approved DB00001 Lepirudin biotech P00734 Prothrombin approved DB00002 Cetuximab biotech P00533 Epidermal growth factor receptor approved DB00002 Cetuximab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved DB00002 Cetuximab biotech P02745 Complement C1q subcomponent subunit A approved DB00002 Cetuximab biotech P02746 Complement C1q subcomponent subunit B approved DB00002 Cetuximab biotech P02747 Complement C1q subcomponent subunit C approved DB00002 Cetuximab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved DB00002 Cetuximab biotech P09871 Complement C1s subcomponent approved DB00002 Cetuximab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00004 Denileukin diftitox biotech P01589 Interleukin-2 receptor subunit alpha approved|investigational DB00004 Denileukin diftitox biotech P14784 Interleukin-2 receptor subunit beta approved|investigational DB00005 Etanercept biotech P01375 Tumor necrosis factor approved|investigational DB00005 Etanercept biotech P20333 Tumor necrosis factor receptor superfamily member 1B approved|investigational DB00005 Etanercept biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational DB00005 Etanercept biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00005 Etanercept biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00005 Etanercept biotech P09871 Complement C1s subcomponent approved|investigational DB00005 Etanercept biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00005 Etanercept biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00005 Etanercept biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00006 Bivalirudin small molecule P00734 Prothrombin approved|investigational DB00008 Peginterferon alfa-2a biotech P48551 Interferon alpha/beta receptor 2 approved|investigational DB00008 Peginterferon alfa-2a biotech P17181 Interferon alpha/beta receptor 1 approved DB00009 Alteplase biotech P00747 Plasminogen approved DB00009 Alteplase biotech P02671 Fibrinogen alpha chain approved DB00009 Alteplase biotech Q03405 Urokinase plasminogen activator surface receptor approved DB00009 Alteplase biotech P05121 Plasminogen activator inhibitor 1 approved|withdrawn DB00010 Sermorelin biotech Q02643 Growth hormone-releasing hormone receptor approved|investigational DB00011 Interferon alfa-n1 biotech P48551 Interferon alpha/beta receptor 2 approved|investigational DB00011 Interferon alfa-n1 biotech P17181 Interferon alpha/beta receptor 1 approved|investigational DB00012 Darbepoetin alfa biotech P19235 Erythropoietin receptor approved|investigational|withdrawn DB00013 Urokinase biotech P00747 Plasminogen approved|investigational|withdrawn DB00013 Urokinase biotech Q03405 Urokinase plasminogen activator surface receptor approved|investigational|withdrawn DB00013 Urokinase biotech P00749 Urokinase-type plasminogen activator approved|investigational|withdrawn DB00013 Urokinase biotech P00750 Tissue-type plasminogen activator approved|investigational|withdrawn DB00013 Urokinase biotech P05121 Plasminogen activator inhibitor 1 approved|investigational|withdrawn DB00013 Urokinase biotech P05120 Plasminogen activator inhibitor 2 approved|investigational|withdrawn DB00013 Urokinase biotech P05154 Plasma serine protease inhibitor approved|investigational|withdrawn DB00013 Urokinase biotech P98164 Low-density lipoprotein receptor-related protein 2 approved|investigational|withdrawn DB00013 Urokinase biotech Q9Y5Y6 Suppressor of tumorigenicity 14 protein approved|investigational|withdrawn DB00013 Urokinase biotech P14543 Nidogen-1 approved DB00014 Goserelin small molecule P22888 Lutropin-choriogonadotropic hormone receptor approved|investigational DB00015 Reteplase biotech P00747 Plasminogen approved|investigational DB00015 Reteplase biotech P02671 Fibrinogen alpha chain approved|investigational DB00015 Reteplase biotech Q03405 Urokinase plasminogen activator surface receptor approved|investigational DB00015 Reteplase biotech P05121 Plasminogen activator inhibitor 1 approved DB00016 Erythropoietin biotech P19235 Erythropoietin receptor approved|investigational DB00017 Salmon Calcitonin biotech P30988 Calcitonin receptor approved DB00019 Pegfilgrastim biotech Q99062 Granulocyte colony-stimulating factor receptor approved|investigational DB00020 Sargramostim biotech P32927 Cytokine receptor common subunit beta approved|investigational DB00020 Sargramostim biotech P34741 Syndecan-2 approved|investigational DB00020 Sargramostim biotech P13727 Bone marrow proteoglycan approved DB00022 Peginterferon alfa-2b biotech P17181 Interferon alpha/beta receptor 1 approved DB00022 Peginterferon alfa-2b biotech P48551 Interferon alpha/beta receptor 2 approved|vet_approved DB00024 Thyrotropin Alfa biotech P16473 Thyrotropin receptor approved|investigational DB00025 Antihemophilic factor, human recombinant biotech P00742 Coagulation factor X approved|investigational DB00025 Antihemophilic factor, human recombinant biotech P04275 von Willebrand factor approved|investigational DB00025 Antihemophilic factor, human recombinant biotech O14832 Phytanoyl-CoA dioxygenase, peroxisomal approved|investigational DB00025 Antihemophilic factor, human recombinant biotech P07307 Asialoglycoprotein receptor 2 approved|investigational DB00025 Antihemophilic factor, human recombinant biotech P11021 Endoplasmic reticulum chaperone BiP {ECO:0000305} approved|investigational DB00025 Antihemophilic factor, human recombinant biotech P27797 Calreticulin approved|investigational DB00025 Antihemophilic factor, human recombinant biotech P27824 Calnexin approved|investigational DB00025 Antihemophilic factor, human recombinant biotech P49257 Protein ERGIC-53 approved|investigational DB00025 Antihemophilic factor, human recombinant biotech Q07954 Prolow-density lipoprotein receptor-related protein 1 approved|investigational DB00025 Antihemophilic factor, human recombinant biotech Q8NI22 Multiple coagulation factor deficiency protein 2 approved DB00026 Anakinra biotech P14778 Interleukin-1 receptor type 1 approved DB00029 Anistreplase biotech P00747 Plasminogen approved DB00029 Anistreplase biotech P02671 Fibrinogen alpha chain approved DB00029 Anistreplase biotech Q03405 Urokinase plasminogen activator surface receptor approved DB00029 Anistreplase biotech P05121 Plasminogen activator inhibitor 1 approved|investigational DB00030 Insulin Human biotech P06213 Insulin receptor approved|investigational DB00030 Insulin Human biotech P08069 Insulin-like growth factor 1 receptor approved|investigational DB00030 Insulin Human biotech P06400 Retinoblastoma-associated protein approved|investigational DB00030 Insulin Human biotech P07339 Cathepsin D approved|investigational DB00030 Insulin Human biotech P14735 Insulin-degrading enzyme approved|investigational DB00030 Insulin Human biotech P16519 Neuroendocrine convertase 2 approved|investigational DB00030 Insulin Human biotech P16870 Carboxypeptidase E approved|investigational DB00030 Insulin Human biotech P29120 Neuroendocrine convertase 1 approved|investigational DB00030 Insulin Human biotech P48745 Protein NOV homolog approved|investigational DB00030 Insulin Human biotech P98164 Low-density lipoprotein receptor-related protein 2 approved|investigational DB00030 Insulin Human biotech Q16270 Insulin-like growth factor-binding protein 7 approved|investigational DB00030 Insulin Human biotech Q96C24 Synaptotagmin-like protein 4 approved DB00031 Tenecteplase biotech P00747 Plasminogen approved DB00031 Tenecteplase biotech P02671 Fibrinogen alpha chain approved DB00031 Tenecteplase biotech Q03405 Urokinase plasminogen activator surface receptor approved DB00031 Tenecteplase biotech P05121 Plasminogen activator inhibitor 1 approved DB00031 Tenecteplase biotech P05120 Plasminogen activator inhibitor 2 approved DB00031 Tenecteplase biotech P05452 Tetranectin approved DB00031 Tenecteplase biotech P05787 Keratin, type II cytoskeletal 8 approved DB00031 Tenecteplase biotech P07355 Annexin A2 approved DB00031 Tenecteplase biotech P27797 Calreticulin approved DB00031 Tenecteplase biotech P27824 Calnexin approved DB00031 Tenecteplase biotech Q07954 Prolow-density lipoprotein receptor-related protein 1 approved DB00032 Menotropins biotech P23945 Follicle-stimulating hormone receptor approved DB00032 Menotropins biotech P22888 Lutropin-choriogonadotropic hormone receptor approved|investigational DB00034 Interferon Alfa-2a, Recombinant biotech P17181 Interferon alpha/beta receptor 1 approved|investigational DB00034 Interferon Alfa-2a, Recombinant biotech P48551 Interferon alpha/beta receptor 2 approved DB00036 Coagulation factor VIIa Recombinant Human biotech P00742 Coagulation factor X approved DB00036 Coagulation factor VIIa Recombinant Human biotech P05981 Serine protease hepsin approved DB00036 Coagulation factor VIIa Recombinant Human biotech P10646 Tissue factor pathway inhibitor approved DB00036 Coagulation factor VIIa Recombinant Human biotech P38435 Vitamin K-dependent gamma-carboxylase approved DB00036 Coagulation factor VIIa Recombinant Human biotech P08709 Coagulation factor VII approved DB00036 Coagulation factor VIIa Recombinant Human biotech P13726 Tissue factor approved|investigational DB00038 Oprelvekin biotech Q14626 Interleukin-11 receptor subunit alpha approved DB00039 Palifermin biotech P21802 Fibroblast growth factor receptor 2 approved DB00039 Palifermin biotech O14786 Neuropilin-1 approved DB00039 Palifermin biotech P11362 Fibroblast growth factor receptor 1 approved DB00039 Palifermin biotech P22455 Fibroblast growth factor receptor 4 approved DB00039 Palifermin biotech P22607 Fibroblast growth factor receptor 3 approved DB00039 Palifermin biotech P98160 Basement membrane-specific heparan sulfate proteoglycan core protein approved DB00040 Glucagon recombinant biotech P47871 Glucagon receptor approved DB00040 Glucagon recombinant biotech O95838 Glucagon-like peptide 2 receptor approved DB00041 Aldesleukin biotech P14784 Interleukin-2 receptor subunit beta approved DB00041 Aldesleukin biotech P01589 Interleukin-2 receptor subunit alpha approved|investigational DB00042 Botulinum Toxin Type B biotech P63027 Vesicle-associated membrane protein 2 approved|investigational DB00042 Botulinum Toxin Type B biotech P23763 Vesicle-associated membrane protein 1 approved|investigational DB00042 Botulinum Toxin Type B biotech Q8N9I0 Synaptotagmin-2 {ECO:0000305} approved|investigational DB00043 Omalizumab biotech P12319 High affinity immunoglobulin epsilon receptor subunit alpha approved DB00044 Lutropin alfa biotech P22888 Lutropin-choriogonadotropic hormone receptor approved DB00046 Insulin Lispro biotech P06213 Insulin receptor approved DB00046 Insulin Lispro biotech P08069 Insulin-like growth factor 1 receptor approved DB00047 Insulin Glargine biotech P06213 Insulin receptor approved DB00047 Insulin Glargine biotech P08069 Insulin-like growth factor 1 receptor approved|investigational DB00048 Collagenase clostridium histolyticum biotech P02452 Collagen alpha-1(I) chain approved|investigational DB00048 Collagenase clostridium histolyticum biotech P02458 Collagen alpha-1(II) chain {ECO:0000305} approved|investigational DB00048 Collagenase clostridium histolyticum biotech P02461 Collagen alpha-1(III) chain approved|investigational DB00048 Collagenase clostridium histolyticum biotech P08123 Collagen alpha-2(I) chain approved|investigational DB00050 Cetrorelix small molecule P22888 Lutropin-choriogonadotropic hormone receptor approved DB00051 Adalimumab biotech P01375 Tumor necrosis factor approved DB00051 Adalimumab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved DB00051 Adalimumab biotech P02745 Complement C1q subcomponent subunit A approved DB00051 Adalimumab biotech P02746 Complement C1q subcomponent subunit B approved DB00051 Adalimumab biotech P02747 Complement C1q subcomponent subunit C approved DB00051 Adalimumab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved DB00051 Adalimumab biotech P09871 Complement C1s subcomponent approved DB00051 Adalimumab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00052 Somatotropin biotech P10912 Growth hormone receptor approved|investigational DB00052 Somatotropin biotech P16471 Prolactin receptor approved DB00054 Abciximab biotech P05106 Integrin beta-3 approved DB00054 Abciximab biotech P08514 Integrin alpha-IIb approved DB00054 Abciximab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved DB00054 Abciximab biotech P02745 Complement C1q subcomponent subunit A approved DB00054 Abciximab biotech P02746 Complement C1q subcomponent subunit B approved DB00054 Abciximab biotech P02747 Complement C1q subcomponent subunit C approved DB00054 Abciximab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved DB00054 Abciximab biotech P09871 Complement C1s subcomponent approved DB00054 Abciximab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved DB00054 Abciximab biotech P04004 Vitronectin approved|investigational|withdrawn DB00055 Drotrecogin alfa biotech P00451 Coagulation factor VIII approved|investigational|withdrawn DB00055 Drotrecogin alfa biotech P12259 Coagulation factor V approved|investigational|withdrawn DB00055 Drotrecogin alfa biotech P05121 Plasminogen activator inhibitor 1 approved|investigational|withdrawn DB00055 Drotrecogin alfa biotech P07204 Thrombomodulin approved|investigational|withdrawn DB00055 Drotrecogin alfa biotech P07225 Vitamin K-dependent protein S approved|investigational|withdrawn DB00055 Drotrecogin alfa biotech P00450 Ceruloplasmin approved|investigational|withdrawn DB00055 Drotrecogin alfa biotech P00734 Prothrombin approved|investigational|withdrawn DB00055 Drotrecogin alfa biotech P05154 Plasma serine protease inhibitor approved|investigational|withdrawn DB00055 Drotrecogin alfa biotech P35237 Serpin B6 approved|investigational|withdrawn DB00055 Drotrecogin alfa biotech P38435 Vitamin K-dependent gamma-carboxylase approved|investigational|withdrawn DB00055 Drotrecogin alfa biotech Q9UNN8 Endothelial protein C receptor approved|investigational DB00056 Gemtuzumab ozogamicin biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00056 Gemtuzumab ozogamicin biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00056 Gemtuzumab ozogamicin biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00056 Gemtuzumab ozogamicin biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00056 Gemtuzumab ozogamicin biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational DB00056 Gemtuzumab ozogamicin biotech P09871 Complement C1s subcomponent approved|investigational DB00056 Gemtuzumab ozogamicin biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00060 Interferon beta-1a biotech P17181 Interferon alpha/beta receptor 1 approved|investigational DB00060 Interferon beta-1a biotech P48551 Interferon alpha/beta receptor 2 approved DB00062 Human Serum Albumin biotech P02649 Apolipoprotein E approved DB00062 Human Serum Albumin biotech P0DJI8 Serum amyloid A-1 protein approved DB00062 Human Serum Albumin biotech P02760 Protein AMBP approved|investigational DB00063 Eptifibatide biotech P05106 Integrin beta-3 approved DB00065 Infliximab biotech P01375 Tumor necrosis factor approved DB00066 Follitropin biotech P23945 Follicle-stimulating hormone receptor approved DB00068 Interferon beta-1b biotech P17181 Interferon alpha/beta receptor 1 approved DB00068 Interferon beta-1b biotech P48551 Interferon alpha/beta receptor 2 approved|investigational DB00069 Interferon alfacon-1 biotech P17181 Interferon alpha/beta receptor 1 approved|investigational DB00069 Interferon alfacon-1 biotech P48551 Interferon alpha/beta receptor 2 approved|investigational DB00070 Hyaluronidase biotech P01137 Transforming growth factor beta-1 approved DB00071 Insulin Pork biotech P06213 Insulin receptor approved DB00071 Insulin Pork biotech P08069 Insulin-like growth factor 1 receptor approved DB00071 Insulin Pork biotech P14735 Insulin-degrading enzyme approved DB00071 Insulin Pork biotech P01920 HLA class II histocompatibility antigen, DQ beta 1 chain approved DB00071 Insulin Pork biotech P06400 Retinoblastoma-associated protein approved DB00071 Insulin Pork biotech P07339 Cathepsin D approved DB00071 Insulin Pork biotech P16870 Carboxypeptidase E approved DB00071 Insulin Pork biotech P16519 Neuroendocrine convertase 2 approved DB00071 Insulin Pork biotech P29120 Neuroendocrine convertase 1 approved DB00071 Insulin Pork biotech P48745 Protein NOV homolog approved DB00071 Insulin Pork biotech P98164 Low-density lipoprotein receptor-related protein 2 approved DB00071 Insulin Pork biotech Q16270 Insulin-like growth factor-binding protein 7 approved DB00071 Insulin Pork biotech Q96C24 Synaptotagmin-like protein 4 approved|investigational DB00072 Trastuzumab biotech P04626 Receptor tyrosine-protein kinase erbB-2 approved|investigational DB00072 Trastuzumab biotech P00533 Epidermal growth factor receptor approved|investigational DB00072 Trastuzumab biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00072 Trastuzumab biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00072 Trastuzumab biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00072 Trastuzumab biotech P09871 Complement C1s subcomponent approved|investigational DB00072 Trastuzumab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00072 Trastuzumab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00072 Trastuzumab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved DB00073 Rituximab biotech P11836 B-lymphocyte antigen CD20 approved DB00073 Rituximab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved DB00073 Rituximab biotech P02745 Complement C1q subcomponent subunit A approved DB00073 Rituximab biotech P02746 Complement C1q subcomponent subunit B approved DB00073 Rituximab biotech P02747 Complement C1q subcomponent subunit C approved DB00073 Rituximab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved DB00073 Rituximab biotech P09871 Complement C1s subcomponent approved DB00073 Rituximab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00074 Basiliximab biotech P01589 Interleukin-2 receptor subunit alpha approved|investigational DB00074 Basiliximab biotech P14784 Interleukin-2 receptor subunit beta approved|investigational DB00074 Basiliximab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational DB00074 Basiliximab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00074 Basiliximab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00074 Basiliximab biotech P09871 Complement C1s subcomponent approved|investigational DB00074 Basiliximab biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00074 Basiliximab biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00074 Basiliximab biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00075 Muromonab biotech P04234 T-cell surface glycoprotein CD3 delta chain approved|investigational DB00075 Muromonab biotech P07766 T-cell surface glycoprotein CD3 epsilon chain approved|investigational DB00075 Muromonab biotech P09693 T-cell surface glycoprotein CD3 gamma chain approved|investigational DB00075 Muromonab biotech P20963 T-cell surface glycoprotein CD3 zeta chain approved|investigational DB00075 Muromonab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00075 Muromonab biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00075 Muromonab biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00075 Muromonab biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00075 Muromonab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational DB00075 Muromonab biotech P09871 Complement C1s subcomponent approved|investigational DB00075 Muromonab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00078 Ibritumomab tiuxetan biotech P11836 B-lymphocyte antigen CD20 approved|investigational DB00078 Ibritumomab tiuxetan biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00078 Ibritumomab tiuxetan biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00078 Ibritumomab tiuxetan biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00078 Ibritumomab tiuxetan biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00078 Ibritumomab tiuxetan biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational DB00078 Ibritumomab tiuxetan biotech P09871 Complement C1s subcomponent approved|investigational DB00078 Ibritumomab tiuxetan biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00081 Tositumomab biotech P11836 B-lymphocyte antigen CD20 approved|investigational DB00081 Tositumomab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00081 Tositumomab biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00081 Tositumomab biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00081 Tositumomab biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00081 Tositumomab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational DB00081 Tositumomab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved DB00082 Pegvisomant biotech P10912 Growth hormone receptor approved|investigational DB00083 Botulinum Toxin Type A biotech P60880 Synaptosomal-associated protein 25 approved|investigational DB00083 Botulinum Toxin Type A biotech P62745 Rho-related GTP-binding protein RhoB approved|investigational DB00086 Streptokinase biotech P00747 Plasminogen approved|investigational DB00086 Streptokinase biotech P25116 Proteinase-activated receptor 1 approved|investigational DB00087 Alemtuzumab biotech P31358 CAMPATH-1 antigen approved|investigational DB00087 Alemtuzumab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00087 Alemtuzumab biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00087 Alemtuzumab biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00087 Alemtuzumab biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00087 Alemtuzumab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational DB00087 Alemtuzumab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved DB00089 Capromab pendetide biotech Q04609 Glutamate carboxypeptidase 2 approved|investigational|vet_approved DB00091 Cyclosporine small molecule P49069 Calcium signal-modulating cyclophilin ligand approved|investigational|vet_approved DB00091 Cyclosporine small molecule P62937 Peptidyl-prolyl cis-trans isomerase A approved|investigational|vet_approved DB00091 Cyclosporine small molecule P30405 Peptidyl-prolyl cis-trans isomerase F, mitochondrial approved|investigational|withdrawn DB00092 Alefacept biotech P06729 T-cell surface antigen CD2 approved|investigational|withdrawn DB00092 Alefacept biotech P02745 Complement C1q subcomponent subunit A approved|investigational|withdrawn DB00092 Alefacept biotech P02746 Complement C1q subcomponent subunit B approved|investigational|withdrawn DB00092 Alefacept biotech P02747 Complement C1q subcomponent subunit C approved|investigational|withdrawn DB00092 Alefacept biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational|withdrawn DB00092 Alefacept biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational|withdrawn DB00092 Alefacept biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|vet_approved DB00094 Urofollitropin biotech P23945 Follicle-stimulating hormone receptor approved|investigational DB00095 Efalizumab biotech P20701 Integrin alpha-L approved|investigational DB00095 Efalizumab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00095 Efalizumab biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00095 Efalizumab biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00095 Efalizumab biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00095 Efalizumab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational DB00095 Efalizumab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved DB00097 Choriogonadotropin alfa biotech P22888 Lutropin-choriogonadotropic hormone receptor approved DB00097 Choriogonadotropin alfa biotech P23945 Follicle-stimulating hormone receptor approved DB00098 Antithymocyte immunoglobulin (rabbit) biotech P06126 T-cell surface glycoprotein CD1a approved DB00098 Antithymocyte immunoglobulin (rabbit) biotech Q95460 Major histocompatibility complex class I-related gene protein approved DB00098 Antithymocyte immunoglobulin (rabbit) biotech P20701 Integrin alpha-L approved DB00098 Antithymocyte immunoglobulin (rabbit) biotech P42081 T-lymphocyte activation antigen CD86 approved DB00098 Antithymocyte immunoglobulin (rabbit) biotech P01730 T-cell surface glycoprotein CD4 approved DB00098 Antithymocyte immunoglobulin (rabbit) biotech P05556 Integrin beta-1 approved DB00098 Antithymocyte immunoglobulin (rabbit) biotech P06756 Integrin alpha-V approved DB00098 Antithymocyte immunoglobulin (rabbit) biotech P05106 Integrin beta-3 approved DB00099 Filgrastim biotech Q99062 Granulocyte colony-stimulating factor receptor approved|investigational DB00100 Coagulation Factor IX (Recombinant) biotech P00742 Coagulation factor X approved|investigational DB00100 Coagulation Factor IX (Recombinant) biotech P03951 Coagulation factor XI approved|investigational DB00100 Coagulation Factor IX (Recombinant) biotech P08709 Coagulation factor VII approved|investigational DB00100 Coagulation Factor IX (Recombinant) biotech P00451 Coagulation factor VIII approved|investigational DB00100 Coagulation Factor IX (Recombinant) biotech P00734 Prothrombin approved|investigational DB00100 Coagulation Factor IX (Recombinant) biotech Q07954 Prolow-density lipoprotein receptor-related protein 1 approved|investigational DB00100 Coagulation Factor IX (Recombinant) biotech P38435 Vitamin K-dependent gamma-carboxylase approved|investigational DB00102 Becaplermin biotech P09619 Platelet-derived growth factor receptor beta approved|investigational DB00102 Becaplermin biotech P16234 Platelet-derived growth factor receptor alpha approved|investigational DB00102 Becaplermin biotech P01023 Alpha-2-macroglobulin approved|investigational DB00104 Octreotide small molecule P35346 Somatostatin receptor type 5 approved DB00105 Interferon Alfa-2b, Recombinant biotech P48551 Interferon alpha/beta receptor 2 approved DB00105 Interferon Alfa-2b, Recombinant biotech P17181 Interferon alpha/beta receptor 1 approved|vet_approved DB00107 Oxytocin biotech P30559 Oxytocin receptor approved|investigational DB00108 Natalizumab biotech P13612 Integrin alpha-4 approved|investigational DB00108 Natalizumab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00108 Natalizumab biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00108 Natalizumab biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00108 Natalizumab biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00108 Natalizumab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational DB00108 Natalizumab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00108 Natalizumab biotech P05362 Intercellular adhesion molecule 1 approved|investigational DB00110 Palivizumab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00110 Palivizumab biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00110 Palivizumab biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00110 Palivizumab biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00110 Palivizumab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational DB00110 Palivizumab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a investigational|withdrawn DB00111 Daclizumab biotech P01589 Interleukin-2 receptor subunit alpha investigational|withdrawn DB00111 Daclizumab biotech P14784 Interleukin-2 receptor subunit beta investigational|withdrawn DB00111 Daclizumab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B investigational|withdrawn DB00111 Daclizumab biotech P02745 Complement C1q subcomponent subunit A investigational|withdrawn DB00111 Daclizumab biotech P02746 Complement C1q subcomponent subunit B investigational|withdrawn DB00111 Daclizumab biotech P02747 Complement C1q subcomponent subunit C investigational|withdrawn DB00111 Daclizumab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A investigational|withdrawn DB00111 Daclizumab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00112 Bevacizumab biotech P15692 Vascular endothelial growth factor A approved|investigational DB00112 Bevacizumab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational DB00112 Bevacizumab biotech P02745 Complement C1q subcomponent subunit A approved|investigational DB00112 Bevacizumab biotech P02746 Complement C1q subcomponent subunit B approved|investigational DB00112 Bevacizumab biotech P02747 Complement C1q subcomponent subunit C approved|investigational DB00112 Bevacizumab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational DB00112 Bevacizumab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational DB00113 Technetium Tc-99m arcitumomab biotech P13688 Carcinoembryonic antigen-related cell adhesion molecule 1 {ECO:0000303|Ref.8} approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q9BYV1 Alanine--glyoxylate aminotransferase 2, mitochondrial approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q99259 Glutamate decarboxylase 1 approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P35520 Cystathionine beta-synthase {ECO:0000305} approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q16719 Kynureninase {ECO:0000255|HAMAP-Rule:MF_03017} approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P34896 Serine hydroxymethyltransferase, cytosolic approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q9Y697 Cysteine desulfurase, mitochondrial approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P17174 Aspartate aminotransferase, cytoplasmic approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P04181 Ornithine aminotransferase, mitochondrial approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P11926 Ornithine decarboxylase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q8N5Z0 Kynurenine/alpha-aminoadipate aminotransferase, mitochondrial approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P80404 4-aminobutyrate aminotransferase, mitochondrial approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q9NVS9 Pyridoxine-5'-phosphate oxidase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule O95470 Sphingosine-1-phosphate lyase 1 {ECO:0000305} approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P17735 Tyrosine aminotransferase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q16773 Kynurenine--oxoglutarate transaminase 1 approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q8IYQ7 Threonine synthase-like 1 approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P06737 Glycogen phosphorylase, liver form approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule O15270 Serine palmitoyltransferase 2 approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q9Y600 Cysteine sulfinic acid decarboxylase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q96A70 Antizyme inhibitor 2 approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P20132 L-serine dehydratase/L-threonine deaminase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule O75600 2-amino-3-ketobutyrate coenzyme A ligase, mitochondrial approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P23378 Glycine dehydrogenase (decarboxylating), mitochondrial {ECO:0000303|PubMed:15489334} approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q9Y617 Phosphoserine aminotransferase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P13196 5-aminolevulinate synthase, nonspecific, mitochondrial approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P21549 Serine--pyruvate aminotransferase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q96GD0 Pyridoxal phosphate phosphatase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule O15269 Serine palmitoyltransferase 1 approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P32929 Cystathionine gamma-lyase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P54687 Branched-chain-amino-acid aminotransferase, cytosolic approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule O15382 Branched-chain-amino-acid aminotransferase, mitochondrial approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule O94903 Pyridoxal phosphate homeostasis protein {ECO:0000255|HAMAP-Rule:MF_03225} approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule O95954 Formimidoyltransferase-cyclodeaminase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P00505 Aspartate aminotransferase, mitochondrial approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P11216 Glycogen phosphorylase, brain form {ECO:0000303|PubMed:3346228} approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P20711 Aromatic-L-amino-acid decarboxylase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q99259 Glutamate decarboxylase 1 approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q6P996 Pyridoxal-dependent decarboxylase domain-containing protein 1 approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q6YP21 Kynurenine--oxoglutarate transaminase 3 approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q6ZQY3 Acidic amino acid decarboxylase GADL1 approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q96I15 Selenocysteine lyase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q8IUZ5 5-phosphohydroxy-L-lysine phospho-lyase approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P34897 Serine hydroxymethyltransferase, mitochondrial approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule P22557 5-aminolevulinate synthase, erythroid-specific, mitochondrial approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q8TD30 Alanine aminotransferase 2 approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q96EN8 Molybdenum cofactor sulfurase {ECO:0000255|HAMAP-Rule:MF_03050} approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q96GA7 Serine dehydratase-like approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q9GZT4 Serine racemase {ECO:0000303|PubMed:11054547} approved|investigational|nutraceutical DB00114 Pyridoxal Phosphate small molecule Q9NUV7 Serine palmitoyltransferase 3 approved|nutraceutical DB00115 Cyanocobalamin small molecule Q99707 Methionine synthase approved|nutraceutical DB00115 Cyanocobalamin small molecule P22033 Methylmalonyl-CoA mutase, mitochondrial approved|nutraceutical DB00115 Cyanocobalamin small molecule Q9UBK8 Methionine synthase reductase approved|nutraceutical DB00115 Cyanocobalamin small molecule Q9Y4U1 Methylmalonic aciduria and homocystinuria type C protein approved|nutraceutical DB00115 Cyanocobalamin small molecule P42898 Methylenetetrahydrofolate reductase {ECO:0000305} approved|investigational|nutraceutical DB00118 Ademetionine small molecule Q14749 Glycine N-methyltransferase approved|investigational|nutraceutical DB00118 Ademetionine small molecule P17707 S-adenosylmethionine decarboxylase proenzyme approved|investigational|nutraceutical DB00118 Ademetionine small molecule P31153 S-adenosylmethionine synthase isoform type-2 approved|investigational|nutraceutical DB00118 Ademetionine small molecule P35520 Cystathionine beta-synthase {ECO:0000305} approved|investigational|nutraceutical DB00118 Ademetionine small molecule Q00266 S-adenosylmethionine synthase isoform type-1 approved|investigational|nutraceutical DB00118 Ademetionine small molecule P21964 Catechol O-methyltransferase approved|investigational|nutraceutical DB00118 Ademetionine small molecule Q8N1G2 Cap-specific mRNA (nucleoside-2'-O-)-methyltransferase 1 approved|investigational|nutraceutical DB00118 Ademetionine small molecule Q9HBK9 Arsenite methyltransferase approved|investigational|nutraceutical DB00121 Biotin small molecule P05166 Propionyl-CoA carboxylase beta chain, mitochondrial approved|investigational|nutraceutical DB00121 Biotin small molecule P50747 Biotin--protein ligase approved|investigational|nutraceutical DB00121 Biotin small molecule Q9Y289 Sodium-dependent multivitamin transporter approved|investigational|nutraceutical DB00121 Biotin small molecule Q9HCC0 Methylcrotonoyl-CoA carboxylase beta chain, mitochondrial approved|investigational|nutraceutical DB00121 Biotin small molecule O00763 Acetyl-CoA carboxylase 2 approved|investigational|nutraceutical DB00121 Biotin small molecule Q96RQ3 Methylcrotonoyl-CoA carboxylase subunit alpha, mitochondrial approved|investigational|nutraceutical DB00121 Biotin small molecule P11498 Pyruvate carboxylase, mitochondrial approved|investigational|nutraceutical DB00121 Biotin small molecule P05165 Propionyl-CoA carboxylase alpha chain, mitochondrial approved|investigational|nutraceutical DB00121 Biotin small molecule Q13085 Acetyl-CoA carboxylase 1 approved|nutraceutical DB00122 Choline small molecule Q9Y5K3 Choline-phosphate cytidylyltransferase B approved|nutraceutical DB00122 Choline small molecule P22303 Acetylcholinesterase approved|nutraceutical DB00122 Choline small molecule P49585 Choline-phosphate cytidylyltransferase A approved|nutraceutical DB00122 Choline small molecule O14939 Phospholipase D2 approved|nutraceutical DB00122 Choline small molecule P06276 Cholinesterase approved|nutraceutical DB00122 Choline small molecule Q13393 Phospholipase D1 approved|nutraceutical DB00122 Choline small molecule Q8TCT1 Phosphoethanolamine/phosphocholine phosphatase approved|nutraceutical DB00122 Choline small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|nutraceutical DB00123 L-Lysine small molecule P30825 High affinity cationic amino acid transporter 1 approved|nutraceutical DB00123 L-Lysine small molecule P52569 Cationic amino acid transporter 2 approved|nutraceutical DB00123 L-Lysine small molecule Q15046 Lysine--tRNA ligase approved|nutraceutical DB00125 L-Arginine small molecule P29474 Nitric oxide synthase, endothelial approved|nutraceutical DB00125 L-Arginine small molecule Q96A70 Antizyme inhibitor 2 approved|nutraceutical DB00125 L-Arginine small molecule P04424 Argininosuccinate lyase approved|nutraceutical DB00125 L-Arginine small molecule P35228 Nitric oxide synthase, inducible approved|nutraceutical DB00125 L-Arginine small molecule P30825 High affinity cationic amino acid transporter 1 approved|nutraceutical DB00125 L-Arginine small molecule P78540 Arginase-2, mitochondrial approved|nutraceutical DB00125 L-Arginine small molecule P00966 Argininosuccinate synthase {ECO:0000305} approved|nutraceutical DB00126 Vitamin C small molecule P09848 Lactase-phlorizin hydrolase approved|nutraceutical DB00126 Vitamin C small molecule O00469 Procollagen-lysine,2-oxoglutarate 5-dioxygenase 2 approved|nutraceutical DB00126 Vitamin C small molecule O14832 Phytanoyl-CoA dioxygenase, peroxisomal approved|nutraceutical DB00126 Vitamin C small molecule O60568 Procollagen-lysine,2-oxoglutarate 5-dioxygenase 3 approved|nutraceutical DB00126 Vitamin C small molecule O75936 Gamma-butyrobetaine dioxygenase approved|nutraceutical DB00126 Vitamin C small molecule P09172 Dopamine beta-hydroxylase approved|nutraceutical DB00126 Vitamin C small molecule P19021 Peptidyl-glycine alpha-amidating monooxygenase approved|nutraceutical DB00126 Vitamin C small molecule P13674 Prolyl 4-hydroxylase subunit alpha-1 approved|nutraceutical DB00126 Vitamin C small molecule Q32P28 Prolyl 3-hydroxylase 1 {ECO:0000312|HGNC:HGNC:19316} approved|nutraceutical DB00126 Vitamin C small molecule Q6N063 2-oxoglutarate and iron-dependent oxygenase domain-containing protein 2 approved|nutraceutical DB00126 Vitamin C small molecule Q8IVL5 Prolyl 3-hydroxylase 2 {ECO:0000312|HGNC:HGNC:19317} approved|nutraceutical DB00126 Vitamin C small molecule Q8IVL6 Prolyl 3-hydroxylase 3 {ECO:0000312|HGNC:HGNC:19318} approved|nutraceutical DB00126 Vitamin C small molecule Q8N543 Prolyl 3-hydroxylase OGFOD1 approved|nutraceutical DB00126 Vitamin C small molecule Q96KS0 Egl nine homolog 2 approved|nutraceutical DB00126 Vitamin C small molecule Q96Q83 Alpha-ketoglutarate-dependent dioxygenase alkB homolog 3 {ECO:0000305} approved|nutraceutical DB00126 Vitamin C small molecule Q9BY66 Lysine-specific demethylase 5D approved|nutraceutical DB00126 Vitamin C small molecule Q9GZT9 Egl nine homolog 1 approved|nutraceutical DB00126 Vitamin C small molecule Q9UHI7 Solute carrier family 23 member 1 approved|nutraceutical DB00126 Vitamin C small molecule Q02809 Procollagen-lysine,2-oxoglutarate 5-dioxygenase 1 approved|nutraceutical DB00126 Vitamin C small molecule Q9H6Z9 Egl nine homolog 3 approved|nutraceutical DB00126 Vitamin C small molecule Q9NVH6 Trimethyllysine dioxygenase, mitochondrial approved|nutraceutical DB00126 Vitamin C small molecule Q9NXG6 Transmembrane prolyl 4-hydroxylase approved|investigational|nutraceutical DB00130 L-Glutamine small molecule P17812 CTP synthase 1 {ECO:0000305} approved|investigational|nutraceutical DB00130 L-Glutamine small molecule Q06203 Amidophosphoribosyltransferase approved|investigational|nutraceutical DB00130 L-Glutamine small molecule P15104 Glutamine synthetase approved|nutraceutical DB00134 Methionine small molecule Q9UBK8 Methionine synthase reductase approved|nutraceutical DB00134 Methionine small molecule Q99707 Methionine synthase approved|nutraceutical DB00134 Methionine small molecule P50579 Methionine aminopeptidase 2 {ECO:0000255|HAMAP-Rule:MF_03175} approved|nutraceutical DB00134 Methionine small molecule Q93088 Betaine--homocysteine S-methyltransferase 1 approved|nutraceutical DB00134 Methionine small molecule Q9H2M3 S-methylmethionine--homocysteine S-methyltransferase BHMT2 approved|nutraceutical DB00136 Calcitriol small molecule P11473 Vitamin D3 receptor approved|nutraceutical DB00136 Calcitriol small molecule P31260 Homeobox protein Hox-A10 approved|nutraceutical DB00136 Calcitriol small molecule P02774 Vitamin D-binding protein approved|investigational|nutraceutical|vet_approved DB00140 Riboflavin small molecule Q969G6 Riboflavin kinase approved|investigational|nutraceutical|vet_approved DB00140 Riboflavin small molecule P30043 Flavin reductase (NADPH) approved|nutraceutical DB00142 Glutamic Acid small molecule Q13255 Metabotropic glutamate receptor 1 approved|nutraceutical DB00142 Glutamic Acid small molecule Q14833 Metabotropic glutamate receptor 4 approved|nutraceutical DB00142 Glutamic Acid small molecule Q16099 Glutamate receptor ionotropic, kainate 4 approved|nutraceutical DB00142 Glutamic Acid small molecule Q16478 Glutamate receptor ionotropic, kainate 5 approved|nutraceutical DB00142 Glutamic Acid small molecule Q14831 Metabotropic glutamate receptor 7 approved|nutraceutical DB00142 Glutamic Acid small molecule O00222 Metabotropic glutamate receptor 8 approved|nutraceutical DB00142 Glutamic Acid small molecule O00341 Excitatory amino acid transporter 5 approved|nutraceutical DB00142 Glutamic Acid small molecule O14841 5-oxoprolinase approved|nutraceutical DB00142 Glutamic Acid small molecule O15067 Phosphoribosylformylglycinamidine synthase approved|nutraceutical DB00142 Glutamic Acid small molecule O15382 Branched-chain-amino-acid aminotransferase, mitochondrial approved|nutraceutical DB00142 Glutamic Acid small molecule O15399 Glutamate receptor ionotropic, NMDA 2D approved|nutraceutical DB00142 Glutamic Acid small molecule O43424 Glutamate receptor ionotropic, delta-2 approved|nutraceutical DB00142 Glutamic Acid small molecule O60391 Glutamate receptor ionotropic, NMDA 3B approved|nutraceutical DB00142 Glutamic Acid small molecule O94925 Glutaminase kidney isoform, mitochondrial approved|nutraceutical DB00142 Glutamic Acid small molecule P00505 Aspartate aminotransferase, mitochondrial approved|nutraceutical DB00142 Glutamic Acid small molecule P07814 Bifunctional glutamate/proline--tRNA ligase approved|nutraceutical DB00142 Glutamic Acid small molecule P08243 Asparagine synthetase [glutamine-hydrolyzing] approved|nutraceutical DB00142 Glutamic Acid small molecule P15104 Glutamine synthetase approved|nutraceutical DB00142 Glutamic Acid small molecule P17174 Aspartate aminotransferase, cytoplasmic approved|nutraceutical DB00142 Glutamic Acid small molecule P17735 Tyrosine aminotransferase approved|nutraceutical DB00142 Glutamic Acid small molecule P38435 Vitamin K-dependent gamma-carboxylase approved|nutraceutical DB00142 Glutamic Acid small molecule P43003 Excitatory amino acid transporter 1 {ECO:0000303|PubMed:16042756, ECO:0000303|PubMed:8647279} approved|nutraceutical DB00142 Glutamic Acid small molecule P43004 Excitatory amino acid transporter 2 approved|nutraceutical DB00142 Glutamic Acid small molecule P43005 Excitatory amino acid transporter 3 approved|nutraceutical DB00142 Glutamic Acid small molecule P48506 Glutamate--cysteine ligase catalytic subunit approved|nutraceutical DB00142 Glutamic Acid small molecule P48664 Excitatory amino acid transporter 4 approved|nutraceutical DB00142 Glutamic Acid small molecule P49915 GMP synthase [glutamine-hydrolyzing] approved|nutraceutical DB00142 Glutamic Acid small molecule P54687 Branched-chain-amino-acid aminotransferase, cytosolic approved|nutraceutical DB00142 Glutamic Acid small molecule P80404 4-aminobutyrate aminotransferase, mitochondrial approved|nutraceutical DB00142 Glutamic Acid small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved|nutraceutical DB00142 Glutamic Acid small molecule Q05932 Folylpolyglutamate synthase, mitochondrial approved|nutraceutical DB00142 Glutamic Acid small molecule Q07075 Glutamyl aminopeptidase approved|nutraceutical DB00142 Glutamic Acid small molecule Q12879 Glutamate receptor ionotropic, NMDA 2A approved|nutraceutical DB00142 Glutamic Acid small molecule Q13224 Glutamate receptor ionotropic, NMDA 2B approved|nutraceutical DB00142 Glutamic Acid small molecule Q5JPH6 Probable glutamate--tRNA ligase, mitochondrial approved|nutraceutical DB00142 Glutamic Acid small molecule Q5TDP6 Lengsin approved|nutraceutical DB00142 Glutamic Acid small molecule Q6IA69 Glutamine-dependent NAD(+) synthetase approved|nutraceutical DB00142 Glutamic Acid small molecule Q6YP21 Kynurenine--oxoglutarate transaminase 3 approved|nutraceutical DB00142 Glutamic Acid small molecule Q8N159 N-acetylglutamate synthase, mitochondrial approved|nutraceutical DB00142 Glutamic Acid small molecule Q8N5Z0 Kynurenine/alpha-aminoadipate aminotransferase, mitochondrial approved|nutraceutical DB00142 Glutamic Acid small molecule Q8TD30 Alanine aminotransferase 2 approved|nutraceutical DB00142 Glutamic Acid small molecule Q9H1K4 Mitochondrial glutamate carrier 2 approved|nutraceutical DB00142 Glutamic Acid small molecule Q9H936 Mitochondrial glutamate carrier 1 approved|nutraceutical DB00142 Glutamic Acid small molecule Q9UDR5 Alpha-aminoadipic semialdehyde synthase, mitochondrial approved|nutraceutical DB00142 Glutamic Acid small molecule Q9UI32 Glutaminase liver isoform, mitochondrial approved|nutraceutical DB00142 Glutamic Acid small molecule Q9ULA0 Aspartyl aminopeptidase approved|nutraceutical DB00142 Glutamic Acid small molecule Q9ULK0 Glutamate receptor ionotropic, delta-1 approved|nutraceutical DB00142 Glutamic Acid small molecule Q9Y646 Carboxypeptidase Q approved|nutraceutical DB00142 Glutamic Acid small molecule Q9Y617 Phosphoserine aminotransferase approved|nutraceutical DB00142 Glutamic Acid small molecule P00367 Glutamate dehydrogenase 1, mitochondrial approved|nutraceutical DB00142 Glutamic Acid small molecule P39086 Glutamate receptor ionotropic, kainate 1 approved|nutraceutical DB00142 Glutamic Acid small molecule P42261 Glutamate receptor 1 approved|nutraceutical DB00142 Glutamic Acid small molecule P48507 Glutamate--cysteine ligase regulatory subunit approved|nutraceutical DB00142 Glutamic Acid small molecule Q04609 Glutamate carboxypeptidase 2 approved|nutraceutical DB00142 Glutamic Acid small molecule Q05329 Glutamate decarboxylase 2 approved|nutraceutical DB00142 Glutamic Acid small molecule Q99259 Glutamate decarboxylase 1 approved|nutraceutical DB00142 Glutamic Acid small molecule O95954 Formimidoyltransferase-cyclodeaminase approved|nutraceutical DB00142 Glutamic Acid small molecule P42262 Glutamate receptor 2 approved|nutraceutical DB00142 Glutamic Acid small molecule P42263 Glutamate receptor 3 approved|nutraceutical DB00142 Glutamic Acid small molecule P48058 Glutamate receptor 4 approved|nutraceutical DB00142 Glutamic Acid small molecule P54886 Delta-1-pyrroline-5-carboxylate synthase approved|nutraceutical DB00142 Glutamic Acid small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved|nutraceutical DB00142 Glutamic Acid small molecule Q13003 Glutamate receptor ionotropic, kainate 3 approved|investigational|nutraceutical DB00143 Glutathione small molecule O14880 Microsomal glutathione S-transferase 3 approved|investigational|nutraceutical DB00143 Glutathione small molecule O95881 Thioredoxin domain-containing protein 12 approved|investigational|nutraceutical DB00143 Glutathione small molecule P08263 Glutathione S-transferase A1 approved|investigational|nutraceutical DB00143 Glutathione small molecule P10620 Microsomal glutathione S-transferase 1 approved|investigational|nutraceutical DB00143 Glutathione small molecule P10768 S-formylglutathione hydrolase approved|investigational|nutraceutical DB00143 Glutathione small molecule P19440 Glutathione hydrolase 1 proenzyme approved|investigational|nutraceutical DB00143 Glutathione small molecule P28161 Glutathione S-transferase Mu 2 approved|investigational|nutraceutical DB00143 Glutathione small molecule P35754 Glutaredoxin-1 approved|investigational|nutraceutical DB00143 Glutathione small molecule P36969 Phospholipid hydroperoxide glutathione peroxidase approved|investigational|nutraceutical DB00143 Glutathione small molecule P46439 Glutathione S-transferase Mu 5 approved|investigational|nutraceutical DB00143 Glutathione small molecule P59796 Glutathione peroxidase 6 approved|investigational|nutraceutical DB00143 Glutathione small molecule Q16775 Hydroxyacylglutathione hydrolase, mitochondrial {ECO:0000303|PubMed:15117945} approved|investigational|nutraceutical DB00143 Glutathione small molecule Q8TED1 Probable glutathione peroxidase 8 approved|investigational|nutraceutical DB00143 Glutathione small molecule Q96SL4 Glutathione peroxidase 7 approved|investigational|nutraceutical DB00143 Glutathione small molecule Q99735 Microsomal glutathione S-transferase 2 approved|investigational|nutraceutical DB00143 Glutathione small molecule Q9H4Y5 Glutathione S-transferase omega-2 approved|investigational|nutraceutical DB00143 Glutathione small molecule Q9NS18 Glutaredoxin-2, mitochondrial approved|investigational|nutraceutical DB00143 Glutathione small molecule Q04760 Lactoylglutathione lyase approved|investigational|nutraceutical DB00143 Glutathione small molecule P00390 Glutathione reductase, mitochondrial approved|investigational|nutraceutical DB00143 Glutathione small molecule P48637 Glutathione synthetase approved|investigational|nutraceutical DB00143 Glutathione small molecule P09488 Glutathione S-transferase Mu 1 approved|investigational|nutraceutical DB00143 Glutathione small molecule Q9Y2Q3 Glutathione S-transferase kappa 1 approved|investigational|nutraceutical DB00143 Glutathione small molecule P21266 Glutathione S-transferase Mu 3 approved|investigational|nutraceutical DB00143 Glutathione small molecule O15217 Glutathione S-transferase A4 approved|investigational|nutraceutical DB00143 Glutathione small molecule Q03013 Glutathione S-transferase Mu 4 approved|investigational|nutraceutical DB00143 Glutathione small molecule Q7RTV2 Glutathione S-transferase A5 approved|investigational|nutraceutical DB00143 Glutathione small molecule P09211 Glutathione S-transferase P approved|investigational|nutraceutical DB00143 Glutathione small molecule P78417 Glutathione S-transferase omega-1 approved|investigational|nutraceutical DB00143 Glutathione small molecule P07203 Glutathione peroxidase 1 approved|investigational|nutraceutical DB00143 Glutathione small molecule P30711 Glutathione S-transferase theta-1 approved|investigational|nutraceutical DB00143 Glutathione small molecule O43708 Maleylacetoacetate isomerase approved|investigational|nutraceutical DB00143 Glutathione small molecule O75715 Epididymal secretory glutathione peroxidase approved|investigational|nutraceutical DB00143 Glutathione small molecule P22352 Glutathione peroxidase 3 approved|investigational|nutraceutical DB00143 Glutathione small molecule P15121 Aldose reductase approved|investigational|nutraceutical DB00143 Glutathione small molecule P14780 Matrix metalloproteinase-9 approved|investigational|nutraceutical DB00143 Glutathione small molecule P08684 Cytochrome P450 3A4 approved|nutraceutical|vet_approved DB00145 Glycine small molecule O75600 2-amino-3-ketobutyrate coenzyme A ligase, mitochondrial approved|nutraceutical|vet_approved DB00145 Glycine small molecule P13196 5-aminolevulinate synthase, nonspecific, mitochondrial approved|nutraceutical|vet_approved DB00145 Glycine small molecule P22557 5-aminolevulinate synthase, erythroid-specific, mitochondrial approved|nutraceutical|vet_approved DB00145 Glycine small molecule P23434 Glycine cleavage system H protein, mitochondrial {ECO:0000303|PubMed:1671321} approved|nutraceutical|vet_approved DB00145 Glycine small molecule P41250 Glycine--tRNA ligase approved|nutraceutical|vet_approved DB00145 Glycine small molecule Q12879 Glutamate receptor ionotropic, NMDA 2A approved|nutraceutical|vet_approved DB00145 Glycine small molecule Q14032 Bile acid-CoA:amino acid N-acyltransferase {ECO:0000303|PubMed:8034703} approved|nutraceutical|vet_approved DB00145 Glycine small molecule P48637 Glutathione synthetase approved|nutraceutical|vet_approved DB00145 Glycine small molecule Q6IB77 Glycine N-acyltransferase {ECO:0000303|PubMed:10630424} approved|nutraceutical|vet_approved DB00145 Glycine small molecule Q7Z2H8 Proton-coupled amino acid transporter 1 approved|nutraceutical|vet_approved DB00145 Glycine small molecule P34897 Serine hydroxymethyltransferase, mitochondrial approved|nutraceutical|vet_approved DB00145 Glycine small molecule Q8WU03 Glycine N-acyltransferase-like protein 2 approved|nutraceutical|vet_approved DB00145 Glycine small molecule Q969I3 Glycine N-acyltransferase-like protein 1 approved|nutraceutical|vet_approved DB00145 Glycine small molecule Q9BYV1 Alanine--glyoxylate aminotransferase 2, mitochondrial approved|nutraceutical|vet_approved DB00145 Glycine small molecule Q9P0Z9 Peroxisomal sarcosine oxidase approved|nutraceutical|vet_approved DB00145 Glycine small molecule O60391 Glutamate receptor ionotropic, NMDA 3B approved|nutraceutical|vet_approved DB00145 Glycine small molecule P23378 Glycine dehydrogenase (decarboxylating), mitochondrial {ECO:0000303|PubMed:15489334} approved|nutraceutical|vet_approved DB00145 Glycine small molecule P48067 Sodium- and chloride-dependent glycine transporter 1 approved|nutraceutical|vet_approved DB00145 Glycine small molecule P23415 Glycine receptor subunit alpha-1 approved|nutraceutical|vet_approved DB00145 Glycine small molecule P21549 Serine--pyruvate aminotransferase approved|nutraceutical|vet_approved DB00145 Glycine small molecule P34896 Serine hydroxymethyltransferase, cytosolic approved|nutraceutical|vet_approved DB00145 Glycine small molecule P23416 Glycine receptor subunit alpha-2 approved|nutraceutical|vet_approved DB00145 Glycine small molecule Q14749 Glycine N-methyltransferase approved|nutraceutical|vet_approved DB00145 Glycine small molecule P50440 Glycine amidinotransferase, mitochondrial approved|nutraceutical DB00146 Calcidiol small molecule P11473 Vitamin D3 receptor approved|nutraceutical|withdrawn DB00150 L-Tryptophan small molecule Q9UGM6 Tryptophan--tRNA ligase, mitochondrial approved|nutraceutical|withdrawn DB00150 L-Tryptophan small molecule P23381 Tryptophan--tRNA ligase, cytoplasmic approved|investigational|nutraceutical|vet_approved DB00152 Thiamine small molecule Q9H3S4 Thiamin pyrophosphokinase 1 approved|investigational|nutraceutical|vet_approved DB00152 Thiamine small molecule O60779 Thiamine transporter 1 approved|nutraceutical DB00153 Ergocalciferol small molecule P11473 Vitamin D3 receptor approved|nutraceutical|vet_approved DB00158 Folic Acid small molecule P41439 Folate receptor gamma approved|nutraceutical|vet_approved DB00158 Folic Acid small molecule P15328 Folate receptor alpha approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule O75911 Short-chain dehydrogenase/reductase 3 approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule P47895 Aldehyde dehydrogenase family 1 member A3 approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule Q6NUM9 All-trans-retinol 13,14-reductase approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule Q8TC12 Retinol dehydrogenase 11 approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule Q9BTZ2 Dehydrogenase/reductase SDR family member 4 approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule Q9HBH5 Retinol dehydrogenase 14 approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule Q9NYR8 Retinol dehydrogenase 8 approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule O95237 Lecithin retinol acyltransferase approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule P09455 Retinol-binding protein 1 approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule Q92781 11-cis retinol dehydrogenase approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule Q8NBN7 Retinol dehydrogenase 13 approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule O94788 Retinal dehydrogenase 2 approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule P00352 Retinal dehydrogenase 1 {ECO:0000305} approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule P12271 Retinaldehyde-binding protein 1 approved|nutraceutical|vet_approved DB00162 Vitamin A small molecule P05090 Apolipoprotein D approved|investigational|nutraceutical|vet_approved DB00165 Pyridoxine small molecule O00764 Pyridoxal kinase approved|investigational|nutraceutical DB00166 Lipoic Acid small molecule O43766 Lipoyl synthase, mitochondrial {ECO:0000255|HAMAP-Rule:MF_03123} approved|investigational|nutraceutical DB00166 Lipoic Acid small molecule Q9Y289 Sodium-dependent multivitamin transporter approved|nutraceutical DB00169 Cholecalciferol small molecule P11473 Vitamin D3 receptor approved|nutraceutical DB00170 Menadione small molecule P38435 Vitamin K-dependent gamma-carboxylase approved|nutraceutical DB00170 Menadione small molecule Q9BQB6 Vitamin K epoxide reductase complex subunit 1 approved|nutraceutical DB00170 Menadione small molecule Q8N0U8 Vitamin K epoxide reductase complex subunit 1-like protein 1 approved|nutraceutical DB00170 Menadione small molecule P00734 Prothrombin approved|nutraceutical DB00170 Menadione small molecule P08709 Coagulation factor VII approved|nutraceutical DB00170 Menadione small molecule P00742 Coagulation factor X approved|nutraceutical DB00170 Menadione small molecule P07225 Vitamin K-dependent protein S approved|nutraceutical DB00170 Menadione small molecule P22891 Vitamin K-dependent protein Z approved|nutraceutical DB00170 Menadione small molecule P16083 Ribosyldihydronicotinamide dehydrogenase [quinone] approved|nutraceutical DB00170 Menadione small molecule P15559 NAD(P)H dehydrogenase [quinone] 1 approved DB00175 Pravastatin small molecule P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase approved|investigational DB00176 Fluvoxamine small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB00176 Fluvoxamine small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB00177 Valsartan small molecule P30556 Type-1 angiotensin II receptor approved DB00178 Ramipril small molecule P12821 Angiotensin-converting enzyme approved|investigational DB00179 Masoprocol small molecule P09917 Arachidonate 5-lipoxygenase approved|investigational DB00179 Masoprocol small molecule P04278 Sex hormone-binding globulin approved|investigational DB00180 Flunisolide small molecule P04150 Glucocorticoid receptor approved DB00181 Baclofen small molecule Q9UBS5 Gamma-aminobutyric acid type B receptor subunit 1 approved DB00181 Baclofen small molecule O75899 Gamma-aminobutyric acid type B receptor subunit 2 approved|illicit|investigational DB00182 Amphetamine small molecule Q05940 Synaptic vesicular amine transporter approved|illicit|investigational DB00182 Amphetamine small molecule Q16568 Cocaine- and amphetamine-regulated transcript protein approved|illicit|investigational DB00182 Amphetamine small molecule P23975 Sodium-dependent noradrenaline transporter approved|illicit|investigational DB00182 Amphetamine small molecule P14416 D(2) dopamine receptor approved|illicit|investigational DB00182 Amphetamine small molecule P27338 Amine oxidase [flavin-containing] B approved|illicit|investigational DB00182 Amphetamine small molecule P31645 Sodium-dependent serotonin transporter approved|illicit|investigational DB00182 Amphetamine small molecule P21397 Amine oxidase [flavin-containing] A approved DB00184 Nicotine small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved DB00184 Nicotine small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved DB00184 Nicotine small molecule P17787 Neuronal acetylcholine receptor subunit beta-2 approved DB00184 Nicotine small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB00184 Nicotine small molecule P32297 Neuronal acetylcholine receptor subunit alpha-3 approved DB00184 Nicotine small molecule Q15825 Neuronal acetylcholine receptor subunit alpha-6 approved DB00184 Nicotine small molecule Q9UGM1 Neuronal acetylcholine receptor subunit alpha-9 approved DB00184 Nicotine small molecule Q05901 Neuronal acetylcholine receptor subunit beta-3 approved DB00184 Nicotine small molecule P30926 Neuronal acetylcholine receptor subunit beta-4 approved DB00184 Nicotine small molecule P11511 Aromatase approved DB00185 Cevimeline small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00185 Cevimeline small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00186 Lorazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00186 Lorazepam small molecule P30536 Translocator protein approved|investigational DB00188 Bortezomib small molecule P28074 Proteasome subunit beta type-5 approved|investigational DB00188 Bortezomib small molecule P20618 Proteasome subunit beta type-1 approved|illicit|withdrawn DB00189 Ethchlorvynol small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB00191 Phentermine small molecule P23975 Sodium-dependent noradrenaline transporter approved|illicit DB00191 Phentermine small molecule P31645 Sodium-dependent serotonin transporter approved|illicit DB00191 Phentermine small molecule P21397 Amine oxidase [flavin-containing] A approved|illicit DB00191 Phentermine small molecule P27338 Amine oxidase [flavin-containing] B approved|investigational DB00193 Tramadol small molecule P35372 Mu-type opioid receptor approved|investigational DB00193 Tramadol small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB00193 Tramadol small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB00193 Tramadol small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB00193 Tramadol small molecule P41143 Delta-type opioid receptor approved|investigational DB00193 Tramadol small molecule P20309 Muscarinic acetylcholine receptor M3 investigational|withdrawn DB00197 Troglitazone small molecule P37231 Peroxisome proliferator-activated receptor gamma investigational|withdrawn DB00197 Troglitazone small molecule O60488 Long-chain-fatty-acid--CoA ligase 4 investigational|withdrawn DB00197 Troglitazone small molecule P05121 Plasminogen activator inhibitor 1 investigational|withdrawn DB00197 Troglitazone small molecule Q99808 Equilibrative nucleoside transporter 1 investigational|withdrawn DB00197 Troglitazone small molecule P62508 Estrogen-related receptor gamma investigational|withdrawn DB00197 Troglitazone small molecule P11474 Steroid hormone receptor ERR1 investigational|withdrawn DB00197 Troglitazone small molecule Q03181 Peroxisome proliferator-activated receptor delta investigational|withdrawn DB00197 Troglitazone small molecule Q07869 Peroxisome proliferator-activated receptor alpha investigational|withdrawn DB00197 Troglitazone small molecule P09211 Glutathione S-transferase P approved DB00198 Oseltamivir small molecule P23141 Liver carboxylesterase 1 approved DB00198 Oseltamivir small molecule Q99519 Sialidase-1 approved|investigational|vet_approved DB00199 Erythromycin small molecule O43193 Motilin receptor approved|investigational|vet_approved DB00199 Erythromycin small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational|vet_approved DB00199 Erythromycin small molecule P02768 Serum albumin approved DB00200 Hydroxocobalamin small molecule Q99707 Methionine synthase approved DB00200 Hydroxocobalamin small molecule P22033 Methylmalonyl-CoA mutase, mitochondrial approved DB00200 Hydroxocobalamin small molecule Q9UBK8 Methionine synthase reductase approved DB00200 Hydroxocobalamin small molecule P20061 Transcobalamin-1 approved DB00200 Hydroxocobalamin small molecule Q9BXJ7 Protein amnionless approved DB00200 Hydroxocobalamin small molecule O60494 Cubilin approved DB00200 Hydroxocobalamin small molecule Q9Y4U1 Methylmalonic aciduria and homocystinuria type C protein approved DB00201 Caffeine small molecule P30542 Adenosine receptor A1 approved DB00201 Caffeine small molecule Q07343 cAMP-specific 3',5'-cyclic phosphodiesterase 4B approved DB00201 Caffeine small molecule P21817 Ryanodine receptor 1 approved DB00201 Caffeine small molecule P54750 Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A approved DB00201 Caffeine small molecule P78527 DNA-dependent protein kinase catalytic subunit approved DB00201 Caffeine small molecule O00329 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform approved DB00201 Caffeine small molecule P42336 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform approved DB00201 Caffeine small molecule P42338 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform approved DB00201 Caffeine small molecule Q14643 Inositol 1,4,5-trisphosphate receptor type 1 approved DB00201 Caffeine small molecule Q13315 Serine-protein kinase ATM approved DB00202 Succinylcholine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00202 Succinylcholine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00202 Succinylcholine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB00203 Sildenafil small molecule O76074 cGMP-specific 3',5'-cyclic phosphodiesterase approved|investigational DB00203 Sildenafil small molecule P18545 Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma approved|investigational DB00203 Sildenafil small molecule Q13956 Retinal cone rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma approved|investigational DB00204 Dofetilide small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB00204 Dofetilide small molecule O95069 Potassium channel subfamily K member 2 approved|investigational DB00204 Dofetilide small molecule Q14500 ATP-sensitive inward rectifier potassium channel 12 approved|investigational|vet_approved DB00205 Pyrimethamine small molecule P00374 Dihydrofolate reductase approved|investigational|vet_approved DB00205 Pyrimethamine small molecule P07686 Beta-hexosaminidase subunit beta approved|investigational DB00206 Reserpine small molecule Q05940 Synaptic vesicular amine transporter approved|investigational DB00206 Reserpine small molecule O15392 Baculoviral IAP repeat-containing protein 5 approved DB00207 Azithromycin small molecule Q9UM07 Protein-arginine deiminase type-4 approved DB00208 Ticlopidine small molecule Q9H244 P2Y purinoceptor 12 approved DB00209 Trospium small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00210 Adapalene small molecule P13631 Retinoic acid receptor gamma approved DB00210 Adapalene small molecule P10826 Retinoic acid receptor beta approved DB00210 Adapalene small molecule P48443 Retinoic acid receptor RXR-gamma approved DB00210 Adapalene small molecule P28702 Retinoic acid receptor RXR-beta approved DB00210 Adapalene small molecule P10276 Retinoic acid receptor alpha approved DB00210 Adapalene small molecule P19793 Retinoic acid receptor RXR-alpha approved DB00211 Midodrine small molecule P25100 Alpha-1D adrenergic receptor approved DB00212 Remikiren small molecule P00797 Renin approved DB00213 Pantoprazole small molecule P20648 Potassium-transporting ATPase alpha chain 1 approved DB00214 Torasemide small molecule Q13621 Solute carrier family 12 member 1 approved DB00215 Citalopram small molecule P31645 Sodium-dependent serotonin transporter approved DB00215 Citalopram small molecule P35367 Histamine H1 receptor approved DB00215 Citalopram small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00215 Citalopram small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB00216 Eletriptan small molecule P28566 5-hydroxytryptamine receptor 1E approved|investigational DB00216 Eletriptan small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational DB00218 Moxifloxacin small molecule P11388 DNA topoisomerase 2-alpha approved DB00219 Oxyphenonium small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00222 Glimepiride small molecule Q09428 ATP-binding cassette sub-family C member 8 approved DB00223 Diflorasone small molecule P04150 Glucocorticoid receptor approved|investigational DB00227 Lovastatin small molecule P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase approved|investigational DB00227 Lovastatin small molecule P20701 Integrin alpha-L approved|investigational DB00227 Lovastatin small molecule Q92769 Histone deacetylase 2 approved|investigational|vet_approved DB00228 Enflurane small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational|vet_approved DB00228 Enflurane small molecule P23415 Glycine receptor subunit alpha-1 approved|investigational|vet_approved DB00228 Enflurane small molecule O15554 Intermediate conductance calcium-activated potassium channel protein 4 approved|investigational|vet_approved DB00228 Enflurane small molecule Q09470 Potassium voltage-gated channel subfamily A member 1 approved|investigational|vet_approved DB00228 Enflurane small molecule P98194 Calcium-transporting ATPase type 2C member 1 approved|investigational|vet_approved DB00228 Enflurane small molecule P42261 Glutamate receptor 1 approved|investigational|vet_approved DB00228 Enflurane small molecule P30049 ATP synthase subunit delta, mitochondrial {ECO:0000305} approved|illicit|investigational DB00230 Pregabalin small molecule O00555 Voltage-dependent P/Q-type calcium channel subunit alpha-1A approved|investigational DB00231 Temazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00231 Temazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|investigational DB00231 Temazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|investigational DB00231 Temazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|investigational DB00231 Temazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|investigational DB00231 Temazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|investigational DB00231 Temazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|investigational DB00231 Temazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|investigational DB00231 Temazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|investigational DB00231 Temazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|investigational DB00231 Temazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|investigational DB00231 Temazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|investigational DB00231 Temazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|investigational DB00231 Temazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|investigational DB00231 Temazepam small molecule P30536 Translocator protein approved|investigational DB00231 Temazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00232 Methyclothiazide small molecule Q13621 Solute carrier family 12 member 1 approved DB00232 Methyclothiazide small molecule P00915 Carbonic anhydrase 1 approved DB00232 Methyclothiazide small molecule P00918 Carbonic anhydrase 2 approved DB00232 Methyclothiazide small molecule P22748 Carbonic anhydrase 4 approved DB00233 Aminosalicylic Acid small molecule P35354 Prostaglandin G/H synthase 2 approved DB00233 Aminosalicylic Acid small molecule O15111 Inhibitor of nuclear factor kappa-B kinase subunit alpha approved DB00233 Aminosalicylic Acid small molecule P09917 Arachidonate 5-lipoxygenase approved|investigational DB00234 Reboxetine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00235 Milrinone small molecule Q14432 cGMP-inhibited 3',5'-cyclic phosphodiesterase A approved DB00239 Oxiconazole small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB00240 Alclometasone small molecule P04150 Glucocorticoid receptor approved|investigational DB00242 Cladribine small molecule P23921 Ribonucleoside-diphosphate reductase large subunit approved|investigational DB00242 Cladribine small molecule P31350 Ribonucleoside-diphosphate reductase subunit M2 approved|investigational DB00242 Cladribine small molecule Q7LG56 Ribonucleoside-diphosphate reductase subunit M2 B approved|investigational DB00242 Cladribine small molecule P09884 DNA polymerase alpha catalytic subunit approved|investigational DB00242 Cladribine small molecule Q07864 DNA polymerase epsilon catalytic subunit A approved|investigational DB00242 Cladribine small molecule P56282 DNA polymerase epsilon subunit 2 approved|investigational DB00242 Cladribine small molecule Q9NRF9 DNA polymerase epsilon subunit 3 approved|investigational DB00242 Cladribine small molecule P00491 Purine nucleoside phosphorylase approved|investigational DB00243 Ranolazine small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|investigational DB00243 Ranolazine small molecule Q15858 Sodium channel protein type 9 subunit alpha {ECO:0000305} approved DB00244 Mesalazine small molecule P35354 Prostaglandin G/H synthase 2 approved DB00244 Mesalazine small molecule P23219 Prostaglandin G/H synthase 1 approved DB00244 Mesalazine small molecule P09917 Arachidonate 5-lipoxygenase approved DB00244 Mesalazine small molecule P37231 Peroxisome proliferator-activated receptor gamma approved DB00244 Mesalazine small molecule O15111 Inhibitor of nuclear factor kappa-B kinase subunit alpha approved DB00244 Mesalazine small molecule O14920 Inhibitor of nuclear factor kappa-B kinase subunit beta approved DB00244 Mesalazine small molecule P05164 Myeloperoxidase approved DB00245 Benzatropine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00245 Benzatropine small molecule P35367 Histamine H1 receptor approved DB00246 Ziprasidone small molecule P14416 D(2) dopamine receptor approved DB00246 Ziprasidone small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00246 Ziprasidone small molecule P35462 D(3) dopamine receptor approved DB00246 Ziprasidone small molecule P21917 D(4) dopamine receptor approved DB00246 Ziprasidone small molecule P28566 5-hydroxytryptamine receptor 1E approved DB00246 Ziprasidone small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00246 Ziprasidone small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00246 Ziprasidone small molecule P35367 Histamine H1 receptor approved DB00246 Ziprasidone small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00246 Ziprasidone small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00246 Ziprasidone small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00246 Ziprasidone small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00247 Methysergide small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00247 Methysergide small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00247 Methysergide small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00247 Methysergide small molecule P28566 5-hydroxytryptamine receptor 1E approved DB00248 Cabergoline small molecule P14416 D(2) dopamine receptor approved DB00248 Cabergoline small molecule P35462 D(3) dopamine receptor approved DB00248 Cabergoline small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00248 Cabergoline small molecule P21917 D(4) dopamine receptor approved DB00248 Cabergoline small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00248 Cabergoline small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00248 Cabergoline small molecule P25100 Alpha-1D adrenergic receptor approved|vet_approved DB00252 Phenytoin small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|vet_approved DB00252 Phenytoin small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|vet_approved DB00252 Phenytoin small molecule Q07699 Sodium channel subunit beta-1 approved|vet_approved DB00252 Phenytoin small molecule Q9NY46 Sodium channel protein type 3 subunit alpha approved DB00253 Medrysone small molecule P04150 Glucocorticoid receptor approved|investigational|vet_approved DB00254 Doxycycline small molecule Q9UM07 Protein-arginine deiminase type-4 approved|investigational|vet_approved DB00254 Doxycycline small molecule P61769 Beta-2-microglobulin approved|investigational DB00255 Diethylstilbestrol small molecule P03372 Estrogen receptor approved|investigational DB00255 Diethylstilbestrol small molecule P62508 Estrogen-related receptor gamma approved|investigational DB00255 Diethylstilbestrol small molecule Q92731 Estrogen receptor beta approved|investigational DB00255 Diethylstilbestrol small molecule P11474 Steroid hormone receptor ERR1 approved|investigational DB00255 Diethylstilbestrol small molecule O95718 Steroid hormone receptor ERR2 {ECO:0000305} approved|investigational DB00255 Diethylstilbestrol small molecule Q15596 Nuclear receptor coactivator 2 approved|investigational DB00255 Diethylstilbestrol small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB00255 Diethylstilbestrol small molecule P10275 Androgen receptor approved|investigational DB00255 Diethylstilbestrol small molecule P04278 Sex hormone-binding globulin approved|vet_approved DB00257 Clotrimazole small molecule O15554 Intermediate conductance calcium-activated potassium channel protein 4 approved|vet_approved DB00257 Clotrimazole small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|vet_approved DB00257 Clotrimazole small molecule Q14994 Nuclear receptor subfamily 1 group I member 3 approved DB00261 Anagrelide small molecule Q14432 cGMP-inhibited 3',5'-cyclic phosphodiesterase A approved|investigational DB00262 Carmustine small molecule P00390 Glutathione reductase, mitochondrial approved DB00266 Dicoumarol small molecule Q9BQB6 Vitamin K epoxide reductase complex subunit 1 approved DB00266 Dicoumarol small molecule P15559 NAD(P)H dehydrogenase [quinone] 1 approved DB00266 Dicoumarol small molecule Q08257 Quinone oxidoreductase approved|investigational DB00268 Ropinirole small molecule P35462 D(3) dopamine receptor approved|investigational DB00268 Ropinirole small molecule P14416 D(2) dopamine receptor approved|investigational DB00268 Ropinirole small molecule P21917 D(4) dopamine receptor approved|investigational DB00268 Ropinirole small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB00268 Ropinirole small molecule P28335 5-hydroxytryptamine receptor 2C investigational|withdrawn DB00269 Chlorotrianisene small molecule P03372 Estrogen receptor approved|investigational DB00270 Isradipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB00270 Isradipine small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved|investigational DB00270 Isradipine small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved|investigational DB00270 Isradipine small molecule O95180 Voltage-dependent T-type calcium channel subunit alpha-1H approved|investigational DB00270 Isradipine small molecule Q9NY47 Voltage-dependent calcium channel subunit alpha-2/delta-2 approved|investigational DB00270 Isradipine small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved|investigational DB00270 Isradipine small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved DB00272 Betazole small molecule P25021 Histamine H2 receptor approved DB00273 Topiramate small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00273 Topiramate small molecule P39086 Glutamate receptor ionotropic, kainate 1 approved DB00273 Topiramate small molecule P00918 Carbonic anhydrase 2 approved DB00273 Topiramate small molecule P22748 Carbonic anhydrase 4 approved DB00273 Topiramate small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00273 Topiramate small molecule P00915 Carbonic anhydrase 1 approved DB00273 Topiramate small molecule P07451 Carbonic anhydrase 3 approved|investigational DB00275 Olmesartan small molecule P30556 Type-1 angiotensin II receptor approved|investigational DB00276 Amsacrine small molecule P11388 DNA topoisomerase 2-alpha approved|investigational DB00276 Amsacrine small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB00276 Amsacrine small molecule P02763 Alpha-1-acid glycoprotein 1 approved|investigational DB00276 Amsacrine small molecule P02768 Serum albumin approved DB00277 Theophylline small molecule P30542 Adenosine receptor A1 approved DB00277 Theophylline small molecule P29275 Adenosine receptor A2b approved DB00277 Theophylline small molecule Q07343 cAMP-specific 3',5'-cyclic phosphodiesterase 4B approved DB00277 Theophylline small molecule O76074 cGMP-specific 3',5'-cyclic phosphodiesterase approved DB00277 Theophylline small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved DB00277 Theophylline small molecule Q14432 cGMP-inhibited 3',5'-cyclic phosphodiesterase A approved DB00277 Theophylline small molecule Q92769 Histone deacetylase 2 approved DB00277 Theophylline small molecule Q99829 Copine-1 {ECO:0000305} approved DB00277 Theophylline small molecule Q8TCT9 Minor histocompatibility antigen H13 approved DB00277 Theophylline small molecule Q15155 Nodal modulator 1 approved DB00277 Theophylline small molecule P09874 Poly [ADP-ribose] polymerase 1 approved DB00277 Theophylline small molecule Q9Y4R7 Tubulin monoglycylase TTLL3 approved|investigational DB00278 Argatroban small molecule P00734 Prothrombin approved|vet_approved DB00279 Liothyronine small molecule P10827 Thyroid hormone receptor alpha approved|vet_approved DB00279 Liothyronine small molecule P10828 Thyroid hormone receptor beta approved|vet_approved DB00279 Liothyronine small molecule P12004 Proliferating cell nuclear antigen approved DB00280 Disopyramide small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB00280 Disopyramide small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00280 Disopyramide small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00280 Disopyramide small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00280 Disopyramide small molecule Q9NZV8 Potassium voltage-gated channel subfamily D member 2 approved DB00280 Disopyramide small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB00280 Disopyramide small molecule P19652 Alpha-1-acid glycoprotein 2 approved|vet_approved DB00281 Lidocaine small molecule Q15858 Sodium channel protein type 9 subunit alpha {ECO:0000305} approved|vet_approved DB00281 Lidocaine small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|vet_approved DB00281 Lidocaine small molecule P00533 Epidermal growth factor receptor approved|vet_approved DB00281 Lidocaine small molecule P35499 Sodium channel protein type 4 subunit alpha approved|vet_approved DB00281 Lidocaine small molecule P02763 Alpha-1-acid glycoprotein 1 approved|vet_approved DB00281 Lidocaine small molecule P19652 Alpha-1-acid glycoprotein 2 approved DB00282 Pamidronate small molecule P14324 Farnesyl pyrophosphate synthase approved|investigational DB00283 Clemastine small molecule P35367 Histamine H1 receptor approved|investigational DB00284 Acarbose small molecule O43451 Maltase-glucoamylase, intestinal approved|investigational DB00284 Acarbose small molecule P10253 Lysosomal alpha-glucosidase approved|investigational DB00284 Acarbose small molecule P14410 Sucrase-isomaltase, intestinal approved DB00285 Venlafaxine small molecule P31645 Sodium-dependent serotonin transporter approved DB00285 Venlafaxine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00286 Conjugated estrogens small molecule P03372 Estrogen receptor approved DB00287 Travoprost small molecule P43088 Prostaglandin F2-alpha receptor approved DB00288 Amcinonide small molecule P04150 Glucocorticoid receptor approved DB00288 Amcinonide small molecule P04083 Annexin A1 approved DB00289 Atomoxetine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00289 Atomoxetine small molecule P31645 Sodium-dependent serotonin transporter approved DB00289 Atomoxetine small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved|investigational DB00290 Bleomycin small molecule P18858 DNA ligase 1 approved|investigational DB00290 Bleomycin small molecule P49916 DNA ligase 3 approved DB00292 Etomidate small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00292 Etomidate small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00293 Raltitrexed small molecule P04818 Thymidylate synthase approved|investigational DB00293 Raltitrexed small molecule Q05932 Folylpolyglutamate synthase, mitochondrial approved|investigational DB00294 Etonogestrel small molecule P06401 Progesterone receptor approved|investigational DB00294 Etonogestrel small molecule P03372 Estrogen receptor approved|investigational DB00295 Morphine small molecule P35372 Mu-type opioid receptor approved|investigational DB00295 Morphine small molecule P41143 Delta-type opioid receptor approved|investigational DB00295 Morphine small molecule Q9Y6Y9 Lymphocyte antigen 96 approved|investigational DB00297 Bupivacaine small molecule P34995 Prostaglandin E2 receptor EP1 subtype approved DB00298 Dapiprazole small molecule P25100 Alpha-1D adrenergic receptor approved DB00302 Tranexamic Acid small molecule P00747 Plasminogen approved DB00304 Desogestrel small molecule P06401 Progesterone receptor approved DB00304 Desogestrel small molecule P03372 Estrogen receptor approved|illicit DB00306 Talbutal small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB00306 Talbutal small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB00306 Talbutal small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB00306 Talbutal small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB00306 Talbutal small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|illicit DB00306 Talbutal small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|illicit DB00306 Talbutal small molecule P42262 Glutamate receptor 2 approved|illicit DB00306 Talbutal small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved|illicit DB00306 Talbutal small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00307 Bexarotene small molecule P19793 Retinoic acid receptor RXR-alpha approved|investigational DB00307 Bexarotene small molecule P28702 Retinoic acid receptor RXR-beta approved|investigational DB00307 Bexarotene small molecule P48443 Retinoic acid receptor RXR-gamma approved DB00308 Ibutilide small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved DB00308 Ibutilide small molecule Q02641 Voltage-dependent L-type calcium channel subunit beta-1 approved DB00308 Ibutilide small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB00308 Ibutilide small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved DB00308 Ibutilide small molecule Q06432 Voltage-dependent calcium channel gamma-1 subunit approved DB00308 Ibutilide small molecule O00180 Potassium channel subfamily K member 1 approved DB00308 Ibutilide small molecule Q9Y257 Potassium channel subfamily K member 6 approved DB00308 Ibutilide small molecule Q9NS40 Potassium voltage-gated channel subfamily H member 7 approved DB00310 Chlorthalidone small molecule Q13621 Solute carrier family 12 member 1 approved|investigational|vet_approved DB00312 Pentobarbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational|vet_approved DB00312 Pentobarbital small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|investigational|vet_approved DB00312 Pentobarbital small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|investigational|vet_approved DB00312 Pentobarbital small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|investigational|vet_approved DB00312 Pentobarbital small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|investigational|vet_approved DB00312 Pentobarbital small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|investigational|vet_approved DB00312 Pentobarbital small molecule P42262 Glutamate receptor 2 approved|investigational|vet_approved DB00312 Pentobarbital small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved|investigational|vet_approved DB00312 Pentobarbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational|vet_approved DB00312 Pentobarbital small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved|investigational|vet_approved DB00312 Pentobarbital small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB00313 Valproic Acid small molecule Q9UKV0 Histone deacetylase 9 approved|investigational DB00313 Valproic Acid small molecule P80404 4-aminobutyrate aminotransferase, mitochondrial approved|investigational DB00313 Valproic Acid small molecule P45954 Short/branched chain specific acyl-CoA dehydrogenase, mitochondrial approved|investigational DB00313 Valproic Acid small molecule Q02218 2-oxoglutarate dehydrogenase, mitochondrial approved|investigational DB00313 Valproic Acid small molecule P51649 Succinate-semialdehyde dehydrogenase, mitochondrial approved|investigational DB00313 Valproic Acid small molecule Q92769 Histone deacetylase 2 approved|investigational DB00313 Valproic Acid small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved|investigational DB00313 Valproic Acid small molecule Q03181 Peroxisome proliferator-activated receptor delta approved|investigational DB00313 Valproic Acid small molecule P37231 Peroxisome proliferator-activated receptor gamma approved DB00316 Acetaminophen small molecule P23219 Prostaglandin G/H synthase 1 approved DB00316 Acetaminophen small molecule P35354 Prostaglandin G/H synthase 2 approved DB00316 Acetaminophen small molecule O00519 Fatty-acid amide hydrolase 1 approved DB00316 Acetaminophen small molecule Q8NER1 Transient receptor potential cation channel subfamily V member 1 approved DB00316 Acetaminophen small molecule P09211 Glutathione S-transferase P approved|investigational DB00317 Gefitinib small molecule P00533 Epidermal growth factor receptor approved|illicit DB00318 Codeine small molecule P35372 Mu-type opioid receptor approved|illicit DB00318 Codeine small molecule P41143 Delta-type opioid receptor approved DB00321 Amitriptyline small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00321 Amitriptyline small molecule P31645 Sodium-dependent serotonin transporter approved DB00321 Amitriptyline small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00321 Amitriptyline small molecule P41143 Delta-type opioid receptor approved DB00321 Amitriptyline small molecule P04629 High affinity nerve growth factor receptor approved DB00321 Amitriptyline small molecule Q16620 BDNF/NT-3 growth factors receptor approved DB00321 Amitriptyline small molecule P25100 Alpha-1D adrenergic receptor approved DB00321 Amitriptyline small molecule P35367 Histamine H1 receptor approved DB00321 Amitriptyline small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00321 Amitriptyline small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00321 Amitriptyline small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00321 Amitriptyline small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00321 Amitriptyline small molecule O43526 Potassium voltage-gated channel subfamily KQT member 2 {ECO:0000305} approved DB00321 Amitriptyline small molecule Q09470 Potassium voltage-gated channel subfamily A member 1 approved DB00321 Amitriptyline small molecule Q9NZV8 Potassium voltage-gated channel subfamily D member 2 approved DB00321 Amitriptyline small molecule P25021 Histamine H2 receptor approved DB00321 Amitriptyline small molecule Q9H3N8 Histamine H4 receptor approved DB00321 Amitriptyline small molecule Q99720 Sigma non-opioid intracellular receptor 1 approved DB00321 Amitriptyline small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00321 Amitriptyline small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00321 Amitriptyline small molecule P35372 Mu-type opioid receptor approved DB00321 Amitriptyline small molecule O43525 Potassium voltage-gated channel subfamily KQT member 3 {ECO:0000305} approved|withdrawn DB00323 Tolcapone small molecule P21964 Catechol O-methyltransferase approved|investigational DB00324 Fluorometholone small molecule P04150 Glucocorticoid receptor approved|illicit DB00327 Hydromorphone small molecule P35372 Mu-type opioid receptor approved|illicit DB00327 Hydromorphone small molecule P41143 Delta-type opioid receptor approved|investigational DB00328 Indomethacin small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB00328 Indomethacin small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB00328 Indomethacin small molecule P14555 Phospholipase A2, membrane associated approved|investigational DB00328 Indomethacin small molecule Q8N8N7 Prostaglandin reductase 2 approved|investigational DB00328 Indomethacin small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|investigational DB00328 Indomethacin small molecule Q04760 Lactoylglutathione lyase approved|investigational DB00328 Indomethacin small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved|investigational DB00328 Indomethacin small molecule P42330 Aldo-keto reductase family 1 member C3 approved DB00331 Metformin small molecule Q9Y478 5'-AMP-activated protein kinase subunit beta-1 approved DB00332 Ipratropium bromide small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00332 Ipratropium bromide small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00332 Ipratropium bromide small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00333 Methadone small molecule P35372 Mu-type opioid receptor approved DB00333 Methadone small molecule P41143 Delta-type opioid receptor approved DB00333 Methadone small molecule Q9Y6Y9 Lymphocyte antigen 96 approved DB00333 Methadone small molecule P19652 Alpha-1-acid glycoprotein 2 approved|investigational DB00334 Olanzapine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB00334 Olanzapine small molecule P14416 D(2) dopamine receptor approved|investigational DB00334 Olanzapine small molecule P35462 D(3) dopamine receptor approved|investigational DB00334 Olanzapine small molecule P21917 D(4) dopamine receptor approved|investigational DB00334 Olanzapine small molecule P28566 5-hydroxytryptamine receptor 1E approved|investigational DB00334 Olanzapine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB00334 Olanzapine small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational DB00334 Olanzapine small molecule P35367 Histamine H1 receptor approved|investigational DB00334 Olanzapine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00334 Olanzapine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00334 Olanzapine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB00334 Olanzapine small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB00334 Olanzapine small molecule P25021 Histamine H2 receptor approved|investigational DB00334 Olanzapine small molecule Q9H3N8 Histamine H4 receptor approved|investigational DB00334 Olanzapine small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00337 Pimecrolimus small molecule P42345 Serine/threonine-protein kinase mTOR approved|investigational DB00337 Pimecrolimus small molecule P62942 Peptidyl-prolyl cis-trans isomerase FKBP1A approved|investigational|vet_approved DB00338 Omeprazole small molecule P20648 Potassium-transporting ATPase alpha chain 1 approved|investigational|vet_approved DB00338 Omeprazole small molecule P35869 Aryl hydrocarbon receptor approved DB00340 Metixene small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00340 Metixene small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00340 Metixene small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00340 Metixene small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00341 Cetirizine small molecule P35367 Histamine H1 receptor approved|withdrawn DB00342 Terfenadine small molecule P35367 Histamine H1 receptor approved|withdrawn DB00342 Terfenadine small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|withdrawn DB00342 Terfenadine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|withdrawn DB00342 Terfenadine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|withdrawn DB00342 Terfenadine small molecule P08173 Muscarinic acetylcholine receptor M4 approved|withdrawn DB00342 Terfenadine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00343 Diltiazem small molecule Q06432 Voltage-dependent calcium channel gamma-1 subunit approved DB00344 Protriptyline small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00344 Protriptyline small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB00346 Alfuzosin small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB00346 Alfuzosin small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB00347 Trimethadione small molecule O43497 Voltage-dependent T-type calcium channel subunit alpha-1G approved|investigational DB00348 Nitisinone small molecule P32754 4-hydroxyphenylpyruvate dioxygenase approved|illicit DB00349 Clobazam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00350 Minoxidil small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB00350 Minoxidil small molecule P00797 Renin approved|investigational|vet_approved DB00351 Megestrol acetate small molecule P06401 Progesterone receptor approved|investigational|vet_approved DB00351 Megestrol acetate small molecule P04150 Glucocorticoid receptor approved DB00354 Buclizine small molecule P35367 Histamine H1 receptor approved DB00354 Buclizine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00356 Chlorzoxazone small molecule Q12791 Calcium-activated potassium channel subunit alpha-1 approved|investigational DB00357 Aminoglutethimide small molecule P11511 Aromatase approved|investigational DB00357 Aminoglutethimide small molecule P05108 Cholesterol side-chain cleavage enzyme, mitochondrial approved|investigational DB00358 Mefloquine small molecule P69905 Hemoglobin subunit alpha approved|investigational DB00360 Sapropterin small molecule P00439 Phenylalanine-4-hydroxylase approved|investigational DB00360 Sapropterin small molecule P29474 Nitric oxide synthase, endothelial approved|investigational DB00360 Sapropterin small molecule P07101 Tyrosine 3-monooxygenase approved|investigational DB00360 Sapropterin small molecule P17752 Tryptophan 5-hydroxylase 1 approved|investigational DB00361 Vinorelbine small molecule P07437 Tubulin beta chain approved DB00363 Clozapine small molecule P14416 D(2) dopamine receptor approved DB00363 Clozapine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00363 Clozapine small molecule P35462 D(3) dopamine receptor approved DB00363 Clozapine small molecule P21917 D(4) dopamine receptor approved DB00363 Clozapine small molecule P28566 5-hydroxytryptamine receptor 1E approved DB00363 Clozapine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00363 Clozapine small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00363 Clozapine small molecule P35367 Histamine H1 receptor approved DB00363 Clozapine small molecule Q9H3N8 Histamine H4 receptor approved DB00363 Clozapine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00363 Clozapine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00363 Clozapine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00363 Clozapine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00363 Clozapine small molecule P09211 Glutathione S-transferase P approved DB00364 Sucralfate small molecule P09038 Fibroblast growth factor 2 approved DB00364 Sucralfate small molecule P01133 Pro-epidermal growth factor approved DB00364 Sucralfate small molecule P02671 Fibrinogen alpha chain approved DB00364 Sucralfate small molecule P02675 Fibrinogen beta chain approved DB00364 Sucralfate small molecule P02679 Fibrinogen gamma chain approved|vet_approved DB00366 Doxylamine small molecule P35367 Histamine H1 receptor approved|vet_approved DB00366 Doxylamine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|vet_approved DB00366 Doxylamine small molecule Q14994 Nuclear receptor subfamily 1 group I member 3 approved|investigational DB00367 Levonorgestrel small molecule P06401 Progesterone receptor approved|investigational DB00367 Levonorgestrel small molecule P18405 3-oxo-5-alpha-steroid 4-dehydrogenase 1 approved|investigational DB00367 Levonorgestrel small molecule P03372 Estrogen receptor approved|investigational DB00367 Levonorgestrel small molecule P10275 Androgen receptor approved|investigational DB00367 Levonorgestrel small molecule P04278 Sex hormone-binding globulin approved DB00368 Norepinephrine small molecule P25100 Alpha-1D adrenergic receptor approved DB00368 Norepinephrine small molecule P13945 Beta-3 adrenergic receptor approved DB00368 Norepinephrine small molecule P00439 Phenylalanine-4-hydroxylase approved DB00368 Norepinephrine small molecule Q05940 Synaptic vesicular amine transporter approved DB00370 Mirtazapine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00370 Mirtazapine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00370 Mirtazapine small molecule P35367 Histamine H1 receptor approved DB00370 Mirtazapine small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00370 Mirtazapine small molecule P14416 D(2) dopamine receptor approved DB00370 Mirtazapine small molecule P35462 D(3) dopamine receptor approved DB00370 Mirtazapine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00370 Mirtazapine small molecule P31645 Sodium-dependent serotonin transporter approved DB00370 Mirtazapine small molecule Q9Y5N1 Histamine H3 receptor approved|illicit DB00371 Meprobamate small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB00371 Meprobamate small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB00371 Meprobamate small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB00371 Meprobamate small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB00371 Meprobamate small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 withdrawn DB00372 Thiethylperazine small molecule P14416 D(2) dopamine receptor withdrawn DB00372 Thiethylperazine small molecule P21917 D(4) dopamine receptor approved|investigational DB00374 Treprostinil small molecule Q03181 Peroxisome proliferator-activated receptor delta approved|investigational DB00374 Treprostinil small molecule Q9H244 P2Y purinoceptor 12 approved DB00376 Trihexyphenidyl small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00376 Trihexyphenidyl small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00376 Trihexyphenidyl small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00376 Trihexyphenidyl small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational|withdrawn DB00378 Dydrogesterone small molecule P06401 Progesterone receptor approved|investigational DB00379 Mexiletine small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|investigational DB00379 Mexiletine small molecule P35869 Aryl hydrocarbon receptor approved|withdrawn DB00380 Dexrazoxane small molecule P11388 DNA topoisomerase 2-alpha approved|withdrawn DB00380 Dexrazoxane small molecule Q02880 DNA topoisomerase 2-beta approved DB00381 Amlodipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved DB00381 Amlodipine small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved DB00381 Amlodipine small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved DB00381 Amlodipine small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved DB00381 Amlodipine small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved DB00381 Amlodipine small molecule Q00975 Voltage-dependent N-type calcium channel subunit alpha-1B approved DB00381 Amlodipine small molecule Q8IZS8 Voltage-dependent calcium channel subunit alpha-2/delta-3 approved DB00381 Amlodipine small molecule P00915 Carbonic anhydrase 1 approved DB00381 Amlodipine small molecule P17405 Sphingomyelin phosphodiesterase investigational|withdrawn DB00382 Tacrine small molecule P22303 Acetylcholinesterase investigational|withdrawn DB00382 Tacrine small molecule P06276 Cholinesterase investigational|withdrawn DB00382 Tacrine small molecule P23141 Liver carboxylesterase 1 approved DB00383 Oxyphencyclimine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00383 Oxyphencyclimine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00383 Oxyphencyclimine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00384 Triamterene small molecule P51170 Amiloride-sensitive sodium channel subunit gamma approved DB00384 Triamterene small molecule P37088 Amiloride-sensitive sodium channel subunit alpha approved DB00384 Triamterene small molecule P51168 Amiloride-sensitive sodium channel subunit beta approved DB00384 Triamterene small molecule P51172 Amiloride-sensitive sodium channel subunit delta approved DB00385 Valrubicin small molecule P11388 DNA topoisomerase 2-alpha approved DB00387 Procyclidine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00387 Procyclidine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00387 Procyclidine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00387 Procyclidine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00388 Phenylephrine small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB00389 Carbimazole small molecule P07202 Thyroid peroxidase {ECO:0000305} approved DB00390 Digoxin small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved|investigational DB00391 Sulpiride small molecule P14416 D(2) dopamine receptor approved|investigational DB00391 Sulpiride small molecule P35462 D(3) dopamine receptor approved|investigational DB00391 Sulpiride small molecule P00918 Carbonic anhydrase 2 approved|investigational DB00391 Sulpiride small molecule P07451 Carbonic anhydrase 3 approved DB00392 Ethopropazine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00392 Ethopropazine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00393 Nimodipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB00393 Nimodipine small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved|investigational DB00393 Nimodipine small molecule O60840 Voltage-dependent L-type calcium channel subunit alpha-1F {ECO:0000305} approved|investigational DB00393 Nimodipine small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved|investigational DB00393 Nimodipine small molecule Q02641 Voltage-dependent L-type calcium channel subunit beta-1 approved|investigational DB00393 Nimodipine small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved|investigational DB00393 Nimodipine small molecule P54284 Voltage-dependent L-type calcium channel subunit beta-3 approved|investigational DB00393 Nimodipine small molecule O00305 Voltage-dependent L-type calcium channel subunit beta-4 {ECO:0000305} approved|investigational DB00393 Nimodipine small molecule P08235 Mineralocorticoid receptor approved|investigational DB00393 Nimodipine small molecule P35869 Aryl hydrocarbon receptor approved|investigational DB00394 Beclomethasone dipropionate small molecule P04150 Glucocorticoid receptor approved DB00395 Carisoprodol small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00395 Carisoprodol small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|vet_approved DB00396 Progesterone small molecule P06401 Progesterone receptor approved|vet_approved DB00396 Progesterone small molecule P03372 Estrogen receptor approved|vet_approved DB00396 Progesterone small molecule P08235 Mineralocorticoid receptor approved|vet_approved DB00396 Progesterone small molecule P05093 Steroid 17-alpha-hydroxylase/17,20 lyase approved|vet_approved DB00396 Progesterone small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|vet_approved DB00396 Progesterone small molecule P02763 Alpha-1-acid glycoprotein 1 approved|vet_approved DB00396 Progesterone small molecule P04150 Glucocorticoid receptor approved|vet_approved DB00396 Progesterone small molecule P10275 Androgen receptor approved|vet_approved DB00396 Progesterone small molecule P04278 Sex hormone-binding globulin approved|investigational DB00398 Sorafenib small molecule P15056 Serine/threonine-protein kinase B-raf approved|investigational DB00398 Sorafenib small molecule P04049 RAF proto-oncogene serine/threonine-protein kinase approved|investigational DB00398 Sorafenib small molecule P35916 Vascular endothelial growth factor receptor 3 approved|investigational DB00398 Sorafenib small molecule P36888 Receptor-type tyrosine-protein kinase FLT3 approved|investigational DB00398 Sorafenib small molecule P09619 Platelet-derived growth factor receptor beta approved|investigational DB00398 Sorafenib small molecule P10721 Mast/stem cell growth factor receptor Kit approved|investigational DB00398 Sorafenib small molecule P11362 Fibroblast growth factor receptor 1 approved|investigational DB00398 Sorafenib small molecule P07949 Proto-oncogene tyrosine-protein kinase receptor Ret {ECO:0000305} approved|investigational DB00398 Sorafenib small molecule P17948 Vascular endothelial growth factor receptor 1 approved DB00399 Zoledronic acid small molecule P14324 Farnesyl pyrophosphate synthase approved DB00399 Zoledronic acid small molecule O95749 Geranylgeranyl pyrophosphate synthase approved|investigational|vet_approved DB00400 Griseofulvin small molecule Q99456 Keratin, type I cytoskeletal 12 approved DB00401 Nisoldipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved DB00401 Nisoldipine small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved DB00401 Nisoldipine small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved DB00401 Nisoldipine small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved DB00401 Nisoldipine small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved|investigational DB00402 Eszopiclone small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00402 Eszopiclone small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|investigational DB00402 Eszopiclone small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|investigational DB00402 Eszopiclone small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|investigational DB00402 Eszopiclone small molecule P30536 Translocator protein approved|investigational DB00402 Eszopiclone small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00403 Ceruletide small molecule P32238 Cholecystokinin receptor type A approved|illicit|investigational DB00404 Alprazolam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00405 Dexbrompheniramine small molecule P35367 Histamine H1 receptor approved DB00408 Loxapine small molecule P14416 D(2) dopamine receptor approved DB00408 Loxapine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00408 Loxapine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00408 Loxapine small molecule P28566 5-hydroxytryptamine receptor 1E approved DB00408 Loxapine small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00408 Loxapine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00408 Loxapine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00408 Loxapine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00408 Loxapine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00408 Loxapine small molecule P35462 D(3) dopamine receptor approved DB00408 Loxapine small molecule P21917 D(4) dopamine receptor approved DB00408 Loxapine small molecule P35367 Histamine H1 receptor approved DB00408 Loxapine small molecule P25021 Histamine H2 receptor approved DB00408 Loxapine small molecule Q9H3N8 Histamine H4 receptor approved DB00408 Loxapine small molecule P31645 Sodium-dependent serotonin transporter approved DB00408 Loxapine small molecule P23975 Sodium-dependent noradrenaline transporter approved|withdrawn DB00409 Remoxipride small molecule P14416 D(2) dopamine receptor approved|withdrawn DB00409 Remoxipride small molecule P21917 D(4) dopamine receptor approved|withdrawn DB00409 Remoxipride small molecule P35462 D(3) dopamine receptor approved|withdrawn DB00409 Remoxipride small molecule P28223 5-hydroxytryptamine receptor 2A approved|withdrawn DB00409 Remoxipride small molecule Q99720 Sigma non-opioid intracellular receptor 1 approved DB00411 Carbachol small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00411 Carbachol small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00411 Carbachol small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB00411 Carbachol small molecule P22303 Acetylcholinesterase approved DB00411 Carbachol small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00411 Carbachol small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB00412 Rosiglitazone small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|investigational DB00412 Rosiglitazone small molecule O60488 Long-chain-fatty-acid--CoA ligase 4 approved|investigational DB00412 Rosiglitazone small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved|investigational DB00412 Rosiglitazone small molecule Q03181 Peroxisome proliferator-activated receptor delta approved|investigational DB00412 Rosiglitazone small molecule P19793 Retinoic acid receptor RXR-alpha approved|investigational DB00412 Rosiglitazone small molecule P28702 Retinoic acid receptor RXR-beta approved|investigational DB00412 Rosiglitazone small molecule P48443 Retinoic acid receptor RXR-gamma approved|investigational DB00413 Pramipexole small molecule P35462 D(3) dopamine receptor approved|investigational DB00413 Pramipexole small molecule P14416 D(2) dopamine receptor approved|investigational DB00413 Pramipexole small molecule P21917 D(4) dopamine receptor approved|investigational DB00413 Pramipexole small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB00413 Pramipexole small molecule P28335 5-hydroxytryptamine receptor 2C approved|vet_approved DB00415 Ampicillin small molecule P46059 Solute carrier family 15 member 1 approved|vet_approved DB00415 Ampicillin small molecule Q02763 Angiopoietin-1 receptor approved|vet_approved DB00417 Phenoxymethylpenicillin small molecule P46059 Solute carrier family 15 member 1 approved|vet_approved DB00418 Secobarbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|vet_approved DB00418 Secobarbital small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|vet_approved DB00418 Secobarbital small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|vet_approved DB00418 Secobarbital small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|vet_approved DB00418 Secobarbital small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|vet_approved DB00418 Secobarbital small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|vet_approved DB00418 Secobarbital small molecule P42262 Glutamate receptor 2 approved|vet_approved DB00418 Secobarbital small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved|vet_approved DB00418 Secobarbital small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved DB00419 Miglustat small molecule Q16739 Ceramide glucosyltransferase approved|vet_approved DB00420 Promazine small molecule P14416 D(2) dopamine receptor approved|vet_approved DB00420 Promazine small molecule P28223 5-hydroxytryptamine receptor 2A approved|vet_approved DB00420 Promazine small molecule P28335 5-hydroxytryptamine receptor 2C approved|vet_approved DB00420 Promazine small molecule P21917 D(4) dopamine receptor approved|vet_approved DB00420 Promazine small molecule P08173 Muscarinic acetylcholine receptor M4 approved|vet_approved DB00420 Promazine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|vet_approved DB00420 Promazine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|vet_approved DB00420 Promazine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|vet_approved DB00420 Promazine small molecule P35367 Histamine H1 receptor approved|vet_approved DB00420 Promazine small molecule P25100 Alpha-1D adrenergic receptor approved DB00421 Spironolactone small molecule P08235 Mineralocorticoid receptor approved DB00421 Spironolactone small molecule P10275 Androgen receptor approved DB00421 Spironolactone small molecule P06401 Progesterone receptor approved DB00421 Spironolactone small molecule P04150 Glucocorticoid receptor approved DB00421 Spironolactone small molecule P18405 3-oxo-5-alpha-steroid 4-dehydrogenase 1 approved DB00421 Spironolactone small molecule P04278 Sex hormone-binding globulin approved DB00421 Spironolactone small molecule Q06432 Voltage-dependent calcium channel gamma-1 subunit approved DB00421 Spironolactone small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB00422 Methylphenidate small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB00422 Methylphenidate small molecule P31645 Sodium-dependent serotonin transporter approved|vet_approved DB00423 Methocarbamol small molecule P00915 Carbonic anhydrase 1 approved DB00424 Hyoscyamine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00424 Hyoscyamine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00424 Hyoscyamine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00424 Hyoscyamine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00425 Zolpidem small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00425 Zolpidem small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB00425 Zolpidem small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB00425 Zolpidem small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved DB00425 Zolpidem small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved DB00427 Triprolidine small molecule P35367 Histamine H1 receptor approved|investigational DB00428 Streptozocin small molecule P11168 Solute carrier family 2, facilitated glucose transporter member 2 approved|investigational DB00428 Streptozocin small molecule O60502 Protein O-GlcNAcase {ECO:0000303|PubMed:11148210, ECO:0000303|PubMed:11788610} approved DB00429 Carboprost Tromethamine small molecule P34995 Prostaglandin E2 receptor EP1 subtype approved|withdrawn DB00431 Lindane small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|withdrawn DB00431 Lindane small molecule P23415 Glycine receptor subunit alpha-1 approved|withdrawn DB00431 Lindane small molecule P23416 Glycine receptor subunit alpha-2 approved|withdrawn DB00431 Lindane small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|withdrawn DB00431 Lindane small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|withdrawn DB00431 Lindane small molecule P06401 Progesterone receptor approved|withdrawn DB00431 Lindane small molecule P03372 Estrogen receptor approved|withdrawn DB00431 Lindane small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB00432 Trifluridine small molecule P04818 Thymidylate synthase approved|vet_approved DB00433 Prochlorperazine small molecule P14416 D(2) dopamine receptor approved DB00434 Cyproheptadine small molecule P35367 Histamine H1 receptor approved DB00434 Cyproheptadine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00434 Cyproheptadine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00434 Cyproheptadine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00434 Cyproheptadine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00434 Cyproheptadine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00434 Cyproheptadine small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00435 Nitric Oxide small molecule P33402 Guanylate cyclase soluble subunit alpha-2 approved DB00435 Nitric Oxide small molecule P04731 Metallothionein-1A approved DB00435 Nitric Oxide small molecule P14902 Indoleamine 2,3-dioxygenase 1 approved DB00436 Bendroflumethiazide small molecule P55017 Solute carrier family 12 member 3 approved DB00436 Bendroflumethiazide small molecule Q12791 Calcium-activated potassium channel subunit alpha-1 approved DB00436 Bendroflumethiazide small molecule P00915 Carbonic anhydrase 1 approved DB00436 Bendroflumethiazide small molecule P00918 Carbonic anhydrase 2 approved DB00436 Bendroflumethiazide small molecule P22748 Carbonic anhydrase 4 approved|withdrawn DB00439 Cerivastatin small molecule P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase approved|vet_approved DB00440 Trimethoprim small molecule P04818 Thymidylate synthase approved|vet_approved DB00440 Trimethoprim small molecule P00374 Dihydrofolate reductase approved DB00441 Gemcitabine small molecule P23921 Ribonucleoside-diphosphate reductase large subunit approved DB00441 Gemcitabine small molecule P04818 Thymidylate synthase approved DB00441 Gemcitabine small molecule P30085 UMP-CMP kinase {ECO:0000255|HAMAP-Rule:MF_03172} approved|vet_approved DB00443 Betamethasone small molecule P04150 Glucocorticoid receptor approved DB00444 Teniposide small molecule P11388 DNA topoisomerase 2-alpha approved DB00445 Epirubicin small molecule O14646 Chromodomain-helicase-DNA-binding protein 1 approved DB00445 Epirubicin small molecule P11388 DNA topoisomerase 2-alpha approved|vet_approved DB00446 Chloramphenicol small molecule P08174 Complement decay-accelerating factor approved|investigational DB00448 Lansoprazole small molecule P20648 Potassium-transporting ATPase alpha chain 1 approved|investigational DB00448 Lansoprazole small molecule P10636 Microtubule-associated protein tau approved DB00449 Dipivefrin small molecule P06276 Cholinesterase approved DB00449 Dipivefrin small molecule P22303 Acetylcholinesterase approved|vet_approved DB00450 Droperidol small molecule P14416 D(2) dopamine receptor approved DB00451 Levothyroxine small molecule P10827 Thyroid hormone receptor alpha approved DB00451 Levothyroxine small molecule P10828 Thyroid hormone receptor beta approved DB00452 Framycetin small molecule P61073 C-X-C chemokine receptor type 4 approved DB00454 Pethidine small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved DB00454 Pethidine small molecule Q13224 Glutamate receptor ionotropic, NMDA 2B approved DB00454 Pethidine small molecule Q12879 Glutamate receptor ionotropic, NMDA 2A approved DB00454 Pethidine small molecule O15399 Glutamate receptor ionotropic, NMDA 2D approved DB00454 Pethidine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00454 Pethidine small molecule P35372 Mu-type opioid receptor approved DB00454 Pethidine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00454 Pethidine small molecule P31645 Sodium-dependent serotonin transporter approved DB00454 Pethidine small molecule P23141 Liver carboxylesterase 1 approved|investigational DB00455 Loratadine small molecule P35367 Histamine H1 receptor approved|investigational DB00455 Loratadine small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB00457 Prazosin small molecule P25100 Alpha-1D adrenergic receptor approved DB00457 Prazosin small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB00457 Prazosin small molecule Q9NS40 Potassium voltage-gated channel subfamily H member 7 approved DB00458 Imipramine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00458 Imipramine small molecule P31645 Sodium-dependent serotonin transporter approved DB00458 Imipramine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00458 Imipramine small molecule P35367 Histamine H1 receptor approved DB00458 Imipramine small molecule P25100 Alpha-1D adrenergic receptor approved DB00458 Imipramine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00458 Imipramine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00458 Imipramine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00458 Imipramine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00458 Imipramine small molecule Q9NZV8 Potassium voltage-gated channel subfamily D member 2 approved DB00458 Imipramine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00458 Imipramine small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00458 Imipramine small molecule P14416 D(2) dopamine receptor approved DB00458 Imipramine small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB00458 Imipramine small molecule O95259 Potassium voltage-gated channel subfamily H member 1 approved DB00458 Imipramine small molecule P19652 Alpha-1-acid glycoprotein 2 approved DB00459 Acitretin small molecule P19793 Retinoic acid receptor RXR-alpha approved DB00459 Acitretin small molecule P10276 Retinoic acid receptor alpha approved DB00459 Acitretin small molecule P10826 Retinoic acid receptor beta approved DB00459 Acitretin small molecule P13631 Retinoic acid receptor gamma approved DB00459 Acitretin small molecule P28702 Retinoic acid receptor RXR-beta approved DB00459 Acitretin small molecule P48443 Retinoic acid receptor RXR-gamma approved DB00459 Acitretin small molecule P09455 Retinol-binding protein 1 approved DB00461 Nabumetone small molecule P35354 Prostaglandin G/H synthase 2 approved DB00461 Nabumetone small molecule P23219 Prostaglandin G/H synthase 1 withdrawn DB00463 Metharbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 withdrawn DB00463 Metharbital small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 withdrawn DB00463 Metharbital small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 withdrawn DB00463 Metharbital small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 withdrawn DB00463 Metharbital small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 withdrawn DB00463 Metharbital small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 withdrawn DB00463 Metharbital small molecule P42262 Glutamate receptor 2 withdrawn DB00463 Metharbital small molecule Q13002 Glutamate receptor ionotropic, kainate 2 withdrawn DB00463 Metharbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00464 Sodium Tetradecyl Sulfate small molecule P07225 Vitamin K-dependent protein S approved DB00465 Ketorolac small molecule P35354 Prostaglandin G/H synthase 2 approved DB00465 Ketorolac small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB00467 Enoxacin small molecule P11388 DNA topoisomerase 2-alpha approved DB00468 Quinine small molecule O15554 Intermediate conductance calcium-activated potassium channel protein 4 approved DB00469 Tenoxicam small molecule P35354 Prostaglandin G/H synthase 2 approved DB00469 Tenoxicam small molecule P23219 Prostaglandin G/H synthase 1 approved|illicit DB00470 Dronabinol small molecule P34972 Cannabinoid receptor 2 approved DB00471 Montelukast small molecule Q9Y271 Cysteinyl leukotriene receptor 1 approved DB00471 Montelukast small molecule P09917 Arachidonate 5-lipoxygenase approved|vet_approved DB00472 Fluoxetine small molecule P31645 Sodium-dependent serotonin transporter approved|vet_approved DB00472 Fluoxetine small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|vet_approved DB00472 Fluoxetine small molecule P28335 5-hydroxytryptamine receptor 2C approved|vet_approved DB00472 Fluoxetine small molecule P61024 Cyclin-dependent kinases regulatory subunit 1 approved DB00474 Methohexital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit|investigational DB00475 Chlordiazepoxide small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00476 Duloxetine small molecule P31645 Sodium-dependent serotonin transporter approved DB00476 Duloxetine small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P14416 D(2) dopamine receptor approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P35367 Histamine H1 receptor approved|investigational|vet_approved DB00477 Chlorpromazine small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P35462 D(3) dopamine receptor approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P21917 D(4) dopamine receptor approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P17405 Sphingomyelin phosphodiesterase approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P02763 Alpha-1-acid glycoprotein 1 approved|investigational|vet_approved DB00477 Chlorpromazine small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational|vet_approved DB00477 Chlorpromazine small molecule Q9H3N8 Histamine H4 receptor approved DB00480 Lenalidomide small molecule Q96SW2 Protein cereblon approved DB00480 Lenalidomide small molecule O14788 Tumor necrosis factor ligand superfamily member 11 approved DB00480 Lenalidomide small molecule P33151 Cadherin-5 approved DB00480 Lenalidomide small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB00481 Raloxifene small molecule P03372 Estrogen receptor approved|investigational DB00481 Raloxifene small molecule Q92731 Estrogen receptor beta approved|investigational DB00481 Raloxifene small molecule P04155 Trefoil factor 1 approved|investigational DB00482 Celecoxib small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB00482 Celecoxib small molecule O15530 3-phosphoinositide-dependent protein kinase 1 approved|investigational DB00482 Celecoxib small molecule P00918 Carbonic anhydrase 2 approved|investigational DB00482 Celecoxib small molecule P07451 Carbonic anhydrase 3 approved|investigational DB00486 Nabilone small molecule P34972 Cannabinoid receptor 2 approved DB00487 Pefloxacin small molecule P11388 DNA topoisomerase 2-alpha approved DB00489 Sotalol small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB00490 Buspirone small molecule P14416 D(2) dopamine receptor approved DB00491 Miglitol small molecule O43451 Maltase-glucoamylase, intestinal approved DB00491 Miglitol small molecule P10253 Lysosomal alpha-glucosidase approved DB00491 Miglitol small molecule Q14697 Neutral alpha-glucosidase AB approved DB00491 Miglitol small molecule Q8TET4 Neutral alpha-glucosidase C approved DB00492 Fosinopril small molecule P12821 Angiotensin-converting enzyme approved DB00493 Cefotaxime small molecule Q4U2R8 Solute carrier family 22 member 6 approved DB00493 Cefotaxime small molecule Q8TCC7 Solute carrier family 22 member 8 approved DB00493 Cefotaxime small molecule Q9NSA0 Solute carrier family 22 member 11 approved DB00493 Cefotaxime small molecule Q9Y694 Solute carrier family 22 member 7 approved DB00493 Cefotaxime small molecule P46059 Solute carrier family 15 member 1 approved DB00493 Cefotaxime small molecule P02768 Serum albumin approved|investigational DB00494 Entacapone small molecule P21964 Catechol O-methyltransferase approved DB00495 Zidovudine small molecule O14746 Telomerase reverse transcriptase approved|investigational DB00496 Darifenacin small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB00496 Darifenacin small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00496 Darifenacin small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00496 Darifenacin small molecule P08173 Muscarinic acetylcholine receptor M4 approved|illicit|investigational DB00497 Oxycodone small molecule P35372 Mu-type opioid receptor approved|illicit|investigational DB00497 Oxycodone small molecule P41143 Delta-type opioid receptor approved|illicit|investigational DB00497 Oxycodone small molecule P02763 Alpha-1-acid glycoprotein 1 approved|investigational DB00498 Phenindione small molecule Q9BQB6 Vitamin K epoxide reductase complex subunit 1 approved|investigational DB00499 Flutamide small molecule P10275 Androgen receptor approved|investigational DB00499 Flutamide small molecule P35869 Aryl hydrocarbon receptor approved|investigational DB00499 Flutamide small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB00500 Tolmetin small molecule P35354 Prostaglandin G/H synthase 2 approved DB00500 Tolmetin small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB00501 Cimetidine small molecule P25021 Histamine H2 receptor approved DB00502 Haloperidol small molecule P14416 D(2) dopamine receptor approved DB00502 Haloperidol small molecule Q13224 Glutamate receptor ionotropic, NMDA 2B approved DB00502 Haloperidol small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00502 Haloperidol small molecule P35462 D(3) dopamine receptor approved DB00502 Haloperidol small molecule Q99705 Melanin-concentrating hormone receptor 1 approved DB00502 Haloperidol small molecule Q05940 Synaptic vesicular amine transporter approved|investigational DB00503 Ritonavir small molecule O75469 Nuclear receptor subfamily 1 group I member 2 withdrawn DB00505 Tridihexethyl small molecule P20309 Muscarinic acetylcholine receptor M3 withdrawn DB00505 Tridihexethyl small molecule P11229 Muscarinic acetylcholine receptor M1 withdrawn DB00505 Tridihexethyl small molecule P08172 Muscarinic acetylcholine receptor M2 approved|vet_approved DB00508 Triflupromazine small molecule P14416 D(2) dopamine receptor approved|vet_approved DB00508 Triflupromazine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|vet_approved DB00508 Triflupromazine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00509 Dextrothyroxine small molecule P10827 Thyroid hormone receptor alpha approved|investigational DB00509 Dextrothyroxine small molecule P10828 Thyroid hormone receptor beta approved|investigational DB00509 Dextrothyroxine small molecule P07202 Thyroid peroxidase {ECO:0000305} approved DB00511 Acetyldigitoxin small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved|investigational DB00513 Aminocaproic Acid small molecule P00747 Plasminogen approved|investigational DB00513 Aminocaproic Acid small molecule P00750 Tissue-type plasminogen activator approved DB00514 Dextromethorphan small molecule Q99720 Sigma non-opioid intracellular receptor 1 approved DB00514 Dextromethorphan small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB00514 Dextromethorphan small molecule P31645 Sodium-dependent serotonin transporter approved DB00514 Dextromethorphan small molecule O00264 Membrane-associated progesterone receptor component 1 approved DB00514 Dextromethorphan small molecule P32297 Neuronal acetylcholine receptor subunit alpha-3 approved DB00514 Dextromethorphan small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved DB00514 Dextromethorphan small molecule P30926 Neuronal acetylcholine receptor subunit beta-4 approved DB00514 Dextromethorphan small molecule P17787 Neuronal acetylcholine receptor subunit beta-2 approved DB00514 Dextromethorphan small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved DB00514 Dextromethorphan small molecule P35372 Mu-type opioid receptor approved DB00514 Dextromethorphan small molecule P41143 Delta-type opioid receptor approved DB00514 Dextromethorphan small molecule P04839 Cytochrome b-245 heavy chain approved DB00514 Dextromethorphan small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00515 Cisplatin small molecule P29372 DNA-3-methyladenine glycosylase approved DB00515 Cisplatin small molecule P01023 Alpha-2-macroglobulin approved DB00515 Cisplatin small molecule P02787 Serotransferrin approved DB00515 Cisplatin small molecule O00244 Copper transport protein ATOX1 approved|vet_approved DB00518 Albendazole small molecule Q71U36 Tubulin alpha-1A chain approved|vet_approved DB00518 Albendazole small molecule P68371 Tubulin beta-4B chain approved DB00519 Trandolapril small molecule P12821 Angiotensin-converting enzyme investigational|withdrawn DB00522 Bentiromide small molecule P05981 Serine protease hepsin approved|investigational DB00523 Alitretinoin small molecule P10276 Retinoic acid receptor alpha approved|investigational DB00523 Alitretinoin small molecule P19793 Retinoic acid receptor RXR-alpha approved|investigational DB00523 Alitretinoin small molecule P10826 Retinoic acid receptor beta approved|investigational DB00523 Alitretinoin small molecule P28702 Retinoic acid receptor RXR-beta approved|investigational DB00523 Alitretinoin small molecule P13631 Retinoic acid receptor gamma approved|investigational DB00523 Alitretinoin small molecule P48443 Retinoic acid receptor RXR-gamma approved|investigational DB00523 Alitretinoin small molecule P17936 Insulin-like growth factor-binding protein 3 approved|investigational DB00523 Alitretinoin small molecule Q15238 Pregnancy-specific beta-1-glycoprotein 5 approved DB00524 Metolazone small molecule P55017 Solute carrier family 12 member 3 approved|vet_approved DB00527 Cinchocaine small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|investigational DB00528 Lercanidipine small molecule Q06432 Voltage-dependent calcium channel gamma-1 subunit approved|investigational DB00530 Erlotinib small molecule P00533 Epidermal growth factor receptor approved|investigational DB00530 Erlotinib small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB00531 Cyclophosphamide small molecule O75469 Nuclear receptor subfamily 1 group I member 2 investigational|withdrawn DB00532 Mephenytoin small molecule Q14524 Sodium channel protein type 5 subunit alpha investigational|withdrawn DB00532 Mephenytoin small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational|withdrawn DB00533 Rofecoxib small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational|withdrawn DB00533 Rofecoxib small molecule P15502 Elastin approved DB00535 Cefdinir small molecule P05164 Myeloperoxidase approved|investigational DB00537 Ciprofloxacin small molecule P11388 DNA topoisomerase 2-alpha approved|investigational DB00537 Ciprofloxacin small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB00539 Toremifene small molecule P03372 Estrogen receptor approved|investigational DB00539 Toremifene small molecule P04278 Sex hormone-binding globulin approved DB00540 Nortriptyline small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00540 Nortriptyline small molecule P31645 Sodium-dependent serotonin transporter approved DB00540 Nortriptyline small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00540 Nortriptyline small molecule P35367 Histamine H1 receptor approved DB00540 Nortriptyline small molecule P25100 Alpha-1D adrenergic receptor approved DB00540 Nortriptyline small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00540 Nortriptyline small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00540 Nortriptyline small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00540 Nortriptyline small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00540 Nortriptyline small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00540 Nortriptyline small molecule P14416 D(2) dopamine receptor approved DB00540 Nortriptyline small molecule O00264 Membrane-associated progesterone receptor component 1 approved|investigational DB00541 Vincristine small molecule P07437 Tubulin beta chain approved|investigational DB00541 Vincristine small molecule P68366 Tubulin alpha-4A chain approved|investigational DB00542 Benazepril small molecule P12821 Angiotensin-converting enzyme approved DB00543 Amoxapine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00543 Amoxapine small molecule P31645 Sodium-dependent serotonin transporter approved DB00543 Amoxapine small molecule P14416 D(2) dopamine receptor approved DB00543 Amoxapine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00543 Amoxapine small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00543 Amoxapine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00543 Amoxapine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00543 Amoxapine small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00543 Amoxapine small molecule P35462 D(3) dopamine receptor approved DB00543 Amoxapine small molecule P21917 D(4) dopamine receptor approved DB00543 Amoxapine small molecule P35367 Histamine H1 receptor approved DB00543 Amoxapine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00543 Amoxapine small molecule Q9H3N8 Histamine H4 receptor approved DB00543 Amoxapine small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00544 Fluorouracil small molecule P04818 Thymidylate synthase approved|investigational DB00545 Pyridostigmine small molecule P22303 Acetylcholinesterase approved|investigational DB00545 Pyridostigmine small molecule P06276 Cholinesterase approved|investigational DB00545 Pyridostigmine small molecule P02768 Serum albumin approved DB00546 Adinazolam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00546 Adinazolam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB00546 Adinazolam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB00546 Adinazolam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved DB00546 Adinazolam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved DB00546 Adinazolam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved DB00546 Adinazolam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved DB00546 Adinazolam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved DB00546 Adinazolam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved DB00546 Adinazolam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved DB00546 Adinazolam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved DB00546 Adinazolam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved DB00546 Adinazolam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved DB00546 Adinazolam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved DB00547 Desoximetasone small molecule P04150 Glucocorticoid receptor approved DB00548 Azelaic Acid small molecule P51857 3-oxo-5-beta-steroid 4-dehydrogenase approved DB00548 Azelaic Acid small molecule P14679 Tyrosinase approved|investigational DB00549 Zafirlukast small molecule Q9Y271 Cysteinyl leukotriene receptor 1 approved|investigational DB00550 Propylthiouracil small molecule P07202 Thyroid peroxidase {ECO:0000305} approved DB00551 Acetohydroxamic Acid small molecule P39900 Macrophage metalloelastase approved|investigational DB00552 Pentostatin small molecule P00813 Adenosine deaminase approved|investigational DB00554 Piroxicam small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB00554 Piroxicam small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB00555 Lamotrigine small molecule Q15878 Voltage-dependent R-type calcium channel subunit alpha-1E approved|investigational DB00555 Lamotrigine small molecule Q99250 Sodium channel protein type 2 subunit alpha approved|investigational DB00555 Lamotrigine small molecule P30542 Adenosine receptor A1 approved|investigational DB00555 Lamotrigine small molecule P14416 D(2) dopamine receptor approved|investigational DB00555 Lamotrigine small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00555 Lamotrigine small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00555 Lamotrigine small molecule P35367 Histamine H1 receptor approved|investigational DB00555 Lamotrigine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00555 Lamotrigine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00557 Hydroxyzine small molecule P35367 Histamine H1 receptor approved|investigational DB00559 Bosentan small molecule P25101 Endothelin-1 receptor {ECO:0000305} approved|investigational DB00559 Bosentan small molecule P24530 Endothelin receptor type B {ECO:0000305} approved|vet_approved DB00561 Doxapram small molecule O14649 Potassium channel subfamily K member 3 approved|vet_approved DB00561 Doxapram small molecule Q9NPC2 Potassium channel subfamily K member 9 approved DB00562 Benzthiazide small molecule P55017 Solute carrier family 12 member 3 approved DB00562 Benzthiazide small molecule P00915 Carbonic anhydrase 1 approved DB00562 Benzthiazide small molecule P00918 Carbonic anhydrase 2 approved DB00562 Benzthiazide small molecule P22748 Carbonic anhydrase 4 approved DB00562 Benzthiazide small molecule Q16790 Carbonic anhydrase 9 approved DB00562 Benzthiazide small molecule O43570 Carbonic anhydrase 12 approved DB00563 Methotrexate small molecule P00374 Dihydrofolate reductase approved|investigational DB00564 Carbamazepine small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|investigational DB00564 Carbamazepine small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|investigational DB00564 Carbamazepine small molecule P17787 Neuronal acetylcholine receptor subunit beta-2 approved|investigational DB00564 Carbamazepine small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB00568 Cinnarizine small molecule P35367 Histamine H1 receptor approved|investigational DB00568 Cinnarizine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB00568 Cinnarizine small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved|investigational DB00568 Cinnarizine small molecule O60840 Voltage-dependent L-type calcium channel subunit alpha-1F {ECO:0000305} approved|investigational DB00568 Cinnarizine small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved|investigational DB00568 Cinnarizine small molecule O43497 Voltage-dependent T-type calcium channel subunit alpha-1G approved|investigational DB00568 Cinnarizine small molecule O95180 Voltage-dependent T-type calcium channel subunit alpha-1H approved|investigational DB00568 Cinnarizine small molecule Q9P0X4 Voltage-dependent T-type calcium channel subunit alpha-1I approved|investigational DB00568 Cinnarizine small molecule P14416 D(2) dopamine receptor approved|investigational DB00568 Cinnarizine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00570 Vinblastine small molecule Q71U36 Tubulin alpha-1A chain approved DB00570 Vinblastine small molecule P07437 Tubulin beta chain approved DB00570 Vinblastine small molecule Q9UJT1 Tubulin delta chain approved DB00570 Vinblastine small molecule P23258 Tubulin gamma-1 chain approved DB00570 Vinblastine small molecule P05412 Transcription factor AP-1 approved|investigational DB00571 Propranolol small molecule P13945 Beta-3 adrenergic receptor approved|vet_approved DB00572 Atropine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|vet_approved DB00572 Atropine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|vet_approved DB00572 Atropine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|vet_approved DB00572 Atropine small molecule P08173 Muscarinic acetylcholine receptor M4 approved|vet_approved DB00572 Atropine small molecule P23415 Glycine receptor subunit alpha-1 approved|vet_approved DB00572 Atropine small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|vet_approved DB00572 Atropine small molecule P17787 Neuronal acetylcholine receptor subunit beta-2 approved DB00573 Fenoprofen small molecule P35354 Prostaglandin G/H synthase 2 approved DB00573 Fenoprofen small molecule P23219 Prostaglandin G/H synthase 1 approved DB00573 Fenoprofen small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved DB00573 Fenoprofen small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|illicit|investigational|withdrawn DB00574 Fenfluramine small molecule P31645 Sodium-dependent serotonin transporter approved|illicit|investigational|withdrawn DB00574 Fenfluramine small molecule P28335 5-hydroxytryptamine receptor 2C approved|illicit|investigational|withdrawn DB00574 Fenfluramine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00575 Clonidine small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB00579 Mazindol small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB00579 Mazindol small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB00579 Mazindol small molecule Q05940 Synaptic vesicular amine transporter approved|investigational|withdrawn DB00580 Valdecoxib small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational|withdrawn DB00580 Valdecoxib small molecule P00918 Carbonic anhydrase 2 approved|investigational|withdrawn DB00580 Valdecoxib small molecule P07451 Carbonic anhydrase 3 approved|investigational DB00583 L-Carnitine small molecule Q9H015 Solute carrier family 22 member 4 approved|investigational DB00583 L-Carnitine small molecule O76082 Solute carrier family 22 member 5 approved|investigational DB00583 L-Carnitine small molecule P43155 Carnitine O-acetyltransferase approved|investigational DB00583 L-Carnitine small molecule O43772 Mitochondrial carnitine/acylcarnitine carrier protein approved|investigational DB00583 L-Carnitine small molecule Q9UKG9 Peroxisomal carnitine O-octanoyltransferase approved|investigational DB00583 L-Carnitine small molecule P23786 Carnitine O-palmitoyltransferase 2, mitochondrial approved|investigational DB00583 L-Carnitine small molecule P50416 Carnitine O-palmitoyltransferase 1, liver isoform approved|investigational DB00583 L-Carnitine small molecule P23141 Liver carboxylesterase 1 approved|investigational DB00583 L-Carnitine small molecule P05164 Myeloperoxidase approved|vet_approved DB00584 Enalapril small molecule P12821 Angiotensin-converting enzyme approved DB00585 Nizatidine small molecule P25021 Histamine H2 receptor approved|vet_approved DB00586 Diclofenac small molecule P35354 Prostaglandin G/H synthase 2 approved|vet_approved DB00586 Diclofenac small molecule P23219 Prostaglandin G/H synthase 1 approved|vet_approved DB00586 Diclofenac small molecule P09917 Arachidonate 5-lipoxygenase approved|vet_approved DB00586 Diclofenac small molecule P35499 Sodium channel protein type 4 subunit alpha approved|vet_approved DB00586 Diclofenac small molecule P78348 Acid-sensing ion channel 1 {ECO:0000303|PubMed:10798398} approved|vet_approved DB00586 Diclofenac small molecule O43526 Potassium voltage-gated channel subfamily KQT member 2 {ECO:0000305} approved|vet_approved DB00586 Diclofenac small molecule O43525 Potassium voltage-gated channel subfamily KQT member 3 {ECO:0000305} approved|vet_approved DB00586 Diclofenac small molecule P14555 Phospholipase A2, membrane associated approved|investigational DB00589 Lisuride small molecule P14416 D(2) dopamine receptor approved|investigational DB00589 Lisuride small molecule P35462 D(3) dopamine receptor approved|investigational DB00589 Lisuride small molecule P21917 D(4) dopamine receptor approved|investigational DB00589 Lisuride small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB00589 Lisuride small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB00589 Lisuride small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00590 Doxazosin small molecule P25100 Alpha-1D adrenergic receptor approved DB00590 Doxazosin small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB00590 Doxazosin small molecule Q9NS40 Potassium voltage-gated channel subfamily H member 7 approved|investigational|vet_approved DB00591 Fluocinolone Acetonide small molecule P04150 Glucocorticoid receptor approved|vet_approved DB00592 Piperazine small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved DB00593 Ethosuximide small molecule O43497 Voltage-dependent T-type calcium channel subunit alpha-1G approved DB00594 Amiloride small molecule P37088 Amiloride-sensitive sodium channel subunit alpha approved DB00594 Amiloride small molecule P51168 Amiloride-sensitive sodium channel subunit beta approved DB00594 Amiloride small molecule P51170 Amiloride-sensitive sodium channel subunit gamma approved DB00594 Amiloride small molecule P51172 Amiloride-sensitive sodium channel subunit delta approved DB00594 Amiloride small molecule P19801 Amiloride-sensitive amine oxidase [copper-containing] approved DB00594 Amiloride small molecule Q16515 Acid-sensing ion channel 2 {ECO:0000303|PubMed:10842183} approved DB00594 Amiloride small molecule P78348 Acid-sensing ion channel 1 {ECO:0000303|PubMed:10798398} approved DB00594 Amiloride small molecule P19634 Sodium/hydrogen exchanger 1 approved DB00594 Amiloride small molecule P00749 Urokinase-type plasminogen activator approved DB00596 Ulobetasol small molecule P04150 Glucocorticoid receptor approved|vet_approved DB00599 Thiopental small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|vet_approved DB00599 Thiopental small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|vet_approved DB00599 Thiopental small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|vet_approved DB00599 Thiopental small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|vet_approved DB00599 Thiopental small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|vet_approved DB00599 Thiopental small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|vet_approved DB00599 Thiopental small molecule P42262 Glutamate receptor 2 approved|vet_approved DB00599 Thiopental small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved|vet_approved DB00599 Thiopental small molecule O00519 Fatty-acid amide hydrolase 1 approved|vet_approved DB00599 Thiopental small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00600 Monobenzone small molecule P14679 Tyrosinase approved|investigational|vet_approved DB00602 Ivermectin small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|investigational DB00603 Medroxyprogesterone acetate small molecule P06401 Progesterone receptor approved|investigational DB00603 Medroxyprogesterone acetate small molecule P03372 Estrogen receptor approved|investigational|withdrawn DB00604 Cisapride small molecule Q13639 5-hydroxytryptamine receptor 4 approved|investigational|withdrawn DB00604 Cisapride small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational|withdrawn DB00604 Cisapride small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB00605 Sulindac small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB00605 Sulindac small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB00605 Sulindac small molecule P15121 Aldose reductase approved|investigational DB00605 Sulindac small molecule P27361 Mitogen-activated protein kinase 3 approved|investigational DB00605 Sulindac small molecule Q03181 Peroxisome proliferator-activated receptor delta approved|investigational DB00605 Sulindac small molecule O60218 Aldo-keto reductase family 1 member B10 approved DB00606 Cyclothiazide small molecule P54710 Sodium/potassium-transporting ATPase subunit gamma approved DB00606 Cyclothiazide small molecule P00915 Carbonic anhydrase 1 approved DB00606 Cyclothiazide small molecule P00918 Carbonic anhydrase 2 approved DB00606 Cyclothiazide small molecule P22748 Carbonic anhydrase 4 approved DB00606 Cyclothiazide small molecule Q6FHJ7 Secreted frizzled-related protein 4 approved|investigational|vet_approved DB00608 Chloroquine small molecule P01375 Tumor necrosis factor approved|investigational|vet_approved DB00608 Chloroquine small molecule Q9NR96 Toll-like receptor 9 approved|illicit|vet_approved DB00611 Butorphanol small molecule P41143 Delta-type opioid receptor approved|illicit|vet_approved DB00611 Butorphanol small molecule P35372 Mu-type opioid receptor approved|investigational DB00613 Amodiaquine small molecule P50135 Histamine N-methyltransferase approved|investigational DB00615 Rifabutin small molecule P07900 Heat shock protein HSP 90-alpha approved|investigational DB00615 Rifabutin small molecule P14625 Endoplasmin approved DB00617 Paramethadione small molecule Q9P0X4 Voltage-dependent T-type calcium channel subunit alpha-1I approved DB00619 Imatinib small molecule P10721 Mast/stem cell growth factor receptor Kit approved DB00619 Imatinib small molecule P04629 High affinity nerve growth factor receptor approved DB00619 Imatinib small molecule P07333 Macrophage colony-stimulating factor 1 receptor approved DB00619 Imatinib small molecule P16234 Platelet-derived growth factor receptor alpha approved DB00619 Imatinib small molecule Q08345 Epithelial discoidin domain-containing receptor 1 approved DB00619 Imatinib small molecule P00519 Tyrosine-protein kinase ABL1 approved DB00619 Imatinib small molecule P09619 Platelet-derived growth factor receptor beta approved|vet_approved DB00620 Triamcinolone small molecule P04150 Glucocorticoid receptor approved|investigational DB00621 Oxandrolone small molecule P10275 Androgen receptor approved|investigational DB00622 Nicardipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB00622 Nicardipine small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved|investigational DB00622 Nicardipine small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved|investigational DB00622 Nicardipine small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved|investigational DB00622 Nicardipine small molecule P54750 Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A approved|investigational DB00622 Nicardipine small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB00622 Nicardipine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00622 Nicardipine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00622 Nicardipine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB00622 Nicardipine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00623 Fluphenazine small molecule P14416 D(2) dopamine receptor approved DB00623 Fluphenazine small molecule P10275 Androgen receptor approved DB00623 Fluphenazine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00623 Fluphenazine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB00624 Testosterone small molecule P10275 Androgen receptor approved|investigational DB00624 Testosterone small molecule P03372 Estrogen receptor approved|investigational DB00624 Testosterone small molecule P08235 Mineralocorticoid receptor approved|vet_approved DB00626 Bacitracin small molecule P14735 Insulin-degrading enzyme approved|vet_approved DB00626 Bacitracin small molecule P01023 Alpha-2-macroglobulin approved|investigational|nutraceutical DB00627 Niacin small molecule Q15274 Nicotinate-nucleotide pyrophosphorylase [carboxylating] approved|investigational|nutraceutical DB00627 Niacin small molecule P40261 Nicotinamide N-methyltransferase approved DB00630 Alendronic acid small molecule P14324 Farnesyl pyrophosphate synthase approved DB00630 Alendronic acid small molecule P29074 Tyrosine-protein phosphatase non-receptor type 4 approved DB00630 Alendronic acid small molecule Q13332 Receptor-type tyrosine-protein phosphatase S approved DB00630 Alendronic acid small molecule P23469 Receptor-type tyrosine-protein phosphatase epsilon approved DB00630 Alendronic acid small molecule P38606 V-type proton ATPase catalytic subunit A approved|investigational DB00631 Clofarabine small molecule P09884 DNA polymerase alpha catalytic subunit approved|investigational DB00631 Clofarabine small molecule P23921 Ribonucleoside-diphosphate reductase large subunit approved|vet_approved DB00635 Prednisone small molecule P04150 Glucocorticoid receptor approved|vet_approved DB00635 Prednisone small molecule P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 approved|investigational DB00636 Clofibrate small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved|withdrawn DB00637 Astemizole small molecule P35367 Histamine H1 receptor approved|withdrawn DB00637 Astemizole small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|withdrawn DB00637 Astemizole small molecule O95259 Potassium voltage-gated channel subfamily H member 1 approved|withdrawn DB00637 Astemizole small molecule P10636 Microtubule-associated protein tau approved|investigational DB00640 Adenosine small molecule P29275 Adenosine receptor A2b approved|investigational DB00640 Adenosine small molecule P30542 Adenosine receptor A1 approved DB00641 Simvastatin small molecule P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase approved DB00641 Simvastatin small molecule P20701 Integrin alpha-L approved|investigational DB00642 Pemetrexed small molecule P04818 Thymidylate synthase approved|investigational DB00642 Pemetrexed small molecule P31939 Bifunctional purine biosynthesis protein PURH approved|investigational DB00642 Pemetrexed small molecule P00374 Dihydrofolate reductase approved|investigational DB00642 Pemetrexed small molecule P22102 Trifunctional purine biosynthetic protein adenosine-3 approved|vet_approved DB00643 Mebendazole small molecule Q71U36 Tubulin alpha-1A chain approved|vet_approved DB00643 Mebendazole small molecule P68371 Tubulin beta-4B chain approved|illicit|investigational|withdrawn DB00647 Dextropropoxyphene small molecule P35372 Mu-type opioid receptor approved|illicit|investigational|withdrawn DB00647 Dextropropoxyphene small molecule P41143 Delta-type opioid receptor approved|illicit|investigational|withdrawn DB00647 Dextropropoxyphene small molecule P23141 Liver carboxylesterase 1 approved DB00648 Mitotane small molecule P15538 Cytochrome P450 11B1, mitochondrial approved DB00648 Mitotane small molecule P10109 Adrenodoxin, mitochondrial approved DB00648 Mitotane small molecule P03372 Estrogen receptor approved DB00648 Mitotane small molecule P06401 Progesterone receptor approved DB00648 Mitotane small molecule P10275 Androgen receptor approved DB00651 Dyphylline small molecule Q07343 cAMP-specific 3',5'-cyclic phosphodiesterase 4B approved DB00651 Dyphylline small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved DB00651 Dyphylline small molecule Q08493 cAMP-specific 3',5'-cyclic phosphodiesterase 4C approved DB00651 Dyphylline small molecule Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D approved DB00651 Dyphylline small molecule P30542 Adenosine receptor A1 approved DB00651 Dyphylline small molecule Q13946 High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A approved DB00651 Dyphylline small molecule Q9NP56 cAMP-specific 3',5'-cyclic phosphodiesterase 7B approved|vet_approved DB00652 Pentazocine small molecule P35372 Mu-type opioid receptor approved|vet_approved DB00652 Pentazocine small molecule Q99720 Sigma non-opioid intracellular receptor 1 approved|investigational|vet_approved DB00653 Magnesium sulfate small molecule Q06432 Voltage-dependent calcium channel gamma-1 subunit approved|investigational|vet_approved DB00653 Magnesium sulfate small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved|investigational|vet_approved DB00653 Magnesium sulfate small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational|vet_approved DB00653 Magnesium sulfate small molecule Q02641 Voltage-dependent L-type calcium channel subunit beta-1 approved|investigational|vet_approved DB00653 Magnesium sulfate small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved|investigational|vet_approved DB00653 Magnesium sulfate small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved|investigational DB00654 Latanoprost small molecule P43088 Prostaglandin F2-alpha receptor approved DB00655 Estrone small molecule P03372 Estrogen receptor approved DB00655 Estrone small molecule Q92731 Estrogen receptor beta approved DB00655 Estrone small molecule P10275 Androgen receptor approved DB00655 Estrone small molecule P11511 Aromatase approved DB00655 Estrone small molecule P04278 Sex hormone-binding globulin approved|investigational DB00656 Trazodone small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB00656 Trazodone small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB00656 Trazodone small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB00656 Trazodone small molecule P35367 Histamine H1 receptor approved|investigational DB00657 Mecamylamine small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved|investigational DB00657 Mecamylamine small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|investigational DB00657 Mecamylamine small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|investigational DB00657 Mecamylamine small molecule P17787 Neuronal acetylcholine receptor subunit beta-2 approved|investigational DB00659 Acamprosate small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00659 Acamprosate small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved|investigational DB00659 Acamprosate small molecule P41594 Metabotropic glutamate receptor 5 approved DB00661 Verapamil small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved DB00661 Verapamil small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved DB00661 Verapamil small molecule O60840 Voltage-dependent L-type calcium channel subunit alpha-1F {ECO:0000305} approved DB00661 Verapamil small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved DB00661 Verapamil small molecule Q02641 Voltage-dependent L-type calcium channel subunit beta-1 approved DB00661 Verapamil small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved DB00661 Verapamil small molecule P54284 Voltage-dependent L-type calcium channel subunit beta-3 approved DB00661 Verapamil small molecule O00305 Voltage-dependent L-type calcium channel subunit beta-4 {ECO:0000305} approved DB00661 Verapamil small molecule Q9P0X4 Voltage-dependent T-type calcium channel subunit alpha-1I approved DB00661 Verapamil small molecule O43497 Voltage-dependent T-type calcium channel subunit alpha-1G approved DB00661 Verapamil small molecule Q00975 Voltage-dependent N-type calcium channel subunit alpha-1B approved DB00661 Verapamil small molecule O00555 Voltage-dependent P/Q-type calcium channel subunit alpha-1A approved DB00661 Verapamil small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB00661 Verapamil small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB00661 Verapamil small molecule P31645 Sodium-dependent serotonin transporter approved DB00661 Verapamil small molecule P25100 Alpha-1D adrenergic receptor approved|vet_approved DB00663 Flumethasone small molecule P04150 Glucocorticoid receptor approved|investigational DB00665 Nilutamide small molecule P10275 Androgen receptor approved|vet_approved DB00668 Epinephrine small molecule P25100 Alpha-1D adrenergic receptor approved|vet_approved DB00668 Epinephrine small molecule P00439 Phenylalanine-4-hydroxylase approved|vet_approved DB00668 Epinephrine small molecule P13945 Beta-3 adrenergic receptor approved|vet_approved DB00668 Epinephrine small molecule P01375 Tumor necrosis factor approved|vet_approved DB00668 Epinephrine small molecule P00441 Superoxide dismutase [Cu-Zn] approved DB00670 Pirenzepine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00672 Chlorpropamide small molecule Q09428 ATP-binding cassette sub-family C member 8 approved|investigational DB00673 Aprepitant small molecule P25103 Substance-P receptor approved DB00674 Galantamine small molecule P22303 Acetylcholinesterase approved DB00674 Galantamine small molecule P02708 Acetylcholine receptor subunit alpha approved DB00674 Galantamine small molecule P11230 Acetylcholine receptor subunit beta approved DB00674 Galantamine small molecule Q07001 Acetylcholine receptor subunit delta approved DB00674 Galantamine small molecule Q04844 Acetylcholine receptor subunit epsilon approved DB00674 Galantamine small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB00674 Galantamine small molecule P32297 Neuronal acetylcholine receptor subunit alpha-3 approved DB00674 Galantamine small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved DB00674 Galantamine small molecule Q15825 Neuronal acetylcholine receptor subunit alpha-6 approved DB00674 Galantamine small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved DB00674 Galantamine small molecule Q9UGM1 Neuronal acetylcholine receptor subunit alpha-9 approved DB00674 Galantamine small molecule P17787 Neuronal acetylcholine receptor subunit beta-2 approved DB00674 Galantamine small molecule Q05901 Neuronal acetylcholine receptor subunit beta-3 approved DB00674 Galantamine small molecule P30926 Neuronal acetylcholine receptor subunit beta-4 approved DB00674 Galantamine small molecule P06276 Cholinesterase approved DB00675 Tamoxifen small molecule P03372 Estrogen receptor approved DB00675 Tamoxifen small molecule Q92731 Estrogen receptor beta approved DB00675 Tamoxifen small molecule P17252 Protein kinase C alpha type approved DB00675 Tamoxifen small molecule P10275 Androgen receptor approved DB00675 Tamoxifen small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB00675 Tamoxifen small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB00675 Tamoxifen small molecule P62508 Estrogen-related receptor gamma approved DB00675 Tamoxifen small molecule P04278 Sex hormone-binding globulin approved DB00678 Losartan small molecule P30556 Type-1 angiotensin II receptor approved|withdrawn DB00679 Thioridazine small molecule P14416 D(2) dopamine receptor approved|withdrawn DB00679 Thioridazine small molecule P28223 5-hydroxytryptamine receptor 2A approved|withdrawn DB00679 Thioridazine small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational|withdrawn DB00680 Moricizine small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB00682 Warfarin small molecule Q9BQB6 Vitamin K epoxide reductase complex subunit 1 approved DB00682 Warfarin small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|illicit DB00683 Midazolam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB00683 Midazolam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB00683 Midazolam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB00683 Midazolam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB00683 Midazolam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|illicit DB00683 Midazolam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|illicit DB00683 Midazolam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|illicit DB00683 Midazolam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|illicit DB00683 Midazolam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|illicit DB00683 Midazolam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|illicit DB00683 Midazolam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|illicit DB00683 Midazolam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|illicit DB00683 Midazolam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|illicit DB00683 Midazolam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|investigational|withdrawn DB00685 Trovafloxacin small molecule P11388 DNA topoisomerase 2-alpha approved DB00686 Pentosan Polysulfate small molecule P09038 Fibroblast growth factor 2 approved DB00686 Pentosan Polysulfate small molecule P05230 Fibroblast growth factor 1 approved DB00686 Pentosan Polysulfate small molecule P08620 Fibroblast growth factor 4 approved|investigational DB00687 Fludrocortisone small molecule P08235 Mineralocorticoid receptor approved|investigational DB00687 Fludrocortisone small molecule P04150 Glucocorticoid receptor approved|investigational DB00687 Fludrocortisone small molecule P10275 Androgen receptor approved|illicit|investigational DB00690 Flurazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit|investigational DB00690 Flurazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit|investigational DB00690 Flurazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit|investigational DB00690 Flurazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit|investigational DB00690 Flurazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|illicit|investigational DB00690 Flurazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|illicit|investigational DB00690 Flurazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|illicit|investigational DB00690 Flurazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|illicit|investigational DB00690 Flurazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|illicit|investigational DB00690 Flurazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|illicit|investigational DB00690 Flurazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|illicit|investigational DB00690 Flurazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|illicit|investigational DB00690 Flurazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|illicit|investigational DB00690 Flurazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved DB00691 Moexipril small molecule P12821 Angiotensin-converting enzyme approved DB00691 Moexipril small molecule Q9BYF1 Angiotensin-converting enzyme 2 approved DB00692 Phentolamine small molecule P25100 Alpha-1D adrenergic receptor approved DB00694 Daunorubicin small molecule P11388 DNA topoisomerase 2-alpha approved DB00694 Daunorubicin small molecule Q02880 DNA topoisomerase 2-beta approved|vet_approved DB00695 Furosemide small molecule Q13621 Solute carrier family 12 member 1 approved|vet_approved DB00695 Furosemide small molecule P00918 Carbonic anhydrase 2 approved DB00696 Ergotamine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00696 Ergotamine small molecule P14416 D(2) dopamine receptor approved DB00696 Ergotamine small molecule P25100 Alpha-1D adrenergic receptor approved DB00696 Ergotamine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00696 Ergotamine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB00697 Tizanidine small molecule Q9Y2I1 Nischarin approved DB00700 Eplerenone small molecule P08235 Mineralocorticoid receptor approved DB00703 Methazolamide small molecule P00915 Carbonic anhydrase 1 approved DB00703 Methazolamide small molecule P00918 Carbonic anhydrase 2 approved DB00703 Methazolamide small molecule P22748 Carbonic anhydrase 4 approved DB00703 Methazolamide small molecule P43166 Carbonic anhydrase 7 approved DB00703 Methazolamide small molecule P07451 Carbonic anhydrase 3 approved|investigational|vet_approved DB00704 Naltrexone small molecule P41143 Delta-type opioid receptor approved|investigational|vet_approved DB00704 Naltrexone small molecule P35372 Mu-type opioid receptor approved|investigational DB00706 Tamsulosin small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB00707 Porfimer sodium small molecule P01130 Low-density lipoprotein receptor approved|investigational DB00708 Sufentanil small molecule P35372 Mu-type opioid receptor approved|investigational DB00708 Sufentanil small molecule P41143 Delta-type opioid receptor approved|investigational DB00710 Ibandronate small molecule P14324 Farnesyl pyrophosphate synthase approved|investigational|vet_approved DB00711 Diethylcarbamazine small molecule P09917 Arachidonate 5-lipoxygenase approved|investigational|vet_approved DB00711 Diethylcarbamazine small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB00712 Flurbiprofen small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB00712 Flurbiprofen small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB00713 Oxacillin small molecule P46059 Solute carrier family 15 member 1 approved|investigational DB00714 Apomorphine small molecule P35462 D(3) dopamine receptor approved|investigational DB00714 Apomorphine small molecule P21917 D(4) dopamine receptor approved|investigational DB00714 Apomorphine small molecule P14416 D(2) dopamine receptor approved|investigational DB00714 Apomorphine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB00714 Apomorphine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB00715 Paroxetine small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB00715 Paroxetine small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB00715 Paroxetine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB00715 Paroxetine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00715 Paroxetine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00715 Paroxetine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB00715 Paroxetine small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB00716 Nedocromil small molecule Q9Y271 Cysteinyl leukotriene receptor 1 approved|investigational DB00716 Nedocromil small molecule Q9NS75 Cysteinyl leukotriene receptor 2 approved|investigational DB00716 Nedocromil small molecule P07900 Heat shock protein HSP 90-alpha approved DB00717 Norethisterone small molecule P06401 Progesterone receptor approved DB00719 Azatadine small molecule P35367 Histamine H1 receptor approved|investigational|vet_approved DB00720 Clodronic Acid small molecule P12235 ADP/ATP translocase 1 approved|investigational|vet_approved DB00720 Clodronic Acid small molecule P05141 ADP/ATP translocase 2 approved|investigational|vet_approved DB00721 Procaine small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved|investigational|vet_approved DB00721 Procaine small molecule Q12791 Calcium-activated potassium channel subunit alpha-1 approved|investigational|vet_approved DB00721 Procaine small molecule P21397 Amine oxidase [flavin-containing] A approved|investigational DB00722 Lisinopril small molecule P12821 Angiotensin-converting enzyme approved|investigational DB00723 Methoxamine small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB00724 Imiquimod small molecule Q9NYK1 Toll-like receptor 7 approved DB00725 Homatropine Methylbromide small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00725 Homatropine Methylbromide small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00725 Homatropine Methylbromide small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00725 Homatropine Methylbromide small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00726 Trimipramine small molecule P31645 Sodium-dependent serotonin transporter approved DB00726 Trimipramine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00726 Trimipramine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00726 Trimipramine small molecule P14416 D(2) dopamine receptor approved DB00726 Trimipramine small molecule P35367 Histamine H1 receptor approved DB00726 Trimipramine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00726 Trimipramine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00728 Rocuronium small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB00728 Rocuronium small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00731 Nateglinide small molecule Q09428 ATP-binding cassette sub-family C member 8 approved|investigational DB00731 Nateglinide small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|vet_approved DB00733 Pralidoxime small molecule P22303 Acetylcholinesterase approved|vet_approved DB00733 Pralidoxime small molecule P06276 Cholinesterase approved|investigational DB00734 Risperidone small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB00734 Risperidone small molecule P14416 D(2) dopamine receptor approved|investigational DB00734 Risperidone small molecule P35462 D(3) dopamine receptor approved|investigational DB00734 Risperidone small molecule P21917 D(4) dopamine receptor approved|investigational DB00734 Risperidone small molecule P35367 Histamine H1 receptor approved|investigational DB00734 Risperidone small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB00734 Risperidone small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00735 Naftifine small molecule Q14534 Squalene monooxygenase approved|investigational DB00736 Esomeprazole small molecule P20648 Potassium-transporting ATPase alpha chain 1 approved DB00737 Meclizine small molecule P35367 Histamine H1 receptor approved DB00737 Meclizine small molecule Q14994 Nuclear receptor subfamily 1 group I member 3 approved|investigational DB00738 Pentamidine small molecule O14717 tRNA (cytosine(38)-C(5))-methyltransferase approved|investigational DB00740 Riluzole small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|vet_approved DB00741 Hydrocortisone small molecule P04150 Glucocorticoid receptor approved|vet_approved DB00741 Hydrocortisone small molecule P04083 Annexin A1 approved|vet_approved DB00741 Hydrocortisone small molecule P80365 Corticosteroid 11-beta-dehydrogenase isozyme 2 approved|vet_approved DB00741 Hydrocortisone small molecule P14060 3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1 approved|investigational DB00746 Deferoxamine small molecule P05067 Amyloid-beta A4 protein approved|investigational DB00747 Scopolamine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00747 Scopolamine small molecule P14410 Sucrase-isomaltase, intestinal approved|investigational DB00747 Scopolamine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00747 Scopolamine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB00747 Scopolamine small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB00747 Scopolamine small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|investigational DB00747 Scopolamine small molecule P17787 Neuronal acetylcholine receptor subunit beta-2 approved DB00748 Carbinoxamine small molecule P35367 Histamine H1 receptor approved|investigational|vet_approved DB00749 Etodolac small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational|vet_approved DB00749 Etodolac small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational|vet_approved DB00749 Etodolac small molecule P19793 Retinoic acid receptor RXR-alpha approved DB00750 Prilocaine small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|investigational DB00751 Epinastine small molecule P35367 Histamine H1 receptor approved|investigational DB00751 Epinastine small molecule P25021 Histamine H2 receptor approved|investigational DB00751 Epinastine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB00751 Epinastine small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational DB00752 Tranylcypromine small molecule P21397 Amine oxidase [flavin-containing] A approved|investigational DB00752 Tranylcypromine small molecule P27338 Amine oxidase [flavin-containing] B approved|vet_approved DB00753 Isoflurane small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|vet_approved DB00753 Isoflurane small molecule P98194 Calcium-transporting ATPase type 2C member 1 approved|vet_approved DB00753 Isoflurane small molecule P23415 Glycine receptor subunit alpha-1 approved|vet_approved DB00753 Isoflurane small molecule P42261 Glutamate receptor 1 approved|vet_approved DB00753 Isoflurane small molecule Q09470 Potassium voltage-gated channel subfamily A member 1 approved|vet_approved DB00753 Isoflurane small molecule P30049 ATP synthase subunit delta, mitochondrial {ECO:0000305} approved|vet_approved DB00753 Isoflurane small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00754 Ethotoin small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB00754 Ethotoin small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational|nutraceutical DB00755 Tretinoin small molecule P28702 Retinoic acid receptor RXR-beta approved|investigational|nutraceutical DB00755 Tretinoin small molecule P48443 Retinoic acid receptor RXR-gamma approved|investigational|nutraceutical DB00755 Tretinoin small molecule P13631 Retinoic acid receptor gamma approved|investigational|nutraceutical DB00755 Tretinoin small molecule P00352 Retinal dehydrogenase 1 {ECO:0000305} approved|investigational|nutraceutical DB00755 Tretinoin small molecule Q8NFJ5 Retinoic acid-induced protein 3 approved|investigational|nutraceutical DB00755 Tretinoin small molecule P51843 Nuclear receptor subfamily 0 group B member 1 approved|investigational|nutraceutical DB00755 Tretinoin small molecule O94788 Retinal dehydrogenase 2 approved|investigational|nutraceutical DB00755 Tretinoin small molecule P49788 Retinoic acid receptor responder protein 1 approved|investigational|nutraceutical DB00755 Tretinoin small molecule P10276 Retinoic acid receptor alpha approved|investigational|nutraceutical DB00755 Tretinoin small molecule P10826 Retinoic acid receptor beta approved|investigational|nutraceutical DB00755 Tretinoin small molecule P31025 Lipocalin-1 approved|investigational|nutraceutical DB00755 Tretinoin small molecule P02753 Retinol-binding protein 4 approved|investigational|nutraceutical DB00755 Tretinoin small molecule Q16654 [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial approved|investigational|nutraceutical DB00755 Tretinoin small molecule P19793 Retinoic acid receptor RXR-alpha approved|investigational|nutraceutical DB00755 Tretinoin small molecule O43174 Cytochrome P450 26A1 approved|investigational|nutraceutical DB00755 Tretinoin small molecule Q9NR63 Cytochrome P450 26B1 approved|withdrawn DB00756 Hexachlorophene small molecule O14521 Succinate dehydrogenase [ubiquinone] cytochrome b small subunit, mitochondrial approved|withdrawn DB00756 Hexachlorophene small molecule P00367 Glutamate dehydrogenase 1, mitochondrial approved|withdrawn DB00756 Hexachlorophene small molecule P03372 Estrogen receptor approved DB00758 Clopidogrel small molecule Q9H244 P2Y purinoceptor 12 approved|vet_approved DB00759 Tetracycline small molecule P04156 Major prion protein approved|vet_approved DB00759 Tetracycline small molecule Q9UM07 Protein-arginine deiminase type-4 approved|withdrawn DB00761 Potassium Chloride small molecule P55011 Solute carrier family 12 member 2 approved|withdrawn DB00761 Potassium Chloride small molecule Q13621 Solute carrier family 12 member 1 approved|withdrawn DB00761 Potassium Chloride small molecule Q9H2X9 Solute carrier family 12 member 5 approved|withdrawn DB00761 Potassium Chloride small molecule Q9UHW9 Solute carrier family 12 member 6 approved|withdrawn DB00761 Potassium Chloride small molecule Q9Y666 Solute carrier family 12 member 7 approved|withdrawn DB00761 Potassium Chloride small molecule Q9UP95 Solute carrier family 12 member 4 approved|investigational DB00762 Irinotecan small molecule P11387 DNA topoisomerase 1 approved|investigational DB00762 Irinotecan small molecule Q969P6 DNA topoisomerase I, mitochondrial approved DB00763 Methimazole small molecule P07202 Thyroid peroxidase {ECO:0000305} approved|vet_approved DB00764 Mometasone small molecule P04150 Glucocorticoid receptor approved|vet_approved DB00764 Mometasone small molecule P06401 Progesterone receptor approved DB00765 Metyrosine small molecule P07101 Tyrosine 3-monooxygenase approved DB00768 Olopatadine small molecule P35367 Histamine H1 receptor approved DB00768 Olopatadine small molecule P23297 Protein S100-A1 approved DB00768 Olopatadine small molecule P04271 Protein S100-B approved DB00768 Olopatadine small molecule Q99584 Protein S100-A13 approved DB00768 Olopatadine small molecule P29034 Protein S100-A2 approved|investigational DB00770 Alprostadil small molecule P34995 Prostaglandin E2 receptor EP1 subtype approved DB00771 Clidinium small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00772 Malathion small molecule P06276 Cholinesterase approved DB00773 Etoposide small molecule P11388 DNA topoisomerase 2-alpha approved DB00773 Etoposide small molecule Q02880 DNA topoisomerase 2-beta approved|investigational DB00774 Hydroflumethiazide small molecule Q13621 Solute carrier family 12 member 1 approved|investigational DB00774 Hydroflumethiazide small molecule P00915 Carbonic anhydrase 1 approved|investigational DB00774 Hydroflumethiazide small molecule P00918 Carbonic anhydrase 2 approved|investigational DB00774 Hydroflumethiazide small molecule P22748 Carbonic anhydrase 4 approved|investigational DB00774 Hydroflumethiazide small molecule Q16790 Carbonic anhydrase 9 approved|investigational DB00774 Hydroflumethiazide small molecule O43570 Carbonic anhydrase 12 approved|investigational DB00774 Hydroflumethiazide small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved|investigational DB00774 Hydroflumethiazide small molecule Q12791 Calcium-activated potassium channel subunit alpha-1 approved DB00775 Tirofiban small molecule P08514 Integrin alpha-IIb approved DB00775 Tirofiban small molecule P05106 Integrin beta-3 approved DB00776 Oxcarbazepine small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB00777 Propiomazine small molecule P35367 Histamine H1 receptor approved DB00777 Propiomazine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00777 Propiomazine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00777 Propiomazine small molecule P14416 D(2) dopamine receptor approved DB00777 Propiomazine small molecule P21917 D(4) dopamine receptor approved DB00777 Propiomazine small molecule P25100 Alpha-1D adrenergic receptor approved DB00777 Propiomazine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00777 Propiomazine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00777 Propiomazine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00777 Propiomazine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational|withdrawn DB00778 Roxithromycin small molecule P08183 Multidrug resistance protein 1 approved DB00780 Phenelzine small molecule P21397 Amine oxidase [flavin-containing] A approved DB00780 Phenelzine small molecule P27338 Amine oxidase [flavin-containing] B approved DB00780 Phenelzine small molecule P80404 4-aminobutyrate aminotransferase, mitochondrial approved DB00780 Phenelzine small molecule Q8TD30 Alanine aminotransferase 2 approved DB00782 Propantheline small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational|vet_approved DB00783 Estradiol small molecule P03372 Estrogen receptor approved|investigational|vet_approved DB00783 Estradiol small molecule Q92731 Estrogen receptor beta approved|investigational|vet_approved DB00783 Estradiol small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational|vet_approved DB00783 Estradiol small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|investigational|vet_approved DB00783 Estradiol small molecule Q15596 Nuclear receptor coactivator 2 approved|investigational|vet_approved DB00783 Estradiol small molecule Q14457 Beclin-1 approved|investigational|vet_approved DB00783 Estradiol small molecule P37059 Estradiol 17-beta-dehydrogenase 2 approved|investigational|vet_approved DB00783 Estradiol small molecule P62508 Estrogen-related receptor gamma approved DB00784 Mefenamic acid small molecule P35354 Prostaglandin G/H synthase 2 approved DB00784 Mefenamic acid small molecule P23219 Prostaglandin G/H synthase 1 approved|vet_approved DB00788 Naproxen small molecule P23219 Prostaglandin G/H synthase 1 approved|vet_approved DB00788 Naproxen small molecule P35354 Prostaglandin G/H synthase 2 approved DB00790 Perindopril small molecule P12821 Angiotensin-converting enzyme approved DB00790 Perindopril small molecule Q6FHJ7 Secreted frizzled-related protein 4 approved|vet_approved DB00792 Tripelennamine small molecule P35367 Histamine H1 receptor approved|vet_approved DB00794 Primidone small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|vet_approved DB00794 Primidone small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|vet_approved DB00794 Primidone small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|vet_approved DB00794 Primidone small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|vet_approved DB00794 Primidone small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|vet_approved DB00794 Primidone small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|vet_approved DB00794 Primidone small molecule P42262 Glutamate receptor 2 approved|vet_approved DB00794 Primidone small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved|vet_approved DB00794 Primidone small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00795 Sulfasalazine small molecule P09917 Arachidonate 5-lipoxygenase approved DB00795 Sulfasalazine small molecule P35354 Prostaglandin G/H synthase 2 approved DB00795 Sulfasalazine small molecule P23219 Prostaglandin G/H synthase 1 approved DB00795 Sulfasalazine small molecule P37231 Peroxisome proliferator-activated receptor gamma approved DB00795 Sulfasalazine small molecule O15111 Inhibitor of nuclear factor kappa-B kinase subunit alpha approved DB00795 Sulfasalazine small molecule O14920 Inhibitor of nuclear factor kappa-B kinase subunit beta approved DB00795 Sulfasalazine small molecule P24557 Thromboxane-A synthase approved DB00795 Sulfasalazine small molecule P04054 Phospholipase A2 approved|vet_approved DB00797 Tolazoline small molecule P35367 Histamine H1 receptor approved|vet_approved DB00797 Tolazoline small molecule P25021 Histamine H2 receptor approved|vet_approved DB00798 Gentamicin small molecule P98164 Low-density lipoprotein receptor-related protein 2 approved|vet_approved DB00798 Gentamicin small molecule P00374 Dihydrofolate reductase approved|investigational DB00799 Tazarotene small molecule P10276 Retinoic acid receptor alpha approved|investigational DB00799 Tazarotene small molecule P28702 Retinoic acid receptor RXR-beta approved|investigational DB00799 Tazarotene small molecule P13631 Retinoic acid receptor gamma approved|investigational DB00799 Tazarotene small molecule P10826 Retinoic acid receptor beta approved DB00800 Fenoldopam small molecule P25100 Alpha-1D adrenergic receptor approved|illicit|withdrawn DB00801 Halazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit|withdrawn DB00801 Halazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit|withdrawn DB00801 Halazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit|withdrawn DB00801 Halazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit|withdrawn DB00801 Halazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|illicit|withdrawn DB00801 Halazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|illicit|withdrawn DB00801 Halazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|illicit|withdrawn DB00801 Halazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|illicit|withdrawn DB00801 Halazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|illicit|withdrawn DB00801 Halazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|illicit|withdrawn DB00801 Halazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|illicit|withdrawn DB00801 Halazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|illicit|withdrawn DB00801 Halazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|illicit|withdrawn DB00801 Halazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|illicit|withdrawn DB00801 Halazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB00802 Alfentanil small molecule P35372 Mu-type opioid receptor approved DB00804 Dicyclomine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00804 Dicyclomine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00805 Minaprine small molecule P21397 Amine oxidase [flavin-containing] A approved DB00805 Minaprine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00805 Minaprine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB00805 Minaprine small molecule P22303 Acetylcholinesterase approved DB00805 Minaprine small molecule P31645 Sodium-dependent serotonin transporter approved DB00805 Minaprine small molecule P14416 D(2) dopamine receptor approved DB00805 Minaprine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00806 Pentoxifylline small molecule Q07343 cAMP-specific 3',5'-cyclic phosphodiesterase 4B approved|investigational DB00806 Pentoxifylline small molecule P30542 Adenosine receptor A1 approved|investigational DB00806 Pentoxifylline small molecule O76074 cGMP-specific 3',5'-cyclic phosphodiesterase approved|investigational DB00806 Pentoxifylline small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved|investigational DB00806 Pentoxifylline small molecule P21589 5'-nucleotidase approved DB00808 Indapamide small molecule P51787 Potassium voltage-gated channel subfamily KQT member 1 {ECO:0000305} approved DB00808 Indapamide small molecule P15382 Potassium voltage-gated channel subfamily E member 1 approved|investigational DB00809 Tropicamide small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB00809 Tropicamide small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00809 Tropicamide small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00809 Tropicamide small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB00810 Biperiden small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00810 Biperiden small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB00811 Ribavirin small molecule P20839 Inosine-5'-monophosphate dehydrogenase 1 {ECO:0000255|HAMAP-Rule:MF_03156} approved DB00811 Ribavirin small molecule P55263 Adenosine kinase approved DB00811 Ribavirin small molecule P12268 Inosine-5'-monophosphate dehydrogenase 2 {ECO:0000255|HAMAP-Rule:MF_03156} approved DB00811 Ribavirin small molecule P49902 Cytosolic purine 5'-nucleotidase approved DB00811 Ribavirin small molecule P22413 Ectonucleotide pyrophosphatase/phosphodiesterase family member 1 approved|vet_approved DB00812 Phenylbutazone small molecule P35354 Prostaglandin G/H synthase 2 approved|vet_approved DB00812 Phenylbutazone small molecule Q16647 Prostacyclin synthase approved|vet_approved DB00812 Phenylbutazone small molecule P23219 Prostaglandin G/H synthase 1 approved|illicit|investigational|vet_approved DB00813 Fentanyl small molecule P35372 Mu-type opioid receptor approved|illicit|investigational|vet_approved DB00813 Fentanyl small molecule P41143 Delta-type opioid receptor approved|vet_approved DB00814 Meloxicam small molecule P35354 Prostaglandin G/H synthase 2 approved|vet_approved DB00814 Meloxicam small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational|vet_approved DB00818 Propofol small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|investigational|vet_approved DB00818 Propofol small molecule P35499 Sodium channel protein type 4 subunit alpha approved|investigational|vet_approved DB00818 Propofol small molecule Q99250 Sodium channel protein type 2 subunit alpha approved|investigational|vet_approved DB00818 Propofol small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|vet_approved DB00819 Acetazolamide small molecule P00915 Carbonic anhydrase 1 approved|vet_approved DB00819 Acetazolamide small molecule P00918 Carbonic anhydrase 2 approved|vet_approved DB00819 Acetazolamide small molecule P22748 Carbonic anhydrase 4 approved|vet_approved DB00819 Acetazolamide small molecule O43570 Carbonic anhydrase 12 approved|vet_approved DB00819 Acetazolamide small molecule Q9ULX7 Carbonic anhydrase 14 approved|vet_approved DB00819 Acetazolamide small molecule P07451 Carbonic anhydrase 3 approved|vet_approved DB00819 Acetazolamide small molecule P43166 Carbonic anhydrase 7 approved|vet_approved DB00819 Acetazolamide small molecule P29972 Aquaporin-1 approved|investigational DB00820 Tadalafil small molecule O76074 cGMP-specific 3',5'-cyclic phosphodiesterase approved|investigational DB00820 Tadalafil small molecule Q9HCR9 Dual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A approved DB00822 Disulfiram small molecule P05091 Aldehyde dehydrogenase, mitochondrial approved DB00822 Disulfiram small molecule P09172 Dopamine beta-hydroxylase approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P30536 Translocator protein approved|illicit|investigational|vet_approved DB00829 Diazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00831 Trifluoperazine small molecule P14416 D(2) dopamine receptor approved|investigational DB00831 Trifluoperazine small molecule P63316 Troponin C, slow skeletal and cardiac muscles approved|investigational DB00831 Trifluoperazine small molecule P26447 Protein S100-A4 approved|investigational DB00834 Mifepristone small molecule P06401 Progesterone receptor approved|investigational DB00834 Mifepristone small molecule P04150 Glucocorticoid receptor approved|investigational DB00834 Mifepristone small molecule P07288 Prostate-specific antigen approved|investigational DB00834 Mifepristone small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB00835 Brompheniramine small molecule P35367 Histamine H1 receptor approved DB00835 Brompheniramine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00835 Brompheniramine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB00835 Brompheniramine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB00835 Brompheniramine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB00836 Loperamide small molecule P35372 Mu-type opioid receptor approved DB00836 Loperamide small molecule P41143 Delta-type opioid receptor approved DB00836 Loperamide small molecule O00555 Voltage-dependent P/Q-type calcium channel subunit alpha-1A approved DB00836 Loperamide small molecule P01189 Pro-opiomelanocortin approved DB00836 Loperamide small molecule Q14994 Nuclear receptor subfamily 1 group I member 3 approved|investigational DB00837 Progabide small molecule Q9UBS5 Gamma-aminobutyric acid type B receptor subunit 1 approved|investigational DB00837 Progabide small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00838 Clocortolone small molecule P04150 Glucocorticoid receptor approved|investigational DB00839 Tolazamide small molecule Q09428 ATP-binding cassette sub-family C member 8 approved DB00841 Dobutamine small molecule P03372 Estrogen receptor approved DB00842 Oxazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00842 Oxazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB00842 Oxazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB00842 Oxazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved DB00842 Oxazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved DB00842 Oxazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved DB00842 Oxazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved DB00842 Oxazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved DB00842 Oxazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved DB00842 Oxazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved DB00842 Oxazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved DB00842 Oxazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved DB00842 Oxazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved DB00842 Oxazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved DB00842 Oxazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00843 Donepezil small molecule P22303 Acetylcholinesterase approved DB00843 Donepezil small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00844 Nalbuphine small molecule P35372 Mu-type opioid receptor approved DB00844 Nalbuphine small molecule P41143 Delta-type opioid receptor approved|investigational DB00845 Clofazimine small molecule O95342 Bile salt export pump approved DB00846 Flurandrenolide small molecule P04150 Glucocorticoid receptor approved|investigational DB00847 Cysteamine small molecule P61278 Somatostatin approved|investigational|vet_approved|withdrawn DB00848 Levamisole small molecule P32297 Neuronal acetylcholine receptor subunit alpha-3 approved DB00849 Methylphenobarbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00849 Methylphenobarbital small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB00849 Methylphenobarbital small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB00849 Methylphenobarbital small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved DB00849 Methylphenobarbital small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved DB00849 Methylphenobarbital small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved DB00849 Methylphenobarbital small molecule P42262 Glutamate receptor 2 approved DB00849 Methylphenobarbital small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved DB00849 Methylphenobarbital small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB00850 Perphenazine small molecule P14416 D(2) dopamine receptor approved|investigational DB00851 Dacarbazine small molecule Q14181 DNA polymerase alpha subunit B approved|investigational DB00851 Dacarbazine small molecule P52209 6-phosphogluconate dehydrogenase, decarboxylating approved DB00852 Pseudoephedrine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00852 Pseudoephedrine small molecule P31645 Sodium-dependent serotonin transporter approved DB00852 Pseudoephedrine small molecule O95644 Nuclear factor of activated T-cells, cytoplasmic 1 approved DB00852 Pseudoephedrine small molecule P01375 Tumor necrosis factor approved DB00852 Pseudoephedrine small molecule P18846 Cyclic AMP-dependent transcription factor ATF-1 approved DB00852 Pseudoephedrine small molecule P60568 Interleukin-2 approved DB00855 Aminolevulinic acid small molecule P13716 Delta-aminolevulinic acid dehydratase approved|investigational|vet_approved DB00857 Terbinafine small molecule Q14534 Squalene monooxygenase approved|vet_approved DB00860 Prednisolone small molecule P04150 Glucocorticoid receptor approved|investigational DB00861 Diflunisal small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB00861 Diflunisal small molecule P23219 Prostaglandin G/H synthase 1 approved DB00862 Vardenafil small molecule O76074 cGMP-specific 3',5'-cyclic phosphodiesterase approved DB00862 Vardenafil small molecule P18545 Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma approved DB00862 Vardenafil small molecule Q13956 Retinal cone rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma approved DB00863 Ranitidine small molecule P25021 Histamine H2 receptor approved DB00863 Ranitidine small molecule P22303 Acetylcholinesterase approved DB00863 Ranitidine small molecule P06276 Cholinesterase approved|investigational DB00864 Tacrolimus small molecule P62942 Peptidyl-prolyl cis-trans isomerase FKBP1A approved|withdrawn DB00866 Alprenolol small molecule P13945 Beta-3 adrenergic receptor approved DB00868 Benzonatate small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB00869 Dorzolamide small molecule P00918 Carbonic anhydrase 2 approved DB00869 Dorzolamide small molecule P22748 Carbonic anhydrase 4 approved DB00869 Dorzolamide small molecule P00915 Carbonic anhydrase 1 approved DB00869 Dorzolamide small molecule P07451 Carbonic anhydrase 3 approved|withdrawn DB00870 Suprofen small molecule P23219 Prostaglandin G/H synthase 1 approved|withdrawn DB00870 Suprofen small molecule P35354 Prostaglandin G/H synthase 2 approved DB00871 Terbutaline small molecule P13945 Beta-3 adrenergic receptor approved DB00873 Loteprednol small molecule P04150 Glucocorticoid receptor approved|investigational|withdrawn DB00875 Flupentixol small molecule P14416 D(2) dopamine receptor approved|investigational|withdrawn DB00875 Flupentixol small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational|withdrawn DB00875 Flupentixol small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB00876 Eprosartan small molecule P30556 Type-1 angiotensin II receptor approved|investigational DB00877 Sirolimus small molecule P42345 Serine/threonine-protein kinase mTOR approved|investigational DB00877 Sirolimus small molecule P62942 Peptidyl-prolyl cis-trans isomerase FKBP1A approved|investigational DB00877 Sirolimus small molecule P09038 Fibroblast growth factor 2 approved|vet_approved DB00880 Chlorothiazide small molecule P55017 Solute carrier family 12 member 3 approved|vet_approved DB00880 Chlorothiazide small molecule P00915 Carbonic anhydrase 1 approved|vet_approved DB00880 Chlorothiazide small molecule P00918 Carbonic anhydrase 2 approved|vet_approved DB00880 Chlorothiazide small molecule P22748 Carbonic anhydrase 4 approved|investigational DB00881 Quinapril small molecule P12821 Angiotensin-converting enzyme approved|investigational DB00882 Clomifene small molecule P03372 Estrogen receptor approved|investigational DB00882 Clomifene small molecule P04278 Sex hormone-binding globulin approved|investigational DB00884 Risedronate small molecule P14324 Farnesyl pyrophosphate synthase approved DB00887 Bumetanide small molecule Q13621 Solute carrier family 12 member 1 approved DB00887 Bumetanide small molecule P55011 Solute carrier family 12 member 2 approved DB00887 Bumetanide small molecule Q9UP95 Solute carrier family 12 member 4 approved DB00887 Bumetanide small molecule Q9H2X9 Solute carrier family 12 member 5 approved DB00887 Bumetanide small molecule P13569 Cystic fibrosis transmembrane conductance regulator approved|investigational DB00890 Dienestrol small molecule P03372 Estrogen receptor approved|investigational DB00890 Dienestrol small molecule P04278 Sex hormone-binding globulin approved DB00895 Benzylpenicilloyl Polylysine small molecule P30273 High affinity immunoglobulin epsilon receptor subunit gamma approved DB00895 Benzylpenicilloyl Polylysine small molecule P12319 High affinity immunoglobulin epsilon receptor subunit alpha approved DB00896 Rimexolone small molecule P04150 Glucocorticoid receptor approved|investigational DB00897 Triazolam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB00897 Triazolam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|investigational DB00897 Triazolam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|investigational DB00897 Triazolam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|investigational DB00897 Triazolam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|investigational DB00897 Triazolam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|investigational DB00897 Triazolam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|investigational DB00897 Triazolam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|investigational DB00897 Triazolam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|investigational DB00897 Triazolam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|investigational DB00897 Triazolam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|investigational DB00897 Triazolam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|investigational DB00897 Triazolam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|investigational DB00897 Triazolam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|investigational DB00897 Triazolam small molecule P30536 Translocator protein approved|investigational DB00897 Triazolam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00898 Ethanol small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB00898 Ethanol small molecule P23415 Glycine receptor subunit alpha-1 approved DB00898 Ethanol small molecule P23416 Glycine receptor subunit alpha-2 approved DB00898 Ethanol small molecule Q02641 Voltage-dependent L-type calcium channel subunit beta-1 approved DB00898 Ethanol small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB00898 Ethanol small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved DB00898 Ethanol small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved DB00898 Ethanol small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB00898 Ethanol small molecule P42261 Glutamate receptor 1 approved DB00898 Ethanol small molecule Q06432 Voltage-dependent calcium channel gamma-1 subunit approved DB00898 Ethanol small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB00898 Ethanol small molecule P42262 Glutamate receptor 2 approved DB00898 Ethanol small molecule P48058 Glutamate receptor 4 approved DB00898 Ethanol small molecule P42263 Glutamate receptor 3 approved DB00898 Ethanol small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved DB00898 Ethanol small molecule P17787 Neuronal acetylcholine receptor subunit beta-2 approved DB00898 Ethanol small molecule P48549 G protein-activated inward rectifier potassium channel 1 approved DB00898 Ethanol small molecule P48051 G protein-activated inward rectifier potassium channel 2 approved DB00898 Ethanol small molecule P19320 Vascular cell adhesion protein 1 approved DB00898 Ethanol small molecule Q99808 Equilibrative nucleoside transporter 1 approved DB00898 Ethanol small molecule P48544 G protein-activated inward rectifier potassium channel 4 approved DB00898 Ethanol small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved DB00898 Ethanol small molecule Q9UGM1 Neuronal acetylcholine receptor subunit alpha-9 approved DB00898 Ethanol small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved DB00898 Ethanol small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved DB00898 Ethanol small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved DB00898 Ethanol small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved DB00898 Ethanol small molecule P30926 Neuronal acetylcholine receptor subunit beta-4 approved DB00898 Ethanol small molecule P32297 Neuronal acetylcholine receptor subunit alpha-3 approved DB00898 Ethanol small molecule Q15825 Neuronal acetylcholine receptor subunit alpha-6 approved DB00898 Ethanol small molecule Q05901 Neuronal acetylcholine receptor subunit beta-3 approved DB00898 Ethanol small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved DB00898 Ethanol small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved DB00898 Ethanol small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved DB00898 Ethanol small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved DB00898 Ethanol small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved DB00898 Ethanol small molecule Q14542 Equilibrative nucleoside transporter 2 approved DB00898 Ethanol small molecule A5X5Y0 5-hydroxytryptamine receptor 3E approved DB00898 Ethanol small molecule O95264 5-hydroxytryptamine receptor 3B approved DB00898 Ethanol small molecule Q70Z44 5-hydroxytryptamine receptor 3D approved DB00898 Ethanol small molecule Q8WXA8 5-hydroxytryptamine receptor 3C approved DB00898 Ethanol small molecule Q9Y698 Voltage-dependent calcium channel gamma-2 subunit approved DB00899 Remifentanil small molecule P35372 Mu-type opioid receptor approved DB00899 Remifentanil small molecule P41143 Delta-type opioid receptor approved DB00900 Didanosine small molecule P00491 Purine nucleoside phosphorylase approved DB00902 Methdilazine small molecule P35367 Histamine H1 receptor approved|investigational DB00903 Etacrynic acid small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved|investigational DB00903 Etacrynic acid small molecule Q13621 Solute carrier family 12 member 1 approved|investigational DB00903 Etacrynic acid small molecule Q9UJU2 Lymphoid enhancer-binding factor 1 approved|investigational DB00903 Etacrynic acid small molecule P09211 Glutathione S-transferase P approved DB00904 Ondansetron small molecule Q13639 5-hydroxytryptamine receptor 4 approved DB00904 Ondansetron small molecule P35372 Mu-type opioid receptor approved|investigational DB00905 Bimatoprost small molecule P43088 Prostaglandin F2-alpha receptor approved|investigational DB00905 Bimatoprost small molecule P34995 Prostaglandin E2 receptor EP1 subtype approved|investigational DB00905 Bimatoprost small molecule P43115 Prostaglandin E2 receptor EP3 subtype approved|investigational DB00905 Bimatoprost small molecule P42330 Aldo-keto reductase family 1 member C3 approved|investigational DB00906 Tiagabine small molecule P30531 Sodium- and chloride-dependent GABA transporter 1 approved|illicit DB00907 Cocaine small molecule P23975 Sodium-dependent noradrenaline transporter approved|illicit DB00907 Cocaine small molecule P31645 Sodium-dependent serotonin transporter approved|illicit DB00907 Cocaine small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|illicit DB00907 Cocaine small molecule Q9UI33 Sodium channel protein type 11 subunit alpha approved|illicit DB00907 Cocaine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|illicit DB00907 Cocaine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|illicit DB00907 Cocaine small molecule Q99720 Sigma non-opioid intracellular receptor 1 approved|illicit DB00907 Cocaine small molecule P23141 Liver carboxylesterase 1 approved|investigational DB00908 Quinidine small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|investigational DB00908 Quinidine small molecule O00180 Potassium channel subfamily K member 1 approved|investigational DB00908 Quinidine small molecule Q9Y257 Potassium channel subfamily K member 6 approved|investigational DB00908 Quinidine small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB00908 Quinidine small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB00909 Zonisamide small molecule Q99250 Sodium channel protein type 2 subunit alpha approved|investigational DB00909 Zonisamide small molecule Q9NY46 Sodium channel protein type 3 subunit alpha approved|investigational DB00909 Zonisamide small molecule P35499 Sodium channel protein type 4 subunit alpha approved|investigational DB00909 Zonisamide small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|investigational DB00909 Zonisamide small molecule Q15858 Sodium channel protein type 9 subunit alpha {ECO:0000305} approved|investigational DB00909 Zonisamide small molecule Q9UI33 Sodium channel protein type 11 subunit alpha approved|investigational DB00909 Zonisamide small molecule Q07699 Sodium channel subunit beta-1 approved|investigational DB00909 Zonisamide small molecule O60939 Sodium channel subunit beta-2 approved|investigational DB00909 Zonisamide small molecule Q8IWT1 Sodium channel subunit beta-4 approved|investigational DB00909 Zonisamide small molecule O43497 Voltage-dependent T-type calcium channel subunit alpha-1G approved|investigational DB00909 Zonisamide small molecule O95180 Voltage-dependent T-type calcium channel subunit alpha-1H approved|investigational DB00909 Zonisamide small molecule Q9P0X4 Voltage-dependent T-type calcium channel subunit alpha-1I approved|investigational DB00909 Zonisamide small molecule P00915 Carbonic anhydrase 1 approved|investigational DB00909 Zonisamide small molecule P00918 Carbonic anhydrase 2 approved|investigational DB00909 Zonisamide small molecule P07451 Carbonic anhydrase 3 approved|investigational DB00909 Zonisamide small molecule P22748 Carbonic anhydrase 4 approved|investigational DB00909 Zonisamide small molecule P35218 Carbonic anhydrase 5A, mitochondrial approved|investigational DB00909 Zonisamide small molecule P23280 Carbonic anhydrase 6 approved|investigational DB00909 Zonisamide small molecule P43166 Carbonic anhydrase 7 approved|investigational DB00909 Zonisamide small molecule P35219 Carbonic anhydrase-related protein approved|investigational DB00909 Zonisamide small molecule Q16790 Carbonic anhydrase 9 approved|investigational DB00909 Zonisamide small molecule Q9NS85 Carbonic anhydrase-related protein 10 approved|investigational DB00909 Zonisamide small molecule O75493 Carbonic anhydrase-related protein 11 approved|investigational DB00909 Zonisamide small molecule O43570 Carbonic anhydrase 12 approved|investigational DB00909 Zonisamide small molecule Q8N1Q1 Carbonic anhydrase 13 approved|investigational DB00909 Zonisamide small molecule Q9ULX7 Carbonic anhydrase 14 approved|investigational DB00909 Zonisamide small molecule P27338 Amine oxidase [flavin-containing] B approved|investigational DB00909 Zonisamide small molecule P21397 Amine oxidase [flavin-containing] A approved|investigational DB00910 Paricalcitol small molecule P11473 Vitamin D3 receptor approved|investigational DB00912 Repaglinide small molecule Q09428 ATP-binding cassette sub-family C member 8 approved|investigational DB00912 Repaglinide small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|illicit DB00913 Anileridine small molecule P35372 Mu-type opioid receptor approved|investigational|withdrawn DB00914 Phenformin small molecule Q13131 5'-AMP-activated protein kinase catalytic subunit alpha-1 approved DB00915 Amantadine small molecule P14416 D(2) dopamine receptor approved DB00916 Metronidazole small molecule Q16850 Lanosterol 14-alpha demethylase approved DB00917 Dinoprostone small molecule P34995 Prostaglandin E2 receptor EP1 subtype approved DB00917 Dinoprostone small molecule P43115 Prostaglandin E2 receptor EP3 subtype approved DB00920 Ketotifen small molecule P35367 Histamine H1 receptor approved DB00920 Ketotifen small molecule P52209 6-phosphogluconate dehydrogenase, decarboxylating approved|illicit|investigational|vet_approved DB00921 Buprenorphine small molecule P35372 Mu-type opioid receptor approved|illicit|investigational|vet_approved DB00921 Buprenorphine small molecule P41143 Delta-type opioid receptor approved|illicit|investigational|vet_approved DB00921 Buprenorphine small molecule P41146 Nociceptin receptor approved|investigational DB00922 Levosimendan small molecule P63316 Troponin C, slow skeletal and cardiac muscles approved|investigational DB00922 Levosimendan small molecule Q14432 cGMP-inhibited 3',5'-cyclic phosphodiesterase A approved DB00924 Cyclobenzaprine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB00925 Phenoxybenzamine small molecule P25100 Alpha-1D adrenergic receptor withdrawn DB00926 Etretinate small molecule P10276 Retinoic acid receptor alpha withdrawn DB00926 Etretinate small molecule P19793 Retinoic acid receptor RXR-alpha withdrawn DB00926 Etretinate small molecule P10826 Retinoic acid receptor beta withdrawn DB00926 Etretinate small molecule P48443 Retinoic acid receptor RXR-gamma withdrawn DB00926 Etretinate small molecule P28702 Retinoic acid receptor RXR-beta withdrawn DB00926 Etretinate small molecule P13631 Retinoic acid receptor gamma approved DB00927 Famotidine small molecule P25021 Histamine H2 receptor approved|investigational DB00928 Azacitidine small molecule P26358 DNA (cytosine-5)-methyltransferase 1 approved DB00929 Misoprostol small molecule P43115 Prostaglandin E2 receptor EP3 subtype approved|investigational DB00933 Mesoridazine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB00933 Mesoridazine small molecule P14416 D(2) dopamine receptor approved|investigational DB00934 Maprotiline small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB00934 Maprotiline small molecule P35367 Histamine H1 receptor approved|investigational DB00934 Maprotiline small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00934 Maprotiline small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00934 Maprotiline small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB00934 Maprotiline small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB00934 Maprotiline small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB00934 Maprotiline small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB00934 Maprotiline small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational DB00934 Maprotiline small molecule P14416 D(2) dopamine receptor approved|investigational DB00935 Oxymetazoline small molecule P25100 Alpha-1D adrenergic receptor approved|investigational|vet_approved DB00936 Salicylic acid small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational|vet_approved DB00936 Salicylic acid small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational|vet_approved DB00936 Salicylic acid small molecule Q04828 Aldo-keto reductase family 1 member C1 approved|illicit DB00937 Diethylpropion small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00938 Salmeterol small molecule P13945 Beta-3 adrenergic receptor approved|vet_approved DB00939 Meclofenamic acid small molecule P23219 Prostaglandin G/H synthase 1 approved|vet_approved DB00939 Meclofenamic acid small molecule P35354 Prostaglandin G/H synthase 2 approved|vet_approved DB00939 Meclofenamic acid small molecule P09917 Arachidonate 5-lipoxygenase approved|vet_approved DB00939 Meclofenamic acid small molecule O43526 Potassium voltage-gated channel subfamily KQT member 2 {ECO:0000305} approved|vet_approved DB00939 Meclofenamic acid small molecule O43525 Potassium voltage-gated channel subfamily KQT member 3 {ECO:0000305} approved|investigational DB00940 Methantheline small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00940 Methantheline small molecule P25021 Histamine H2 receptor approved DB00941 Hexafluronium small molecule P06276 Cholinesterase approved DB00944 Demecarium small molecule P22303 Acetylcholinesterase approved DB00944 Demecarium small molecule P06276 Cholinesterase approved|vet_approved DB00945 Acetylsalicylic acid small molecule P23219 Prostaglandin G/H synthase 1 approved|vet_approved DB00945 Acetylsalicylic acid small molecule P35354 Prostaglandin G/H synthase 2 approved|vet_approved DB00945 Acetylsalicylic acid small molecule Q04828 Aldo-keto reductase family 1 member C1 approved|vet_approved DB00945 Acetylsalicylic acid small molecule Q13131 5'-AMP-activated protein kinase catalytic subunit alpha-1 approved|vet_approved DB00945 Acetylsalicylic acid small molecule P25101 Endothelin-1 receptor {ECO:0000305} approved|vet_approved DB00945 Acetylsalicylic acid small molecule O14920 Inhibitor of nuclear factor kappa-B kinase subunit beta approved|vet_approved DB00945 Acetylsalicylic acid small molecule P04637 Cellular tumor antigen p53 approved|vet_approved DB00945 Acetylsalicylic acid small molecule P11021 Endoplasmic reticulum chaperone BiP {ECO:0000305} approved|vet_approved DB00945 Acetylsalicylic acid small molecule P51812 Ribosomal protein S6 kinase alpha-3 approved|vet_approved DB00945 Acetylsalicylic acid small molecule P25963 NF-kappa-B inhibitor alpha approved|vet_approved DB00945 Acetylsalicylic acid small molecule Q00653 Nuclear factor NF-kappa-B p100 subunit approved|investigational DB00946 Phenprocoumon small molecule Q9BQB6 Vitamin K epoxide reductase complex subunit 1 approved|investigational DB00947 Fulvestrant small molecule P03372 Estrogen receptor approved DB00949 Felbamate small molecule Q13224 Glutamate receptor ionotropic, NMDA 2B approved DB00949 Felbamate small molecule Q12879 Glutamate receptor ionotropic, NMDA 2A approved|investigational DB00950 Fexofenadine small molecule P35367 Histamine H1 receptor approved|investigational DB00951 Isoniazid small molecule P10632 Cytochrome P450 2C8 approved|investigational DB00951 Isoniazid small molecule P08684 Cytochrome P450 3A4 approved|investigational DB00951 Isoniazid small molecule P33261 Cytochrome P450 2C19 approved|illicit DB00956 Hydrocodone small molecule P35372 Mu-type opioid receptor approved|illicit DB00956 Hydrocodone small molecule P41143 Delta-type opioid receptor approved|investigational DB00957 Norgestimate small molecule P06401 Progesterone receptor approved|investigational DB00957 Norgestimate small molecule P03372 Estrogen receptor approved|investigational DB00957 Norgestimate small molecule P10275 Androgen receptor approved|vet_approved DB00959 Methylprednisolone small molecule P04150 Glucocorticoid receptor approved|investigational DB00960 Pindolol small molecule P13945 Beta-3 adrenergic receptor approved|illicit|investigational DB00962 Zaleplon small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit|investigational DB00962 Zaleplon small molecule P30536 Translocator protein approved DB00963 Bromfenac small molecule P35354 Prostaglandin G/H synthase 2 approved DB00963 Bromfenac small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB00966 Telmisartan small molecule P30556 Type-1 angiotensin II receptor approved|investigational DB00966 Telmisartan small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|investigational DB00967 Desloratadine small molecule P35367 Histamine H1 receptor approved|investigational DB00970 Dactinomycin small molecule P11388 DNA topoisomerase 2-alpha approved DB00972 Azelastine small molecule P35367 Histamine H1 receptor approved DB00973 Ezetimibe small molecule P35610 Sterol O-acyltransferase 1 approved DB00973 Ezetimibe small molecule Q9UHC9 NPC1-like intracellular cholesterol transporter 1 {ECO:0000312|HGNC:HGNC:7898} approved DB00973 Ezetimibe small molecule P15144 Aminopeptidase N {ECO:0000305} approved DB00975 Dipyridamole small molecule Q9Y233 cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A approved DB00975 Dipyridamole small molecule P00813 Adenosine deaminase approved DB00975 Dipyridamole small molecule O76074 cGMP-specific 3',5'-cyclic phosphodiesterase approved DB00975 Dipyridamole small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved DB00975 Dipyridamole small molecule P53805 Calcipressin-1 approved DB00975 Dipyridamole small molecule P02763 Alpha-1-acid glycoprotein 1 approved DB00977 Ethinyl Estradiol small molecule P03372 Estrogen receptor approved DB00977 Ethinyl Estradiol small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB00977 Ethinyl Estradiol small molecule P04278 Sex hormone-binding globulin approved|investigational DB00978 Lomefloxacin small molecule P11388 DNA topoisomerase 2-alpha approved DB00979 Cyclopentolate small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB00981 Physostigmine small molecule P22303 Acetylcholinesterase approved|investigational DB00981 Physostigmine small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|investigational DB00981 Physostigmine small molecule P17787 Neuronal acetylcholine receptor subunit beta-2 approved DB00982 Isotretinoin small molecule P10276 Retinoic acid receptor alpha approved|investigational DB00983 Formoterol small molecule P13945 Beta-3 adrenergic receptor approved DB00985 Dimenhydrinate small molecule P35367 Histamine H1 receptor approved|investigational|vet_approved DB00986 Glycopyrronium small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational|vet_approved DB00986 Glycopyrronium small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational|vet_approved DB00986 Glycopyrronium small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB00987 Cytarabine small molecule P06746 DNA polymerase beta approved DB00988 Dopamine small molecule P14416 D(2) dopamine receptor approved DB00988 Dopamine small molecule P35462 D(3) dopamine receptor approved DB00988 Dopamine small molecule P21917 D(4) dopamine receptor approved DB00988 Dopamine small molecule P09172 Dopamine beta-hydroxylase approved DB00988 Dopamine small molecule P34969 5-hydroxytryptamine receptor 7 approved DB00988 Dopamine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB00988 Dopamine small molecule P31645 Sodium-dependent serotonin transporter approved DB00988 Dopamine small molecule O95264 5-hydroxytryptamine receptor 3B approved DB00988 Dopamine small molecule P00441 Superoxide dismutase [Cu-Zn] approved DB00988 Dopamine small molecule Q05940 Synaptic vesicular amine transporter approved|investigational DB00989 Rivastigmine small molecule P22303 Acetylcholinesterase approved|investigational DB00989 Rivastigmine small molecule P06276 Cholinesterase approved|investigational DB00990 Exemestane small molecule P11511 Aromatase approved DB00991 Oxaprozin small molecule P23219 Prostaglandin G/H synthase 1 approved DB00991 Oxaprozin small molecule P35354 Prostaglandin G/H synthase 2 approved DB00993 Azathioprine small molecule P00492 Hypoxanthine-guanine phosphoribosyltransferase approved DB00993 Azathioprine small molecule P63000 Ras-related C3 botulinum toxin substrate 1 approved|vet_approved DB00994 Neomycin small molecule P41180 Extracellular calcium-sensing receptor {ECO:0000305} approved|investigational DB00995 Auranofin small molecule P30044 Peroxiredoxin-5, mitochondrial approved|investigational DB00995 Auranofin small molecule O14920 Inhibitor of nuclear factor kappa-B kinase subunit beta approved|investigational DB00996 Gabapentin small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved|investigational DB00996 Gabapentin small molecule Q9NY47 Voltage-dependent calcium channel subunit alpha-2/delta-2 approved|investigational DB00996 Gabapentin small molecule Q00975 Voltage-dependent N-type calcium channel subunit alpha-1B approved|investigational DB00996 Gabapentin small molecule P30542 Adenosine receptor A1 approved|investigational DB00996 Gabapentin small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved|investigational DB00996 Gabapentin small molecule Q9UBS5 Gamma-aminobutyric acid type B receptor subunit 1 approved|investigational DB00996 Gabapentin small molecule O75899 Gamma-aminobutyric acid type B receptor subunit 2 approved|investigational DB00997 Doxorubicin small molecule P11388 DNA topoisomerase 2-alpha approved|investigational DB00997 Doxorubicin small molecule Q14978 Nucleolar and coiled-body phosphoprotein 1 {ECO:0000305} approved|vet_approved DB00999 Hydrochlorothiazide small molecule P55017 Solute carrier family 12 member 3 approved|vet_approved DB00999 Hydrochlorothiazide small molecule P00915 Carbonic anhydrase 1 approved|vet_approved DB00999 Hydrochlorothiazide small molecule P00918 Carbonic anhydrase 2 approved|vet_approved DB00999 Hydrochlorothiazide small molecule P22748 Carbonic anhydrase 4 approved|vet_approved DB00999 Hydrochlorothiazide small molecule Q16790 Carbonic anhydrase 9 approved|vet_approved DB00999 Hydrochlorothiazide small molecule O43570 Carbonic anhydrase 12 approved|vet_approved DB00999 Hydrochlorothiazide small molecule Q12791 Calcium-activated potassium channel subunit alpha-1 approved|vet_approved DB01001 Salbutamol small molecule P13945 Beta-3 adrenergic receptor approved DB01003 Cromoglicic acid small molecule Q12791 Calcium-activated potassium channel subunit alpha-1 approved DB01003 Cromoglicic acid small molecule P25815 Protein S100-P approved DB01005 Hydroxyurea small molecule P23921 Ribonucleoside-diphosphate reductase large subunit approved|investigational DB01006 Letrozole small molecule P11511 Aromatase approved DB01007 Tioconazole small molecule Q16850 Lanosterol 14-alpha demethylase approved|vet_approved DB01009 Ketoprofen small molecule P23219 Prostaglandin G/H synthase 1 approved|vet_approved DB01009 Ketoprofen small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB01011 Metyrapone small molecule P15538 Cytochrome P450 11B1, mitochondrial approved DB01012 Cinacalcet small molecule P41180 Extracellular calcium-sensing receptor {ECO:0000305} approved|investigational DB01014 Balsalazide small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|investigational DB01014 Balsalazide small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB01014 Balsalazide small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB01014 Balsalazide small molecule P09917 Arachidonate 5-lipoxygenase approved DB01015 Sulfamethoxazole small molecule P09211 Glutathione S-transferase P approved DB01016 Glyburide small molecule Q09428 ATP-binding cassette sub-family C member 8 approved DB01016 Glyburide small molecule P48544 G protein-activated inward rectifier potassium channel 4 approved DB01016 Glyburide small molecule O60706 ATP-binding cassette sub-family C member 9 approved DB01016 Glyburide small molecule O95342 Bile salt export pump approved DB01016 Glyburide small molecule O95477 ATP-binding cassette sub-family A member 1 approved DB01016 Glyburide small molecule P13569 Cystic fibrosis transmembrane conductance regulator approved DB01016 Glyburide small molecule P50416 Carnitine O-palmitoyltransferase 1, liver isoform approved|investigational DB01017 Minocycline small molecule P01584 Interleukin-1 beta approved|investigational DB01017 Minocycline small molecule P09917 Arachidonate 5-lipoxygenase approved|investigational DB01017 Minocycline small molecule P14780 Matrix metalloproteinase-9 approved|investigational DB01017 Minocycline small molecule P15692 Vascular endothelial growth factor A approved|investigational DB01017 Minocycline small molecule P29466 Caspase-1 approved|investigational DB01017 Minocycline small molecule P99999 Cytochrome c approved DB01019 Bethanechol small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB01019 Bethanechol small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB01019 Bethanechol small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB01019 Bethanechol small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB01020 Isosorbide Mononitrate small molecule P33402 Guanylate cyclase soluble subunit alpha-2 approved|vet_approved DB01021 Trichlormethiazide small molecule Q13621 Solute carrier family 12 member 1 approved|vet_approved DB01021 Trichlormethiazide small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved|vet_approved DB01021 Trichlormethiazide small molecule P00915 Carbonic anhydrase 1 approved|vet_approved DB01021 Trichlormethiazide small molecule P00918 Carbonic anhydrase 2 approved|vet_approved DB01021 Trichlormethiazide small molecule P22748 Carbonic anhydrase 4 approved|investigational DB01022 Phylloquinone small molecule P38435 Vitamin K-dependent gamma-carboxylase approved|investigational DB01023 Felodipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB01023 Felodipine small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved|investigational DB01023 Felodipine small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved|investigational DB01023 Felodipine small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved|investigational DB01023 Felodipine small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved|investigational DB01023 Felodipine small molecule O95180 Voltage-dependent T-type calcium channel subunit alpha-1H approved|investigational DB01023 Felodipine small molecule Q9NY47 Voltage-dependent calcium channel subunit alpha-2/delta-2 approved|investigational DB01023 Felodipine small molecule P54750 Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A approved|investigational DB01023 Felodipine small molecule P08235 Mineralocorticoid receptor approved|investigational DB01023 Felodipine small molecule P02585 Troponin C, skeletal muscle approved|investigational DB01023 Felodipine small molecule P63316 Troponin C, slow skeletal and cardiac muscles approved DB01024 Mycophenolic acid small molecule P20839 Inosine-5'-monophosphate dehydrogenase 1 {ECO:0000255|HAMAP-Rule:MF_03156} approved DB01024 Mycophenolic acid small molecule P12268 Inosine-5'-monophosphate dehydrogenase 2 {ECO:0000255|HAMAP-Rule:MF_03156} approved|investigational DB01025 Amlexanox small molecule Q99584 Protein S100-A13 approved|investigational DB01025 Amlexanox small molecule P05230 Fibroblast growth factor 1 approved|investigational DB01026 Ketoconazole small molecule P10275 Androgen receptor approved|investigational DB01026 Ketoconazole small molecule P11511 Aromatase approved|investigational DB01026 Ketoconazole small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB01026 Ketoconazole small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB01026 Ketoconazole small molecule Q14994 Nuclear receptor subfamily 1 group I member 3 approved|investigational|vet_approved DB01028 Methoxyflurane small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational|vet_approved DB01028 Methoxyflurane small molecule P42261 Glutamate receptor 1 approved|investigational|vet_approved DB01028 Methoxyflurane small molecule P23415 Glycine receptor subunit alpha-1 approved|investigational|vet_approved DB01028 Methoxyflurane small molecule P98194 Calcium-transporting ATPase type 2C member 1 approved|investigational|vet_approved DB01028 Methoxyflurane small molecule Q09470 Potassium voltage-gated channel subfamily A member 1 approved|investigational|vet_approved DB01028 Methoxyflurane small molecule P30049 ATP synthase subunit delta, mitochondrial {ECO:0000305} approved|investigational|vet_approved DB01028 Methoxyflurane small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB01029 Irbesartan small molecule P30556 Type-1 angiotensin II receptor approved|investigational DB01029 Irbesartan small molecule P05412 Transcription factor AP-1 approved|investigational DB01030 Topotecan small molecule P11387 DNA topoisomerase 1 approved|investigational DB01030 Topotecan small molecule Q969P6 DNA topoisomerase I, mitochondrial approved|investigational DB01032 Probenecid small molecule Q4U2R8 Solute carrier family 22 member 6 approved|investigational DB01032 Probenecid small molecule Q9NSA0 Solute carrier family 22 member 11 approved|investigational DB01032 Probenecid small molecule Q8TCC7 Solute carrier family 22 member 8 approved|investigational DB01032 Probenecid small molecule Q96RD7 Pannexin-1 approved DB01033 Mercaptopurine small molecule P00492 Hypoxanthine-guanine phosphoribosyltransferase approved DB01033 Mercaptopurine small molecule Q06203 Amidophosphoribosyltransferase approved DB01033 Mercaptopurine small molecule P20839 Inosine-5'-monophosphate dehydrogenase 1 {ECO:0000255|HAMAP-Rule:MF_03156} approved DB01035 Procainamide small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB01035 Procainamide small molecule P26358 DNA (cytosine-5)-methyltransferase 1 approved DB01035 Procainamide small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB01036 Tolterodine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB01036 Tolterodine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB01036 Tolterodine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB01036 Tolterodine small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational|vet_approved DB01037 Selegiline small molecule P27338 Amine oxidase [flavin-containing] B approved|investigational|vet_approved DB01037 Selegiline small molecule P21397 Amine oxidase [flavin-containing] A approved DB01039 Fenofibrate small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved DB01039 Fenofibrate small molecule P37231 Peroxisome proliferator-activated receptor gamma approved DB01039 Fenofibrate small molecule Q03181 Peroxisome proliferator-activated receptor delta approved DB01039 Fenofibrate small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational|withdrawn DB01041 Thalidomide small molecule Q96SW2 Protein cereblon approved|investigational|withdrawn DB01041 Thalidomide small molecule P01375 Tumor necrosis factor approved|investigational|withdrawn DB01041 Thalidomide small molecule P19838 Nuclear factor NF-kappa-B p105 subunit approved|investigational|withdrawn DB01041 Thalidomide small molecule P21802 Fibroblast growth factor receptor 2 approved|investigational|withdrawn DB01041 Thalidomide small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational|withdrawn DB01041 Thalidomide small molecule P02763 Alpha-1-acid glycoprotein 1 approved|investigational DB01043 Memantine small molecule Q12879 Glutamate receptor ionotropic, NMDA 2A approved|investigational DB01043 Memantine small molecule Q13224 Glutamate receptor ionotropic, NMDA 2B approved|investigational DB01043 Memantine small molecule P14416 D(2) dopamine receptor approved|investigational DB01043 Memantine small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved DB01045 Rifampicin small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB01045 Rifampicin small molecule Q9Y6L6 Solute carrier organic anion transporter family member 1B1 approved DB01045 Rifampicin small molecule P46721 Solute carrier organic anion transporter family member 1A2 approved DB01045 Rifampicin small molecule Q16850 Lanosterol 14-alpha demethylase approved DB01045 Rifampicin small molecule P02768 Serum albumin approved DB01045 Rifampicin small molecule O94956 Solute carrier organic anion transporter family member 2B1 approved|investigational DB01046 Lubiprostone small molecule P51788 Chloride channel protein 2 approved|investigational DB01047 Fluocinonide small molecule P04150 Glucocorticoid receptor approved|investigational DB01047 Fluocinonide small molecule Q99835 Smoothened homolog approved|investigational DB01048 Abacavir small molecule P18465 HLA class I histocompatibility antigen, B-57 alpha chain approved DB01050 Ibuprofen small molecule P35354 Prostaglandin G/H synthase 2 approved DB01050 Ibuprofen small molecule P23219 Prostaglandin G/H synthase 1 approved DB01050 Ibuprofen small molecule P10415 Apoptosis regulator Bcl-2 approved DB01050 Ibuprofen small molecule P07204 Thrombomodulin approved DB01050 Ibuprofen small molecule P00750 Tissue-type plasminogen activator approved DB01050 Ibuprofen small molecule P12104 Fatty acid-binding protein, intestinal approved DB01050 Ibuprofen small molecule P37231 Peroxisome proliferator-activated receptor gamma approved DB01050 Ibuprofen small molecule P13569 Cystic fibrosis transmembrane conductance regulator approved DB01050 Ibuprofen small molecule P46059 Solute carrier family 15 member 1 approved DB01050 Ibuprofen small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved|vet_approved DB01053 Benzylpenicillin small molecule Q8TCC7 Solute carrier family 22 member 8 approved|vet_approved DB01053 Benzylpenicillin small molecule P46059 Solute carrier family 15 member 1 approved|investigational DB01054 Nitrendipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB01054 Nitrendipine small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved|investigational DB01054 Nitrendipine small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved|investigational DB01054 Nitrendipine small molecule Q06432 Voltage-dependent calcium channel gamma-1 subunit approved|investigational DB01054 Nitrendipine small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved|investigational DB01054 Nitrendipine small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved|investigational DB01054 Nitrendipine small molecule Q9NY47 Voltage-dependent calcium channel subunit alpha-2/delta-2 approved|investigational DB01054 Nitrendipine small molecule O95180 Voltage-dependent T-type calcium channel subunit alpha-1H approved DB01056 Tocainide small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB01057 Echothiophate small molecule P06276 Cholinesterase approved DB01059 Norfloxacin small molecule P11388 DNA topoisomerase 2-alpha approved|investigational DB01062 Oxybutynin small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB01062 Oxybutynin small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB01062 Oxybutynin small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB01063 Acetophenazine small molecule P14416 D(2) dopamine receptor approved DB01063 Acetophenazine small molecule P10275 Androgen receptor approved|investigational DB01064 Isoprenaline small molecule P13945 Beta-3 adrenergic receptor approved|investigational DB01064 Isoprenaline small molecule P28482 Mitogen-activated protein kinase 1 approved|investigational DB01064 Isoprenaline small molecule P27986 Phosphatidylinositol 3-kinase regulatory subunit alpha approved|investigational DB01064 Isoprenaline small molecule O00459 Phosphatidylinositol 3-kinase regulatory subunit beta approved|investigational DB01064 Isoprenaline small molecule Q92569 Phosphatidylinositol 3-kinase regulatory subunit gamma approved|investigational DB01064 Isoprenaline small molecule P00441 Superoxide dismutase [Cu-Zn] approved|nutraceutical|vet_approved DB01065 Melatonin small molecule P03372 Estrogen receptor approved|nutraceutical|vet_approved DB01065 Melatonin small molecule Q92753 Nuclear receptor ROR-beta approved|nutraceutical|vet_approved DB01065 Melatonin small molecule P05164 Myeloperoxidase approved|nutraceutical|vet_approved DB01065 Melatonin small molecule P27797 Calreticulin approved|nutraceutical|vet_approved DB01065 Melatonin small molecule P16083 Ribosyldihydronicotinamide dehydrogenase [quinone] approved|investigational DB01067 Glipizide small molecule Q09428 ATP-binding cassette sub-family C member 8 approved|investigational DB01067 Glipizide small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|illicit DB01068 Clonazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01068 Clonazepam small molecule P30536 Translocator protein approved|illicit DB01068 Clonazepam small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB01069 Promethazine small molecule P35367 Histamine H1 receptor approved|investigational DB01069 Promethazine small molecule P14416 D(2) dopamine receptor approved|investigational DB01069 Promethazine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB01069 Promethazine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB01069 Promethazine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB01069 Promethazine small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB01069 Promethazine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB01069 Promethazine small molecule P25021 Histamine H2 receptor approved DB01070 Dihydrotachysterol small molecule P11473 Vitamin D3 receptor approved DB01071 Mequitazine small molecule P35367 Histamine H1 receptor approved DB01073 Fludarabine small molecule P23921 Ribonucleoside-diphosphate reductase large subunit approved DB01073 Fludarabine small molecule P09884 DNA polymerase alpha catalytic subunit approved DB01073 Fludarabine small molecule P27707 Deoxycytidine kinase approved|investigational DB01074 Perhexiline small molecule P50416 Carnitine O-palmitoyltransferase 1, liver isoform approved|investigational DB01074 Perhexiline small molecule P23786 Carnitine O-palmitoyltransferase 2, mitochondrial approved|investigational DB01074 Perhexiline small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB01075 Diphenhydramine small molecule P35367 Histamine H1 receptor approved|investigational DB01075 Diphenhydramine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB01076 Atorvastatin small molecule P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase approved DB01076 Atorvastatin small molecule P27487 Dipeptidyl peptidase 4 approved DB01076 Atorvastatin small molecule P35869 Aryl hydrocarbon receptor approved DB01077 Etidronic acid small molecule Q13332 Receptor-type tyrosine-protein phosphatase S approved DB01077 Etidronic acid small molecule P38606 V-type proton ATPase catalytic subunit A approved DB01078 Deslanoside small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved|investigational|withdrawn DB01079 Tegaserod small molecule Q13639 5-hydroxytryptamine receptor 4 approved|investigational|withdrawn DB01079 Tegaserod small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational|withdrawn DB01079 Tegaserod small molecule P28223 5-hydroxytryptamine receptor 2A approved DB01080 Vigabatrin small molecule Q9UBS5 Gamma-aminobutyric acid type B receptor subunit 1 approved DB01080 Vigabatrin small molecule P80404 4-aminobutyrate aminotransferase, mitochondrial approved|illicit DB01081 Diphenoxylate small molecule P35372 Mu-type opioid receptor approved|illicit DB01081 Diphenoxylate small molecule P41143 Delta-type opioid receptor approved|vet_approved DB01082 Streptomycin small molecule Q9UM07 Protein-arginine deiminase type-4 approved|investigational DB01083 Orlistat small molecule P16233 Pancreatic triacylglycerol lipase approved|investigational DB01083 Orlistat small molecule P07098 Gastric triacylglycerol lipase approved|investigational DB01083 Orlistat small molecule P49327 Fatty acid synthase approved DB01084 Emedastine small molecule P35367 Histamine H1 receptor approved|investigational DB01085 Pilocarpine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB01085 Pilocarpine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB01085 Pilocarpine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB01085 Pilocarpine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB01087 Primaquine small molecule P08729 Keratin, type II cytoskeletal 7 approved DB01087 Primaquine small molecule P16083 Ribosyldihydronicotinamide dehydrogenase [quinone] approved|investigational DB01088 Iloprost small molecule P34995 Prostaglandin E2 receptor EP1 subtype approved|investigational DB01088 Iloprost small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved|investigational DB01088 Iloprost small molecule Q07343 cAMP-specific 3',5'-cyclic phosphodiesterase 4B approved|investigational DB01088 Iloprost small molecule Q08493 cAMP-specific 3',5'-cyclic phosphodiesterase 4C approved|investigational DB01088 Iloprost small molecule Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D approved|investigational DB01088 Iloprost small molecule P00750 Tissue-type plasminogen activator approved DB01089 Deserpidine small molecule Q05940 Synaptic vesicular amine transporter approved DB01091 Butenafine small molecule Q14534 Squalene monooxygenase approved DB01092 Ouabain small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved DB01092 Ouabain small molecule P50993 Sodium/potassium-transporting ATPase subunit alpha-2 approved DB01092 Ouabain small molecule P13637 Sodium/potassium-transporting ATPase subunit alpha-3 approved DB01095 Fluvastatin small molecule P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase approved|investigational DB01097 Leflunomide small molecule Q02127 Dihydroorotate dehydrogenase (quinone), mitochondrial approved|investigational DB01097 Leflunomide small molecule P35869 Aryl hydrocarbon receptor approved|investigational DB01097 Leflunomide small molecule Q14289 Protein-tyrosine kinase 2-beta approved DB01098 Rosuvastatin small molecule P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase approved|investigational DB01099 Flucytosine small molecule P26358 DNA (cytosine-5)-methyltransferase 1 approved DB01100 Pimozide small molecule P14416 D(2) dopamine receptor approved DB01100 Pimozide small molecule P35462 D(3) dopamine receptor approved DB01100 Pimozide small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB01101 Capecitabine small molecule P04818 Thymidylate synthase approved DB01102 Arbutamine small molecule P13945 Beta-3 adrenergic receptor approved|investigational DB01103 Quinacrine small molecule O60733 85/88 kDa calcium-independent phospholipase A2 approved|investigational DB01103 Quinacrine small molecule Q15111 Inactive phospholipase C-like protein 1 approved DB01104 Sertraline small molecule P31645 Sodium-dependent serotonin transporter approved DB01104 Sertraline small molecule O00264 Membrane-associated progesterone receptor component 1 approved|illicit|investigational|withdrawn DB01105 Sibutramine small molecule P23975 Sodium-dependent noradrenaline transporter approved|illicit|investigational|withdrawn DB01105 Sibutramine small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB01106 Levocabastine small molecule P35367 Histamine H1 receptor approved|investigational DB01106 Levocabastine small molecule O95665 Neurotensin receptor type 2 approved|illicit|withdrawn DB01107 Methyprylon small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit|withdrawn DB01107 Methyprylon small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational|vet_approved|withdrawn DB01108 Trilostane small molecule P14060 3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1 approved|investigational|vet_approved|withdrawn DB01108 Trilostane small molecule P26439 3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2 approved|investigational|vet_approved|withdrawn DB01108 Trilostane small molecule P03372 Estrogen receptor approved|investigational|vet_approved|withdrawn DB01108 Trilostane small molecule Q92731 Estrogen receptor beta approved|investigational DB01109 Heparin small molecule P01008 Antithrombin-III approved|investigational DB01109 Heparin small molecule P00742 Coagulation factor X approved|investigational DB01109 Heparin small molecule P16109 P-selectin approved|investigational DB01109 Heparin small molecule P22455 Fibroblast growth factor receptor 4 approved|investigational DB01109 Heparin small molecule P08620 Fibroblast growth factor 4 approved|investigational DB01109 Heparin small molecule O95750 Fibroblast growth factor 19 approved|investigational DB01109 Heparin small molecule P11362 Fibroblast growth factor receptor 1 approved|investigational DB01109 Heparin small molecule P05230 Fibroblast growth factor 1 approved|investigational DB01109 Heparin small molecule P21802 Fibroblast growth factor receptor 2 approved|investigational DB01109 Heparin small molecule P09038 Fibroblast growth factor 2 approved|investigational DB01109 Heparin small molecule P14210 Hepatocyte growth factor approved|investigational|vet_approved DB01110 Miconazole small molecule P29474 Nitric oxide synthase, endothelial approved|investigational|vet_approved DB01110 Miconazole small molecule P35228 Nitric oxide synthase, inducible approved|investigational|vet_approved DB01110 Miconazole small molecule Q12791 Calcium-activated potassium channel subunit alpha-1 approved|investigational|vet_approved DB01110 Miconazole small molecule Q16558 Calcium-activated potassium channel subunit beta-1 approved|investigational|vet_approved DB01110 Miconazole small molecule Q9Y691 Calcium-activated potassium channel subunit beta-2 approved|investigational|vet_approved DB01110 Miconazole small molecule Q9NPA1 Calcium-activated potassium channel subunit beta-3 approved|investigational|vet_approved DB01110 Miconazole small molecule Q86W47 Calcium-activated potassium channel subunit beta-4 approved|investigational|vet_approved DB01110 Miconazole small molecule O15554 Intermediate conductance calcium-activated potassium channel protein 4 approved|investigational|vet_approved DB01110 Miconazole small molecule Q92952 Small conductance calcium-activated potassium channel protein 1 approved|investigational|vet_approved DB01110 Miconazole small molecule Q9H2S1 Small conductance calcium-activated potassium channel protein 2 approved|investigational|vet_approved DB01110 Miconazole small molecule Q9UGI6 Small conductance calcium-activated potassium channel protein 3 approved|investigational|vet_approved DB01110 Miconazole small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational|vet_approved DB01110 Miconazole small molecule Q9NS40 Potassium voltage-gated channel subfamily H member 7 approved|investigational|vet_approved DB01110 Miconazole small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB01113 Papaverine small molecule Q07343 cAMP-specific 3',5'-cyclic phosphodiesterase 4B approved|investigational DB01113 Papaverine small molecule Q9Y233 cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A approved DB01114 Chlorphenamine small molecule P35367 Histamine H1 receptor approved DB01114 Chlorphenamine small molecule P31645 Sodium-dependent serotonin transporter approved DB01114 Chlorphenamine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB01115 Nifedipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved DB01115 Nifedipine small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved DB01115 Nifedipine small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved DB01115 Nifedipine small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved DB01115 Nifedipine small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved DB01115 Nifedipine small molecule Q09470 Potassium voltage-gated channel subfamily A member 1 approved DB01115 Nifedipine small molecule O95180 Voltage-dependent T-type calcium channel subunit alpha-1H approved DB01115 Nifedipine small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB01117 Atovaquone small molecule Q02127 Dihydroorotate dehydrogenase (quinone), mitochondrial approved|investigational DB01118 Amiodarone small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB01118 Amiodarone small molecule O95180 Voltage-dependent T-type calcium channel subunit alpha-1H approved|investigational DB01118 Amiodarone small molecule Q9NY47 Voltage-dependent calcium channel subunit alpha-2/delta-2 approved|investigational DB01118 Amiodarone small molecule P10827 Thyroid hormone receptor alpha approved|investigational DB01118 Amiodarone small molecule P10828 Thyroid hormone receptor beta approved|investigational DB01118 Amiodarone small molecule P37231 Peroxisome proliferator-activated receptor gamma approved DB01119 Diazoxide small molecule P00915 Carbonic anhydrase 1 approved DB01119 Diazoxide small molecule P00918 Carbonic anhydrase 2 approved DB01119 Diazoxide small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved DB01119 Diazoxide small molecule Q12791 Calcium-activated potassium channel subunit alpha-1 approved DB01119 Diazoxide small molecule P55017 Solute carrier family 12 member 3 approved DB01120 Gliclazide small molecule Q09428 ATP-binding cassette sub-family C member 8 approved DB01120 Gliclazide small molecule P15692 Vascular endothelial growth factor A approved DB01122 Ambenonium small molecule P22303 Acetylcholinesterase approved|investigational DB01124 Tolbutamide small molecule Q09428 ATP-binding cassette sub-family C member 8 approved|investigational DB01126 Dutasteride small molecule P18405 3-oxo-5-alpha-steroid 4-dehydrogenase 1 approved DB01127 Econazole small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB01128 Bicalutamide small molecule P10275 Androgen receptor approved|investigational DB01129 Rabeprazole small molecule P20648 Potassium-transporting ATPase alpha chain 1 approved|investigational DB01130 Prednicarbate small molecule P04150 Glucocorticoid receptor approved DB01131 Proguanil small molecule P00374 Dihydrofolate reductase approved|investigational DB01132 Pioglitazone small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|investigational DB01132 Pioglitazone small molecule Q03181 Peroxisome proliferator-activated receptor delta approved|investigational DB01132 Pioglitazone small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved|investigational DB01132 Pioglitazone small molecule P27338 Amine oxidase [flavin-containing] B approved|investigational|vet_approved DB01133 Tiludronic acid small molecule P38606 V-type proton ATPase catalytic subunit A approved|investigational|vet_approved DB01133 Tiludronic acid small molecule P18031 Tyrosine-protein phosphatase non-receptor type 1 approved DB01135 Doxacurium chloride small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB01135 Doxacurium chloride small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB01136 Carvedilol small molecule O95298 NADH dehydrogenase [ubiquinone] 1 subunit C2 approved|investigational DB01136 Carvedilol small molecule P15692 Vascular endothelial growth factor A approved|investigational DB01136 Carvedilol small molecule P17302 Gap junction alpha-1 protein approved|investigational DB01136 Carvedilol small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB01136 Carvedilol small molecule P19320 Vascular cell adhesion protein 1 approved|investigational DB01136 Carvedilol small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB01136 Carvedilol small molecule P16581 E-selectin approved|investigational DB01136 Carvedilol small molecule Q16665 Hypoxia-inducible factor 1-alpha {ECO:0000303|PubMed:7539918} approved|investigational DB01136 Carvedilol small molecule P48050 Inward rectifier potassium channel 4 approved|investigational DB01137 Levofloxacin small molecule P11388 DNA topoisomerase 2-alpha approved DB01138 Sulfinpyrazone small molecule Q92887 Canalicular multispecific organic anion transporter 1 approved DB01138 Sulfinpyrazone small molecule P33527 Multidrug resistance-associated protein 1 approved DB01138 Sulfinpyrazone small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB01142 Doxepin small molecule P35367 Histamine H1 receptor approved|investigational DB01142 Doxepin small molecule P25021 Histamine H2 receptor approved|investigational DB01142 Doxepin small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB01142 Doxepin small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB01142 Doxepin small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB01142 Doxepin small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB01142 Doxepin small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB01142 Doxepin small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB01142 Doxepin small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB01142 Doxepin small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB01142 Doxepin small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB01142 Doxepin small molecule P14416 D(2) dopamine receptor approved|investigational DB01142 Doxepin small molecule Q9H3N8 Histamine H4 receptor approved|investigational DB01142 Doxepin small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB01143 Amifostine small molecule P22413 Ectonucleotide pyrophosphatase/phosphodiesterase family member 1 approved|investigational DB01144 Diclofenamide small molecule P00915 Carbonic anhydrase 1 approved|investigational DB01144 Diclofenamide small molecule P00918 Carbonic anhydrase 2 approved|investigational DB01144 Diclofenamide small molecule P22748 Carbonic anhydrase 4 approved|investigational DB01144 Diclofenamide small molecule P43166 Carbonic anhydrase 7 approved|investigational DB01144 Diclofenamide small molecule P07451 Carbonic anhydrase 3 approved|investigational DB01146 Diphenylpyraline small molecule P35367 Histamine H1 receptor approved DB01148 Flavoxate small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB01148 Flavoxate small molecule P11229 Muscarinic acetylcholine receptor M1 approved|withdrawn DB01149 Nefazodone small molecule P28223 5-hydroxytryptamine receptor 2A approved|withdrawn DB01149 Nefazodone small molecule P28335 5-hydroxytryptamine receptor 2C approved|withdrawn DB01149 Nefazodone small molecule P31645 Sodium-dependent serotonin transporter approved|withdrawn DB01149 Nefazodone small molecule P23975 Sodium-dependent noradrenaline transporter approved|withdrawn DB01149 Nefazodone small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB01151 Desipramine small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB01151 Desipramine small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB01151 Desipramine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB01151 Desipramine small molecule P17405 Sphingomyelin phosphodiesterase approved|investigational DB01151 Desipramine small molecule P35367 Histamine H1 receptor approved|investigational DB01151 Desipramine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB01151 Desipramine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB01151 Desipramine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB01151 Desipramine small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB01151 Desipramine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB01151 Desipramine small molecule P14416 D(2) dopamine receptor approved|vet_approved DB01154 Thiamylal small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01156 Bupropion small molecule P23975 Sodium-dependent noradrenaline transporter approved DB01156 Bupropion small molecule P32297 Neuronal acetylcholine receptor subunit alpha-3 approved|investigational DB01157 Trimetrexate small molecule P00374 Dihydrofolate reductase approved|vet_approved DB01159 Halothane small molecule O14649 Potassium channel subfamily K member 3 approved|vet_approved DB01159 Halothane small molecule Q9NPC2 Potassium channel subfamily K member 9 approved|vet_approved DB01159 Halothane small molecule Q12791 Calcium-activated potassium channel subunit alpha-1 approved|vet_approved DB01159 Halothane small molecule O60391 Glutamate receptor ionotropic, NMDA 3B approved|vet_approved DB01159 Halothane small molecule Q12879 Glutamate receptor ionotropic, NMDA 2A approved|vet_approved DB01159 Halothane small molecule P23415 Glycine receptor subunit alpha-1 approved|vet_approved DB01159 Halothane small molecule P08100 Rhodopsin approved|vet_approved DB01159 Halothane small molecule P48051 G protein-activated inward rectifier potassium channel 2 approved|vet_approved DB01159 Halothane small molecule P48549 G protein-activated inward rectifier potassium channel 1 approved|vet_approved DB01159 Halothane small molecule O15554 Intermediate conductance calcium-activated potassium channel protein 4 approved|vet_approved DB01159 Halothane small molecule P30049 ATP synthase subunit delta, mitochondrial {ECO:0000305} approved|vet_approved DB01159 Halothane small molecule P98194 Calcium-transporting ATPase type 2C member 1 approved|vet_approved DB01159 Halothane small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|vet_approved DB01159 Halothane small molecule P59768 Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2 approved|vet_approved DB01159 Halothane small molecule Q6W5P4 Neuropeptide S receptor approved|vet_approved DB01159 Halothane small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01162 Terazosin small molecule P25100 Alpha-1D adrenergic receptor approved DB01162 Terazosin small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB01162 Terazosin small molecule Q9NS40 Potassium voltage-gated channel subfamily H member 7 approved DB01164 Calcium Chloride small molecule Q99584 Protein S100-A13 approved DB01165 Ofloxacin small molecule P11388 DNA topoisomerase 2-alpha approved|investigational DB01166 Cilostazol small molecule Q14432 cGMP-inhibited 3',5'-cyclic phosphodiesterase A approved|investigational DB01167 Itraconazole small molecule Q16850 Lanosterol 14-alpha demethylase approved|investigational DB01168 Procarbazine small molecule P21397 Amine oxidase [flavin-containing] A approved|investigational DB01169 Arsenic trioxide small molecule O14920 Inhibitor of nuclear factor kappa-B kinase subunit beta approved|investigational DB01169 Arsenic trioxide small molecule Q16881 Thioredoxin reductase 1, cytoplasmic approved|investigational DB01169 Arsenic trioxide small molecule P05412 Transcription factor AP-1 approved|investigational DB01169 Arsenic trioxide small molecule P24385 G1/S-specific cyclin-D1 approved|investigational DB01169 Arsenic trioxide small molecule P27361 Mitogen-activated protein kinase 3 approved|investigational DB01169 Arsenic trioxide small molecule P28482 Mitogen-activated protein kinase 1 approved|investigational DB01169 Arsenic trioxide small molecule P31749 RAC-alpha serine/threonine-protein kinase approved|investigational DB01169 Arsenic trioxide small molecule P38936 Cyclin-dependent kinase inhibitor 1 approved|investigational DB01169 Arsenic trioxide small molecule Q13547 Histone deacetylase 1 approved|investigational DB01169 Arsenic trioxide small molecule P29590 Protein PML approved DB01170 Guanethidine small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB01171 Moclobemide small molecule P21397 Amine oxidase [flavin-containing] A approved|investigational DB01171 Moclobemide small molecule P21397 Amine oxidase [flavin-containing] A approved|investigational DB01171 Moclobemide small molecule P27338 Amine oxidase [flavin-containing] B approved DB01173 Orphenadrine small molecule O15399 Glutamate receptor ionotropic, NMDA 2D approved DB01173 Orphenadrine small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved DB01173 Orphenadrine small molecule O60391 Glutamate receptor ionotropic, NMDA 3B approved DB01173 Orphenadrine small molecule P35367 Histamine H1 receptor approved DB01173 Orphenadrine small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB01174 Phenobarbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB01174 Phenobarbital small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|investigational DB01174 Phenobarbital small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|investigational DB01174 Phenobarbital small molecule P42262 Glutamate receptor 2 approved|investigational DB01174 Phenobarbital small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved|investigational DB01174 Phenobarbital small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved|investigational DB01174 Phenobarbital small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB01175 Escitalopram small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB01175 Escitalopram small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB01175 Escitalopram small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB01175 Escitalopram small molecule P35367 Histamine H1 receptor approved DB01176 Cyclizine small molecule P35367 Histamine H1 receptor approved DB01176 Cyclizine small molecule P49888 Estrogen sulfotransferase approved DB01177 Idarubicin small molecule P11388 DNA topoisomerase 2-alpha approved|investigational|withdrawn DB01178 Chlormezanone small molecule P30536 Translocator protein approved DB01179 Podofilox small molecule P11388 DNA topoisomerase 2-alpha approved DB01179 Podofilox small molecule P68366 Tubulin alpha-4A chain approved DB01179 Podofilox small molecule P07437 Tubulin beta chain approved DB01180 Rescinnamine small molecule P12821 Angiotensin-converting enzyme approved DB01181 Ifosfamide small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB01182 Propafenone small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB01182 Propafenone small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|vet_approved DB01183 Naloxone small molecule P35372 Mu-type opioid receptor approved|vet_approved DB01183 Naloxone small molecule P41143 Delta-type opioid receptor approved|vet_approved DB01183 Naloxone small molecule P16220 Cyclic AMP-responsive element-binding protein 1 approved|vet_approved DB01183 Naloxone small molecule P03372 Estrogen receptor approved|vet_approved DB01183 Naloxone small molecule O00206 Toll-like receptor 4 approved|vet_approved DB01183 Naloxone small molecule P23141 Liver carboxylesterase 1 approved|investigational|vet_approved DB01184 Domperidone small molecule P14416 D(2) dopamine receptor approved|investigational|vet_approved DB01184 Domperidone small molecule P35462 D(3) dopamine receptor approved|illicit DB01185 Fluoxymesterone small molecule P10275 Androgen receptor approved|illicit DB01185 Fluoxymesterone small molecule P03372 Estrogen receptor approved|illicit DB01185 Fluoxymesterone small molecule P16471 Prolactin receptor approved|illicit DB01185 Fluoxymesterone small molecule P04150 Glucocorticoid receptor approved|illicit DB01185 Fluoxymesterone small molecule P80365 Corticosteroid 11-beta-dehydrogenase isozyme 2 approved|investigational|vet_approved|withdrawn DB01186 Pergolide small molecule P14416 D(2) dopamine receptor approved|investigational|vet_approved|withdrawn DB01186 Pergolide small molecule P35462 D(3) dopamine receptor approved|investigational|vet_approved|withdrawn DB01186 Pergolide small molecule P21917 D(4) dopamine receptor approved|investigational|vet_approved|withdrawn DB01186 Pergolide small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational|vet_approved|withdrawn DB01186 Pergolide small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational|vet_approved|withdrawn DB01186 Pergolide small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB01188 Ciclopirox small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved DB01189 Desflurane small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01189 Desflurane small molecule P23415 Glycine receptor subunit alpha-1 approved DB01189 Desflurane small molecule P42261 Glutamate receptor 1 approved DB01189 Desflurane small molecule Q09470 Potassium voltage-gated channel subfamily A member 1 approved DB01189 Desflurane small molecule P98194 Calcium-transporting ATPase type 2C member 1 approved DB01189 Desflurane small molecule P30049 ATP synthase subunit delta, mitochondrial {ECO:0000305} approved|illicit|investigational|withdrawn DB01191 Dexfenfluramine small molecule P31645 Sodium-dependent serotonin transporter approved|illicit|investigational|withdrawn DB01191 Dexfenfluramine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB01194 Brinzolamide small molecule P00918 Carbonic anhydrase 2 approved DB01194 Brinzolamide small molecule P00915 Carbonic anhydrase 1 approved DB01194 Brinzolamide small molecule P22748 Carbonic anhydrase 4 approved DB01194 Brinzolamide small molecule P35218 Carbonic anhydrase 5A, mitochondrial approved DB01194 Brinzolamide small molecule P07451 Carbonic anhydrase 3 approved|withdrawn DB01195 Flecainide small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|withdrawn DB01195 Flecainide small molecule P35499 Sodium channel protein type 4 subunit alpha approved|withdrawn DB01195 Flecainide small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB01196 Estramustine small molecule P11137 Microtubule-associated protein 2 approved|investigational DB01196 Estramustine small molecule P78559 Microtubule-associated protein 1A approved|investigational DB01196 Estramustine small molecule P03372 Estrogen receptor approved|investigational DB01196 Estramustine small molecule Q92731 Estrogen receptor beta approved DB01197 Captopril small molecule P12821 Angiotensin-converting enzyme approved DB01197 Captopril small molecule P08253 72 kDa type IV collagenase approved DB01197 Captopril small molecule P14780 Matrix metalloproteinase-9 approved DB01197 Captopril small molecule P09960 Leukotriene A-4 hydrolase approved DB01198 Zopiclone small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01198 Zopiclone small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB01198 Zopiclone small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB01198 Zopiclone small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved DB01198 Zopiclone small molecule P30536 Translocator protein approved DB01199 Tubocurarine small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB01199 Tubocurarine small molecule P22303 Acetylcholinesterase approved DB01199 Tubocurarine small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|investigational DB01200 Bromocriptine small molecule P14416 D(2) dopamine receptor approved|investigational DB01200 Bromocriptine small molecule P35462 D(3) dopamine receptor approved|investigational DB01200 Bromocriptine small molecule P21917 D(4) dopamine receptor approved|investigational DB01200 Bromocriptine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB01200 Bromocriptine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB01200 Bromocriptine small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB01200 Bromocriptine small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational DB01202 Levetiracetam small molecule Q7L0J3 Synaptic vesicle glycoprotein 2A approved|investigational DB01202 Levetiracetam small molecule Q00975 Voltage-dependent N-type calcium channel subunit alpha-1B approved|investigational DB01204 Mitoxantrone small molecule P11388 DNA topoisomerase 2-alpha approved DB01205 Flumazenil small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01205 Flumazenil small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved DB01205 Flumazenil small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved DB01205 Flumazenil small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB01208 Sparfloxacin small molecule P11388 DNA topoisomerase 2-alpha approved|investigational DB01209 Dezocine small molecule P35372 Mu-type opioid receptor approved DB01211 Clarithromycin small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB01211 Clarithromycin small molecule Q9Y6L6 Solute carrier organic anion transporter family member 1B1 approved DB01212 Ceftriaxone small molecule Q9NSA0 Solute carrier family 22 member 11 approved DB01212 Ceftriaxone small molecule Q4U2R8 Solute carrier family 22 member 6 approved DB01212 Ceftriaxone small molecule Q8TCC7 Solute carrier family 22 member 8 approved DB01212 Ceftriaxone small molecule P46059 Solute carrier family 15 member 1 approved|vet_approved DB01213 Fomepizole small molecule P00325 Alcohol dehydrogenase 1B approved|vet_approved DB01213 Fomepizole small molecule P04040 Catalase approved|illicit DB01215 Estazolam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01215 Estazolam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB01215 Estazolam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB01215 Estazolam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB01215 Estazolam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|illicit DB01215 Estazolam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|illicit DB01215 Estazolam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|illicit DB01215 Estazolam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|illicit DB01215 Estazolam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|illicit DB01215 Estazolam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|illicit DB01215 Estazolam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|illicit DB01215 Estazolam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|illicit DB01215 Estazolam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|illicit DB01215 Estazolam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|illicit DB01215 Estazolam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01216 Finasteride small molecule P18405 3-oxo-5-alpha-steroid 4-dehydrogenase 1 approved DB01216 Finasteride small molecule P51857 3-oxo-5-beta-steroid 4-dehydrogenase approved|investigational DB01217 Anastrozole small molecule P11511 Aromatase approved DB01218 Halofantrine small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB01219 Dantrolene small molecule P21817 Ryanodine receptor 1 approved|investigational DB01220 Rifaximin small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|vet_approved DB01221 Ketamine small molecule P25103 Substance-P receptor approved|vet_approved DB01221 Ketamine small molecule P14416 D(2) dopamine receptor approved|vet_approved DB01221 Ketamine small molecule P41143 Delta-type opioid receptor approved|vet_approved DB01221 Ketamine small molecule P23975 Sodium-dependent noradrenaline transporter approved|vet_approved DB01221 Ketamine small molecule P35372 Mu-type opioid receptor approved|vet_approved DB01221 Ketamine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|vet_approved DB01221 Ketamine small molecule P28223 5-hydroxytryptamine receptor 2A approved|vet_approved DB01221 Ketamine small molecule P06276 Cholinesterase approved|vet_approved DB01221 Ketamine small molecule P29475 Nitric oxide synthase, brain approved DB01222 Budesonide small molecule P04150 Glucocorticoid receptor approved DB01223 Aminophylline small molecule Q14432 cGMP-inhibited 3',5'-cyclic phosphodiesterase A approved DB01223 Aminophylline small molecule P30542 Adenosine receptor A1 approved DB01223 Aminophylline small molecule Q92769 Histone deacetylase 2 approved DB01224 Quetiapine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB01224 Quetiapine small molecule P14416 D(2) dopamine receptor approved DB01224 Quetiapine small molecule P28566 5-hydroxytryptamine receptor 1E approved DB01224 Quetiapine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB01224 Quetiapine small molecule P34969 5-hydroxytryptamine receptor 7 approved DB01224 Quetiapine small molecule P35462 D(3) dopamine receptor approved DB01224 Quetiapine small molecule P21917 D(4) dopamine receptor approved DB01224 Quetiapine small molecule P35367 Histamine H1 receptor approved DB01224 Quetiapine small molecule P25100 Alpha-1D adrenergic receptor approved DB01224 Quetiapine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB01224 Quetiapine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB01224 Quetiapine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB01224 Quetiapine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB01225 Enoxaparin small molecule P01008 Antithrombin-III approved DB01225 Enoxaparin small molecule P00742 Coagulation factor X approved DB01226 Mivacurium small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB01226 Mivacurium small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB01226 Mivacurium small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB01226 Mivacurium small molecule P06276 Cholinesterase approved|investigational DB01227 Levomethadyl Acetate small molecule P35372 Mu-type opioid receptor approved|investigational DB01227 Levomethadyl Acetate small molecule P30926 Neuronal acetylcholine receptor subunit beta-4 approved|investigational DB01227 Levomethadyl Acetate small molecule P32297 Neuronal acetylcholine receptor subunit alpha-3 approved|investigational|withdrawn DB01228 Encainide small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|vet_approved DB01229 Paclitaxel small molecule P10415 Apoptosis regulator Bcl-2 approved|vet_approved DB01229 Paclitaxel small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|vet_approved DB01229 Paclitaxel small molecule P27816 Microtubule-associated protein 4 approved|vet_approved DB01229 Paclitaxel small molecule P11137 Microtubule-associated protein 2 approved|vet_approved DB01229 Paclitaxel small molecule P10636 Microtubule-associated protein tau approved|investigational DB01233 Metoclopramide small molecule P14416 D(2) dopamine receptor approved|investigational DB01233 Metoclopramide small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB01233 Metoclopramide small molecule Q13639 5-hydroxytryptamine receptor 4 approved|investigational DB01233 Metoclopramide small molecule P22303 Acetylcholinesterase approved|investigational|vet_approved DB01234 Dexamethasone small molecule P04150 Glucocorticoid receptor approved|investigational|vet_approved DB01234 Dexamethasone small molecule P51843 Nuclear receptor subfamily 0 group B member 1 approved|investigational|vet_approved DB01234 Dexamethasone small molecule P04083 Annexin A1 approved|investigational|vet_approved DB01234 Dexamethasone small molecule P35228 Nitric oxide synthase, inducible approved|investigational|vet_approved DB01234 Dexamethasone small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB01235 Levodopa small molecule P14416 D(2) dopamine receptor approved DB01235 Levodopa small molecule P35462 D(3) dopamine receptor approved DB01235 Levodopa small molecule P21917 D(4) dopamine receptor approved|vet_approved DB01236 Sevoflurane small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|vet_approved DB01236 Sevoflurane small molecule P23415 Glycine receptor subunit alpha-1 approved|vet_approved DB01236 Sevoflurane small molecule P42261 Glutamate receptor 1 approved|vet_approved DB01236 Sevoflurane small molecule Q09470 Potassium voltage-gated channel subfamily A member 1 approved|vet_approved DB01236 Sevoflurane small molecule P98194 Calcium-transporting ATPase type 2C member 1 approved|vet_approved DB01236 Sevoflurane small molecule P30049 ATP synthase subunit delta, mitochondrial {ECO:0000305} approved|vet_approved DB01236 Sevoflurane small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01237 Bromodiphenhydramine small molecule P35367 Histamine H1 receptor approved|investigational DB01238 Aripiprazole small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB01238 Aripiprazole small molecule P14416 D(2) dopamine receptor approved|investigational DB01238 Aripiprazole small molecule P28566 5-hydroxytryptamine receptor 1E approved|investigational DB01238 Aripiprazole small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB01238 Aripiprazole small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational DB01238 Aripiprazole small molecule P35462 D(3) dopamine receptor approved|investigational DB01238 Aripiprazole small molecule P21917 D(4) dopamine receptor approved|investigational DB01238 Aripiprazole small molecule P35367 Histamine H1 receptor approved|investigational DB01238 Aripiprazole small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB01238 Aripiprazole small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB01238 Aripiprazole small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB01238 Aripiprazole small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational|withdrawn DB01239 Chlorprothixene small molecule P14416 D(2) dopamine receptor approved|investigational|withdrawn DB01239 Chlorprothixene small molecule P35462 D(3) dopamine receptor approved|investigational|withdrawn DB01239 Chlorprothixene small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational|withdrawn DB01239 Chlorprothixene small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational|withdrawn DB01239 Chlorprothixene small molecule P35367 Histamine H1 receptor approved|investigational|withdrawn DB01239 Chlorprothixene small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational|withdrawn DB01239 Chlorprothixene small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational|withdrawn DB01239 Chlorprothixene small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational|withdrawn DB01239 Chlorprothixene small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB01240 Epoprostenol small molecule Q9H244 P2Y purinoceptor 12 approved DB01240 Epoprostenol small molecule Q16647 Prostacyclin synthase approved DB01241 Gemfibrozil small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved|investigational|vet_approved DB01242 Clomipramine small molecule P31645 Sodium-dependent serotonin transporter approved|investigational|vet_approved DB01242 Clomipramine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational|vet_approved DB01242 Clomipramine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational|vet_approved DB01242 Clomipramine small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational|vet_approved DB01242 Clomipramine small molecule P09211 Glutathione S-transferase P approved|withdrawn DB01244 Bepridil small molecule O00555 Voltage-dependent P/Q-type calcium channel subunit alpha-1A approved|withdrawn DB01244 Bepridil small molecule O95180 Voltage-dependent T-type calcium channel subunit alpha-1H approved|withdrawn DB01244 Bepridil small molecule Q9NY47 Voltage-dependent calcium channel subunit alpha-2/delta-2 approved|withdrawn DB01244 Bepridil small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved|withdrawn DB01244 Bepridil small molecule P51787 Potassium voltage-gated channel subfamily KQT member 1 {ECO:0000305} approved|withdrawn DB01244 Bepridil small molecule P63316 Troponin C, slow skeletal and cardiac muscles approved|withdrawn DB01244 Bepridil small molecule P54750 Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A approved|withdrawn DB01244 Bepridil small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|vet_approved DB01246 Alimemazine small molecule P35367 Histamine H1 receptor approved DB01247 Isocarboxazid small molecule P21397 Amine oxidase [flavin-containing] A approved DB01247 Isocarboxazid small molecule P27338 Amine oxidase [flavin-containing] B approved|investigational DB01248 Docetaxel small molecule P10415 Apoptosis regulator Bcl-2 approved|investigational DB01248 Docetaxel small molecule P11137 Microtubule-associated protein 2 approved|investigational DB01248 Docetaxel small molecule P27816 Microtubule-associated protein 4 approved|investigational DB01248 Docetaxel small molecule P10636 Microtubule-associated protein tau approved|investigational DB01248 Docetaxel small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB01250 Olsalazine small molecule P51580 Thiopurine S-methyltransferase {ECO:0000303|PubMed:18484748} approved DB01250 Olsalazine small molecule P01579 Interferon gamma approved|investigational DB01251 Gliquidone small molecule Q09428 ATP-binding cassette sub-family C member 8 approved|investigational DB01252 Mitiglinide small molecule Q09428 ATP-binding cassette sub-family C member 8 approved|investigational DB01252 Mitiglinide small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|investigational DB01254 Dasatinib small molecule P00519 Tyrosine-protein kinase ABL1 approved|investigational DB01254 Dasatinib small molecule P12931 Proto-oncogene tyrosine-protein kinase Src approved|investigational DB01254 Dasatinib small molecule P29317 Ephrin type-A receptor 2 approved|investigational DB01254 Dasatinib small molecule P06239 Tyrosine-protein kinase Lck approved|investigational DB01254 Dasatinib small molecule P07947 Tyrosine-protein kinase Yes approved|investigational DB01254 Dasatinib small molecule P10721 Mast/stem cell growth factor receptor Kit approved|investigational DB01254 Dasatinib small molecule P09619 Platelet-derived growth factor receptor beta approved|investigational DB01254 Dasatinib small molecule P51692 Signal transducer and activator of transcription 5B approved|investigational DB01254 Dasatinib small molecule P42684 Tyrosine-protein kinase ABL2 approved|investigational DB01254 Dasatinib small molecule P06241 Tyrosine-protein kinase Fyn approved|investigational DB01254 Dasatinib small molecule Q06187 Tyrosine-protein kinase BTK approved|investigational DB01254 Dasatinib small molecule Q92570 Nuclear receptor subfamily 4 group A member 3 approved|investigational DB01254 Dasatinib small molecule P11274 Breakpoint cluster region protein approved|investigational DB01254 Dasatinib small molecule P41240 Tyrosine-protein kinase CSK approved|investigational DB01254 Dasatinib small molecule P54756 Ephrin type-A receptor 5 approved|investigational DB01254 Dasatinib small molecule P54760 Ephrin type-B receptor 4 approved|investigational DB01254 Dasatinib small molecule P09769 Tyrosine-protein kinase Fgr approved|investigational DB01254 Dasatinib small molecule P42685 Tyrosine-protein kinase FRK approved|investigational DB01254 Dasatinib small molecule P11142 Heat shock cognate 71 kDa protein approved|investigational DB01254 Dasatinib small molecule P07948 Tyrosine-protein kinase Lyn approved|investigational DB01254 Dasatinib small molecule Q16539 Mitogen-activated protein kinase 14 approved|investigational DB01254 Dasatinib small molecule Q06203 Amidophosphoribosyltransferase approved|investigational DB01257 Eculizumab biotech P01031 Complement C5 approved|investigational DB01259 Lapatinib small molecule P00533 Epidermal growth factor receptor approved|investigational DB01259 Lapatinib small molecule P04626 Receptor tyrosine-protein kinase erbB-2 approved|investigational DB01260 Desonide small molecule P04150 Glucocorticoid receptor approved|investigational DB01261 Sitagliptin small molecule P27487 Dipeptidyl peptidase 4 approved|investigational DB01262 Decitabine small molecule P26358 DNA (cytosine-5)-methyltransferase 1 approved DB01267 Paliperidone small molecule P28223 5-hydroxytryptamine receptor 2A approved DB01267 Paliperidone small molecule P14416 D(2) dopamine receptor approved DB01267 Paliperidone small molecule P35367 Histamine H1 receptor approved DB01267 Paliperidone small molecule P21917 D(4) dopamine receptor approved DB01267 Paliperidone small molecule P35462 D(3) dopamine receptor approved DB01267 Paliperidone small molecule P28335 5-hydroxytryptamine receptor 2C approved DB01267 Paliperidone small molecule P08684 Cytochrome P450 3A4 approved DB01267 Paliperidone small molecule P10635 Cytochrome P450 2D6 approved DB01267 Paliperidone small molecule P20815 Cytochrome P450 3A5 approved DB01267 Paliperidone small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational DB01268 Sunitinib small molecule P09619 Platelet-derived growth factor receptor beta approved|investigational DB01268 Sunitinib small molecule P17948 Vascular endothelial growth factor receptor 1 approved|investigational DB01268 Sunitinib small molecule P10721 Mast/stem cell growth factor receptor Kit approved|investigational DB01268 Sunitinib small molecule P35916 Vascular endothelial growth factor receptor 3 approved|investigational DB01268 Sunitinib small molecule P36888 Receptor-type tyrosine-protein kinase FLT3 approved|investigational DB01268 Sunitinib small molecule P07333 Macrophage colony-stimulating factor 1 receptor approved|investigational DB01268 Sunitinib small molecule P16234 Platelet-derived growth factor receptor alpha approved|investigational DB01269 Panitumumab biotech P00533 Epidermal growth factor receptor approved DB01270 Ranibizumab biotech P15692 Vascular endothelial growth factor A approved DB01271 Idursulfase biotech O60664 Perilipin-3 approved|investigational DB01273 Varenicline small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|investigational DB01273 Varenicline small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|investigational DB01273 Varenicline small molecule P32297 Neuronal acetylcholine receptor subunit alpha-3 approved|investigational DB01273 Varenicline small molecule Q15825 Neuronal acetylcholine receptor subunit alpha-6 approved|investigational DB01273 Varenicline small molecule P17787 Neuronal acetylcholine receptor subunit beta-2 approved DB01275 Hydralazine small molecule P13674 Prolyl 4-hydroxylase subunit alpha-1 approved|investigational DB01277 Mecasermin biotech P08069 Insulin-like growth factor 1 receptor approved|investigational DB01277 Mecasermin biotech P17936 Insulin-like growth factor-binding protein 3 approved|investigational DB01277 Mecasermin biotech P06213 Insulin receptor approved|investigational DB01277 Mecasermin biotech P11717 Cation-independent mannose-6-phosphate receptor approved|investigational DB01278 Pramlintide biotech P30988 Calcitonin receptor approved|investigational DB01278 Pramlintide biotech O60894 Receptor activity-modifying protein 1 approved|investigational DB01278 Pramlintide biotech O60895 Receptor activity-modifying protein 2 approved|investigational DB01278 Pramlintide biotech O60896 Receptor activity-modifying protein 3 approved|investigational DB01279 Galsulfase biotech O60664 Perilipin-3 approved|investigational DB01280 Nelarabine small molecule P09884 DNA polymerase alpha catalytic subunit approved DB01281 Abatacept biotech P33681 T-lymphocyte activation antigen CD80 approved DB01281 Abatacept biotech P42081 T-lymphocyte activation antigen CD86 approved|investigational DB01282 Carbetocin small molecule P30559 Oxytocin receptor approved|investigational DB01283 Lumiracoxib small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB01283 Lumiracoxib small molecule P23219 Prostaglandin G/H synthase 1 approved DB01284 Tetracosactide small molecule Q01718 Adrenocorticotropic hormone receptor approved|investigational|vet_approved DB01285 Corticotropin biotech Q01718 Adrenocorticotropic hormone receptor approved|investigational DB01288 Fenoterol small molecule P13945 Beta-3 adrenergic receptor approved|investigational DB01296 Glucosamine small molecule P14780 Matrix metalloproteinase-9 approved|investigational DB01296 Glucosamine small molecule Q00653 Nuclear factor NF-kappa-B p100 subunit approved|investigational DB01296 Glucosamine small molecule P01375 Tumor necrosis factor approved|investigational DB01296 Glucosamine small molecule P01579 Interferon gamma approved DB01303 Oxtriphylline small molecule Q14432 cGMP-inhibited 3',5'-cyclic phosphodiesterase A approved DB01303 Oxtriphylline small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved DB01303 Oxtriphylline small molecule P30542 Adenosine receptor A1 approved DB01303 Oxtriphylline small molecule Q92769 Histone deacetylase 2 approved DB01306 Insulin Aspart biotech P06213 Insulin receptor approved DB01307 Insulin Detemir biotech P06213 Insulin receptor approved DB01309 Insulin Glulisine biotech P06213 Insulin receptor approved|investigational DB01320 Fosphenytoin small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB01324 Polythiazide small molecule P55017 Solute carrier family 12 member 3 approved DB01325 Quinethazone small molecule P00915 Carbonic anhydrase 1 approved DB01325 Quinethazone small molecule P00918 Carbonic anhydrase 2 approved DB01325 Quinethazone small molecule Q13621 Solute carrier family 12 member 1 approved DB01325 Quinethazone small molecule P55011 Solute carrier family 12 member 2 approved DB01325 Quinethazone small molecule P55017 Solute carrier family 12 member 3 approved DB01327 Cefazolin small molecule P27169 Serum paraoxonase/arylesterase 1 {ECO:0000303|PubMed:7916578} approved DB01327 Cefazolin small molecule P40933 Interleukin-15 approved DB01327 Cefazolin small molecule P60568 Interleukin-2 approved DB01337 Pancuronium small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB01337 Pancuronium small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB01337 Pancuronium small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB01338 Pipecuronium small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB01338 Pipecuronium small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB01338 Pipecuronium small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB01339 Vecuronium small molecule Q15822 Neuronal acetylcholine receptor subunit alpha-2 approved DB01340 Cilazapril small molecule P12821 Angiotensin-converting enzyme approved|investigational DB01345 Potassium small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved DB01348 Spirapril small molecule P12821 Angiotensin-converting enzyme approved DB01349 Tasosartan small molecule P30556 Type-1 angiotensin II receptor approved|illicit DB01351 Amobarbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01351 Amobarbital small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB01351 Amobarbital small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB01351 Amobarbital small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB01351 Amobarbital small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|illicit DB01351 Amobarbital small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|illicit DB01351 Amobarbital small molecule P42262 Glutamate receptor 2 approved|illicit DB01351 Amobarbital small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved|illicit DB01352 Aprobarbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01352 Aprobarbital small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB01352 Aprobarbital small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB01352 Aprobarbital small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB01352 Aprobarbital small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|illicit DB01352 Aprobarbital small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|illicit DB01352 Aprobarbital small molecule P42262 Glutamate receptor 2 approved|illicit DB01352 Aprobarbital small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved|illicit DB01353 Butethal small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01353 Butethal small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB01353 Butethal small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB01353 Butethal small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB01353 Butethal small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved|illicit DB01353 Butethal small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|illicit DB01353 Butethal small molecule P42262 Glutamate receptor 2 approved|illicit DB01353 Butethal small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved DB01354 Heptabarbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01354 Heptabarbital small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB01354 Heptabarbital small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB01354 Heptabarbital small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved DB01354 Heptabarbital small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved DB01354 Heptabarbital small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved DB01354 Heptabarbital small molecule P42262 Glutamate receptor 2 approved DB01354 Heptabarbital small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved DB01355 Hexobarbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01355 Hexobarbital small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB01355 Hexobarbital small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB01355 Hexobarbital small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved DB01355 Hexobarbital small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 approved DB01355 Hexobarbital small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved DB01355 Hexobarbital small molecule P42262 Glutamate receptor 2 approved DB01355 Hexobarbital small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved DB01356 Lithium small molecule P49841 Glycogen synthase kinase-3 beta approved DB01356 Lithium small molecule P29218 Inositol monophosphatase 1 approved DB01356 Lithium small molecule O14732 Inositol monophosphatase 2 approved DB01356 Lithium small molecule P42263 Glutamate receptor 3 approved DB01364 Ephedrine small molecule P23975 Sodium-dependent noradrenaline transporter approved DB01364 Ephedrine small molecule Q05940 Synaptic vesicular amine transporter approved DB01364 Ephedrine small molecule P22303 Acetylcholinesterase approved DB01367 Rasagiline small molecule P27338 Amine oxidase [flavin-containing] B approved DB01367 Rasagiline small molecule P10415 Apoptosis regulator Bcl-2 approved|investigational DB01370 Aluminium small molecule P02787 Serotransferrin approved|investigational DB01370 Aluminium small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved|investigational DB01370 Aluminium small molecule P06870 Kallikrein-1 approved|investigational DB01370 Aluminium small molecule P05067 Amyloid-beta A4 protein approved|nutraceutical DB01373 Calcium small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|nutraceutical DB01373 Calcium small molecule P98194 Calcium-transporting ATPase type 2C member 1 approved|nutraceutical DB01373 Calcium small molecule P02585 Troponin C, skeletal muscle approved|nutraceutical DB01373 Calcium small molecule P63316 Troponin C, slow skeletal and cardiac muscles approved|nutraceutical DB01373 Calcium small molecule Q01082 Spectrin beta chain, non-erythrocytic 1 approved|nutraceutical DB01373 Calcium small molecule P04271 Protein S100-B approved|nutraceutical DB01373 Calcium small molecule P20810 Calpastatin approved|nutraceutical DB01373 Calcium small molecule P49747 Cartilage oligomeric matrix protein approved|nutraceutical DB01373 Calcium small molecule P19801 Amiloride-sensitive amine oxidase [copper-containing] approved|nutraceutical DB01373 Calcium small molecule Q99584 Protein S100-A13 approved|nutraceutical DB01373 Calcium small molecule P05187 Alkaline phosphatase, placental type approved|nutraceutical DB01373 Calcium small molecule P05109 Protein S100-A8 approved|nutraceutical DB01373 Calcium small molecule P06702 Protein S100-A9 approved|nutraceutical DB01373 Calcium small molecule P29034 Protein S100-A2 approved|nutraceutical DB01373 Calcium small molecule P00450 Ceruloplasmin approved|nutraceutical DB01373 Calcium small molecule P12644 Bone morphogenetic protein 4 approved|nutraceutical DB01373 Calcium small molecule P08493 Matrix Gla protein approved|nutraceutical DB01373 Calcium small molecule O75340 Programmed cell death protein 6 approved|nutraceutical DB01378 Magnesium small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved|investigational DB01380 Cortisone acetate small molecule P04150 Glucocorticoid receptor approved|investigational|nutraceutical DB01381 Ginkgo biloba small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational|nutraceutical DB01381 Ginkgo biloba small molecule P14555 Phospholipase A2, membrane associated approved|investigational|nutraceutical DB01381 Ginkgo biloba small molecule P23415 Glycine receptor subunit alpha-1 approved|investigational|nutraceutical DB01381 Ginkgo biloba small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational|nutraceutical DB01381 Ginkgo biloba small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|investigational DB01382 Glycodiazine small molecule Q09428 ATP-binding cassette sub-family C member 8 approved DB01384 Paramethasone small molecule P04150 Glucocorticoid receptor investigational|withdrawn DB01388 Mibefradil small molecule O43497 Voltage-dependent T-type calcium channel subunit alpha-1G investigational|withdrawn DB01388 Mibefradil small molecule O95180 Voltage-dependent T-type calcium channel subunit alpha-1H investigational|withdrawn DB01388 Mibefradil small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C investigational|withdrawn DB01388 Mibefradil small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D investigational|withdrawn DB01388 Mibefradil small molecule O60840 Voltage-dependent L-type calcium channel subunit alpha-1F {ECO:0000305} investigational|withdrawn DB01388 Mibefradil small molecule Q9P0X4 Voltage-dependent T-type calcium channel subunit alpha-1I investigational|withdrawn DB01388 Mibefradil small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S investigational|withdrawn DB01388 Mibefradil small molecule Q02641 Voltage-dependent L-type calcium channel subunit beta-1 investigational|withdrawn DB01388 Mibefradil small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 investigational|withdrawn DB01388 Mibefradil small molecule P54284 Voltage-dependent L-type calcium channel subunit beta-3 investigational|withdrawn DB01388 Mibefradil small molecule O00305 Voltage-dependent L-type calcium channel subunit beta-4 {ECO:0000305} approved|investigational|vet_approved DB01392 Yohimbine small molecule P14416 D(2) dopamine receptor approved|investigational|vet_approved DB01392 Yohimbine small molecule P35462 D(3) dopamine receptor approved|investigational|vet_approved DB01392 Yohimbine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational|vet_approved DB01392 Yohimbine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB01393 Bezafibrate small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved|investigational DB01393 Bezafibrate small molecule Q03181 Peroxisome proliferator-activated receptor delta approved|investigational DB01393 Bezafibrate small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|investigational DB01393 Bezafibrate small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB01393 Bezafibrate small molecule P19793 Retinoic acid receptor RXR-alpha approved|investigational DB01393 Bezafibrate small molecule P28702 Retinoic acid receptor RXR-beta approved|investigational DB01393 Bezafibrate small molecule P48443 Retinoic acid receptor RXR-gamma approved DB01394 Colchicine small molecule P07437 Tubulin beta chain approved DB01395 Drospirenone small molecule P06401 Progesterone receptor approved DB01395 Drospirenone small molecule P08235 Mineralocorticoid receptor approved DB01395 Drospirenone small molecule P10275 Androgen receptor approved|investigational DB01396 Digitoxin small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved DB01399 Salsalate small molecule P35354 Prostaglandin G/H synthase 2 approved DB01399 Salsalate small molecule P23219 Prostaglandin G/H synthase 1 approved|vet_approved DB01400 Neostigmine small molecule P22303 Acetylcholinesterase approved|investigational DB01403 Methotrimeprazine small molecule P14416 D(2) dopamine receptor approved|investigational DB01403 Methotrimeprazine small molecule P35462 D(3) dopamine receptor approved|investigational DB01403 Methotrimeprazine small molecule P21917 D(4) dopamine receptor approved|investigational DB01403 Methotrimeprazine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB01403 Methotrimeprazine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB01403 Methotrimeprazine small molecule P35367 Histamine H1 receptor approved|investigational DB01403 Methotrimeprazine small molecule P11229 Muscarinic acetylcholine receptor M1 approved|investigational DB01403 Methotrimeprazine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational DB01403 Methotrimeprazine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB01403 Methotrimeprazine small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB01403 Methotrimeprazine small molecule P25100 Alpha-1D adrenergic receptor approved DB01406 Danazol small molecule P03372 Estrogen receptor approved DB01406 Danazol small molecule P10275 Androgen receptor approved DB01406 Danazol small molecule P06401 Progesterone receptor approved DB01406 Danazol small molecule P13500 C-C motif chemokine 2 approved|investigational|vet_approved DB01407 Clenbuterol small molecule P13945 Beta-3 adrenergic receptor approved|investigational|vet_approved DB01407 Clenbuterol small molecule P01375 Tumor necrosis factor approved DB01409 Tiotropium small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB01409 Tiotropium small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB01409 Tiotropium small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB01409 Tiotropium small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB01410 Ciclesonide small molecule P04150 Glucocorticoid receptor approved|investigational DB01411 Pranlukast small molecule Q9Y271 Cysteinyl leukotriene receptor 1 approved|investigational DB01411 Pranlukast small molecule P01375 Tumor necrosis factor approved|investigational DB01411 Pranlukast small molecule P05113 Interleukin-5 approved|investigational DB01411 Pranlukast small molecule P19838 Nuclear factor NF-kappa-B p105 subunit approved|investigational DB01411 Pranlukast small molecule Q02817 Mucin-2 approved|investigational DB01412 Theobromine small molecule P30542 Adenosine receptor A1 approved|investigational DB01412 Theobromine small molecule Q07343 cAMP-specific 3',5'-cyclic phosphodiesterase 4B approved|investigational DB01418 Acenocoumarol small molecule Q9BQB6 Vitamin K epoxide reductase complex subunit 1 approved DB01422 Nitroxoline small molecule P50579 Methionine aminopeptidase 2 {ECO:0000255|HAMAP-Rule:MF_03175} approved DB01425 Alizapride small molecule P14416 D(2) dopamine receptor approved|investigational DB01426 Ajmaline small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB01427 Amrinone small molecule Q14432 cGMP-inhibited 3',5'-cyclic phosphodiesterase A approved DB01427 Amrinone small molecule Q07343 cAMP-specific 3',5'-cyclic phosphodiesterase 4B approved DB01427 Amrinone small molecule P01375 Tumor necrosis factor approved DB01429 Aprindine small molecule Q14524 Sodium channel protein type 5 subunit alpha approved DB01430 Almitrine small molecule P05023 Sodium/potassium-transporting ATPase subunit alpha-1 approved DB01431 Allylestrenol small molecule P06401 Progesterone receptor approved DB01431 Allylestrenol small molecule P03372 Estrogen receptor approved|investigational DB01435 Antipyrine small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB01435 Antipyrine small molecule P23219 Prostaglandin G/H synthase 1 approved|nutraceutical DB01436 Alfacalcidol small molecule P11473 Vitamin D3 receptor approved|nutraceutical DB01436 Alfacalcidol small molecule O15528 25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrial approved|nutraceutical DB01436 Alfacalcidol small molecule P19793 Retinoic acid receptor RXR-alpha approved|illicit DB01437 Glutethimide small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01437 Glutethimide small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit|investigational DB01452 Heroin small molecule P35372 Mu-type opioid receptor approved|illicit|investigational DB01452 Heroin small molecule P41143 Delta-type opioid receptor approved|illicit|investigational DB01452 Heroin small molecule P23141 Liver carboxylesterase 1 approved|illicit DB01466 Ethylmorphine small molecule P35372 Mu-type opioid receptor illicit DB01483 Barbital small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 illicit DB01483 Barbital small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 illicit DB01483 Barbital small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 illicit DB01483 Barbital small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 illicit DB01483 Barbital small molecule P43681 Neuronal acetylcholine receptor subunit alpha-4 illicit DB01483 Barbital small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 illicit DB01483 Barbital small molecule P42262 Glutamate receptor 2 illicit DB01483 Barbital small molecule Q13002 Glutamate receptor ionotropic, kainate 2 approved|illicit DB01544 Flunitrazepam small molecule P30536 Translocator protein approved|illicit DB01544 Flunitrazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB01544 Flunitrazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB01544 Flunitrazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB01544 Flunitrazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01544 Flunitrazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|illicit DB01544 Flunitrazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|illicit|investigational DB01558 Bromazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit|investigational DB01558 Bromazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit|investigational DB01558 Bromazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit|investigational DB01558 Bromazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit|investigational DB01558 Bromazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|illicit|investigational DB01558 Bromazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|illicit|investigational DB01558 Bromazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|illicit|investigational DB01558 Bromazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|illicit|investigational DB01558 Bromazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|illicit|investigational DB01558 Bromazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|illicit|investigational DB01558 Bromazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|illicit|investigational DB01558 Bromazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|illicit|investigational DB01558 Bromazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|illicit|investigational DB01558 Bromazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|illicit DB01559 Clotiazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01559 Clotiazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB01559 Clotiazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB01559 Clotiazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB01559 Clotiazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|illicit DB01559 Clotiazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|illicit DB01559 Clotiazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|illicit DB01559 Clotiazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|illicit DB01559 Clotiazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|illicit DB01559 Clotiazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|illicit DB01559 Clotiazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|illicit DB01559 Clotiazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|illicit DB01559 Clotiazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|illicit DB01559 Clotiazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|illicit DB01567 Fludiazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01567 Fludiazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB01567 Fludiazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB01567 Fludiazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB01567 Fludiazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|illicit DB01567 Fludiazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|illicit DB01567 Fludiazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|illicit DB01567 Fludiazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|illicit DB01567 Fludiazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|illicit DB01567 Fludiazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|illicit DB01567 Fludiazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|illicit DB01567 Fludiazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|illicit DB01567 Fludiazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|illicit DB01567 Fludiazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|illicit DB01576 Dextroamphetamine small molecule Q05940 Synaptic vesicular amine transporter approved|illicit DB01576 Dextroamphetamine small molecule P23975 Sodium-dependent noradrenaline transporter approved|illicit DB01577 Methamphetamine small molecule P31645 Sodium-dependent serotonin transporter approved|illicit DB01577 Methamphetamine small molecule P23975 Sodium-dependent noradrenaline transporter approved|illicit DB01577 Methamphetamine small molecule Q05940 Synaptic vesicular amine transporter approved|illicit DB01577 Methamphetamine small molecule P21397 Amine oxidase [flavin-containing] A approved|illicit DB01577 Methamphetamine small molecule P27338 Amine oxidase [flavin-containing] B approved DB01580 Oxprenolol small molecule P13945 Beta-3 adrenergic receptor approved|investigational DB01586 Ursodeoxycholic acid small molecule P52895 Aldo-keto reductase family 1 member C2 approved DB01587 Ketazolam small molecule P30536 Translocator protein approved DB01587 Ketazolam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01587 Ketazolam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved DB01587 Ketazolam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved DB01587 Ketazolam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved DB01587 Ketazolam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|illicit DB01588 Prazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01588 Prazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB01588 Prazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB01588 Prazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB01588 Prazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|illicit DB01588 Prazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|illicit DB01588 Prazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|illicit DB01588 Prazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|illicit DB01588 Prazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|illicit DB01588 Prazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|illicit DB01588 Prazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|illicit DB01588 Prazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|illicit DB01588 Prazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|illicit DB01588 Prazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|illicit DB01588 Prazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01589 Quazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|illicit DB01589 Quazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved|illicit DB01589 Quazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved|illicit DB01589 Quazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved|illicit DB01589 Quazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved|illicit DB01589 Quazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved|illicit DB01589 Quazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved|illicit DB01589 Quazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved|illicit DB01589 Quazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved|illicit DB01589 Quazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved|illicit DB01589 Quazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved|illicit DB01589 Quazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved|illicit DB01589 Quazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved|illicit DB01589 Quazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|illicit DB01589 Quazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01590 Everolimus small molecule P42345 Serine/threonine-protein kinase mTOR approved DB01591 Solifenacin small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB01591 Solifenacin small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB01591 Solifenacin small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB01591 Solifenacin small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB01592 Iron small molecule P02786 Transferrin receptor protein 1 approved DB01592 Iron small molecule Q9GZT9 Egl nine homolog 1 approved DB01592 Iron small molecule Q9BY41 Histone deacetylase 8 approved DB01592 Iron small molecule Q9NZD4 Alpha-hemoglobin-stabilizing protein approved DB01592 Iron small molecule P69905 Hemoglobin subunit alpha approved DB01592 Iron small molecule Q16595 Frataxin, mitochondrial approved DB01592 Iron small molecule P02794 Ferritin heavy chain approved DB01592 Iron small molecule P39748 Flap endonuclease 1 {ECO:0000255|HAMAP-Rule:MF_03140} approved DB01592 Iron small molecule Q96FI4 Endonuclease 8-like 1 approved DB01592 Iron small molecule Q969S2 Endonuclease 8-like 2 approved DB01592 Iron small molecule P06746 DNA polymerase beta approved DB01592 Iron small molecule P00450 Ceruloplasmin approved DB01592 Iron small molecule P02787 Serotransferrin approved|investigational DB01593 Zinc small molecule P16455 Methylated-DNA--protein-cysteine methyltransferase approved|investigational DB01593 Zinc small molecule P04075 Fructose-bisphosphate aldolase A approved|investigational DB01593 Zinc small molecule P68104 Elongation factor 1-alpha 1 approved|investigational DB01593 Zinc small molecule P06733 Alpha-enolase approved|investigational DB01593 Zinc small molecule O14556 Glyceraldehyde-3-phosphate dehydrogenase, testis-specific approved|investigational DB01593 Zinc small molecule P15531 Nucleoside diphosphate kinase A approved|investigational DB01593 Zinc small molecule P07237 Protein disulfide-isomerase approved|investigational DB01593 Zinc small molecule P30101 Protein disulfide-isomerase A3 approved|investigational DB01593 Zinc small molecule Q06830 Peroxiredoxin-1 approved|investigational DB01593 Zinc small molecule P78330 Phosphoserine phosphatase approved|investigational DB01593 Zinc small molecule P60174 Triosephosphate isomerase approved|investigational DB01593 Zinc small molecule P03372 Estrogen receptor approved|investigational DB01593 Zinc small molecule P02795 Metallothionein-2 approved|investigational DB01593 Zinc small molecule O14618 Copper chaperone for superoxide dismutase approved|investigational DB01593 Zinc small molecule Q13547 Histone deacetylase 1 approved|investigational DB01593 Zinc small molecule P56524 Histone deacetylase 4 approved|investigational DB01593 Zinc small molecule P29372 DNA-3-methyladenine glycosylase approved|investigational DB01593 Zinc small molecule P00441 Superoxide dismutase [Cu-Zn] approved|investigational DB01593 Zinc small molecule Q9BY41 Histone deacetylase 8 approved|investigational DB01593 Zinc small molecule O15304 Apoptosis regulatory protein Siva approved|investigational DB01593 Zinc small molecule P23415 Glycine receptor subunit alpha-1 approved|investigational DB01593 Zinc small molecule Q00987 E3 ubiquitin-protein ligase Mdm2 approved|investigational DB01593 Zinc small molecule P46939 Utrophin approved|investigational DB01593 Zinc small molecule P45381 Aspartoacylase approved|investigational DB01593 Zinc small molecule P05109 Protein S100-A8 approved|investigational DB01593 Zinc small molecule P06702 Protein S100-A9 approved|investigational DB01593 Zinc small molecule P14780 Matrix metalloproteinase-9 approved|investigational DB01593 Zinc small molecule O15350 Tumor protein p73 approved|investigational DB01593 Zinc small molecule P29034 Protein S100-A2 approved|investigational DB01593 Zinc small molecule P04637 Cellular tumor antigen p53 approved|investigational DB01593 Zinc small molecule P25713 Metallothionein-3 approved|investigational DB01593 Zinc small molecule O75340 Programmed cell death protein 6 approved|investigational DB01593 Zinc small molecule Q8N907 DAN domain family member 5 approved|investigational DB01593 Zinc small molecule P04731 Metallothionein-1A approved|investigational DB01593 Zinc small molecule P04217 Alpha-1B-glycoprotein approved|investigational DB01593 Zinc small molecule P01023 Alpha-2-macroglobulin approved|investigational DB01593 Zinc small molecule P01019 Angiotensinogen approved|investigational DB01593 Zinc small molecule P02765 Alpha-2-HS-glycoprotein approved|investigational DB01593 Zinc small molecule P02743 Serum amyloid P-component approved|investigational DB01593 Zinc small molecule P02647 Apolipoprotein A-I approved|investigational DB01593 Zinc small molecule P02652 Apolipoprotein A-II approved|investigational DB01593 Zinc small molecule P02649 Apolipoprotein E approved|investigational DB01593 Zinc small molecule O14791 Apolipoprotein L1 approved|investigational DB01593 Zinc small molecule P02746 Complement C1q subcomponent subunit B approved|investigational DB01593 Zinc small molecule P02747 Complement C1q subcomponent subunit C approved|investigational DB01593 Zinc small molecule P09871 Complement C1s subcomponent approved|investigational DB01593 Zinc small molecule P01024 Complement C3 approved|investigational DB01593 Zinc small molecule P0C0L5 Complement C4-B approved|investigational DB01593 Zinc small molecule P04003 C4b-binding protein alpha chain approved|investigational DB01593 Zinc small molecule P20851 C4b-binding protein beta chain approved|investigational DB01593 Zinc small molecule P01031 Complement C5 approved|investigational DB01593 Zinc small molecule P46736 Lys-63-specific deubiquitinase BRCC36 approved|investigational DB01593 Zinc small molecule P07357 Complement component C8 alpha chain approved|investigational DB01593 Zinc small molecule P07358 Complement component C8 beta chain approved|investigational DB01593 Zinc small molecule P00751 Complement factor B approved|investigational DB01593 Zinc small molecule P08603 Complement factor H approved|investigational DB01593 Zinc small molecule P05156 Complement factor I approved|investigational DB01593 Zinc small molecule P10909 Clusterin approved|investigational DB01593 Zinc small molecule P00450 Ceruloplasmin approved|investigational DB01593 Zinc small molecule P15169 Carboxypeptidase N catalytic chain approved|investigational DB01593 Zinc small molecule P15924 Desmoplakin approved|investigational DB01593 Zinc small molecule P00748 Coagulation factor XII approved|investigational DB01593 Zinc small molecule P05160 Coagulation factor XIII B chain approved|investigational DB01593 Zinc small molecule P00734 Prothrombin approved|investigational DB01593 Zinc small molecule O75636 Ficolin-3 approved|investigational DB01593 Zinc small molecule P02671 Fibrinogen alpha chain approved|investigational DB01593 Zinc small molecule P02751 Fibronectin approved|investigational DB01593 Zinc small molecule P06396 Gelsolin approved|investigational DB01593 Zinc small molecule P69905 Hemoglobin subunit alpha approved|investigational DB01593 Zinc small molecule P68871 Hemoglobin subunit beta approved|investigational DB01593 Zinc small molecule P01876 Immunoglobulin heavy constant alpha 1 {ECO:0000303|PubMed:11340299, ECO:0000303|Ref.11} approved|investigational DB01593 Zinc small molecule P19823 Inter-alpha-trypsin inhibitor heavy chain H2 approved|investigational DB01593 Zinc small molecule Q06033 Inter-alpha-trypsin inhibitor heavy chain H3 approved|investigational DB01593 Zinc small molecule Q14624 Inter-alpha-trypsin inhibitor heavy chain H4 approved|investigational DB01593 Zinc small molecule P14923 Junction plakoglobin approved|investigational DB01593 Zinc small molecule P01042 Kininogen-1 approved|investigational DB01593 Zinc small molecule P04264 Keratin, type II cytoskeletal 1 approved|investigational DB01593 Zinc small molecule P13645 Keratin, type I cytoskeletal 10 approved|investigational DB01593 Zinc small molecule P02533 Keratin, type I cytoskeletal 14 approved|investigational DB01593 Zinc small molecule P08779 Keratin, type I cytoskeletal 16 approved|investigational DB01593 Zinc small molecule P35908 Keratin, type II cytoskeletal 2 epidermal approved|investigational DB01593 Zinc small molecule P13647 Keratin, type II cytoskeletal 5 approved|investigational DB01593 Zinc small molecule P02538 Keratin, type II cytoskeletal 6A approved|investigational DB01593 Zinc small molecule P35527 Keratin, type I cytoskeletal 9 approved|investigational DB01593 Zinc small molecule P19652 Alpha-1-acid glycoprotein 2 approved|investigational DB01593 Zinc small molecule Q96PD5 N-acetylmuramoyl-L-alanine amidase approved|investigational DB01593 Zinc small molecule P27169 Serum paraoxonase/arylesterase 1 {ECO:0000303|PubMed:7916578} approved|investigational DB01593 Zinc small molecule P20742 Pregnancy zone protein approved|investigational DB01593 Zinc small molecule P31151 Protein S100-A7 approved|investigational DB01593 Zinc small molecule P49908 Selenoprotein P {ECO:0000303|PubMed:27645994} approved|investigational DB01593 Zinc small molecule P01009 Alpha-1-antitrypsin approved|investigational DB01593 Zinc small molecule P01011 Alpha-1-antichymotrypsin approved|investigational DB01593 Zinc small molecule P05546 Heparin cofactor 2 approved|investigational DB01593 Zinc small molecule P04278 Sex hormone-binding globulin approved|investigational DB01593 Zinc small molecule P02787 Serotransferrin approved|investigational DB01593 Zinc small molecule P02766 Transthyretin approved|investigational DB01593 Zinc small molecule P04004 Vitronectin approved|investigational DB01593 Zinc small molecule P51693 Amyloid-like protein 1 approved|investigational DB01593 Zinc small molecule Q06481 Amyloid-like protein 2 approved|investigational DB01593 Zinc small molecule P05067 Amyloid-beta A4 protein approved|investigational DB01593 Zinc small molecule P09874 Poly [ADP-ribose] polymerase 1 approved DB01594 Cinolazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01594 Cinolazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB01594 Cinolazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB01594 Cinolazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved DB01594 Cinolazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved DB01594 Cinolazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved DB01594 Cinolazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved DB01594 Cinolazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved DB01594 Cinolazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved DB01594 Cinolazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved DB01594 Cinolazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved DB01594 Cinolazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved DB01594 Cinolazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved DB01594 Cinolazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved DB01595 Nitrazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB01595 Nitrazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB01595 Nitrazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB01595 Nitrazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved DB01595 Nitrazepam small molecule P18505 Gamma-aminobutyric acid receptor subunit beta-1 approved DB01595 Nitrazepam small molecule P28472 Gamma-aminobutyric acid receptor subunit beta-3 approved DB01595 Nitrazepam small molecule Q8N1C3 Gamma-aminobutyric acid receptor subunit gamma-1 approved DB01595 Nitrazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved DB01595 Nitrazepam small molecule Q99928 Gamma-aminobutyric acid receptor subunit gamma-3 approved DB01595 Nitrazepam small molecule O14764 Gamma-aminobutyric acid receptor subunit delta approved DB01595 Nitrazepam small molecule P78334 Gamma-aminobutyric acid receptor subunit epsilon approved DB01595 Nitrazepam small molecule O00591 Gamma-aminobutyric acid receptor subunit pi approved DB01595 Nitrazepam small molecule P24046 Gamma-aminobutyric acid receptor subunit rho-1 approved DB01595 Nitrazepam small molecule P28476 Gamma-aminobutyric acid receptor subunit rho-2 approved|investigational DB01599 Probucol small molecule O95477 ATP-binding cassette sub-family A member 1 approved|investigational DB01599 Probucol small molecule P23141 Liver carboxylesterase 1 approved DB01600 Tiaprofenic acid small molecule P35354 Prostaglandin G/H synthase 2 approved DB01600 Tiaprofenic acid small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB01608 Propericiazine small molecule P10275 Androgen receptor approved DB01611 Hydroxychloroquine small molecule Q9NYK1 Toll-like receptor 7 approved DB01611 Hydroxychloroquine small molecule Q9NR96 Toll-like receptor 9 approved|investigational DB01613 Erythrityl Tetranitrate small molecule P20594 Atrial natriuretic peptide receptor 2 approved|vet_approved DB01614 Acepromazine small molecule P14416 D(2) dopamine receptor approved|vet_approved DB01614 Acepromazine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB01618 Molindone small molecule P14416 D(2) dopamine receptor approved DB01618 Molindone small molecule P28223 5-hydroxytryptamine receptor 2A approved DB01618 Molindone small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB01619 Phenindamine small molecule P35367 Histamine H1 receptor approved DB01620 Pheniramine small molecule P35367 Histamine H1 receptor approved DB01620 Pheniramine small molecule Q14994 Nuclear receptor subfamily 1 group I member 3 approved|investigational DB01621 Pipotiazine small molecule P14416 D(2) dopamine receptor approved|investigational DB01621 Pipotiazine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB01622 Thioproperazine small molecule P14416 D(2) dopamine receptor approved DB01622 Thioproperazine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB01623 Thiothixene small molecule P14416 D(2) dopamine receptor approved DB01623 Thiothixene small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB01624 Zuclopenthixol small molecule P14416 D(2) dopamine receptor approved|investigational DB01624 Zuclopenthixol small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB01624 Zuclopenthixol small molecule P35367 Histamine H1 receptor approved|vet_approved DB01625 Isopropamide small molecule P20309 Muscarinic acetylcholine receptor M3 approved|vet_approved DB01625 Isopropamide small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB01626 Pargyline small molecule P27338 Amine oxidase [flavin-containing] B approved DB01626 Pargyline small molecule P21397 Amine oxidase [flavin-containing] A approved|investigational DB01628 Etoricoxib small molecule P35354 Prostaglandin G/H synthase 2 approved DB01656 Roflumilast small molecule Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D approved DB01656 Roflumilast small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved DB01656 Roflumilast small molecule Q07343 cAMP-specific 3',5'-cyclic phosphodiesterase 4B approved DB01656 Roflumilast small molecule Q08493 cAMP-specific 3',5'-cyclic phosphodiesterase 4C experimental|investigational DB01677 Fumaric Acid small molecule P23368 NAD-dependent malic enzyme, mitochondrial experimental|investigational DB01677 Fumaric Acid small molecule P16930 Fumarylacetoacetase experimental|investigational DB01698 Rutin small molecule P42330 Aldo-keto reductase family 1 member C3 experimental|investigational DB01698 Rutin small molecule P16152 Carbonyl reductase [NADPH] 1 approved|investigational|nutraceutical DB01708 Prasterone small molecule P03372 Estrogen receptor approved|investigational|nutraceutical DB01708 Prasterone small molecule Q92731 Estrogen receptor beta approved|investigational|nutraceutical DB01708 Prasterone small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational|nutraceutical DB01708 Prasterone small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved|investigational|nutraceutical DB01708 Prasterone small molecule P10275 Androgen receptor approved|investigational|nutraceutical DB01708 Prasterone small molecule P14061 Estradiol 17-beta-dehydrogenase 1 approved|investigational|nutraceutical DB01708 Prasterone small molecule Q06520 Bile salt sulfotransferase approved|investigational|nutraceutical DB01708 Prasterone small molecule O00204 Sulfotransferase family cytosolic 2B member 1 approved|investigational|nutraceutical DB01708 Prasterone small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved|investigational|nutraceutical DB01708 Prasterone small molecule Q99720 Sigma non-opioid intracellular receptor 1 approved|investigational|nutraceutical DB01708 Prasterone small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational|nutraceutical DB01708 Prasterone small molecule Q14994 Nuclear receptor subfamily 1 group I member 3 experimental DB02266 Flufenamic Acid small molecule P35354 Prostaglandin G/H synthase 2 experimental DB02266 Flufenamic Acid small molecule P23219 Prostaglandin G/H synthase 1 experimental DB02266 Flufenamic Acid small molecule P42330 Aldo-keto reductase family 1 member C3 experimental DB02266 Flufenamic Acid small molecule P10275 Androgen receptor experimental DB02266 Flufenamic Acid small molecule Q07869 Peroxisome proliferator-activated receptor alpha experimental DB02266 Flufenamic Acid small molecule P37231 Peroxisome proliferator-activated receptor gamma approved DB02300 Calcipotriol small molecule P11473 Vitamin D3 receptor approved|investigational DB02325 Isopropyl Alcohol small molecule O60942 mRNA-capping enzyme approved|investigational DB02325 Isopropyl Alcohol small molecule Q9BV57 1,2-dihydroxy-3-keto-5-methylthiopentene dioxygenase {ECO:0000255|HAMAP-Rule:MF_03154} approved|investigational DB02325 Isopropyl Alcohol small molecule P30793 GTP cyclohydrolase 1 approved|investigational DB02325 Isopropyl Alcohol small molecule P43026 Growth/differentiation factor 5 approved|investigational DB02325 Isopropyl Alcohol small molecule P07998 Ribonuclease pancreatic approved|investigational DB02325 Isopropyl Alcohol small molecule P14555 Phospholipase A2, membrane associated approved|investigational DB02325 Isopropyl Alcohol small molecule P17900 Ganglioside GM2 activator approved|investigational DB02325 Isopropyl Alcohol small molecule Q13231 Chitotriosidase-1 approved|investigational DB02325 Isopropyl Alcohol small molecule Q7Z4W1 L-xylulose reductase approved|investigational DB02325 Isopropyl Alcohol small molecule P30041 Peroxiredoxin-6 approved|investigational DB02325 Isopropyl Alcohol small molecule P01375 Tumor necrosis factor approved|investigational DB02325 Isopropyl Alcohol small molecule P13686 Tartrate-resistant acid phosphatase type 5 approved|investigational DB02325 Isopropyl Alcohol small molecule P23526 Adenosylhomocysteinase approved|investigational DB02325 Isopropyl Alcohol small molecule Q13838 Spliceosome RNA helicase DDX39B experimental DB02329 Carbenoxolone small molecule P28845 Corticosteroid 11-beta-dehydrogenase isozyme 1 withdrawn DB02383 Tolrestat small molecule P15121 Aldose reductase withdrawn DB02383 Tolrestat small molecule P14550 Alcohol dehydrogenase [NADP(+)] withdrawn DB02383 Tolrestat small molecule O60218 Aldo-keto reductase family 1 member B10 approved|investigational DB02546 Vorinostat small molecule Q13547 Histone deacetylase 1 approved|investigational DB02546 Vorinostat small molecule Q92769 Histone deacetylase 2 approved|investigational DB02546 Vorinostat small molecule O15379 Histone deacetylase 3 approved|investigational DB02546 Vorinostat small molecule Q9UBN7 Histone deacetylase 6 approved|investigational DB02546 Vorinostat small molecule Q9BY41 Histone deacetylase 8 experimental DB02640 Fumagillin small molecule P50579 Methionine aminopeptidase 2 {ECO:0000255|HAMAP-Rule:MF_03175} approved DB02659 Cholic Acid small molecule P22830 Ferrochelatase, mitochondrial approved DB02659 Cholic Acid small molecule P62508 Estrogen-related receptor gamma approved DB02659 Cholic Acid small molecule P51161 Gastrotropin approved DB02659 Cholic Acid small molecule P13073 Cytochrome c oxidase subunit 4 isoform 1, mitochondrial approved DB02659 Cholic Acid small molecule P20674 Cytochrome c oxidase subunit 5A, mitochondrial approved DB02659 Cholic Acid small molecule P10606 Cytochrome c oxidase subunit 5B, mitochondrial approved DB02659 Cholic Acid small molecule P09669 Cytochrome c oxidase subunit 6C approved DB02659 Cholic Acid small molecule P24311 Cytochrome c oxidase subunit 7B, mitochondrial approved DB02659 Cholic Acid small molecule P15954 Cytochrome c oxidase subunit 7C, mitochondrial approved DB02659 Cholic Acid small molecule P10176 Cytochrome c oxidase subunit 8A, mitochondrial approved DB02659 Cholic Acid small molecule Q02221 Cytochrome c oxidase subunit 6A2, mitochondrial approved DB02659 Cholic Acid small molecule P14854 Cytochrome c oxidase subunit 6B1 approved DB02659 Cholic Acid small molecule P24310 Cytochrome c oxidase subunit 7A1, mitochondrial approved DB02659 Cholic Acid small molecule P04054 Phospholipase A2 approved DB02659 Cholic Acid small molecule P23141 Liver carboxylesterase 1 approved|investigational DB02701 Nicotinamide small molecule P00338 L-lactate dehydrogenase A chain approved|investigational DB02701 Nicotinamide small molecule P09874 Poly [ADP-ribose] polymerase 1 approved|investigational DB02701 Nicotinamide small molecule Q9NXA8 NAD-dependent protein deacylase sirtuin-5, mitochondrial {ECO:0000255|HAMAP-Rule:MF_03160} approved|investigational DB02701 Nicotinamide small molecule Q10588 ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 2 illicit|investigational DB02901 Stanolone small molecule P14061 Estradiol 17-beta-dehydrogenase 1 illicit|investigational DB02901 Stanolone small molecule P10275 Androgen receptor illicit|investigational DB02901 Stanolone small molecule P03372 Estrogen receptor illicit|investigational DB02901 Stanolone small molecule P08235 Mineralocorticoid receptor approved DB02925 Piretanide small molecule Q13621 Solute carrier family 12 member 1 approved DB03128 Acetylcholine small molecule P22303 Acetylcholinesterase approved DB03128 Acetylcholine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB03128 Acetylcholine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB03128 Acetylcholine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB03128 Acetylcholine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB03128 Acetylcholine small molecule P36544 Neuronal acetylcholine receptor subunit alpha-7 approved|experimental DB03255 Phenol small molecule P02768 Serum albumin approved|investigational DB03615 Ribostamycin small molecule P07237 Protein disulfide-isomerase approved DB03754 Tromethamine small molecule Q8WVQ1 Soluble calcium-activated nucleotidase 1 approved DB03754 Tromethamine small molecule Q96FI4 Endonuclease 8-like 1 approved DB03754 Tromethamine small molecule P17707 S-adenosylmethionine decarboxylase proenzyme approved DB03754 Tromethamine small molecule P15692 Vascular endothelial growth factor A approved DB03754 Tromethamine small molecule P07585 Decorin withdrawn DB03783 Phenacetin small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB03793 Benzoic Acid small molecule P14920 D-amino-acid oxidase approved|investigational DB03793 Benzoic Acid small molecule P52758 2-iminobutanoate/2-iminopropanoate deaminase {ECO:0000305|PubMed:22094463} approved|investigational DB03793 Benzoic Acid small molecule P51151 Ras-related protein Rab-9A approved|investigational DB03793 Benzoic Acid small molecule P30044 Peroxiredoxin-5, mitochondrial approved|investigational DB03793 Benzoic Acid small molecule P46059 Solute carrier family 15 member 1 experimental|investigational DB04106 Fotemustine small molecule Q16881 Thioredoxin reductase 1, cytoplasmic approved|experimental DB04173 Fructose small molecule P49789 Bis(5'-adenosyl)-triphosphatase approved|investigational DB04209 Dequalinium small molecule P98170 E3 ubiquitin-protein ligase XIAP approved|investigational DB04209 Dequalinium small molecule P29973 cGMP-gated cation channel alpha-1 approved|investigational DB04209 Dequalinium small molecule Q12791 Calcium-activated potassium channel subunit alpha-1 approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule Q96RQ9 L-amino-acid oxidase approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule P14174 Macrophage migration inhibitory factor approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule Q9GZU7 Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule O14964 Hepatocyte growth factor-regulated tyrosine kinase substrate approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule P40926 Malate dehydrogenase, mitochondrial approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule P15086 Carboxypeptidase B approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule P62312 U6 snRNA-associated Sm-like protein LSm6 approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule Q9HB21 Pleckstrin homology domain-containing family A member 1 approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule P07741 Adenine phosphoribosyltransferase approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule Q9BZX2 Uridine-cytidine kinase 2 approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule Q9Y275 Tumor necrosis factor ligand superfamily member 13B approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule Q93088 Betaine--homocysteine S-methyltransferase 1 approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule P15121 Aldose reductase approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule Q9BY32 Inosine triphosphate pyrophosphatase {ECO:0000255|HAMAP-Rule:MF_03148} approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule O75390 Citrate synthase, mitochondrial approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule Q9Y663 Heparan sulfate glucosamine 3-O-sulfotransferase 3A1 approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule O76074 cGMP-specific 3',5'-cyclic phosphodiesterase approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule P12931 Proto-oncogene tyrosine-protein kinase Src approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule P07998 Ribonuclease pancreatic approved|nutraceutical|vet_approved DB04272 Citric Acid small molecule Q14749 Glycine N-methyltransferase approved|investigational DB04335 Inosine small molecule P00491 Purine nucleoside phosphorylase approved|investigational DB04339 Carbocisteine small molecule P09211 Glutathione S-transferase P approved DB04552 Niflumic Acid small molecule P04054 Phospholipase A2 approved DB04552 Niflumic Acid small molecule P35354 Prostaglandin G/H synthase 2 approved DB04552 Niflumic Acid small molecule P23219 Prostaglandin G/H synthase 1 approved DB04552 Niflumic Acid small molecule O60656 UDP-glucuronosyltransferase 1-9 approved|investigational|vet_approved DB04573 Estriol small molecule P03372 Estrogen receptor approved|investigational|vet_approved DB04573 Estriol small molecule Q92731 Estrogen receptor beta approved|investigational|vet_approved DB04573 Estriol small molecule P04278 Sex hormone-binding globulin approved DB04576 Fleroxacin small molecule P11388 DNA topoisomerase 2-alpha experimental DB04599 Aniracetam small molecule P28223 5-hydroxytryptamine receptor 2A experimental DB04599 Aniracetam small molecule P14416 D(2) dopamine receptor experimental DB04599 Aniracetam small molecule P42262 Glutamate receptor 2 experimental DB04599 Aniracetam small molecule P42263 Glutamate receptor 3 experimental|investigational DB04630 Aldosterone small molecule P08235 Mineralocorticoid receptor experimental|investigational DB04630 Aldosterone small molecule P04150 Glucocorticoid receptor experimental|investigational DB04660 Choline alfoscerate small molecule P17900 Ganglioside GM2 activator approved|investigational|withdrawn DB04743 Nimesulide small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational|withdrawn DB04743 Nimesulide small molecule P02788 Lactotransferrin approved|investigational DB04786 Suramin small molecule P41231 P2Y purinoceptor 2 approved|investigational DB04786 Suramin small molecule Q9NXA8 NAD-dependent protein deacylase sirtuin-5, mitochondrial {ECO:0000255|HAMAP-Rule:MF_03160} approved|investigational DB04786 Suramin small molecule P23945 Follicle-stimulating hormone receptor approved|investigational DB04786 Suramin small molecule P21817 Ryanodine receptor 1 approved|investigational DB04786 Suramin small molecule P00734 Prothrombin approved|investigational DB04786 Suramin small molecule P14555 Phospholipase A2, membrane associated approved|investigational|withdrawn DB04817 Metamizole small molecule P23219 Prostaglandin G/H synthase 1 withdrawn DB04820 Nialamide small molecule P27338 Amine oxidase [flavin-containing] B withdrawn DB04820 Nialamide small molecule P21397 Amine oxidase [flavin-containing] A withdrawn DB04820 Nialamide small molecule P21964 Catechol O-methyltransferase withdrawn DB04821 Nomifensine small molecule P23975 Sodium-dependent noradrenaline transporter withdrawn DB04821 Nomifensine small molecule P27338 Amine oxidase [flavin-containing] B withdrawn DB04821 Nomifensine small molecule P21397 Amine oxidase [flavin-containing] A withdrawn DB04821 Nomifensine small molecule P05164 Myeloperoxidase withdrawn DB04821 Nomifensine small molecule P31645 Sodium-dependent serotonin transporter withdrawn DB04821 Nomifensine small molecule Q05940 Synaptic vesicular amine transporter approved|withdrawn DB04824 Phenolphthalein small molecule O60656 UDP-glucuronosyltransferase 1-9 approved|withdrawn DB04824 Phenolphthalein small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|withdrawn DB04824 Phenolphthalein small molecule Q14994 Nuclear receptor subfamily 1 group I member 3 approved|withdrawn DB04824 Phenolphthalein small molecule P03372 Estrogen receptor approved|withdrawn DB04824 Phenolphthalein small molecule P04278 Sex hormone-binding globulin withdrawn DB04825 Prenylamine small molecule Q9H1R3 Myosin light chain kinase 2, skeletal/cardiac muscle withdrawn DB04832 Zimelidine small molecule P31645 Sodium-dependent serotonin transporter withdrawn DB04832 Zimelidine small molecule P27338 Amine oxidase [flavin-containing] B withdrawn DB04832 Zimelidine small molecule P21397 Amine oxidase [flavin-containing] A illicit|withdrawn DB04836 Amineptine small molecule P23975 Sodium-dependent noradrenaline transporter illicit|withdrawn DB04836 Amineptine small molecule P31645 Sodium-dependent serotonin transporter approved|withdrawn DB04837 Clofedanol small molecule P35367 Histamine H1 receptor approved DB04838 Cyclandelate small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved DB04838 Cyclandelate small molecule P23141 Liver carboxylesterase 1 approved|investigational DB04839 Cyproterone acetate small molecule P10275 Androgen receptor approved|investigational DB04839 Cyproterone acetate small molecule P07288 Prostate-specific antigen approved|investigational DB04840 Debrisoquin small molecule P23975 Sodium-dependent noradrenaline transporter approved DB04841 Flunarizine small molecule O43497 Voltage-dependent T-type calcium channel subunit alpha-1G approved DB04841 Flunarizine small molecule O95180 Voltage-dependent T-type calcium channel subunit alpha-1H approved DB04841 Flunarizine small molecule Q9P0X4 Voltage-dependent T-type calcium channel subunit alpha-1I approved DB04841 Flunarizine small molecule P35367 Histamine H1 receptor approved|investigational DB04842 Fluspirilene small molecule P14416 D(2) dopamine receptor approved|investigational DB04842 Fluspirilene small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB04842 Fluspirilene small molecule Q06432 Voltage-dependent calcium channel gamma-1 subunit approved DB04843 Mepenzolate small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB04843 Mepenzolate small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB04844 Tetrabenazine small molecule Q05940 Synaptic vesicular amine transporter approved|investigational DB04844 Tetrabenazine small molecule P14416 D(2) dopamine receptor approved|investigational DB04845 Ixabepilone small molecule Q13509 Tubulin beta-3 chain approved DB04855 Dronedarone small molecule P25100 Alpha-1D adrenergic receptor approved DB04855 Dronedarone small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB04855 Dronedarone small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved DB04855 Dronedarone small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved DB04855 Dronedarone small molecule O60840 Voltage-dependent L-type calcium channel subunit alpha-1F {ECO:0000305} approved DB04855 Dronedarone small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved DB04855 Dronedarone small molecule Q02641 Voltage-dependent L-type calcium channel subunit beta-1 approved DB04855 Dronedarone small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved DB04855 Dronedarone small molecule P54284 Voltage-dependent L-type calcium channel subunit beta-3 approved DB04855 Dronedarone small molecule O00305 Voltage-dependent L-type calcium channel subunit beta-4 {ECO:0000305} approved DB04855 Dronedarone small molecule O95069 Potassium channel subfamily K member 2 approved|investigational DB04865 Omacetaxine mepesuccinate small molecule P39023 60S ribosomal protein L3 approved|investigational DB04868 Nilotinib small molecule P00519 Tyrosine-protein kinase ABL1 approved|investigational DB04868 Nilotinib small molecule P10721 Mast/stem cell growth factor receptor Kit approved DB04871 Lorcaserin small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB04876 Vildagliptin small molecule P27487 Dipeptidyl peptidase 4 approved|investigational DB04878 Voglibose small molecule O43451 Maltase-glucoamylase, intestinal approved|investigational DB04880 Enoximone small molecule Q14432 cGMP-inhibited 3',5'-cyclic phosphodiesterase A investigational DB04884 Dapoxetine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB04894 Vapreotide small molecule P35346 Somatostatin receptor type 5 approved|investigational DB04894 Vapreotide small molecule P25103 Substance-P receptor approved|investigational DB04895 Pegaptanib biotech O14786 Neuropilin-1 approved|investigational DB04896 Milnacipran small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB04896 Milnacipran small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB04896 Milnacipran small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved|investigational|withdrawn DB04898 Ximelagatran small molecule P00734 Prothrombin approved|investigational DB04899 Nesiritide biotech P20594 Atrial natriuretic peptide receptor 2 approved|investigational DB04899 Nesiritide biotech P17342 Atrial natriuretic peptide receptor 3 approved|investigational DB04908 Flibanserin small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB04908 Flibanserin small molecule P21917 D(4) dopamine receptor approved|investigational DB04920 Clevidipine small molecule O60840 Voltage-dependent L-type calcium channel subunit alpha-1F {ECO:0000305} approved|investigational DB04920 Clevidipine small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved|investigational DB04920 Clevidipine small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved|investigational DB04920 Clevidipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C investigational DB04924 Itopride small molecule P14416 D(2) dopamine receptor investigational DB04924 Itopride small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational DB04930 Permethrin small molecule P03372 Estrogen receptor approved|investigational DB04930 Permethrin small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB04931 Afamelanotide small molecule Q01726 Melanocyte-stimulating hormone receptor approved|investigational DB04932 Defibrotide biotech P30542 Adenosine receptor A1 approved|investigational DB04932 Defibrotide biotech P29275 Adenosine receptor A2b approved|investigational DB04938 Ospemifene small molecule P03372 Estrogen receptor approved DB04946 Iloperidone small molecule P28223 5-hydroxytryptamine receptor 2A approved DB04946 Iloperidone small molecule P14416 D(2) dopamine receptor approved DB04946 Iloperidone small molecule P35462 D(3) dopamine receptor approved DB04946 Iloperidone small molecule P21917 D(4) dopamine receptor approved DB04946 Iloperidone small molecule P34969 5-hydroxytryptamine receptor 7 approved DB04946 Iloperidone small molecule P35367 Histamine H1 receptor approved|investigational DB04951 Pirfenidone small molecule P09958 Furin approved|investigational DB04953 Ezogabine small molecule O43526 Potassium voltage-gated channel subfamily KQT member 2 {ECO:0000305} approved|investigational DB04953 Ezogabine small molecule O43525 Potassium voltage-gated channel subfamily KQT member 3 {ECO:0000305} approved|investigational DB04953 Ezogabine small molecule P56696 Potassium voltage-gated channel subfamily KQT member 4 approved|investigational DB04953 Ezogabine small molecule Q9NR82 Potassium voltage-gated channel subfamily KQT member 5 investigational DB04956 Afelimomab biotech P01375 Tumor necrosis factor approved DB05013 Ingenol Mebutate small molecule Q05655 Protein kinase C delta type approved DB05013 Ingenol Mebutate small molecule P17252 Protein kinase C alpha type approved|investigational DB05015 Belinostat small molecule Q13547 Histone deacetylase 1 approved|investigational DB05099 Ancrod small molecule P02671 Fibrinogen alpha chain investigational DB05168 Vintafolide small molecule P41439 Folate receptor gamma investigational DB05168 Vintafolide small molecule P15328 Folate receptor alpha approved DB05246 Methsuximide small molecule O43497 Voltage-dependent T-type calcium channel subunit alpha-1G investigational DB05254 Fibrinolysin biotech P05121 Plasminogen activator inhibitor 1 investigational DB05254 Fibrinolysin biotech P00749 Urokinase-type plasminogen activator approved|investigational DB05259 Glatiramer Acetate biotech P04229 HLA class II histocompatibility antigen, DRB1-1 beta chain approved|investigational DB05266 Ibudilast small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved|investigational DB05266 Ibudilast small molecule Q07343 cAMP-specific 3',5'-cyclic phosphodiesterase 4B approved|investigational DB05266 Ibudilast small molecule Q08493 cAMP-specific 3',5'-cyclic phosphodiesterase 4C approved|investigational DB05266 Ibudilast small molecule Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D approved|investigational DB05266 Ibudilast small molecule Q14432 cGMP-inhibited 3',5'-cyclic phosphodiesterase A approved DB05271 Rotigotine small molecule P35462 D(3) dopamine receptor approved DB05271 Rotigotine small molecule P21917 D(4) dopamine receptor approved DB05271 Rotigotine small molecule P14416 D(2) dopamine receptor approved DB05294 Vandetanib small molecule P15692 Vascular endothelial growth factor A approved DB05294 Vandetanib small molecule P00533 Epidermal growth factor receptor approved DB05294 Vandetanib small molecule Q13882 Protein-tyrosine kinase 6 approved DB05294 Vandetanib small molecule Q02763 Angiopoietin-1 receptor approved DB05294 Vandetanib small molecule P07949 Proto-oncogene tyrosine-protein kinase receptor Ret {ECO:0000305} approved DB05332 Romiplostim biotech P40238 Thrombopoietin receptor approved|investigational DB05351 Dexlansoprazole small molecule P20648 Potassium-transporting ATPase alpha chain 1 approved|investigational DB05351 Dexlansoprazole small molecule P51164 Potassium-transporting ATPase subunit beta approved|investigational DB05381 Histamine small molecule P35367 Histamine H1 receptor approved|investigational DB05381 Histamine small molecule P25021 Histamine H2 receptor approved|investigational DB05381 Histamine small molecule Q9Y5N1 Histamine H3 receptor approved|investigational DB05381 Histamine small molecule Q9H3N8 Histamine H4 receptor approved|investigational DB05381 Histamine small molecule Q05940 Synaptic vesicular amine transporter approved|withdrawn DB05521 Telaprevir small molecule Q9Y6L6 Solute carrier organic anion transporter family member 1B1 approved|withdrawn DB05521 Telaprevir small molecule O94956 Solute carrier organic anion transporter family member 2B1 approved|investigational DB05541 Brivaracetam small molecule Q7L0J3 Synaptic vesicle glycoprotein 2A approved|investigational DB05630 Sodium stibogluconate small molecule P11387 DNA topoisomerase 1 approved|investigational DB05676 Apremilast small molecule Q08499 cAMP-specific 3',5'-cyclic phosphodiesterase 4D approved|investigational DB05676 Apremilast small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved|investigational DB05676 Apremilast small molecule Q07343 cAMP-specific 3',5'-cyclic phosphodiesterase 4B approved|investigational DB05676 Apremilast small molecule P01375 Tumor necrosis factor approved|investigational DB05676 Apremilast small molecule P60568 Interleukin-2 approved|investigational DB05676 Apremilast small molecule P01579 Interferon gamma approved|investigational DB05676 Apremilast small molecule P29474 Nitric oxide synthase, endothelial approved|investigational DB05773 Trastuzumab emtansine biotech P04626 Receptor tyrosine-protein kinase erbB-2 approved DB05812 Abiraterone small molecule P05093 Steroid 17-alpha-hydroxylase/17,20 lyase approved|investigational DB05829 Parathyroid hormone biotech P49190 Parathyroid hormone 2 receptor approved|investigational DB06016 Cariprazine small molecule P35462 D(3) dopamine receptor approved|investigational DB06016 Cariprazine small molecule P14416 D(2) dopamine receptor approved|investigational DB06016 Cariprazine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB06016 Cariprazine small molecule P35367 Histamine H1 receptor approved|investigational|withdrawn DB06144 Sertindole small molecule P14416 D(2) dopamine receptor approved|investigational|withdrawn DB06144 Sertindole small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational|withdrawn DB06144 Sertindole small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational|withdrawn DB06144 Sertindole small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational|withdrawn DB06144 Sertindole small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB06148 Mianserin small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB06148 Mianserin small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB06148 Mianserin small molecule P35367 Histamine H1 receptor approved|investigational DB06148 Mianserin small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB06148 Mianserin small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB06148 Mianserin small molecule Q9H3N8 Histamine H4 receptor approved|investigational DB06148 Mianserin small molecule P35462 D(3) dopamine receptor approved|investigational DB06148 Mianserin small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational DB06148 Mianserin small molecule P14416 D(2) dopamine receptor approved|investigational DB06151 Acetylcysteine small molecule P48637 Glutathione synthetase approved|investigational DB06151 Acetylcysteine small molecule Q03154 Aminoacylase-1 approved|investigational DB06151 Acetylcysteine small molecule O14920 Inhibitor of nuclear factor kappa-B kinase subunit beta approved|investigational DB06151 Acetylcysteine small molecule O15111 Inhibitor of nuclear factor kappa-B kinase subunit alpha approved|investigational DB06151 Acetylcysteine small molecule Q13224 Glutamate receptor ionotropic, NMDA 2B approved|investigational DB06151 Acetylcysteine small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved|investigational DB06151 Acetylcysteine small molecule Q12879 Glutamate receptor ionotropic, NMDA 2A approved|investigational DB06151 Acetylcysteine small molecule O15399 Glutamate receptor ionotropic, NMDA 2D approved|investigational DB06168 Canakinumab biotech P01584 Interleukin-1 beta investigational DB06174 Noscapine small molecule Q99720 Sigma non-opioid intracellular receptor 1 approved|investigational DB06176 Romidepsin small molecule Q13547 Histone deacetylase 1 approved|investigational DB06176 Romidepsin small molecule Q92769 Histone deacetylase 2 approved|investigational DB06176 Romidepsin small molecule P56524 Histone deacetylase 4 approved|investigational DB06176 Romidepsin small molecule Q9UBN7 Histone deacetylase 6 approved|investigational DB06176 Romidepsin small molecule P33527 Multidrug resistance-associated protein 1 approved DB06186 Ipilimumab biotech P16410 Cytotoxic T-lymphocyte protein 4 approved|investigational DB06196 Icatibant small molecule P30411 B2 bradykinin receptor approved|investigational DB06196 Icatibant small molecule P15144 Aminopeptidase N {ECO:0000305} approved DB06201 Rufinamide small molecule P41594 Metabotropic glutamate receptor 5 approved DB06201 Rufinamide small molecule Q15858 Sodium channel protein type 9 subunit alpha {ECO:0000305} approved|investigational DB06202 Lasofoxifene small molecule P03372 Estrogen receptor approved|investigational DB06202 Lasofoxifene small molecule Q92731 Estrogen receptor beta approved|investigational DB06202 Lasofoxifene small molecule P34972 Cannabinoid receptor 2 approved DB06203 Alogliptin small molecule P27487 Dipeptidyl peptidase 4 approved DB06204 Tapentadol small molecule P35372 Mu-type opioid receptor approved DB06204 Tapentadol small molecule P23975 Sodium-dependent noradrenaline transporter approved DB06204 Tapentadol small molecule P41143 Delta-type opioid receptor approved DB06204 Tapentadol small molecule P31645 Sodium-dependent serotonin transporter approved DB06207 Silodosin small molecule P25100 Alpha-1D adrenergic receptor approved DB06209 Prasugrel small molecule Q9H244 P2Y purinoceptor 12 approved DB06210 Eltrombopag small molecule P40238 Thrombopoietin receptor approved DB06216 Asenapine small molecule P14416 D(2) dopamine receptor approved DB06216 Asenapine small molecule P28223 5-hydroxytryptamine receptor 2A approved DB06216 Asenapine small molecule P28335 5-hydroxytryptamine receptor 2C approved DB06216 Asenapine small molecule P34969 5-hydroxytryptamine receptor 7 approved DB06216 Asenapine small molecule P35462 D(3) dopamine receptor approved DB06216 Asenapine small molecule P21917 D(4) dopamine receptor approved DB06216 Asenapine small molecule P35367 Histamine H1 receptor approved DB06216 Asenapine small molecule P25021 Histamine H2 receptor approved|investigational DB06217 Vernakalant small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|investigational DB06217 Vernakalant small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved DB06218 Lacosamide small molecule Q15858 Sodium channel protein type 9 subunit alpha {ECO:0000305} approved DB06218 Lacosamide small molecule Q9NY46 Sodium channel protein type 3 subunit alpha approved DB06228 Rivaroxaban small molecule P00742 Coagulation factor X approved|investigational|withdrawn DB06230 Nalmefene small molecule P35372 Mu-type opioid receptor approved|investigational|withdrawn DB06230 Nalmefene small molecule P41143 Delta-type opioid receptor investigational DB06233 Ridaforolimus small molecule P42345 Serine/threonine-protein kinase mTOR approved DB06237 Avanafil small molecule O76074 cGMP-specific 3',5'-cyclic phosphodiesterase approved|withdrawn DB06243 Eflornithine small molecule P11926 Ornithine decarboxylase approved|investigational DB06262 Droxidopa small molecule P25100 Alpha-1D adrenergic receptor approved|investigational DB06262 Droxidopa small molecule P13945 Beta-3 adrenergic receptor approved|investigational DB06262 Droxidopa small molecule P00439 Phenylalanine-4-hydroxylase approved|investigational DB06263 Amrubicin small molecule P11388 DNA topoisomerase 2-alpha investigational DB06266 Lonidamine small molecule P13569 Cystic fibrosis transmembrane conductance regulator investigational DB06266 Lonidamine small molecule P19367 Hexokinase-1 approved|investigational DB06267 Udenafil small molecule O76074 cGMP-specific 3',5'-cyclic phosphodiesterase approved|investigational|withdrawn DB06268 Sitaxentan small molecule P25101 Endothelin-1 receptor {ECO:0000305} approved|investigational|withdrawn DB06268 Sitaxentan small molecule P24530 Endothelin receptor type B {ECO:0000305} approved|investigational DB06271 Sulodexide biotech P05546 Heparin cofactor 2 approved|investigational DB06271 Sulodexide biotech P01008 Antithrombin-III approved DB06273 Tocilizumab biotech P08887 Interleukin-6 receptor subunit alpha approved|investigational DB06274 Alvimopan small molecule P35372 Mu-type opioid receptor approved|investigational DB06274 Alvimopan small molecule P41143 Delta-type opioid receptor approved DB06282 Levocetirizine small molecule P35367 Histamine H1 receptor approved DB06287 Temsirolimus small molecule P42345 Serine/threonine-protein kinase mTOR approved|investigational DB06288 Amisulpride small molecule P14416 D(2) dopamine receptor approved|investigational DB06288 Amisulpride small molecule P35462 D(3) dopamine receptor approved|investigational DB06288 Amisulpride small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational DB06288 Amisulpride small molecule P28223 5-hydroxytryptamine receptor 2A approved DB06292 Dapagliflozin small molecule P31639 Sodium/glucose cotransporter 2 approved DB06335 Saxagliptin small molecule P27487 Dipeptidyl peptidase 4 investigational DB06358 Iclaprim small molecule P00374 Dihydrofolate reductase approved DB06366 Pertuzumab biotech P04626 Receptor tyrosine-protein kinase erbB-2 approved|investigational DB06372 Rilonacept biotech P01584 Interleukin-1 beta approved|investigational DB06372 Rilonacept biotech P01583 Interleukin-1 alpha approved|investigational DB06372 Rilonacept biotech P18510 Interleukin-1 receptor antagonist protein approved|investigational DB06401 Bazedoxifene small molecule P03372 Estrogen receptor approved|investigational DB06401 Bazedoxifene small molecule Q92731 Estrogen receptor beta approved|investigational DB06403 Ambrisentan small molecule P25101 Endothelin-1 receptor {ECO:0000305} approved|investigational DB06403 Ambrisentan small molecule P24530 Endothelin receptor type B {ECO:0000305} approved DB06404 Human C1-esterase inhibitor biotech P09871 Complement C1s subcomponent approved DB06404 Human C1-esterase inhibitor biotech P00748 Coagulation factor XII approved DB06404 Human C1-esterase inhibitor biotech P00734 Prothrombin approved DB06404 Human C1-esterase inhibitor biotech P03951 Coagulation factor XI approved DB06404 Human C1-esterase inhibitor biotech P00750 Tissue-type plasminogen activator approved DB06410 Doxercalciferol small molecule P11473 Vitamin D3 receptor approved|illicit DB06412 Oxymetholone small molecule P10275 Androgen receptor approved DB06441 Cangrelor small molecule Q9H244 P2Y purinoceptor 12 investigational DB06470 clomethiazole small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 investigational DB06479 Propentofylline small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved DB06480 Prucalopride small molecule Q13639 5-hydroxytryptamine receptor 4 approved DB06589 Pazopanib small molecule P17948 Vascular endothelial growth factor receptor 1 approved DB06589 Pazopanib small molecule P35916 Vascular endothelial growth factor receptor 3 approved DB06589 Pazopanib small molecule P16234 Platelet-derived growth factor receptor alpha approved DB06589 Pazopanib small molecule P09619 Platelet-derived growth factor receptor beta approved DB06589 Pazopanib small molecule P10721 Mast/stem cell growth factor receptor Kit approved DB06589 Pazopanib small molecule P22607 Fibroblast growth factor receptor 3 approved DB06589 Pazopanib small molecule Q08881 Tyrosine-protein kinase ITK/TSK approved DB06589 Pazopanib small molecule P05230 Fibroblast growth factor 1 approved DB06589 Pazopanib small molecule Q9UQQ2 SH2B adapter protein 3 approved|investigational DB06594 Agomelatine small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB06602 Reslizumab biotech P05113 Interleukin-5 approved|investigational DB06603 Panobinostat small molecule Q13547 Histone deacetylase 1 approved DB06605 Apixaban small molecule P00742 Coagulation factor X approved|investigational|withdrawn DB06607 Catumaxomab biotech P16422 Epithelial cell adhesion molecule approved|investigational|withdrawn DB06607 Catumaxomab biotech P12318 Low affinity immunoglobulin gamma Fc region receptor II-a approved|investigational|withdrawn DB06607 Catumaxomab biotech P08637 Low affinity immunoglobulin gamma Fc region receptor III-A approved|investigational|withdrawn DB06607 Catumaxomab biotech O75015 Low affinity immunoglobulin gamma Fc region receptor III-B approved|investigational|withdrawn DB06607 Catumaxomab biotech P07766 T-cell surface glycoprotein CD3 epsilon chain approved|investigational DB06612 Mepolizumab biotech P05113 Interleukin-5 approved DB06616 Bosutinib small molecule P11274 Breakpoint cluster region protein approved DB06616 Bosutinib small molecule P00519 Tyrosine-protein kinase ABL1 approved DB06616 Bosutinib small molecule P07948 Tyrosine-protein kinase Lyn approved DB06616 Bosutinib small molecule P08631 Tyrosine-protein kinase HCK approved DB06616 Bosutinib small molecule P12931 Proto-oncogene tyrosine-protein kinase Src approved DB06616 Bosutinib small molecule P24941 Cyclin-dependent kinase 2 approved DB06616 Bosutinib small molecule Q02750 Dual specificity mitogen-activated protein kinase kinase 1 approved DB06616 Bosutinib small molecule P36507 Dual specificity mitogen-activated protein kinase kinase 2 approved DB06616 Bosutinib small molecule Q9Y2U5 Mitogen-activated protein kinase kinase kinase 2 approved DB06616 Bosutinib small molecule Q13555 Calcium/calmodulin-dependent protein kinase type II subunit gamma approved|investigational DB06626 Axitinib small molecule P17948 Vascular endothelial growth factor receptor 1 approved|investigational DB06626 Axitinib small molecule P35916 Vascular endothelial growth factor receptor 3 investigational DB06634 Casopitant small molecule P08684 Cytochrome P450 3A4 investigational DB06634 Casopitant small molecule P25103 Substance-P receptor approved DB06637 Dalfampridine small molecule Q09470 Potassium voltage-gated channel subfamily A member 1 approved DB06637 Dalfampridine small molecule P17658 Potassium voltage-gated channel subfamily A member 6 approved DB06637 Dalfampridine small molecule Q14721 Potassium voltage-gated channel subfamily B member 1 {ECO:0000312|HGNC:HGNC:6231} approved DB06637 Dalfampridine small molecule Q92953 Potassium voltage-gated channel subfamily B member 2 {ECO:0000312|HGNC:HGNC:6232} approved DB06637 Dalfampridine small molecule P48547 Potassium voltage-gated channel subfamily C member 1 approved DB06637 Dalfampridine small molecule Q96PR1 Potassium voltage-gated channel subfamily C member 2 {ECO:0000312|HGNC:HGNC:6234} approved DB06637 Dalfampridine small molecule Q14003 Potassium voltage-gated channel subfamily C member 3 approved DB06637 Dalfampridine small molecule Q9NZV8 Potassium voltage-gated channel subfamily D member 2 approved DB06643 Denosumab biotech O14788 Tumor necrosis factor ligand superfamily member 11 approved DB06650 Ofatumumab biotech P11836 B-lymphocyte antigen CD20 approved DB06663 Pasireotide small molecule P32745 Somatostatin receptor type 3 approved DB06663 Pasireotide small molecule P35346 Somatostatin receptor type 5 approved DB06674 Golimumab biotech P01375 Tumor necrosis factor approved|investigational DB06681 Belatacept biotech P42081 T-lymphocyte activation antigen CD86 approved|investigational DB06681 Belatacept biotech P33681 T-lymphocyte activation antigen CD80 approved|investigational DB06688 Sipuleucel-T biotech P15309 Prostatic acid phosphatase approved DB06689 Ethanolamine Oleate small molecule P00748 Coagulation factor XII approved|vet_approved DB06691 Mepyramine small molecule P35367 Histamine H1 receptor approved|investigational|withdrawn DB06692 Aprotinin biotech P07477 Trypsin-1 approved|investigational|withdrawn DB06692 Aprotinin biotech P00747 Plasminogen approved|investigational|withdrawn DB06692 Aprotinin biotech P06870 Kallikrein-1 approved|investigational DB06694 Xylometazoline small molecule P25100 Alpha-1D adrenergic receptor approved DB06695 Dabigatran etexilate small molecule P00734 Prothrombin approved|investigational DB06698 Betahistine small molecule P35367 Histamine H1 receptor approved|investigational DB06698 Betahistine small molecule Q9Y5N1 Histamine H3 receptor approved|investigational DB06700 Desvenlafaxine small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB06700 Desvenlafaxine small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB06701 Dexmethylphenidate small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational DB06701 Dexmethylphenidate small molecule P31645 Sodium-dependent serotonin transporter approved DB06702 Fesoterodine small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB06702 Fesoterodine small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB06702 Fesoterodine small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB06702 Fesoterodine small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB06706 Isometheptene small molecule Q05940 Synaptic vesicular amine transporter approved DB06710 Methyltestosterone small molecule P10275 Androgen receptor approved DB06710 Methyltestosterone small molecule P03372 Estrogen receptor approved|investigational DB06712 Nilvadipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB06712 Nilvadipine small molecule P54289 Voltage-dependent calcium channel subunit alpha-2/delta-1 approved|investigational DB06712 Nilvadipine small molecule Q08289 Voltage-dependent L-type calcium channel subunit beta-2 approved|investigational DB06712 Nilvadipine small molecule Q01668 Voltage-dependent L-type calcium channel subunit alpha-1D approved|investigational DB06712 Nilvadipine small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved|investigational DB06712 Nilvadipine small molecule Q8IZS8 Voltage-dependent calcium channel subunit alpha-2/delta-3 approved|investigational DB06713 Norelgestromin small molecule P06401 Progesterone receptor approved|investigational DB06713 Norelgestromin small molecule P02768 Serum albumin approved|investigational DB06713 Norelgestromin small molecule P10275 Androgen receptor approved|investigational DB06719 Buserelin biotech P22888 Lutropin-choriogonadotropic hormone receptor approved|investigational DB06720 Velaglucerase alfa biotech P04062 Glucosylceramidase approved|investigational DB06725 Lornoxicam small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB06725 Lornoxicam small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB06736 Aceclofenac small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB06736 Aceclofenac small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB06738 Ketobemidone small molecule P35372 Mu-type opioid receptor approved|investigational DB06738 Ketobemidone small molecule P41143 Delta-type opioid receptor approved|investigational DB06738 Ketobemidone small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved DB06739 Seratrodast small molecule P21731 Thromboxane A2 receptor approved|investigational DB06751 Drotaverine small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved|investigational DB06751 Drotaverine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|nutraceutical DB06756 Glycine betaine small molecule P10415 Apoptosis regulator Bcl-2 approved DB06766 Alcaftadine small molecule P35367 Histamine H1 receptor approved DB06772 Cabazitaxel small molecule P68366 Tubulin alpha-4A chain approved|investigational DB06773 Human calcitonin biotech P12814 Alpha-actinin-1 approved DB06774 Capsaicin small molecule Q8NER1 Transient receptor potential cation channel subfamily V member 1 approved DB06774 Capsaicin small molecule Q99623 Prohibitin-2 approved DB06775 Carglumic Acid small molecule P31327 Carbamoyl-phosphate synthase [ammonia], mitochondrial approved DB06777 Chenodeoxycholic acid small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB06777 Chenodeoxycholic acid small molecule P52895 Aldo-keto reductase family 1 member C2 approved DB06779 Dalteparin small molecule P01008 Antithrombin-III approved DB06779 Dalteparin small molecule P15692 Vascular endothelial growth factor A approved DB06779 Dalteparin small molecule P10646 Tissue factor pathway inhibitor approved DB06779 Dalteparin small molecule P16109 P-selectin approved DB06781 Difluprednate small molecule P04150 Glucocorticoid receptor approved DB06782 Dimercaprol small molecule P05067 Amyloid-beta A4 protein approved|investigational|withdrawn DB06786 Halcinonide small molecule Q99835 Smoothened homolog approved DB06787 Hexocyclium small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB06787 Hexocyclium small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB06787 Hexocyclium small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB06787 Hexocyclium small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB06789 Hydroxyprogesterone caproate small molecule P06401 Progesterone receptor approved DB06791 Lanreotide small molecule P35346 Somatostatin receptor type 5 approved|vet_approved DB06795 Mafenide small molecule P23280 Carbonic anhydrase 6 approved DB06800 Methylnaltrexone small molecule P35372 Mu-type opioid receptor approved|investigational DB06802 Nepafenac small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB06802 Nepafenac small molecule P35354 Prostaglandin G/H synthase 2 approved DB06809 Plerixafor small molecule P61073 C-X-C chemokine receptor type 4 approved|investigational DB06813 Pralatrexate small molecule P00374 Dihydrofolate reductase approved|investigational DB06813 Pralatrexate small molecule P04818 Thymidylate synthase approved DB06822 Tinzaparin small molecule P01008 Antithrombin-III approved DB06822 Tinzaparin small molecule P13612 Integrin alpha-4 approved DB06822 Tinzaparin small molecule P48061 Stromal cell-derived factor 1 experimental DB07477 Felbinac small molecule P07711 Cathepsin L1 experimental DB07637 Dibromotyrosine small molecule P19235 Erythropoietin receptor experimental DB08329 Sulthiame small molecule P00918 Carbonic anhydrase 2 approved DB08439 Parecoxib small molecule P35354 Prostaglandin G/H synthase 2 approved DB08439 Parecoxib small molecule P02788 Lactotransferrin investigational DB08486 Efaproxiral small molecule P69905 Hemoglobin subunit alpha investigational DB08486 Efaproxiral small molecule P68871 Hemoglobin subunit beta approved|investigational DB08604 Triclosan small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved|investigational DB08604 Triclosan small molecule P10275 Androgen receptor approved|investigational DB08604 Triclosan small molecule Q14994 Nuclear receptor subfamily 1 group I member 3 approved|investigational DB08604 Triclosan small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|investigational DB08604 Triclosan small molecule P07202 Thyroid peroxidase {ECO:0000305} approved DB08799 Antazoline small molecule P35367 Histamine H1 receptor approved DB08800 Chloropyramine small molecule P35367 Histamine H1 receptor approved|investigational DB08801 Dimetindene small molecule P35367 Histamine H1 receptor approved|investigational DB08801 Dimetindene small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB08802 Isothipendyl small molecule P35367 Histamine H1 receptor approved|investigational DB08806 Roxatidine acetate small molecule P25021 Histamine H2 receptor approved DB08807 Bopindolol small molecule P13945 Beta-3 adrenergic receptor approved DB08808 Bupranolol small molecule P13945 Beta-3 adrenergic receptor approved DB08811 Tofisopam small molecule P27815 cAMP-specific 3',5'-cyclic phosphodiesterase 4A approved DB08811 Tofisopam small molecule Q9Y233 cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A approved DB08811 Tofisopam small molecule Q14432 cGMP-inhibited 3',5'-cyclic phosphodiesterase A approved DB08811 Tofisopam small molecule O00408 cGMP-dependent 3',5'-cyclic phosphodiesterase approved|investigational DB08813 Nadroparin small molecule P01008 Antithrombin-III approved|investigational DB08813 Nadroparin small molecule P16109 P-selectin approved|investigational DB08813 Nadroparin small molecule P01100 Proto-oncogene c-Fos approved|investigational DB08813 Nadroparin small molecule P01106 Myc proto-oncogene protein approved|investigational DB08814 Triflusal small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB08814 Triflusal small molecule P19838 Nuclear factor NF-kappa-B p105 subunit approved|investigational DB08814 Triflusal small molecule P35228 Nitric oxide synthase, inducible approved|investigational DB08814 Triflusal small molecule Q9Y233 cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A approved|investigational DB08815 Lurasidone small molecule P14416 D(2) dopamine receptor approved|investigational DB08815 Lurasidone small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB08815 Lurasidone small molecule P34969 5-hydroxytryptamine receptor 7 approved DB08816 Ticagrelor small molecule Q9H244 P2Y purinoceptor 12 approved|vet_approved DB08818 Hyaluronic acid small molecule P16070 CD44 antigen approved|vet_approved DB08818 Hyaluronic acid small molecule P05362 Intercellular adhesion molecule 1 approved|vet_approved DB08818 Hyaluronic acid small molecule O75330 Hyaluronan mediated motility receptor approved|vet_approved DB08818 Hyaluronic acid small molecule O14594 Neurocan core protein approved|vet_approved DB08818 Hyaluronic acid small molecule P13611 Versican core protein approved|vet_approved DB08818 Hyaluronic acid small molecule Q07021 Complement component 1 Q subcomponent-binding protein, mitochondrial approved|vet_approved DB08818 Hyaluronic acid small molecule P10915 Hyaluronan and proteoglycan link protein 1 approved|vet_approved DB08818 Hyaluronic acid small molecule Q96S86 Hyaluronan and proteoglycan link protein 3 approved|vet_approved DB08818 Hyaluronic acid small molecule Q86UW8 Hyaluronan and proteoglycan link protein 4 approved|vet_approved DB08818 Hyaluronic acid small molecule Q14520 Hyaluronan-binding protein 2 approved|vet_approved DB08818 Hyaluronic acid small molecule Q6UX15 Layilin approved|vet_approved DB08818 Hyaluronic acid small molecule Q8WWQ8 Stabilin-2 approved|vet_approved DB08818 Hyaluronic acid small molecule P98066 Tumor necrosis factor-inducible gene 6 protein approved|vet_approved DB08818 Hyaluronic acid small molecule Q9BZV3 Interphotoreceptor matrix proteoglycan 2 approved|vet_approved DB08818 Hyaluronic acid small molecule Q5JVS0 Intracellular hyaluronan-binding protein 4 {ECO:0000303|PubMed:10887182} approved DB08819 Tafluprost small molecule P43088 Prostaglandin F2-alpha receptor approved DB08820 Ivacaftor small molecule P13569 Cystic fibrosis transmembrane conductance regulator approved|investigational DB08822 Azilsartan medoxomil small molecule P30556 Type-1 angiotensin II receptor approved|investigational DB08828 Vismodegib small molecule Q99835 Smoothened homolog approved DB08835 Spaglumic Acid small molecule Q04609 Glutamate carboxypeptidase 2 experimental|investigational DB08836 Temocapril small molecule P12821 Angiotensin-converting enzyme approved DB08860 Pitavastatin small molecule P04035 3-hydroxy-3-methylglutaryl-coenzyme A reductase approved|investigational DB08862 Cholecystokinin small molecule P32238 Cholecystokinin receptor type A approved|investigational DB08862 Cholecystokinin small molecule P04049 RAF proto-oncogene serine/threonine-protein kinase approved|investigational DB08862 Cholecystokinin small molecule P27361 Mitogen-activated protein kinase 3 approved|investigational DB08862 Cholecystokinin small molecule P01133 Pro-epidermal growth factor approved|investigational DB08862 Cholecystokinin small molecule P05771 Protein kinase C beta type approved DB08864 Rilpivirine small molecule O75469 Nuclear receptor subfamily 1 group I member 2 approved DB08865 Crizotinib small molecule Q9UM73 ALK tyrosine kinase receptor approved DB08865 Crizotinib small molecule P08581 Hepatocyte growth factor receptor approved DB08867 Ulipristal small molecule P06401 Progesterone receptor approved DB08867 Ulipristal small molecule P04150 Glucocorticoid receptor approved DB08867 Ulipristal small molecule P10275 Androgen receptor approved|investigational DB08868 Fingolimod small molecule Q9H228 Sphingosine 1-phosphate receptor 5 approved|investigational DB08868 Fingolimod small molecule Q13547 Histone deacetylase 1 approved|investigational DB08869 Tesamorelin small molecule Q02643 Growth hormone-releasing hormone receptor approved|investigational DB08870 Brentuximab vedotin biotech P28908 Tumor necrosis factor receptor superfamily member 8 {ECO:0000312|HGNC:HGNC:11923} approved|investigational DB08871 Eribulin small molecule P10415 Apoptosis regulator Bcl-2 approved|investigational DB08875 Cabozantinib small molecule P08581 Hepatocyte growth factor receptor approved|investigational DB08875 Cabozantinib small molecule P07949 Proto-oncogene tyrosine-protein kinase receptor Ret {ECO:0000305} approved DB08877 Ruxolitinib small molecule P23458 Tyrosine-protein kinase JAK1 approved DB08877 Ruxolitinib small molecule O60674 Tyrosine-protein kinase JAK2 approved DB08879 Belimumab biotech Q9Y275 Tumor necrosis factor ligand superfamily member 13B approved DB08880 Teriflunomide small molecule Q02127 Dihydroorotate dehydrogenase (quinone), mitochondrial approved DB08881 Vemurafenib small molecule P15056 Serine/threonine-protein kinase B-raf approved DB08882 Linagliptin small molecule P27487 Dipeptidyl peptidase 4 approved DB08883 Perampanel small molecule P42261 Glutamate receptor 1 approved DB08885 Aflibercept biotech P15692 Vascular endothelial growth factor A approved DB08885 Aflibercept biotech P49765 Vascular endothelial growth factor B approved DB08888 Ocriplasmin biotech P02751 Fibronectin approved DB08888 Ocriplasmin biotech P01023 Alpha-2-macroglobulin approved DB08888 Ocriplasmin biotech P08697 Alpha-2-antiplasmin approved|investigational DB08889 Carfilzomib small molecule P28074 Proteasome subunit beta type-5 approved|investigational DB08889 Carfilzomib small molecule P28062 Proteasome subunit beta type-8 approved|investigational DB08889 Carfilzomib small molecule P20618 Proteasome subunit beta type-1 approved|investigational DB08889 Carfilzomib small molecule P49721 Proteasome subunit beta type-2 approved|investigational DB08889 Carfilzomib small molecule P40306 Proteasome subunit beta type-10 approved DB08890 Linaclotide small molecule P25092 Heat-stable enterotoxin receptor approved DB08893 Mirabegron small molecule P13945 Beta-3 adrenergic receptor approved|investigational DB08894 Peginesatide biotech P19235 Erythropoietin receptor approved|investigational DB08895 Tofacitinib small molecule P23458 Tyrosine-protein kinase JAK1 approved|investigational DB08895 Tofacitinib small molecule O60674 Tyrosine-protein kinase JAK2 approved|investigational DB08895 Tofacitinib small molecule P52333 Tyrosine-protein kinase JAK3 approved|investigational DB08895 Tofacitinib small molecule P29597 Non-receptor tyrosine-protein kinase TYK2 approved DB08896 Regorafenib small molecule P17948 Vascular endothelial growth factor receptor 1 approved DB08896 Regorafenib small molecule P35916 Vascular endothelial growth factor receptor 3 approved DB08896 Regorafenib small molecule P10721 Mast/stem cell growth factor receptor Kit approved DB08896 Regorafenib small molecule P16234 Platelet-derived growth factor receptor alpha approved DB08896 Regorafenib small molecule P09619 Platelet-derived growth factor receptor beta approved DB08896 Regorafenib small molecule P11362 Fibroblast growth factor receptor 1 approved DB08896 Regorafenib small molecule P21802 Fibroblast growth factor receptor 2 approved DB08896 Regorafenib small molecule Q02763 Angiopoietin-1 receptor approved DB08896 Regorafenib small molecule Q16832 Discoidin domain-containing receptor 2 approved DB08896 Regorafenib small molecule P04629 High affinity nerve growth factor receptor approved DB08896 Regorafenib small molecule P29317 Ephrin type-A receptor 2 approved DB08896 Regorafenib small molecule P04049 RAF proto-oncogene serine/threonine-protein kinase approved DB08896 Regorafenib small molecule P15056 Serine/threonine-protein kinase B-raf approved DB08896 Regorafenib small molecule Q15759 Mitogen-activated protein kinase 11 approved DB08896 Regorafenib small molecule P42685 Tyrosine-protein kinase FRK approved DB08896 Regorafenib small molecule P00519 Tyrosine-protein kinase ABL1 approved DB08896 Regorafenib small molecule P07949 Proto-oncogene tyrosine-protein kinase receptor Ret {ECO:0000305} approved DB08897 Aclidinium small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB08897 Aclidinium small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB08897 Aclidinium small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB08897 Aclidinium small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB08899 Enzalutamide small molecule P10275 Androgen receptor approved DB08900 Teduglutide biotech O95838 Glucagon-like peptide 2 receptor approved|investigational DB08901 Ponatinib small molecule P00519 Tyrosine-protein kinase ABL1 approved|investigational DB08901 Ponatinib small molecule P11274 Breakpoint cluster region protein approved|investigational DB08901 Ponatinib small molecule P10721 Mast/stem cell growth factor receptor Kit approved|investigational DB08901 Ponatinib small molecule P07949 Proto-oncogene tyrosine-protein kinase receptor Ret {ECO:0000305} approved|investigational DB08901 Ponatinib small molecule Q02763 Angiopoietin-1 receptor approved|investigational DB08901 Ponatinib small molecule P36888 Receptor-type tyrosine-protein kinase FLT3 approved|investigational DB08901 Ponatinib small molecule P11362 Fibroblast growth factor receptor 1 approved|investigational DB08901 Ponatinib small molecule P21802 Fibroblast growth factor receptor 2 approved|investigational DB08901 Ponatinib small molecule P22607 Fibroblast growth factor receptor 3 approved|investigational DB08901 Ponatinib small molecule P22455 Fibroblast growth factor receptor 4 approved|investigational DB08901 Ponatinib small molecule P06239 Tyrosine-protein kinase Lck approved|investigational DB08901 Ponatinib small molecule P12931 Proto-oncogene tyrosine-protein kinase Src approved|investigational DB08901 Ponatinib small molecule P07948 Tyrosine-protein kinase Lyn approved|investigational DB08901 Ponatinib small molecule P16234 Platelet-derived growth factor receptor alpha approved DB08904 Certolizumab pegol biotech P01375 Tumor necrosis factor approved DB08906 Fluticasone furoate small molecule P04150 Glucocorticoid receptor approved DB08907 Canagliflozin small molecule P31639 Sodium/glucose cotransporter 2 approved DB08907 Canagliflozin small molecule P13866 Sodium/glucose cotransporter 1 approved|investigational DB08908 Dimethyl fumarate small molecule Q14145 Kelch-like ECH-associated protein 1 approved|investigational DB08908 Dimethyl fumarate small molecule Q04206 Transcription factor p65 approved DB08910 Pomalidomide small molecule Q96SW2 Protein cereblon approved DB08910 Pomalidomide small molecule P01375 Tumor necrosis factor approved DB08910 Pomalidomide small molecule P35354 Prostaglandin G/H synthase 2 approved DB08911 Trametinib small molecule Q02750 Dual specificity mitogen-activated protein kinase kinase 1 approved DB08911 Trametinib small molecule P36507 Dual specificity mitogen-activated protein kinase kinase 2 approved|investigational DB08912 Dabrafenib small molecule P15056 Serine/threonine-protein kinase B-raf approved|investigational DB08912 Dabrafenib small molecule P04049 RAF proto-oncogene serine/threonine-protein kinase approved|investigational DB08912 Dabrafenib small molecule P57059 Serine/threonine-protein kinase SIK1 approved|investigational DB08912 Dabrafenib small molecule Q8NG66 Serine/threonine-protein kinase Nek11 approved|investigational DB08912 Dabrafenib small molecule P53667 LIM domain kinase 1 approved DB08916 Afatinib small molecule P00533 Epidermal growth factor receptor approved DB08916 Afatinib small molecule P04626 Receptor tyrosine-protein kinase erbB-2 approved DB08916 Afatinib small molecule Q15303 Receptor tyrosine-protein kinase erbB-4 approved DB08931 Riociguat small molecule P33402 Guanylate cyclase soluble subunit alpha-2 approved DB08932 Macitentan small molecule P25101 Endothelin-1 receptor {ECO:0000305} approved DB08932 Macitentan small molecule P24530 Endothelin receptor type B {ECO:0000305} approved|investigational DB08935 Obinutuzumab biotech P11836 B-lymphocyte antigen CD20 approved DB08936 Chlorcyclizine small molecule P35367 Histamine H1 receptor approved|investigational|withdrawn DB08954 Ifenprodil small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved|investigational|withdrawn DB08954 Ifenprodil small molecule Q13224 Glutamate receptor ionotropic, NMDA 2B approved|withdrawn DB08964 Gemeprost small molecule P43115 Prostaglandin E2 receptor EP3 subtype approved|investigational DB08995 Diosmin small molecule P35869 Aryl hydrocarbon receptor approved|withdrawn DB08996 Dimetacrine small molecule P22303 Acetylcholinesterase approved|investigational DB09014 Captodiame small molecule P28335 5-hydroxytryptamine receptor 2C approved|investigational DB09014 Captodiame small molecule Q99720 Sigma non-opioid intracellular receptor 1 approved|investigational DB09014 Captodiame small molecule P35462 D(3) dopamine receptor approved DB09016 Butriptyline small molecule P31645 Sodium-dependent serotonin transporter approved DB09016 Butriptyline small molecule P35367 Histamine H1 receptor approved DB09016 Butriptyline small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB09018 Bromopride small molecule P14416 D(2) dopamine receptor approved|investigational DB09026 Aliskiren small molecule P00797 Renin approved DB09029 Secukinumab biotech Q16552 Interleukin-17A approved DB09030 Vorapaxar small molecule P25116 Proteinase-activated receptor 1 approved|investigational DB09031 Miltefosine small molecule P08183 Multidrug resistance protein 1 approved DB09033 Vedolizumab biotech P13612 Integrin alpha-4 approved DB09033 Vedolizumab biotech P26010 Integrin beta-7 approved|investigational DB09036 Siltuximab biotech P05231 Interleukin-6 approved DB09038 Empagliflozin small molecule P31639 Sodium/glucose cotransporter 2 approved DB09039 Eliglustat small molecule Q16739 Ceramide glucosyltransferase approved DB09049 Naloxegol small molecule P35372 Mu-type opioid receptor approved|investigational DB09052 Blinatumomab biotech P15391 B-lymphocyte antigen CD19 approved|investigational DB09052 Blinatumomab biotech P04234 T-cell surface glycoprotein CD3 delta chain approved DB09053 Ibrutinib small molecule Q06187 Tyrosine-protein kinase BTK approved DB09063 Ceritinib small molecule Q9UM73 ALK tyrosine kinase receptor approved|investigational DB09064 Ciprofibrate small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved|investigational DB09068 Vortioxetine small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB09068 Vortioxetine small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational DB09069 Trimetazidine small molecule P09110 3-ketoacyl-CoA thiolase, peroxisomal approved|investigational DB09070 Tibolone small molecule P03372 Estrogen receptor approved|investigational DB09073 Palbociclib small molecule P11802 Cyclin-dependent kinase 4 approved|investigational DB09073 Palbociclib small molecule Q00534 Cyclin-dependent kinase 6 approved DB09074 Olaparib small molecule P09874 Poly [ADP-ribose] polymerase 1 approved DB09074 Olaparib small molecule Q9UGN5 Poly [ADP-ribose] polymerase 2 approved DB09074 Olaparib small molecule Q9Y6F1 Poly [ADP-ribose] polymerase 3 approved DB09076 Umeclidinium small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB09076 Umeclidinium small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB09076 Umeclidinium small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB09076 Umeclidinium small molecule P08173 Muscarinic acetylcholine receptor M4 approved|investigational DB09078 Lenvatinib small molecule P17948 Vascular endothelial growth factor receptor 1 approved|investigational DB09078 Lenvatinib small molecule P35916 Vascular endothelial growth factor receptor 3 approved|investigational DB09078 Lenvatinib small molecule P11362 Fibroblast growth factor receptor 1 approved|investigational DB09078 Lenvatinib small molecule P21802 Fibroblast growth factor receptor 2 approved|investigational DB09078 Lenvatinib small molecule P22607 Fibroblast growth factor receptor 3 approved|investigational DB09078 Lenvatinib small molecule P22455 Fibroblast growth factor receptor 4 approved|investigational DB09078 Lenvatinib small molecule P10721 Mast/stem cell growth factor receptor Kit approved DB09079 Nintedanib small molecule P17948 Vascular endothelial growth factor receptor 1 approved DB09079 Nintedanib small molecule P35916 Vascular endothelial growth factor receptor 3 approved DB09079 Nintedanib small molecule P11362 Fibroblast growth factor receptor 1 approved DB09079 Nintedanib small molecule P21802 Fibroblast growth factor receptor 2 approved DB09079 Nintedanib small molecule P22607 Fibroblast growth factor receptor 3 approved DB09079 Nintedanib small molecule P36888 Receptor-type tyrosine-protein kinase FLT3 approved DB09079 Nintedanib small molecule P06239 Tyrosine-protein kinase Lck approved DB09079 Nintedanib small molecule P07948 Tyrosine-protein kinase Lyn approved DB09079 Nintedanib small molecule P12931 Proto-oncogene tyrosine-protein kinase Src approved|vet_approved DB09085 Tetracaine small molecule P21817 Ryanodine receptor 1 approved|vet_approved DB09085 Tetracaine small molecule Q92736 Ryanodine receptor 2 approved DB09089 Trimebutine small molecule P35372 Mu-type opioid receptor approved DB09089 Trimebutine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved DB09089 Trimebutine small molecule Q12791 Calcium-activated potassium channel subunit alpha-1 approved DB09089 Trimebutine small molecule O43497 Voltage-dependent T-type calcium channel subunit alpha-1G approved DB09090 Pinaverium small molecule Q13698 Voltage-dependent L-type calcium channel subunit alpha-1S approved|withdrawn DB09091 Tixocortol small molecule P04150 Glucocorticoid receptor approved|withdrawn DB09091 Tixocortol small molecule Q92769 Histone deacetylase 2 approved|withdrawn DB09092 Xanthinol small molecule P39023 60S ribosomal protein L3 approved|withdrawn DB09092 Xanthinol small molecule Q13423 NAD(P) transhydrogenase, mitochondrial approved|withdrawn DB09092 Xanthinol small molecule P04406 Glyceraldehyde-3-phosphate dehydrogenase approved|withdrawn DB09092 Xanthinol small molecule P50213 Isocitrate dehydrogenase [NAD] subunit alpha, mitochondrial approved|withdrawn DB09092 Xanthinol small molecule Q02218 2-oxoglutarate dehydrogenase, mitochondrial approved|withdrawn DB09092 Xanthinol small molecule P40926 Malate dehydrogenase, mitochondrial approved|investigational|withdrawn DB09095 Difluocortolone small molecule P12429 Annexin A3 approved|investigational|withdrawn DB09095 Difluocortolone small molecule P04150 Glucocorticoid receptor approved|investigational DB09097 Quinagolide small molecule P14416 D(2) dopamine receptor approved|investigational|withdrawn DB09098 Somatrem biotech P10912 Growth hormone receptor approved|investigational|withdrawn DB09098 Somatrem biotech P08069 Insulin-like growth factor 1 receptor approved|investigational|withdrawn DB09103 Ancestim biotech P10721 Mast/stem cell growth factor receptor Kit approved DB09107 Methoxy polyethylene glycol-epoetin beta biotech P19235 Erythropoietin receptor approved|investigational DB09112 Nitrous acid small molecule P69905 Hemoglobin subunit alpha approved|investigational DB09112 Nitrous acid small molecule P68871 Hemoglobin subunit beta approved|investigational DB09112 Nitrous acid small molecule P02144 Myoglobin approved|withdrawn DB09116 Calcium carbimide small molecule P48448 Aldehyde dehydrogenase family 3 member B2 approved DB09118 Stiripentol small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB09118 Stiripentol small molecule P00338 L-lactate dehydrogenase A chain approved DB09118 Stiripentol small molecule P07195 L-lactate dehydrogenase B chain approved DB09119 Eslicarbazepine acetate small molecule Q99571 P2X purinoceptor 4 approved|investigational DB09120 Zucapsaicin small molecule Q8NER1 Transient receptor potential cation channel subfamily V member 1 approved|withdrawn DB09121 Aurothioglucose small molecule Q08828 Adenylate cyclase type 1 approved|withdrawn DB09121 Aurothioglucose small molecule Q08462 Adenylate cyclase type 2 approved|withdrawn DB09121 Aurothioglucose small molecule O95622 Adenylate cyclase type 5 approved DB09123 Dienogest small molecule P06401 Progesterone receptor approved DB09123 Dienogest small molecule P10275 Androgen receptor approved DB09124 Medrogestone small molecule P06401 Progesterone receptor approved|vet_approved DB09126 Chorionic Gonadotropin (Human) biotech P22888 Lutropin-choriogonadotropic hormone receptor approved|investigational DB09128 Brexpiprazole small molecule P14416 D(2) dopamine receptor approved|investigational DB09128 Brexpiprazole small molecule P28223 5-hydroxytryptamine receptor 2A approved|vet_approved DB09140 Oxygen small molecule Q9Y5S8 NADPH oxidase 1 approved|vet_approved DB09140 Oxygen small molecule P69905 Hemoglobin subunit alpha approved|vet_approved DB09140 Oxygen small molecule P68871 Hemoglobin subunit beta approved|investigational DB09143 Sonidegib small molecule Q99835 Smoothened homolog approved DB09146 Iron saccharate small molecule P69905 Hemoglobin subunit alpha approved DB09148 Florbetaben (18F) small molecule P05067 Amyloid-beta A4 protein approved|investigational DB09149 Florbetapir (18F) small molecule P05067 Amyloid-beta A4 protein approved|investigational DB09151 Flutemetamol (18F) small molecule P05067 Amyloid-beta A4 protein approved DB09166 Etizolam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB09166 Etizolam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB09166 Etizolam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB09166 Etizolam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved DB09166 Etizolam small molecule P25105 Platelet-activating factor receptor approved DB09167 Dosulepin small molecule P28223 5-hydroxytryptamine receptor 2A approved DB09167 Dosulepin small molecule P35367 Histamine H1 receptor approved DB09167 Dosulepin small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB09167 Dosulepin small molecule P08172 Muscarinic acetylcholine receptor M2 approved DB09167 Dosulepin small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB09167 Dosulepin small molecule P08173 Muscarinic acetylcholine receptor M4 approved DB09167 Dosulepin small molecule P23975 Sodium-dependent noradrenaline transporter approved DB09167 Dosulepin small molecule P31645 Sodium-dependent serotonin transporter approved|investigational|withdrawn DB09185 Viloxazine small molecule P23975 Sodium-dependent noradrenaline transporter withdrawn DB09194 Etoperidone small molecule P14416 D(2) dopamine receptor withdrawn DB09194 Etoperidone small molecule P35367 Histamine H1 receptor withdrawn DB09194 Etoperidone small molecule P11229 Muscarinic acetylcholine receptor M1 withdrawn DB09194 Etoperidone small molecule P28223 5-hydroxytryptamine receptor 2A withdrawn DB09194 Etoperidone small molecule P28335 5-hydroxytryptamine receptor 2C approved|illicit DB09209 Pholcodine small molecule P35372 Mu-type opioid receptor approved|illicit DB09209 Pholcodine small molecule P41143 Delta-type opioid receptor approved|investigational DB09213 Dexibuprofen small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB09213 Dexibuprofen small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB09213 Dexibuprofen small molecule P10415 Apoptosis regulator Bcl-2 approved|investigational DB09213 Dexibuprofen small molecule P07204 Thrombomodulin approved|investigational DB09213 Dexibuprofen small molecule P00750 Tissue-type plasminogen activator approved|investigational DB09213 Dexibuprofen small molecule P12104 Fatty acid-binding protein, intestinal approved|investigational DB09213 Dexibuprofen small molecule P37231 Peroxisome proliferator-activated receptor gamma approved|investigational DB09213 Dexibuprofen small molecule P13569 Cystic fibrosis transmembrane conductance regulator approved|investigational DB09214 Dexketoprofen small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB09214 Dexketoprofen small molecule P35354 Prostaglandin G/H synthase 2 withdrawn DB09215 Droxicam small molecule P23219 Prostaglandin G/H synthase 1 withdrawn DB09215 Droxicam small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB09216 Tolfenamic Acid small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB09216 Tolfenamic Acid small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB09220 Nicorandil small molecule O60706 ATP-binding cassette sub-family C member 9 approved|investigational DB09224 Melperone small molecule P14416 D(2) dopamine receptor approved|investigational|withdrawn DB09225 Zotepine small molecule P14416 D(2) dopamine receptor approved|investigational|withdrawn DB09225 Zotepine small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational|withdrawn DB09225 Zotepine small molecule P34969 5-hydroxytryptamine receptor 7 approved|investigational|withdrawn DB09225 Zotepine small molecule P23975 Sodium-dependent noradrenaline transporter approved|investigational|withdrawn DB09225 Zotepine small molecule P31645 Sodium-dependent serotonin transporter approved DB09227 Barnidipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB09228 Conestat alfa biotech P09871 Complement C1s subcomponent approved|investigational DB09228 Conestat alfa biotech P00748 Coagulation factor XII approved|investigational DB09228 Conestat alfa biotech P00734 Prothrombin approved|investigational DB09228 Conestat alfa biotech P03951 Coagulation factor XI approved|investigational DB09228 Conestat alfa biotech P00750 Tissue-type plasminogen activator approved|investigational DB09231 Benidipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB09231 Benidipine small molecule Q00975 Voltage-dependent N-type calcium channel subunit alpha-1B approved|investigational DB09231 Benidipine small molecule O43497 Voltage-dependent T-type calcium channel subunit alpha-1G approved|investigational DB09232 Cilnidipine small molecule Q00975 Voltage-dependent N-type calcium channel subunit alpha-1B approved|investigational DB09232 Cilnidipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB09236 Lacidipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB09238 Manidipine small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB09238 Manidipine small molecule O43497 Voltage-dependent T-type calcium channel subunit alpha-1G approved|investigational DB09241 Methylene blue small molecule P33402 Guanylate cyclase soluble subunit alpha-2 approved|investigational DB09241 Methylene blue small molecule P29475 Nitric oxide synthase, brain approved|investigational DB09242 Moxonidine small molecule Q9Y2I1 Nischarin approved DB09245 Toloxatone small molecule P21397 Amine oxidase [flavin-containing] A approved|investigational DB09258 Bemiparin small molecule P00742 Coagulation factor X approved|investigational DB09258 Bemiparin small molecule P01008 Antithrombin-III approved|investigational DB09258 Bemiparin small molecule P05546 Heparin cofactor 2 approved|investigational DB09266 Technetium Tc-99m tilmanocept small molecule P22897 Macrophage mannose receptor 1 approved|investigational|nutraceutical DB09270 Ubidecarenone small molecule P56181 NADH dehydrogenase [ubiquinone] flavoprotein 3, mitochondrial approved|investigational|nutraceutical DB09270 Ubidecarenone small molecule P31040 Succinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrial approved|investigational DB09279 Fimasartan small molecule P30556 Type-1 angiotensin II receptor approved DB09280 Lumacaftor small molecule P13569 Cystic fibrosis transmembrane conductance regulator approved|investigational DB09282 Molsidomine small molecule P33402 Guanylate cyclase soluble subunit alpha-2 approved DB09283 Trapidil small molecule P54750 Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A approved DB09285 Morniflumate small molecule P09917 Arachidonate 5-lipoxygenase approved DB09285 Morniflumate small molecule P35354 Prostaglandin G/H synthase 2 approved DB09285 Morniflumate small molecule Q15722 Leukotriene B4 receptor 1 approved DB09285 Morniflumate small molecule P21731 Thromboxane A2 receptor approved|investigational DB09286 Pipamperone small molecule P14416 D(2) dopamine receptor approved|investigational DB09286 Pipamperone small molecule P28223 5-hydroxytryptamine receptor 2A approved|investigational DB09286 Pipamperone small molecule P21917 D(4) dopamine receptor approved|investigational DB09286 Pipamperone small molecule P35462 D(3) dopamine receptor approved|investigational DB09288 Propacetamol small molecule P23219 Prostaglandin G/H synthase 1 approved|investigational DB09288 Propacetamol small molecule P35354 Prostaglandin G/H synthase 2 approved|investigational DB09288 Propacetamol small molecule Q8NER1 Transient receptor potential cation channel subfamily V member 1 approved|investigational DB09289 Tianeptine small molecule P31645 Sodium-dependent serotonin transporter approved|investigational DB09289 Tianeptine small molecule P42261 Glutamate receptor 1 approved DB09292 Sacubitril small molecule P08473 Neprilysin approved|investigational|vet_approved DB09300 Butylscopolamine small molecule P20309 Muscarinic acetylcholine receptor M3 approved|investigational|vet_approved DB09300 Butylscopolamine small molecule P08172 Muscarinic acetylcholine receptor M2 approved|investigational|nutraceutical DB09301 Chondroitin sulfate small molecule P23560 Brain-derived neurotrophic factor approved|investigational|nutraceutical DB09301 Chondroitin sulfate small molecule P39905 Glial cell line-derived neurotrophic factor approved|investigational|nutraceutical DB09301 Chondroitin sulfate small molecule P15692 Vascular endothelial growth factor A approved|investigational|nutraceutical DB09301 Chondroitin sulfate small molecule P13500 C-C motif chemokine 2 approved DB09338 Mersalyl small molecule P05186 Alkaline phosphatase, tissue-nonspecific isozyme approved DB09338 Mersalyl small molecule P29972 Aquaporin-1 approved DB09338 Mersalyl small molecule P53985 Monocarboxylate transporter 1 approved DB09357 Dexpanthenol small molecule P20309 Muscarinic acetylcholine receptor M3 approved DB09369 Polyestradiol phosphate small molecule P03372 Estrogen receptor approved DB09371 Norethynodrel small molecule P03372 Estrogen receptor approved DB09371 Norethynodrel small molecule P10275 Androgen receptor approved DB09371 Norethynodrel small molecule P04278 Sex hormone-binding globulin approved DB09389 Norgestrel small molecule P06401 Progesterone receptor approved DB09389 Norgestrel small molecule P18405 3-oxo-5-alpha-steroid 4-dehydrogenase 1 approved DB09389 Norgestrel small molecule P10275 Androgen receptor approved|investigational DB09462 Glycerin small molecule Q03181 Peroxisome proliferator-activated receptor delta approved|investigational DB09462 Glycerin small molecule P09211 Glutathione S-transferase P approved|investigational DB09462 Glycerin small molecule Q9NPH2 Inositol-3-phosphate synthase 1 approved|investigational DB09462 Glycerin small molecule P00325 Alcohol dehydrogenase 1B approved|investigational DB09462 Glycerin small molecule Q14643 Inositol 1,4,5-trisphosphate receptor type 1 approved|investigational DB09462 Glycerin small molecule P09466 Glycodelin approved|investigational DB09462 Glycerin small molecule P17050 Alpha-N-acetylgalactosaminidase approved|investigational DB09462 Glycerin small molecule P37173 TGF-beta receptor type-2 approved|investigational DB09462 Glycerin small molecule P84077 ADP-ribosylation factor 1 approved|investigational DB09462 Glycerin small molecule O43252 Bifunctional 3'-phosphoadenosine 5'-phosphosulfate synthase 1 approved|investigational DB09462 Glycerin small molecule O14717 tRNA (cytosine(38)-C(5))-methyltransferase approved|vet_approved DB09472 Sodium sulfate small molecule P00918 Carbonic anhydrase 2 approved|vet_approved DB09472 Sodium sulfate small molecule P00915 Carbonic anhydrase 1 approved|investigational DB09481 Magnesium carbonate small molecule Q05586 Glutamate receptor ionotropic, NMDA 1 approved DB09488 Acrivastine small molecule P35367 Histamine H1 receptor approved|investigational DB09526 Hydroquinone small molecule P14679 Tyrosinase approved|investigational DB09559 Necitumumab biotech P00533 Epidermal growth factor receptor approved DB09564 Insulin Degludec biotech P06213 Insulin receptor approved DB11071 Phenyl salicylate small molecule P03372 Estrogen receptor approved DB11075 Hypromellose small molecule P16422 Epithelial cell adhesion molecule approved DB11081 Aluminum chloride small molecule P00367 Glutamate dehydrogenase 1, mitochondrial approved DB11085 Resorcinol small molecule P07202 Thyroid peroxidase {ECO:0000305} approved DB11093 Calcium Citrate small molecule P41180 Extracellular calcium-sensing receptor {ECO:0000305} approved DB11093 Calcium Citrate small molecule P27797 Calreticulin approved DB11093 Calcium Citrate small molecule Q99828 Calcium and integrin-binding protein 1 approved DB11093 Calcium Citrate small molecule O75340 Programmed cell death protein 6 approved DB11093 Calcium Citrate small molecule P30626 Sorcin approved DB11093 Calcium Citrate small molecule Q99653 Calcineurin B homologous protein 1 approved DB11093 Calcium Citrate small molecule P09486 SPARC approved DB11093 Calcium Citrate small molecule P27824 Calnexin approved DB11093 Calcium Citrate small molecule P35556 Fibrillin-2 approved DB11093 Calcium Citrate small molecule P04271 Protein S100-B approved DB11093 Calcium Citrate small molecule O14958 Calsequestrin-2 approved DB11093 Calcium Citrate small molecule Q15493 Regucalcin approved DB11093 Calcium Citrate small molecule Q9UBV8 Peflin {ECO:0000303|PubMed:10486255} approved DB11093 Calcium Citrate small molecule P06703 Protein S100-A6 approved DB11093 Calcium Citrate small molecule P13693 Translationally-controlled tumor protein approved DB11093 Calcium Citrate small molecule O75838 Calcium and integrin-binding family member 2 approved DB11093 Calcium Citrate small molecule Q99584 Protein S100-A13 approved DB11093 Calcium Citrate small molecule P31415 Calsequestrin-1 approved DB11093 Calcium Citrate small molecule Q02818 Nucleobindin-1 approved DB11093 Calcium Citrate small molecule P80303 Nucleobindin-2 approved DB11093 Calcium Citrate small molecule Q75N90 Fibrillin-3 approved DB11093 Calcium Citrate small molecule P28676 Grancalcin approved DB11093 Calcium Citrate small molecule Q9ULU8 Calcium-dependent secretion activator 1 approved DB11093 Calcium Citrate small molecule Q96FQ6 Protein S100-A16 approved DB11093 Calcium Citrate small molecule Q13938 Calcyphosin approved DB11093 Calcium Citrate small molecule Q86UW7 Calcium-dependent secretion activator 2 approved DB11093 Calcium Citrate small molecule Q96L12 Calreticulin-3 approved DB11093 Calcium Citrate small molecule Q9ULB1 Neurexin-1 approved DB11093 Calcium Citrate small molecule P62166 Neuronal calcium sensor 1 approved|illicit DB11130 Opium small molecule P41143 Delta-type opioid receptor approved|illicit DB11130 Opium small molecule P35372 Mu-type opioid receptor approved|vet_approved DB11156 Pyrantel small molecule Q9HC97 G-protein coupled receptor 35 approved|vet_approved DB11156 Pyrantel small molecule P11229 Muscarinic acetylcholine receptor M1 approved DB11157 Anthralin small molecule P35908 Keratin, type II cytoskeletal 2 epidermal approved DB11157 Anthralin small molecule Q9UQF2 C-Jun-amino-terminal kinase-interacting protein 1 approved DB11157 Anthralin small molecule Q99456 Keratin, type I cytoskeletal 12 approved DB11181 Homatropine small molecule P23141 Liver carboxylesterase 1 approved|investigational DB11300 Thrombin small molecule P25116 Proteinase-activated receptor 1 approved DB11348 Calcium Phosphate small molecule P41180 Extracellular calcium-sensing receptor {ECO:0000305} approved DB11348 Calcium Phosphate small molecule P27797 Calreticulin approved DB11348 Calcium Phosphate small molecule Q99828 Calcium and integrin-binding protein 1 approved DB11348 Calcium Phosphate small molecule O75340 Programmed cell death protein 6 approved DB11348 Calcium Phosphate small molecule P30626 Sorcin approved DB11348 Calcium Phosphate small molecule Q99653 Calcineurin B homologous protein 1 approved DB11348 Calcium Phosphate small molecule P09486 SPARC approved DB11348 Calcium Phosphate small molecule P27824 Calnexin approved DB11348 Calcium Phosphate small molecule P35556 Fibrillin-2 approved DB11348 Calcium Phosphate small molecule P04271 Protein S100-B approved DB11348 Calcium Phosphate small molecule O14958 Calsequestrin-2 approved DB11348 Calcium Phosphate small molecule Q15493 Regucalcin approved DB11348 Calcium Phosphate small molecule Q9UBV8 Peflin {ECO:0000303|PubMed:10486255} approved DB11348 Calcium Phosphate small molecule P06703 Protein S100-A6 approved DB11348 Calcium Phosphate small molecule P13693 Translationally-controlled tumor protein approved DB11348 Calcium Phosphate small molecule O75838 Calcium and integrin-binding family member 2 approved DB11348 Calcium Phosphate small molecule Q99584 Protein S100-A13 approved DB11348 Calcium Phosphate small molecule P31415 Calsequestrin-1 approved DB11348 Calcium Phosphate small molecule Q02818 Nucleobindin-1 approved DB11348 Calcium Phosphate small molecule P80303 Nucleobindin-2 approved DB11348 Calcium Phosphate small molecule Q75N90 Fibrillin-3 approved DB11348 Calcium Phosphate small molecule P28676 Grancalcin approved DB11348 Calcium Phosphate small molecule Q9ULU8 Calcium-dependent secretion activator 1 approved DB11348 Calcium Phosphate small molecule Q96FQ6 Protein S100-A16 approved DB11348 Calcium Phosphate small molecule Q13938 Calcyphosin approved DB11348 Calcium Phosphate small molecule Q86UW7 Calcium-dependent secretion activator 2 approved DB11348 Calcium Phosphate small molecule Q96L12 Calreticulin-3 approved DB11348 Calcium Phosphate small molecule Q9ULB1 Neurexin-1 approved DB11348 Calcium Phosphate small molecule P62166 Neuronal calcium sensor 1 approved|investigational|vet_approved DB11386 Chlorobutanol small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB11560 Lesinurad small molecule Q9NSA0 Solute carrier family 22 member 11 approved DB11577 Indigotindisulfonic Acid small molecule P35869 Aryl hydrocarbon receptor approved|investigational DB11582 Thiocolchicoside small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved|investigational DB11582 Thiocolchicoside small molecule P23415 Glycine receptor subunit alpha-1 approved|investigational DB11582 Thiocolchicoside small molecule O14788 Tumor necrosis factor ligand superfamily member 11 approved DB11590 Thimerosal small molecule Q99707 Methionine synthase approved DB11590 Thimerosal small molecule P54710 Sodium/potassium-transporting ATPase subunit gamma approved|investigational DB11591 Bilastine small molecule P35367 Histamine H1 receptor approved DB11598 Antithrombin III human biotech P01008 Antithrombin-III approved|investigational DB11606 Susoctocog alfa biotech P04275 von Willebrand factor approved DB11614 Rupatadine small molecule P25105 Platelet-activating factor receptor approved DB11614 Rupatadine small molecule P35367 Histamine H1 receptor approved DB11619 Gestrinone small molecule P04278 Sex hormone-binding globulin approved DB11619 Gestrinone small molecule P06401 Progesterone receptor approved DB11619 Gestrinone small molecule P04150 Glucocorticoid receptor approved DB11619 Gestrinone small molecule P10275 Androgen receptor approved DB11619 Gestrinone small molecule P03372 Estrogen receptor approved DB11626 Tasonermin biotech P19438 Tumor necrosis factor receptor superfamily member 1A approved DB11626 Tasonermin biotech P20333 Tumor necrosis factor receptor superfamily member 1B approved|investigational DB11633 Isavuconazole small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB11633 Isavuconazole small molecule Q13936 Voltage-dependent L-type calcium channel subunit alpha-1C approved|investigational DB11633 Isavuconazole small molecule P48051 G protein-activated inward rectifier potassium channel 2 approved|investigational DB11633 Isavuconazole small molecule P51787 Potassium voltage-gated channel subfamily KQT member 1 {ECO:0000305} approved|investigational DB11633 Isavuconazole small molecule Q14524 Sodium channel protein type 5 subunit alpha approved|investigational DB11638 Artenimol small molecule P63261 Actin, cytoplasmic 2 approved|investigational DB11638 Artenimol small molecule P49419 Alpha-aminoadipic semialdehyde dehydrogenase approved|investigational DB11638 Artenimol small molecule P07355 Annexin A2 approved|investigational DB11638 Artenimol small molecule P25705 ATP synthase subunit alpha, mitochondrial {ECO:0000305} approved|investigational DB11638 Artenimol small molecule O75964 ATP synthase subunit g, mitochondrial approved|investigational DB11638 Artenimol small molecule P48047 ATP synthase subunit O, mitochondrial approved|investigational DB11638 Artenimol small molecule P20810 Calpastatin approved|investigational DB11638 Artenimol small molecule P49368 T-complex protein 1 subunit gamma approved|investigational DB11638 Artenimol small molecule P23528 Cofilin-1 approved|investigational DB11638 Artenimol small molecule O00299 Chloride intracellular channel protein 1 approved|investigational DB11638 Artenimol small molecule P21291 Cysteine and glycine-rich protein 1 approved|investigational DB11638 Artenimol small molecule Q16555 Dihydropyrimidinase-related protein 2 approved|investigational DB11638 Artenimol small molecule P15924 Desmoplakin approved|investigational DB11638 Artenimol small molecule P68104 Elongation factor 1-alpha 1 approved|investigational DB11638 Artenimol small molecule P06733 Alpha-enolase approved|investigational DB11638 Artenimol small molecule P21333 Filamin-A approved|investigational DB11638 Artenimol small molecule Q9C0B1 Alpha-ketoglutarate-dependent dioxygenase FTO approved|investigational DB11638 Artenimol small molecule P11413 Glucose-6-phosphate 1-dehydrogenase approved|investigational DB11638 Artenimol small molecule O14556 Glyceraldehyde-3-phosphate dehydrogenase, testis-specific approved|investigational DB11638 Artenimol small molecule P06744 Glucose-6-phosphate isomerase approved|investigational DB11638 Artenimol small molecule P22626 Heterogeneous nuclear ribonucleoproteins A2/B1 approved|investigational DB11638 Artenimol small molecule Q14103 Heterogeneous nuclear ribonucleoprotein D0 approved|investigational DB11638 Artenimol small molecule P61978 Heterogeneous nuclear ribonucleoprotein K approved|investigational DB11638 Artenimol small molecule Q5SSJ5 Heterochromatin protein 1-binding protein 3 approved|investigational DB11638 Artenimol small molecule P04792 Heat shock protein beta-1 approved|investigational DB11638 Artenimol small molecule P46940 Ras GTPase-activating-like protein IQGAP1 approved|investigational DB11638 Artenimol small molecule Q92945 Far upstream element-binding protein 2 approved|investigational DB11638 Artenimol small molecule P00338 L-lactate dehydrogenase A chain approved|investigational DB11638 Artenimol small molecule P07195 L-lactate dehydrogenase B chain approved|investigational DB11638 Artenimol small molecule P09382 Galectin-1 approved|investigational DB11638 Artenimol small molecule P27816 Microtubule-associated protein 4 approved|investigational DB11638 Artenimol small molecule P40925 Malate dehydrogenase, cytoplasmic approved|investigational DB11638 Artenimol small molecule P55786 Puromycin-sensitive aminopeptidase approved|investigational DB11638 Artenimol small molecule P07737 Profilin-1 approved|investigational DB11638 Artenimol small molecule P00558 Phosphoglycerate kinase 1 approved|investigational DB11638 Artenimol small molecule P14618 Pyruvate kinase PKM approved|investigational DB11638 Artenimol small molecule P62937 Peptidyl-prolyl cis-trans isomerase A approved|investigational DB11638 Artenimol small molecule Q06830 Peroxiredoxin-1 approved|investigational DB11638 Artenimol small molecule P27635 60S ribosomal protein L10 {ECO:0000305} approved|investigational DB11638 Artenimol small molecule P50914 60S ribosomal protein L14 approved|investigational DB11638 Artenimol small molecule Q07020 60S ribosomal protein L18 approved|investigational DB11638 Artenimol small molecule P62750 60S ribosomal protein L23a approved|investigational DB11638 Artenimol small molecule P42766 60S ribosomal protein L35 approved|investigational DB11638 Artenimol small molecule P36578 60S ribosomal protein L4 approved|investigational DB11638 Artenimol small molecule P62277 40S ribosomal protein S13 approved|investigational DB11638 Artenimol small molecule P08708 40S ribosomal protein S17 {ECO:0000305} approved|investigational DB11638 Artenimol small molecule P62269 40S ribosomal protein S18 approved|investigational DB11638 Artenimol small molecule P39019 40S ribosomal protein S19 approved|investigational DB11638 Artenimol small molecule P46782 40S ribosomal protein S5 approved|investigational DB11638 Artenimol small molecule P62753 40S ribosomal protein S6 approved|investigational DB11638 Artenimol small molecule P62241 40S ribosomal protein S8 approved|investigational DB11638 Artenimol small molecule P46781 40S ribosomal protein S9 approved|investigational DB11638 Artenimol small molecule Q15637 Splicing factor 1 approved|investigational DB11638 Artenimol small molecule P23246 Splicing factor, proline- and glutamine-rich approved|investigational DB11638 Artenimol small molecule P62316 Small nuclear ribonucleoprotein Sm D2 approved|investigational DB11638 Artenimol small molecule P37108 Signal recognition particle 14 kDa protein approved|investigational DB11638 Artenimol small molecule Q08170 Serine/arginine-rich splicing factor 4 approved|investigational DB11638 Artenimol small molecule P37802 Transgelin-2 approved|investigational DB11638 Artenimol small molecule P60174 Triosephosphate isomerase approved|investigational DB11638 Artenimol small molecule P09493 Tropomyosin alpha-1 chain approved|investigational DB11638 Artenimol small molecule Q71U36 Tubulin alpha-1A chain approved|investigational DB11638 Artenimol small molecule P08670 Vimentin approved|investigational DB11638 Artenimol small molecule Q15942 Zyxin approved|investigational DB11638 Artenimol small molecule P11142 Heat shock cognate 71 kDa protein approved|investigational DB11638 Artenimol small molecule Q9BUF5 Tubulin beta-6 chain approved|investigational DB11638 Artenimol small molecule P04350 Tubulin beta-4A chain approved|investigational DB11638 Artenimol small molecule P07437 Tubulin beta chain approved|investigational DB11638 Artenimol small molecule P04075 Fructose-bisphosphate aldolase A approved|investigational DB11638 Artenimol small molecule P04406 Glyceraldehyde-3-phosphate dehydrogenase approved|investigational DB11638 Artenimol small molecule P99999 Cytochrome c approved|investigational DB11638 Artenimol small molecule P18669 Phosphoglycerate mutase 1 approved|investigational DB11638 Artenimol small molecule P35579 Myosin-9 approved|investigational DB11638 Artenimol small molecule P07237 Protein disulfide-isomerase approved|investigational DB11638 Artenimol small molecule P17844 Probable ATP-dependent RNA helicase DDX5 approved|investigational DB11638 Artenimol small molecule P34897 Serine hydroxymethyltransferase, mitochondrial approved|investigational DB11638 Artenimol small molecule Q13838 Spliceosome RNA helicase DDX39B approved|investigational DB11638 Artenimol small molecule P06748 Nucleophosmin approved|investigational DB11638 Artenimol small molecule P02768 Serum albumin approved|investigational DB11639 Dibotermin alfa biotech Q13873 Bone morphogenetic protein receptor type-2 approved|investigational DB11639 Dibotermin alfa biotech P36894 Bone morphogenetic protein receptor type-1A approved|investigational DB11642 Pitolisant small molecule Q9Y5N1 Histamine H3 receptor approved|investigational DB11642 Pitolisant small molecule Q12809 Potassium voltage-gated channel subfamily H member 2 approved|investigational DB11994 Diacerein small molecule Q13133 Oxysterols receptor LXR-alpha approved|investigational DB11994 Diacerein small molecule P55055 Oxysterols receptor LXR-beta approved|investigational DB11994 Diacerein small molecule P09917 Arachidonate 5-lipoxygenase approved|investigational DB11994 Diacerein small molecule P08684 Cytochrome P450 3A4 approved|investigational DB11994 Diacerein small molecule P05181 Cytochrome P450 2E1 approved|investigational DB11994 Diacerein small molecule P11712 Cytochrome P450 2C9 approved|investigational DB11994 Diacerein small molecule P10635 Cytochrome P450 2D6 investigational|withdrawn DB12319 Benzbromarone small molecule P11712 Cytochrome P450 2C9 investigational|withdrawn DB12319 Benzbromarone small molecule P33261 Cytochrome P450 2C19 investigational DB12465 Ketanserin small molecule P28223 5-hydroxytryptamine receptor 2A investigational DB12478 Piribedil small molecule P14416 D(2) dopamine receptor investigational DB12478 Piribedil small molecule P35462 D(3) dopamine receptor investigational DB13003 Cortivazol small molecule P04150 Glucocorticoid receptor approved|investigational DB13025 Tiapride small molecule P14416 D(2) dopamine receptor approved|investigational DB13025 Tiapride small molecule P35462 D(3) dopamine receptor approved|investigational DB13025 Tiapride small molecule P35367 Histamine H1 receptor approved|investigational DB13133 Von Willebrand Factor Human biotech P00451 Coagulation factor VIII approved|investigational DB13133 Von Willebrand Factor Human biotech P02452 Collagen alpha-1(I) chain approved|investigational DB13144 Lenograstim biotech Q99062 Granulocyte colony-stimulating factor receptor approved|investigational DB13151 Anti-inhibitor coagulant complex biotech P00742 Coagulation factor X approved|investigational DB13151 Anti-inhibitor coagulant complex biotech P00734 Prothrombin approved|investigational DB13151 Anti-inhibitor coagulant complex biotech P02671 Fibrinogen alpha chain approved|investigational DB13151 Anti-inhibitor coagulant complex biotech P02675 Fibrinogen beta chain approved|investigational DB13151 Anti-inhibitor coagulant complex biotech P00488 Coagulation factor XIII A chain approved|investigational DB13151 Anti-inhibitor coagulant complex biotech P12259 Coagulation factor V approved|investigational DB13151 Anti-inhibitor coagulant complex biotech P00451 Coagulation factor VIII approved|investigational DB13151 Anti-inhibitor coagulant complex biotech P08709 Coagulation factor VII approved DB13158 Clobetasone small molecule P04150 Glucocorticoid receptor experimental DB13166 Zofenopril small molecule P12821 Angiotensin-converting enzyme approved|withdrawn DB13167 Alclofenac small molecule P35354 Prostaglandin G/H synthase 2 approved DB13179 Troleandomycin small molecule O75469 Nuclear receptor subfamily 1 group I member 2 nutraceutical DB13191 Phosphocreatine small molecule Q14353 Guanidinoacetate N-methyltransferase nutraceutical DB13191 Phosphocreatine small molecule P48029 Sodium- and chloride-dependent creatine transporter 1 nutraceutical DB13191 Phosphocreatine small molecule P06732 Creatine kinase M-type nutraceutical DB13191 Phosphocreatine small molecule P12532 Creatine kinase U-type, mitochondrial nutraceutical DB13191 Phosphocreatine small molecule P12277 Creatine kinase B-type {ECO:0000305} approved DB13192 Antihemophilic factor human biotech P00742 Coagulation factor X experimental DB13520 Metergoline small molecule Q99250 Sodium channel protein type 2 subunit alpha approved|experimental DB13615 Mifamurtide small molecule O00206 Toll-like receptor 4 approved|experimental DB13615 Mifamurtide small molecule Q9HC29 Nucleotide-binding oligomerization domain-containing protein 2 approved|experimental|investigational DB13783 Acemetacin small molecule P23219 Prostaglandin G/H synthase 1 approved|experimental|investigational DB13783 Acemetacin small molecule P35354 Prostaglandin G/H synthase 2 approved DB13872 Lormetazepam small molecule P47869 Gamma-aminobutyric acid receptor subunit alpha-2 approved DB13872 Lormetazepam small molecule P18507 Gamma-aminobutyric acid receptor subunit gamma-2 approved DB13872 Lormetazepam small molecule P34903 Gamma-aminobutyric acid receptor subunit alpha-3 approved DB13872 Lormetazepam small molecule P31644 Gamma-aminobutyric acid receptor subunit alpha-5 approved DB13872 Lormetazepam small molecule P14867 Gamma-aminobutyric acid receptor subunit alpha-1 approved DB13873 Fenofibric acid small molecule Q07869 Peroxisome proliferator-activated receptor alpha approved DB13873 Fenofibric acid small molecule P37231 Peroxisome proliferator-activated receptor gamma approved DB13873 Fenofibric acid small molecule Q03181 Peroxisome proliferator-activated receptor delta approved DB13873 Fenofibric acid small molecule O75469 Nuclear receptor subfamily 1 group I member 2 experimental DB13919 Candesartan small molecule P30556 Type-1 angiotensin II receptor