124 81503 55512 GAA 2548 DRUGGABLE GENOME, ENZYME GNF-PF-4322 CHEMBL604100 81504 55513 BRCA2 675 CLINICALLY ACTIONABLE Irinotecan IRINOTECAN 26842236 81505 55514 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE ORAL CONTRACEPTIVE 15763593 81506 55515 RGS5 8490 NA leucovorin LEUCOVORIN 25069475 81507 55516 CASP8 841 DRUGGABLE GENOME, PROTEASE, ENZYME, CLINICALLY ACTIONABLE inhibitor 178103122 EMRICASAN 81508 55517 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Dihydropyrrolopyrazole derivative 1 81509 55518 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1201572 ETANERCEPT 81512 55519 TARDBP 23435 TUMOR SUPPRESSOR SJ000066425 CHEMBL600255 81513 55520 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME (S)-THIORPHAN (S)-THIORPHAN 81514 55521 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME AMBENONIUM AMBENONIUM 81516 55522 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Heterocyclic derivative 11 81518 55523 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 20 81519 55524 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Nalbuphine NALBUPHINE 81520 55525 ALDH1A1 216 DRUGGABLE GENOME, ENZYME LY-367265 CHEMBL1079460 81523 55526 ALDH1A1 216 DRUGGABLE GENOME, ENZYME TYRPHOSTIN A9 TYRPHOSTIN A9 81524 55527 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME GW441756X GW441756X 81525 55528 PDE4A 5141 DRUGGABLE GENOME, ENZYME LEO-32731 81526 55529 MAPT 4137 DRUGGABLE GENOME RESVERATROL RESVERATROL 81527 55530 AKR1B1 231 DRUGGABLE GENOME, ENZYME RANIRESTAT RANIRESTAT 81528 55531 PRKACA 5566 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE SB-202190 SB-202190 81529 55532 CBX1 10951 NA TCMDC-124176 CHEMBL588038 81532 55533 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE TDR77578 CHEMBL1364172 81534 55534 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor 135649662 81535 55535 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE DIPHENOXYLATE DIPHENOXYLATE 81536 55536 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME OSI-632 OSI-632 81537 55537 RACGAP1 29127 NA FAGARONINE FAGARONINE 81538 55538 HEXB 3074 ENZYME RABEPRAZOLE RABEPRAZOLE 9593221 81539 55539 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME ALSTERPAULLONE ALSTERPAULLONE 81541 55540 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649924 81542 55541 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DITHIAZANINE IODIDE DITHIAZANINE IODIDE 81545 55542 MYD88 4615 CLINICALLY ACTIONABLE ST2825 81546 55543 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor PLX3397 PEXIDARTINIB 81547 55544 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Sorafenib SORAFENIB 23629727,25363205 81548 55545 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE REL-3,5-DICAFFEOYLQUINIC ACID CHEMBL249447 22921742 81550 55546 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-45174 CHEMBL221047 17432842 81551 55547 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR IMMUNOTOXIN 7670112 81552 55548 ADRM1 11047 ENZYME inhibitor CHEMBL2103884 OPROZOMIB 81553 55549 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Palbociclib PALBOCICLIB 81554 55550 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ISOKAEMPFERIDE ISOKAEMPFERIDE 81555 55551 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PHENACYL CHLORIDE PHENACYL CHLORIDE 81556 55552 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-123984 CHEMBL532909 81559 55553 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE unspecified ERBB3 antibody 27196767 81560 55554 TUBB 203068 DRUGGABLE GENOME inhibitor 178103419 ERIBULIN 81561 55555 BRCA2 675 CLINICALLY ACTIONABLE Rucaparib RUCAPARIB 26779812,27002934 81562 55556 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME PICTILISIB PICTILISIB 81563 55557 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE inhibitor HESPERADIN HESPERADIN 19035792 81564 55558 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Talacotuzumab TALACOTUZUMAB 81565 55559 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME HARMOL HARMOL 81566 55560 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565923 81567 55561 AKR1D1 6718 DRUGGABLE GENOME, ENZYME cholic acid 81568 55562 PBK 55872 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, ENZYME PHA-767491 CHEMBL225519 81569 55563 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL70418 CLOBAZAM 81570 55564 PIK3C2A 5286 ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, TRANSPORTER inhibitor BEZ235 DACTOLISIB 81571 55565 APOBEC3G 60489 ENZYME, DRUGGABLE GENOME CY-208243 CHEMBL313737 81572 55566 TUBA3D 113457 DRUGGABLE GENOME CHEMBL2103826 DAVUNETIDE 81574 55567 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Imatinib IMATINIB 26758680 81579 55568 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 mycophenolic acid 24220207 81580 55569 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE CEP-2563 DIHYDROCHLORIDE 15292715 81581 55570 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PD-0166285 PD-0166285 81582 55571 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE 6-MERCAPTOPURINE MERCAPTOPURINE 16614955 81584 55572 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME WORTMANNIN WORTMANNIN 81585 55573 PTGS1 5742 ENZYME, DRUGGABLE GENOME DIFLUNISAL DIFLUNISAL 81586 55574 PTK6 5753 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, KINASE, TYROSINE KINASE, ENZYME TAK-715 TAK-715 81589 55575 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HER-2 Protein AutoVac 81590 55576 CAMK2D 817 TRANSCRIPTION FACTOR, TRANSPORTER, ENZYME, ION CHANNEL, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME 681640 CHEMBL379975 81591 55577 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE DAUNOMYCIN DAUNORUBICIN 10510309 81592 55578 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Dabrafenib DABRAFENIB 81593 55579 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE DIHYDROXIDINE DIHYDROXIDINE 81594 55580 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE LGK974 WNT-974 24277854 81595 55581 RAPGEF3 10411 ENZYME DIPYRIDAMOLE DIPYRIDAMOLE 81596 55582 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR MERCAPTOPURINE MERCAPTOPURINE 81598 55583 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE METHYL 4-(3-METHOXYBENZAMIDO)BENZOATE CHEMBL1214407 81599 55584 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ILORASERTIB ILORASERTIB 81600 55585 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ISOETHARINE MESYLATE ISOETHARINE MESYLATE 81601 55586 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER SPIRONOLACTONE SPIRONOLACTONE 16740618 81602 55587 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME 3-HYDROXYANTHRANILIC ACID CHEMBL445304 81603 55588 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME PROSTAGLANDIN E1 8213257 81604 55589 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR TCMDC-123532 CHEMBL547833 81605 55590 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Telapristone 81606 55591 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE ETHACRYNIC ACID ETHACRYNIC ACID 81607 55592 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CP-31398 26250460 81609 55593 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE AMPEROZIDE HYDROCHLORIDE AMPEROZIDE HYDROCHLORIDE 81611 55594 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE AZD2461 27550455 81612 55595 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Trimegestone/ethinyl estradiol 81613 55596 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE BYL719 ALPELISIB 27604488 81615 55597 GSTM1 2944 DRUGGABLE GENOME, ENZYME CPT-11 IRINOTECAN HYDROCHLORIDE 16865249 81616 55598 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW441756X GW441756X 81617 55599 CXCL8 3576 DRUGGABLE GENOME METHYLENE BLUE 12500513 81618 55600 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SERICETIN DIACETATE SERICETIN DIACETATE 81620 55601 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE venlafaxine VENLAFAXINE 18695978 81621 55602 PSMB10 5699 PROTEASE, DRUGGABLE GENOME CARFILZOMIB CARFILZOMIB 24524217 81622 55603 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 404859050 81623 55604 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL605 PROCAINAMIDE HYDROCHLORIDE 81624 55605 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 81625 55606 ILK 3611 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME US8754233, 2-(3-Amino-1H-pyrazol-4-yl)-5-fluoro-benzothiazole-6-sulfonic acid amide 81627 55607 GAA 2548 DRUGGABLE GENOME, ENZYME GNF-PF-5037 CHEMBL585828 81628 55608 PAK1 5058 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME inhibitor 249565832 81629 55609 MAPT 4137 DRUGGABLE GENOME KAEMPFEROL KAEMPFEROL 81632 55610 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER URSODEOXYCHOLIC ACID 15885361 81633 55611 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Oxandrolone OXANDROLONE 81634 55612 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME CRS-207 81635 55613 CTH 1491 ENZYME 5-Hydrazino-1H-tetrazole 81636 55614 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650620 81637 55615 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE GLIMEPIRIDE GLIMEPIRIDE 14686960 81639 55616 PTK2 5747 TYROSINE KINASE, DRUGGABLE GENOME, KINASE, G PROTEIN COUPLED RECEPTOR, ENZYME LINIFANIB LINIFANIB 81641 55617 ACTR2 10097 NA MCP-1 16004967 81643 55618 CHUK 1147 SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR 2,6-DIDEHYDROPEPEROMIN B 2,6-DIDEHYDROPEPEROMIN B 19559609 81644 55619 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 249565637 BMS-911543 81645 55620 TNFRSF1B 7133 DRUGGABLE GENOME DIDANOSINE DIDANOSINE 9430255 81646 55621 PDE4D 5144 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL190 THEOPHYLLINE 81647 55622 ETS2 2114 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR gemcitabine GEMCITABINE 31616045 81648 55623 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 AMOXICILLIN AMOXICILLIN 22931300 81649 55624 HTT 3064 DRUGGABLE GENOME FUCHSIN, BASIC FUCHSIN, BASIC 81650 55625 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR MITONAFIDE MITONAFIDE 81652 55626 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR GIVINOSTAT GIVINOSTAT 81653 55627 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor BYL719 ALPELISIB 81656 55628 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR angiotensin II 10594793 81657 55629 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR TRICLOFENOL TRICLOFENOL 81659 55630 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DIHYDROCAPSAICIN DIHYDROCAPSAICIN 81660 55631 PTGS1 5742 ENZYME, DRUGGABLE GENOME NEPAFENAC NEPAFENAC 81662 55632 UGT1A10 54575 DRUGGABLE GENOME, ENZYME risperidone RISPERIDONE 81663 55633 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-A7 81664 55634 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE BENFLUOREX HYDROCHLORIDE BENFLUOREX HYDROCHLORIDE 81665 55635 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 siponimod SIPONIMOD 81666 55636 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER hydroxocobalamin HYDROXOCOBALAMIN 81667 55637 CACNA1H 8912 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL2103836 IMAGABALIN 81668 55638 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-Figure3bI 81669 55639 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Cycloalkyl nitrile pyrazole carboxamide derivative 1 81671 55640 ERCC1 2067 CLINICALLY ACTIONABLE, DNA REPAIR PLATINUM COMPOUND 19488864 81672 55641 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME DIHYDROGAMBOGIC ACID DIHYDROGAMBOGIC ACID 81675 55642 POLI 11201 DNA REPAIR SANGUINARIUM CHLORIDE SANGUINARIUM CHLORIDE 81676 55643 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE MK-2461 MK-2461 81679 55644 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 252166594 VS-5584 81680 55645 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-12 81681 55646 PNP 4860 ENZYME, DRUGGABLE GENOME Forodesine FORODESINE 81682 55647 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL1946170 REGORAFENIB 81684 55648 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME DSP-8658 81685 55649 PTGS2 5743 DRUGGABLE GENOME, ENZYME NS-398 NS-398 21775152,19172146,16480277,25453792 81686 55650 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE AT9283 AT-9283 81687 55651 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL970 HALAZEPAM 81688 55652 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE Acebilustat ACEBILUSTAT 81689 55653 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL CC8464 81690 55654 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL3545282 KC-706 81691 55655 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE midostaurin MIDOSTAURIN 81692 55656 KCNA3 3738 DRUGGABLE GENOME, ION CHANNEL blocker 135652277 81693 55657 HDGF 3068 DRUGGABLE GENOME, GROWTH FACTOR PROTEIN KINASE C INHIBITOR 11149024 81694 55658 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Succinylcholine SUXAMETHONIUM 81696 55659 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE TRICHOSTATIN TRICHOSTATIN 19966789 81697 55660 RAPGEF3 10411 ENZYME 1,4-DIMETHOXYANTHRAQUINONE 1,4-DIMETHOXYANTHRAQUINONE 81699 55661 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR antagonist 135650883 RALOXIFENE 81700 55662 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR 2-CHLOROADENOSINE CHEMBL285819 81702 55663 POLI 11201 DNA REPAIR DNDI1417149 CHEMBL1622802 81705 55664 TUBB2B 347733 DRUGGABLE GENOME inhibitor CHEMBL1743082 TRASTUZUMAB EMTANSINE 81708 55665 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE EP-51389 81713 55666 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CHEMBL1257 ENFLURANE 81715 55667 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor SELUMETINIB SELUMETINIB 81716 55668 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-32e 81717 55669 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 WIN-55212-2 WIN-552122 81719 55670 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE erythromycin ERYTHROMYCIN 18695978 81720 55671 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE AP32788 81722 55672 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME BERKELEYTRIONE BERKELEYTRIONE 17970594 81723 55673 USP1 7398 DNA REPAIR, PROTEASE, ENZYME L-165041 CHEMBL153057 81724 55674 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor GDC-0941 PICTILISIB 81725 55675 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE THIOPHENE THIOPHENE 81726 55676 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME D-DOPA CHEMBL211670 81727 55677 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME NORHARMANE NORHARMANE 81729 55678 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor BI847325 81730 55679 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME SB-203580 SB-203580 81731 55680 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE AVX-470 81732 55681 HMGCR 3156 ENZYME, DRUGGABLE GENOME PRAVASTATIN PRAVASTATIN 81733 55682 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist CHEMBL2062262 METARAMINOL BITARTRATE 81734 55683 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-15 81735 55684 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor BAY86-9766 REFAMETINIB 81736 55685 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME CHEMBL1372 OXIGLUTATIONE 81737 55686 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME Sulfasalazine SULFASALAZINE 81738 55687 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Ad5CMV-p53 gene 15608394 81739 55688 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-124557 CHEMBL530682 81742 55689 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME 7-METHOXY-BAPTIGENIN CHEMBL583578 81743 55690 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 223366076 81745 55691 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME DEMECARIUM BROMIDE 81747 55692 GMNN 51053 DRUGGABLE GENOME ROTENONE ROTENONE 81748 55693 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR NSC-319994 CHEMBL1329443 81750 55694 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE SNS-314 SNS-314 81751 55695 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR LEVONORGESTREL LEVONORGESTREL 81752 55696 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME ALPRAZOLAM ALPRAZOLAM 22137933 81754 55697 ABCC1 4363 DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER CYTOKINES 15654950 81756 55698 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652751 81757 55699 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200328 DULOXETINE HYDROCHLORIDE 81758 55700 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 363894201 TENALISIB 81759 55701 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CHLOROTHALONIL CHLOROTHALONIL 81760 55702 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PF-4989216 24240111 81761 55703 CYP4B1 1580 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME TCDD 2829388 81762 55704 BAZ2B 29994 NA OXOGLAUCINE OXOGLAUCINE 81764 55705 HDAC11 79885 DRUGGABLE GENOME, ENZYME 4-(4-AMINOPHENYL)BUTANOIC ACID CHEMBL1650245 24044874 81765 55706 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL3707353 RG7893 81769 55707 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Bb21217 81770 55708 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ARQ 087 81772 55709 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-123650 CHEMBL580727 81773 55710 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 329968373 81774 55711 RXRG 6258 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME TRETINOIN TRETINOIN 81775 55712 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 81778 55713 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME HAEMATOXYLIN HAEMATOXYLIN 81780 55714 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL modulator CHEMBL1200349 81781 55715 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME deutetrabenazine DEUTETRABENAZINE 81782 55716 POSTN 10631 DRUGGABLE GENOME ANTISERUM 10404027 81783 55717 ALOX15 246 ENZYME, DRUGGABLE GENOME NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 17869117 81784 55718 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TAS3681 81785 55719 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME NSC-37173 CHEMBL221733 81788 55720 CYB5R2 51700 DRUGGABLE GENOME rasburicase RASBURICASE 81790 55721 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITOR 26561417 81791 55722 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ARN-509 APALUTAMIDE 81792 55723 TUBB2B 347733 DRUGGABLE GENOME CHEMBL2103826 DAVUNETIDE 81794 55724 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DOCOSATETRA-7Z,10Z,13Z,16Z-ENOYL ETHANOLAMIDE CHEMBL321585 81796 55725 LTB4R 1241 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100358 81799 55726 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME GNF-PF-5159 CHEMBL1493528 81800 55727 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Tricyclic heterocycle derivative 1 81801 55728 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL3545272 LAS190792 81802 55729 HSPA4 3308 NA LITHIUM LITHIUM 12732732,16179524,16797496 81803 55730 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE TAK-733 TAK-733 26439693 81804 55731 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER FURAZOLIDONE FURAZOLIDONE 81805 55732 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME doxorubicin DOXORUBICIN 29938344,20179710 81807 55733 BCR 613 TUMOR SUPPRESSOR, SERINE THREONINE KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE, KINASE, ENZYME, DRUGGABLE GENOME Busulfan BUSULFAN 81809 55734 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody CIXUTUMUMAB CIXUTUMUMAB 81811 55735 POLI 11201 DNA REPAIR CATECHOL CATECHOL 81814 55736 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE LY3023414 SAMOTOLISIB 27439478 81815 55737 ALDH1A1 216 DRUGGABLE GENOME, ENZYME DNDI1417076 CHEMBL1526167 81816 55738 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME AZD-8165 AZD-8165 81817 55739 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CENISERTIB CENISERTIB 81818 55740 MSLN 10232 SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME SS1(DSFV)-PE38 81819 55741 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME U0126 23298836 81820 55742 PLA2G10 8399 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2105659 VARESPLADIB METHYL 81821 55743 SLC29A4 222962 EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 135650099 CIMETIDINE 81822 55744 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME PAZOPANIB PAZOPANIB 81823 55745 IMPDH1 3614 ENZYME, DRUGGABLE GENOME mycophenolate mofetil 20649757,20136638,21142914,20679962,17851563,22960765 81825 55746 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL3039518 BATEFENTEROL 81826 55747 MPHOSPH8 54737 NA PROMETHAZINE HYDROCHLORIDE PROMETHAZINE HYDROCHLORIDE 81827 55748 HDAC10 83933 ENZYME, DRUGGABLE GENOME, DNA REPAIR SUBEROHYDROXAMIC ACID SUBEROHYDROXAMIC ACID 16921367 81828 55749 STK11 6794 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, ENZYME, TUMOR SUPPRESSOR, DRUG RESISTANCE Phenformin PHENFORMIN 26574479 81829 55750 SLC12A5 57468 DRUGGABLE GENOME, TRANSPORTER BUMETANIDE BUMETANIDE 81830 55751 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178103477 81831 55752 NRG1 3084 GROWTH FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE CARBOPLATIN CARBOPLATIN 23390248 81832 55753 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME US8598210, Table XV, 5 81835 55754 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Tacrine-dihydropyridine hybrid derivative 1 81836 55755 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME SRT3025 81840 55756 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL16 PHENYTOIN 81841 55757 MAPT 4137 DRUGGABLE GENOME ZAPA ZAPA 81842 55758 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME REDIOCIDE A REDIOCIDE A 22650618 81843 55759 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-42 81845 55760 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME N/A 26768652 81846 55761 PMEL 6490 DRUGGABLE GENOME IFN 15980237 81847 55762 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Dabrafenib DABRAFENIB 81849 55763 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME INDIGO INDIGO 81850 55764 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Aryl alkanolamine derivative 1 81851 55765 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CAPSAZEPINE CAPSAZEPINE 81852 55766 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LEE011 RIBOCICLIB 81853 55767 LAMA4 3910 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 81855 55768 NPPC 4880 DRUGGABLE GENOME, HORMONE ACTIVITY BMN-111 VOSORITIDE 81856 55769 ALOX5 240 DRUGGABLE GENOME, ENZYME PF-4191834 PF-4191834 81857 55770 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX 1-O-ACETYLGEOPYXIN A CHEMBL1902074 81860 55771 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME GNF-PF-388 CHEMBL582278 81861 55772 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE Tezacaftor TEZACAFTOR 81863 55773 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX SJ000100732 CHEMBL592819 81865 55774 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE inhibitor 178102312 81866 55775 GAA 2548 DRUGGABLE GENOME, ENZYME NODAKENIN NODAKENIN 81867 55776 NR1H2 7376 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME gefitinib GEFITINIB 31664190 81868 55777 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-19 81869 55778 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650109 CLOBENPROPIT 81871 55779 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR JNK INHIBITOR VIII CHEMBL210618 81872 55780 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-135810 CHEMBL1605629 81874 55781 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR UMECLIDINIUM BROMIDE UMECLIDINIUM BROMIDE 19317446 81875 55782 BCHE 590 DRUGGABLE GENOME, ENZYME Tetra-hydro-isoquinoline derivative 3 81876 55783 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 404859074 81877 55784 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Osimertinib OSIMERTINIB 81878 55785 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE MK-2206 MK-2206 81879 55786 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME PAC-1 PAC-1 19708658,16936720 81880 55787 EML4 27436 CLINICALLY ACTIONABLE, KINASE TPX-0005 81881 55788 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DICHLORVOS DICHLORVOS 81883 55789 NOS2 4843 DRUGGABLE GENOME, ENZYME CAPTOPRIL CAPTOPRIL 15680268 81886 55790 BAZ2B 29994 NA GOSSYPOL GOSSYPOL 81887 55791 GMNN 51053 DRUGGABLE GENOME SPICLOMAZINE SPICLOMAZINE 81889 55792 IRAK4 51135 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 249565764 81891 55793 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NAFRONYL OXALATE NAFRONYL OXALATE 81892 55794 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR PHA-767491 CHEMBL225519 81894 55795 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 quinidine QUINIDINE 11353757,9187528 81900 55796 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE BMS-387032 BMS-387032 81901 55797 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 178102316 CHEMBL1908395 81904 55798 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME antibody 249565931 LABETUZUMAB 81905 55799 MAPT 4137 DRUGGABLE GENOME ATHRAQUINONES A ATHRAQUINONES A 81906 55800 GJA1 2697 ION CHANNEL VITAMIN A 16292552 81907 55801 DNER 92737 NA GS-5829 ALOBRESIB 81911 55802 DDR2 4921 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TYROSINE KINASE ERLOTINIB ERLOTINIB 22328973,23932362,18938156 81913 55803 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ETHACRYNIC ACID ETHACRYNIC ACID 81914 55804 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL CNS-7056 REMIMAZOLAM 81915 55805 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE GV1001 TERTOMOTIDE 81916 55806 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE SAFINAMIDE SAFINAMIDE 81917 55807 ALDH1A1 216 DRUGGABLE GENOME, ENZYME KAVAIN KAVAIN 81918 55808 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME AZD6244 SELUMETINIB 81919 55809 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYL ISOBUTYL KETONE METHYL ISOBUTYL KETONE 81920 55810 HSPA4 3308 NA VITAMIN C 12927909 81923 55811 PGF 5228 GROWTH FACTOR, DRUGGABLE GENOME inhibitor CHEMBL2108313 CONBERCEPT 81924 55812 CYP2R1 120227 CYTOCHROME P450, DRUGGABLE GENOME, ENZYME peginterferon alfa-2b 81926 55813 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CAPTAMINE CAPTAMINE 81927 55814 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PRIMIDONE PRIMIDONE 81931 55815 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE ANABOLIC STEROID 12943056 81935 55816 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 310264754 OMIPALISIB 81937 55817 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME GW441756X GW441756X 81938 55818 TXK 7294 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 249565826 81939 55819 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE RISPERIDONE RISPERIDONE 17052361 81940 55820 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 7-CHLOROKYNURENIC ACID 7-CHLOROKYNURENIC ACID 81941 55821 PRKCB 5579 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSPORTER activator 178104015 81942 55822 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Imidazo cyclohexylamine derivative 2 81943 55823 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor CHEMBL3137318 TALAZOPARIB TOSYLATE 81944 55824 COMT 1312 DRUGGABLE GENOME, ENZYME risperidone RISPERIDONE 19451915,22935916 81946 55825 BAZ2B 29994 NA SJ000128325 CHEMBL602718 81947 55826 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Dihydropyrido pyrazinone compound 2 81950 55827 ATAD5 79915 NA CID 1225609 CHEMBL444376 81952 55828 LSS 4047 ENZYME, DRUGGABLE GENOME inhibitor 178103328 81954 55829 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417614 CHEMBL1567571 81955 55830 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE CYCLOSERINE CYCLOSERINE 81957 55831 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CARBOQUONE CARBOQUONE 81959 55832 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 178102290 AT-7519 81960 55833 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING ROTENONE ROTENONE 16680159 81962 55834 MAPT 4137 DRUGGABLE GENOME A-23187 CALCIMYCIN 81963 55835 LTA 4049 DRUGGABLE GENOME abacavir ABACAVIR 81966 55836 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR HALS 1283360 81969 55837 TSPO 706 DRUGGABLE GENOME LORAZEPAM LORAZEPAM 81970 55838 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE CEDIRANIB CEDIRANIB 81971 55839 ALDH1A1 216 DRUGGABLE GENOME, ENZYME SB-415286 CHEMBL322970 81972 55840 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME RDEA119 81973 55841 PTGS1 5742 ENZYME, DRUGGABLE GENOME NAPROXCINOD NAPROXCINOD 81974 55842 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME PMID28270021-Compound-WO2016054807Example1 81977 55843 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PATIDEGIB PATIDEGIB 22550175 81979 55844 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-57 81980 55845 KDM4A 9682 DRUGGABLE GENOME, ENZYME SJ000018298 CHEMBL591412 81981 55846 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LIOTHYRONINE LIOTHYRONINE 22931300 81982 55847 HNF1A 6927 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR opioids 26233334 81983 55848 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME OXIDOPAMINE HYDROCHLORIDE OXIDOPAMINE HYDROCHLORIDE 81985 55849 UNC13D 201294 NA Emapalumab-lzsg EMAPALUMAB 81986 55850 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME HEMICHOLINIUM-3 HEMICHOLINIUM-3 81988 55851 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE allosteric modulator 178102576 CHELERYTHRINE 81990 55852 RAB9A 9367 ENZYME, DRUGGABLE GENOME NSC-102045 CHEMBL483633 81991 55853 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR PYRITHIONE ZINC PYRITHIONE ZINC 81992 55854 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE PD-0166285 PD-0166285 81993 55855 PTGES2 80142 ENZYME inhibitor 252827470 81994 55856 PTGES 9536 DRUGGABLE GENOME, ENZYME CELECOXIB CELECOXIB 19884011,24183739,19053751 81995 55857 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE APG-1252 81996 55858 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AR-12286 VEROSUDIL 81998 55859 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565596 FILGOTINIB 81999 55860 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME Dihydrothieno [2,3-e]indazole derivative 4 82000 55861 GART 2618 ENZYME, DRUGGABLE GENOME LOMETREXOL LOMETREXOL 22243528 82001 55862 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR Blisibimod BLISIBIMOD 82002 55863 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL2105738 GALETERONE 82003 55864 ATXN2 6311 NA INDIRUBIN-3-MONOXIME INDIRUBIN-3-MONOXIME 82006 55865 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ELETRIPTAN ELETRIPTAN 82007 55866 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor MOTESANIB MOTESANIB 82008 55867 MPHOSPH8 54737 NA CHLORPROMAZINE HYDROCHLORIDE CHLORPROMAZINE HYDROCHLORIDE 82009 55868 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor VATALANIB VATALANIB 82010 55869 HCN3 57657 DRUGGABLE GENOME, ION CHANNEL blocker 135652734 82011 55870 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR FINASTERIDE FINASTERIDE 82012 55871 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE IMATINIB IMATINIB 82013 55872 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BERGAMOTTIN BERGAMOTTIN 82015 55873 PTGES 9536 DRUGGABLE GENOME, ENZYME CURCUMIN CURCUMIN 25686392 82018 55874 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SHIKONIN SHIKONIN 82019 55875 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR ROMIDEPSIN ROMIDEPSIN 82020 55876 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME E-2609 ELENBECESTAT 24556009 82021 55877 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME TYRPHOSTIN 47 TYRPHOSTIN 47 82022 55878 ITGB5 3693 CELL SURFACE, DRUGGABLE GENOME antagonist CHEMBL1743032 INTETUMUMAB 82023 55879 LIG1 3978 DNA REPAIR, DRUGGABLE GENOME BLEOMYCIN BLEOMYCIN 82025 55880 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER codeine CODEINE 22398969 82027 55881 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR NOREPINEPHRINE NOREPINEPHRINE 82028 55882 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR pertuzumab PERTUZUMAB 82029 55883 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TREQUINSIN HYDROCHLORIDE TREQUINSIN HYDROCHLORIDE 82030 55884 SLC22A5 6584 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME CARNITINE CARNITINE 21422191 82031 55885 COMT 1312 DRUGGABLE GENOME, ENZYME morphine MORPHINE 11054766,12595695,28006928,15927391,23686330,21398039,23302985,26902643,29474345,23773341,9259381,25155931,25185591,19514130,28745577,27027462 82032 55886 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PMID26924192-Compound-22 82035 55887 TNFRSF14 8764 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME 178101591 82036 55888 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651350 TAMSULOSIN 82037 55889 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL424133 LY-518674 82038 55890 ITGB2 3689 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL2109224 ROVELIZUMAB 82039 55891 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL agonist 178100898 82040 55892 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CLOMETHIAZOLE CLOMETHIAZOLE 82042 55893 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE 5-AZACYTIDINE AZACITIDINE 2425967 82044 55894 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE GEFITINIB GEFITINIB 20151670 82047 55895 CLOCK 9575 ENZYME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX lithium LITHIUM 21047205 82048 55896 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE S-222611 S-222611 24837299,25434923 82049 55897 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE PHA-767491 CHEMBL225519 82051 55898 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NITROFURAZONE NITROFURAZONE 82053 55899 RAPGEF3 10411 ENZYME MYRICETIN MYRICETIN 82056 55900 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE TAMATINIB R-406 82057 55901 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE LETROZOLE LETROZOLE 18256205 82059 55902 CLDN18 51208 KINASE, DRUGGABLE GENOME CAR-CLD18 T cell 82060 55903 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PF-03446962 ASCRINVACUMAB 21467543 82061 55904 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 178100867 82062 55905 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX FENTICLOR FENTICLOR 82063 55906 F2R 2149 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE antagonist 178100505 82064 55907 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR CHLOROTHALONIL CHLOROTHALONIL 82066 55908 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor CUDC-101 CUDC-101 82068 55909 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PURPUROGALLIN PURPUROGALLIN 82069 55910 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Arformoterol ARFORMOTEROL 82071 55911 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE KOPARIN KOPARIN 82072 55912 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR HALOPERIDOL HALOPERIDOL 12393228 82073 55913 GGPS1 9453 DRUGGABLE GENOME, ENZYME inhibitor 135650017 CHEMBL494897 82075 55914 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SP-600125 SP-600125 82077 55915 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR BAICALEIN BAICALEIN 82078 55916 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR sirolimus SIROLIMUS 22094953 82079 55917 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME NSC-601359 CHEMBL1306524 82080 55918 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME VENLAFAXINE VENLAFAXINE 82081 55919 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Ranolazine RANOLAZINE 82082 55920 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NANAOMYCIN NANAOMYCIN 82084 55921 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL738 THIOPENTAL SODIUM 82085 55922 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE antagonist 135650686 82087 55923 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-P5 82091 55924 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHOLECALCIFEROL CHOLECALCIFEROL 82092 55925 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME agonist 178103125 82093 55926 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LAMOTRIGINE LAMOTRIGINE 22931300 82094 55927 ALOX15 246 ENZYME, DRUGGABLE GENOME DICHLOROPHEN DICHLOROPHEN 82095 55928 CBFB 865 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR D-DOPA CHEMBL211670 82096 55929 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 381118846 82097 55930 P4HA1 5033 DRUGGABLE GENOME, ENZYME Lufironil LUFIRONIL 82098 55931 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PAPAVERINE PAPAVERINE 82099 55932 MAP3K5 4217 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSCRIPTION FACTOR, ENZYME inhibitor 404859049 82103 55933 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME PYROGALLOL PYROGALLOL 82105 55934 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor ORANTINIB ORANTINIB 82106 55935 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FISETIN FISETIN 8759170 82109 55936 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME Pegfilgrastim PEGFILGRASTIM 82110 55937 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL Pyrimidine derivative 1 82111 55938 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PLX8394 PLX8394 82113 55939 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR 2-HYDROXYPHENAZINE 5,10-DIOXIDE CHEMBL179611 82115 55940 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651741 82116 55941 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist CHEMBL1767407 DENUFOSOL TETRASODIUM 82117 55942 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme24Paprotrain 82118 55943 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER GNF-PF-1852 CHEMBL533293 82119 55944 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE COVA322 82123 55945 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE PMID26394986-Compound-11 82125 55946 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER GARLIC GARLIC 11466175 82126 55947 P3H3 10536 DRUGGABLE GENOME sertraline SERTRALINE 30324302 82127 55948 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME LINIFANIB LINIFANIB 82128 55949 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE SUNITINIB SUNITINIB 19755855,19366796,21482694,18955458 82129 55950 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3545145 WX-554 82130 55951 TFF2 7032 DRUGGABLE GENOME VT-111 82131 55952 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR VITAMIN K 1336373 82132 55953 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ILORASERTIB ILORASERTIB 82133 55954 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE lomitapide LOMITAPIDE 82134 55955 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 223366039 82136 55956 ALDH7A1 501 ENZYME, DRUGGABLE GENOME NM-702 82137 55957 MAPT 4137 DRUGGABLE GENOME NSC-601359 CHEMBL1306524 82139 55958 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BETA-HYDRASTINE CHEMBL462731 82140 55959 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR allosteric modulator 135650027 82141 55960 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENMEDIPHAM PHENMEDIPHAM 82143 55961 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME BL-8040 BKT140 82145 55962 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-3012 CHEMBL582715 82147 55963 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Docetaxel DOCETAXEL 23801166,27052654,25185099 82148 55964 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX agonist CHEMBL705 ALITRETINOIN 82150 55965 PRDX5 25824 ENZYME Motexafin gadolinium 82152 55966 ATXN2 6311 NA SJ000113257 CHEMBL528694 82153 55967 GLCCI1 113263 NA glucocorticoids 21991891 82154 55968 USP1 7398 DNA REPAIR, PROTEASE, ENZYME HISTAMINE HISTAMINE 82155 55969 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DASATINIB DASATINIB 82158 55970 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102568 82161 55971 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PHENDIMETRAZINE PHENDIMETRAZINE 82163 55972 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-7 82166 55973 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME AMIFOSTINE AMIFOSTINE 12751907 82167 55974 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME inhibitor YM155 82170 55975 GSR 2936 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, ENZYME ORAL CONTRACEPTIVE 12340474 82172 55976 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Pembrolizumab PEMBROLIZUMAB 82173 55977 CES2 8824 DRUGGABLE GENOME, ENZYME mycophenolic acid 24220207 82175 55978 ADAM10 102 ENZYME, CELL SURFACE, TRANSPORTER, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE Aderbasib ADERBASIB 82177 55979 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME GSK-269962A GSK-269962A 82178 55980 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SB-202190 SB-202190 82179 55981 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor 315661265 82180 55982 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ALCAFTADINE ALCAFTADINE 82181 55983 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor PI-103 PI-103 82184 55984 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LONIDAMINE LONIDAMINE 82185 55985 BMP7 655 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR daunorubicin DAUNORUBICIN 26590194 82186 55986 TPBG 7162 CELL SURFACE, DRUGGABLE GENOME antibody 374883835 82187 55987 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DIPHENHYDRAMINE DIPHENHYDRAMINE 22931300 82188 55988 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME PMID27967267-Compound-36 82189 55989 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201002 CARTEOLOL HYDROCHLORIDE 82192 55990 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor 249565728 82193 55991 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PEG-SN38 82194 55992 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL2096631 CLORAZEPATE DIPOTASSIUM 82195 55993 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME (2S)-2'-METHOXYKURARINONE CHEMBL496451 18565755 82196 55994 HGF 3082 PROTEASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, GROWTH FACTOR, KINASE, ENZYME inhibitor CHEMBL1743018 FICLATUZUMAB 82197 55995 EIF3A 8661 NA cisplatin CISPLATIN 23127338 82198 55996 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PHA-793887 PHA-793887 82199 55997 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER GNF-PF-2968 CHEMBL582473 82200 55998 SLC25A4 291 DRUGGABLE GENOME, TRANSPORTER CLODRONATE CLODRONIC ACID 82201 55999 MGLL 11343 DRUGGABLE GENOME, ENZYME Carbamate derivative 12 82202 56000 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PX-866 SONOLISIB 22693357 82203 56001 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 BERBERINE CHLORIDE BERBERINE CHLORIDE 82204 56002 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 223366138 82206 56003 PDE4B 5142 DRUGGABLE GENOME, ENZYME HT-0712 HT-0712 82207 56004 BRD3 8019 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR inhibitor 187051820 82208 56005 MAPT 4137 DRUGGABLE GENOME TYRPHOSTIN 25 TYRPHOSTIN 25 82210 56006 NOS2 4843 DRUGGABLE GENOME, ENZYME rifampin RIFAMPIN 22341855 82211 56007 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TOXAPHENE TOXAPHENE 82212 56008 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR AUS-131 AUS-131 82213 56009 LGALS1 3956 KINASE, DRUGGABLE GENOME US8703720, Reference Compound 1 82215 56010 FZD5 7855 G PROTEIN COUPLED RECEPTOR, KINASE, CELL SURFACE antagonist CHEMBL2364652 VANTICTUMAB 82216 56011 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178102585 DOVITINIB 82218 56012 SOD1 6647 ENZYME, DRUGGABLE GENOME DOXYCYCLINE DOXYCYCLINE 82219 56013 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ANTI CD3 11599102 82220 56014 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME THYROXINE THYROXINE 82221 56015 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME EPIGALOCATECHIN GALLATE EPIGALOCATECHIN GALLATE 82223 56016 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME RESVERATROL RESVERATROL 16525036 82224 56017 FABP5 2171 NUCLEAR HORMONE RECEPTOR PMID27109571-Compound-31 82225 56018 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651002 82226 56019 ALDH1A1 216 DRUGGABLE GENOME, ENZYME BI-87E7 CHEMBL523200 82227 56020 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME SPINASAPONIN A METHYL ESTER SPINASAPONIN A METHYL ESTER 20951582 82228 56021 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ZINC 03369470 CHEMBL599013 82229 56022 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PHENYLBUTANOIC ACID PHENYLBUTANOIC ACID 24044874 82230 56023 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR TOREMIFENE TOREMIFENE 2147123 82231 56024 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR antagonist AT-406 AT-406 82233 56025 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DITHIAZANINE DITHIAZANINE 82234 56026 CDKN1A 1026 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME FLUTAMIDE FLUTAMIDE 16281084 82236 56027 ATAD5 79915 NA CID 4101591 CHEMBL428789 82237 56028 GSK3A 2931 DRUGGABLE GENOME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE, ENZYME AZAKENPAULLONE AZAKENPAULLONE 82239 56029 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL30219 METHOHEXITAL SODIUM 82240 56030 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 REMOXIPRIDE REMOXIPRIDE 22931300 82241 56031 BAZ2B 29994 NA inhibitor 252166518 82243 56032 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR inhibitor 363894217 VORUCICLIB 82244 56033 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TYROSINE KINASE INHIBITOR SU5402 21119661 82245 56034 CRTC2 200186 KINASE INK128 SAPANISERTIB 82246 56035 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE ABCIXIMAB ABCIXIMAB 82248 56036 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BIMU-1 82249 56037 PDE4B 5142 DRUGGABLE GENOME, ENZYME IPL455 82250 56038 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL blocker 178100875 PICROTOXIN 82251 56039 PDE4D 5144 DRUGGABLE GENOME, ENZYME diuretics 23778321 82252 56040 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-123764 CHEMBL533226 82253 56041 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME LY-2811376 LY-2811376 82255 56042 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE JNJ-7706621 JNJ-7706621 82256 56043 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME GOSSYPOL GOSSYPOL 82257 56044 TUBA1C 84790 DRUGGABLE GENOME NSC-753575 CHEMBL2036119 22543234 82259 56045 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME HALOBETASOL PROPIONATE 82260 56046 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565856 82261 56047 ALB 213 TRANSPORTER, DRUGGABLE GENOME COCHINCHINENIN C COCHINCHINENIN C 25734332 82262 56048 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR ACRIFLAVINE CHLORIDE ACRIFLAVINE 82263 56049 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Nilutamide NILUTAMIDE 82265 56050 NOS1 4842 DRUGGABLE GENOME, ENZYME ENZYME INHIBITOR 9595494 82266 56051 RGS4 5999 DRUGGABLE GENOME MITOXANTRONE MITOXANTRONE 82267 56052 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor 318164849 CDP840 82268 56053 SMN2 6607 DRUGGABLE GENOME GENISTEIN GENISTEIN 82270 56054 CASP1 834 DRUGGABLE GENOME, ENZYME, PROTEASE GNF-PF-67 CHEMBL578512 82271 56055 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor BAY80-6946 COPANLISIB 82272 56056 TLR7 51284 DRUGGABLE GENOME LOXORIBINE LOXORIBINE 82273 56057 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL3544906 BENZPHETAMINE HYDROCHLORIDE 82275 56058 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-124685 CHEMBL587579 82277 56059 FASN 2194 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE TAXOL PACLITAXEL 15657900 82279 56060 E2F1 1869 TRANSCRIPTION FACTOR PS-341 BORTEZOMIB 11489836 82280 56061 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE AESCULIOSIDE IIID AESCULIOSIDE IIID 20371180 82281 56062 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TOK-001 GALETERONE 82282 56063 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE Fostamatinib FOSTAMATINIB 82283 56064 MVK 4598 KINASE, ENZYME inhibitor 135650204 82284 56065 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ENTRECTINIB ENTRECTINIB 82287 56066 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 381744915 82288 56067 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE BEVACIZUMAB BEVACIZUMAB 26921265 82290 56068 GPR68 8111 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 385612200 82291 56069 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE highly active antiretroviral therapy (haart) 82292 56070 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BENZOTHIAZYL DISULFIDE BENZOTHIAZYL DISULFIDE 82293 56071 TP73 7161 DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR CDDP CISPLATIN 11689148 82297 56072 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SB-202190 SB-202190 22951114 82298 56073 PTGS2 5743 DRUGGABLE GENOME, ENZYME ETODOLAC ETODOLAC 82299 56074 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRICLOCARBAN TRICLOCARBAN 82300 56075 GAA 2548 DRUGGABLE GENOME, ENZYME ESCULETIN ESCULETIN 82301 56076 TNFSF13B 10673 DRUGGABLE GENOME, TRANSCRIPTION FACTOR antibody BELIMUMAB BELIMUMAB 82303 56077 PDE4A 5141 DRUGGABLE GENOME, ENZYME AN2728 CRISABOROLE 82304 56078 BRD9 65980 ENZYME inhibitor 315661231 82305 56079 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Tyrosine kinase inhibitor - NS 82307 56080 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME CARBINOXAMINE CARBINOXAMINE 82309 56081 CRBN 51185 ENZYME, DRUG RESISTANCE CC-220 IBERDOMIDE HYDROCHLORIDE 82310 56082 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE DC/I540/KLH vaccine 82311 56083 F7 2155 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 252166701 82313 56084 KDM4A 9682 DRUGGABLE GENOME, ENZYME S-166659 CHEMBL252417 82315 56085 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor BGJ398 INFIGRATINIB 82317 56086 GLS 2744 ENZYME CEFQUINOME CEFQUINOME 82319 56087 BIRC2 329 TUMOR SUPPRESSOR, KINASE, DRUGGABLE GENOME antagonist 223366043 82321 56088 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650533 LOXAPINE 82325 56089 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TCMDC-124059 CHEMBL530733 82327 56090 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Erlotinib ERLOTINIB 82329 56091 NR1D1 9572 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME agonist 310264682 SR9009 82332 56092 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME BI-87E7 CHEMBL523200 82334 56093 IL2RG 3561 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME INTERLEUKIN-2 82335 56094 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-19063 CHEMBL1310138 82337 56095 MT1A 4489 NA oxaliplatin OXALIPLATIN 24924344 82338 56096 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Bis-aminopyrimidine derivative 1 82339 56097 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 4-FORMYL-BENZOIC ACID CHEMBL113897 82340 56098 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME Tricyclic compound 9 82343 56099 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GW305074X GW305074X 82344 56100 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR HEMATOXYLIN HEMATOXYLIN 82347 56101 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 178101602 CRIZOTINIB 82348 56102 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Si306 27196762 82349 56103 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AMARANTH AMARANTH 82351 56104 PSMB5 5693 PROTEASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545432 IXAZOMIB CITRATE 82352 56105 PTPN1 5770 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, ENZYME, KINASE KQ-791 82354 56106 GJA3 2700 ION CHANNEL, TRANSPORTER inhibitor 178100972 CARBENOXOLONE 82357 56107 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME INAMRINONE INAMRINONE 82359 56108 AQP9 366 ION CHANNEL DHT ANDROSTANOLONE 15850448 82360 56109 IL24 11009 DRUGGABLE GENOME, KINASE INGN 242 82361 56110 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL408513 BELINOSTAT 82362 56111 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE VS-5584 VS-5584 23270925 82363 56112 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CEFOPERAZONE CEFOPERAZONE 22931300 82364 56113 GABPA 2551 TRANSCRIPTION FACTOR CSA CYCLOSPORINE 16612258 82365 56114 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178102745 82366 56115 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 363894208 ILORASERTIB 82367 56116 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METIXENE METHIXENE 82368 56117 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor 178103109 TRAMETINIB 82370 56118 EDN1 1906 HORMONE ACTIVITY, DRUGGABLE GENOME irbesartan IRBESARTAN 15188945 82371 56119 TYMSOS 494514 NA platinum PLATINUM 25677447 82372 56120 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR inhibitor 178102296 DORAMAPIMOD 82373 56121 GABBR2 9568 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL LESOGABERAN LESOGABERAN 82375 56122 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE DORAMAPIMOD DORAMAPIMOD 82377 56123 CRTC2 200186 KINASE NVP-BEZ235 DACTOLISIB 82378 56124 CCNA2 890 DRUGGABLE GENOME, KINASE GENISTEIN GENISTEIN 9664138 82379 56125 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor AZD1480 AZD-1480 82380 56126 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME PIPERINE PIPERINE 82385 56127 CTSS 1520 DRUGGABLE GENOME, PROTEASE, ENZYME inhibitor 178103149 82387 56128 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER TERFENADINE TERFENADINE 10213372 82388 56129 TRPC4 7223 ION CHANNEL, KINASE, DRUGGABLE GENOME, CELL SURFACE activator 381744968 82389 56130 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ISOPROTERENOL ISOPROTERENOL 82390 56131 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR APICIDIN APICIDIN 19705846 82391 56132 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE KU-0063794 26546619 82392 56133 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER QPI-1002 TEPRASIRAN 82393 56134 GSTA1 2938 ENZYME, DRUGGABLE GENOME prednisone PREDNISONE 29938344,19448608 82395 56135 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE GM-CSF REGRAMOSTIM 12574393 82396 56136 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE salmeterol SALMETEROL 18695978 82398 56137 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 desloratadine DESLORATADINE 9187528 82399 56138 VKORC1 79001 DRUGGABLE GENOME, ENZYME fluindione FLUINDIONE 21883387 82400 56139 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME MLN-8054 MLN-8054 82401 56140 ATXN2 6311 NA SJ000119988 CHEMBL589694 82402 56141 CBR3 874 ENZYME, DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, CLINICALLY ACTIONABLE fluorouracil FLUOROURACIL 82403 56142 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE Anti-CD45 mabs 82404 56143 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Sonidegib SONIDEGIB 26546616,26823493,25759019,26124204 82405 56144 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE Everolimus EVEROLIMUS 26546619 82406 56145 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE ANTI-CD3 MONOCLONAL ANTIBODY 82407 56146 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME APOGOSSYPOL APOGOSSYPOL 19555126 82408 56147 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TRIFLUPERIDOL TRIFLUPERIDOL 82409 56148 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Gold-complexed thiosaccharide derivative 2 82410 56149 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR DRF 10945 82411 56150 PHKG2 5261 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE BAY-613606 CHEMBL541400 82412 56151 POLI 11201 DNA REPAIR SULFURETIN SULFURETIN 82413 56152 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL856 PRIMIDONE 82415 56153 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL FLURAZEPAM FLURAZEPAM 82416 56154 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TOZASERTIB TOZASERTIB 82417 56155 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE PURVALANOLA PURVALANOLA 82419 56156 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR CD271 18394312 82420 56157 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER 6-AZAURIDINE 6-AZAURIDINE 82421 56158 MERTK 10461 KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 363894214 SITRAVATINIB 82422 56159 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE KENPAULLONE KENPAULLONE 82424 56160 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME GO-6976 GO-6976 82425 56161 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME SEN0014196 82426 56162 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME LYCOPENE LYCOPENE 82427 56163 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME JNJ-7706621 JNJ-7706621 82428 56164 SPP1 6696 DRUGGABLE GENOME CALCITONIN CALCITONIN 8013390 82429 56165 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200935 DARIFENACIN HYDROBROMIDE 82432 56166 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-41 82433 56167 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Cobimetinib COBIMETINIB 82435 56168 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME EPZ004777 23138183 82436 56169 DYRK1B 9149 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME PHA-767491 CHEMBL225519 82438 56170 HDAC8 55869 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR HINOKITIOL HINOKITIOL 82439 56171 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR DIACEREIN DIACEREIN 82440 56172 ITGA4 3676 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME ELND-004 82441 56173 USP5 8078 ENZYME, PROTEASE inhibitor 252166869 82442 56174 GAA 2548 DRUGGABLE GENOME, ENZYME DOPAMINE HYDROCHLORIDE DOPAMINE HYDROCHLORIDE 82443 56175 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME LINIFANIB LINIFANIB 82444 56176 PRLR 5618 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, KINASE agonist 178101593 82446 56177 HSPA4 3308 NA CHLORPROMAZINE CHLORPROMAZINE 12857801 82447 56178 STAG2 10735 CLINICALLY ACTIONABLE, DRUG RESISTANCE Veliparib VELIPARIB 21852505,24356817 82448 56179 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135652667 ATROPINE 82449 56180 HIPK2 28996 TYROSINE KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME VADIMEZAN VADIMEZAN 82450 56181 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-32 82451 56182 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL2103829 FAXELADOL 82452 56183 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US20130116324 2 82454 56184 ITGB1 3688 DRUGGABLE GENOME, KINASE, CELL SURFACE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE VOLOCIXIMAB VOLOCIXIMAB 82456 56185 RBP4 5950 DRUGGABLE GENOME US9434727, 93 82457 56186 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME flibanserin FLIBANSERIN 82459 56187 TARDBP 23435 TUMOR SUPPRESSOR GNF-PF-5554 CHEMBL580130 82460 56188 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LINTITRIPT LINTITRIPT 82463 56189 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME NEOSTIGMINE NEOSTIGMINE 82465 56190 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME carbamazepine CARBAMAZEPINE 17638512,21738081 82466 56191 ATXN2 6311 NA VER-3323 CHEMBL309760 82467 56192 POR 5447 ENZYME, DRUGGABLE GENOME tacrolimus TACROLIMUS 23097010,25322286,26829596,30323313,24113216,26227094,21770725,24921414,24739669,25271728,24061445,28094348,29878980,29399716 82469 56193 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE PRN1371 82471 56194 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR DNDI1417467 CHEMBL1997335 82472 56195 CHRNA1 1134 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE antagonist 178100810 82473 56196 IMPDH2 3615 DRUGGABLE GENOME, ENZYME MYCOPHENOLIC ACID 82474 56197 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4364 CHEMBL528647 82475 56198 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE PF-04217903 PF-04217903 82477 56199 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR letrozole LETROZOLE 82478 56200 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME ATI-502 topical 82479 56201 TUBB3 10381 DRUGGABLE GENOME CHEMBL2108628 PACLITAXEL POLIGLUMEX 82481 56202 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PROPRANOLOL HYDROCHLORIDE PROPRANOLOL HYDROCHLORIDE 82483 56203 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CISPLATIN CISPLATIN 25081901 82484 56204 TDO2 6999 ENZYME, DRUGGABLE GENOME 2,3-diamino-benzo[b]thiophene derivative 3 82489 56205 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-33 82490 56206 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Benzamide derivative 12 82491 56207 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 178102286 QUIZARTINIB 82493 56208 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist 135649971 ATENOLOL 82495 56209 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 385612180 82496 56210 P2RY6 5031 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL antagonist 135650661 82497 56211 HTT 3064 DRUGGABLE GENOME Indole-based analog 11 82498 56212 FAAH 2166 ENZYME, DRUGGABLE GENOME inhibitor 315661162 82499 56213 BDKRB1 623 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME 178100640 82500 56214 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 benzbromarone BENZBROMARONE 25876828,20962433 82501 56215 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Beta blocking agents, non-selective 82503 56216 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051792 PANOBINOSTAT 82505 56217 PLG 5340 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE Desmoteplase DESMOTEPLASE 82506 56218 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201641 INSULIN ZINC SUSP EXTENDED RECOMBINANT HUMAN 82507 56219 ATXN2 6311 NA FLAVOKAWAIN B FLAVOKAWAIN B 82508 56220 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE WITHAFERIN A WITHAFERIN A 20726569 82509 56221 SCTR 6344 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME RG1068 82510 56222 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE fluvastatin FLUVASTATIN 82511 56223 PIM2 11040 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME LGH-447 LGH-447 82512 56224 USP1 7398 DNA REPAIR, PROTEASE, ENZYME 4-METHOXYDALBERGIONE 4-METHOXYDALBERGIONE 82513 56225 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME TRAMETINIB TRAMETINIB 82514 56226 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME GLPG0634 82516 56227 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE JNJ-7706621 JNJ-7706621 82517 56228 CBX1 10951 NA NSC-66209 CHEMBL175266 82518 56229 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME 7,3'-DIMETHOXYFLAVONE 7,3'-DIMETHOXYFLAVONE 82521 56230 CAMK2G 818 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME TAMATINIB R-406 82523 56231 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE E-3810 RABEPRAZOLE SODIUM 82526 56232 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist,antagonist 135649978 82527 56233 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR EOTAXIN 10706854 82528 56234 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135652673 BUPRENORPHINE 82529 56235 STXBP2 6813 NA Emapalumab-lzsg EMAPALUMAB 82531 56236 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1255654 TETRACAINE HYDROCHLORIDE 82532 56237 MAD1L1 8379 NA paclitaxel PACLITAXEL 23407047 82533 56238 HDAC7 51564 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME, ENZYME MOCETINOSTAT MOCETINOSTAT 23829483,26287310 82534 56239 POLI 11201 DNA REPAIR D-DOPA CHEMBL211670 82535 56240 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME RAPAMYCIN SIROLIMUS 10515383 82536 56241 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor CHEMBL3188267 CAPMATINIB 82541 56242 UMPS 7372 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE leucovorin LEUCOVORIN 20647221,16818689 82543 56243 TUBB 203068 DRUGGABLE GENOME BNC-105 82544 56244 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE cotinine COTININE 23223006 82546 56245 ATXN2 6311 NA SJ000001592 CHEMBL591834 82547 56246 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE CARBOXYLATED GLUCOSAMINE CARBOXYLATED GLUCOSAMINE 16616490 82549 56247 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Benzothiazine derivative 1 82550 56248 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1230607 PHA-793887 82551 56249 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE GNF-PF-2301 CHEMBL578061 82556 56250 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL41306 CNS-5161 82557 56251 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL592445 GEDATOLISIB 82558 56252 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-74 82559 56253 PTGS2 5743 DRUGGABLE GENOME, ENZYME Nabumetone NABUMETONE 82560 56254 ALOX5 240 DRUGGABLE GENOME, ENZYME BF-389 82561 56255 LAG3 3902 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE GSK2831781 GSK2831781 82563 56256 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE antibody MEDI-575 TOVETUMAB 82565 56257 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AMLODIPINE AMLODIPINE 82566 56258 LYN 4067 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE TAE-684 TAE-684 82567 56259 DEPTOR 64798 KINASE inhibitor MLN0128 SAPANISERTIB 82568 56260 POLK 51426 DNA REPAIR, ENZYME TYRPHOSTIN 51 TYRPHOSTIN 51 82570 56261 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE LINSITINIB LINSITINIB 82577 56262 MAPT 4137 DRUGGABLE GENOME AG-126 CHEMBL77387 82578 56263 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME Thiazolidine dione crystalline derivative 1 82580 56264 SCNN1B 6338 DRUGGABLE GENOME, ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE TRIAMTERENE TRIAMTERENE 82581 56265 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME PEMBROLIZUMAB PEMBROLIZUMAB 28451792 82583 56266 FAAH 2166 ENZYME, DRUGGABLE GENOME Azole derivative 3 82584 56267 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE ARQ 087 82585 56268 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2,4,6-TRIBROMOPHENOL CHEMBL220087 82586 56269 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME PENTAMIDINE DIISETHIONATE PENTAMIDINE ISETHIONATE 82587 56270 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 252166680 82589 56271 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME LICOFLAVANONE A LICOFLAVANONE A 20022509 82590 56272 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Nalfurafine hcl 82592 56273 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antagonist 252166738 82594 56274 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COUMESTROL COUMESTROL 82596 56275 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 178102553 82598 56276 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR ZINC 03369470 CHEMBL599013 82599 56277 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TESTOSTERONE BUCICLATE 82600 56278 TTK 7272 SERINE THREONINE KINASE, TYROSINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME Tricyclic isoxazoloquinazoline derivative 2 82601 56279 IGF1 3479 GROWTH FACTOR, HORMONE ACTIVITY, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE MEDI-573 DUSIGITUMAB 82602 56280 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME Cetuximab CETUXIMAB 22797062 82604 56281 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR PH-797804 PH-797804 82605 56282 PDE4C 5143 DRUGGABLE GENOME, ENZYME inhibitor 178103171 82606 56283 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE OTELIXIZUMAB OTELIXIZUMAB 82607 56284 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TCMDC-123605 CHEMBL547285 82608 56285 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TRACAZOLATE TRACAZOLATE 82611 56286 TXNRD1 7296 DRUGGABLE GENOME Binuclear gold(I) compound 2 82614 56287 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR VORINOSTAT VORINOSTAT 82616 56288 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR agonist 310264680 LIQUIRTIGENIN 82619 56289 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-61 82620 56290 EIF2AK4 440275 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME ziprasidone ZIPRASIDONE 24751813 82621 56291 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL2146146 ATROPINE SULFATE 82622 56292 EPHB4 2050 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545155 JI-101 82624 56293 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME DIETHYLSTILBESTROL DIETHYLSTILBESTROL 1980008 82625 56294 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE DEZOCINE DEZOCINE 82626 56295 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor CHEMBL608533 MIDOSTAURIN 82628 56296 RPS6KA3 6197 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR Pyrrolo[2,3-d]pyrimidine derivative 35 82631 56297 KAT2B 8850 ENZYME, DRUGGABLE GENOME DIETHYL-2-PENTADECYLIDENEMALONATE CHEMBL404916 18434144,21292492 82632 56298 GLA 2717 ENZYME, DRUGGABLE GENOME PSEUDOEPHEDRINE PSEUDOEPHEDRINE 82633 56299 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME METHYLCELLULOSE METHYLCELLULOSE 11516172 82634 56300 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 12 82637 56301 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PMID25726713-Compound-31 82638 56302 CCL21 6366 DRUGGABLE GENOME MIP-1BETA 10737895 82639 56303 FOXO3 2309 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE SYRINGARESINOL SYRINGARESINOL 25479772 82640 56304 POLK 51426 DNA REPAIR, ENZYME L-690330 L-690330 82641 56305 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Aromatic bicyclic compound 2 82644 56306 STAT3 6774 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, KINASE Pyrazole derivative 64 82646 56307 GJB5 2709 ION CHANNEL inhibitor 135652731 82647 56308 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545052 FIMEPINOSTAT 82649 56309 POLB 5423 DNA REPAIR, DRUGGABLE GENOME SJ000044417 CHEMBL609438 82651 56310 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE VATALANIB VATALANIB 82652 56311 CBR3 874 ENZYME, DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, CLINICALLY ACTIONABLE anthracyclines and related substances 18457324 82654 56312 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PF-562271 PF-00562271 82656 56313 PSMA7 5688 PROTEASE, DRUGGABLE GENOME inhibitor BORTEZOMIB BORTEZOMIB 82657 56314 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE 6-OHDA 17855652 82658 56315 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL598797 CUDC-101 82659 56316 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1200561 DOXAZOSIN MESYLATE 82660 56317 MT-RNR1 4549 KINASE gentamicin GENTAMICIN 18830133,16875663,9164619,19682603,16631122,21495045,16458854,12031626,16375862,9831149,17637808,22475488,11857751,27397648,9779807,7689389,20111055,9111378,27427311,17698030,11313749,20416460,16168391,24703164,9950117,21504270,11174059,8285309,18790089,15917167,20353758,16955413,16380089,14699607,17999439,14755216,17341440,19376484,15708009,25515069,15555598,11079536,17434445 82661 56318 PTAFR 5724 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 135649879 CHEMBL317090 82662 56319 KDM4A 9682 DRUGGABLE GENOME, ENZYME GNF-PF-1644 CHEMBL600734 82663 56320 SMN2 6607 DRUGGABLE GENOME INDOPROFEN INDOPROFEN 82665 56321 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor AZD1480 AZD-1480 82667 56322 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CHEMBL1257 ENFLURANE 82668 56323 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME SB-203580 SB-203580 82669 56324 TUBA1B 10376 DRUGGABLE GENOME inhibitor CHEMBL1096380 PLINABULIN 82672 56325 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME ENTRECTINIB ENTRECTINIB 82673 56326 ALOX15B 247 DRUGGABLE GENOME, ENZYME PD-404182 CHEMBL595227 82674 56327 HLA-A 3105 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME amoxicillin AMOXICILLIN 9609616 82675 56328 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME DOPAMINE DOPAMINE 82676 56329 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME busulfan BUSULFAN 82678 56330 ACO1 48 ENZYME N-ACETYLCYSTEINE ACETYLCYSTEINE 10037708 82679 56331 KDM4A 9682 DRUGGABLE GENOME, ENZYME CEPHALOCHROMIN CEPHALOCHROMIN 82681 56332 APH1A 51107 DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID28350212-Compound-13 82685 56333 PRKCI 5584 KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL494089 GSK-690693 82687 56334 BIRC3 330 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL3039522 BIRINAPANT 82688 56335 PIM3 415116 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE US8759338, 2 82690 56336 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PIOGLITAZONE PIOGLITAZONE 17063547 82692 56337 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 82694 56338 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 315661142 PF-03463275 82696 56339 CSNK1A1 1452 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SB-431542 SB-431542 82698 56340 SMN2 6607 DRUGGABLE GENOME 2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE 2,3-DIHYDROXY-6,7-DICHLOROQUINOXALINE 82699 56341 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Argatroban ARGATROBAN 82700 56342 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME activator 135651450 82702 56343 ABCB11 8647 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE 178101266 82704 56344 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BROMOXYNIL BROMOXYNIL 82705 56345 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 187051829 82706 56346 FABP4 2167 DRUGGABLE GENOME inhibitor 252827455 82708 56347 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 387065609 82709 56348 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor CHEMBL2107358 OBATOCLAX MESYLATE 82711 56349 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME LEVOTHYROXINE LEVOTHYROXINE 82712 56350 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME FMS/TRK TYROSINE KINASE INHIBITOR PLX7486 TOSYLATE 29880614 82713 56351 GAPVD1 26130 NA interferon beta-1b 27001119 82714 56352 HTT 3064 DRUGGABLE GENOME SANGUINARIUM SANGUINARIUM 82715 56353 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CHLORPROPAMIDE CHLORPROPAMIDE 22931300 82716 56354 CA9 768 DRUGGABLE GENOME, ENZYME PMID30074415-Compound-GS3 82718 56355 PDE5A 8654 ENZYME, DRUGGABLE GENOME TADALAFIL TADALAFIL 82720 56356 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Camptothecin CAMPTOTHECIN 82721 56357 CTSK 1513 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE, ENZYME inhibitor 223366191 BALICATIB 82722 56358 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME agonist 178103549 PEGFILGRASTIM 82723 56359 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME Pentacea 20093855 82724 56360 IL1B 3553 KINASE, DRUGGABLE GENOME ANTIDEPRESSANT 11752890 82725 56361 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DOLASTATIN 12 DOLASTATIN 12 82726 56362 GSTT1 2952 DRUGGABLE GENOME amoxicillin AMOXICILLIN 82727 56363 GRIK2 2898 DRUGGABLE GENOME, ION CHANNEL TALBUTAL TALBUTAL 82728 56364 BCHE 590 DRUGGABLE GENOME, ENZYME PMID29757691-Compound-8b 82729 56365 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE ONO-7475 82730 56366 MAPT 4137 DRUGGABLE GENOME BITHIONOLATE SODIUM BITHIONOLATE SODIUM 82731 56367 POLB 5423 DNA REPAIR, DRUGGABLE GENOME PURPUROGALLIN PURPUROGALLIN 82734 56368 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CYTARABINE HYDROCHLORIDE CYTARABINE HYDROCHLORIDE 82735 56369 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL2326966 SF-1126 82736 56370 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME PMID28621580-Compound-WO2013036866C66 82738 56371 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GEMFIBROZIL GEMFIBROZIL 82740 56372 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GITOXIGENIN GITOXIGENIN 82741 56373 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Anti-HER3/EGFR DAF 82743 56374 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE BROMOETHANE BROMOETHANE 22503207 82744 56375 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL572881 MOTESANIB 82747 56376 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR modulator CHEMBL10041 AFIMOXIFENE 82748 56377 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR peginterferon alfa-2b 82749 56378 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME YTTRIUM-90 EDOTREOTIDE 82750 56379 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SR-13668 SR-13668 17602463 82751 56380 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR MAPK INHIBITORS 15316935 82753 56381 GUCY1A2 2977 ENZYME, DRUGGABLE GENOME NCX 1510 82754 56382 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME BENZO(K)FLUORANTHENE BENZO(K)FLUORANTHENE 82755 56383 PSMD7 5713 PROTEASE inhibitor CHEMBL3545432 IXAZOMIB CITRATE 82756 56384 TPCN1 53373 ION CHANNEL, DRUGGABLE GENOME activator 178100233 82758 56385 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE EPI-743 VATIQUINONE 82759 56386 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER AMOXAPINE AMOXAPINE 82760 56387 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1233528 VOLASERTIB 82763 56388 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME thiotepa THIOTEPA 17638512 82764 56389 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME inhibitor 178101542 SULFASALAZINE 82765 56390 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR inhibitor CHEMBL2108718 SEMULOPARIN SODIUM 82766 56391 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME cyclophosphamide CYCLOPHOSPHAMIDE 26773420,24128861,29938344,17638512,20179710,19005482,11470993,28181240,21821736 82768 56392 RGS4 5999 DRUGGABLE GENOME BETA-LAPACHONE LAPACHONE 82769 56393 GRK6 2870 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE inhibitor 249565822 BALANOL 82772 56394 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID29338548-Compound-27 82773 56395 GRM8 2918 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 381744921 82774 56396 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME MTOR KINASE INHIBITOR AZD8055 26544513 82776 56397 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE LAUROGUADINE LAUROGUADINE 82777 56398 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Quinolone derivative 1 82778 56399 RUNX1 861 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FUSARIC ACID FUSARIC ACID 82779 56400 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE pamaquine 23530079 82780 56401 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GAMBOGIC ACID GAMBOGIC ACID 21486005 82782 56402 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102298 BMS-387032 82784 56403 KIF11 3832 DRUGGABLE GENOME inhibitor CHEMBL2105661 LITRONESIB 82787 56404 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME DOVITINIB DOVITINIB 82789 56405 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL2096631 CLORAZEPATE DIPOTASSIUM 82790 56406 BAZ2B 29994 NA EMODIC ACID EMODIC ACID 82793 56407 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 249565751 82794 56408 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL956 SUPROFEN 82797 56409 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 252166679 82798 56410 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR desipramine DESIPRAMINE 82799 56411 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME PICTILISIB BISMESYLATE 23845441 82800 56412 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE EPISIALIN 11903603 82802 56413 C3 718 PROTEASE INHIBITOR, DRUGGABLE GENOME, CELL SURFACE clozapine CLOZAPINE 26503818 82803 56414 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CROMOLYN SODIUM CROMOLYN SODIUM 82805 56415 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SJ000124275 CHEMBL602150 82808 56416 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ALLOPURINOL ALLOPURINOL 22931300 82809 56417 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE unspecified IGF-1R antibody 27196767 82810 56418 ALDH1A1 216 DRUGGABLE GENOME, ENZYME 1,2,3,4,5,6-HEXABROMO-CYCLOHEXANE CHEMBL444236 82813 56419 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102290 AT-7519 82814 56420 GMNN 51053 DRUGGABLE GENOME NSC-102042 CHEMBL273103 82815 56421 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE TRIPHENYLSTANNANOL TRIPHENYLSTANNANOL 82816 56422 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650152 CYPROHEPTADINE 82817 56423 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL679 EPINEPHRINE 82818 56424 MAOA 4128 DRUGGABLE GENOME, ENZYME PMID29324067-Compound-25 82820 56425 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE IL-1 7688736 82821 56426 CXCL8 3576 DRUGGABLE GENOME PENTOXIFYLLINE PENTOXIFYLLINE 12576442 82822 56427 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200781 CITALOPRAM HYDROBROMIDE 82823 56428 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE IRESSA IRESSA 16470840 82824 56429 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor PANOBINOSTAT PANOBINOSTAT 82825 56430 TUBA1B 10376 DRUGGABLE GENOME LARGAZOLE LARGAZOLE 20491440 82826 56431 NR5A2 2494 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR agonist 385612242 82829 56432 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR antagonist 223366066 GDC-0152 82832 56433 HPD 3242 ENZYME, DRUGGABLE GENOME Nitisinone NITISINONE 82833 56434 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CARMUSTINE CARMUSTINE 82834 56435 STAT6 6778 TRANSCRIPTION FACTOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 363894136 82835 56436 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor 53801036 82836 56437 ERCC2 2068 KINASE, TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME etoposide ETOPOSIDE 82837 56438 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME agonist CHEMBL3707402 PF-06372865 82840 56439 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Amuvatinib AMUVATINIB 24326130 82841 56440 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME inhibitor PF00562271 82842 56441 SCNN1G 6340 ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE triamterene TRIAMTERENE 23788015 82843 56442 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE OSI-632 OSI-632 82846 56443 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE NSC-56452 CHEMBL1358137 22944332 82847 56444 ALDH2 217 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ethanol ALCOHOL 31002879,15902904,16679777 82848 56445 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR AST-487 AST-487 82850 56446 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME NSC-720622 CHEMBL1287980 82855 56447 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR KD3010 KD3010 82856 56448 HMOX1 3162 ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 252827530 82857 56449 ITGB3 3690 DRUGGABLE GENOME, CELL SURFACE inhibitor CILENGITIDE CILENGITIDE 82858 56450 GMNN 51053 DRUGGABLE GENOME GNF-PF-3696 CHEMBL598885 82859 56451 SQLE 6713 DRUGGABLE GENOME, ENZYME Epigallocatechin gallate 82861 56452 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE PMID28048944-Compound-19 82862 56453 PRKD2 25865 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PF-562271 PF-00562271 82865 56454 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Propafenone PROPAFENONE 82866 56455 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME N-(cyanomethyl)-4-(2-(phenylamino)pyrimidin-4-yl)benzamide derivative 1 82868 56456 TG 7038 DRUGGABLE GENOME, HORMONE ACTIVITY VACCINE 10390298 82870 56457 GLS 2744 ENZYME PMID30273516-Compound-40 82871 56458 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR THIOMERSAL THIMEROSAL 82872 56459 IMPDH1 3614 ENZYME, DRUGGABLE GENOME MYCOPHENOLATE MOFETIL 82876 56460 HMGCR 3156 ENZYME, DRUGGABLE GENOME inhibitor 135650602 MEVASTATIN 82877 56461 ATAD5 79915 NA DINALINE DINALINE 82880 56462 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 3-HYDROXYFLAVONOL CHEMBL242172 82881 56463 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR PALBOCICLIB PALBOCICLIB 26715889,21278246,24495407,26528855,23898052 82882 56464 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 178102315 RUXOLITINIB 82883 56465 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE OESTRADIOL ESTRADIOL 10325261 82886 56466 CDKN2D 1032 KINASE TRICHOSTATIN A 15107822 82887 56467 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR YKP-GI 82888 56468 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR PHA-767491 CHEMBL225519 82891 56469 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR OXYTETRACYCLINE HYDROCHLORIDE OXYTETRACYCLINE HYDROCHLORIDE 82892 56470 DTYMK 1841 KINASE ETHANOL ALCOHOL 11923581 82893 56471 UQCRB 7381 NA TERPESTACIN TERPESTACIN 21215626 82894 56472 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE RM-1929 CETUXIMAB SAROTALOCAN 82896 56473 NPR3 4883 DRUGGABLE GENOME NESIRITIDE NESIRITIDE 82899 56474 TUBB2A 7280 DRUGGABLE GENOME VINCRISTINE VINCRISTINE 82900 56475 POLK 51426 DNA REPAIR, ENZYME GALUTEOLIN GALUTEOLIN 82901 56476 PPIA 5478 DRUGGABLE GENOME, ENZYME SCY-635 SCY 635 82902 56477 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178100330 82904 56478 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING RETINYLRETINOATE RETINYLRETINOATE 18511283 82905 56479 SLC47A2 146802 TRANSPORTER, CLINICALLY ACTIONABLE, DRUGGABLE GENOME rucaparib RUCAPARIB 82906 56480 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME HYDROCORTISONE HYDROCORTISONE 82907 56481 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 178102027 82908 56482 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR LUTEOLIN LUTEOLIN 82909 56483 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME PMID25684022-Compound-WO2012135799 42(1.4) 82910 56484 MAFK 7975 ENZYME, TRANSCRIPTION FACTOR isoniazid ISONIAZID 22341855,29036176 82912 56485 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR lapatinib LAPATINIB 82913 56486 CA9 768 DRUGGABLE GENOME, ENZYME FERULIC ACID 82914 56487 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651146 82915 56488 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (+)-VENTILOQUINONE L METHYL ETHER CHEMBL594259 19783445 82918 56489 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR L-ornithine phenylacetate 82920 56490 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE BKM120 BUPARLISIB 24470511,23948973,23940356,28539475 82921 56491 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME DIAZEPAM DIAZEPAM 82922 56492 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 MIBEFRADIL MIBEFRADIL 21447734 82923 56493 KLK4 9622 PROTEASE, DRUGGABLE GENOME, ENZYME inhibitor 252827531 82924 56494 TGFB1 7040 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CELL SURFACE, GROWTH FACTOR GOSSYPOL GOSSYPOL 15015581 82926 56495 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL AVP-786 82927 56496 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Dabrafenib DABRAFENIB 27312529 82928 56497 ANPEP 290 NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, PROTEASE, ENZYME PL37 82929 56498 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME TAMATINIB R-406 82930 56499 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 252827484 82931 56500 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FURATHIOCARB FURATHIOCARB 82932 56501 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-19 82933 56502 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TELENZEPINE TELENZEPINE 82934 56503 BUB1 699 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 315661211 82935 56504 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR R(-)-PROPYLNORAPOMORPHINE HCL CHEMBL538542 82936 56505 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PIMOZIDE PIMOZIDE 82938 56506 DGAT1 8694 ENZYME, DRUGGABLE GENOME PF-04620110 PF-04620110 23871442 82939 56507 LAMA3 3909 DRUGGABLE GENOME CHEMBL2095222 OCRIPLASMIN 82940 56508 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DODINE DODINE 82941 56509 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor 249565884 A-443654 82942 56510 GMNN 51053 DRUGGABLE GENOME TCMDC-124009 CHEMBL1366623 82943 56511 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME GNF-PF-4832 CHEMBL601137 82944 56512 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 GENTAMICIN GENTAMICIN 22931300 82945 56513 TAT 6898 ENZYME 17 BETA-ESTRADIOL 2887201 82946 56514 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 inhibitor 135650454 KETOCONAZOLE 82949 56515 MKNK2 2872 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 178102632 82950 56516 POLI 11201 DNA REPAIR DAUNORUBICIN HYDROCHLORIDE DAUNORUBICIN HYDROCHLORIDE 82952 56517 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR CHEMOPREVENTIVE 15313408 82954 56518 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE GEMCITABINE GEMCITABINE 29338080 82955 56519 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Alpelisib ALPELISIB 82956 56520 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE DASATINIB DASATINIB 20537386,26758680,15705718,19779040,16775234,24367893,18191450,25686603,25207766,18818391,16772610 82957 56521 BRPF3 27154 DRUGGABLE GENOME 252166774 82958 56522 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME antibody 178103386 RITUXIMAB 82959 56523 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE HER-2-targeting CAR T Cells 82960 56524 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 363894199 82961 56525 CA7 766 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL18 ETHOXZOLAMIDE 82964 56526 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ETOPOSIDE ETOPOSIDE 82965 56527 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135649997 82966 56528 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME HALOPROGIN HALOPROGIN 82967 56529 SMN2 6607 DRUGGABLE GENOME 2-(4-METHOXYPHENYL)BENZO[D]THIAZOLE CHEMBL460508 82968 56530 TSHR 7253 CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, CELL SURFACE TCMDC-123781 CHEMBL581194 82969 56531 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE BMS-754807 BMS-754807 19778024 82971 56532 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR IMIPRAMINE HYDROCHLORIDE IMIPRAMINE HYDROCHLORIDE 82973 56533 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PACLITAXEL PACLITAXEL 16459017 82975 56534 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FEBANTEL FEBANTEL 82976 56535 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FIDUXOSIN HYDROCHLORIDE FIDUXOSIN HYDROCHLORIDE 82979 56536 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME SULFOBROMOPHTHALEIN SULFOBROMOPHTHALEIN 82980 56537 TRPC4 7223 ION CHANNEL, KINASE, DRUGGABLE GENOME, CELL SURFACE blocker 381744966 CLEMIZOLE 82981 56538 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE propoxyphene PROPOXYPHENE 18695978 82983 56539 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL723 CARVEDILOL 82985 56540 TGFBR1 7046 DRUGGABLE GENOME, ENZYME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, CELL SURFACE, TUMOR SUPPRESSOR LY3200882 82986 56541 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Indium-111 82988 56542 HBEGF 1839 CELL SURFACE, GROWTH FACTOR, DRUGGABLE GENOME KHK-2866 KHK-2866 82989 56543 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 XANTHOXYLIN XANTHOXYLIN 82991 56544 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME TACRINE TACRINE 82992 56545 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR LINIFANIB LINIFANIB 82994 56546 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GAMOLENIC ACID GAMOLENIC ACID 82995 56547 HMMR 3161 KINASE, CELL SURFACE, DRUGGABLE GENOME cyclophosphamide CYCLOPHOSPHAMIDE 82997 56548 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE SF1126 18172313,24634413 82999 56549 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE WZ4002 25964297,26036643,25870145,25948633 83000 56550 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor SODIUM PHENYLBUTYRATE 83001 56551 MAPT 4137 DRUGGABLE GENOME 1,4-DIMETHOXYANTHRAQUINONE 1,4-DIMETHOXYANTHRAQUINONE 83002 56552 TARDBP 23435 TUMOR SUPPRESSOR PHENYLETHENYLSEMICARBAZONE PHENYLETHENYLSEMICARBAZONE 83003 56553 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR SULOCHRIN SULOCHRIN 83006 56554 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR DINITRO CRESOL DINITRO CRESOL 83008 56555 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE AG-1879 CHEMBL406845 83009 56556 CAST 831 PROTEASE INHIBITOR EPINEPHRINE EPINEPHRINE 10863002 83010 56557 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Roxadustat ROXADUSTAT 83011 56558 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ESOXYBUTYNIN ESOXYBUTYNIN 83015 56559 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Triamcinolone TRIAMCINOLONE 83017 56560 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE OXAPIUM IODIDE OXAPIUM IODIDE 83018 56561 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649962 83020 56562 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE ORAL CONTRACEPTIVE 12376514 83021 56563 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 MAPROTILINE MAPROTILINE 22931300 83022 56564 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME WITHAFERIN A WITHAFERIN A 24079846 83023 56565 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SB590885 SB590885 20538618,27523909 83024 56566 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE JNJ-26483327 JNJ-26483327 83025 56567 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE GUGGULSTERONE GUGGULSTERONE 83027 56568 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL CM-2395 83028 56569 ARG1 383 ENZYME 2-AMINOHOMOHISTIDINE CHEMBL1099168 20441173 83029 56570 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MITOGLITAZONE MITOGLITAZONE 83030 56571 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 RIMCAZOLE RIMCAZOLE 83031 56572 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor SODIUM PHENYLBUTYRATE 83032 56573 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor HESPERADIN HESPERADIN 19035792 83033 56574 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE PMID26882240-Compound-8 83034 56575 CTSV 1515 ENZYME, DRUGGABLE GENOME, PROTEASE inhibitor 405067337 83035 56576 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME 2,3,4-TRIHYDROXYBENZOPHENONE CHEMBL1527 83036 56577 RACGAP1 29127 NA TCMDC-139459 CHEMBL86464 83037 56578 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME SIB-1757 CHEMBL88553 83038 56579 ALOX15 246 ENZYME, DRUGGABLE GENOME PYRITHIONE ZINC PYRITHIONE ZINC 83039 56580 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 miconazole MICONAZOLE 9187528 83040 56581 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3544942 RONICICLIB 83041 56582 TCF7L2 6934 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR sirolimus SIROLIMUS 23041303,21857094 83042 56583 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MESALAMINE MESALAMINE 83044 56584 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR T091317 T091317 83046 56585 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PLICAMYCIN PLICAMYCIN 22931300 83047 56586 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 27 83048 56587 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR RALOXIFENE RALOXIFENE 20659801 83049 56588 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME ROTTLERIN ROTTLERIN 83050 56589 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 252827451 SAR-260301 83051 56590 TNKS 8658 DRUGGABLE GENOME, ENZYME BGB-290 PAMIPARIB 83052 56591 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor STA-9090 GANETESPIB 83053 56592 TNFRSF10B 8795 DRUGGABLE GENOME, CELL SURFACE agonist 178101758 83054 56593 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Pyridine derivative 19 83055 56594 SLC19A1 6573 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME inhibitor 310264671 83057 56595 PDE5A 8654 ENZYME, DRUGGABLE GENOME SILDENAFIL SILDENAFIL 83059 56596 POLI 11201 DNA REPAIR INDOCYANINE GREEN SODIUM INDOCYANINE GREEN 83060 56597 KDM4A 9682 DRUGGABLE GENOME, ENZYME ZM-39923 HCL CHEMBL538798 83061 56598 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MIBEFRADIL MIBEFRADIL 83063 56599 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CEFACLOR CEFACLOR 83064 56600 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME BENZO(K)FLUORANTHENE BENZO(K)FLUORANTHENE 83066 56601 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 315661159 ECHOTHIOPHATE 83068 56602 ENO2 2026 CELL SURFACE PROPOFOL PROPOFOL 16027086 83069 56603 LTF 4057 CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, PROTEASE Parecoxib PARECOXIB 83070 56604 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GSK1120212 TRAMETINIB 27876675 83071 56605 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102345 NEFLAMAPIMOD 83073 56606 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE PKF118-310 28611108 83074 56607 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME Imidazopyridine derivative 3 83075 56608 HPD 3242 ENZYME, DRUGGABLE GENOME NITISINONE NITISINONE 83076 56609 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565633 DACTOLISIB 83077 56610 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME EUPAFOLIN EUPAFOLIN 83079 56611 PLTP 5360 DRUGGABLE GENOME SIMVASTATIN SIMVASTATIN 11566255 83080 56612 IDE 3416 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, ENZYME, PROTEASE PRO-001 83081 56613 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL109480 TANESPIMYCIN 83083 56614 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TCMDC-123579 CHEMBL533954 83084 56615 PAK2 5062 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor 135652717 STAUROSPORINE 83087 56616 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4242 CHEMBL584514 83088 56617 FZD1 8321 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, KINASE antibody 381118907 VANTICTUMAB 83090 56618 ALOX15 246 ENZYME, DRUGGABLE GENOME DNDI1417309 CHEMBL1341830 83093 56619 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME agonist 178103125 83094 56620 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-56 83095 56621 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ZERANOL ZERANOL 83096 56622 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME PMID25482888-Compound-72 83098 56623 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME E324 E324 83099 56624 TOP2B 7155 DRUGGABLE GENOME, ENZYME TAS-103 CHEMBL488755 83100 56625 RPS6KA6 27330 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME CID 138805970 83101 56626 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Fluorophenyl-substituted heterocyclic amide analog 1 83102 56627 CD274 29126 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE atezolizumab ATEZOLIZUMAB 83103 56628 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME COLFORSIN COLFORSIN 83104 56629 MAOB 4129 DRUGGABLE GENOME, ENZYME Pargyline PARGYLINE 83105 56630 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RETINOL RETINOL 83106 56631 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Quinidine QUINIDINE 83108 56632 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100429 83109 56633 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Lapatinib LAPATINIB 83110 56634 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL MIDAZOLAM MIDAZOLAM 83112 56635 ALOX15 246 ENZYME, DRUGGABLE GENOME RO-318220 BISINDOLYLMALEIMIDE IX 83114 56636 ABCC4 10257 ABC TRANSPORTER, DRUGGABLE GENOME, TRANSPORTER RIMONABANT RIMONABANT 21511945 83115 56637 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PREDNISOLONE SODIUM SUCCINATE PREDNISOLONE SODIUM SUCCINATE 83116 56638 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE XL765 83118 56639 HPGDS 27306 ENZYME, DRUGGABLE GENOME HQL-79 CHEMBL574003 20684598 83120 56640 SIRT5 23408 ENZYME GW7647 GW7647 83122 56641 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ZEBULARINE ZEBULARINE 16239434 83123 56642 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CEP-8983 23428903 83125 56643 GUCY1A1 2982 ENZYME, DRUGGABLE GENOME RIOCIGUAT RIOCIGUAT 83127 56644 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL DIAZEPAM DIAZEPAM 83128 56645 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CAPSAICIN CAPSAICIN 17979524 83129 56646 MTF1 4520 TRANSCRIPTION FACTOR LOR-253 APTO-253 83131 56647 IL1B 3553 KINASE, DRUGGABLE GENOME PENTAMIDINE PENTAMIDINE 8370344 83132 56648 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135650736 NORTRIPTYLINE 83133 56649 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-73 83134 56650 SENP6 26054 ENZYME, PROTEASE, DRUGGABLE GENOME TCMDC-125543 CHEMBL546170 83136 56651 ROS1 6098 TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR SB-202190 SB-202190 83139 56652 IFI27 3429 NUCLEAR HORMONE RECEPTOR TGFBETA1 15086558 83140 56653 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417024 CHEMBL1462710 83142 56654 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PH-797804 PH-797804 83143 56655 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME GSK2126458 OMIPALISIB 22389471 83144 56656 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME N-phenyl-pyrimidin-4-amine derivative 1 83146 56657 KDM4A 9682 DRUGGABLE GENOME, ENZYME MMV007764 CHEMBL609628 83147 56658 MTHFR 4524 ENZYME, CLINICALLY ACTIONABLE fluorouracil FLUOROURACIL 27738344,18245544,12083967,17700593,24167597,29845393,27864592,18299612,20819423,27995989,19384296,29134491,23314736,20638924,25331073,20385995,27557140,24980946,26967565,23407049,26014925,23736036 83148 56659 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 83149 56660 POLK 51426 DNA REPAIR, ENZYME DAUNORUBICIN DAUNORUBICIN 83150 56661 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-50690 CHEMBL1388703 83151 56662 USP2 9099 DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR, PROTEASE IODOACETAMIDE IODOACETAMIDE 83153 56663 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 178102417 83154 56664 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-26 83155 56665 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 318164820 83156 56666 SLC46A1 113235 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME methotrexate METHOTREXATE 21317831 83157 56667 TRPM4 54795 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME blocker,inhibitor 135651446 ADENOSINE TRIPHOSPHATE 83159 56668 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME TAMIBAROTENE TAMIBAROTENE 83160 56669 SMN1 6606 DRUGGABLE GENOME NSC-102045 CHEMBL483633 83162 56670 CXCL8 3576 DRUGGABLE GENOME RU 41740 9304405 83163 56671 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PERUVOSIDE PERUVOSIDE 83164 56672 SACM1L 22908 NA bupropion BUPROPION 22041458 83165 56673 SMARCB1 6598 CLINICALLY ACTIONABLE CFI-400945 CFI-400945 28398638 83166 56674 TNFRSF11B 4982 DRUGGABLE GENOME TRAIL 11912131,12915677 83167 56675 ADAMTS1 9510 ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, PROTEASE hmg coa reductase inhibitors 21037509 83169 56676 UGT1A10 54575 DRUGGABLE GENOME, ENZYME methotrexate METHOTREXATE 29791011 83173 56677 SOD1 6647 ENZYME, DRUGGABLE GENOME ISIS-SOD1RX TOFERSEN 83176 56678 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR GANODERMANONTRIOL GANODERMANONTRIOL 22014750 83177 56679 TSPO 706 DRUGGABLE GENOME CLONAZEPAM CLONAZEPAM 83178 56680 LTA4H 4048 ENZYME, DRUGGABLE GENOME, PROTEASE 4-(4-METHOXYPHENOXY)PHENOL CHEMBL444161 18952425 83183 56681 CXCL10 3627 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE ZIDOVUDINE ZIDOVUDINE 11141242 83184 56682 POLK 51426 DNA REPAIR, ENZYME RAFOXANIDE RAFOXANIDE 83185 56683 TUBB2B 347733 DRUGGABLE GENOME COLCHICINE COLCHICINE 23750455,25805446,24502232,25061803,25937236,24773591,25938266 83186 56684 ALDH5A1 7915 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL109 VALPROIC ACID 83188 56685 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135650212 DULOXETINE 83190 56686 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME BENZBROMARONE BENZBROMARONE 83191 56687 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME AUY922 24398328 83194 56688 GRIK4 2900 DRUGGABLE GENOME, ION CHANNEL agonist 178101134 83198 56689 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NILUTAMIDE NILUTAMIDE 83199 56690 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Pyrazinylpyridine derivative 1 83200 56691 TMEM97 27346 NA Bicyclo-heptan-2-amine derivative 1 83205 56692 PON1 5444 ENZYME, TRANSPORTER, DRUGGABLE GENOME simvastatin SIMVASTATIN 18430057,16238680,19904013 83206 56693 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR POMIFERIN POMIFERIN 83207 56694 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE GLYBURIDE GLYBURIDE 8224371 83208 56695 ALDH1A1 216 DRUGGABLE GENOME, ENZYME chloroacetaldehyde 83211 56696 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SECURININE SECURININE 83213 56697 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CLOTRIMAZOLE CLOTRIMAZOLE 83214 56698 CFTR 1080 DRUGGABLE GENOME, ABC TRANSPORTER, ION CHANNEL, TRANSPORTER, CELL SURFACE, CLINICALLY ACTIONABLE activator 178101130 83215 56699 CARM1 10498 ENZYME, METHYL TRANSFERASE, DRUGGABLE GENOME inhibitor 315661333 BIIB021 83217 56700 SMN1 6606 DRUGGABLE GENOME KENPAULLONE KENPAULLONE 83218 56701 ATAD5 79915 NA GNF-PF-1947 CHEMBL585591 83219 56702 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL1370 BUDESONIDE 83220 56703 GMNN 51053 DRUGGABLE GENOME BROMOCICLEN BROMOCICLEN 83221 56704 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ISOCYANATO-CYCLOHEXANE CHEMBL26886 83222 56705 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ALFUZOSIN ALFUZOSIN 83223 56706 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Bortezomib BORTEZOMIB 21216929 83224 56707 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME SHINFLAVANONE SHINFLAVANONE 20022509 83225 56708 WRN 7486 CLINICALLY ACTIONABLE, DNA REPAIR, ENZYME SJ000044511 CHEMBL592124 83226 56709 CHST11 50515 ENZYME, DRUGGABLE GENOME CHONDROITIN 11056388 83227 56710 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 triazolam TRIAZOLAM 83228 56711 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TYRPHOSTIN 47 TYRPHOSTIN 47 83231 56712 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME inhibitor 315661180 ZOTIRACICLIB 83232 56713 ALDH1A1 216 DRUGGABLE GENOME, ENZYME CATECHOL CATECHOL 83233 56714 PTGS2 5743 DRUGGABLE GENOME, ENZYME Mefenamic acid 83234 56715 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE triazolam TRIAZOLAM 83235 56716 PTGFR 5737 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Tafluprost TAFLUPROST 83236 56717 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE Dihydrotestosterone ANDROSTANOLONE 83239 56718 RARB 5915 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME ALITRETINOIN ALITRETINOIN 83241 56719 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME RESMINOSTAT RESMINOSTAT 83242 56720 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RO-137410 CHEMBL275311 18951029 83244 56721 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ALPHA-ENDORPHIN CHEMBL255300 17616524 83245 56722 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CYC-116 CYC-116 20462263 83246 56723 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR SR9011 SR9011 23656296 83247 56724 ABHD6 57406 PHOSPHOLIPASE, ENZYME inhibitor 375973250 83248 56725 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALEXIDINE DIHYDROCHLORIDE ALEXIDINE DIHYDROCHLORIDE 83249 56726 KDM5A 5927 CLINICALLY ACTIONABLE, ENZYME, NUCLEAR HORMONE RECEPTOR AKOS020330656 83250 56727 MAPT 4137 DRUGGABLE GENOME DNDI1416917 CHEMBL1335833 83251 56728 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER NORDIHYDROGUAIARETIC ACID NORDIHYDROGUAIARETIC ACID 83253 56729 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE SORBIC ACID SORBIC ACID 83255 56730 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652604 83257 56731 GMNN 51053 DRUGGABLE GENOME GNF-PF-4967 CHEMBL585827 83260 56732 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651211 83262 56733 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME SRA737 27167172 83264 56734 CA9 768 DRUGGABLE GENOME, ENZYME Curcumin CURCUMIN 83265 56735 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Estrone ESTRONE 83269 56736 RARG 5916 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX PMID27336223-Compound-15 83270 56737 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 tramadol TRAMADOL 24849324 83272 56738 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME STAUROSPORINE STAUROSPORINE 83273 56739 USP1 7398 DNA REPAIR, PROTEASE, ENZYME CONGO RED CONGO RED 83274 56740 CACNB4 785 DRUGGABLE GENOME, ION CHANNEL ARVERAPAMIL 83275 56741 ANKS1B 56899 NA amisulpride AMISULPRIDE 28332719 83276 56742 GMNN 51053 DRUGGABLE GENOME GW7647 GW7647 83277 56743 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Pyrrolidinyl urea derivative 9 83279 56744 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DRONEDARONE DRONEDARONE 83281 56745 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR APOMORPHINE APOMORPHINE 83282 56746 ALDH1A1 216 DRUGGABLE GENOME, ENZYME RO-106-9920 CHEMBL271023 83284 56747 ATAD5 79915 NA GNF-PF-1644 CHEMBL600734 83285 56748 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650026 BROMOCRIPTINE 83287 56749 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME blocker 135652059 83288 56750 MAP3K20 51776 KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME TOZASERTIB TOZASERTIB 83289 56751 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW805758X GW805758X 83293 56752 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Cediranib CEDIRANIB 26802156 83294 56753 PDE4B 5142 DRUGGABLE GENOME, ENZYME ETAZOLATE ETAZOLATE 83295 56754 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME 4-(thiazol-5-yl)-pyrimidine derivative 2 83296 56755 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE M2698 MSC-2363318A 83298 56756 POLB 5423 DNA REPAIR, DRUGGABLE GENOME NSC-367089 CHEMBL1543865 83299 56757 BCHE 590 DRUGGABLE GENOME, ENZYME Eptastigmine EPTASTIGMINE 83300 56758 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR inhibitor CHEMBL1213490 ROMIDEPSIN 83301 56759 CYB5R1 51706 DRUGGABLE GENOME isosorbide mononitrate 83302 56760 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME GRAMINE GRAMINE 83303 56761 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 328083458 83304 56762 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL3545003 MSC-2363318A 83307 56763 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR PMID25553724-Compound-US2012820715110 83310 56764 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE OMEPRAZOLE OMEPRAZOLE 83311 56765 ADA 100 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE DIPYRIDAMOLE DIPYRIDAMOLE 83312 56766 UGT1A10 54575 DRUGGABLE GENOME, ENZYME SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 83314 56767 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR SNX-5422 CHEMBL553939 83315 56768 TAC1 6863 DRUGGABLE GENOME GLYCYRRHETINIC ACID 10529487 83316 56769 TSPO 706 DRUGGABLE GENOME Benzoxazepine analog 1 83317 56770 NR1D2 9975 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 178101166 83318 56771 PIP5K1A 8394 KINASE, DRUGGABLE GENOME, ENZYME inhibitor 252166654 83319 56772 SLC18A2 6571 DRUGGABLE GENOME, TRANSPORTER TETRABENAZINE TETRABENAZINE 83320 56773 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE 4-HYDROXYEVODIAMINE CHEMBL2171794 22867019 83321 56774 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 CP-55940 CP-55940 83322 56775 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE Saruplase SARUPLASE 83323 56776 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ENOBOSARM ENOBOSARM 21506597 83324 56777 USP1 7398 DNA REPAIR, PROTEASE, ENZYME OTILONIUM OTILONIUM 83325 56778 POLK 51426 DNA REPAIR, ENZYME TRICETIN TRICETIN 83326 56779 PPP3CC 5533 TRANSCRIPTION FACTOR VOCLOSPORIN VOCLOSPORIN 83327 56780 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR KENPAULLONE KENPAULLONE 83328 56781 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Lidocaine LIDOCAINE 83329 56782 VAMP2 6844 DRUGGABLE GENOME BOTULINUM TOXIN TYPE B 83330 56783 KAT2B 8850 ENZYME, DRUGGABLE GENOME inhibitor 178103615 83331 56784 PDE10A 10846 ENZYME, DRUGGABLE GENOME Imidazo[5,1-c]pyrido[2,3-e][1,2,4]triazine derivative 5 83332 56785 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER cisplatin CISPLATIN 29938344,22016816,23746184,21332314,20530282 83334 56786 HTT 3064 DRUGGABLE GENOME HYCANTHONE HYCANTHONE 83335 56787 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL Pregabalin PREGABALIN 83338 56788 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE BMS-509744 CHEMBL209148 83339 56789 PTGS2 5743 DRUGGABLE GENOME, ENZYME etoricoxib ETORICOXIB 19602986 83340 56790 CACNA1E 777 DRUGGABLE GENOME, ION CHANNEL blocker 135652744 83342 56791 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL58323 ERLOSAMIDE 83343 56792 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME antagonist 252827399 RESVERATROL 83344 56793 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TAE226 26090892 83347 56794 MME 4311 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME inhibitor 178103120 DAGLUTRIL 83348 56795 RAB9A 9367 ENZYME, DRUGGABLE GENOME 6-HYDROXYFLAVONE 6-HYDROXYFLAVONE 83349 56796 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME BMS-345541 BMS-345541 83350 56797 BAZ2B 29994 NA HEXACHLOROPHENE HEXACHLOROPHENE 83351 56798 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE NSC-107022 CHEMBL1601846 83353 56799 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE GNF-PF-4967 CHEMBL585827 83354 56800 MAP3K8 1326 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 178102673 83355 56801 NAE1 8883 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1231160 PEVONEDISTAT 83356 56802 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID28048944-Compound-5 83357 56803 IKBKG 8517 KINASE, DRUGGABLE GENOME pyrimethamine PYRIMETHAMINE 83358 56804 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Ibrutinib IBRUTINIB 27256378,28830912 83359 56805 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE PAZOPANIB PAZOPANIB 83360 56806 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME allosteric modulator 135652725 VINCAMINE 83363 56807 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MPC-3100 83364 56808 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE TENIPOSIDE TENIPOSIDE 9842975 83365 56809 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Quinestrol QUINESTROL 83366 56810 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME METHDILAZINE METHDILAZINE 83368 56811 DAPK3 1613 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME PALBOCICLIB PALBOCICLIB 83369 56812 CD38 952 CELL SURFACE, DRUGGABLE GENOME HUMAX-CD38 DARATUMUMAB 83370 56813 TGFB2 7042 GROWTH FACTOR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor CHEMBL2108967 LERDELIMUMAB 83371 56814 EDNRA 1909 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100778 AMBRISENTAN 83373 56815 XDH 7498 DRUGGABLE GENOME, ENZYME MITOMYCIN-C 3023600 83374 56816 ARG1 383 ENZYME inhibitor 315661102 83375 56817 RAB9A 9367 ENZYME, DRUGGABLE GENOME TENONITROZOLE TENONITROZOLE 83376 56818 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE allosteric modulator 178102544 83377 56819 CYP2C8 1558 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME rosiglitazone ROSIGLITAZONE 17178266,23426382,27271184 83378 56820 AKR1D1 6718 DRUGGABLE GENOME, ENZYME FINASTERIDE FINASTERIDE 83379 56821 SERPINC1 462 DRUGGABLE GENOME, PROTEASE INHIBITOR ARDEPARIN 83380 56822 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME XYLOMETAZOLINE XYLOMETAZOLINE 83382 56823 TNFRSF12A 51330 DRUGGABLE GENOME 178101760 83383 56824 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME METHYSERGIDE METHYSERGIDE 83384 56825 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 318164805 PZM21 83385 56826 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLOROXURON CHLOROXURON 83386 56827 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE 5,7-DIHYDROXY-4-METHYLCOUMARIN 5,7-DIHYDROXY-4-METHYLCOUMARIN 83387 56828 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 249565745 83390 56829 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME 6-AMINONICOTINAMIDE 6-AMINONICOTINAMIDE 153476 83392 56830 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR DIPHENHYDRAMINE HYDROCHLORIDE DIPHENHYDRAMINE HYDROCHLORIDE 83393 56831 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME CHEMBL681 ETOMIDATE 83394 56832 EGLN3 112399 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL2338329 ROXADUSTAT 83395 56833 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 53801076 83397 56834 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME antibody BEVACIZUMAB BEVACIZUMAB 83398 56835 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor PI-103 PI-103 83399 56836 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME ELTROMBOPAG ELTROMBOPAG 21422191 83401 56837 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TENONITROZOLE TENONITROZOLE 83402 56838 GFER 2671 DRUGGABLE GENOME, ENZYME, GROWTH FACTOR GALLIC ACID METHYL ESTER GALLIC ACID METHYL ESTER 83403 56839 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE N/A 83408 56840 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE SULINDAC SULINDAC 12414619 83409 56841 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID28092474-Compound-32l 83410 56842 CLK4 57396 SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, ENZYME JNJ-7706621 JNJ-7706621 83412 56843 HTT 3064 DRUGGABLE GENOME inhibitor CHEMBL1200631 83416 56844 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SIB-1757 CHEMBL88553 83417 56845 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX TCMDC-125086 CHEMBL532504 83418 56846 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CHLORHEXIDINE CHLORHEXIDINE 83419 56847 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FEPRAZONE FEPRAZONE 83422 56848 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Fexofenadine FEXOFENADINE 83423 56849 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME ASTEMIZOLE ASTEMIZOLE 83425 56850 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor PAZOPANIB PAZOPANIB 83426 56851 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3187723 BINIMETINIB 83427 56852 PTGS1 5742 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL704 MESALAMINE 83431 56853 CRTC2 200186 KINASE cyclosporine CYCLOSPORINE 26644205 83432 56854 MAOB 4129 DRUGGABLE GENOME, ENZYME inhibitor 405560268 LINEZOLID 83433 56855 SMN2 6607 DRUGGABLE GENOME 7,2'-DIHYDROXYFLAVONE CHEMBL475908 83434 56856 NR1H3 10062 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651388 83435 56857 PRKCE 5581 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ION CHANNEL, TRANSCRIPTION FACTOR, ENZYME BRYOSTATIN-1 83436 56858 GMNN 51053 DRUGGABLE GENOME CALCIMYCIN CALCIMYCIN 83437 56859 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL1563 DAUNORUBICIN HYDROCHLORIDE 83438 56860 MAPT 4137 DRUGGABLE GENOME RESERPINE RESERPINE 83440 56861 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE Azacitidine AZACITIDINE 24077805 83441 56862 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE EKI-285 17085664,20942962,25948633 83442 56863 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SB-222200 SB-222200 83444 56864 HTR4 3360 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR DA-6886 DA-6886 83447 56865 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 384403645 83449 56866 SLC12A5 57468 DRUGGABLE GENOME, TRANSPORTER inhibitor 178101380 83450 56867 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR CHLORAMBUCIL CHLORAMBUCIL 83451 56868 B4GALT2 8704 ENZYME clopidogrel CLOPIDOGREL 83452 56869 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Bevacizumab BEVACIZUMAB 28632865,21216929,23828442,25363205 83453 56870 POLK 51426 DNA REPAIR, ENZYME 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 83455 56871 TNFRSF1B 7133 DRUGGABLE GENOME CYT-6091 83456 56872 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 2',4'-DIHYDROXY FLAVONE CHEMBL1374610 83458 56873 S1PR3 1903 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME US8524917, 12 83460 56874 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Carboplatin CARBOPLATIN 21216929 83461 56875 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME AG-555 CHEMBL53898 83462 56876 PSEN1 5663 ENZYME, TRANSPORTER, PROTEASE, DRUGGABLE GENOME, CELL SURFACE inhibitor 178103910 RG-4733 83463 56877 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME ALSTERPAULLONE ALSTERPAULLONE 83465 56878 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE MUSTARD 16489579 83466 56879 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 348353623 83468 56880 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER Cremophor EL 83469 56881 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME cotinine COTININE 18004205 83471 56882 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Fluorouracil FLUOROURACIL 28784859,27626067,26432108 83472 56883 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL122 ROFECOXIB 83474 56884 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135651739 83477 56885 TSPO 706 DRUGGABLE GENOME Iodophenyl-N-methyl-N-fluoroalkyl-3-isoquinoline carboxamide derivative 1 83478 56886 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CI-1040 CI-1040 20580230 83479 56887 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE TRAIL 12730676,14977850 83481 56888 SLC16A7 9194 DRUGGABLE GENOME, TRANSPORTER inhibitor 252827475 83484 56889 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3301612 ENCORAFENIB 83485 56890 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME KRH-3955 CHEMBL2062277 19451305 83486 56891 MTTP 4547 DRUGGABLE GENOME atorvastatin ATORVASTATIN 15864113 83487 56892 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor CHEMBL3545133 JNJ-26483327 83489 56893 RPS6KA1 6195 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor 328083458 83490 56894 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME Isoquinoline 1,3-dione derivative 1 83491 56895 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE HALOPERIDOL HALOPERIDOL 16002093 83492 56896 BAZ2B 29994 NA DOXORUBICIN HYDROCHLORIDE DOXORUBICIN HYDROCHLORIDE 83494 56897 RGS4 5999 DRUGGABLE GENOME BENSERAZIDE BENSERAZIDE 83495 56898 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR DACTINOMYCIN DACTINOMYCIN 83496 56899 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX BETA-LAPACHONE LAPACHONE 83499 56900 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALISOL A-23 ACETATE CHEMBL2059711 24915879 83500 56901 SCARB1 949 TRANSPORTER, CELL SURFACE, DRUGGABLE GENOME fenofibrate FENOFIBRATE 83501 56902 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL1922094 APITOLISIB 83502 56903 GSTP1 2950 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME oxaliplatin OXALIPLATIN 10728587,22188361,17409936,9498276,27995989,17401013,19203783,15093273,12435115,11307147,11751440,20530282,16707601,21449681,15213713 83503 56904 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME OLEOYL DOPAMINE OLEOYL DOPAMINE 83504 56905 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Pyrimidine derivative 8 83506 56906 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 KEPONE KEPONE 83507 56907 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL698 TETRACAINE 83508 56908 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL1230609 FORETINIB 83509 56909 HBB 3043 DRUGGABLE GENOME, ENZYME MENADIONE MENADIONE 83510 56910 CD69 969 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME tocilizumab TOCILIZUMAB 27339827 83511 56911 HSPA4 3308 NA PHENYLEPHRINE PHENYLEPHRINE 8047983 83513 56912 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME ERYTHROPOIETIN EPOETIN BETA 10590051 83514 56913 ASXL1 171023 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR Decitabine DECITABINE 25224413 83516 56914 GLO1 2739 ENZYME, DRUGGABLE GENOME NARINGENIN NARINGENIN 83518 56915 BAZ2B 29994 NA 2-AMINOPHENOXAZINONE CHEMBL146710 83519 56916 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE IRINOTECAN IRINOTECAN 25788273 83520 56917 PTGER1 5731 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650094 CICAPROST 83521 56918 CDK6 1021 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE ALVOCIDIB ALVOCIDIB 83522 56919 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ADAPALENE ADAPALENE 83523 56920 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE PHA-739358 DANUSERTIB 83526 56921 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL1094408 NMS-1286937 83529 56922 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE ABP 980 83530 56923 RAB9A 9367 ENZYME, DRUGGABLE GENOME SJ000202381 CHEMBL591598 83531 56924 TNFRSF11B 4982 DRUGGABLE GENOME letrozole LETROZOLE 83533 56925 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME 5-FU FLUOROURACIL 15067352 83534 56926 PPID 5481 DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING, KINASE 1313212-89-3 83535 56927 F7 2155 ENZYME, DRUGGABLE GENOME, PROTEASE Eptacog alfa intravenous 83536 56928 SMN2 6607 DRUGGABLE GENOME (E)-2-STYRYLCHROMONE CHEMBL388823 83538 56929 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME INDOCYANINE GREEN SODIUM INDOCYANINE GREEN 83539 56930 POLB 5423 DNA REPAIR, DRUGGABLE GENOME 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 83541 56931 BARD1 580 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR OLAPARIB OLAPARIB 28389374,27197561 83542 56932 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE NN-818 83543 56933 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE ENPIROLINE ENPIROLINE 83544 56934 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 lumefantrine LUMEFANTRINE 83545 56935 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 4101591 CHEMBL428789 83546 56936 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 328083491 SB590885 83547 56937 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE PF-562271 PF-00562271 83548 56938 TUBA3D 113457 DRUGGABLE GENOME ABT-751 ABT-751 25468039 83549 56939 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR RETINYL ACETATE RETINYL ACETATE 83551 56940 KDM4A 9682 DRUGGABLE GENOME, ENZYME ALEXIDINE HYDROCHLORIDE ALEXIDINE HYDROCHLORIDE 83552 56941 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE NAVARIXIN NAVARIXIN 17181143 83555 56942 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Panitumumab PANITUMUMAB 28514312 83556 56943 SUMO1 7341 ENZYME, DNA REPAIR, TRANSCRIPTION FACTOR BINDING ASTERRIC ACID ASTERRIC ACID 83557 56944 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-11 83558 56945 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE STREPTONIGRIN STREPTONIGRIN 83559 56946 MUC16 94025 DRUGGABLE GENOME ETOPOSIDE ETOPOSIDE 1988893 83562 56947 TH 7054 ENZYME, DRUGGABLE GENOME L-Tyrosine TYROSINE 83563 56948 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 83564 56949 THBD 7056 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME PROSTAGLANDIN E1 7684300 83565 56950 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650055 CARBACHOL 83567 56951 PROS1 5627 DRUGGABLE GENOME Progesterone PROGESTERONE 83568 56952 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE MEPENZOLATE MEPENZOLATE 83569 56953 NRP1 8829 DRUGGABLE GENOME RG7347 26090340 83570 56954 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL1743050 OLOKIZUMAB 83571 56955 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE POMIFERIN POMIFERIN 83573 56956 APOD 347 DRUGGABLE GENOME, ENZYME RETINOIDS 8943263 83574 56957 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR HAPLAMINE HAPLAMINE 83575 56958 RXFP1 59350 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE NECA NECA 83576 56959 CDK5 1020 SERINE THREONINE KINASE, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME PURPUROGALLIN PURPUROGALLIN 83577 56960 HDAC2 3066 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, TRANSCRIPTION FACTOR ROMIDEPSIN ROMIDEPSIN 83578 56961 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE CYTOFAB 83579 56962 ATAD5 79915 NA FASUDIL HYDROCHLORIDE FASUDIL HYDROCHLORIDE 83580 56963 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME IFN 10505750,17239402 83581 56964 TSPO 706 DRUGGABLE GENOME Adinazolam ADINAZOLAM 83582 56965 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL3545422 MIRANSERTIB 83583 56966 ALOX5 240 DRUGGABLE GENOME, ENZYME Tipelukast TIPELUKAST 83584 56967 CYP4A11 1579 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME spironolactone SPIRONOLACTONE 83585 56968 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME SORAFENIB SORAFENIB 83586 56969 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Mitotane MITOTANE 83587 56970 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 83588 56971 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME MUNDULONE ACETATE MUNDULONE ACETATE 83589 56972 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE salmeterol SALMETEROL 23126384,15500895,19800676,19932356,24279851,18156033 83590 56973 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE AZD8055 AZD-8055 28446642 83591 56974 SMN1 6606 DRUGGABLE GENOME DNDI1417031 CHEMBL1333049 83592 56975 CXCL2 2920 DRUGGABLE GENOME DEFEROXAMINE DEFEROXAMINE 17883261 83593 56976 GMNN 51053 DRUGGABLE GENOME NSC-158389 CHEMBL192626 83594 56977 CFH 3075 DRUGGABLE GENOME bevacizumab BEVACIZUMAB 26439641,23584701,23204795,22840423,22594510,23559864,24070809,26411831,23842101,23337555 83595 56978 CXCL8 3576 DRUGGABLE GENOME ANTIHISTAMINE TERFENADINE 8919641 83596 56979 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL3218576 COPANLISIB 83598 56980 TGFBR3 7049 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME RETINOIC ACID 8143777 83599 56981 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER TDR78826 CHEMBL1500913 83602 56982 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME BL-8040 BKT140 83603 56983 ABCB11 8647 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE GS-9256 GS-9256 22244938 83605 56984 BCL2A1 597 DRUGGABLE GENOME inhibitor CHEMBL2107358 OBATOCLAX MESYLATE 83606 56985 MCL1 4170 DRUGGABLE GENOME, CLINICALLY ACTIONABLE ZINC 02849675 CHEMBL605959 83609 56986 ALDH1A1 216 DRUGGABLE GENOME, ENZYME ROFECOXIB ROFECOXIB 83610 56987 APOA1 335 CELL SURFACE, ENZYME, DRUGGABLE GENOME ETHANOL ALCOHOL 10956052 83613 56988 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE HEGF 83615 56989 NUAK1 9891 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565819 83617 56990 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME CHEMBL2105675 TAFAMIDIS MEGLUMINE 83618 56991 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CC-90003 83622 56992 RAB9A 9367 ENZYME, DRUGGABLE GENOME GNF-PF-2307 CHEMBL421088 83623 56993 SOST 50964 DRUGGABLE GENOME Romosozumab ROMOSOZUMAB 83624 56994 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103491 83626 56995 MARCHF8 220972 ENZYME Grippol Plus 83627 56996 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 3,4-DIMETHOXYDALBERGIONE 3,4-DIMETHOXYDALBERGIONE 83628 56997 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR Prednisolone PREDNISOLONE 83631 56998 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL FLUDIAZEPAM FLUDIAZEPAM 83632 56999 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME SBI-087 83634 57000 TUBA1A 7846 DRUGGABLE GENOME CHEMBL2304041 SAGOPILONE 83636 57001 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DABRAFENIB DABRAFENIB 25452114 83637 57002 RPL10 6134 CLINICALLY ACTIONABLE TRANSFORMING GROWTH FACTOR 15345329 83638 57003 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLOROBENZILATE CHLOROBENZILATE 83639 57004 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE CENISERTIB CENISERTIB 83644 57005 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER STREPTONIGRIN STREPTONIGRIN 12027749 83645 57006 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 Erdafitinib   83646 57007 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR METHOTRIMEPRAZINE LEVOMEPROMAZINE 83647 57008 PDE4C 5143 DRUGGABLE GENOME, ENZYME DYPHYLLINE DYPHYLLINE 83648 57009 FXN 2395 TRANSPORTER, ENZYME ERYTHROPOIETIN EPOETIN BETA 16269021 83649 57010 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME GNF-PF-3561 CHEMBL599712 83651 57011 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE ENTRECTINIB ENTRECTINIB 83653 57012 CBX1 10951 NA SJ000147784 CHEMBL590186 83655 57013 ADK 132 DRUGGABLE GENOME, ENZYME, KINASE inhibitor 178101823 83656 57014 MAPKAPK2 9261 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE inhibitor 178102631 83657 57015 P2RX7 5027 NUCLEAR HORMONE RECEPTOR, ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE PMID27724045-Compound-33 83658 57016 PTGS2 5743 DRUGGABLE GENOME, ENZYME Coxibs 19602986 83660 57017 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME OMEPRAZOLE OMEPRAZOLE 83663 57018 SLC28A1 9154 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE URIDINE URIDINE 23388705 83666 57019 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Imidazo isoindole derivative 1 83668 57020 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR 2,4,6-TRIBROMOPHENOL CHEMBL220087 83671 57021 DGAT1 8694 ENZYME, DRUGGABLE GENOME PMID25470667-Compound-PF-04620110 83672 57022 MAPT 4137 DRUGGABLE GENOME PHENSERINE PHENSERINE 83673 57023 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor 249565925 83674 57024 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR LETROZOLE LETROZOLE 83675 57025 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102569 83676 57026 HKDC1 80201 DRUGGABLE GENOME, KINASE DNDI1417941 CHEMBL2095095 83677 57027 COL18A1 80781 DRUGGABLE GENOME VITAMIN C 12792883 83678 57028 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR AR-A014418 CHEMBL259850 83680 57029 MUC2 4583 DRUGGABLE GENOME 5-AZA-2'-DEOXYCYTIDINE 11893907,16112420 83682 57030 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER CAPSAICIN CAPSAICIN 16674925 83683 57031 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR CORT-125134 CORT 125134 83684 57032 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME BVD-523 ULIXERTINIB 83685 57033 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME inhibitor 310264675 CUDC-101 83686 57034 FAAH 2166 ENZYME, DRUGGABLE GENOME Heteroaryl-substituted urea derivative 2 83687 57035 PTK2B 2185 DRUGGABLE GENOME, KINASE, ION CHANNEL, G PROTEIN COUPLED RECEPTOR, TYROSINE KINASE, ENZYME CENISERTIB CENISERTIB 83688 57036 MAPT 4137 DRUGGABLE GENOME DALBERGIONE, 4-METHOXY-4'-HYDROXY- DALBERGIONE, 4-METHOXY-4'-HYDROXY- 83689 57037 SMN2 6607 DRUGGABLE GENOME PHENAMIL PHENAMIL 83690 57038 VEGFB 7423 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR inhibitor ENDOSTATIN (84-114)-NH2 (JKC367) 83691 57039 MAPT 4137 DRUGGABLE GENOME ANGUSTIBALIN ANGUSTIBALIN 83693 57040 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME activator 135651429 83695 57041 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME KUSHENOL A KUSHENOL A 18565755 83696 57042 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE ISOVELLERAL ISOVELLERAL 83697 57043 SOAT1 6646 DRUGGABLE GENOME LOVASTATIN LOVASTATIN 2268271 83699 57044 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE REGORAFENIB REGORAFENIB 27371698,25239608 83700 57045 KIF11 3832 DRUGGABLE GENOME AZD-4877 AZD-4877 83701 57046 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE inhibitor 178103969 CERITINIB 83702 57047 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME VIOXX ROFECOXIB 14627349 83704 57048 HCAR2 338442 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE Vitamin B3 83706 57049 RAB9A 9367 ENZYME, DRUGGABLE GENOME DNDI1417597 CHEMBL1330352 83707 57050 ALDH1A1 216 DRUGGABLE GENOME, ENZYME AG-34 CHEMBL80155 83708 57051 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE LAPATINIB LAPATINIB 83709 57052 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 187051799 DACINOSTAT 83710 57053 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE N/A 83711 57054 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL2007641 PERTUZUMAB 83712 57055 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ALDRIN ALDRIN 83713 57056 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME TAK-733 TAK-733 26439693 83716 57057 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CHEMBL2108041 OCRELIZUMAB 83718 57058 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME Dimenhydrinate DIMENHYDRINATE 83719 57059 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650013 BNTX 83720 57060 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE AMFONELIC ACID AMFONELIC ACID 83721 57061 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE ETANERCEPT ETANERCEPT 83722 57062 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 178103890 TRIMIPRAMINE 83724 57063 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor CHEMBL3545225 INCB-047986 83726 57064 PVALB 5816 NA SALINE SODIUM CHLORIDE 9133585 83729 57065 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178102727 83731 57066 RYR2 6262 B30_2 SPRY DOMAIN, DRUGGABLE GENOME, ION CHANNEL ARM210 83733 57067 TLR7 51284 DRUGGABLE GENOME agonist 178101700 IMIQUIMOD 83734 57068 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE MSC2156119J 25256830 83736 57069 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TAMATINIB R-406 83737 57070 GAPDH 2597 DRUGGABLE GENOME, ENZYME TAMOXIFEN TAMOXIFEN 9883985 83739 57071 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME ER-319711-15 83741 57072 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE TOZASERTIB TOZASERTIB 83742 57073 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 TYRPHOSTIN AG 879 TYRPHOSTIN AG 879 83743 57074 ATAD5 79915 NA RUTAECARPINE RUTAECARPINE 83744 57075 RACGAP1 29127 NA 3-O-METHYLQUERCETIN 3-O-METHYLQUERCETIN 83745 57076 PSMA3 5684 PROTEASE, DRUGGABLE GENOME inhibitor CHEMBL451887 CARFILZOMIB 83746 57077 PDE4A 5141 DRUGGABLE GENOME, ENZYME SUN13834 83747 57078 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE TRAMADOL TRAMADOL 83748 57079 ATAD5 79915 NA GNF-PF-1008 CHEMBL602424 83750 57080 TNFRSF1A 7132 CELL SURFACE, DRUGGABLE GENOME CYT-6091 83751 57081 RXRA 6256 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CLOROPHENE CLOROPHENE 83752 57082 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME EVT-103 83754 57083 HP 3240 DRUGGABLE GENOME, PROTEASE, ENZYME VACCINE 8228935 83755 57084 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME TAK-715 TAK-715 83756 57085 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER TARIQUIDAR TARIQUIDAR 21657271 83757 57086 TCN1 6947 DRUGGABLE GENOME VITAMIN-B12 526444,3018464,1285639,6164603,8438881,474643,1176445,10207776,3332101,2235967,1504859 83759 57087 MAOA 4128 DRUGGABLE GENOME, ENZYME MOCLOBEMIDE MOCLOBEMIDE 83760 57088 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME MYRICETIN MYRICETIN 83762 57089 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME QUETIAPINE QUETIAPINE 83763 57090 NUDT1 4521 DNA REPAIR, ENZYME 8-oxo-dgtp 26238318 83765 57091 GLS 2744 ENZYME PIRARUBICIN PIRARUBICIN 83766 57092 GUCY1A1 2982 ENZYME, DRUGGABLE GENOME positive modulator CHEMBL2107834 RIOCIGUAT 83767 57093 PRKDC 5591 TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 178102584 83769 57094 BCL2L10 10017 DRUGGABLE GENOME inhibitor CHEMBL2107358 OBATOCLAX MESYLATE 83770 57095 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL521851 PICTILISIB 83772 57096 HTT 3064 DRUGGABLE GENOME DNDI1416934 CHEMBL1989750 83773 57097 CCND2 894 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE LY2835219 ABEMACICLIB 83774 57098 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR TOLAZOLINE TOLAZOLINE 83777 57099 S100A9 6280 DRUGGABLE GENOME, KINASE, ENZYME Tasquinimod TASQUINIMOD 24162378 83779 57100 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE MARIMASTAT MARIMASTAT 83780 57101 USP1 7398 DNA REPAIR, PROTEASE, ENZYME ALLOXAN ALLOXAN 83781 57102 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-741905 CHEMBL407113 83783 57103 HTT 3064 DRUGGABLE GENOME MMV007764 CHEMBL609628 83784 57104 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE MITOXANTRONE DIHYDROCHLORIDE MITOXANTRONE HYDROCHLORIDE 83785 57105 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER Seliciclib SELICICLIB 22862161,26826118 83786 57106 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GFT-505 ELAFIBRANOR 83787 57107 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME meperidine MEPERIDINE 17638512,11470993 83788 57108 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME PHENAMIPHOS PHENAMIPHOS 83789 57109 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 249565839 83790 57110 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 249565924 83791 57111 SLCO2B1 11309 TRANSPORTER, DRUGGABLE GENOME SILYDIANIN SILYDIANIN 23401473 83793 57112 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR THEOPHYLLINE THEOPHYLLINE 83795 57113 EREG 2069 KINASE, GROWTH FACTOR, DRUGGABLE GENOME LY3016859 83798 57114 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE MET-ENKEPHALIN CHEMBL13786 17616524 83801 57115 PDE4A 5141 DRUGGABLE GENOME, ENZYME ETAZOLATE ETAZOLATE 83803 57116 GATA2 2624 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX FASUDIL FASUDIL 22541434 83804 57117 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR GENTAMICIN GENTAMICIN 10536212 83806 57118 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME AZD5153 AZD-5153 27573426 83809 57119 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME TAK-070 83810 57120 IMPDH2 3615 DRUGGABLE GENOME, ENZYME inhibitor 178103451 THIOGUANINE 83811 57121 GMNN 51053 DRUGGABLE GENOME DNDI1417649 CHEMBL1994034 83812 57122 POLI 11201 DNA REPAIR PINAFIDE PINAFIDE 83814 57123 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 SULPIRIDE SULPIRIDE 22931300 83815 57124 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR dexamethasone DEXAMETHASONE 15883634,15864137,20727239,18827005,10320522 83816 57125 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CYCLOHEXIMIDE CYCLOHEXIMIDE 83818 57126 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE agonist 135650735 NORMORPHINE 83819 57127 CXCR4 7852 DRUG RESISTANCE, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CTCE-0214 83820 57128 RPS6KB1 6198 CELL SURFACE, SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME, CLINICALLY ACTIONABLE VATALANIB VATALANIB 83822 57129 MAP2K7 5609 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TYROSINE KINASE, ENZYME inhibitor TRAMETINIB TRAMETINIB 83827 57130 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME Volasertib VOLASERTIB 83828 57131 DCLK1 9201 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 249565887 83829 57132 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME TENONITROZOLE TENONITROZOLE 83830 57133 GRIN2D 2906 ION CHANNEL, DRUGGABLE GENOME blocker 178101050 KETAMINE 83831 57134 GNAS 2778 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR, DRUG RESISTANCE, TRANSPORTER DNDI1417319 CHEMBL1392244 83833 57135 GMNN 51053 DRUGGABLE GENOME SJ000114740 CHEMBL592068 83834 57136 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL2105708 PONATINIB HYDROCHLORIDE 83835 57137 DYRK2 8445 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME, TRANSCRIPTION FACTOR PMID28766366-Compound-Scheme21Right 83837 57138 GLCCI1 113263 NA flunisolide FLUNISOLIDE 21991891 83838 57139 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME PMID27774824-Compound-Figure2Example4 83840 57140 PLAU 5328 PROTEASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE inhibitor 178103111 UPAMOSTAT 83843 57141 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR 4-TRIETHYLSILYLPHENOL CHEMBL2313445 23214428 83844 57142 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE Pyridine derivative 18 83845 57143 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE FLUOCINOLONE ACETONIDE 16454812 83846 57144 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR PRAZOSIN PRAZOSIN 83847 57145 FN1 2335 DRUGGABLE GENOME CHEMBL2109589 L19TNFA 83848 57146 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME PMID29671355-Compound-11 83849 57147 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000032150 CHEMBL607140 83850 57148 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Gedatolisib GEDATOLISIB 24042735,25673820,25688157,21325073 83854 57149 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX JTC-801 CHEMBL140979 83855 57150 BAZ2B 29994 NA ISOKAEMPFERIDE ISOKAEMPFERIDE 83857 57151 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE SB-203580 SB-203580 83858 57152 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME N-(3,4-DICHLOROPHENYL)BENZAMIDE CHEMBL560296 83861 57153 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR GNF-PF-4370 CHEMBL600971 83862 57154 RGS4 5999 DRUGGABLE GENOME 4-CHLOROMERCURIBENZOIC ACID 4-CHLOROMERCURIBENZOIC ACID 83863 57155 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 249565645 MK-2461 83864 57156 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE inhibitor BGJ398 INFIGRATINIB 83865 57157 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE inhibitor ABIRATERONE ACETATE ZYTIGA 83866 57158 KDM4A 9682 DRUGGABLE GENOME, ENZYME NAFRONYL OXALATE NAFRONYL OXALATE 83867 57159 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE modulator CHEMBL3545417 GLPG0492 83869 57160 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GSK2636771 GSK-2636771 26117819,23674493,26577700,26645196 83870 57161 IKBKB 3551 SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME SC-514 CHEMBL193093 18702457 83871 57162 MELK 9833 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE SP-600125 SP-600125 83872 57163 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE DEXANABINOL DEXANABINOL 83875 57164 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417156 CHEMBL1504679 83878 57165 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL452 CLONAZEPAM 83879 57166 KDM4A 9682 DRUGGABLE GENOME, ENZYME EMBELIN EMBELIN 83880 57167 HSPB1 3315 DRUGGABLE GENOME ROFECOXIB ROFECOXIB 16041694 83881 57168 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR U-0124 CHEMBL97858 83882 57169 ALOX15B 247 DRUGGABLE GENOME, ENZYME FENTICLOR FENTICLOR 83883 57170 SH2B1 25970 KINASE paliperidone PALIPERIDONE 28694205 83884 57171 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE EFAVIRENZ EFAVIRENZ 21189339,17172311 83885 57172 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE METHOTREXATE METHOTREXATE 12972956 83888 57173 PLAUR 5329 DRUGGABLE GENOME, ENZYME, CELL SURFACE PHORBOL MYRISTATE ACETATE 9531044 83890 57174 GJB1 2705 ION CHANNEL, DRUGGABLE GENOME, TRANSPORTER inhibitor 135650269 83891 57175 TUBB6 84617 DRUGGABLE GENOME PODOFILOX PODOFILOX 17765552,24953821,21402478 83892 57176 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME antagonist 178100733 83893 57177 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CID 739615 CHEMBL260560 83894 57178 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER corticosteroids 83895 57179 RGS4 5999 DRUGGABLE GENOME METHYLERGONOVINE METHYLERGONOVINE 83897 57180 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE inhibitor 318164841 NETARSUDIL 83898 57181 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE 13-CIS-RETINOIC ACID 10621853 83899 57182 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME Ruxolitinib RUXOLITINIB 83901 57183 GABRB2 2561 DRUGGABLE GENOME, ION CHANNEL CHLORDIAZEPOXIDE CHLORDIAZEPOXIDE 83902 57184 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME inhibitor 404858998 83903 57185 TPM3 7170 KINASE, CLINICALLY ACTIONABLE RETINOID 8522994 83904 57186 CDKN2C 1031 CLINICALLY ACTIONABLE, KINASE ANTISENSE OLIGONUCLEOTIDES 12821941 83905 57187 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE PONATINIB PONATINIB 20513156 83906 57188 KIF11 3832 DRUGGABLE GENOME ISPINESIB ISPINESIB 83909 57189 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE inhibitor REGORAFENIB REGORAFENIB 83913 57190 COL1A2 1278 DRUGGABLE GENOME TRANSFORMING GROWTH FACTOR 14520013 83914 57191 CBX1 10951 NA E-64 E-64 83915 57192 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME raloxifene RALOXIFENE 19364970,19852077,18349289,12181437,17058217,12969965,1651156,18466101,14647407,20562211,19390945,17728214,12019197,10381366,11037804 83916 57193 BCHE 590 DRUGGABLE GENOME, ENZYME DEMECARIUM BROMIDE 83917 57194 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR MERCURIC CHLORIDE MERCURIC CHLORIDE 83918 57195 ASS1 445 ENZYME, DRUG RESISTANCE PEGARGIMINASE PEGARGIMINASE 27735949 83920 57196 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antagonist CHEMBL1743006 DALOTUZUMAB 83922 57197 IFNAR1 3454 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE INTERFERON ALFACON-1 83923 57198 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1201454 ALSEROXYLON 83924 57199 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID29671355-Compound-42 83925 57200 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650846 PRACTOLOL 83926 57201 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID28394193-Compound-56 83927 57202 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR (E),(E)-2,4-DECACIENAL CHEMBL443949 83930 57203 TSPO 706 DRUGGABLE GENOME Imidazopyridine derivative 2 83935 57204 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 (+)-HYDRASTINE CHEMBL1256868 83936 57205 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR ARRY-614 PEXMETINIB 83938 57206 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE Cetuximab CETUXIMAB 27149458 83940 57207 PDE5A 8654 ENZYME, DRUGGABLE GENOME UDENAFIL UDENAFIL 83941 57208 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 178103904 BARASERTIB 83942 57209 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MENADIONE MENADIONE 83944 57210 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME XMT-1536 XMT-1536 83945 57211 PLA2G1B 5319 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME, CELL SURFACE RETINOIDS 3218613 83946 57212 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE TRAMETINIB TRAMETINIB 25952648 83947 57213 POLI 11201 DNA REPAIR ELLIPTECINE ELLIPTECINE 83949 57214 PRKCZ 5590 DRUGGABLE GENOME, KINASE, TRANSPORTER, ENZYME, SERINE THREONINE KINASE inhibitor 249565865 83950 57215 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME PENTACHLOROPHENOL PENTACHLOROPHENOL 83951 57216 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME RESMINOSTAT RESMINOSTAT 83952 57217 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE Ganetespib GANETESPIB 26483207 83953 57218 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE RG-1530 RG-1530 83954 57219 GALNT14 79623 ENZYME mitoxantrone MITOXANTRONE 31611591,21635146 83956 57220 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME inhibitor CUDC-101 CUDC-101 83957 57221 EIF2AK3 9451 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Indoline derivative 2 83958 57222 POLI 11201 DNA REPAIR HYDROXYZINE PAMOATE HYDROXYZINE PAMOATE 83962 57223 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 135650192 DIPHENHYDRAMINE 83964 57224 TARDBP 23435 TUMOR SUPPRESSOR CHLORHEXIDINE CHLORHEXIDINE 83965 57225 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR CAFFEINE CAFFEINE 83966 57226 GMNN 51053 DRUGGABLE GENOME SJ000071854 CHEMBL602127 83968 57227 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME APIGENIN APIGENIN 83969 57228 MAPKAPK3 7867 ENZYME, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR LAUROGUADINE LAUROGUADINE 83970 57229 FOLR1 2348 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME DEXAMETHASONE DEXAMETHASONE 15899836 83971 57230 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME THIOPHANATE METHYL THIOPHANATE METHYL 83973 57231 KDM4A 9682 DRUGGABLE GENOME, ENZYME BAS-8770954 CHEMBL478324 83974 57232 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PD0166285 11719452 83975 57233 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR OLEOYLETHANOLAMIDE OLEOYLETHANOLAMIDE 83978 57234 NSD2 7468 CLINICALLY ACTIONABLE, METHYL TRANSFERASE, ENZYME DNDI1417156 CHEMBL1504679 83979 57235 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178103275 83980 57236 APOB 338 DRUGGABLE GENOME, CLINICALLY ACTIONABLE SPC4955 83981 57237 TPMT 7172 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME cyclosporine CYCLOSPORINE 16044099,15476481 83982 57238 MMP7 4316 NEUTRAL ZINC METALLOPEPTIDASE, DRUGGABLE GENOME, ENZYME, PROTEASE inhibitor 178101905 MARIMASTAT 83983 57239 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE ALKS 37 83984 57240 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME PF-562271 PF-00562271 83985 57241 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR FASUDIL FASUDIL 83987 57242 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR ZINC SULFATE 16962724 83988 57243 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME BELVARAFENIB 83990 57244 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TOTAROL TOTAROL 83991 57245 MAOB 4129 DRUGGABLE GENOME, ENZYME NAPHTHOQUINONE NAPHTHOQUINONE 22071524 83992 57246 MMP9 4318 DRUGGABLE GENOME, PROTEASE, ENZYME, NEUTRAL ZINC METALLOPEPTIDASE, DRUG RESISTANCE AE-941 83993 57247 PDPK1 5170 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME GNF-PF-2301 CHEMBL578061 83994 57248 BCHE 590 DRUGGABLE GENOME, ENZYME BUPIVACAINE BUPIVACAINE 14631501 83995 57249 MPHOSPH8 54737 NA METHIOTHEPIN MESYLATE METHIOTHEPIN MESYLATE 83996 57250 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR ANISOTROPINE METHYLBROMIDE 83998 57251 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 ATHRAQUINONES A ATHRAQUINONES A 84001 57252 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME CADMIUM DICHLORIDE CADMIUM DICHLORIDE 84002 57253 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE DIGOXIGENIN DIGOXIGENIN 84005 57254 ADORA2B 136 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651063 84006 57255 NOS1 4842 DRUGGABLE GENOME, ENZYME ANTIDEPRESSANTS 12480166 84011 57256 MARK2 2011 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME APAP ACETAMINOPHEN 17654741 84013 57257 PSMC1 5700 PROTEASE inhibitor CARFILZOMIB CARFILZOMIB 84016 57258 PDE3A 5139 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL932 DIPYRIDAMOLE 84017 57259 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NICARDIPINE HYDROCHLORIDE NICARDIPINE HYDROCHLORIDE 84018 57260 ATP2B1 490 DRUGGABLE GENOME, TRANSPORTER, ENZYME Antihypertensives 25385345 84019 57261 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME 2-HYDRAZINYLBENZO[D]THIAZOLE CHEMBL1933308 24262887 84020 57262 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME RAZOXANE RAZOXANE 84022 57263 HLA-C 3107 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE gemcitabine GEMCITABINE 31616045 84023 57264 LIPA 3988 ENZYME, DRUGGABLE GENOME GLUCAGON GLUCAGON 8900456 84025 57265 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME SJ000032081 CHEMBL590184 84026 57266 DPYS 1807 ENZYME DEXRAZOXANE DEXRAZOXANE 7902252 84028 57267 CBX1 10951 NA NAPROXEN NAPROXEN 84029 57268 MGLL 11343 DRUGGABLE GENOME, ENZYME N-PHENYLMALEIMIDE CHEMBL76012 19583260 84031 57269 DHFR 1719 DRUGGABLE GENOME, ENZYME 1954U89 84032 57270 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PENTABROMOPHENOL PENTABROMOPHENOL 84034 57271 MMP14 4323 PROTEASE, DRUGGABLE GENOME, ENZYME GM6001 84035 57272 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME PD-0118057 CHEMBL521083 84036 57273 BRD2 6046 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 187051825 84038 57274 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME SULINDAC SULFIDE 15657353 84039 57275 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE AZD-2115 84041 57276 AXL 558 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, KINASE, TYROSINE KINASE, CELL SURFACE ENTRECTINIB ENTRECTINIB 84043 57277 PANX1 24145 ION CHANNEL inhibitor 135650269 84044 57278 POLK 51426 DNA REPAIR, ENZYME PENTAMIDINE DIISETHIONATE PENTAMIDINE ISETHIONATE 84045 57279 BACE1 23621 DRUGGABLE GENOME, PROTEASE, CELL SURFACE, ENZYME JNJ-54861911 ATABECESTAT 84046 57280 TUBA1B 10376 DRUGGABLE GENOME VINORELBINE BASE VINORELBINE 25768699 84047 57281 POLI 11201 DNA REPAIR METHYLDOPA METHYLDOPA 84048 57282 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE inhibitor 178102585 DOVITINIB 84050 57283 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME VORINOSTAT VORINOSTAT 84051 57284 PTGS2 5743 DRUGGABLE GENOME, ENZYME inhibitor 178103871 SUPROFEN 84053 57285 POLB 5423 DNA REPAIR, DRUGGABLE GENOME CEFOTAXIME SODIUM CEFOTAXIME SODIUM 84054 57286 LIPG 9388 DRUGGABLE GENOME, ENZYME, LIPASE, CELL SURFACE, PHOSPHOLIPASE inhibitor 178103308 84055 57287 POLK 51426 DNA REPAIR, ENZYME GNF-PF-1969 CHEMBL601364 84057 57288 SMS 6611 DRUGGABLE GENOME 2-hydroxyoleic acid 84059 57289 HLA-DRB1 3123 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME azathioprine AZATHIOPRINE 25217962 84060 57290 CLK2 1196 SERINE THREONINE KINASE, TYROSINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor 340590250 LORECIVIVINT 84062 57291 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR GDC-0425 RG-7602 84063 57292 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR inhibitor 404859150 HALICIN 84064 57293 TBP 6908 TRANSCRIPTION FACTOR VP-16 ETOPOSIDE PHOSPHATE 1646402 84066 57294 ATAD5 79915 NA PECTOLINARIGENIN PECTOLINARIGENIN 84067 57295 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE docetaxel DOCETAXEL 20157331 84070 57296 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE IFN 10462502 84072 57297 BCHE 590 DRUGGABLE GENOME, ENZYME inhibitor 178103299 TACRINE 84073 57298 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME FLUPIRTINE FLUPIRTINE 84076 57299 SLC12A4 6560 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSPORTER BUMETANIDE BUMETANIDE 84077 57300 PTGS2 5743 DRUGGABLE GENOME, ENZYME nimesulide NIMESULIDE 84078 57301 P4HB 5034 THIOREDOXIN, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE DIHYDRODAPHNODORIN B DIHYDRODAPHNODORIN B 84081 57302 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE BIZELESIN BIZELESIN 10933811 84082 57303 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Segesterone acetate and ethinyl estradiol vaginal system 84084 57304 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE flutamide FLUTAMIDE 84085 57305 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CGP-71683A CGP-71683A 84087 57306 BAZ2B 29994 NA QUINOLINIC ACID QUINOLINIC ACID 84088 57307 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PSC-833 10609555 84089 57308 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR inhibitor CHEMBL3545218 VORUCICLIB 84091 57309 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME PMID28621580-Compound-WO2015089220C70 84094 57310 CACNA2D2 9254 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL1628502 GABAPENTIN ENACARBIL 84095 57311 GMNN 51053 DRUGGABLE GENOME TANSHINONE I TANSHINONE I 84097 57312 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME AG-1879 CHEMBL406845 84099 57313 TUBA1B 10376 DRUGGABLE GENOME CHEMBL2304041 SAGOPILONE 84100 57314 TRPM3 80036 ION CHANNEL, DRUGGABLE GENOME blocker 135652740 84101 57315 TXNRD1 7296 DRUGGABLE GENOME PMID27977313-Compound-45 84103 57316 CEACAM5 1048 CELL SURFACE, DRUGGABLE GENOME CALCIUM GLUCONATE 709521 84108 57317 GMNN 51053 DRUGGABLE GENOME ENPIROLINE ENPIROLINE 84109 57318 IMPDH1 3614 ENZYME, DRUGGABLE GENOME Urea and carbamate bioisostere derivative 9 84110 57319 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE FLUTAMIDE FLUTAMIDE 84112 57320 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE TCMDC-125758 CHEMBL546797 84113 57321 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT PYRROLIDINE DITHIOCARBAMIC ACID, AMMONIUM SALT 84114 57322 ALOX5 240 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1201013 OLSALAZINE SODIUM 84115 57323 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR PREDNISONE PREDNISONE 84118 57324 FER 2241 KINASE, DRUGGABLE GENOME, ENZYME, TYROSINE KINASE SOTRASTAURIN SOTRASTAURIN 84119 57325 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR Barusiban BARUSIBAN 84120 57326 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE olaparib OLAPARIB 84121 57327 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME sertraline SERTRALINE 26830411 84123 57328 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR LY3214996 84124 57329 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR THIORPHAN THIORPHAN 84125 57330 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL741 LAMOTRIGINE 84126 57331 AKT3 10000 DRUGGABLE GENOME, KINASE, ENZYME, DRUG RESISTANCE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE allosteric modulator 249565628 MK-2206 84127 57332 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME NSD-644 84129 57333 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Bosutinib BOSUTINIB 84131 57334 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE AZD-4017 AZD-4017 84132 57335 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE Pyrrolo[2,3-d]pyrimidine derivative 4 84133 57336 NEK2 4751 ENZYME, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE DOVITINIB DOVITINIB 84138 57337 PTGS2 5743 DRUGGABLE GENOME, ENZYME MELOXICAM MELOXICAM 84139 57338 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor 385612234 84140 57339 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE inhibitor CHEMBL2387080 TASELISIB 84141 57340 MAOB 4129 DRUGGABLE GENOME, ENZYME 8-{[(4-BROMOPHENYL)METHYL]SULFANYL}CAFFEINE CHEMBL1927670 22055712 84144 57341 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE DIFENOCONAZOLE DIFENOCONAZOLE 84145 57342 KCNQ5 56479 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL113461 TEDISAMIL 84148 57343 CHEK2 11200 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SP-600125 SP-600125 84151 57344 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE 3-oxo-2,3-dihydro-1H-indazole-4-carboxamide derivative 3 84155 57345 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PYRITHIONE PYRITHIONE 84157 57346 ICAM1 3383 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME APC-8015F 84158 57347 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR EPZ005687 23023262 84161 57348 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME VER-49009 CHEMBL365617 84163 57349 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME TCMDC-123723 CHEMBL525103 84164 57350 MS4A2 2206 EXTERNAL SIDE OF PLASMA MEMBRANE R112 84165 57351 IMPDH1 3614 ENZYME, DRUGGABLE GENOME inhibitor CHEMBL727 THIOGUANINE 84166 57352 RAB27A 5873 ENZYME Emapalumab-lzsg EMAPALUMAB 84168 57353 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PYRITHIONE ZINC PYRITHIONE ZINC 84170 57354 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME Cyclohexyl azetidine derivative 1 84172 57355 HTT 3064 DRUGGABLE GENOME PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 84173 57356 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CARDAMOMIN CARDAMOMIN 84174 57357 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME inhibitor 178103213 84175 57358 PDE5A 8654 ENZYME, DRUGGABLE GENOME SLX-2101 84177 57359 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME AUTO2 84178 57360 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME SLAZINIC ACID SLAZINIC ACID 84180 57361 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR agonist 178103650 ETHINYL ESTRADIOL 84181 57362 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR HYDRAMETHYLNON HYDRAMETHYLNON 84184 57363 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE TCMDC-125810 CHEMBL528119 84185 57364 MAOB 4129 DRUGGABLE GENOME, ENZYME [18F]FLUORORASAGILINE [18F]FLUORORASAGILINE 22436387 84186 57365 TMEM97 27346 NA Piperazinyl norbenzomorphane compound 4 84187 57366 ECE1 1889 DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, PROTEASE inhibitor 178103176 84188 57367 BAX 581 TUMOR SUPPRESSOR, DRUGGABLE GENOME LEVODOPA LEVODOPA 15672541 84190 57368 HBB 3043 DRUGGABLE GENOME, ENZYME 8-AZAGUANINE 8-AZAGUANINE 84191 57369 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417457 CHEMBL1530911 84194 57370 DDC 1644 ENZYME, DRUGGABLE GENOME CARBIDOPA CARBIDOPA 84195 57371 KDM4A 9682 DRUGGABLE GENOME, ENZYME ATHRAQUINONES A ATHRAQUINONES A 84196 57372 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR inhibitor CHEMBL2178577 AZD-5363 84197 57373 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE RG-1530 RG-1530 84198 57374 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor CHEMBL603469 LESTAURTINIB 84200 57375 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000031505 CHEMBL589479 84201 57376 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL NIFEDIPINE NIFEDIPINE 84203 57377 MARK3 4140 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DIMETHYLADENINE DIMETHYLADENINE 84204 57378 MAP2K1 5604 ENZYME, DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, DRUG RESISTANCE, TYROSINE KINASE, NUCLEAR HORMONE RECEPTOR inhibitor CHEMBL1097999 E-6201 84205 57379 SCNN1G 6340 ION CHANNEL, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE blocker CHEMBL3545352 P-1037 84207 57380 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE leucovorin LEUCOVORIN 22486600 84208 57381 CDC25B 994 DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE NSC-71881 CHEMBL357170 22524450 84209 57382 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME EUPAFOLIN EUPAFOLIN 84211 57383 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE tolbutamide TOLBUTAMIDE 84212 57384 KDM4A 9682 DRUGGABLE GENOME, ENZYME TERPYRIDINE TERPYRIDINE 84213 57385 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME RESCINNAMINE RESCINNAMINE 84214 57386 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR LISOFYLLINE LISOFYLLINE 9227316 84216 57387 PORCN 64840 ENZYME, DRUGGABLE GENOME, TRANSPORTER LGK974 WNT-974 84217 57388 PSMB7 5695 DRUGGABLE GENOME, PROTEASE inhibitor CHEMBL451887 CARFILZOMIB 84218 57389 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 135649654 84219 57390 SMAD2 4087 KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX CURCUMIN CURCUMIN 23145932 84220 57391 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL DEUTERATED DEXTROMETHORPHAN 84221 57392 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TYRPHOSTIN 25 TYRPHOSTIN 25 84222 57393 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR everolimus EVEROLIMUS 84223 57394 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE BIIB037 84224 57395 CELF4 56853 NA iloperidone ILOPERIDONE 18521091 84227 57396 POLI 11201 DNA REPAIR ACETOSIDE ACETOSIDE 84228 57397 POLI 11201 DNA REPAIR NSC-228155 CHEMBL505670 84229 57398 ACE2 59272 ENZYME, TRANSPORTER, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, CELL SURFACE, PROTEASE captopril CAPTOPRIL 17473847 84231 57399 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME inhibitor 315661286 ULIXERTINIB 84234 57400 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TERFENADINE TERFENADINE 84235 57401 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor GDC-0941 PICTILISIB 84236 57402 SLC25A4 291 DRUGGABLE GENOME, TRANSPORTER inhibitor 53801038 84238 57403 MAOB 4129 DRUGGABLE GENOME, ENZYME SELEGILINE SELEGILINE 84240 57404 NFKB2 4791 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR FRENTIZOLE FRENTIZOLE 84242 57405 NT5E 4907 ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME VESNARINONE VESNARINONE 9133521 84243 57406 MDM2 4193 CLINICALLY ACTIONABLE, ENZYME, TUMOR SUPPRESSOR, DRUGGABLE GENOME JNJ-26854165 SERDEMETAN 84244 57407 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE GDC0879 19276360 84245 57408 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME Crizotinib CRIZOTINIB 84246 57409 USP1 7398 DNA REPAIR, PROTEASE, ENZYME PERFLUNAFENE PERFLUNAFENE 84247 57410 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CIS-4-AMINOCROTONIC ACID CHEMBL32307 84248 57411 MINK1 50488 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE SP-600125 SP-600125 84249 57412 SYK 6850 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL3545138 PRT-2607 84250 57413 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL285674 ESTAZOLAM 84251 57414 FABP4 2167 DRUGGABLE GENOME PMID27109571-Compound-27 84252 57415 CDA 978 ENZYME, DRUGGABLE GENOME CYTOSINE ARABINOSIDE 14744791 84253 57416 HDAC4 9759 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR, ENZYME PMID29671355-Compound-71b 84254 57417 A2M 2 ENZYME, TRANSPORTER, DRUGGABLE GENOME, PROTEASE INHIBITOR THROMBIN THROMBIN 2432677 84255 57418 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 PD-123319 CHEMBL157946 84256 57419 UGT1A1 54658 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME DAIDZEIN DAIDZEIN 21030469 84257 57420 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY ZP2929 84258 57421 GUCY2C 2984 DRUGGABLE GENOME, KINASE agonist 178101777 84259 57422 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-720622 CHEMBL1287980 84260 57423 ACVR1 90 DRUGGABLE GENOME, ENZYME, KINASE, SERINE THREONINE KINASE DACTOLISIB DACTOLISIB 84261 57424 SLC29A1 2030 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME FLUDARABINE FLUDARABINE 23388705 84262 57425 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME ethambutol ETHAMBUTOL 28389387 84265 57426 SIRT1 23411 TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME SURAMIN SURAMIN 21215647 84266 57427 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME PARAPLATIN CARBOPLATIN 84267 57428 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650493 84268 57429 PAX8 7849 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE PINAFIDE PINAFIDE 84269 57430 MGMT 4255 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DNA REPAIR, ENZYME TEMOZOLOMIDE TEMOZOLOMIDE 30782343,25910840,15758010,21365007,17442989,21331613 84271 57431 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME Avatrombopag AVATROMBOPAG 84272 57432 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME exemestane EXEMESTANE 84275 57433 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL1200464 PROPARACAINE HYDROCHLORIDE 84277 57434 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 310264749 SERABELISIB 84279 57435 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME PIMOZIDE PIMOZIDE 84280 57436 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE METHYL 4-(3-METHOXYBENZAMIDO)BENZOATE CHEMBL1214407 84282 57437 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR Gemcitabine GEMCITABINE 25156567 84283 57438 KCNQ1 3784 DRUGGABLE GENOME, ION CHANNEL, CELL SURFACE tacrolimus TACROLIMUS 21355884 84284 57439 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE AME-527 84286 57440 NECTIN4 81607 DRUGGABLE GENOME Enfortumab Vedotin-ejfv 84287 57441 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR IODOQUINOL IODOQUINOL 84288 57442 HDAC3 8841 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME inhibitor 252166578 ABEXINOSTAT 84289 57443 PDE9A 5152 DRUGGABLE GENOME, ENZYME inhibitor 178101953 84290 57444 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME enalapril ENALAPRIL 26002049 84291 57445 CSNK1G3 1456 SERINE THREONINE KINASE, DRUGGABLE GENOME, KINASE, ENZYME GS 6201 GS 6201 84292 57446 GPT 2875 ENZYME GLUCAGON GLUCAGON 9808480 84294 57447 PGR 5241 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Anastrozole ANASTROZOLE 84295 57448 TNK2 10188 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME US8481733, 118 84297 57449 KDM4A 9682 DRUGGABLE GENOME, ENZYME FLUPIRTINE MALEATE FLUPIRTINE MALEATE 84298 57450 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Palonosetron PALONOSETRON 84299 57451 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor PLX3397 PEXIDARTINIB 84300 57452 SULT1A1 6817 DRUGGABLE GENOME, ENZYME conjugated estrogens 16985250 84302 57453 BCHE 590 DRUGGABLE GENOME, ENZYME Protexia 84305 57454 NFKBIL1 4795 NA IFN 16362817 84307 57455 PDE4A 5141 DRUGGABLE GENOME, ENZYME GPD-1116 84308 57456 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER OSM-S-85 CHEMBL1494650 84309 57457 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 DANTROLENE DANTROLENE 22931300 84310 57458 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME EVT-201 84311 57459 TUBB4B 10383 DRUGGABLE GENOME CHEMBL2105643 FOSBRETABULIN TROMETHAMINE 84312 57460 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL2103827 DROXIDOPA 84313 57461 TARDBP 23435 TUMOR SUPPRESSOR CLOROPHENE CLOROPHENE 84314 57462 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Dextromethorphan Polistirex 84316 57463 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR ALDOSTERONE ALDOSTERONE 16759088 84320 57464 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME NSAIDS 17270149 84322 57465 POLK 51426 DNA REPAIR, ENZYME APIGENIN APIGENIN 84324 57466 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR PURMORPHAMINE PURMORPHAMINE 16408088 84327 57467 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR SJ000143975 CHEMBL196585 84329 57468 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALTRENOGEST ALTRENOGEST 84330 57469 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR ZINC SULFATE 15715661 84331 57470 TNNC1 7134 DRUGGABLE GENOME BEPRIDIL BEPRIDIL 84333 57471 NTRK2 4915 KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE RXDX 101 84336 57472 CSNK1G1 53944 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME LINIFANIB LINIFANIB 84338 57473 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE EPIANDROSTERONE EPIANDROSTERONE 84339 57474 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HINOKITIOL HINOKITIOL 84340 57475 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 223365978 AEE-788 84341 57476 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-659162 CHEMBL471005 84342 57477 DYRK3 8444 TYROSINE KINASE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SB-220025 SB-220025 84343 57478 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME agonist CHEMBL2105765 LIPEGFILGRASTIM 84345 57479 VEGFB 7423 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR LENALIDOMIDE LENALIDOMIDE 84347 57480 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 trimipramine TRIMIPRAMINE 14520122 84352 57481 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SK-7068 CHEMBL152543 84353 57482 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE inhibitor CHEMBL491473 CEDIRANIB 84355 57483 MAP2K4 6416 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, SERINE THREONINE KINASE, ENZYME inhibitor DABRAFENIB MESYLATE 84356 57484 CBX1 10951 NA PICEATANNOL PICEATANNOL 84357 57485 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME SSR128129E 23597562 84358 57486 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME DIGITOXIN DIGITOXIN 16309315 84362 57487 NOS1 4842 DRUGGABLE GENOME, ENZYME PHENYLEPHRINE PHENYLEPHRINE 12124213 84366 57488 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME (+)-7,9-DEOXYTHYSANONE CHEMBL607534 19783445 84368 57489 CYP1B1 1545 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450, CLINICALLY ACTIONABLE inhibitor 252827406 84369 57490 CHEK1 1111 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DNA REPAIR inhibitor 336446935 PREXASERTIB 84370 57491 SCN2B 6327 ION CHANNEL, DRUGGABLE GENOME ZONISAMIDE ZONISAMIDE 84371 57492 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENFORMIN HYDROCHLORIDE PHENFORMIN HYDROCHLORIDE 84372 57493 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE TRIAMCINOLONE TRIAMCINOLONE 4077022 84373 57494 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CYCLIC ADENOSINE MONOPHOSPHATE CYCLIC ADENOSINE MONOPHOSPHATE 84376 57495 KAT2A 2648 TUMOR SUPPRESSOR, ENZYME TRAZODONE TRAZODONE 84378 57496 GMNN 51053 DRUGGABLE GENOME GROSSHEIMIN GROSSHEIMIN 84379 57497 PDE10A 10846 ENZYME, DRUGGABLE GENOME 1,2,4-triazole [4,3-a]quinoxaline derivative 1 84381 57498 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Ipatasertib IPATASERTIB 24141624 84385 57499 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 249565858 84387 57500 FN1 2335 DRUGGABLE GENOME CHEMBL2109412 L19SIP 131I 84388 57501 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 ETHINYL ESTRADIOL ETHINYL ESTRADIOL 22931300 84389 57502 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 HYDROXYZINE HYDROXYZINE 22931300 84390 57503 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE Topotecan TOPOTECAN 84391 57504 MAPK14 1432 TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1090090 VX-702 84392 57505 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE PYRROLIDINE DITHIOCARBAMATE PYRROLIDINE DITHIOCARBAMATE 84393 57506 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR EPLERENONE EPLERENONE 84395 57507 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE warfarin WARFARIN 18695978 84396 57508 HLA-DRB5 3127 DRUGGABLE GENOME, CLINICALLY ACTIONABLE clavulanate CLAVULANIC ACID 10535882 84400 57509 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE Trametinib TRAMETINIB 84402 57510 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BEVANTOLOL BEVANTOLOL 84404 57511 RNASEH2A 10535 ENZYME TRANSFORMING GROWTH FACTOR 7547241 84405 57512 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 13 84406 57513 DNMT1 1786 DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PMID27376512-Compound-asCEBP-2 84407 57514 SMAD4 4089 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, DRUG RESISTANCE, KINASE Alectinib ALECTINIB 28476735 84409 57515 CDKN1B 1027 DRUG RESISTANCE, TUMOR SUPPRESSOR, CLINICALLY ACTIONABLE, KINASE EPO EPOETIN ALFA 15122318 84410 57516 FRK 2444 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, ENZYME inhibitor CHEMBL403989 TG100-801 84411 57517 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 DERRUSTONE DERRUSTONE 84412 57518 VDAC3 7419 KINASE PRLX93936 84413 57519 SETD2 29072 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE Oligooxopiperazine derivative 1 84414 57520 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 381118818 84415 57521 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ACTB1003 84416 57522 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE DEXAMETHASONE DEXAMETHASONE 1587399 84418 57523 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME ZSTK474 26137449 84419 57524 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL1200802 TALBUTAL 84422 57525 DMD 1756 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Biostrophin 84424 57526 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE AZINPHOS-ETHYL AZINPHOS-ETHYL 84428 57527 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL3545195 LY-3009120 84430 57528 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 315661180 ZOTIRACICLIB 84431 57529 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR LEVODOPA LEVODOPA 84432 57530 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 AMINOPURVALANOL AMINOPURVALANOL 84434 57531 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PT-101 CHEMBL316796 84435 57532 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE imatinib IMATINIB 27426203 84436 57533 KMT2A 4297 METHYL TRANSFERASE, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME MMV000704 CHEMBL582478 84437 57534 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE nilotinib NILOTINIB 84439 57535 KLK3 354 DRUGGABLE GENOME, PROTEASE, ENZYME RETINOIC ACID 15447848 84440 57536 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor AZD8931 SAPITINIB 84441 57537 ATAD5 79915 NA CAFFEIC ACID PHENETHYL ESTER CAFFEIC ACID PHENETHYL ESTER 84442 57538 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE CLOROPHENE CLOROPHENE 84443 57539 MAPK12 6300 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR sorafenib SORAFENIB 20124951 84445 57540 GMNN 51053 DRUGGABLE GENOME HELENALIN HELENALIN 84446 57541 BAZ2B 29994 NA DNDI1417614 CHEMBL1567571 84448 57542 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME blocker 178100875 PICROTOXIN 84449 57543 EPO 2056 HORMONE ACTIVITY, CELL SURFACE, DRUGGABLE GENOME CHELATORS 1501748 84450 57544 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME SELUMETINIB SELUMETINIB 84451 57545 PTGS2 5743 DRUGGABLE GENOME, ENZYME ASPIRIN ASPIRIN 84453 57546 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE PALMATINE CHLORIDE HYDRATE PALMATINE CHLORIDE HYDRATE 84454 57547 NTRK1 4914 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE N-acylpiperidine ether derivative 4 84455 57548 APOBEC3A 200315 ENZYME, DRUGGABLE GENOME STILONIUM IODIDE STILONIUM IODIDE 84456 57549 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME DOCETAXEL DOCETAXEL 23200175,27876675,26125448,28492898 84458 57550 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE SU11274 19783361,15064724,19723643 84459 57551 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL856 PRIMIDONE 84460 57552 CSNK2A1 1457 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, TUMOR SUPPRESSOR ALSTERPAULLONE ALSTERPAULLONE 84461 57553 CCL20 6364 DRUGGABLE GENOME GSK3050002 GSK-3050002 84462 57554 IL3RA 3563 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE MB-102 RELMAPIRAZIN 84464 57555 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR HYDROCORTISONE HYDROCORTISONE 16759088 84467 57556 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR GNF-PF-67 CHEMBL578512 84469 57557 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME simvastatin SIMVASTATIN 24598718,19842935 84470 57558 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE IMATINIB IMATINIB 84472 57559 NOTCH3 4854 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME OMP-59R5 TAREXTUMAB 84475 57560 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor 328083504 84476 57561 KCND3 3752 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL2107762 NERISPIRDINE 84477 57562 IGF1R 3480 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TYROSINE KINASE antibody FIGITUMUMAB FIGITUMUMAB 84478 57563 KCNN4 3783 ION CHANNEL, DRUGGABLE GENOME ASP-0819 84481 57564 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME agonist CHEMBL1201656 INSULIN SUSP ISOPHANE PURIFIED PORK 84483 57565 FZD6 8323 CELL SURFACE, G PROTEIN COUPLED RECEPTOR, KINASE agonist 381745008 84484 57566 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-76 84486 57567 MAP4K4 9448 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ALSTERPAULLONE ALSTERPAULLONE 84487 57568 MAOA 4128 DRUGGABLE GENOME, ENZYME MOCLOBEMIDE MOCLOBEMIDE 84488 57569 CDKN2A 1029 CLINICALLY ACTIONABLE, DRUG RESISTANCE, KINASE, TUMOR SUPPRESSOR PANITUMUMAB PANITUMUMAB 23746666 84490 57570 SNW1 22938 NA TRANSFORMING GROWTH FACTOR 15149847 84491 57571 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 NEOSTIGMINE BROMIDE NEOSTIGMINE BROMIDE 22931300 84492 57572 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX DNDI1417165 CHEMBL1406948 84493 57573 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR 2,4-DINITRO-PHENYLAMINE CHEMBL354318 84494 57574 MPHOSPH8 54737 NA THIOLACTOMYCIN THIOLACTOMYCIN 84495 57575 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE TYRPHOSTIN AG-1478 TYRPHOSTIN AG-1478 21718029 84496 57576 ITGAL 3683 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME EFALIZUMAB EFALIZUMAB 84497 57577 CDK10 8558 DRUGGABLE GENOME, KINASE, TRANSCRIPTION FACTOR, ENZYME, SERINE THREONINE KINASE inhibitor CHEMBL445813 AT-7519 84498 57578 G6PD 2539 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE carmustine CARMUSTINE 539595 84499 57579 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE GSK2578215A CHEMBL2204495 22863203 84500 57580 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER pravastatin PRAVASTATIN 19667110 84501 57581 POLI 11201 DNA REPAIR THUNBERGINOL B THUNBERGINOL B 84502 57582 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE SUNITINIB SUNITINIB 29760553 84504 57583 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 84508 57584 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE VANDETANIB VANDETANIB 84509 57585 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NSC-8186 CHEMBL122355 84511 57586 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE PD-0166285 PD-0166285 84512 57587 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE SB-264865 CHEMBL1785002 84513 57588 SERPINE1 5054 DRUGGABLE GENOME, PROTEASE INHIBITOR EPIRUBICIN EPIRUBICIN 16444429 84514 57589 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME MURAGLITAZAR MURAGLITAZAR 84516 57590 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME inhibitor 404859044 84522 57591 IFNAR2 3455 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE Sifalimumab SIFALIMUMAB 84524 57592 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR CLOSANTEL CLOSANTEL 84526 57593 ALDH1A1 216 DRUGGABLE GENOME, ENZYME AM-630 CHEMBL181633 84527 57594 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE PCSK9 Adnectin 84528 57595 CYB5R3 1727 DRUGGABLE GENOME, ENZYME lidocaine and tetracaine 84529 57596 MAPT 4137 DRUGGABLE GENOME RALOXIFENE HYDROCHLORIDE RALOXIFENE HYDROCHLORIDE 84530 57597 TTR 7276 HORMONE ACTIVITY, DRUGGABLE GENOME Inotersen INOTERSEN 84531 57598 LPAR1 1902 G PROTEIN COUPLED RECEPTOR, CELL SURFACE, DRUGGABLE GENOME, KINASE agonist 135649710 84532 57599 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1094785 CARMOTEROL 84533 57600 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER PENTACHLOROPHENOL PENTACHLOROPHENOL 84535 57601 SMN1 6606 DRUGGABLE GENOME 2-(3',4'-METHYLENEDIOXYPHENYL)QUINOLINE CHEMBL502774 84539 57602 SCN9A 6335 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL698 TETRACAINE 84541 57603 ROCK2 9475 KINASE, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE GO-6976 GO-6976 84542 57604 SOCS3 9021 KINASE, CLINICALLY ACTIONABLE ANTISENSE OLIGONUCLEOTIDES 15939448 84544 57605 ITGB5 3693 CELL SURFACE, DRUGGABLE GENOME GLPG0187 GLPG-0187 84546 57606 APBA1 320 NA SLAZINIC ACID SLAZINIC ACID 84547 57607 CAMK1D 57118 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME 681640 CHEMBL379975 84548 57608 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME HARMINE HARMINE 84549 57609 RAB9A 9367 ENZYME, DRUGGABLE GENOME PHENELZINE PHENELZINE 84550 57610 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME INS-20 84551 57611 TUBA3C 7278 DRUGGABLE GENOME MAYTANSINOL MAYTANSINOL 563462 84553 57612 DDIT3 1649 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR 6-DIAZO-5-OXO-L-NORLEUCINE 6-DIAZO-5-OXO-L-NORLEUCINE 10377266 84554 57613 RACGAP1 29127 NA GNF-PF-1919 CHEMBL576409 84555 57614 PIK3C2G 5288 PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE inhibitor PKI-587 GEDATOLISIB 84557 57615 STK3 6788 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GW843682X GW843682X 84558 57616 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DNDI1417827 CHEMBL1363249 84559 57617 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME Ganetespib GANETESPIB 24398428,25077897 84560 57618 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 223365899 METHYLNALTREXONE 84561 57619 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR HEPARIN SODIUM 9101641 84562 57620 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME PMID28092474-Compound-33p 84565 57621 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565626 SCH-900776 84566 57622 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GW827396X GW827396X 84568 57623 SENP7 57337 ENZYME, DRUGGABLE GENOME, PROTEASE 6,4'-DIHYDROXYFLAVONE CHEMBL484663 84569 57624 EPHA2 1969 DRUGGABLE GENOME, CELL SURFACE, KINASE, TYROSINE KINASE, CLINICALLY ACTIONABLE ILORASERTIB ILORASERTIB 84570 57625 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200961 BROMPHENIRAMINE MALEATE 84571 57626 ALDH1A1 216 DRUGGABLE GENOME, ENZYME FUMARPROTOCETRARIC ACID FUMARPROTOCETRARIC ACID 84572 57627 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE PF-04691502 PF-04691502 84573 57628 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME MINOXIDIL MINOXIDIL 22931300 84574 57629 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME inhibitor 249565579 APITOLISIB 84575 57630 FGFR3 2261 CELL SURFACE, TYROSINE KINASE, KINASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 223366040 84576 57631 COL1A1 1277 CLINICALLY ACTIONABLE, DRUGGABLE GENOME COLLAGENASE COLLAGENASE CLOSTRIDIUM HISTOLYTICUM 84577 57632 IGF2 3481 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, HORMONE ACTIVITY, GROWTH FACTOR, DRUGGABLE GENOME FLUOXETINE FLUOXETINE 8265809 84578 57633 CCND2 894 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE 5-AZA-2-DEOXYCYTIDINE 12771922 84582 57634 NAT1 9 ENZYME, DRUGGABLE GENOME CHEMBL1345 GUANETHIDINE MONOSULFATE 84583 57635 ALDH1A1 216 DRUGGABLE GENOME, ENZYME PROPACHLOR PROPACHLOR 84584 57636 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE sunitinib SUNITINIB 19248971,12538485 84585 57637 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NITROXOLINE NITROXOLINE 84587 57638 CHRM3 1131 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 187051786 SOLIFENACIN 84588 57639 CACNB4 785 DRUGGABLE GENOME, ION CHANNEL VERAPAMIL VERAPAMIL 84589 57640 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist CHEMBL1200550 ANTAZOLINE PHOSPHATE 84590 57641 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565806 SILMITASERTIB 84591 57642 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE ALCLOFENAC ALCLOFENAC 84593 57643 EPHX2 2053 DRUGGABLE GENOME, ENZYME inhibitor 374883889 84596 57644 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME Dinaciclib DINACICLIB 26627013 84597 57645 NDUFV1 4723 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 84598 57646 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE METHYLTHIOURACIL METHYLTHIOURACIL 84599 57647 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Org-24461 CHEMBL59821 84600 57648 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE IMATINIB IMATINIB 84601 57649 RRM2 6241 DRUGGABLE GENOME, ENZYME Gemcitabine prodrug 84602 57650 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR CHENODIOL CHENODIOL 25162837,25247751,22018919,22014750,24387325,22126372,21459580,21309576,17963371 84603 57651 GMNN 51053 DRUGGABLE GENOME GNF-PF-4227 CHEMBL585654 84604 57652 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE TRAMETINIB TRAMETINIB 27922010 84605 57653 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TEN010 84606 57654 CDK4 1019 KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR Isoquinoline 1,3-dione derivative 1 84607 57655 RGS4 5999 DRUGGABLE GENOME AC-55649 CHEMBL425027 84608 57656 SIRT2 22933 TRANSCRIPTION FACTOR BINDING, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME, KINASE, TRANSCRIPTION FACTOR BDBM50363780 84611 57657 VDAC1 7416 NA OLESOXIME OLESOXIME 84612 57658 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Paliperidone PALIPERIDONE 84614 57659 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME GNF-PF-5134 CHEMBL602969 84617 57660 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME 6-CHLORONICOTINIC ACID 6-CHLORONICOTINIC ACID 84619 57661 THRB 7068 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist 135651405 TIRATRICOL 84621 57662 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME inhibitor 178102336 BOSUTINIB 84622 57663 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE IPI-145 DUVELISIB 84624 57664 GALR2 8811 G PROTEIN COUPLED RECEPTOR, KINASE, DRUGGABLE GENOME agonist 178100712 84625 57665 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ANETHOLTRITHION ANETHOLTRITHION 84626 57666 MAP4K2 5871 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE 681640 CHEMBL379975 84627 57667 GBA 2629 DRUGGABLE GENOME, ENZYME DOMIPHEN BROMIDE DOMIPHEN BROMIDE 84628 57668 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thiazole carboxamide derivative 3 84629 57669 ADRB1 153 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR catecholamines 17541557 84631 57670 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME BAS-8770949 CHEMBL476025 84633 57671 NOS1AP 9722 NA repaglinide REPAGLINIDE 84635 57672 GSTM1 2944 DRUGGABLE GENOME, ENZYME trimethoprim TRIMETHOPRIM 11191886 84636 57673 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 53801065 NIFEDIPINE 84637 57674 PDE4C 5143 DRUGGABLE GENOME, ENZYME ZINC584606052 84640 57675 SMN1 6606 DRUGGABLE GENOME BENZENE-1,2-DIAMINE CHEMBL70582 84641 57676 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME LIOTHYRONINE LIOTHYRONINE 22931300 84642 57677 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME CARBETAPENTANE CITRATE CARBETAPENTANE CITRATE 84644 57678 SLK 9748 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, KINASE GW843682X GW843682X 84645 57679 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY ALPHA-ADRENERGIC ANTAGONIST 6123933 84646 57680 CXCR2 3579 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE modulator CHEMBL191413 REPARIXIN 84647 57681 POLK 51426 DNA REPAIR, ENZYME SLAZINIC ACID SLAZINIC ACID 84648 57682 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE 6-OHDA 3084169 84649 57683 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR 5-FU FLUOROURACIL 18702703 84650 57684 TARDBP 23435 TUMOR SUPPRESSOR BENZOPHENONE-THIOSEMICARBAZONE BENZOPHENONE-THIOSEMICARBAZONE 84651 57685 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE 681640 CHEMBL379975 84652 57686 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR PHENYLMERCURIC ACETATE PHENYLMERCURIC ACETATE 84653 57687 PDE3A 5139 ENZYME, DRUGGABLE GENOME CILOSTAZOL CILOSTAZOL 84654 57688 FYN 2534 DRUGGABLE GENOME, CELL SURFACE, TYROSINE KINASE, KINASE, ENZYME ZM-447439 CHEMBL202721 84655 57689 CAMK1D 57118 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME SOTRASTAURIN SOTRASTAURIN 84656 57690 TBK1 29110 ENZYME, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME PMID26293650-Compound-35 84657 57691 TSPO 706 DRUGGABLE GENOME PMID27607364-Compound-65 84659 57692 PSMC3IP 29893 NUCLEAR HORMONE RECEPTOR inhibitor CARFILZOMIB CARFILZOMIB 84660 57693 TRPV4 59341 ION CHANNEL, CELL SURFACE, DRUGGABLE GENOME blocker 178101030 84661 57694 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER SANGUINARINE SULFATE SANGUINARINE SULFATE 84662 57695 MAPT 4137 DRUGGABLE GENOME BISSALICYL FUMARATE BISSALICYL FUMARATE 84664 57696 GJA1 2697 ION CHANNEL SELENIUM 16240671 84665 57697 ABCB11 8647 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE hmg coa reductase inhibitors 84666 57698 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE CIS-(Z)-FLUPENTHIXOL DIHYDROCHLORIDE CHEMBL1256995 84668 57699 F2 2147 PROTEASE, EXTERNAL SIDE OF PLASMA MEMBRANE, GROWTH FACTOR, DRUGGABLE GENOME, ENZYME ANTITHROMBIN 84669 57700 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-34 84670 57701 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR AZT ZIDOVUDINE 10433557 84672 57702 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE Sympathomimetics 84674 57703 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL PRAZEPAM PRAZEPAM 84675 57704 CES1 1066 DRUGGABLE GENOME, ENZYME SN-38 7-ETHYL-10-HYDROXYCAMPTOTHECIN 84676 57705 SLC5A1 6523 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 178101315 DAPAGLIFLOZIN 84677 57706 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME epirubicin EPIRUBICIN 84678 57707 S1PR5 53637 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 336446955 ASP-4058 84679 57708 HTT 3064 DRUGGABLE GENOME CMS-024-02 84681 57709 LPAR3 23566 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 178100857 84682 57710 FEN1 2237 DNA REPAIR, DRUGGABLE GENOME, ENZYME RO-410960 CHEMBL1256291 84683 57711 KCNT2 343450 ION CHANNEL, DRUGGABLE GENOME activator 135650716 84684 57712 DKK1 22943 GROWTH FACTOR, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor CHEMBL2109381 BHQ-880 84685 57713 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor 249565634 BGT-226 84686 57714 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Ranibizumab RANIBIZUMAB 84687 57715 BMP7 655 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, GROWTH FACTOR doxorubicin DOXORUBICIN 26590194 84688 57716 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 178102306 FORETINIB 84689 57717 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR TAMOXIFEN CITRATE TAMOXIFEN CITRATE 84690 57718 TF 7018 CELL SURFACE, DRUGGABLE GENOME EP-2167 84692 57719 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR 5,6,7,8,4'-PENTAHYDROXYFLAVONE CHEMBL234338 84693 57720 BRCA1 672 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, ENZYME, DRUGGABLE GENOME, DRUG RESISTANCE rucaparib RUCAPARIB 84695 57721 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE PONATINIB PONATINIB 25239608 84696 57722 GMNN 51053 DRUGGABLE GENOME 1,3-DIBENZYLTHIOUREA CHEMBL1388908 84697 57723 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE OSIMERTINIB OSIMERTINIB 29386539 84698 57724 BRCA2 675 CLINICALLY ACTIONABLE NIRAPARIB NIRAPARIB 84699 57725 CEL 1056 CELL SURFACE, DRUGGABLE GENOME, ENZYME Taurocholic Acid 84700 57726 TARDBP 23435 TUMOR SUPPRESSOR ARTEMISININ ARTEMISININ 84702 57727 SRC 6714 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME GW441756X GW441756X 84706 57728 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE inhibitor 310264740 ENSARTINIB 84707 57729 AHR 196 NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME NAPHTHALEN-1-YLAMINE CHEMBL57394 84709 57730 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE (R)-NIPHATENONE B CHEMBL1946014 22148427 84710 57731 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor DINACICLIB DINACICLIB 84711 57732 GJB6 10804 ION CHANNEL inhibitor 135652731 84712 57733 MAPK9 5601 KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PMID25991433-Compound-A9 84713 57734 SST 6750 HORMONE ACTIVITY, DRUGGABLE GENOME Cysteamine CYSTEAMINE 84714 57735 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CLOSTEBOL CLOSTEBOL 84715 57736 ALDH1A1 216 DRUGGABLE GENOME, ENZYME VANILLIN VANILLIN 84716 57737 LRRK2 120892 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE DNL201 84718 57738 CSF2 1437 DRUGGABLE GENOME, GROWTH FACTOR inhibitor CHEMBL2109433 OTILIMAB 84719 57739 BAZ2B 29994 NA inhibitor 252166514 84720 57740 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CD20-CAR-T Cells 84721 57741 CASP6 839 DRUGGABLE GENOME, PROTEASE, ENZYME METHYLDOPA METHYLDOPA 84722 57742 HDAC9 9734 TRANSCRIPTION FACTOR BINDING, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TACEDINALINE TACEDINALINE 18692397 84725 57743 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME RG-1530 RG-1530 84726 57744 PSMC3 5702 NA inhibitor CHEMBL3545432 IXAZOMIB CITRATE 84728 57745 SCN1A 6323 DRUGGABLE GENOME, ION CHANNEL blocker CHEMBL1769 PROPOXYCAINE HYDROCHLORIDE 84729 57746 TNFRSF17 608 CLINICALLY ACTIONABLE, DRUGGABLE GENOME C-CAR088 84730 57747 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR GSK126 27135738 84731 57748 SLC39A14 23516 TRANSPORTER nortriptyline NORTRIPTYLINE 20970119 84732 57749 FGFR2 2263 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, CELL SURFACE NINTEDANIB NINTEDANIB 84735 57750 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME diazepam DIAZEPAM 17638512,11470993 84736 57751 CPB2 1361 DRUGGABLE GENOME, ENZYME, PROTEASE SAR-104772 84737 57752 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TCMDC-123598 CHEMBL547269 84739 57753 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CLEMASTINE CLEMASTINE 84742 57754 CXCL8 3576 DRUGGABLE GENOME CEFTRIAXONE CEFTRIAXONE 8011012 84743 57755 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME BENZYDAMINE BENZYDAMINE 84744 57756 PTPRC 5788 CLINICALLY ACTIONABLE, TUMOR SUPPRESSOR, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME, PROTEIN PHOSPHATASE, KINASE infliximab INFLIXIMAB 20309874,23007924 84745 57757 FGFR4 2264 CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, ENZYME, DRUG RESISTANCE, TYROSINE KINASE inhibitor CHEMBL274654 ORANTINIB 84746 57758 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE VATALANIB VATALANIB 84748 57759 BAZ2B 29994 NA HAEMATOXYLIN HAEMATOXYLIN 84750 57760 AQP4 361 ION CHANNEL, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME ACETAZOLAMIDE ACETAZOLAMIDE 18572411 84751 57761 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-71033 CHEMBL116548 84755 57762 SCN7A 6332 ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1201486 QUINIDINE POLYGALACTURONATE 84756 57763 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE VE-822 BERZOSERTIB 84757 57764 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER PERVILLEINE D PERVILLEINE D 11754602 84758 57765 JUN 3725 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR BINDING IRISOLIDONE IRISOLIDONE 17996449 84759 57766 MGLL 11343 DRUGGABLE GENOME, ENZYME Pyrazole derivative 85 84760 57767 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 84761 57768 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME NCI-17383 CHEMBL188641 84762 57769 MAPK10 5602 KINASE, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE PMID25991433-Compound-F2 84763 57770 MAP2K5 5607 KINASE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME, DRUGGABLE GENOME inhibitor PD 0325901 84765 57771 PRKD3 23683 KINASE, ENZYME, SERINE THREONINE KINASE, DRUGGABLE GENOME inhibitor CHEMBL3545332 CEP-2563 84766 57772 IL6R 3570 EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME tocilizumab TOCILIZUMAB 24978393,27958380 84767 57773 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME GSK-269962A GSK-269962A 84768 57774 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME MADOLIN U MADOLIN U 84769 57775 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME ABT-263 NAVITOCLAX 27659046 84770 57776 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE docetaxel DOCETAXEL 21151855,23188068,18294295 84773 57777 BRD4 23476 CLINICALLY ACTIONABLE, KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME DOCETAXEL DOCETAXEL 16542442 84774 57778 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE CLOFIBRATE CLOFIBRATE 8557642 84775 57779 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE NSC-747265 CHEMBL595682 84776 57780 INSR 3643 CLINICALLY ACTIONABLE, TYROSINE KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, ENZYME, DRUGGABLE GENOME Mitoglitazone MITOGLITAZONE 84778 57781 NR3C2 4306 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR antagonist 178100449 84779 57782 BCL2 596 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE RIBAVIRIN RIBAVIRIN 15902734,16190549 84780 57783 ADK 132 DRUGGABLE GENOME, ENZYME, KINASE abacavir ABACAVIR 24625462 84781 57784 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor 178102572 84785 57785 PSMC2 5701 PROTEASE, TRANSCRIPTION FACTOR inhibitor BORTEZOMIB BORTEZOMIB 84787 57786 OPCML 4978 DRUGGABLE GENOME methylphenidate METHYLPHENIDATE 29382897 84788 57787 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ETHACRIDINE LACTATE ETHACRIDINE LACTATE 84790 57788 TOP2B 7155 DRUGGABLE GENOME, ENZYME XR-5000 84793 57789 ALDH1A1 216 DRUGGABLE GENOME, ENZYME METHYSERGIDE METHYSERGIDE 84794 57790 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Pralidoxime Chloride 84795 57791 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103816 MITOXANTRONE 84796 57792 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME NMS-1286937 NMS-1286937 84797 57793 GMNN 51053 DRUGGABLE GENOME FEBANTEL FEBANTEL 84798 57794 PCSK9 255738 DRUGGABLE GENOME, ENZYME, CELL SURFACE, PROTEASE REGN727 ALIROCUMAB 84800 57795 EPCAM 4072 CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME ING-1 ING-1 84801 57796 PIK3R3 8503 KINASE, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor CHEMBL3544999 SAMOTOLISIB 84802 57797 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL QUAZEPAM QUAZEPAM 84803 57798 KLF5 688 TRANSCRIPTION FACTOR COMPLEX, TRANSCRIPTION FACTOR, DRUGGABLE GENOME TCMDC-125567 CHEMBL530049 84804 57799 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR ZIRAM ZIRAM 84805 57800 XRCC4 7518 KINASE Platinum compounds 28796378 84807 57801 MYC 4609 TRANSCRIPTION FACTOR, CLINICALLY ACTIONABLE LIF 1906157 84808 57802 CRTC1 23373 CLINICALLY ACTIONABLE PKI-587 GEDATOLISIB 84809 57803 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor SNS-314 SNS-314 84810 57804 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Recombinant human Erbb3 fragment therapeutic tumor vaccine 84811 57805 ADAMTS4 9507 ENZYME, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE US9206139, 4 84812 57806 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR INAMRINONE INAMRINONE 84813 57807 DDC 1644 ENZYME, DRUGGABLE GENOME IPX066 84815 57808 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE 1,7-O-DIACETYLMETHYLGEOPYXIN A CHEMBL1889303 84816 57809 CA1 759 DRUGGABLE GENOME, ENZYME MEDRONIC ACID MEDRONIC ACID 24813742 84817 57810 CREBBP 1387 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, ENZYME, TRANSCRIPTION FACTOR, DRUG RESISTANCE, DRUGGABLE GENOME OXOGLAUCINE OXOGLAUCINE 84821 57811 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 178102626 84822 57812 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CINACALCET HYDROCHLORIDE CINACALCET HYDROCHLORIDE 84823 57813 CACNA1A 773 ION CHANNEL, DRUGGABLE GENOME celecoxib CELECOXIB 22336956 84824 57814 GNAQ 2776 CLINICALLY ACTIONABLE, DRUG RESISTANCE PD-0325901 PD-0325901 24141786 84825 57815 ALOX15B 247 DRUGGABLE GENOME, ENZYME PYRITHIONE ZINC PYRITHIONE ZINC 84826 57816 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME MADOLIN T MADOLIN T 84829 57817 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL BROMAZEPAM BROMAZEPAM 84834 57818 PAK4 10298 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME JNJ-7706621 JNJ-7706621 84836 57819 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME SFLT-01 84837 57820 CD3E 916 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE inhibitor CHEMBL2108811 VISILIZUMAB 84838 57821 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE KENPAULLONE KENPAULLONE 84841 57822 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR MTX METHOTREXATE 12210990 84842 57823 FFAR4 338557 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651503 84843 57824 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE agonist 178100889 84845 57825 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Radiotherapy 25589492,26846818,24130052 84846 57826 ANXA1 301 CELL SURFACE, DRUGGABLE GENOME LOTEPREDNOL ETABONATE 84849 57827 POLK 51426 DNA REPAIR, ENZYME 3,4,5-TRIHYDROXY-BENZOIC ACID PHENETHYL ESTER CHEMBL151146 84850 57828 GCG 2641 DRUGGABLE GENOME, HORMONE ACTIVITY PENICILLAMINE PENICILLAMINE 11485378 84851 57829 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID29473428-Compound-41 84852 57830 MAOB 4129 DRUGGABLE GENOME, ENZYME Heteroaryl-cyclopropylamine derivative 3 84853 57831 SNCA 6622 DRUGGABLE GENOME, TRANSPORTER AG-1879 CHEMBL406845 84855 57832 CDH1 999 CLINICALLY ACTIONABLE, DRUGGABLE GENOME Lapatinib LAPATINIB 26487584 84858 57833 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX NSC-105827 CHEMBL171699 84859 57834 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TRIFLOXYSTROBIN TRIFLOXYSTROBIN 84860 57835 DMD 1756 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Eteplirsen ETEPLIRSEN 84862 57836 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME activator 135651544 84863 57837 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR MELPHALAN MELPHALAN 84864 57838 BAZ2B 29994 NA DNDI1417080 CHEMBL1498652 84865 57839 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR ISOSPAGLUMIC ACID ISOSPAGLUMIC ACID 84866 57840 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL450 METHARBITAL 84867 57841 APP 351 DRUGGABLE GENOME, PROTEASE INHIBITOR, CELL SURFACE CHEMBL1743004 CRENEZUMAB 84868 57842 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 LEUPROLIDE LEUPROLIDE 22931300 84869 57843 TRPM2 7226 ION CHANNEL, DRUGGABLE GENOME blocker 135649885 84870 57844 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME ADINAZOLAM ADINAZOLAM 84871 57845 PIK3CD 5293 KINASE, DRUGGABLE GENOME, ENZYME, PHOSPHATIDYLINOSITOL 3 KINASE, CLINICALLY ACTIONABLE inhibitor 249565692 84875 57846 RECQL 5965 DRUGGABLE GENOME, DNA REPAIR, ENZYME GW7074 CHEMBL72365 84876 57847 MUC16 94025 DRUGGABLE GENOME IFN 8217487 84877 57848 PARP3 10039 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE, DNA REPAIR inhibitor CHEMBL1173055 RUCAPARIB 84880 57849 LIF 3976 GROWTH FACTOR, DRUGGABLE GENOME 5-AZA-2'-DEOXYCYTIDINE 14647063 84881 57850 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME CAMPTOTHECIN CAMPTOTHECIN 16962673 84883 57851 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR PYRONIN Y PYRONIN Y 84886 57852 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR ACTEIN ACTEIN 84887 57853 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PIFITHRIN-ALPHA CHEMBL198759 84889 57854 LDLR 3949 ENZYME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME TGF 1464611 84890 57855 SMO 6608 DRUG RESISTANCE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, G PROTEIN COUPLED RECEPTOR Isoflavone derivative 8 84894 57856 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE TRASTUZUMAB DERUXTECAN 31047804,31047803 84895 57857 MAPT 4137 DRUGGABLE GENOME SULFASALAZINE SULFASALAZINE 84896 57858 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME SU-6656 CHEMBL605003 84900 57859 POLK 51426 DNA REPAIR, ENZYME ANTHRALIN ANTHRALIN 84901 57860 MAPK1 5594 SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, TRANSCRIPTION FACTOR GNF-PF-3756 CHEMBL597035 84902 57861 AR 367 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, DRUG RESISTANCE CHLOROXINE CHLOROXINE 84903 57862 FAS 355 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME THROMBIN THROMBIN 16271051 84904 57863 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102313 NERATINIB 84905 57864 CRMP1 1400 NA METHIMAZOLE METHIMAZOLE 11694350 84907 57865 NPY1R 4886 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135649992 84909 57866 BAZ2B 29994 NA AURINTRICARBOXYLIC ACID AURINTRICARBOXYLIC ACID 84910 57867 MARK4 57787 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor HESPERADIN HESPERADIN 19035792 84911 57868 HRAS 3265 CLINICALLY ACTIONABLE, DRUG RESISTANCE, TUMOR SUPPRESSOR, DRUGGABLE GENOME, ENZYME SCH772984 27222538 84912 57869 CYBB 1536 ION CHANNEL, TRANSPORTER, DRUGGABLE GENOME, ENZYME inhibitor 363894226 84914 57870 TUBB3 10381 DRUGGABLE GENOME inhibitor CHEMBL289351 FOSBRETABULIN DISODIUM 84915 57871 CYP2E1 1571 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 cyclophosphamide CYCLOPHOSPHAMIDE 22188361 84916 57872 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER ZIRAM ZIRAM 84917 57873 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 RIMCAZOLE RIMCAZOLE 84918 57874 P2RY2 5029 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, ION CHANNEL agonist 135651593 84919 57875 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE GSK-299115A GSK-299115A 84920 57876 HSD11B1 3290 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 3-EPICOROSOLIC ACID METHYL ESTER CHEMBL604538 20100662 84922 57877 OXTR 5021 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135651080 RELCOVAPTAN 84923 57878 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 385612184 84924 57879 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME inhibitor CHEMBL574737 UCN-01 84928 57880 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178102302 CANERTINIB 84929 57881 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE inhibitor CHEMBL1921976 ORTERONEL 84930 57882 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 315661275 OLMUTINIB 84933 57883 MMP3 4314 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE, ENZYME inhibitor 178101905 MARIMASTAT 84934 57884 GLI1 2735 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR Isoflavone derivative 4 84935 57885 CYP2B6 1555 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME mephenytoin MEPHENYTOIN 17638512,11470993 84936 57886 ITGAV 3685 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE antagonist CHEMBL1743032 INTETUMUMAB 84937 57887 KDM4A 9682 DRUGGABLE GENOME, ENZYME DNDI1417076 CHEMBL1526167 84938 57888 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR CONICASTEROL D CONICASTEROL D 21428459 84942 57889 NT5C2 22978 ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE cytarabine CYTARABINE 84944 57890 CAPN2 824 PROTEASE, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE Epoxysuccinate derivative 9 84945 57891 CHRM2 1129 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135650782 OXOTREMORINE 84946 57892 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR ICI 182780 12021046 84947 57893 CDK7 1022 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102566 84948 57894 BAZ2B 29994 NA SJ000111875 CHEMBL590949 84949 57895 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE Topotecan TOPOTECAN 21216929 84950 57896 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME blocker CHEMBL1200728 GUANIDINE HYDROCHLORIDE 84951 57897 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME APOMORPHINE HYDROCHLORIDE HEMIHYDRATE APOMORPHINE HYDROCHLORIDE HEMIHYDRATE 84952 57898 AURKA 6790 SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME, DRUG RESISTANCE, DRUGGABLE GENOME inhibitor 252166565 84953 57899 MET 4233 KINASE, TYROSINE KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, DRUG RESISTANCE BMS-754807 BMS-754807 19778024 84955 57900 MAPT 4137 DRUGGABLE GENOME TCMDC-125602 CHEMBL580183 84957 57901 RAPGEF3 10411 ENZYME ESTROPIPATE ESTROPIPATE 84959 57902 GMNN 51053 DRUGGABLE GENOME CHLORQUINALDOL CHLORQUINALDOL 84960 57903 PTGDR 5729 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 53801020 84963 57904 GABRE 2564 DRUGGABLE GENOME, ION CHANNEL LORAZEPAM LORAZEPAM 84965 57905 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR NAFTOPIDIL NAFTOPIDIL 84966 57906 H19 283120 CLINICALLY ACTIONABLE HORMONES 8785513 84968 57907 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE RUCAPARIB RUCAPARIB 84970 57908 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor GEFITINIBIRESSA GEFITINIB 84971 57909 ABCG1 9619 TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME fluorouracil FLUOROURACIL 26352872 84972 57910 IL1B 3553 KINASE, DRUGGABLE GENOME omeprazole OMEPRAZOLE 16815316,21054464,14638340 84973 57911 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CEFOPERAZONE CEFOPERAZONE 22931300 84974 57912 NR1H4 9971 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, KINASE, TRANSCRIPTION FACTOR PMID29649907-Compound-3 84975 57913 PARP1 142 ENZYME, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE, DRUG RESISTANCE inhibitor VELIPARIB VELIPARIB 84976 57914 KCNQ3 3786 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME activator 135650896 EZOGABINE 84977 57915 ERBB3 2065 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE, DRUG RESISTANCE PATRITUMAB DERUXTECAN 84978 57916 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 PENTOSALEN PENTOSALEN 84979 57917 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME METHANESULFONIC ACID METHYL ESTER METHANESULFONIC ACID METHYL ESTER 22455312 84980 57918 XIAP 331 ENZYME, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, PROTEASE INHIBITOR, TUMOR SUPPRESSOR UCN-01 UCN-01 12738674,15255949 84981 57919 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR TRIAMCINOLONE TRIAMCINOLONE 84984 57920 IKBKE 9641 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 249565742 84985 57921 GABRB1 2560 ION CHANNEL, DRUGGABLE GENOME HALAZEPAM HALAZEPAM 84986 57922 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist CHEMBL2103876 MAPRACORAT 84988 57923 CACNB3 784 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ION CHANNEL modulator CHEMBL940 GABAPENTIN 84990 57924 DPP7 29952 PROTEASE, ENZYME, DRUGGABLE GENOME US8470836, 6 84991 57925 ATAD5 79915 NA GNF-PF-1872 CHEMBL600103 84993 57926 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX MMV666022 CHEMBL599100 84994 57927 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR BUTORPHANOL BUTORPHANOL 84995 57928 TFPI 7035 CELL SURFACE, DRUGGABLE GENOME, PROTEASE INHIBITOR Tifacogin TIFACOGIN 84996 57929 RARA 5914 TRANSCRIPTION FACTOR COMPLEX, NUCLEAR HORMONE RECEPTOR, CELL SURFACE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME agonist 178103534 TAZAROTENE 84998 57930 VCAM1 7412 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME CYCLOSPORINE CYCLOSPORINE 7694584 85000 57931 IL6 3569 DRUG RESISTANCE, DRUGGABLE GENOME, GROWTH FACTOR Olokizumab OLOKIZUMAB 24641941 85002 57932 NPC1 4864 TRANSPORTER, DRUGGABLE GENOME DNDI1417085 CHEMBL1522984 85003 57933 PIK3R1 5295 CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE GSK2126458 OMIPALISIB 85004 57934 GMNN 51053 DRUGGABLE GENOME AG-494 CHEMBL56731 85005 57935 HSP90AB1 3326 TRANSCRIPTION FACTOR, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TUMOR SUPPRESSOR DIPYRIDAMOLE DIPYRIDAMOLE 85007 57936 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME N-ACETYLGLUCOSAMINE THIAZOLINE CHEMBL257158 20822912 85008 57937 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR agonist 178103640 BETAMETHASONE 85009 57938 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist 135650749 85010 57939 TDP1 55775 DRUGGABLE GENOME, ENZYME, DNA REPAIR CARMINE CARMINE 85011 57940 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME nilotinib NILOTINIB 24322003 85012 57941 HTR1D 3352 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist 135650903 RISPERIDONE 85013 57942 AGTR1 185 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR S-474474 85015 57943 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE mycophenolic acid 24220207 85017 57944 ALDH1A1 216 DRUGGABLE GENOME, ENZYME NSC-92207 CHEMBL139935 85018 57945 ABCC2 1244 TRANSPORTER, DRUGGABLE GENOME, ABC TRANSPORTER, CELL SURFACE simvastatin SIMVASTATIN 22186618 85019 57946 PSENEN 55851 DRUGGABLE GENOME inhibitor CHEMBL520733 SEMAGACESTAT 85020 57947 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME Pyrimidine derivative 32 85022 57948 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Amoxapine AMOXAPINE 85025 57949 B2M 567 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE THYROGLOBULIN THYROGLOBULIN 9609129 85026 57950 GABRP 2568 DRUGGABLE GENOME, ION CHANNEL CHEMBL2068724 ACAMPROSATE CALCIUM 85027 57951 CYP3A5 1577 ENZYME, CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE sildenafil SILDENAFIL 18695978 85029 57952 GMNN 51053 DRUGGABLE GENOME DNDI1417457 CHEMBL1530911 85030 57953 DSE 29940 ENZYME prednisolone PREDNISOLONE 85032 57954 ESR1 2099 DRUG RESISTANCE, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, KINASE, TRANSCRIPTION FACTOR Dienestrol DIENESTROL 85033 57955 PIM1 5292 TRANSCRIPTION FACTOR BINDING, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor CHEMBL3545423 AZD-1208 85035 57956 TOP2B 7155 DRUGGABLE GENOME, ENZYME Sabarubicin SABARUBICIN 85036 57957 EGLN1 54583 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME PYRIDINE-2,4-DICARBOXYLIC ACID CHEMBL316034 26022078,23234607 85037 57958 PRKCD 5580 ENZYME, DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, TRANSCRIPTION FACTOR DOVITINIB DOVITINIB 85038 57959 MUC2 4583 DRUGGABLE GENOME GPI-0100 15837210 85039 57960 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME colchicine COLCHICINE 25645282 85040 57961 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME LINSIDOMINE LINSIDOMINE 85043 57962 GMNN 51053 DRUGGABLE GENOME COLCHICEINE COLCHICEINE 85044 57963 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE PONATINIB PONATINIB 24407160 85045 57964 TOP1 7150 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE N-METHYLCALOTHRIXIN B N-METHYLCALOTHRIXIN B 19203291 85048 57965 NME2 4831 KINASE PROGESTERONE PROGESTERONE 15674352 85049 57966 APC 324 CLINICALLY ACTIONABLE iCRT-3 21393571 85050 57967 CACNA2D3 55799 ION CHANNEL, DRUGGABLE GENOME modulator CHEMBL940 GABAPENTIN 85051 57968 MPHOSPH8 54737 NA GW7647 GW7647 85053 57969 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Flumatinib FLUMATINIB 85055 57970 PIN1 5300 ENZYME, KINASE, TUMOR SUPPRESSOR, DRUGGABLE GENOME S-(P-AZIDOPHENACYL)GLUTATHIONE CHEMBL1256813 85056 57971 GRIN1 2902 ION CHANNEL, DRUGGABLE GENOME, CELL SURFACE agonist 178100907 85057 57972 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 JNJ-16259685 CHEMBL174588 85062 57973 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor CHEMBL1614710 OSI-930 85063 57974 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor 252166729 AZD-8186 85066 57975 DPP4 1803 PROTEASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME ARI-2243 85068 57976 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE inhibitor 315661216 PLX8394 85069 57977 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME ROSIGLITAZONE ROSIGLITAZONE 85070 57978 CD63 967 CELL SURFACE, DRUGGABLE GENOME, KINASE NSAIDS 15608437 85071 57979 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE SORAFENIB SORAFENIB 19671763,17699867,19461405,20970876 85072 57980 SIK2 23235 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME inhibitor 178102305 DASATINIB 85073 57981 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME DIMERCAPROL DIMERCAPROL 85075 57982 RORC 6097 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR AZACITIDINE AZACITIDINE 85076 57983 EPHX1 2052 ENZYME, DRUGGABLE GENOME carbamazepine CARBAMAZEPINE 15692831,22188362,26314341,25495409,19620853 85078 57984 IDO1 3620 ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME Pyridine derivative 1 85080 57985 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 178102555 JNJ-7706621 85082 57986 THPO 7066 GROWTH FACTOR, HORMONE ACTIVITY, DRUGGABLE GENOME L-741626 CHEMBL445102 85083 57987 AKT2 208 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, TRANSPORTER, TRANSCRIPTION FACTOR, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR GDC-0068 IPATASERTIB 85084 57988 TNF 7124 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE mycophenolate mofetil 18444945 85085 57989 SOCS1 8651 CLINICALLY ACTIONABLE, KINASE IL-2 ALDESLEUKIN 12928391 85087 57990 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX MITONAFIDE MITONAFIDE 85088 57991 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME AZD-1080 AZD-1080 85091 57992 DROSHA 29102 NA prednisone PREDNISONE 24614921 85092 57993 SLC6A9 6536 TRANSPORTER, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE Organon-2 85093 57994 TOP2B 7155 DRUGGABLE GENOME, ENZYME Amsacrine AMSACRINE 85094 57995 RIPK1 8737 KINASE, SERINE THREONINE KINASE, DRUGGABLE GENOME, ENZYME inhibitor 381118842 85095 57996 CXCL8 3576 DRUGGABLE GENOME DEOXYSPERGUALIN 9507569 85096 57997 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 pazopanib PAZOPANIB 22341567 85098 57998 SPHK1 8877 ENZYME, KINASE, LIPID KINASE, DRUGGABLE GENOME VPC45129 CHEMBL554130 19632123 85100 57999 GMNN 51053 DRUGGABLE GENOME BERGAPTOL BERGAPTOL 85102 58000 SLC22A3 6581 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, TRANSPORTER inhibitor 252827483 DISPROCYNIUM24 85104 58001 FFAR4 338557 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135651436 85105 58002 FAAH 2166 ENZYME, DRUGGABLE GENOME Azole derivative 2 85106 58003 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 CID 663143 CHEMBL1342336 85107 58004 PDGFRA 5156 TYROSINE KINASE, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUG RESISTANCE AXITINIB AXITINIB 85109 58005 HSP90B1 7184 DRUGGABLE GENOME inhibitor 315661287 SEMAPIMOD 85110 58006 RRM2 6241 DRUGGABLE GENOME, ENZYME LOR-2040 85111 58007 OPRM1 4988 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, KINASE buprenorphine BUPRENORPHINE 30549211 85113 58008 ACHE 43 ENZYME, CELL SURFACE, DRUGGABLE GENOME Isoflurophate ISOFLUROPHATE 85114 58009 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME TRASTUZUMAB TRASTUZUMAB 16452223 85116 58010 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR CDT-fenofibrate 85117 58011 GMNN 51053 DRUGGABLE GENOME CLANFENUR CLANFENUR 85118 58012 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR raloxifene RALOXIFENE 10692979,12608943,18443790,19020788,15739035,12162507 85121 58013 NR3C1 2908 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR, ENZYME, TRANSCRIPTION FACTOR antagonist 178100448 85122 58014 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME SJ000180366 CHEMBL609036 85123 58015 FGFR1 2260 KINASE, DRUG RESISTANCE, TYROSINE KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 249565645 MK-2461 85124 58016 CD2 914 CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME IL-2 ALDESLEUKIN 7519476 85125 58017 PAH 5053 DRUGGABLE GENOME, ENZYME Phenylalanine hydroxylase 85126 58018 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SB-222200 SB-222200 85129 58019 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE AC480 AC-480 21576284 85132 58020 FLT1 2321 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE PD-0166285 PD-0166285 85133 58021 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME TAE-684 TAE-684 85134 58022 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME SIMVASTATIN SIMVASTATIN 85135 58023 TRPA1 8989 DRUGGABLE GENOME, ION CHANNEL activator 135651250 85136 58024 SMN1 6606 DRUGGABLE GENOME NABUMETONE NABUMETONE 85137 58025 GNA11 2767 CLINICALLY ACTIONABLE Trametinib TRAMETINIB 22733540 85138 58026 LTBR 4055 DRUGGABLE GENOME HCBE-11 HCBE-11 85139 58027 POLI 11201 DNA REPAIR GW7647 GW7647 85143 58028 TARDBP 23435 TUMOR SUPPRESSOR 2-PHENYL-1H-INDOLE 2-PHENYL-1H-INDOLE 85145 58029 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME KAEMPFERIDE KAEMPFERIDE 25190466 85148 58030 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME XANTHYLETIN XANTHYLETIN 85150 58031 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE THIOGUANINE THIOGUANINE 85151 58032 ACVRL1 94 KINASE, SERINE THREONINE KINASE, CELL SURFACE, DRUGGABLE GENOME, ENZYME inhibitor 252166689 85152 58033 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR Alitretinoin ALITRETINOIN 85154 58034 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor PAZOPANIB PAZOPANIB 85155 58035 ATAD5 79915 NA DNDI1416955 CHEMBL1327172 85157 58036 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE inhibitor 178101619 ERLOTINIB 85158 58037 ABCG2 9429 TRANSPORTER, ABC TRANSPORTER, DRUGGABLE GENOME methotrexate METHOTREXATE 20386493,18237272,27217051,29791011,25778468,18256692,21317831 85159 58038 CYP2C9 1559 DRUGGABLE GENOME, ENZYME, CYTOCHROME P450 GENTAMICIN GENTAMICIN 22931300 85162 58039 IDH1 3417 ENZYME, CLINICALLY ACTIONABLE HEXACHLOROPHENE HEXACHLOROPHENE 85163 58040 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME inhibitor 249565698 85164 58041 HTT 3064 DRUGGABLE GENOME NSC-102042 CHEMBL273103 85165 58042 PLCG1 5335 ENZYME, KINASE, PHOSPHOLIPASE, DRUGGABLE GENOME aspirin ASPIRIN 26398624 85167 58043 NOTCH1 4851 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSPORTER, CELL SURFACE JQ1 28151717 85168 58044 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE imatinib IMATINIB 85169 58045 SLC6A4 6532 TRANSPORTER, DRUGGABLE GENOME inhibitor 135651367 ZOTEPINE 85170 58046 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE inhibitor 223366064 SARACATINIB 85171 58047 DMD 1756 CELL SURFACE, TRANSPORTER, DRUGGABLE GENOME Golodirsen GOLODIRSEN 85173 58048 MAPT 4137 DRUGGABLE GENOME HAEMATOXYLIN HAEMATOXYLIN 85174 58049 CP 1356 DRUGGABLE GENOME, ENZYME FREUNDS ADJUVANT 7741265 85175 58050 NDUFAF4 29078 NA inhibitor CHEMBL3545320 ME-344 85177 58051 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME CID 2093195 CHEMBL411085 85178 58052 XBP1 7494 TRANSCRIPTION FACTOR, ENZYME, CLINICALLY ACTIONABLE, DRUGGABLE GENOME GNF-PF-1859 CHEMBL1520837 85179 58053 SIGMAR1 10280 DRUGGABLE GENOME, ION CHANNEL Benzamide derivative 9 85180 58054 PIK3CA 5290 PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, KINASE, ENZYME, SERINE THREONINE KINASE, DRUG RESISTANCE inhibitor CHEMBL3545379 SERABELISIB 85181 58055 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 187051804 RESMINOSTAT 85182 58056 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME IPRONIAZID IPRONIAZID 22931300 85183 58057 ODC1 4953 DRUGGABLE GENOME, ENZYME Difluoromethylornithine 85184 58058 VEGFA 7422 CLINICALLY ACTIONABLE, GROWTH FACTOR, CELL SURFACE, DRUGGABLE GENOME Carbamide derivative 16 85187 58059 TP53 7157 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX, TUMOR SUPPRESSOR, DRUGGABLE GENOME, KINASE, DRUG RESISTANCE, TRANSPORTER CID 739615 CHEMBL260560 85189 58060 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR ATOVAQUONE ATOVAQUONE 85191 58061 MAPT 4137 DRUGGABLE GENOME DIMETHYL GAMBOGATE DIMETHYL GAMBOGATE 85193 58062 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CYCLOHEXANONE OXIME CYCLOHEXANONE OXIME 85197 58063 RB1 5925 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE, KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR, TRANSCRIPTION FACTOR COMPLEX Everolimus EVEROLIMUS 28151717 85198 58064 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE BENZAMIL BENZAMIL 85199 58065 ADRB2 154 KINASE, G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE agonist CHEMBL1201153 ISOETHARINE MESYLATE 85200 58066 ABCB1 5243 CLINICALLY ACTIONABLE, TRANSPORTER, DRUGGABLE GENOME, ENZYME, CELL SURFACE, DRUG RESISTANCE, ABC TRANSPORTER dicloxacillin DICLOXACILLIN 15778422,18576903 85204 58067 HCAR3 8843 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102426 85205 58068 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME agonist CHEMBL408 TROGLITAZONE 85207 58069 MS4A1 931 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, DRUGGABLE GENOME IBRITUMOMAB IBRITUMOMAB TIUXETAN 85208 58070 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE 4-PHENYLAMINO-[1,2]NAPHTHOQUINONE CHEMBL299853 85209 58071 HDAC1 3065 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ROMIDEPSIN ROMIDEPSIN 85211 58072 POLK 51426 DNA REPAIR, ENZYME BAICALEIN BAICALEIN 85213 58073 PRSS3 5646 ENZYME, PROTEASE, DRUGGABLE GENOME BORTEZOMIB BORTEZOMIB 20875739 85215 58074 MAPK3 5595 TRANSCRIPTION FACTOR, KINASE, DRUGGABLE GENOME, SERINE THREONINE KINASE, ENZYME GAMBOGIC AMIDE GAMBOGIC AMIDE 17911251 85216 58075 THBS1 7057 EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME antibody CVX-045 85217 58076 AURKB 9212 ENZYME, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, HISTONE MODIFICATION, DRUGGABLE GENOME, KINASE inhibitor PF-03814735 PF-03814735 85220 58077 MTOR 2475 DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, ENZYME TCMDC-124166 CHEMBL528712 85222 58078 POLK 51426 DNA REPAIR, ENZYME PURPURIN PURPURIN 85224 58079 NDUFB11 54539 ENZYME inhibitor CHEMBL1703 METFORMIN HYDROCHLORIDE 85225 58080 PDE4A 5141 DRUGGABLE GENOME, ENZYME SOTB07 85227 58081 FDFT1 2222 DRUGGABLE GENOME, ENZYME inhibitor 249565677 SQ109 85228 58082 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR CIS/TRANS-ISOEUGENOL CIS/TRANS-ISOEUGENOL 85229 58083 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE DOVITINIB DOVITINIB 85230 58084 RACGAP1 29127 NA ACRIFLAVINE CHLORIDE ACRIFLAVINE 85231 58085 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME PURPUROGALLIN PURPUROGALLIN 85232 58086 GHR 2690 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, CELL SURFACE Somatropin recombinant 85233 58087 NFKB1 4790 KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME HYDROQUINONE HYDROQUINONE 85234 58088 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE sorafenib SORAFENIB 28362716 85235 58089 LNPEP 4012 DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, TRANSPORTER, PROTEASE inhibitor CHEMBL2103847 TOSEDOSTAT 85236 58090 CACNA2D1 781 DRUGGABLE GENOME, ION CHANNEL AMLODIPINE AMLODIPINE 85237 58091 SMN2 6607 DRUGGABLE GENOME DEHYDROVARIABILIN DEHYDROVARIABILIN 85238 58092 CD3D 915 DRUGGABLE GENOME, EXTERNAL SIDE OF PLASMA MEMBRANE, KINASE VISILIZUMAB VISILIZUMAB 85239 58093 APEX1 328 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, DRUGGABLE GENOME ELLAGIC ACID ELLAGIC ACID 85240 58094 GSK3B 2932 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR inhibitor 354702282 85241 58095 NOS2 4843 DRUGGABLE GENOME, ENZYME STEROID HORMONE 7532809 85242 58096 F2RL3 9002 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 381744950 85243 58097 MAPK8 5599 DRUGGABLE GENOME, SERINE THREONINE KINASE, KINASE, ENZYME, TRANSCRIPTION FACTOR PMID25991433-Compound-G2 85244 58098 IL10 3586 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, GROWTH FACTOR SHO-SAIKO-TO 9185758 85245 58099 ATR 545 SERINE THREONINE KINASE, DNA REPAIR, CLINICALLY ACTIONABLE, ENZYME, KINASE, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE OLAPARIB OLAPARIB 85247 58100 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR PG102 85249 58101 LPL 4023 DRUGGABLE GENOME, LIPASE, PHOSPHOLIPASE, CELL SURFACE ISOTRETINOIN ISOTRETINOIN 2931603 85252 58102 PDK1 5163 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME Thieno[3,2-c]pyridine-7-carboxamide derivative 1 85253 58103 PDGFRB 5159 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE, CELL SURFACE inhibitor TELATINIB TELATINIB 85256 58104 ENPP2 5168 ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BINDING inhibitor 336446947 ZIRITAXESTAT 85258 58105 MAPT 4137 DRUGGABLE GENOME 3-METHYLCHOLANTHRENE 3-METHYLCHOLANTHRENE 85259 58106 TNFRSF4 7293 DRUGGABLE GENOME, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE TRemelimumab + MEDI0562 85260 58107 CSNK1G2 1455 KINASE, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME CENISERTIB CENISERTIB 85261 58108 CD40 958 CLINICALLY ACTIONABLE, CELL SURFACE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR FLUDARABINE FLUDARABINE 9450802 85262 58109 ARAF 369 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, ENZYME SORAFENIB SORAFENIB 26619011,24569458 85263 58110 MARCHF8 220972 ENZYME Celtura 85264 58111 PPARG 5468 CLINICALLY ACTIONABLE, NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME (-)-GRACILIOETHER C CHEMBL2178583 22934537 85265 58112 IRAK1 3654 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME, TRANSCRIPTION FACTOR SNS-314 SNS-314 85266 58113 KDM4A 9682 DRUGGABLE GENOME, ENZYME NSC-8186 CHEMBL122355 85269 58114 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME DNDI1417221 CHEMBL1459280 85271 58115 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR 7-BENZYLOXYCOUMARIN 7-BENZYLOXYCOUMARIN 85272 58116 CMKLR1 1240 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 135651571 85273 58117 CSF3R 1441 CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME RUXOLITINIB RUXOLITINIB 25180155,24081659 85276 58118 CMKLR1 1240 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 354702254 85278 58119 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 doxorubicin DOXORUBICIN 9187528 85281 58120 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor 223366209 CEP-32496 85282 58121 POLB 5423 DNA REPAIR, DRUGGABLE GENOME ZAFIRLUKAST ZAFIRLUKAST 85283 58122 TNIK 23043 ENZYME, DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE CEP-1347 CEP-1347 24044867 85284 58123 HSD17B10 3028 DRUGGABLE GENOME, SHORT CHAIN DEHYDROGENASE REDUCTASE, ENZYME CARBARIL CARBARIL 85285 58124 HSPA4 3308 NA HYDRALAZINE HYDRALAZINE 12047041 85287 58125 THBS2 7058 DRUGGABLE GENOME ADRENOCORTICOTROPIC HORMONE 8698834 85288 58126 PTPN12 5782 PROTEIN PHOSPHATASE, DRUGGABLE GENOME, KINASE GNF-PF-231 CHEMBL601167 85289 58127 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE lamivudine LAMIVUDINE 85290 58128 BAZ2B 29994 NA CB7969312 CHEMBL599255 85291 58129 EZH2 2146 CLINICALLY ACTIONABLE, ENZYME, METHYL TRANSFERASE, NUCLEAR HORMONE RECEPTOR, TRANSCRIPTION FACTOR PMID26882240-Compound-1 85292 58130 PTGS2 5743 DRUGGABLE GENOME, ENZYME ETHYL EICOSAPENTAENOIC ACID 85293 58131 MAOB 4129 DRUGGABLE GENOME, ENZYME PMID25399762-Compound-Table1-C14 85294 58132 BCL2L1 598 CLINICALLY ACTIONABLE, DRUGGABLE GENOME PMID27744724-Compound-27 85295 58133 TYK2 7297 KINASE, DRUGGABLE GENOME, TYROSINE KINASE, CLINICALLY ACTIONABLE, ENZYME inhibitor 178102304 TOFACITINIB 85296 58134 BAZ2B 29994 NA TCMDC-125556 CHEMBL587092 85298 58135 TPP1 1200 PROTEASE, ENZYME, DRUGGABLE GENOME Cerliponase Alfa 85299 58136 TLR7 51284 DRUGGABLE GENOME IMO-3100 85300 58137 SLC2A4 6517 DRUGGABLE GENOME, TRANSPORTER, EXTERNAL SIDE OF PLASMA MEMBRANE OMAPATRILAT OMAPATRILAT 15776120 85301 58138 FDPS 2224 DRUGGABLE GENOME, ENZYME, CLINICALLY ACTIONABLE ZOLEDRONATE ZOLEDRONIC ACID 85303 58139 POLH 5429 CLINICALLY ACTIONABLE, ENZYME, DNA REPAIR TYRPHOSTIN 25 TYRPHOSTIN 25 85305 58140 CYP3A4 1576 ENZYME, DRUGGABLE GENOME, CYTOCHROME P450 SIMVASTATIN SIMVASTATIN 22931300 85306 58141 HDAC6 10013 ENZYME, TRANSCRIPTION FACTOR, TRANSCRIPTION FACTOR BINDING, DRUGGABLE GENOME PMID29671355-Compound-65a 85307 58142 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 310264762 85308 58143 JAK1 3716 CLINICALLY ACTIONABLE, DRUG RESISTANCE, DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME PMID27774824-Compound-Figure3Example18 85309 58144 ERBB2 2064 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, DRUG RESISTANCE, TYROSINE KINASE Lapatinib LAPATINIB 85310 58145 SLCO1B1 10599 TRANSPORTER, DRUGGABLE GENOME gemtuzumab ozogamicin 22584460 85313 58146 HPGD 3248 DRUGGABLE GENOME, ENZYME, SHORT CHAIN DEHYDROGENASE REDUCTASE 3-METHOXYCATECHOL 3-METHOXYCATECHOL 85315 58147 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TANESPIMYCIN TANESPIMYCIN 85316 58148 TERT 7015 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, RNA DIRECTED DNA POLYMERASE, DRUG RESISTANCE 2,7-BIS[3-(PROPYLAMINO)PROPIONAMIDO]ANTHRAQUINONE CHEMBL481160 18571928 85317 58149 TNKS2 80351 DRUGGABLE GENOME, ENZYME inhibitor 404859120 85318 58150 PSMB1 5689 PROTEASE, DRUGGABLE GENOME, ENZYME OPROZOMIB OPROZOMIB 85320 58151 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102266 EDOTREOTIDE 85322 58152 ADAMTS4 9507 ENZYME, DRUGGABLE GENOME, NEUTRAL ZINC METALLOPEPTIDASE, PROTEASE US9206139, 5 85324 58153 KIT 3815 CLINICALLY ACTIONABLE, KINASE, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, TYROSINE KINASE, DRUG RESISTANCE, EXTERNAL SIDE OF PLASMA MEMBRANE inhibitor AMUVATINIB AMUVATINIB 85328 58154 SSTR2 6752 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME agonist 178102267 85329 58155 LCK 3932 KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TYROSINE KINASE TAMATINIB R-406 85330 58156 NCSTN 23385 DRUGGABLE GENOME, CLINICALLY ACTIONABLE LY-411575 CHEMBL392068 23181502,19443228 85331 58157 HIF1A 3091 TRANSPORTER, TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, TRANSCRIPTION FACTOR COMPLEX, CLINICALLY ACTIONABLE RESVERATROL RESVERATROL 85332 58158 PPARA 5465 TRANSCRIPTION FACTOR, ENZYME, DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR phenprocoumon PHENPROCOUMON 25461249 85333 58159 FCGR3A 2214 EXTERNAL SIDE OF PLASMA MEMBRANE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE HEPARIN HEPARIN 18492254 85334 58160 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME inhibitor SORAFENIB SORAFENIB 85335 58161 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR antagonist CHEMBL1718 NALOXONE HYDROCHLORIDE 85337 58162 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME SJ000111093 CHEMBL585045 85338 58163 ABCC3 8714 DRUG RESISTANCE, DRUGGABLE GENOME, TRANSPORTER, ABC TRANSPORTER, CLINICALLY ACTIONABLE CEFAMANDOLE CEFAMANDOLE 22166395 85339 58164 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE Prinomastat PRINOMASTAT 85340 58165 ROCK1 6093 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE inhibitor 249565717 85342 58166 ESR2 2100 DRUGGABLE GENOME, TRANSCRIPTION FACTOR, NUCLEAR HORMONE RECEPTOR TAMOXIFEN TAMOXIFEN 20659801 85344 58167 PLA2G2A 5320 PHOSPHOLIPASE, DRUGGABLE GENOME, ENZYME HEPARIN HEPARIN 7883954 85345 58168 NRAS 4893 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME AZD9291 OSIMERTINIB 25870145 85348 58169 ATAD5 79915 NA SJ000044417 CHEMBL609438 85349 58170 MAP2K2 5605 KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, TYROSINE KINASE, ENZYME MEK162 BINIMETINIB 85350 58171 CP 1356 DRUGGABLE GENOME, ENZYME PROTOPORPHYRIN PROTOPORPHYRIN 6214811 85351 58172 ERN1 2081 DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, KINASE US8614253, 32-4 85352 58173 LAG3 3902 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, EXTERNAL SIDE OF PLASMA MEMBRANE Anti-LAG3 85353 58174 BCHE 590 DRUGGABLE GENOME, ENZYME OPIOIDS 8961166 85354 58175 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME ciprofloxacin CIPROFLOXACIN 27469576 85355 58176 CDK9 1025 SERINE THREONINE KINASE, TUMOR SUPPRESSOR, DNA REPAIR, KINASE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR, ENZYME inhibitor 178102568 85358 58177 CASP3 836 DRUGGABLE GENOME, PROTEASE, ENZYME TELEOCIDIN B TELEOCIDIN B 21696964 85359 58178 KRAS 3845 CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME CH5132799 PA-799 22159814,21558396 85361 58179 PTEN 5728 PTEN FAMILY, ENZYME, PROTEIN PHOSPHATASE, DRUG RESISTANCE, CLINICALLY ACTIONABLE, KINASE BEZ235 DACTOLISIB 27974663,26206338,28446642,26232337,22662154 85363 58180 LIMK1 3984 KINASE, DRUGGABLE GENOME, ENZYME, SERINE THREONINE KINASE DASATINIB DASATINIB 85364 58181 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE STIBOGLUCONATE STIBOGLUCONATE 85365 58182 HSP90AA1 3320 CLINICALLY ACTIONABLE, DRUGGABLE GENOME, TRANSCRIPTION FACTOR NSC-402083 CHEMBL1546228 85366 58183 AKT1 207 SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSPORTER, TRANSCRIPTION FACTOR, DRUG RESISTANCE inhibitor 249565861 85367 58184 CASP7 840 PROTEASE, DRUGGABLE GENOME, ENZYME 3-HYDROXYANTHRANILIC ACID CHEMBL445304 85368 58185 POLI 11201 DNA REPAIR AG-494 CHEMBL56731 85369 58186 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME GSK-269962A GSK-269962A 85370 58187 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR TRIPHENYLSTANNANOL TRIPHENYLSTANNANOL 85371 58188 NFE2L2 4780 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR TECTOQUINONE TECTOQUINONE 85373 58189 ARSA 410 DRUGGABLE GENOME, ENZYME DNQX DNQX 85374 58190 MMP2 4313 NEUTRAL ZINC METALLOPEPTIDASE, ENZYME, DRUGGABLE GENOME, PROTEASE Metastat INCYCLINIDE 85375 58191 RAF1 5894 DRUGGABLE GENOME, KINASE, ENZYME, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE carboplatin CARBOPLATIN 21636554 85376 58192 PLK1 5347 TRANSCRIPTION FACTOR, KINASE, TUMOR SUPPRESSOR, SERINE THREONINE KINASE, ENZYME, DRUGGABLE GENOME TAK-960 TAK-960 85377 58193 CD163 9332 DRUGGABLE GENOME, KINASE, EXTERNAL SIDE OF PLASMA MEMBRANE FLUTICASONE PROPIONATE 9712057 85378 58194 CDK2 1017 DNA REPAIR, TRANSCRIPTION FACTOR COMPLEX, SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME HGF 11909963 85379 58195 DYRK1A 1859 DRUGGABLE GENOME, KINASE, ENZYME, TYROSINE KINASE, SERINE THREONINE KINASE PMID28766366-Compound-Scheme27LeucettamineB 85380 58196 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME IMETIT DIHYDROBROMIDE IMETIT DIHYDROBROMIDE 85382 58197 IMPDH2 3615 DRUGGABLE GENOME, ENZYME inhibitor CHEMBL1200955 MYCOPHENOLATE MOFETIL HYDROCHLORIDE 85383 58198 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor 178103421 ETOPOSIDE 85385 58199 SMAD3 4088 DRUGGABLE GENOME, KINASE, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR COMPLEX METHYLTHIONINIUM CHLORIDE METHYLTHIONINIUM CHLORIDE 85388 58200 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE Afatinib AFATINIB 85391 58201 RXRB 6257 DRUGGABLE GENOME, NUCLEAR HORMONE RECEPTOR agonist CHEMBL75133 IRX-4204 85392 58202 RGS4 5999 DRUGGABLE GENOME LANSOPRAZOLE LANSOPRAZOLE 85393 58203 GATA3 2625 CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR cytarabine CYTARABINE 24141364 85395 58204 YES1 7525 DRUGGABLE GENOME, KINASE, TYROSINE KINASE, ENZYME, CLINICALLY ACTIONABLE VEMURAFENIB VEMURAFENIB 85397 58205 ADRA1A 148 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135650746 NS-49 85398 58206 CBX1 10951 NA GNF-PF-372 CHEMBL580155 85400 58207 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME ARACHIDONOYL DOPAMINE ARACHIDONOYL DOPAMINE 85401 58208 CYP17A1 1586 DRUGGABLE GENOME, CYTOCHROME P450, ENZYME, CLINICALLY ACTIONABLE Seviteronel SEVITERONEL 85402 58209 NQO1 1728 ENZYME, DRUGGABLE GENOME, CLINICALLY ACTIONABLE cisplatin CISPLATIN 12370763 85403 58210 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME TROLOX TROLOX 85405 58211 BDNF 627 DRUGGABLE GENOME, GROWTH FACTOR Ergot alkaloids 25096645 85406 58212 KDM4A 9682 DRUGGABLE GENOME, ENZYME QUINOXALINE-2-CARBOXYLIC ACID CHEMBL151797 85408 58213 CDK14 5218 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, TUMOR SUPPRESSOR, ENZYME inhibitor CHEMBL488436 AZD-5438 85409 58214 GMNN 51053 DRUGGABLE GENOME 2-HYDROXYESTRADIOL CHEMBL467987 85410 58215 DPYSL2 1808 NA Lacosamide ERLOSAMIDE 85411 58216 POLB 5423 DNA REPAIR, DRUGGABLE GENOME D-DOPA CHEMBL211670 85412 58217 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE GNF-PF-2301 CHEMBL578061 85413 58218 PPARD 5467 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR BEZAFIBRATE BEZAFIBRATE 85415 58219 VDR 7421 NUCLEAR HORMONE RECEPTOR, DRUGGABLE GENOME, TRANSCRIPTION FACTOR CAFFEINE CAFFEINE 11684540 85416 58220 EHMT2 10919 METHYL TRANSFERASE, ENZYME, DRUGGABLE GENOME PROTOAPIGENONE PROTOAPIGENONE 85418 58221 NTRK3 4916 CLINICALLY ACTIONABLE, ENZYME, TYROSINE KINASE, KINASE, DRUG RESISTANCE, DRUGGABLE GENOME LAROTRECTINIB LAROTRECTINIB 29880614,29623306,30204247,31905241,29606586,29466156,30624546,29920189 85419 58222 PTPN11 5781 DRUGGABLE GENOME, KINASE, PROTEIN PHOSPHATASE, ENZYME, CLINICALLY ACTIONABLE PD98059 17942397 85420 58223 BRAF 673 KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, DRUG RESISTANCE, ENZYME, DRUGGABLE GENOME ASN003 85421 58224 GMNN 51053 DRUGGABLE GENOME PIRIQUALONE PIRIQUALONE 85422 58225 BAZ2B 29994 NA FLUPIRTINE MALEATE FLUPIRTINE MALEATE 85423 58226 OPRK1 4986 DRUGGABLE GENOME, G PROTEIN COUPLED RECEPTOR agonist 135652142 85425 58227 GABRB3 2562 ION CHANNEL, DRUGGABLE GENOME positive modulator CHEMBL285674 ESTAZOLAM 85426 58228 CYP2D6 1565 CYTOCHROME P450, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME Escitalopram ESCITALOPRAM 85427 58229 HRH1 3269 G PROTEIN COUPLED RECEPTOR, DRUGGABLE GENOME antagonist 178100784 85429 58230 CCND1 595 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, TRANSCRIPTION FACTOR, KINASE, DRUG RESISTANCE PROTEIN SYNTHESIS INHIBITOR 9094091 85430 58231 TOP2A 7153 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME epirubicin EPIRUBICIN 85431 58232 PIK3CB 5291 CLINICALLY ACTIONABLE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, KINASE, G PROTEIN COUPLED RECEPTOR inhibitor CHEMBL3544966 GSK-1059615 85432 58233 ATM 472 CLINICALLY ACTIONABLE, SERINE THREONINE KINASE, KINASE, ENZYME, DRUGGABLE GENOME, PHOSPHATIDYLINOSITOL 3 KINASE, TUMOR SUPPRESSOR, DRUG RESISTANCE BMN673 85433 58234 MAP4K5 11183 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, ENZYME ENTRECTINIB ENTRECTINIB 85436 58235 EGFR 1956 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, CELL SURFACE, TYROSINE KINASE, DRUG RESISTANCE antibody 387065587 JNJ-61186372 85437 58236 TARDBP 23435 TUMOR SUPPRESSOR ANDROSTERONE ANDROSTERONE 85438 58237 GABRG2 2566 DRUGGABLE GENOME, ION CHANNEL positive modulator CHEMBL451 CHLORDIAZEPOXIDE 85442 58238 JAK2 3717 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, DRUGGABLE GENOME, DRUG RESISTANCE, ENZYME inhibitor 315661260 AC-430 85443 58239 POR 5447 ENZYME, DRUGGABLE GENOME sunitinib SUNITINIB 28117434 85444 58240 CTDSP1 58190 DRUGGABLE GENOME, PROTEIN PHOSPHATASE ISOPROPAMIDE IODIDE ISOPROPAMIDE IODIDE 85445 58241 AKR1C1 1645 DRUGGABLE GENOME, ENZYME PROGESTERONE PROGESTERONE 6584862,12604236,3463506,2547059,6950669,3859707,179793,6288675 85447 58242 SCN11A 11280 DRUGGABLE GENOME, ION CHANNEL, KINASE blocker CHEMBL2107771 RALFINAMIDE 85448 58243 CDK1 983 SERINE THREONINE KINASE, KINASE, DNA REPAIR, TRANSCRIPTION FACTOR, DRUGGABLE GENOME, ENZYME PHA-767491 CHEMBL225519 85449 58244 TAOK1 57551 SERINE THREONINE KINASE, KINASE, DRUGGABLE GENOME, DNA REPAIR, ENZYME PALBOCICLIB PALBOCICLIB 85450 58245 CSF1R 1436 CLINICALLY ACTIONABLE, KINASE, TYROSINE KINASE, CELL SURFACE, DRUGGABLE GENOME BAY-613606 CHEMBL541400 85452 58246 BIRC5 332 DRUG RESISTANCE, TUMOR SUPPRESSOR, PROTEASE INHIBITOR, DRUGGABLE GENOME ISIS 23722 85453 58247 CDK8 1024 DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME, KINASE, SERINE THREONINE KINASE, TRANSCRIPTION FACTOR, TUMOR SUPPRESSOR TCMDC-125758 CHEMBL546797 85455 58248 GRIN2B 2904 CELL SURFACE, ION CHANNEL, DRUGGABLE GENOME H-Gly-PMe-Glu-OH 85456 58249 PIK3C3 5289 KINASE, PHOSPHATIDYLINOSITOL 3 KINASE, DRUGGABLE GENOME, CLINICALLY ACTIONABLE, ENZYME inhibitor BGJ398 INFIGRATINIB 85457 58250 ABL1 25 ENZYME, TYROSINE KINASE, TUMOR SUPPRESSOR, KINASE, CLINICALLY ACTIONABLE, DRUGGABLE GENOME, DRUG RESISTANCE Azaindole derivative 2 85458 58251 CACNA1D 776 ION CHANNEL, CLINICALLY ACTIONABLE, DRUGGABLE GENOME inhibitor 135651166 85459 58252 PRKCA 5578 DRUGGABLE GENOME, KINASE, SERINE THREONINE KINASE, CLINICALLY ACTIONABLE, ENZYME RESVERATROL RESVERATROL 21880495 85460 58253 P4HB 5034 THIOREDOXIN, DRUGGABLE GENOME, ENZYME, EXTERNAL SIDE OF PLASMA MEMBRANE GNF-PF-2976 CHEMBL579956